|
AGC
|
AKT1
|
AKT1_HUMAN
|
6BUUA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 478 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6BUUB
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 477 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6NPZA
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 478 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6NPZB
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
141 - 477 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4GV1A
|
1.49 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0XZ |
Type1 |
144 - 477 |
0 |
TPO308 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OCBA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XM1 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OCBB
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XM1 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKLA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMR |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKMA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SM9 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3CQUA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQU |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3CQWA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQW |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3MV5A
|
2.47 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3MVHA
|
2.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WFE |
Type1 |
145 - 476 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6CCYA
|
2.18 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX4 |
Type1 |
144 - 983 |
0 |
TPO308 |
N199S,S396P,E397S,T433V |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKKA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMH |
Type1.5_Front |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UVYA
|
2.11 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XOO |
Allosteric |
3 - 439 |
0 |
None |
E17K |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW2A
|
2.2 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
XOO |
Allosteric |
4 - 437 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW9A
|
1.9 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XQ2 |
Allosteric |
3 - 428 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW7A
|
1.972 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 439 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3O96A
|
2.7 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
IQO |
Allosteric |
2 - 429 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHHA
|
2.7 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
G4Q |
Allosteric |
2 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHJA
|
2.3 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4H |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9WA
|
2.3 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
L1Z |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EJNA
|
2.19 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
0R4 |
Type1 |
4 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
5KCVA
|
2.7 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
6S1 |
Allosteric |
6 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7APJA
|
2.05 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
none-none |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
3 - 439 |
0 |
None |
S2N |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
9ZBKE
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-none |
none-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
A1AID |
Allosteric |
141 - 478 |
0 |
None |
S473C |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHFA
|
2.9 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
G4K |
Allosteric |
3 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHGA
|
2.3 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4T |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHIA
|
2.7 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4N |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9XA
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
L1W |
Allosteric |
3 - 443 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7NH4A
|
2.3 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
UCE |
Allosteric |
4 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7NH5A
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
UC8 |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2JDOA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I5S |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2UW9A
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVP |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2X39A
|
1.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X39 |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2XH5A
|
2.72 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X37 |
Type1 |
146 - 479 |
0 |
TPO309 |
R467Q,T468E,H469M,P471E,Q472D,S474D,S476I,S478D,I479W |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
9C1WA
|
2.0 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 440 |
0 |
None |
P115A,G116A |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
8Q61A
|
2.32 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
K06 |
Type3 |
1 - 435 |
0 |
None |
N2D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZKA
|
2.3 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 441 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZOA
|
2.75 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZNA
|
2.5 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRVA
|
2.8 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
147 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRYA
|
2.8 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
none-none |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnio |
No_ligand |
No_ligand |
146 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UVCA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PV |
Type1 |
30 - 536 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5HE1A
|
3.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZS2 |
Type1 |
29 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
6C2YA
|
2.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EJS |
Type1 |
30 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3V5WA
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PR |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG3A
|
2.896 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFM |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG4A
|
2.31 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFV |
Type1 |
31 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UKKA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8DJ |
Type1.5_Front |
30 - 667 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
6U7CA
|
2.44 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q1Y |
Type1.5_Front |
30 - 669 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3CIKA
|
2.75 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 669 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7PWDA
|
2.6 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8DS |
Type1 |
27 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3KRWA
|
2.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
30 - 671 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3KRXA
|
3.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
30 - 671 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
4YHJB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
25 - 527 |
0 |
None |
C563S,C578S |
G protein-coupled receptor kinase 4 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKOA
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRKA
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARA |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRLA
|
2.73 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARB |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRPA
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARF |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
4TNDA
|
1.802 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 543 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
AF-P34947-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
4TNBA
|
2.113 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
15 - 543 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9MX2A
|
3.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
6PJXA
|
1.96 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
E104K,R304H,G438E |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
8UAQA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3F |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRFA
|
2.84 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ5 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRIA
|
2.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ8 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRJA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ9 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYNA
|
2.72 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYNB
|
2.72 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
MASTL
|
GWL_HUMAN
|
8V5HA
|
2.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
A1AAE |
Type1 |
29 - 847 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
MASTL
|
GWL_HUMAN
|
5LOHA
|
3.1 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aanon |
APEdist_nnno |
STU |
Type1 |
30 - 854 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
MASTL
|
GWL_HUMAN
|
5LOHB
|
3.1 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
none-out |
nonTYR |
APEdihe_aannn |
APEdist_nnno |
STU |
Type1 |
30 - 854 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1H1WA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5ACKA
|
1.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
73 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXA
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXB
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
77 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXC
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXD
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
76 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXE
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
1F8 |
Allosteric |
76 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXF
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXG
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXH
|
2.204 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
74 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZB
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
73 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZC
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
74 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZD
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
73 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1Z5MA
|
2.17 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LI8 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE0A
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
39Z |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE1A
|
2.14 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
517 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE2A
|
2.13 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
464 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JNZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUUA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JOZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUYA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JPZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU9A
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI3 |
Type1 |
72 - 357 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UVRA
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI8 |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUNA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JMZ |
Type1 |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2XCHA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
CKG |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HKMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
61Y |
Type1 |
76 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HNGA
|
3.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
62O |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HO7A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
63L |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HO8A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
63E |
Type1 |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1OKYA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STU |
Type1 |
72 - 360 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1OKZA
|
2.51 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
UCN |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU3A
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LY4 |
Type1 |
73 - 360 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU7A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI2 |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU8A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI1 |
Type1 |
72 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAYA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MP6 |
Type1 |
76 - 362 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAYB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MP6 |
Type1 |
76 - 362 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RWPA
|
1.92 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ABQ |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RWQA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3RW |
Type1 |
72 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3H9OA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
9BD |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2R7BA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
253 |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3IONA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
8H1 |
Type1 |
75 - 359 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3IOPA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8I1 |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCQA
|
2.501 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q0 |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCSA
|
2.487 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q1 |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3PWYA
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
SYP |
Type1 |
71 - 359 |
0 |
None |
E166C,C260S |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2XCKA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MH4 |
Type1 |
76 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCXA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q2 |
Type1.5_Back |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCYA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
3Q3 |
Type1.5_Front |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD3A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q5 |
Type1.5_Front |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAXA
|
1.75 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MP7 |
Type2 |
76 - 360 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4A
|
1.8 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
76 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4B
|
1.8 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
51 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTDA
|
2.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
605 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTGA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2V9 |
Type1 |
605 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTHA
|
1.8 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-in |
in-in |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
DRN |
Type1 |
606 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTIA
|
1.93 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MI1 |
Type1 |
606 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
4CRSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
AGS |
ATPlike |
646 - 984 |
0 |
SEP755,TPO816,TPO958 |
None |
Serine/threonine-protein kinase N2 |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE6A
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE6B
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE9A
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE9B
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
7Y1GB
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I5G |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DC6A
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3I |
Type1 |
16 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DC6B
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3I |
Type1 |
16 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AMBA
|
2.25 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
4 - 351 |
0 |
SEP11,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8X5LA
|
2.75 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
RKD |
Type1 |
17 - 351 |
0 |
SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8X5LB
|
2.75 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
RKD |
Type1 |
17 - 334 |
0 |
SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7E
|
3.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7G
|
3.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDDA
|
6.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDEA
|
5.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZJA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6J9 |
Allosteric |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZJB
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6J9 |
Allosteric |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSA
|
4.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSC
|
4.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSE
|
4.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSG
|
4.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7A
|
3.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJB
|
2.49 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJFA
|
7.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJFB
|
7.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJGA
|
6.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJGB
|
6.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3VQHA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQB |
Type1 |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ1A
|
1.768 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVX |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ2A
|
2.019 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVV |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ9A
|
1.87 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S3N |
Type1 |
11 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJAA
|
1.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4L7 |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJBA
|
1.949 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8BQ |
Type1 |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
7Y1GA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I5G |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6C0UA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EE4 |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
4RA4A
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3KZ |
Type1 |
332 - 666 |
0 |
TPO497,TPO638,SEP657 |
C619S |
Protein kinase C alpha type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE2A
|
2.95 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE3A
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE4A
|
2.68 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE4B
|
2.68 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
2I0EA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
PDS |
Type1 |
339 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
9S9TA
|
3.425 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LY4 |
Type1 |
340 - 667 |
0 |
TPO500,TPO642,SEP661 |
D427N |
Protein kinase C beta type |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
3TXOA
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
07U |
Type1 |
353 - 679 |
0 |
TPO656 |
S675E |
Protein kinase C eta type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3YI
|
3.68 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
248 - 585 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3XA
|
2.591 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3XB
|
2.591 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZA
|
3.261 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8WA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8WB
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4Q9ZA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZW |
Type1 |
375 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4Q9ZB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZW |
Type1 |
374 - 704 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4RA5A
|
2.61 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3L0 |
Type1 |
374 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4RA5B
|
2.61 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3L0 |
Type1 |
375 - 701 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4UA
|
1.99 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX6 |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4UB
|
1.99 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX6 |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4WA
|
2.23 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZJ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4WB
|
2.23 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZJ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4TA
|
2.08 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PCG,
ATP
|
Allosteric,
ATPlike
|
204 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4TB
|
2.08 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PCG,
ATP
|
Allosteric,
ATPlike
|
204 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4VA
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
EXZ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4VB
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EXZ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BDLA
|
1.96 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iiio |
No_ligand |
No_ligand |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6C0TA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EE4 |
Type1.5_Front |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMA
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZA
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZB
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZC
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZD
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMB
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3ND |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMC
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
3ND |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMD
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3ND |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFA
|
2.45 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4V |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFB
|
2.45 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
B4V |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFC
|
2.45 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4V |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFD
|
2.45 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4V |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGA
|
2.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4Y |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGB
|
2.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
B4Y |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGC
|
2.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4Y |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGD
|
2.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4Y |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHA
|
3.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5G |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHB
|
3.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHC
|
3.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHD
|
3.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
6E9WA
|
2.96 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0P |
Type1 |
9 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
6E9WB
|
2.96 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
J0P |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26D
|
2.744 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
6 - 399 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
8ZH5A
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26A
|
2.744 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86K |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7A
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiio |
07Q |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7B
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
07Q |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7C
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
07Q |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7D
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
07Q |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SA
|
2.286 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0HD |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SB
|
2.286 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
0HD |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SC
|
2.286 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0HD |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SD
|
2.286 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
0HD |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7JOUA
|
3.318 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ESMA
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ESMB
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
M77 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETKB
|
2.96 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
HFS |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETRB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
Y27 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3D9VB
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
H52 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVCB
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
4KH |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVEB
|
3.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
4KK |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5BMLB
|
2.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
4TW |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5UZJB
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
8UV |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
07R |
Type1.5_Back |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5HVUB
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
65R |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKSB
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
6U1 |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKTB
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
6U2 |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26C
|
2.744 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86K |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJC
|
2.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oiio |
07R |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJB
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJD
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25A
|
2.337 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
86G |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25B
|
2.337 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
86G |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25C
|
2.337 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86G |
Type1 |
13 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25D
|
2.337 |
Inactive |
None‑None |
DFGAsp-rot-none |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
9 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MC
|
2.65 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MD
|
2.65 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QA
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QB
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
No_ligand |
No_ligand |
28 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QC
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QD
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RA
|
3.33 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RC
|
3.33 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PA
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O1V |
Type1 |
27 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PB
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnio |
O1V |
Type1 |
27 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PC
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O1V |
Type1 |
28 - 416 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PD
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
O1V |
Type1 |
26 - 416 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8YB
|
3.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
YEA |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8ZA
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEI |
Type1 |
31 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8ZB
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
YEI |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X92A
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEW |
Type1 |
29 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X92B
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_noio |
YEW |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTA
|
2.93 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTB
|
2.93 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTC
|
2.93 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTD
|
2.93 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
3SG |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9HFPA
|
2.92 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IUI |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4L6QA
|
2.79 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1WU |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4L6QB
|
2.79 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1WU |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RB
|
3.33 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
O1S |
Type1 |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MB
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
O1S |
Type1 |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8XB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
YDW |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8YA
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
YEA |
Type1 |
31 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVA
|
2.586 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVC
|
2.586 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_onno |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVF
|
2.586 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVG
|
2.586 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_innn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVH
|
2.586 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTA
|
2.214 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTC
|
2.214 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTF
|
2.214 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTG
|
2.214 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_innn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTH
|
2.214 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_niio |
5YS |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NB
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6ND
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NF
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NG
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
5YK |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OB
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OD
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_inii |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OE
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OF
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PA
|
2.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_onoo |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PB
|
2.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PC
|
2.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PD
|
2.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QA
|
2.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QB
|
2.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QC
|
2.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QD
|
2.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8A
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
A1H6L |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8B
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H6L |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8C
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H6L |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8D
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
A1H6L |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OG
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1.5_Front |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6ED6B
|
2.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
J0P |
Type1.5_Front |
28 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RD
|
3.33 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_onno |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUA
|
3.02 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUC
|
3.02 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSA
|
2.71 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSB
|
2.71 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSC
|
2.71 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSD
|
2.71 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-none |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
Z8O |
Type1.5_Front |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUB
|
3.02 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUD
|
3.02 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
8XOVA
|
2.55 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
ANP |
ATPlike |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7QA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ACP |
ATPlike |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7RA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
STU |
Type1 |
53 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7SA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
P01 |
Type1 |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NW5A
|
1.94 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2NR |
Type1 |
51 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NW6A
|
1.74 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2NS |
Type1 |
51 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOA
|
2.75 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
45 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOE
|
2.75 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOI
|
2.75 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_onnn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOK
|
2.75 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOC
|
2.75 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
46 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOG
|
2.75 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aanni |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8EQ5A
|
1.8 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
QCT |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8R58A
|
2.31 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
QCT |
Type1 |
49 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYA
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
58 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYB
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
59 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYC
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
61 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYD
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYE
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
64 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYF
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 345 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYG
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYH
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYI
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYJ
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
65 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NUSA
|
2.39 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2NK |
Type1 |
53 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9LA
|
2.15 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
583 |
Type1 |
49 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KA
|
2.55 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KB
|
2.55 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
in-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
1VZOA
|
1.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
24 - 345 |
0 |
None |
S212D |
Ribosomal protein S6 kinase alpha-5 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G77A
|
2.499 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
Allosteric,
ATPlike
|
51 - 349 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G77B
|
2.499 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
Allosteric,
ATPlike
|
51 - 349 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G76B
|
3.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
51 - 349 |
0 |
SEP232 |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G78A
|
2.5 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ANP |
ATPlike |
51 - 349 |
0 |
None |
S232E |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G78B
|
2.5 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ANP |
ATPlike |
51 - 349 |
0 |
None |
S232E |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G76A
|
3.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
ATPlike,
Allosteric
|
51 - 349 |
0 |
SEP232 |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLPA
|
2.79 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
none-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
72B |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L3JA
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 375 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L3LA
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 375 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N91A
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1RJ |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N91B
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1RJ |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N93A
|
2.74 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
1SK |
Type1 |
87 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N93B
|
2.74 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1SK |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A62A
|
2.35 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
STU |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WE4A
|
1.995 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF5A
|
2.099 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FZ8 |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF6A
|
2.031 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FZ9 |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L45A
|
2.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L42A
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
5FI |
Type1 |
84 - 417 |
0 |
None |
S403E,A404E,N405Q,Q406E,V407M,L409R,G410D,T412E,V414I,P416D,S417W |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L46A
|
3.01 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
80 - 417 |
0 |
TPO412 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF8A
|
1.975 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
F76 |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF9A
|
2.035 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FS7 |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L43A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412A |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L44A
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412A |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLOA
|
2.527 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3T3 |
Type1 |
85 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A60A
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
STU |
Type1 |
85 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A61A
|
3.43 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
STU |
Type1 |
87 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF7A
|
1.85 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
FS9 |
Type1 |
83 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLOB
|
2.527 |
Inactive |
None‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
STU |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A60B
|
2.8 |
Inactive |
None‑None |
DFGAsp-rot-out |
none-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
STU |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
2R5TA
|
1.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
ANP |
ATPlike |
82 - 378 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
3HDMA
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
MMG |
Type1 |
81 - 378 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
3HDNA
|
3.1 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
GMG |
Type1 |
82 - 374 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
7PUEA
|
2.506 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
86H |
Type1 |
82 - 376 |
0 |
None |
R192A,S422D |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4A
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4B
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4C
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4D
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4E
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 372 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4F
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32C
|
ST32C_HUMAN
|
AF-Q86UX6-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
No_ligand |
No_ligand |
85 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase 32C |
|
AGC
|
STK38
|
STK38_HUMAN
|
6BXIA
|
2.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
82 - 414 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
|
AGC
|
STK38
|
STK38_HUMAN
|
6BXIB
|
2.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
83 - 414 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4C3PD
|
2.69 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_nooo |
ACP |
ATPlike |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8GUWA
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP |
ATPlike |
506 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8GUWB
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
ADP |
ATPlike |
507 - 390 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8GUWC
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ADP |
ATPlike |
506 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DPVA
|
2.285 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
5DN,
SKE
|
Allosteric,
Type1
|
127 - 389 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DR6A
|
2.534 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
5E1,
SKE
|
Allosteric,
Type1
|
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTWA
|
3.302 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
ZZL |
Type1 |
128 - 389 |
0 |
None |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3E5AA
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
125 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2NP8A
|
2.25 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
CC3 |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4BYIA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
FH3 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ONEA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nooo |
9YQ |
Type1 |
127 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DT0A
|
2.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
SKE |
Type1 |
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UODA
|
2.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
0C3 |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UP2A
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
0C8 |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEAA
|
2.45 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
NHI |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AAFA
|
2.78 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
NL4 |
Type1 |
126 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AAGA
|
2.85 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
6F2 |
Type1 |
127 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6GRAA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
F8Z |
Type1.5_Front |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4BN1A
|
2.499 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
126 - 388 |
0 |
TPO287,TPO288 |
V174M |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1MQ4A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DNRA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ATP |
ATPlike |
126 - 390 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DT3A
|
2.33 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ATP |
ATPlike |
127 - 390 |
0 |
TPO287 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1OL7A
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
127 - 390 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5G15A
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ACP |
ATPlike |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2DWBA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPFA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ACP |
ATPlike |
128 - 392 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DRDA
|
2.13 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
ATP |
ATPlike |
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEEA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
124 - 394 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPIA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ANP |
ATPlike |
104 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4CEGA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1OL6A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ATP |
ATPlike |
128 - 388 |
0 |
None |
D274N |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPLA
|
1.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ANP,
R7D
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPLB
|
1.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ANP,
R7D
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPMA
|
1.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
AMP,
R74
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPMB
|
1.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
AMP,
R74
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORLA
|
1.69 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A4W
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORNA
|
2.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5E
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OROA
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORPA
|
2.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5K
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORRA
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5Q
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORSA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5W
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORTA
|
2.56 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5Z
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORVA
|
1.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A65
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORWA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6E
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORXA
|
1.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORYA
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
AY4
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORZA
|
1.92 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6W
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS0A
|
1.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6Z
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS1A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A7H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS2A
|
1.92 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
ADP,
A7K
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS3A
|
1.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A7N
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS4A
|
1.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A8H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS6A
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A7Q
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OSEA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A98
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OSFA
|
1.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A9E
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OSDA
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A9B
|
ATPlike,
Allosteric
|
125 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS5A
|
1.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A8K
|
ATPlike,
Allosteric
|
125 - 392 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R49A
|
2.209 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
JSB
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4AA
|
1.937 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JRT
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4BA
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JSN
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4CA
|
2.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JRQ
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4DA
|
2.009 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JRW
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9SUYA
|
2.27 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
ADP,
A1JQV
|
ATPlike,
Allosteric
|
8 - 389 |
0 |
None |
D274N |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8OF5A
|
1.97 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ADP,
MPO
|
ATPlike,
Allosteric
|
126 - 390 |
0 |
None |
C290A,N332A,Q335A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C14A
|
1.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ADP,
T5L,
T0L
|
ATPlike,
Allosteric,
Allosteric
|
126 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C15A
|
2.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
T4C,
T5L
|
ATPlike,
Allosteric,
Allosteric
|
126 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1FA
|
1.924 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
T5L,
T2O
|
ATPlike,
Allosteric,
Allosteric
|
126 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1IA
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
T1L,
T5L
|
ATPlike,
Allosteric,
Allosteric
|
126 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DN3A
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
5DN,
ATP
|
Allosteric,
ATPlike
|
125 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1EA
|
2.798 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
T0X,
ATP
|
Allosteric,
ATPlike
|
127 - 388 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DT4A
|
2.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
5DN,
ATP
|
Allosteric,
ATPlike
|
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1MA
|
2.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
T4X,
ADP
|
Allosteric,
ATPlike
|
127 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DOSA
|
2.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
5DN,
ATP
|
Allosteric,
ATPlike
|
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DR2A
|
2.46 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
5E1,
ATP
|
Allosteric,
ATPlike
|
128 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1DA
|
2.115 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
T2F,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1GA
|
1.96 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
T3I,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1HA
|
2.233 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
T3U,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1KA
|
2.43 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
T4O,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8SSPA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PDO,
627
|
Allosteric,
Type1
|
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPEA
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8NA
|
3.135 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioo |
No_ligand |
No_ligand |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8NB
|
3.135 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
No_ligand |
No_ligand |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8NC
|
3.135 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8ND
|
3.135 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8JG8A
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
C74 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3HA6A
|
2.36 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2JZ |
Type1 |
125 - 388 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3MYGA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
EML |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3VAPA
|
2.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0FY |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1CA
|
3.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
L0C |
Type1 |
127 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1DA
|
2.97 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0D |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1EA
|
2.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0E |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1FA
|
2.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0F |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1GA
|
2.71 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0G |
Type1 |
127 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ZANA
|
2.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
9A6 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4O0SA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADN |
Type1 |
126 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2XNGA
|
2.605 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
A0H |
Type1 |
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JAJA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
XU1 |
Type1 |
125 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2X6DA
|
2.796 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
X6D |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2X6EA
|
3.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
YM4 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZS0A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
4QV |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6I2UA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
COA |
Type1 |
127 - 391 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2XRUA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
400 |
Type1 |
126 - 389 |
0 |
None |
T288E |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO4A
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
0C0 |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO5A
|
2.701 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
0BX |
Type1 |
124 - 390 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UP7A
|
3.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
0C9 |
Type1 |
124 - 387 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEBA
|
3.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
NHJ |
Type1 |
125 - 388 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEDA
|
3.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
NHU |
Type1 |
124 - 388 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JBOA
|
2.493 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
WPH |
Type1 |
126 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3NRMA
|
3.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
NRM |
Type1 |
126 - 388 |
0 |
None |
T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3R21A
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
D36 |
Type1 |
127 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AADA
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5GX |
Type1 |
127 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2XNEA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ASH |
Type1 |
127 - 388 |
0 |
None |
D274N |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DR9A
|
2.47 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
SKE,
5E2
|
Type1,
Allosteric
|
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3M11A
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
AKI |
Type1.5_Front |
126 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JBPA
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
YPH |
Type1.5_Front |
126 - 390 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8MA
|
1.853 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
CJ5 |
Type1 |
125 - 390 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8PR7D
|
2.76 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-none |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
ADP |
ATPlike |
126 - 388 |
0 |
None |
D274N,C290A,N332A,Q335A,T347A,D350A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9QVZA
|
2.39 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
ADP,
LI
|
ATPlike,
Allosteric
|
124 - 390 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4C3PA
|
2.69 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ACP |
ATPlike |
125 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6DA
|
2.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ANP |
ATPlike |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ODTA
|
2.021 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
ADP |
ATPlike |
126 - 392 |
0 |
None |
D274N,C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OBJA
|
2.901 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
ATP,
9QK
|
ATPlike,
Allosteric
|
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9GUCA
|
2.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
ADP,
AMP
|
ATPlike,
Allosteric
|
124 - 391 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8JF4A
|
2.893 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
C0N |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8JMXA
|
2.95 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnno |
E47 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7AYIA
|
2.86 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
S9K |
Type1 |
125 - 392 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J4ZB
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
626 |
Type1 |
126 - 395 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4O0WA
|
2.6 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nioo |
ADN |
Type1 |
125 - 391 |
0 |
None |
H254Y |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0ZA
|
2.92 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
45B |
Type1 |
128 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DHFA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnoo |
0K6 |
Type1 |
128 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DHFB
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnoo |
0K6 |
Type1 |
128 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4PRJA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnoo |
2VU |
Type1 |
125 - 388 |
0 |
None |
K124A,Q154N,A203S,R251K,T287A,T288A,E336D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AAEA
|
3.11 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
7HD |
Type1 |
126 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4O0UA
|
2.6 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ADN |
Type1 |
126 - 391 |
0 |
None |
H254R |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UZDA
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
QMN |
Type1.5_Front |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UZDB
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
QMN |
Type1.5_Front |
125 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UYNA
|
1.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
Y3M |
Type1.5_Front |
125 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4C3RA
|
2.79 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ACP |
ATPlike |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C83B
|
2.55 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ACP |
ATPlike |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5L8JA
|
1.68 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ADP |
ATPlike |
126 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5L8KA
|
1.79 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ADP |
ATPlike |
126 - 392 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5L8LA
|
1.67 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
ADP |
ATPlike |
126 - 389 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8PR7A
|
2.76 |
Inactive |
DFGinter‑None |
DFGAsp-rot-none |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ADP |
ATPlike |
124 - 389 |
0 |
None |
D274N,C290A,N332A,Q335A,T347A,D350A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6XKAA
|
2.65 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
No_ligand |
No_ligand |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVA
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
ZZL |
Type1 |
125 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVB
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ZZL |
Type1 |
126 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVC
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ZZL |
Type1 |
126 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVD
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
ZZL |
Type1 |
125 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5EW9A
|
2.181 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
5VC |
Type1 |
127 - 390 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C2RA
|
1.96 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
EG7 |
Type1 |
128 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C2TA
|
1.73 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
EGJ |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W16A
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
P9J |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J50A
|
3.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
627 |
Type1 |
128 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J50B
|
3.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
627 |
Type1 |
128 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZTRA
|
2.85 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
4RJ |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6Z4YA
|
2.25 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
Q7Q |
Type1 |
124 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPGA
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
35R |
Type1 |
127 - 387 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPGD
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nooo |
35R |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8SSOA
|
1.97 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
627 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8SSOD
|
1.97 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
627 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1MUOA
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
ADN |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J4ZA
|
2.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
626 |
Type1 |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UNZA
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BZ |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UNZB
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BZ |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO6A
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BY |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO6B
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BY |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOHA
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C4 |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOHB
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C4 |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOJA
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C5 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOJB
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C5 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOKA
|
2.951 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C6 |
Type1 |
125 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOKB
|
2.951 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C6 |
Type1 |
125 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOLA
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C7 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOLB
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C7 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3FDNA
|
1.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
MMH |
Type1 |
126 - 394 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3K5UA
|
2.35 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
PFQ |
Type1 |
126 - 394 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JBQA
|
2.3 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
VX6 |
Type1 |
126 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3LAUA
|
2.1 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
OFI |
Type1 |
125 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UZHA
|
2.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
JVE |
Type1 |
125 - 392 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0YA
|
2.5 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
48B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H10A
|
2.2 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
97B |
Type1 |
124 - 391 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H10B
|
2.2 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
97B |
Type1 |
125 - 391 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H10D
|
2.2 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
97B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3P9JA
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
P9J |
Type1 |
126 - 388 |
0 |
None |
T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W10A
|
2.7 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
RO9 |
Type1 |
126 - 388 |
0 |
None |
T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3R22A
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
D37 |
Type1 |
126 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9KDSA
|
2.5 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
A1EFT |
Type1 |
126 - 391 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCA
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
127 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCB
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
125 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCC
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
125 - 393 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCD
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
127 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCE
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
127 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCF
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
126 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7FICA
|
2.32 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
5YZ |
Type1 |
127 - 391 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9BZGA
|
1.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
OG0 |
Type1 |
127 - 388 |
0 |
TPO288 |
C290A,C393S |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9BZLB
|
1.81 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
OGR |
Type1 |
127 - 388 |
0 |
TPO288 |
C290A,C393S |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9KS6A
|
2.75 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-na |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
A1EG1 |
Type1 |
127 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZTQA
|
2.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
4RM |
Type1.5_Back |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZTSA
|
2.9 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
4RK |
Type1.5_Back |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3EFWA
|
2.29 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
AK8 |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3EFWB
|
2.29 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
AK8 |
Type1.5_Front |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O50A
|
2.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
LJE |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O50B
|
2.0 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LJE |
Type1.5_Front |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6HJJA
|
2.13 |
Inactive |
DFGinter‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
G7T |
Type1.5_Front |
127 - 393 |
0 |
None |
L210C,C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6EA
|
2.1 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
HPM |
Type1.5_Back |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPJA
|
2.1 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
ANP |
ATPlike |
104 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPHA
|
2.14 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
ANP |
ATPlike |
7 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JAIA
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
XU2 |
Type1 |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7AYHA
|
2.8 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
S9H |
Type1 |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7O2VA
|
3.1 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
V0K |
Type1 |
117 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O51A
|
3.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
LJF |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6HJKA
|
2.4 |
Inactive |
DFGout‑None |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
G7W |
Type1.5_Front |
127 - 391 |
0 |
None |
L210C,C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C83A
|
2.55 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ACP |
ATPlike |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WQEA
|
2.5 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-none |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ADP,
ADP,
ADP
|
ATPlike,
ATPlike,
ATPlike
|
127 - 388 |
0 |
None |
S155R |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OBRA
|
2.62 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
9QT,
SKE
|
Allosteric,
Type1
|
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CC
|
2.45 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
N15 |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CE
|
2.45 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
N15 |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2X81A
|
2.91 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ZZL |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W18A
|
2.5 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
N13 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W18B
|
2.5 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
N13 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4B0GA
|
2.5 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VEK |
Type1 |
126 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4BYJA
|
2.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FH5 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0ZB
|
2.92 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
45B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0ZC
|
2.92 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
45B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3COHA
|
2.7 |
Inactive |
None‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
83H |
Type1 |
128 - 388 |
0 |
None |
K124A,Q154N,A203S,R251K,T287A,T288A,E336D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3COHB
|
2.7 |
Inactive |
None‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
83H |
Type1 |
128 - 388 |
0 |
None |
K124A,Q154N,A203S,R251K,T287A,T288A,E336D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3QBNA
|
3.5 |
Inactive |
None‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
E9Z |
Type1 |
126 - 388 |
0 |
None |
V279C,C290S,C393S |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CA
|
2.45 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
N15 |
Type1.5_Back |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CG
|
2.45 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
N15 |
Type1.5_Back |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6EB
|
2.1 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnni |
HPM |
Type1.5_Front |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKB
|
AURKB_HUMAN
|
4AF3A
|
2.75 |
Inactive |
DFGinter‑None |
DFGAsp-rot-none |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VX6 |
Type1 |
70 - 338 |
0 |
None |
None |
Aurora kinase B |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
9ESAAAA
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
32 - 306 |
0 |
None |
R195A,R196A,K197A |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
9ESABBB
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
32 - 306 |
0 |
None |
R195A,R196A,K197A |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
6GR9A
|
2.25 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
37 - 305 |
0 |
TPO39,TPO198 |
None |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
6GR8A
|
1.75 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
F8Z |
Type1.5_Front |
36 - 303 |
0 |
TPO39,TPO198 |
None |
Aurora kinase C |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG9A
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ATP |
ATPlike |
10 - 314 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG9B
|
2.4 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
ATP |
ATPlike |
14 - 314 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FGBA
|
2.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
10 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG8A
|
2.2 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-none |
none-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
ATP |
ATPlike |
10 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG8B
|
2.2 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-none |
none-out |
nonTYR |
APEdihe_aaino |
APEdist_nnno |
ATP |
ATPlike |
14 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6QP5A
|
1.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
13 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T28AAA
|
1.55 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
M92 |
Type1 |
12 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
8BFSA
|
1.95 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QNR |
Type1 |
12 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
8BFMA
|
1.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QI6,
QI6
|
Type1,
Type3
|
12 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T6FA
|
1.97 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MMW |
Type1 |
12 - 329 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T6FB
|
1.97 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MMW |
Type1 |
12 - 329 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T29AAA
|
1.484 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
M8Z |
Type1 |
12 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
2JC6A
|
2.3 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QPP |
Type1 |
11 - 313 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
2JC6C
|
2.3 |
Inactive |
None‑None |
DFGAsp-rot-none |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QPP |
Type1 |
11 - 313 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1G
|
KCC1G_HUMAN
|
2JAMA
|
1.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
J60 |
Type1 |
18 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1G |
|
CAMK
|
CAMK1G
|
KCC1G_HUMAN
|
2JAMB
|
1.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
J60 |
Type1 |
16 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1G |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
7 - 274 |
0 |
None |
Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJPB
|
2.56 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
7 - 273 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJTA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJRA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6X5QA
|
2.14 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL1A
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL1B
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL2A
|
2.56 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UISA
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 273 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6W4OO
|
4.8 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 301 |
0 |
None |
K42M |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6W4PH
|
6.6 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 301 |
0 |
None |
K42M |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
3SOAA
|
3.55 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DB8 |
Type1 |
7 - 474 |
0 |
None |
K42M,D135N,T306V |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2D
|
D6R938_HUMAN
|
8USOA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 475 |
0 |
None |
D364C |
calcium/calmodulin-dependent protein kinase |
|
CAMK
|
CAMK2D
|
D6R938_HUMAN
|
8USOC
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 477 |
0 |
None |
D364C |
calcium/calmodulin-dependent protein kinase |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
2WELA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
K88 |
Type1 |
10 - 316 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK4
|
KCC4_HUMAN
|
2W4OA
|
2.17 |
Inactive |
None‑None |
DFGAsp-rot-out |
none-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
DKI |
Type1 |
34 - 337 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type IV |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CCFA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H1N |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CCFB
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H1N |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OOPA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
5 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3JVSA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AGY |
Allosteric |
2 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9PA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
77A |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3PA3A
|
1.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C70 |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3PA4A
|
1.59 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C72 |
Type1 |
6 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3PA5A
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C73 |
Type1 |
3 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4JIKA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1KO |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDJA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDJ |
Type1 |
8 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDJB
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDJ |
Type1 |
9 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDKA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDK |
Type1 |
3 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
6FC8A
|
1.61 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D4Q |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
6FCFA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D58 |
Type1 |
9 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
6FCKA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D4Z |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM5A
|
2.03 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM5 |
Type1 |
8 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM6A
|
2.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM6 |
Type1 |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2HXQA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
373 |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2HY0A
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
306 |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OORA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
3 - 283 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJMA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TW2 |
Type1 |
5 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUJA
|
2.299 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BYL |
Type1 |
9 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9NA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
76A |
Type1.5_Back |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTLA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H0K |
Type1.5_Back |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2CN5A
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ADP |
ATPlike |
209 - 504 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WB
|
3.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WD
|
3.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WF
|
3.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WH
|
3.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XK9A
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
XK9 |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCFA
|
1.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
YCF |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2W0JA
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ZAT |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2W7XA
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
D1A |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCQA
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
UPX |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCSA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
NXP |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YIQA
|
1.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
YIQ |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YIRA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YIR |
Type1 |
210 - 509 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCRA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
HCW |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2CN8A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_ooon |
DBQ |
Type1 |
212 - 503 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTCA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
VGM |
Type1 |
211 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTDA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaino |
APEdist_oooo |
ZZK |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTIA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
WTI |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTJA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
WTJ |
Type1 |
209 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XBJA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
XBJ |
Type1 |
211 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XM8A
|
3.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
B4W |
Type1 |
211 - 503 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XM9A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LWH |
Type1 |
211 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9RA
|
2.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
RU5 |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9SA
|
2.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
RU9 |
Type1 |
211 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9TA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A9T |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9UA
|
2.48 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A9U |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDAA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
VFB |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDBA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
ODO |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDCA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ODH |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDDA
|
2.67 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
Z0O |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDEA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CWS |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDFA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
H3R |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDGA
|
2.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
P3J |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDHA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
WVI |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDIA
|
2.32 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HAU |
Type1 |
210 - 515 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDJA
|
3.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
Z2M |
Type1 |
211 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDKA
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
RQQ |
Type1 |
211 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YITA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
YIT |
Type1.5_Back |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6UA
|
3.0 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
out-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
89 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6UB
|
3.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
89 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WA
|
3.25 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WC
|
3.25 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WE
|
3.25 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WG
|
3.25 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1WVYA
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STU |
Type1 |
4 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9INVA
|
1.61 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
HCC |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9INWA
|
1.52 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1L2V |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2W4JA
|
1.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1IG1A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 294 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKKA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 293 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKLA
|
1.62 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 294 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3EH9A
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3EHAA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3F5GA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3F5UA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3DFCB
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
Q23K |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU4A
|
1.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU5A
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU6A
|
1.49 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU7A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4PF4A
|
1.13 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 275 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PC
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
2 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV1A
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6IN4A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKSA
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKTA
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKTB
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iooo |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3DGKA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
Q23K |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2XZSA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 312 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2XZSB
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 302 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6QMOA
|
1.87 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
4 - 302 |
0 |
None |
S289E,S308A |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6QN4A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
S289E,S308E |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4UV0A
|
2.49 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 302 |
0 |
None |
S289C |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2X0GA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
3 - 320 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6FHAA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
4 - 302 |
0 |
None |
S289A,S308A |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1WVXA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
BD4 |
Type1 |
2 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2YAKA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
OSV |
Type1 |
2 - 278 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUTA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2AN |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUVA
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
AGI |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUXA
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KMP |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUZA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
GEN |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV0A
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
47X |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV2A
|
1.502 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KMP |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV3A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KMP |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV4A
|
1.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
GEN |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6AARA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
9TF |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
7CCWA
|
1.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STL |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE6A
|
1.701 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8KZ |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE7A
|
1.849 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3RL |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE8A
|
1.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
P5O |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9INXA
|
1.72 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1L2W |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1P4FA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
86Q |
Type1 |
2 - 293 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9N1TA
|
1.43 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BU8 |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9N2MA
|
1.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BVM |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9N2OA
|
1.49 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BVL |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4YO4A
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
4FT |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4YPDA
|
1.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
DKG |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9DUBA
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BB7 |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9O73A
|
1.49 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
86Q |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9MIUA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BLJ |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU8A
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3GU |
Type1 |
2 - 277 |
0 |
None |
L93G |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GUBA
|
1.71 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
GUB |
Type1 |
2 - 277 |
0 |
None |
L93G |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9DUEA
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BB6,
BO3
|
Type1,
Allosteric
|
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUUA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LU2 |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUWA
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
QUE |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUYA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MRI |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
7CCUA
|
1.649 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STL |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
7CCVA
|
1.753 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
PIT |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE5A
|
1.803 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
EZE |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3ZXTA
|
2.65 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ACP |
ATPlike |
7 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PB
|
2.65 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
57 - 275 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PD
|
2.65 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
56 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKA
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKB
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 325 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKC
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKD
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 325 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKE
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 324 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKF
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKG
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 324 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKH
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 315 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
6PAWF
|
2.953 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 327 |
0 |
None |
S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6NB
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6OA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6OB
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 277 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
3BHYA
|
1.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
7CP |
Type1 |
9 - 283 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
3BQRA
|
1.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
4RB |
Type1 |
9 - 284 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6NA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
U7E |
Type1 |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
2J90A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
IZA |
Type1 |
5 - 278 |
0 |
SEP50,TPO265 |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
2J90B
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
IZA |
Type1 |
12 - 280 |
0 |
SEP50,TPO265 |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7F3GB
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RXT |
Type1 |
383 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYRA
|
2.206 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 701 |
0 |
None |
P675L |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYRB
|
2.206 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 700 |
0 |
None |
P675L |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYQA
|
2.141 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 701 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYQB
|
2.141 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 700 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KXWA
|
3.002 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XBD |
Type1 |
382 - 648 |
0 |
TPO484 |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KXWB
|
3.002 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XBD |
Type1 |
382 - 649 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
HUNK
|
HUNK_HUMAN
|
AF-P57058-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 328 |
0 |
None |
None |
Hormonally up-regulated neu tumor-associated kinase |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4A
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 351 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4B
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 351 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4C
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
48 - 351 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4D
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 349 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4E
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 353 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4F
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 353 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4G
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 348 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4H
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 358 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4I
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 347 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4J
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 350 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4K
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 348 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4L
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 354 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NY3A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ADP |
ATPlike |
46 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2PZYD
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnoo |
No_ligand |
No_ligand |
43 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
4TYHA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 400 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2OZAA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 390 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAA
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-none |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 399 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAC
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 397 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAE
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 394 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAG
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 397 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1KWPA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
46 - 385 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1KWPB
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
44 - 378 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2ONLC
|
4.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oooo |
No_ligand |
No_ligand |
46 - 393 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2ONLD
|
4.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
No_ligand |
No_ligand |
46 - 393 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6A
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6B
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6C
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6D
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6E
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6F
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3FPMA
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
793 |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2P3GX
|
3.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
F10 |
Type1 |
45 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3FYJX
|
3.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B97 |
Type1 |
45 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3FYKX
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B98 |
Type1 |
45 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
7NRYX
|
3.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B97 |
Type1 |
45 - 366 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBOA
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
P4O |
Type1 |
44 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPL
|
3.31 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
9R59A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1JH4 |
Type1 |
48 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NXKD
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnoo |
STU |
Type1 |
43 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CB
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CC
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CD
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CE
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CF
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CG
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CH
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 343 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CI
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 343 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CJ
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 343 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CK
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CL
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XA
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B97,
MW8
|
Type1,
Allosteric
|
44 - 330 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XD
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
B97,
MW8
|
Type1,
Allosteric
|
44 - 331 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XE
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
B97,
MW8
|
Type1,
Allosteric
|
45 - 329 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XF
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B97,
MW8
|
Type1,
Allosteric
|
45 - 329 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
AF-Q16644-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
No_ligand |
No_ligand |
35 - 312 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
6C9DA
|
2.499 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
53 - 795 |
0 |
None |
T215E,K761S,R764S |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
6C9DB
|
2.499 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
53 - 795 |
0 |
None |
T215E,K761S,R764S |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKA
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
No_ligand |
No_ligand |
55 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKB
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
53 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKC
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
53 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKD
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKE
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKF
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKG
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
No_ligand |
No_ligand |
55 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKH
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECB
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECD
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5EAKB
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
24R |
Type1 |
51 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECC
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5EAKA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nioo |
24R |
Type1 |
47 - 362 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
8TXYA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
SJ0 |
Type1 |
48 - 363 |
0 |
None |
I59L,K66V,V81I,L97I,V113I,M129T,S133K,G134N,S197G |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
8TXYB
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
SJ0 |
Type1 |
47 - 363 |
0 |
None |
I59L,K66V,V81I,L97I,V113I,M129T,S133K,G134N,S197G |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ7A
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6Z2 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ8A
|
3.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
6Z5 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ8B
|
3.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6Z5 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ7B
|
3.2 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6Z2 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOIA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
X3Q |
Type1 |
51 - 368 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E,V205K |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOKA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
X5N |
Type1 |
51 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E,V205K |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOKB
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
X5N |
Type1 |
51 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E,V205K |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
7P1LA
|
1.95 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
V5E |
Type1 |
50 - 365 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9YR9A
|
2.402 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooi |
A1CZY |
Type1 |
49 - 366 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9ZZWA
|
2.76 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1C86 |
Type1 |
49 - 366 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9VFOA
|
2.5 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooi |
A1ER0 |
Type1 |
51 - 368 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9VGRA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooi |
A1ER9 |
Type1 |
51 - 368 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9VIRA
|
2.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooi |
A1ESF |
Type1 |
51 - 368 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9YSQA
|
2.4 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1CZY |
Type1 |
51 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9YSQB
|
2.4 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1CZY |
Type1 |
50 - 366 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOJA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooi |
X5I,
BEZ
|
Type1,
Allosteric
|
50 - 370 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9YR9B
|
2.402 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1CZY |
Type1 |
49 - 366 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
9ZZWB
|
2.76 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
in-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1C86 |
Type1 |
49 - 366 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
2QNJA
|
2.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
No_ligand |
No_ligand |
44 - 366 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
2QNJB
|
2.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
No_ligand |
No_ligand |
44 - 367 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
3FE3A
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_iooo |
No_ligand |
No_ligand |
50 - 366 |
0 |
None |
T211A,S215A |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
3FE3B
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_iooo |
No_ligand |
No_ligand |
50 - 366 |
0 |
None |
T211A,S215A |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOHA
|
2.15 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
No_ligand |
No_ligand |
48 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
7P1LB
|
1.95 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
V5E |
Type1 |
50 - 365 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOHB
|
2.15 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
X4W |
Type1 |
48 - 370 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOLA
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
X4H |
Type1 |
51 - 370 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOLB
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnni |
X4H |
Type1 |
50 - 367 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
8XFLA
|
3.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 370 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
5ES1A
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
5RC |
Type1 |
54 - 370 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
8XFLB
|
3.0 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 370 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4BL1A
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ANP |
ATPlike |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TX3A
|
2.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
7MY |
Type1 |
1 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWUA
|
2.603 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
No_ligand |
No_ligand |
1 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWUB
|
2.603 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
No_ligand |
No_ligand |
1 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWZA
|
2.631 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
45R |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
6GVXB
|
2.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
TAK |
Type1 |
1 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4BKZA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1WS |
Type1 |
2 - 334 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5M5AA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
KSA |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAGA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
7KC |
Type1 |
3 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAHA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
7KD |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
9F31A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H9M |
Type1 |
1 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2TA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nooi |
3I7 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2VB
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
45R |
Type1 |
2 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WA
|
1.92 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WB
|
1.92 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WD
|
1.92 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnii |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMRA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
QBB |
Type1 |
6 - 333 |
0 |
None |
T167A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TVTA
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
7LV |
Type1.5_Back |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWLA
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
H91 |
Type1.5_Back |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAFA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
XIN |
Type1.5_Back |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMPB
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
5QM |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMQA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
B5S |
Type1.5_Back |
5 - 333 |
0 |
None |
T167A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5IHCA
|
2.14 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6BB |
Type1 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWYA
|
2.91 |
Inactive |
DFGin‑None |
DFGAsp-rot-none |
out-out |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
7LY |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAIA
|
2.15 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5U5 |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4IXPA
|
2.749 |
Inactive |
DFGinter‑BABtrans |
DFGAsp-rot-none |
out-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
2 - 335 |
0 |
None |
K40R,D150A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMTA
|
1.98 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
47W |
Type1 |
3 - 333 |
0 |
None |
N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMUA
|
2.02 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
0V0 |
Type1 |
3 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5K00A
|
1.77 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
out-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6PV |
Type2 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
6VXRA
|
2.1 |
Inactive |
None‑None |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F7D |
Type1 |
1 - 332 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWYB
|
2.91 |
Inactive |
None‑None |
DFGAsp-rot-in |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7LY |
Type1 |
2 - 332 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TX3B
|
2.9 |
Inactive |
None‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
7MY |
Type1 |
1 - 334 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
2HW6A
|
2.5 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
39 - 376 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
2HW6B
|
2.5 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
40 - 375 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
5WVDA
|
3.0 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7UX |
Type1 |
41 - 375 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
5WVDB
|
3.0 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7UX |
Type1 |
41 - 374 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
8XFMA
|
2.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
A1LU6 |
Type1 |
73 - 372 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2HW7A
|
2.71 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
STU |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJ5A
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4G |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJEA
|
3.36 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4A |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJHA
|
3.6 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ET8 |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJWA
|
3.38 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
FYV |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJYA
|
3.05 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4J |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CK3A
|
2.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F67 |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CK6A
|
3.32 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
N45 |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CKIA
|
2.95 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
FZJ |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
9HRCA
|
3.161 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
A1IWO |
Type1 |
72 - 375 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2AC5A
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
72 - 370 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
8P9BA
|
2.59 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
X8K |
Type1 |
72 - 369 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2AC3A
|
2.1 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
No_ligand |
No_ligand |
72 - 369 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6JLRA
|
2.901 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BV9 |
Type1 |
72 - 369 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MYLK4
|
MYLK4_HUMAN
|
2X4FA
|
2.67 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
16X |
Type1 |
80 - 373 |
0 |
None |
None |
Myosin light chain kinase family member 4 |
|
CAMK
|
MYLK4
|
MYLK4_HUMAN
|
2X4FB
|
2.67 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
16X |
Type1 |
81 - 370 |
0 |
None |
None |
Myosin light chain kinase family member 4 |
|
CAMK
|
OBSCN-2
|
OBSCN_HUMAN
|
AF-Q5VST9-K2A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioi |
No_ligand |
No_ligand |
7664 - 7932 |
0 |
None |
None |
Obscurin |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5RC
|
3.52 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TC
|
3.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TG
|
3.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TK
|
3.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TO
|
3.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKC
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKG
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKK
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKO
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8XYAC
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8XYBC
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5MC
|
3.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5PC
|
3.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5PG
|
3.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QC
|
4.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QG
|
4.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QK
|
4.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QO
|
4.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JB
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JC
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JD
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RBLA
|
2.55 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3O7 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RC2A
|
2.096 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3O8 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RC3A
|
2.338 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3OA |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RC4A
|
2.651 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3OK |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4I41A
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
MIX,
MIX
|
Type1,
Allosteric
|
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7OOXA
|
1.97 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5TOEA
|
2.301 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7GK |
Type1 |
34 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5TELA
|
2.214 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7AJ |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KGGA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6SO |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4MBIA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
26K |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2O63A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MYC |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBTA
|
2.23 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0F9 |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBXA
|
2.03 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0FO |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XIYA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIY |
Type1 |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3DCVA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
55E |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3WE8A
|
1.954 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RUI |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4GW8A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3RA |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R0HA
|
1.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8UB |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R0QA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XGB |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R1KA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XHI |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4RA
|
2.13 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MQ |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4XA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MT |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N5LA
|
1.97 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8NZ |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6KZIA
|
2.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RTX |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4IAAA
|
2.85 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RTZ |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4XH6A
|
2.04 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HUL |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
8X72A
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
ANP |
ATPlike |
37 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2OU7A
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
ANP |
ATPlike |
37 - 328 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2V5QA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
No_ligand |
No_ligand |
39 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2V5QB
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
No_ligand |
No_ligand |
39 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2YACA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
937 |
Type1 |
39 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
3KB7A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iooo |
071 |
Type1 |
39 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4A4LA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
939 |
Type1 |
39 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4A4OA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
664 |
Type1 |
39 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8BA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCP |
Type1 |
37 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8BB
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiio |
A1JCP |
Type1 |
37 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8CA
|
2.243 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
38 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8CB
|
2.243 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
38 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4J52A
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
1J3 |
Type1 |
38 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4J53A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
1J4 |
Type1 |
38 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2RKUA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
37 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
8BJTA
|
2.188 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iooo |
8X7 |
Type1 |
39 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
3THBA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
3TA |
Type1 |
42 - 328 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2OWBA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
626 |
Type1 |
37 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
3FC2A
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
IBI |
Type1 |
37 - 329 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9D0PA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
8X7 |
Type1 |
37 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1WAAA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCP |
Type1 |
38 - 334 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1WBBB
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCP |
Type1 |
38 - 325 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1XA
|
2.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
39 - 334 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1XB
|
2.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
39 - 326 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1YAAA
|
2.602 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCQ |
Type1 |
38 - 334 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1YBBB
|
2.602 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCQ |
Type1 |
38 - 325 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
5TA6A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
79D |
Type1 |
37 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
5TA8A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
79C |
Type1 |
37 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I5MA
|
1.801 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
R78 |
Type1 |
71 - 354 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I5PA
|
1.738 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
1D1 |
Type1 |
71 - 354 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I6BA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
11G |
Type1 |
71 - 355 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I6FA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
1C7 |
Type1 |
71 - 355 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I6HA
|
1.91 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
1C8 |
Type1 |
71 - 355 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
9O63A
|
2.26 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1CAD |
Type1 |
2 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
3COKA
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-none |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
2 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
3COKB
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
2 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
9Y9BA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1CTX |
Type1 |
2 - 267 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
9Y9NA
|
1.81 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1CTV |
Type1 |
4 - 267 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
4JXFA
|
2.4 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
631 |
Type1 |
4 - 267 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
4YURA
|
2.65 |
Inactive |
DFGin‑None |
DFGAsp-rot-none |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
4J7 |
Type1 |
5 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9FA
|
2.924 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R34,
STU
|
Allosteric,
Type1
|
22 - 558 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7JIJA
|
5.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
22 - 559 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9GA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R93,
STU
|
Allosteric,
Type1
|
22 - 558 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9HA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R34,
STU
|
Allosteric,
Type1
|
22 - 558 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
AF-Q13131-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 287 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7JHHA
|
3.92 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
22 - 559 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7JHGA
|
3.47 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
TAK |
Type1 |
22 - 559 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7M74A
|
3.93 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
TAK |
Type1 |
22 - 559 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4RERA
|
4.047 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
20 - 559 |
0 |
TPO183 |
E480G,E483A,K485A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4REWA
|
4.58 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
STU |
Type1 |
20 - 559 |
0 |
None |
E480G,E483A,K485A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4REDA
|
2.95 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
22 - 360 |
0 |
None |
K52A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4REDB
|
2.95 |
Inactive |
DFGinter‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
22 - 360 |
0 |
None |
K52A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5ISOA
|
2.63 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
9 - 551 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5ISOC
|
2.63 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
9 - 550 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6B1UC
|
2.77 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
CG7
|
Type1,
Allosteric
|
9 - 552 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
AF-P54646-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 276 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4ZHXA
|
2.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4O7 |
Type1 |
9 - 550 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFFA
|
3.924 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU |
Type1 |
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
8BIKA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
QTN
|
Type1,
Allosteric
|
8 - 551 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
8BIKD
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
QTN
|
Type1,
Allosteric
|
9 - 551 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6B2EA
|
3.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
STU,
CG7
|
Type1,
Allosteric
|
9 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFEA
|
3.023 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFEC
|
3.023 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
10 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
7MYJA
|
2.95 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4O7,
ZQV
|
Type1,
Allosteric
|
7 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
7MYJC
|
2.95 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
4O7 |
Type1 |
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5EZVA
|
2.99 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU,
C1V
|
Type1,
Allosteric
|
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5EZVC
|
2.99 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
C1V
|
Type1,
Allosteric
|
9 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4ZHXC
|
2.99 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
4O7,
C1V
|
Type1,
Allosteric
|
9 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6B1UA
|
2.77 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
CG7
|
Type1,
Allosteric
|
8 - 550 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFFC
|
3.924 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU,
C1V
|
Type1,
Allosteric
|
10 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
2H6DA
|
1.85 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
10 - 278 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
2YZAA
|
3.02 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
10 - 278 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
9IC2A
|
2.5 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
A1I1Y |
Type1 |
8 - 279 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
3AQVA
|
2.08 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
TAK |
Type1 |
7 - 279 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6BX6A
|
2.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
EDJ |
Type1 |
13 - 277 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
2WNTA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanin |
APEdist_oooo |
No_ligand |
No_ligand |
416 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
2WNTB
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
415 - 709 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
3RNYA
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
418 - 707 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
3RNYB
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
419 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
8WF4A
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanin |
APEdist_oooo |
No_ligand |
No_ligand |
416 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
8WF4B
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiin |
APEdist_oooo |
No_ligand |
No_ligand |
415 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
4NIFA
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
413 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
4NIFD
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_ooon |
No_ligand |
No_ligand |
413 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4D9TA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
0JG |
Type1 |
415 - 713 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4D9UA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
0JH |
Type1 |
408 - 714 |
0 |
None |
K591E |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
8XEYA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
403 - 714 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4JG8A
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oooo |
1LE |
Type1 |
415 - 714 |
0 |
None |
T493M |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4JG6A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
1LB |
Type1 |
406 - 712 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4JG7A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
1LC |
Type1 |
405 - 713 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4VB
|
1.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XWA |
Type1 |
61 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4VC
|
1.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XWA |
Type1 |
61 - 385 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OA
|
2.725 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OC
|
2.725 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OE
|
2.725 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OG
|
2.725 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OI
|
2.725 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OK
|
2.725 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QA
|
2.838 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QC
|
2.838 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QE
|
2.838 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QG
|
2.838 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QI
|
2.838 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QK
|
2.838 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4VA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XWA |
Type1 |
62 - 385 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8OKUA
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VRU |
Type1 |
60 - 392 |
0 |
None |
T221D |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8OKUB
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VRU |
Type1 |
60 - 390 |
0 |
None |
T221D |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UA
|
2.416 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
61 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UC
|
2.416 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UE
|
2.416 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
61 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UG
|
2.416 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SNRK
|
SNRK_HUMAN
|
5YKSA
|
2.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 344 |
0 |
None |
None |
SNF-related serine/threonine-protein kinase |
|
CAMK
|
SNRK
|
SNRK_HUMAN
|
5YKSB
|
2.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 344 |
0 |
None |
None |
SNF-related serine/threonine-protein kinase |
|
CAMK
|
STK11
|
STK11_HUMAN
|
2WTKC
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-none |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
47 - 342 |
0 |
None |
D194A |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK11
|
STK11_HUMAN
|
2WTKF
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-none |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
45 - 340 |
0 |
None |
D194A |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK11
|
STK11_HUMAN
|
8VSUC
|
2.86 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 347 |
0 |
None |
None |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUEB
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
F7I |
Type1 |
59 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUFA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
F8I |
Type1 |
50 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUFB
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
F8I |
Type1 |
55 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUEA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
F7I |
Type1 |
50 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6QF4A
|
2.495 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
ADP |
ATPlike |
18 - 308 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7Q7DA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ATP |
ATPlike |
25 - 297 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7Q7EA
|
2.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ATP |
ATPlike |
25 - 297 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
3LM0A
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
EBD |
Type1 |
25 - 304 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6Y6FA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
OD2 |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6Y6HA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
OBW |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6ZJFA
|
1.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
QM2 |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7AKGA
|
2.08 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
38O |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
3LM5A
|
2.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
QUE |
Type1.5_Back |
25 - 301 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK33
|
STK33_HUMAN
|
8VF6A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
A1AAY |
Type1 |
100 - 382 |
0 |
None |
None |
Serine/threonine-protein kinase 33 |
|
CAMK
|
STK33
|
STK33_HUMAN
|
8VF6B
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
A1AAY |
Type1 |
99 - 383 |
0 |
None |
None |
Serine/threonine-protein kinase 33 |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
9OTYC
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
10 - 299 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
7WTTA
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 305 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
5FQDC
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
5FQDF
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
8G66C
|
3.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iini |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7GA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
AMP |
ATPlike |
8 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7GB
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
AMP |
ATPlike |
7 - 293 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5IH4A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXOA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXOB
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7MA
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7NA
|
1.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7NB
|
1.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7OA
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7PA
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
9B3SA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 415 |
0 |
SEP411 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
9B3SB
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 414 |
0 |
SEP411 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXPB
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
K171E |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXNA
|
1.551 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 291 |
0 |
None |
R178C |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXNB
|
1.551 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
R178C |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8IZCA
|
1.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S93 |
Type1 |
5 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5IH5A
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AUE |
Type1 |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RCGA
|
1.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
K0E |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9A
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9C
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9D
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4HGTA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
15G |
Type1 |
9 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4HNFB
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
5 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8VXDA
|
2.47 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1AD7 |
Type1 |
1 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8VXDB
|
2.47 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnii |
A1AD7 |
Type1 |
2 - 298 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVA
|
2.154 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D5Q |
Type1 |
8 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVC
|
2.154 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D5Q |
Type1 |
6 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVF
|
2.154 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D5Q |
Type1 |
7 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBCA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QJ |
Type1 |
2 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6GZMA
|
1.59 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
LCI |
Type1 |
5 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBKD
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1QG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKA
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKE
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKI
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKK
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKO
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKQ
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKS
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKU
|
2.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HNIA
|
2.74 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HNIB
|
2.74 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4G16A
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
0VM |
Type1 |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4G17A
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
0VN |
Type1 |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4HGLA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
0YO |
Type1 |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZRA
|
1.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
BRK |
Type1 |
36 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZSA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
BRQ |
Type1 |
36 - 333 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZTA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
23D |
Type1 |
37 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4HGSA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
15G |
Type1.5_Back |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
8XPZA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
20 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7QHWAAA
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CGI |
Type1 |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7QHWCCC
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CGI |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7Q8VA
|
2.13 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IV |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7Q8WA
|
2.02 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IO |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTMA
|
2.54 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F8E |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTMB
|
2.54 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F8E |
Type1 |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
9HHWA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IU7 |
Type1 |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTKA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DTQ |
Type1.5_Back |
22 - 311 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8YA
|
1.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IV |
Type1 |
6 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8YB
|
1.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IV |
Type1 |
7 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8ZA
|
1.57 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IK |
Type1 |
6 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8ZB
|
1.57 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IK |
Type1 |
7 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q90A
|
1.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IS |
Type1 |
6 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q90B
|
1.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IS |
Type1 |
7 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9A
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
21 - 342 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9B
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9C
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
ATPlike |
24 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9D
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
ATPlike |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
9ZKGB
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ACN,
GG0,
GG0
|
Allosteric,
Allosteric,
Allosteric
|
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
AF-Q99986-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
29 - 334 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2LAVA
|
999.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0C
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUC
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWC
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6C
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMC
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMC
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHC
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWA
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWC
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4A
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4C
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHC
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42A
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42C
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
9ZKGA
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 342 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2RSVA
|
999.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 396 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8E1 |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFB
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8E1 |
Type1 |
51 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFC
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8E1 |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFD
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8E1 |
Type1 |
39 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5A
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
REB |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5B
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
REB |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5C
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
REB |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5D
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
REB |
Type1 |
25 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
7DZ |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFB
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
7DZ |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0B
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
E1D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWB
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
E8D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6B
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
E8V |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6D
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E8V |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMB
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F7D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMD
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F7D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
F87 |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHA
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
F8Y |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHB
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F8Y |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHD
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F8Y |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWB
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
FBY |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWD
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
FBY |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4B
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
G6J |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4D
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
G6J |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
RTJ |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUB
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RTJ |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUD
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RTJ |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42B
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
YD9 |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42D
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
YD9 |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFC
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
7DZ |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFD
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
7DZ |
Type1.5_Back |
25 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0D
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E1D |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUB
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
E5M |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUD
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
E5M |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
E8D |
Type1.5_Back |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWD
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E8D |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
E8V |
Type1.5_Back |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMA
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
EA7 |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMB
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EA7 |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMD
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EA7 |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXB
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F87 |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXC
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
FCS |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXD
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F87 |
Type1.5_Back |
24 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPNA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KWJ |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPNB
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
KWJ |
Type1.5_Back |
24 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPNC
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KWJ |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPND
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
KWJ |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUC
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
VBD |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHB
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
RYA |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHD
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RYA |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
9ZKGC
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
A1C2O |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
9ZKGD
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
A1C2O |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2KTYA
|
999.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 360 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2KULA
|
999.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 360 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
5UU1A
|
2.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
7DZ |
Type1.5_Back |
14 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
6NCGA
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KJD |
Type1.5_Back |
14 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
6NCGB
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
KJD |
Type1.5_Back |
16 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
9SKQA
|
3.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iiii |
ANP |
ATPlike |
3 - 288 |
0 |
TPO161 |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC3A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
7NJ0B
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 290 |
0 |
TPO161 |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4Y72A
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
LZ9 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
5HQ0A
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
LZ9 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
5LQFA
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
4SP |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
5LQFD
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
4SP |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU2A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
F9Z |
Type1 |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU3A
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FB8 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU4A
|
2.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
FC8 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6A
|
2.6 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6C
|
2.6 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6E
|
2.6 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6G
|
2.6 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7C
|
2.75 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7E
|
2.75 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7G
|
2.75 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
1 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU6A
|
2.33 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
1QK |
Type1 |
1 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7A
|
2.75 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FB8 |
Type1 |
1 - 293 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZB
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZC
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZD
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
437 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZE
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
435 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZF
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
9I9IK
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
440 - 740 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU2H
|
3.13 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVQ |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU4B
|
3.09 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU4H
|
3.09 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU5B
|
3.134 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RMF |
Type1 |
713 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU5H
|
3.134 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
713 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU9H
|
3.51 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUAB
|
3.193 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVH |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUAE
|
3.193 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RVH |
Type1 |
715 - 1033 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUAH
|
3.193 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RVH |
Type1 |
715 - 1034 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUCB
|
3.85 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKO |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUDB
|
3.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RP9 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUDH
|
3.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RP9 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUEH
|
3.25 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVU |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUIB
|
3.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RV6 |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUIH
|
3.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RV6 |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BULH
|
3.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSU |
Type1 |
715 - 1034 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUNB
|
3.08 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RNF |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUNH
|
3.08 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RNF |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUOB
|
3.58 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RLC |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BURE
|
3.64 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQU |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUSH
|
3.26 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMX |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUTB
|
3.25 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ5 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUTH
|
3.25 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RQ5 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
7NXKA
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
UUB |
Type1 |
715 - 1040 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9FMRE
|
3.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RMF |
Type1 |
714 - 1042 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9FMRH
|
3.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
714 - 1044 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4CXAA
|
3.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
718 - 1050 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4NSTA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
716 - 1046 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4NSTC
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
717 - 1045 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4UN0C
|
3.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiii |
No_ligand |
No_ligand |
719 - 1036 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4UN0D
|
3.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiii |
No_ligand |
No_ligand |
723 - 1024 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4CXAC
|
3.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
718 - 1048 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU2E
|
3.13 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUDE
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUGE
|
3.53 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6B3EA
|
3.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CJM |
Type1 |
717 - 1036 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6B3EC
|
3.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CJM |
Type1 |
719 - 1036 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
5ACBC
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5I1 |
Type1 |
716 - 1040 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
5ACBD
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5I1 |
Type1 |
718 - 1044 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9JK1A
|
2.72 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1EB3 |
Type1 |
717 - 1039 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9JK1B
|
2.72 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1EB3 |
Type1 |
715 - 1039 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6TD3B
|
3.46 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RC8 |
Type1 |
715 - 1047 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6TD3H
|
3.46 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiii |
RC8 |
Type1 |
715 - 1047 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU1E
|
2.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU4E
|
3.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU6E
|
3.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQE |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU7E
|
3.245 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RS5 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU9E
|
3.51 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUBB
|
3.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
RNU |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUBE
|
3.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
RNU |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUCE
|
3.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKO |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUEE
|
3.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RVU |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUFE
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RW6 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUHE
|
3.79 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RR9 |
Type1 |
715 - 1034 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUIE
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
RV6 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUJE
|
3.62 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RUW |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUKE
|
3.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RWE |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUNE
|
3.08 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RNF |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUOE
|
3.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RLC |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUPB
|
3.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RWN |
Type1 |
715 - 1027 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUPE
|
3.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
RWN |
Type1 |
715 - 1027 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUQB
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ9 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUQE
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ9 |
Type1 |
715 - 1027 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BURB
|
3.64 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQU |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUSB
|
3.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RMX |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUTE
|
3.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ5 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6CKXA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8M1 |
Type1 |
722 - 1024 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6CKXC
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8M1 |
Type1 |
722 - 1024 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
7NXKC
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
UUB |
Type1 |
717 - 1040 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUGH
|
3.53 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU1B
|
2.98 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU1H
|
2.98 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU2B
|
3.13 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVQ |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU3B
|
3.42 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSI |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU3H
|
3.42 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RSI |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU5E
|
3.134 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RMF |
Type1 |
713 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU6B
|
3.45 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQE |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU6H
|
3.45 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQE |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU9B
|
3.51 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUBH
|
3.42 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooo |
APEdist_iiii |
RNU |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUCH
|
3.85 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RKO |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUEB
|
3.25 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RVU |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUFB
|
3.3 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RW6 |
Type1 |
715 - 1033 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUFH
|
3.3 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RW6 |
Type1 |
715 - 1032 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUGB
|
3.53 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RPW |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUHB
|
3.79 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RR9 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUHH
|
3.79 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RR9 |
Type1 |
715 - 1033 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUJB
|
3.62 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RUW |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUJH
|
3.62 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RUW |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUKB
|
3.41 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RWE |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUKH
|
3.41 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RWE |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BULB
|
3.4 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSU |
Type1 |
715 - 1039 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUMB
|
3.36 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6X |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUMH
|
3.36 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6X |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUOH
|
3.58 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RLC |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUQH
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ9 |
Type1 |
715 - 1035 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BURH
|
3.64 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQU |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUSE
|
3.26 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RMX |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9FMRB
|
3.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
714 - 1047 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
5EFQA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
695 - 1025 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
5EFQC
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
697 - 1031 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
7NXJA
|
2.36 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5I1 |
Type1 |
695 - 1023 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
7NXJC
|
2.36 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5I1 |
Type1 |
695 - 1017 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
5G6VA
|
2.2 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
919 |
Type2 |
163 - 474 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
3MTLA
|
2.4 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FEF |
Type1 |
163 - 473 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
5G6VB
|
2.2 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
919 |
Type2 |
163 - 475 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8BZOA
|
3.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-none |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5NEVA
|
2.97 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
72L |
Type1 |
1 - 295 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5NEVC
|
2.97 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
72L |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOOA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOOC
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOMC
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
H84S,Q85M,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FINA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FINC
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FQ1B
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oioo |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CCHA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9I9JK
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ADP |
ATPlike |
6 - 284 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9I9KK
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
2 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9QCVK
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ANP |
ATPlike |
1 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOQA
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOQC
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOJA
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 298 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOJC
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8VQ3A
|
1.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
A1AC4 |
Allosteric |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8VQ4A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
A1AC5 |
Allosteric |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2JGZA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 288 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9HIUB
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9HIWB
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9HJ1B
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1F5QA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1F5QC
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1JSUA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKVA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKVC
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKWA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKWC
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL1A
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL1C
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL2A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL2C
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1URCA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1URCC
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2V22A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2V22C
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WFYA
|
2.53 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WFYC
|
2.53 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WHBA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WHBC
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IF1A
|
2.61 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IF1C
|
2.61 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6P3WA
|
2.54 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6P3WC
|
2.54 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7B5LL
|
3.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
13 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7B5RL
|
3.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
13 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8ROZA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 298 |
0 |
PTR15,TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9D0WC
|
2.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5UQ2A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5UQ3A
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9QCXK
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6SG4A
|
2.43 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
28 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6SG4C
|
2.43 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 295 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H24A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H27C
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOPA
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOPC
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 296 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOIC
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 296 |
0 |
TPO160 |
K89D,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PKDA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UCN |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5LMKC
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6ZK |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9GLAA
|
2.18 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YNK |
Type1 |
2 - 294 |
0 |
TPO160 |
E8D,K9F,I10L,T14Q,Y15F,V64I,L83M,H84E,Q85T,K88E,K89V,Q131N |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EORA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SP |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EORC
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4SP |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FVVA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
107 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FVVC
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiii |
107 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5NA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
CK8 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5NC
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK8 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5OA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
CK2 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5OC
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
CK2 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5VA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK4 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5VC
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK4 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5XA
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oioi |
MTW |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5XC
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
MTW |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2I40A
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnii |
BLZ |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2I40C
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
BLZ |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UUEA
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
MTZ |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UUEC
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
MTZ |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZBA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_iioi |
C75 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZBC
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
C75 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WEVA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
CK7 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WEVC
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK7 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2X1NA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
X1N |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2X1NC
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioi |
X1N |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EJ1A
|
3.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
5BP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EJ1C
|
3.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
5BP |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EOCC
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
T2A |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3TIYA
|
1.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
TIY |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FX3A
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
60K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FX3C
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
60K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8CURA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
OW6 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9NYRD
|
3.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1B7G |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8H6PA
|
2.44 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
WZU |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DDQC
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DOGA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
NNN |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DOGC
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NNN |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6JGMA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
AQG |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8B54A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
P2V |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4NJ3A
|
1.848 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
2KD |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOSA
|
2.57 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOSC
|
2.57 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9QJJB
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
NK3 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1QA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2A6 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7MKXA
|
3.08 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZGY |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTWA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X3A |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QU0A
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X40 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R9DA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X6B |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R9OA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
Z71 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RZBA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
02Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1VYWA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
292 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2BPMA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
529 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C4GA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
514 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WIHA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
P48 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WIPA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
P49 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WIPC
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
P49 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WPAA
|
2.51 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
889 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WXVA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
WXV |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WXVC
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
WXV |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOKA
|
2.57 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4SP |
Type1 |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOKC
|
2.57 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4SP |
Type1 |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOLA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOLC
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3F5XA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
EZV |
Type1.5_Back |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3F5XC
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EZV |
Type1.5_Back |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PXFA
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
2AN,
2AN
|
Allosteric,
Type3
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PXZA
|
1.7 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
2AN,
2AN,
JWS
|
Allosteric,
Type3,
Type1
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6YL6A
|
1.7 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
F80C,C177A |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7UXIA
|
2.07 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
No_ligand |
No_ligand |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5OO3A
|
1.73 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
9ZB |
Type1 |
2 - 294 |
0 |
None |
F80C,C177A |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6YL1A
|
1.66 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
OWN |
Type1 |
1 - 298 |
0 |
None |
F80C,C177A |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6YLKA
|
1.65 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
OY2 |
Type1 |
1 - 298 |
0 |
None |
F80C,C177A |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1DM2A
|
2.1 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
HMD |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1G5SA
|
2.61 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
I17 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1P2AA
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5BN |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PF8A
|
2.51 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
SU9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2B52A
|
1.88 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
D42 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2B55A
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
D31 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2BHEA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
BRY |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2BHHA
|
2.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
RYU |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2BTSA
|
1.99 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
U32 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5YA
|
2.25 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
MTW |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2FVDA
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
LIA |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2J9MA
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
PY8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTNA
|
2.2 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
LZ7 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTQA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
LZA |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTTA
|
1.68 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
LZD |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VU3A
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
LZE |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3TI1A
|
1.99 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
B49 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3TIZA
|
2.02 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
3TI |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3UNJA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
0BX |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3UNKA
|
2.1 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
0BY |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANGA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
WY3 |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7M2FA
|
1.632 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
YOS |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9D0UA
|
2.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
A1A1H |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8ERDA
|
1.33 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
WQ6 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6INLA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
AJR |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3NA
|
1.63 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
SCZ |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VV9A
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
IM9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2W17A
|
2.15 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
I19 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3SW7A
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
19K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BZDA
|
1.83 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
D6I |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKOA
|
1.55 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
20K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EZVA
|
1.99 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
EZV |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7RA5A
|
1.67 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
3I3 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8YNGA
|
1.82 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
A1D6S |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8YPWA
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
A1D6Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8YQEA
|
1.94 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
A1D60 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9JJ5A
|
1.71 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1EB0 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9UAUA
|
1.47 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
A1EOM |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9UAWA
|
1.72 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
A1EOO |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9UGFA
|
1.64 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
A1EO5 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PXYA
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
JWS |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PY0A
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
SU9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QQGA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X06 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QQHA
|
1.87 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X0A |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QQKA
|
1.86 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X02 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QRTA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X14 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QRUA
|
1.95 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X19 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTQA
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X35 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTRA
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
X36 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTUA
|
1.82 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X44 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTXA
|
1.95 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X43 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTZA
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X42 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QWKA
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X62 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QXPA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X64 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R8MA
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
Z19 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R8ZA
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
Z63 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RAKA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
03Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RALA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
04Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RJCA
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
06Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RK9A
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
09Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RMFA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
20Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RNIA
|
1.95 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
21Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RPVA
|
1.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
26Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RPYA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
27Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3S1HA
|
1.75 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
56Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3SQQA
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
99Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4ERWA
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
STU |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EZ3A
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
0S0 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4GCJA
|
1.42 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
X64 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUHA
|
1.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
FB8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4D1ZA
|
1.851 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-none |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
WG8,
WG8
|
Type1,
Allosteric
|
3 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5FP5A
|
2.16 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-none |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
1Y6,
1Y6
|
Type1,
Allosteric
|
1 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5FP6A
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
MFZ,
MFZ
|
Type1,
Allosteric
|
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PXQA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
2AN,
2AN,
2AN
|
Type1,
Allosteric,
Type3
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PY1A
|
2.05 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
SU9,
2AN,
2AN
|
Type1,
Allosteric,
Type3
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7RWEA
|
1.59 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
none-none |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
7TH,
7TH
|
Type1,
Type3
|
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7SA0A
|
1.59 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
8KQ,
8KQ
|
Type1,
Type3
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8FOWA
|
1.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
1QK,
7TW
|
Type1,
Type3
|
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8FP0A
|
1.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
RRC,
7TW
|
Type1,
Type3
|
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EZ7A
|
2.49 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
STU,
2AN,
2AN
|
Type1,
Type3,
Allosteric
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7RXOA
|
1.38 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
80E |
Type3 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7S4TA
|
1.91 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
88O |
Type3 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7S7AA
|
1.7 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
8FI |
Type3 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7S84A
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
8IL |
Type3 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7S85A
|
1.98 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
8IQ |
Type3 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7S9XA
|
1.69 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
8KF |
Type3 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7RWFA
|
1.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
7TW |
Type3 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7UG1A
|
1.84 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
N5R,
N5R
|
Type3,
Allosteric
|
1 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKUA
|
1.47 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
60K,
60K
|
Allosteric,
Type1
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1AQ1A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
STU |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1DI8A
|
2.2 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
DTQ |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FVTA
|
2.2 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
106 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1GIHA
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1PU |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1JVPP
|
1.53 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
89E |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1KE5A
|
2.2 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
LS1 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1KE6A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
LS2 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1KE7A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
LS3 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1KE8A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
LS4 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1KE9A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
LS5 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1R78A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
FMD |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2XNBA
|
1.85 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Y8L |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BGHA
|
1.95 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
3I6 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IEVA
|
2.03 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
R0N |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKWA
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
62K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7NVQA
|
2.05 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
STU |
Type1 |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4HA
|
1.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HGH |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1GIIA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1PU |
Type1 |
1 - 298 |
0 |
None |
F82H,L83V,K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1HCKA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8FP5A
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ATP |
ATPlike |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1B38A
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1B39A
|
2.1 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5OO0A
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
9YZ |
Allosteric |
2 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5OSJA
|
1.83 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
AAK |
Allosteric |
2 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4KA
|
1.06 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HHW,
HHW
|
Allosteric,
Allosteric
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1HCLA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PW2A
|
1.95 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANOA
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EK3A
|
1.34 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7UXKA
|
2.63 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OITA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
HDT |
Type1 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1CKPA
|
2.05 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
PVB |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H0VA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
UN4 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H0WA
|
2.1 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
207 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1JSVA
|
1.96 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
U55 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXIA
|
1.95 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK1 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXJA
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK2 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXKA
|
2.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
CK3 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXLA
|
2.5 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
CK4 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXMA
|
2.53 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK5 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXNA
|
2.5 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK6 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXPA
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1VYZA
|
2.21 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
N5B |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1W0XC
|
2.2 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
OLO |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1WCCA
|
2.2 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
CIG |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1Y8YA
|
1.996 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
CT7 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1Y91A
|
2.15 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CT9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1YKRA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
628 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2A0CX
|
1.95 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2A4LA
|
2.4 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
RRC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2B53A
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
D23 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2B54A
|
1.85 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
D05 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2BTRA
|
1.85 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
U73 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C68A
|
1.95 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
CT6 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C69A
|
2.1 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CT8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6IA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
DT1 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6KA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
DT2 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6LA
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
DT4 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6MA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
DT5 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CLXA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
F18 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2DUVA
|
2.2 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
371 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2EXMA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ZIP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R64A
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
740 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZNA
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
C96 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2V0DA
|
2.2 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
C53 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTAA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LZ1 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTHA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LZ2 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTIA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
LZ3 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTJA
|
2.2 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
LZ4 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTLA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LZ5 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTMA
|
2.25 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LZM |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTOA
|
2.19 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LZ8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTPA
|
2.15 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
LZ9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTRA
|
1.89 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LZB |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2VTSA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LZC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2W1HA
|
2.15 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0F |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2XMYA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
CDK |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3FZ1A
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
B98 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3LE6A
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
2BZ |
Type1 |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3LFNA
|
2.28 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A27 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3LFQA
|
2.03 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A28 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3LFSA
|
2.4 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A07 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3NS9A
|
1.78 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
NS9 |
Type1 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3S2PA
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
PMU |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3ULIA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
1N3 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3WBLA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
PDY |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4LYNA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1YG |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4RJ3A
|
1.63 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-na |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
3QS |
Type1 |
1 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANDA
|
2.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
5JE |
Type1 |
2 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANEA
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
SZL |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANIA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
ES4 |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANJA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
ZXC |
Type1 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5ANKA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
RJI |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IEYA
|
1.66 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
6AE |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5JQ8A
|
1.94 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
I73 |
Type1 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6OQIA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
N14 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8ERNA
|
1.64 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
WQK |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5K4JA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
6QB |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1E1VA
|
1.95 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CMG |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1E1XA
|
1.85 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
NW1 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1GZ8A
|
1.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
MBP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OIQA
|
2.31 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
HDU |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OIRA
|
1.91 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-na |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HDY |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1URWA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
I1P |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1V1KA
|
2.31 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
3FP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1W8CA
|
2.05 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
N69 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3FA
|
1.5 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
SC8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3GA
|
1.55 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
SC9 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3HA
|
1.5 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
SCE |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3IA
|
1.28 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
SCF |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3JA
|
1.65 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
SCJ |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3KA
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
SCQ |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3MA
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
SCX |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3OA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
2SC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3PA
|
1.66 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
3SC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3QA
|
1.35 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
5SC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2W06A
|
2.04 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
FRV |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3IG7A
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
EFP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4ACMA
|
1.63 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
7YG |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EK4A
|
1.26 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
1CK |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EK5A
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
03K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EK6A
|
1.52 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
10K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EK8A
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
16K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKGA
|
1.51 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
4CK |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKIA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
09K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKJA
|
1.63 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
11K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKLA
|
1.26 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK2 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKPA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
LS5 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKSA
|
1.55 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
46K |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKTA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
48K |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKVA
|
1.7 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
61K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PJ8A
|
1.96 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
404 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7VDUA
|
1.53 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-na |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
65L |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8OY2A
|
2.618 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
W5W |
Type1 |
2 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QQLA
|
1.85 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X03 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QZFA
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X66 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R8LA
|
1.9 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z30 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R8PA
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z46 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5MHQA
|
1.3 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-na |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
8QT |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4CA
|
1.73 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HH8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1GIJA
|
2.2 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
2PU |
Type1 |
1 - 298 |
0 |
None |
F82H,L83V,K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2DS1A
|
2.0 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
1CD |
Type1 |
1 - 298 |
0 |
None |
F82H,L83V,K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4DA
|
1.07 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HHT,
HHT,
HHT,
HHT,
HHT,
HHT
|
Type1,
Allosteric,
Allosteric,
Allosteric,
Allosteric,
Allosteric
|
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H01A
|
1.79 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-na |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
FAL,
FBL
|
Type1,
Type1
|
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H00A
|
1.6 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
FAP,
FCP
|
Type1,
Type1
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H07A
|
1.85 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
MFP,
MFQ
|
Type1,
Type1
|
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H08A
|
1.8 |
Inactive |
DFGin‑BLBtrans |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
BYP,
BWP
|
Type1,
Type1
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8BYAA
|
3.38 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
16 - 296 |
0 |
TPO159 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5UQ1C
|
3.201 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5OO1A
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
9Z2 |
Type1 |
4 - 298 |
0 |
None |
F80C,C177A |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PYEA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
PM1 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2W05A
|
1.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
FRT |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5D1JA
|
1.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
56H |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QL8A
|
1.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X01 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QWJA
|
1.75 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X6A |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QX4A
|
1.92 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X4B |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R9HA
|
2.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
Z67 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RK5A
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
07Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RK7A
|
1.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
08Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RKBA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
12Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RM6A
|
1.6 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
18Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3S0OA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
50Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8RU8A
|
1.51 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
I74 |
Type1 |
1 - 298 |
0 |
None |
I10L,T14Q,V64I,K88E,K89V,D92K,Q131N |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EZRA
|
1.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
EZR,
EZR
|
Type1,
Allosteric
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5A14A
|
2.0 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LQ5,
LQ5
|
Type2,
Allosteric
|
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q3FA
|
1.18 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HEW |
Allosteric |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q49A
|
1.0 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
HGQ |
Allosteric |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1BUHA
|
2.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3PXRA
|
2.0 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4IA
|
1.11 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
HGK |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5OSMA
|
1.77 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
AEQ |
Type1 |
1 - 296 |
0 |
None |
F80C,C177A |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8UV0A
|
1.55 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XKU |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4GA
|
0.98 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
HJK |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PXOA
|
1.96 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CK7 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6OA
|
2.1 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
4SP |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZOA
|
2.3 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
C62 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4D1XA
|
2.1 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ESJ |
Type1 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4KD1A
|
1.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
1QK |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IEXA
|
2.03 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
6AF |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5JQ5A
|
1.94 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
I74 |
Type1 |
3 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9FR2A
|
1.6 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
A1IE9 |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3LA
|
1.65 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnnn |
SCW |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2R3RA
|
1.47 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
6SC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3IGGA
|
1.8 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
EFQ |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3SW4A
|
1.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
18K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKQA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
42K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FKRA
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
45K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QQFA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X07 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QQJA
|
1.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X11 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTSA
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
X46 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QX2A
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X63 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QXOA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X65 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QZGA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X67 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QZHA
|
1.95 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X69 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QZIA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X72 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R1QA
|
1.85 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X75 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R1SA
|
1.8 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X73 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R1YA
|
1.8 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X76 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R28A
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
XA0 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R6XA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X84 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R71A
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X86 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R73A
|
1.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X87 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R7EA
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
X88 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R7IA
|
1.85 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
X9I |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R7UA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
X96 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R7VA
|
1.95 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z02 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R7YA
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z04 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R83A
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z14 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R8UA
|
2.0 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z31 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R8VA
|
1.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z62 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R9NA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
Z68 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RAHA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
O1Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RAIA
|
1.7 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X85 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RM7A
|
1.85 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
19Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3ROYA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
22Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RPOA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
24Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3RPRA
|
1.75 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
25Z |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3S00A
|
1.8 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
Z60 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUKA
|
1.3 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
FC8 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q48A
|
1.03 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
HHQ |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4AA
|
1.13 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HGW |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4BA
|
1.12 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HHN |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4EA
|
1.06 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
HH5 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4FA
|
1.21 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
26D |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q4JA
|
1.05 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
HHB |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7ZPCA
|
1.4 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
JLC |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9GNOA
|
1.16 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
A1INI |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q3BA
|
1.11 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
PYZ,
PYZ
|
Type1,
Type1
|
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6Q3CA
|
1.29 |
Inactive |
None‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
BYZ,
BYZ
|
Type1,
Type1
|
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
7SJ3A
|
2.51 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6ZV |
Type1 |
2 - 295 |
0 |
TPO172 |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
3G33A
|
3.0 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
5 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
3G33C
|
3.0 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
No_ligand |
No_ligand |
5 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
6P8GB
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
No_ligand |
No_ligand |
18 - 299 |
0 |
None |
G43E,G47E |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
6P8HB
|
3.19 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
18 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
2W99B
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
No_ligand |
No_ligand |
2 - 295 |
0 |
None |
G43E,G47E,T172A |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
2W9ZB
|
2.45 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
2 - 295 |
0 |
None |
G43E,G47E,T172A |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
2W96B
|
2.3 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
4 - 295 |
0 |
None |
G43E,G47E,T172D |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
9CSKB
|
2.253 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
A1AZ4 |
Type1 |
4 - 295 |
0 |
None |
G43E,G47E |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
9CSKD
|
2.253 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1AZ4 |
Type1 |
4 - 295 |
0 |
None |
G43E,G47E |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
6P8EB
|
2.3 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
18 - 299 |
0 |
None |
G43E,G47E |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
6P8FB
|
2.89 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
18 - 299 |
0 |
None |
G43E,G47E |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
2W9FB
|
2.85 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 295 |
0 |
None |
G43E,G47E,T172F |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
5FWKK
|
3.9 |
Inactive |
None‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_iioo |
No_ligand |
No_ligand |
87 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
5FWLK
|
9.0 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_iioo |
No_ligand |
No_ligand |
5 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
5FWMK
|
8.0 |
Inactive |
None‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_iioo |
No_ligand |
No_ligand |
5 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK4
|
CDK4_HUMAN
|
5FWPK
|
7.2 |
Inactive |
None‑None |
DFGAsp-rot-out |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_iioo |
No_ligand |
No_ligand |
87 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 4 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1H4LA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 287 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1H4LB
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 287 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1UNLB
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
D144N |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
3O0GA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
D144N |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDPA
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
65L |
Type1 |
2 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDPB
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
65L |
Type1 |
3 - 288 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDQA
|
2.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
64V |
Type1 |
2 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDQB
|
2.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
64V |
Type1 |
3 - 288 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDRA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
63I |
Type1 |
2 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDRB
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
63I |
Type1 |
3 - 288 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
7VDSA
|
3.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
61U |
Type1 |
2 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
4AU8A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
Z3R |
Type1 |
2 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
4AU8B
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
Z3R |
Type1 |
2 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1UNGA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ALH |
Type1 |
1 - 292 |
0 |
None |
D144N |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1UNHA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IXM |
Type1 |
2 - 288 |
0 |
None |
D144N |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1UNHB
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IXM |
Type1 |
2 - 288 |
0 |
None |
D144N |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK5
|
CDK5_HUMAN
|
1UNLA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RRC |
Type1 |
1 - 292 |
0 |
None |
D144N |
Cyclin-dependent kinase 5 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1JOWB
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 300 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1XO2B
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_iiii |
FSE |
Type1 |
11 - 305 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
2EUFB
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LQQ |
Type1 |
10 - 305 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
2F2CB
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AP9 |
Type1 |
9 - 305 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
4TTHB
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
24V |
Type1 |
15 - 304 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1BLXA
|
1.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
5 - 309 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
6OQLA
|
2.707 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
N1A |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
6OQOA
|
1.977 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
N1J |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
8I0MA
|
2.777 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
NJ6 |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
3NUPA
|
2.6 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3NU |
Type1 |
12 - 300 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
3NUXA
|
2.7 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
3NV |
Type1 |
10 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
4AUAA
|
2.31 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
4AU |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
4EZ5A
|
2.7 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0RS |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
5L2IA
|
2.75 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
LQQ |
Type1 |
10 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
5L2SA
|
2.27 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
6ZV |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
5L2TA
|
2.37 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
6ZZ |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
9D8UA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
A1AZ4 |
Type1 |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
9PE7A
|
2.05 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
A1CIF |
Type1 |
10 - 301 |
0 |
None |
E21V,K26T,T106R,Q149E |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
9PE8A
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
A1AZ4 |
Type1 |
10 - 301 |
0 |
None |
E21V,K26T,T106R,Q149E |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1G3NA
|
2.9 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1G3NE
|
2.9 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1BI7A
|
3.4 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
10 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1BI8A
|
2.8 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1BI8C
|
2.8 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
11 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
6XBZJ
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AGS |
ATPlike |
10 - 312 |
0 |
SEP164 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
7EGB8
|
3.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 312 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
7ENC8
|
4.13 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
7LBME
|
4.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 312 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
7NVR8
|
4.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 312 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R99A
|
1.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ANP |
ATPlike |
10 - 311 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P6YJ
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AGS |
ATPlike |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9I9IJ
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
12 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9I9JJ
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ADP |
ATPlike |
11 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9I9KJ
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ADP |
ATPlike |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9QCVJ
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ANP |
ATPlike |
10 - 346 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9SKQJ
|
3.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ANP |
ATPlike |
9 - 346 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9SA
|
2.78 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_niii |
PE3,
PE3,
YPK
|
Allosteric,
Allosteric,
Type1
|
8 - 312 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8BVW8
|
4.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P79J
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9QCXJ
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
9 - 346 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9AA
|
1.71 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
I74 |
Type1 |
10 - 311 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9OA
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
YN3 |
Type1 |
10 - 312 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9OB
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
YN3 |
Type1 |
10 - 312 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9UA
|
1.937 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
YNK |
Type1 |
10 - 311 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9UB
|
1.937 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
YNK |
Type1 |
10 - 311 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8ORMJ
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V0G |
Type1 |
10 - 312 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P6VJ
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I74 |
Type1 |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P77J
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I73 |
Type1 |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8S0RJ
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H46 |
Type1 |
10 - 312 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8S0TJ
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YNK |
Type1 |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9QJNJ
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NK3 |
Type1 |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P7LJ
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
WD9 |
Type1 |
10 - 311 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9HIXJ
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_niii |
V0G |
Type1 |
10 - 312 |
0 |
None |
D97N |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
9HJ0J
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I74 |
Type1 |
12 - 310 |
0 |
None |
D97N |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P73J
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
X50,
X58
|
Type1,
Type1
|
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P4ZA
|
2.75 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
WZ8 |
Type1 |
11 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8P4ZB
|
2.75 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
WZ8 |
Type1 |
10 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
1UA2A
|
3.02 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
ATP |
ATPlike |
13 - 311 |
0 |
TPO170 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
1UA2B
|
3.02 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ATP |
ATPlike |
13 - 311 |
0 |
TPO170 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
1UA2C
|
3.02 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ATP |
ATPlike |
13 - 311 |
0 |
TPO170 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
1UA2D
|
3.02 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ATP |
ATPlike |
13 - 311 |
0 |
TPO170 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9BA
|
2.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ANP |
ATPlike |
1 - 311 |
0 |
None |
S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9BB
|
2.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ANP |
ATPlike |
3 - 310 |
0 |
None |
S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9BC
|
2.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
ANP |
ATPlike |
8 - 311 |
0 |
None |
S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9BD
|
2.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
ANP |
ATPlike |
9 - 311 |
0 |
None |
S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8R9SB
|
2.78 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_niii |
PE3,
PE3,
YPK
|
Allosteric,
Allosteric,
Type1
|
9 - 312 |
0 |
None |
W132R,S164D,T170E |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
6O9L8
|
7.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
7EGC8
|
3.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
7ENA8
|
4.07 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8BYQ8
|
4.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
No_ligand |
No_ligand |
13 - 310 |
0 |
None |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8GXQHI
|
5.04 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-na |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
K41A |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8GXSHI
|
4.16 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
K41A |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
6XD3J
|
3.3 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
V0G |
Type1 |
10 - 312 |
0 |
SEP164 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8PYRA
|
2.15 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
46 - 311 |
0 |
SEP164,TPO170 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK7
|
CDK7_HUMAN
|
8PYRE
|
2.15 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 310 |
0 |
SEP164,TPO170 |
None |
Cyclin-dependent kinase 7 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5HBJA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5Y8 |
Type1 |
1 - 361 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5ICPA
|
2.18 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
69Z |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5IDNA
|
2.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
6A7 |
Type1 |
1 - 363 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5XQXA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
8CC |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5XS2A
|
2.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
8D6 |
Type1 |
1 - 363 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6QTJA
|
2.48 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
JHK |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
9H8CA
|
2.573 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
A1IS8 |
Type1 |
1 - 361 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
9H8SA
|
2.157 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1ITF |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
8TQ2A
|
3.8 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
8TQCA
|
3.8 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
8TQWA
|
8.2 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4G6LA
|
2.7 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5FGKA
|
2.36 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5XG |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5HBEA
|
2.38 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
5Y6 |
Type1 |
1 - 361 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5HNBA
|
2.35 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
62M |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5I5ZA
|
2.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
68U |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5IDPA
|
2.65 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6A6 |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7SA
|
2.2 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
0SW |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5BNJA
|
2.64 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
4TV |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6QTGA
|
2.7 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
JH8 |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4CRLA
|
2.4 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
C1I |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5CEIA
|
2.24 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
50R |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6R3SA
|
2.19 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
JRE |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6Y0AA
|
2.19 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
JRE |
Type1 |
1 - 362 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6T41A
|
2.45 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MFE |
Type1 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5HBHA
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
5Y7 |
Type1 |
1 - 361 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
3RGFA
|
2.2 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BAX |
Type2 |
1 - 353 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F6UA
|
2.1 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
0SR |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F6WA
|
2.39 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
0SS |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7LA
|
2.9 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
0SO |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7NA
|
2.65 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
0SV |
Type2 |
1 - 361 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5HVYA
|
2.39 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
66X |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6TPAA
|
2.8 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
NZ8,
NZ5,
NZ5,
NZ5
|
Type2,
Allosteric,
Allosteric,
Allosteric
|
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F6SA
|
2.6 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0SQ |
Type3 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7JA
|
2.6 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0SU |
Type3 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F70A
|
3.0 |
Inactive |
None‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0ST |
Type3 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
3BLHA
|
2.48 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 325 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
3TNIA
|
3.234 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 325 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
8I0LA
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NJ6 |
Type1 |
6 - 326 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
7NWKA
|
2.81 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
UT5 |
Type1 |
7 - 326 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
3BLRA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CPB |
Type1 |
7 - 326 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
4BCGA
|
3.085 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T3C |
Type1 |
7 - 327 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
4BCHA
|
2.958 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T7Z |
Type1 |
7 - 327 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
4BCIA
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T3E |
Type1 |
5 - 326 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
4BCJA
|
3.162 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T9N |
Type1 |
6 - 326 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
8K5RA
|
3.751 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VQE |
Type1 |
5 - 327 |
0 |
TPO186 |
S7D,V8N,K44R,Y138F,K280A,D307E,N311E |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDK9
|
CDK9_HUMAN
|
6Z45A
|
3.37 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
Q6E |
Type1 |
5 - 328 |
0 |
TPO186 |
None |
Cyclin-dependent kinase 9 |
|
CMGC
|
CDKL2
|
CDKL2_HUMAN
|
4BBMB
|
2.0 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-in |
out-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
TC0 |
Type1 |
1 - 308 |
0 |
None |
T159D,Y161E |
Cyclin-dependent kinase-like 2 |
|
CMGC
|
CDKL2
|
CDKL2_HUMAN
|
4AAAA
|
1.53 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
DKI |
Type1 |
1 - 302 |
0 |
None |
T159D,Y161E |
Cyclin-dependent kinase-like 2 |
|
CMGC
|
CDKL2
|
CDKL2_HUMAN
|
8S6IA
|
1.72 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
A1H5G |
Type1 |
1 - 305 |
0 |
None |
None |
Cyclin-dependent kinase-like 2 |
|
CMGC
|
CDKL2
|
CDKL2_HUMAN
|
4BBMA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
TC0 |
Type1 |
1 - 308 |
0 |
None |
T159D,Y161E |
Cyclin-dependent kinase-like 2 |
|
CMGC
|
CDKL3
|
CDKL3_HUMAN
|
3ZDUA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
38R |
Type1 |
1 - 309 |
0 |
None |
T158D,Y160E |
Cyclin-dependent kinase-like 3 |
|
CMGC
|
CDKL5
|
CDKL5_HUMAN
|
4BGQA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
38R |
Type1 |
9 - 302 |
0 |
None |
T169D,Y171E |
Cyclin-dependent kinase-like 5 |
|
CMGC
|
CDKL5
|
CDKL5_HUMAN
|
8CIEA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
US0 |
Type1 |
13 - 303 |
0 |
None |
None |
Cyclin-dependent kinase-like 5 |
|
CMGC
|
CDKL5
|
CDKL5_HUMAN
|
9EPUA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
A1H6P |
Type1 |
12 - 303 |
0 |
None |
None |
Cyclin-dependent kinase-like 5 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6KHDC
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
3NG |
Type1 |
150 - 479 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
AF-P49759-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
153 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
2VAGA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaino |
APEdist_oioo |
V25 |
Type1 |
148 - 481 |
0 |
SEP341,TPO342 |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
5J1VC
|
2.52 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oion |
6FD |
Type1 |
148 - 483 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6FT9C
|
1.87 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_oioo |
E6W |
Type1 |
148 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6G33A
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaino |
APEdist_oioo |
5ID |
Type1 |
148 - 482 |
0 |
SEP341,TPO342 |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6G33B
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iioo |
5ID |
Type1 |
148 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6G33C
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oioi |
5ID |
Type1 |
148 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6I5KA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_oioo |
H3H |
Type1 |
148 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6I5LA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_oioo |
H3Q |
Type1 |
148 - 483 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6Q8PB
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oion |
HQB |
Type1 |
148 - 483 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6RAAA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
JWN |
Type1 |
148 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6TW2E
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanao |
APEdist_oioo |
V25 |
Type1 |
148 - 484 |
0 |
SEP341,TPO342 |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6Z50A
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q7K |
Type1 |
149 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
8P04A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaono |
APEdist_nnni |
WAK |
Type1 |
148 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
8P08A
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_iioo |
WAZ |
Type1 |
148 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
8UWNA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaino |
APEdist_oioo |
XQX |
Type1 |
148 - 482 |
0 |
SEP341,TPO342 |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6KHDB
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
3NG |
Type1 |
149 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
5J1WC
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_oioo |
6FB,
6FB
|
Type1,
Allosteric
|
148 - 483 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK1
|
CLK1_HUMAN
|
6KHDA
|
2.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_ioon |
3NG |
Type1 |
149 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK1 |
|
CMGC
|
CLK2
|
CLK2_HUMAN
|
6KHEA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NG |
Type1 |
144 - 485 |
0 |
None |
None |
Dual specificity protein kinase CLK2 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6FT7A
|
2.02 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E6Q |
Type1 |
129 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6FT7B
|
2.02 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E6Q |
Type1 |
129 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6RCTA
|
2.32 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiii |
JWN |
Type1 |
135 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6RCTB
|
2.32 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiii |
JWN |
Type1 |
134 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6Z52A
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
Q8T |
Type1 |
129 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6Z52B
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
Q8T |
Type1 |
129 - 482 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6Z53A
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
Q7Z |
Type1 |
134 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6Z54A
|
1.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
Q7H |
Type1 |
134 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
3RAWB
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
3RA |
Type1 |
136 - 484 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6Z2VA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
KHC |
Type1 |
134 - 480 |
0 |
None |
A319V |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
6KHFA
|
2.598 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
3NG |
Type1 |
142 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
9EZ3A
|
2.7 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
A1H74 |
Type2 |
136 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
2EXEA
|
2.35 |
Inactive |
None‑None |
DFGAsp-rot-in |
none-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
198 - 479 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
|
CMGC
|
CLK4
|
CLK4_HUMAN
|
AF-Q9HAZ1-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
151 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK4 |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3JUHA
|
1.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
2 - 335 |
0 |
None |
V66A,M163L |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4NH1A
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ACP |
ATPlike |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4NH1B
|
3.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ACP |
ATPlike |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
2PVRA
|
1.605 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
2 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3WOWA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
1JWHA
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
2 - 337 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3U87A
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8AECA
|
1.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP,
LW3
|
ATPlike,
Allosteric
|
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7ZY5A
|
1.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1NP |
Allosteric |
2 - 327 |
0 |
None |
R21S |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HL0A
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVS |
Allosteric |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6FVFA
|
1.47 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
503,
ATP
|
Allosteric,
ATPlike
|
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6FVGA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E8K,
ATP
|
Allosteric,
ATPlike
|
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5OULA
|
1.34 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
AWE,
AWE,
AWE,
AWE,
AWE,
AWE
|
Allosteric,
Allosteric,
Allosteric,
Allosteric,
Type1,
Allosteric
|
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HYHA
|
1.96 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
SY4,
3NG
|
Allosteric,
Type1
|
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HKSA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVR,
A1IVR
|
Allosteric,
Type1
|
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HL0B
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVS,
A1IVS
|
Allosteric,
Type1
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3W8LA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 329 |
0 |
None |
I57V |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3Q04A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3FWQA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3FWQB
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4IB5A
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4IB5C
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6SPXA
|
1.994 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7B8IA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7B8IB
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3QA0A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3QA0B
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
1JWHB
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 336 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5CVGA
|
1.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 329 |
0 |
None |
R21S |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4DGLC
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 335 |
0 |
None |
Y125R |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4DGLD
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 330 |
0 |
None |
Y125R |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7PSUA
|
1.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7PSUB
|
1.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6SPWA
|
1.599 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9RCYA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 330 |
0 |
None |
R21Q |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9RCYB
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 329 |
0 |
None |
R21Q |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9RCXA
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 331 |
0 |
None |
T127M |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9RCXB
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 330 |
0 |
None |
T127M |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4MD9F
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 330 |
0 |
None |
F121E |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4MD9K
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 330 |
0 |
None |
F121E |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4MD9L
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 330 |
0 |
None |
F121E |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4MD9M
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 332 |
0 |
None |
F121E |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9RFNA
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 331 |
0 |
None |
E264D |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9RFNB
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 331 |
0 |
None |
E264D |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5ZN3A
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 329 |
0 |
None |
C147A,H148S,C220A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6L24A
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1 |
2 - 335 |
0 |
None |
H115Y,V116I |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6Q4QB
|
1.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
BEZ |
Type1 |
3 - 329 |
0 |
None |
R21S |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9I0ZA
|
1.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IYU |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9I11A
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IYW |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9I12A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IYX |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5KU8B
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6XK |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3RPSA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4B0 |
Type1 |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3U9CA
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
04G |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3U9CB
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
04G |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4RLLA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E91 |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4UBAA
|
2.995 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3G5 |
Type1 |
2 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4UBAB
|
2.995 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3G5 |
Type1 |
2 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5CQUA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
JRJ |
Type1 |
2 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5CQWA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JRJ |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5CQWB
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JRJ |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5M44A
|
2.71 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7EY |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5M4CA
|
1.935 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7EY |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5M4IA
|
2.218 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7FC |
Type1 |
3 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5N9KA
|
1.643 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8QK |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5N9LA
|
1.79 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8QH |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5N9NA
|
1.841 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
KC5 |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HBNB
|
1.59 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FXB |
Type1 |
3 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7A4BA
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QXW |
Type1 |
2 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7A4BB
|
2.06 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QXW |
Type1 |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7A4CA
|
2.502 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QWW |
Type1 |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7A4CB
|
2.502 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QWW |
Type1 |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7B8HA
|
1.34 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NIO |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3NGAA
|
2.71 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3NGAB
|
2.71 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3U4UA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
LNH |
Type1 |
2 - 328 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4GUBA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0Y4 |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5H8BA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5Y2 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5H8BB
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5Y2 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5H8EB
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5Y3 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5H8GA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5Y4 |
Type1 |
3 - 328 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5KWHB
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6XT |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5T1HA
|
2.11 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
75E |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5T1HB
|
2.11 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
75E |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6QY7B
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
041 |
Type1 |
2 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8BGCA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QIA |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8BGCB
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QIA |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8P06A
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
WAU |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8P07B
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
WAP |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8PVOA
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FW3 |
Type1 |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8PVOB
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FW3 |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8PVPA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FWU |
Type1 |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8PVPB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FWU |
Type1 |
4 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8QWYA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
X59 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8QWZA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
X5E |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPVA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6H |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPVB
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6H |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPXA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1H6E |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPXB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6E |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPYA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6G |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPYB
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6G |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPZA
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1H6I |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EPZB
|
2.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6I |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EZGA
|
2.18 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1H8C |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9EZGB
|
2.18 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1H8C |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3Q9XB
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EMO |
Type1 |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3Q9YA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TXQ |
Type1 |
3 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
4KWPA
|
1.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EXX |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HNYA
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
GHT |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HOQA
|
1.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
FER |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HORA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
GJK |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HOTA
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CIY |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HOUA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
V55 |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6RB1A
|
1.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
JWQ |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6RCBA
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
JYZ |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6RCMA
|
1.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
K0N |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6RFEA
|
1.54 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
K0Z |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6RFFA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
K1B |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8C6LA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
TO6 |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8C6NA
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
TN0 |
Type1 |
3 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
2ZJWA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
REF |
Type1 |
1 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3AMYA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
AGI |
Type1 |
2 - 328 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3WIKA
|
1.995 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
LCT |
Type1 |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5B0XA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
HCK |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6A1CA
|
1.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
9NX |
Type1 |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6JWAA
|
1.781 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5ID |
Type1 |
2 - 328 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6L1ZA
|
1.908 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1 |
2 - 330 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3PE1A
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
3 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3PE2A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E1B |
Type1 |
3 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
3R0TA
|
1.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
FU9 |
Type1 |
3 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5N1VA
|
2.52 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8GQ |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5N1VB
|
2.52 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8GQ |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7AY9A
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
S92 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7AY9B
|
2.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
S92 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7AYAA
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
S8W |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7AYAB
|
2.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
S8W |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6HMEB
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
FXB |
Type1 |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6TEIA
|
1.756 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
N4N |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6TEIB
|
1.756 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
N4N |
Type1 |
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8QQBA
|
2.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
WJE |
Type1 |
2 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9H9DA
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1ITG |
Type1 |
2 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9H9DB
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1ITG |
Type1 |
2 - 329 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6Z83AAA
|
2.171 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QBE |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6Z83BBB
|
2.171 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QBE |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8C5QA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
TL0 |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
8C5QB
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
TL0 |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HKPB
|
2.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVQ |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QRHB
|
2.59 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9M |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QRIB
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9N |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QRJA
|
2.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9O |
Type1 |
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QRJB
|
2.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9O |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSRA
|
2.83 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I90 |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSSA
|
2.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9Z |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSSB
|
2.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9Z |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSTA
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I91 |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSUB
|
2.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I92 |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSVB
|
2.78 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I93 |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6L23A
|
1.974 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1 |
2 - 335 |
0 |
None |
V116I |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6YUMAAA
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PQ8 |
Type1 |
3 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6YUMGGG
|
2.75 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PQ8 |
Type1 |
3 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6TLPA
|
1.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7M0 |
Type1 |
2 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6YPGA
|
1.51 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
N5Q |
Type1 |
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7I8NA
|
1.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1BZX |
Type1 |
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7I8PA
|
1.25 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1BZV |
Type1 |
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QQXA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I9L |
Type1 |
3 - 329 |
0 |
None |
R21S,K74A,K75A,K76A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5NQCA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1KP,
1KP
|
Type1,
Allosteric
|
4 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7X4HA
|
1.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8BH,
8BH
|
Type1,
Allosteric
|
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7AT5A
|
1.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RXE,
42J
|
Type1,
Allosteric
|
2 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7AT5B
|
1.77 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RXE,
42J
|
Type1,
Allosteric
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HYHB
|
1.96 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG,
SY4
|
Type1,
Allosteric
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HZHA
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG,
T9Y
|
Type1,
Allosteric
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HZHB
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG,
T9Y
|
Type1,
Allosteric
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HKSB
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVR,
A1IVR
|
Type1,
Allosteric
|
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HL7B
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVT,
A1IVT
|
Type1,
Allosteric
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9HL7C
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IVT,
A1IVT
|
Type1,
Allosteric
|
2 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6TLRA
|
1.64 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NKE,
NKE
|
Type1,
Type1
|
2 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6L22A
|
2.123 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1.5_Back |
2 - 335 |
0 |
None |
H115Y |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
5OWHA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B0K |
Type1.5_Back |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
7BU4A
|
1.702 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
Y49 |
Type1.5_Back |
2 - 335 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
6L21A
|
2.055 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1.5_Back |
2 - 332 |
0 |
None |
H160A |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A1
|
CSK21_HUMAN
|
9QSTB
|
2.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I91 |
Type1 |
3 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
8QCGA
|
1.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
7 - 330 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
8Q77A
|
1.255 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
LN3,
LN3
|
Allosteric,
Type1
|
7 - 334 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
8QBUA
|
1.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
42J,
3NG
|
Allosteric,
Type1
|
6 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9IHIA
|
1.23 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
SY4,
3NG
|
Allosteric,
Type1
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q9BA
|
1.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VN9,
3NG
|
Allosteric,
Type1
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9QB6A
|
1.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RDV,
3NG
|
Allosteric,
Type1
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7AT9A
|
1.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
42J,
4B0,
42J
|
Allosteric,
Type1,
Allosteric
|
6 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9QABA
|
0.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RA7,
3NG,
RA7
|
Allosteric,
Type1,
Allosteric
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6L20A
|
3.087 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1 |
8 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6L20D
|
3.087 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
E3U |
Type1 |
8 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7XYHA
|
2.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8BH |
Type1 |
8 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7XYHB
|
2.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8BH |
Type1 |
8 - 332 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
5OOIA
|
1.998 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
9YE |
Type1 |
5 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
5OOIB
|
1.998 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
9YE |
Type1 |
7 - 331 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6HMBA
|
1.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
7 - 334 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6HMCA
|
1.03 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
FXB |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6HMQA
|
0.97 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4B0 |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6TE2A
|
0.922 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
N4N |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6TEWA
|
1.082 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
N5Q |
Type1 |
8 - 332 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
6TGUA
|
0.833 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
N92 |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7A1BA
|
1.287 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QXW |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7A1ZA
|
1.024 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QWN |
Type1 |
7 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7A22A
|
1.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QWW |
Type1 |
6 - 333 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
7A2HA
|
1.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QX2 |
Type1 |
7 - 331 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
8Q9SA
|
1.352 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QBE |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
8QCDA
|
1.03 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
TBS |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
8QF1A
|
1.32 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
GNP |
Type1 |
7 - 329 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9FBIA
|
1.161 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NIO |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9FBIB
|
1.161 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NIO |
Type1 |
5 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9GXYA
|
1.16 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IKB |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9H96A
|
1.04 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1ITG |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9R57A
|
1.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7M0 |
Type1 |
7 - 334 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9R5DA
|
1.02 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JC0 |
Type1 |
7 - 334 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9R5FA
|
1.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JCX |
Type1 |
6 - 334 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
5M56A
|
2.237 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7FC |
Type1 |
2 - 332 |
0 |
None |
D39G,C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q8QA
|
0.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I4N |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q9CA
|
1.66 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R9D |
Type1 |
7 - 334 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9QAKA
|
0.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1I5I |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9QB0A
|
1.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
U8X |
Type1 |
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9HK5A
|
1.491 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
7 - 334 |
0 |
None |
P32V,V83I,T101I,C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q9AA
|
1.03 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG,
A1I4V
|
Type1,
Allosteric
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q9DA
|
0.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG,
R9G
|
Type1,
Allosteric
|
7 - 332 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9QAGA
|
1.01 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG,
RBJ
|
Type1,
Allosteric
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q8CA
|
0.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
T9Y,
T9Y,
T9Y
|
Type1,
Allosteric,
Allosteric
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
9Q9GA
|
0.94 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R9J,
R9J,
R9J
|
Type1,
Allosteric,
Allosteric
|
7 - 333 |
0 |
None |
C336S |
Casein kinase II subunit alpha' |
|
CMGC
|
CSNK2A2
|
CSK22_HUMAN
|
3E3BX
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CCK |
Type1 |
1 - 334 |
0 |
None |
None |
Casein kinase II subunit alpha' |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6UIPB
|
3.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q8J |
Type1 |
136 - 478 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6UIPC
|
3.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
Q8J |
Type1 |
131 - 477 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7A4OB
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
ATPlike |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EILC
|
2.465 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
No_ligand |
No_ligand |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7A52A
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QYB |
Type1 |
148 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7OY6C
|
2.38 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
39I |
Type1 |
135 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AJVA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKK |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AJVB
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKK |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AJYA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKZ |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AJYB
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKZ |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AK2A
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RHH |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AK2B
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RHH |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AKAA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RK2 |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AKAB
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RK2 |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AKBA
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RJZ |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AKBB
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RJZ |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AKEA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RK8 |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7AKEB
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RK8 |
Type1 |
148 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
4MQ2D
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
2C4 |
Type1 |
135 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
8R8EA
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
YOX |
Type1 |
135 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHSA
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
4VZ |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHSC
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4VZ |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHSD
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
4VZ |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHTA
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4WD |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHTB
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4WD |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHTC
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
4WD |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7FHTD
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
4WD |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANQA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
EHB |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANQB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
EHB |
Type1 |
133 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANQC
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
EHB |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANQD
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
EHB |
Type1 |
136 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANRB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
HRM |
Type1 |
133 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANRC
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
HRM |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
3ANRD
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
HRM |
Type1 |
134 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
4NCTA
|
2.597 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
2K2 |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
4NCTB
|
2.597 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
2K2 |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
4NCTC
|
2.597 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
2K2 |
Type1 |
134 - 479 |
0 |
SEP301,PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
4NCTD
|
2.597 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
2K2 |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A3XA
|
2.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
QIV |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A3XB
|
2.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
QIV |
Type1 |
133 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A3XC
|
2.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
QIV |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A3XD
|
2.26 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
QIV |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A4EC
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
7QQ |
Type1 |
134 - 473 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A4LB
|
2.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
ZC3 |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A4LC
|
2.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
ZC3 |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A4QA
|
2.37 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
Y3L |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A4QC
|
2.37 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
Y3L |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A4TC
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
AJG |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
5A54C
|
2.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
5PW |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIFB
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
B5T |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIFC
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
B5T |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIFD
|
2.22 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
B5T |
Type1 |
134 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIJA
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5Z |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EILB
|
2.465 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6B |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EILD
|
2.465 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6B |
Type1 |
134 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIPA
|
2.56 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B7B |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIPC
|
2.56 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
B7B |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIQA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6Z |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIQB
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
B6Z |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIQC
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
B6Z |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIRA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6H |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIRB
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
B6H |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIRC
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6H |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIRD
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
B6H |
Type1 |
134 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EISA
|
2.36 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6N |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EISC
|
2.36 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6N |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIVA
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6Q |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIVB
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
B6Q |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIVC
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
B6Q |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIVD
|
2.68 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B6Q |
Type1 |
134 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EJ4A
|
2.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B7W |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EJ4B
|
2.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B7W |
Type1 |
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EJ4D
|
2.88 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
B7W |
Type1 |
134 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6YF8C
|
3.198 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
OPW |
Type1 |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7A4WB
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
QYH |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7A55B
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
QZ2 |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7A5BB
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
MFR |
Type1 |
134 - 481 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7O7KA
|
1.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6ZV,
LI
|
Type1,
Allosteric
|
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
7O7KB
|
1.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
6ZV,
LI
|
Type1,
Allosteric
|
133 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6EIJC
|
2.42 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
B5Z |
Type1.5_Front |
135 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
6UIPA
|
3.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q8J |
Type1 |
131 - 479 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
9FT2A
|
2.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IE6 |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
9FT3A
|
2.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IE7 |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
9FT4A
|
3.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IFJ |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
9FT6A
|
3.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IE8 |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1A
|
DYR1A_HUMAN
|
9FUFA
|
2.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1IFO |
Type1 |
134 - 480 |
0 |
PTR321 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
|
CMGC
|
DYRK1B
|
DYR1B_HUMAN
|
8C2ZA
|
1.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
QS0 |
Type1 |
88 - 434 |
0 |
PTR273 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
9MC0A
|
2.87 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1ENX |
Type1 |
151 - 537 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
3K2LA
|
2.36 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
146 - 543 |
0 |
SEP232,TPO381,PTR382,SEP442,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DG4A
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H5R |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DH9A
|
2.194 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7F |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DHCA
|
2.592 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H99 |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DHHA
|
2.486 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7L |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DHKA
|
2.341 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7O |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DHNA
|
2.38 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7R |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DHOA
|
3.29 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7U |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DJOA
|
2.499 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H80 |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DL6A
|
2.648 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H96 |
Type1 |
215 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DH3A
|
2.33 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7C |
Type1 |
213 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7DHVA
|
2.679 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
H7X |
Type1 |
212 - 538 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
4AZFA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3RA |
Type1 |
146 - 536 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
9MC0B
|
2.87 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1ENX |
Type1 |
151 - 537 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7EJVB
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YK2 |
Type1 |
153 - 543 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
3KVWA
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
IRB |
Type1 |
146 - 536 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
5ZTNA
|
2.496 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CUR |
Type1 |
146 - 536 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
5ZTNB
|
2.496 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CUR |
Type1 |
146 - 536 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
6HDPA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
FZ5 |
Type1 |
146 - 542 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
6HDRA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CC9 |
Type1 |
146 - 536 |
0 |
PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
7AKFA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RK5 |
Type1 |
146 - 535 |
0 |
SEP232,PTR382,SEP458 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
5LXCA
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7AA |
Type1 |
153 - 536 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
5LXCB
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7AA |
Type1 |
153 - 538 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
5LXDA
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7A7 |
Type1 |
153 - 538 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
5LXDB
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
7A7 |
Type1 |
153 - 538 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
6K0JA
|
2.352 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CQO |
Type1 |
212 - 536 |
0 |
PTR382,SEP458 |
E256N,L349A |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
9KQYA
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
151 - 537 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
8HLTB
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XSE |
Type1 |
151 - 537 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
DYRK2
|
DYRK2_HUMAN
|
9KQYB
|
3.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1L6I |
Type1 |
151 - 537 |
0 |
PTR382 |
None |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
|
CMGC
|
GSK3A
|
GSK3A_HUMAN
|
7SXGA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D1E |
Type1 |
103 - 445 |
0 |
PTR279 |
None |
Glycogen synthase kinase-3 alpha |
|
CMGC
|
GSK3A
|
GSK3A_HUMAN
|
7SXFA
|
1.94 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6VL |
Type1 |
101 - 444 |
0 |
PTR279 |
None |
Glycogen synthase kinase-3 alpha |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6Y9SA
|
2.03 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
OHK |
Type1 |
35 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6Y9SB
|
2.03 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
OHK |
Type1 |
35 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
4NM0A
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
26 - 383 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
8XN6B
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
26 - 386 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
9X2VA
|
1.39 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiii |
PG6 |
Allosteric |
35 - 383 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
1I09B
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
37 - 382 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6HK7A
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
G8N |
Type1 |
36 - 382 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
7SXHA
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D1E |
Type1 |
37 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
3F7ZA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
34O |
Type1 |
35 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
3SD0A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
TSK |
Type1 |
35 - 384 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
3ZDIA
|
2.645 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
UGJ |
Type1 |
36 - 384 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
4B7TA
|
2.772 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CWT |
Type1 |
35 - 384 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6HK3A
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
G8B |
Type1 |
35 - 384 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6Y9RA
|
2.08 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
OH8 |
Type1 |
35 - 384 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
1O9UA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADZ |
Type1 |
35 - 384 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
9PE9A
|
2.11 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1CIF |
Type1 |
36 - 382 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
9PE9B
|
2.11 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1CIF |
Type1 |
36 - 382 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
7Z1FA
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
28 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
7Z1FB
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
38 - 382 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
8AV1A
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O9L |
Type1 |
27 - 381 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
8AV1B
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O9L |
Type1 |
27 - 381 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6GN1A
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiii |
F4N |
Type1 |
36 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6GN1B
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiii |
F4N |
Type1 |
36 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
2O5KA
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiii |
HBM |
Type1 |
35 - 384 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
1UV5A
|
2.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
BRW |
Type1 |
35 - 383 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6GJOA
|
2.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
F1B |
Type1 |
35 - 383 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
6GJOB
|
2.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
F1B |
Type1 |
35 - 383 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
3M1SA
|
3.134 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
DW1 |
Type1 |
35 - 385 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
9HUKA
|
3.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IXL |
Type1 |
25 - 385 |
0 |
None |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
4J71A
|
2.31 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1JX |
Type1 |
36 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
4J71B
|
2.31 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1JX |
Type1 |
36 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
5HLNB
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
65C |
Type1 |
37 - 383 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
5OY4B
|
3.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4K |
Type1.5_Back |
30 - 384 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
GSK3B
|
GSK3B_HUMAN
|
8QJIA
|
3.02 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VNG |
Type1 |
36 - 381 |
0 |
PTR216 |
None |
Glycogen synthase kinase-3 beta |
|
CMGC
|
HIPK2
|
HIPK2_HUMAN
|
6P5SA
|
2.194 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3NG |
Type1 |
185 - 535 |
0 |
PTR361,SEP441 |
None |
Homeodomain-interacting protein kinase 2 |
|
CMGC
|
HIPK3
|
HIPK3_HUMAN
|
7O7JA
|
2.81 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6ZV |
Type1 |
184 - 551 |
0 |
PTR359 |
None |
Homeodomain-interacting protein kinase 3 |
|
CMGC
|
HIPK3
|
HIPK3_HUMAN
|
7O7IA
|
2.5 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
184 - 550 |
0 |
PTR359 |
None |
Homeodomain-interacting protein kinase 3 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PVUE
|
3.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
24 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
1WZYA
|
2.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oioo |
F29 |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
1TVOA
|
2.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
FRZ |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4H3QA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioo |
ANP |
ATPlike |
9 - 360 |
0 |
None |
R77A,C161S,I255G,E314A |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZ5A
|
3.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
ADP |
ATPlike |
11 - 357 |
0 |
None |
T185E |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZ5B
|
3.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
ADP |
ATPlike |
11 - 357 |
0 |
None |
T185E |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZ5C
|
3.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
ADP |
ATPlike |
11 - 357 |
0 |
None |
T185E |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZ5D
|
3.19 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
ADP |
ATPlike |
11 - 357 |
0 |
None |
T185E |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
2Y9QA
|
1.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
9 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FMQA
|
2.098 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
9 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4NIFB
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
9 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4NIFE
|
2.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
10 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PSRA
|
1.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
1 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
3TEIA
|
2.404 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
10 - 358 |
0 |
None |
R77A,E314A |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4H3PA
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
11 - 359 |
0 |
None |
R77A,E314A |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4H3PD
|
2.3 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ANP |
ATPlike |
11 - 359 |
0 |
None |
R77A,E314A |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
9TYGB
|
2.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
ADP |
ATPlike |
11 - 360 |
0 |
None |
T185V |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PSTA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
AN2,
DC6
|
ATPlike,
Allosteric
|
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PSWA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
AN2,
D2I
|
ATPlike,
Allosteric
|
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PSYA
|
2.55 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
AN2,
EI0
|
ATPlike,
Allosteric
|
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PT0A
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
ANP,
EAI
|
ATPlike,
Allosteric
|
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PT1A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP,
E2A
|
ATPlike,
Allosteric
|
11 - 359 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PT5A
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP,
D5R
|
ATPlike,
Allosteric
|
10 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8R5FA
|
1.65 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ANP,
Y3H
|
ATPlike,
Allosteric
|
11 - 359 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7W5OB
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_ioii |
6GI |
Allosteric |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8PT3A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
D7O,
ANP
|
Allosteric,
ATPlike
|
10 - 359 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QAHA
|
1.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
HVB,
HVB
|
Allosteric,
Allosteric
|
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QALA
|
1.57 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
HV2,
HV2
|
Allosteric,
Allosteric
|
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6NBSA
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
KJ7,
KJ4
|
Allosteric,
Allosteric
|
10 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOGA
|
1.603 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N29,
N29,
N29
|
Allosteric,
Allosteric,
Type1
|
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G8XA
|
1.76 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
EQT,
EQT
|
Allosteric,
Type1
|
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QA1A
|
1.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
HVK,
HVK,
HVK,
HVK,
HVK,
HVK,
HVK
|
Allosteric,
Type1,
Allosteric,
Allosteric,
Allosteric,
Allosteric,
Allosteric
|
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QA4A
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
HRZ,
HRZ,
HRZ,
HRZ
|
Allosteric,
Type1,
Allosteric,
Type3
|
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZ7A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
11 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZ7C
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
No_ligand |
No_ligand |
11 - 359 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZAA
|
1.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
No_ligand |
No_ligand |
11 - 358 |
0 |
TPO185,PTR187 |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4IZAC
|
1.93 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-none |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
11 - 358 |
0 |
TPO185,PTR187 |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6Q7SA
|
1.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QA3A
|
1.57 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP2B
|
2.23 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
No_ligand |
No_ligand |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
9TYIB
|
3.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
11 - 360 |
0 |
None |
T185V |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7E73A
|
2.28 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
11 - 357 |
0 |
None |
Y36H |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7E75A
|
2.481 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
10 - 358 |
0 |
None |
G37C |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6D5YA
|
2.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
13 - 357 |
0 |
None |
G169D |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
1PMEA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
SB2 |
Type1 |
16 - 360 |
0 |
None |
I103L,Q105T,D106H,E109G,T110A |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6DMGA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK6 |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4XJ0A
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_ioii |
41B |
Type1 |
12 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4XJ0B
|
2.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_ioii |
41B |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8ZJVA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5ID |
Type1 |
10 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5K4IA
|
1.76 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
6QB |
Type1 |
9 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
3SA0A
|
1.595 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
NRA |
Type1 |
4 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FUXA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E75 |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FUYA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK2 |
Type1 |
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FV0A
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK3 |
Type1 |
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FV1A
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK4 |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FV2A
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK5 |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FV3A
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK6 |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4FV7A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E94 |
Type1 |
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4G6NA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EK0 |
Type1 |
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4G6OA
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E28 |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4N0SA
|
1.799 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
DHC |
Type1 |
6 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4ZXTA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
CAQ |
Type1 |
7 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5LCKA
|
1.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
6TT |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G54A
|
2.05 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6H3 |
Type1 |
10 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5LCJA
|
1.78 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
6TS |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G91A
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EQW |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G92A
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ERZ |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G93A
|
1.67 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EU2 |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G97A
|
1.9 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EQZ |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9AA
|
1.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ESQ |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9MA
|
1.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ESW |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6GDQA
|
1.86 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EVK |
Type1 |
10 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6GJBA
|
1.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F0H |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6Q7KA
|
1.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2AI |
Type1 |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QAWA
|
1.84 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
HVE |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6RQ4A
|
1.96 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
KE8 |
Type1 |
19 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7NR3A
|
1.897 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
UO5 |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO2A
|
1.796 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
NXI |
Type1 |
13 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO3A
|
1.778 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
NYX |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO4A
|
1.825 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N8U |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO5A
|
1.595 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N6K |
Type1 |
15 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO6A
|
1.811 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N9F |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO7A
|
1.61 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N3X |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO8A
|
1.697 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N5U |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AO9A
|
1.624 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N4F |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOBA
|
1.623 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
NB3 |
Type1 |
18 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOCA
|
1.62 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N3O |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOEA
|
1.687 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N6U |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOFA
|
1.615 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N4U |
Type1 |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOJA
|
1.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N8L |
Type1 |
10 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
3W55A
|
3.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnoo |
1FM |
Type1 |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5AX3A
|
2.984 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aanii |
APEdist_iion |
5ID |
Type1 |
10 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7W5OA
|
2.35 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_ioii |
5ID |
Type1 |
11 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7XC1B
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_ioii |
5ID |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4O6EA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
2SH |
Type1 |
13 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP1A
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
EMU |
Type1 |
12 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP1B
|
2.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
EMU |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP2A
|
2.23 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
36R |
Type1 |
12 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP3A
|
2.599 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioi |
36Q |
Type1 |
12 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP3B
|
2.599 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
36Q |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP4A
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
36O |
Type1 |
13 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP4B
|
2.2 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
36O |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP6A
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
36N |
Type1 |
12 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP6B
|
3.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
36N |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP7A
|
2.249 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
363 |
Type1 |
13 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP7B
|
2.249 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
363 |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP8A
|
2.446 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
362 |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP8B
|
2.446 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
362 |
Type1 |
13 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QP9A
|
2.001 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
35X |
Type1 |
13 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QPAA
|
2.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
35W |
Type1 |
12 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QPAB
|
2.85 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
35W |
Type1 |
12 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4ZZMA
|
1.89 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
CQ6 |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4ZZNA
|
1.33 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
CQ8 |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4ZZOA
|
1.63 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
CQ3 |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
2OJGA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
19A |
Type1 |
19 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
2OJIA
|
2.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
33A |
Type1 |
15 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
2OJJA
|
2.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
82A |
Type1 |
15 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
9LNRA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1EKR |
Type1 |
9 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NGUA
|
2.74 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8X2 |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHFA
|
2.14 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8X5 |
Type1 |
12 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHHA
|
1.94 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8XH |
Type1 |
11 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHJA
|
2.12 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8XE |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHLA
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8XB |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHOA
|
2.24 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8XN |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHPA
|
1.99 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8XK |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5NHVA
|
2.0 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8QB |
Type1 |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6SLGA
|
1.33 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
LHZ |
Type1 |
18 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
5WP1A
|
1.4 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
B7S,
BEZ
|
Type1,
Allosteric
|
15 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6Q7TA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
HOW,
HOW
|
Type1,
Allosteric
|
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QAGA
|
2.07 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
HUH,
HUH
|
Type1,
Allosteric
|
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOAA
|
1.62 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N83,
OZU
|
Type1,
Allosteric
|
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AODA
|
1.62 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
NY0,
NYI
|
Type1,
Allosteric
|
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOHA
|
1.6 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
N96,
N96
|
Type1,
Allosteric
|
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
8AOIA
|
1.602 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
NX0,
NX0
|
Type1,
Allosteric
|
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7XC1A
|
2.09 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_ioii |
5ID,
B8Z
|
Type1,
Allosteric
|
10 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7X4UA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5ID,
8DK,
BTB
|
Type1,
Allosteric,
Allosteric
|
10 - 359 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
4QTAA
|
1.45 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
38Z |
Type1.5_Front |
10 - 358 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9DA
|
1.8 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ER8 |
Type1.5_Front |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9HA
|
1.73 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ERW |
Type1.5_Front |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9JA
|
1.98 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ERK |
Type1.5_Front |
8 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9KA
|
1.94 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ESK |
Type1.5_Front |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6G9NA
|
1.76 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
ESN |
Type1.5_Front |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6GDMA
|
1.91 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F3Z |
Type1.5_Front |
8 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6GE0A
|
1.82 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EVQ |
Type1.5_Front |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6GJDA
|
1.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F0E |
Type1.5_Front |
10 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7AUVA
|
1.76 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RYW |
Type1.5_Front |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7NQQA
|
1.943 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
UMN |
Type1.5_Front |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7NQWA
|
1.775 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
UNW |
Type1.5_Front |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7NR5A
|
1.766 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
UOH |
Type1.5_Front |
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7NR8A
|
1.627 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
UOE |
Type1.5_Front |
11 - 356 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
7NR9A
|
1.906 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
UOW |
Type1.5_Front |
11 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
6QAQA
|
1.58 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HVQ,
HVQ
|
Type3,
Allosteric
|
11 - 357 |
0 |
None |
None |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK1
|
MK01_HUMAN
|
9TYHB
|
3.4 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-in |
in-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
ADP |
ATPlike |
11 - 360 |
0 |
None |
T185V |
Mitogen-activated protein kinase 1 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8WGFA
|
1.85 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ANP |
ATPlike |
44 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4KKEA
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
AMP |
ATPlike |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EQ9B
|
1.83 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ACP |
ATPlike |
47 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
1JNKA
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ANP |
ATPlike |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EQ9A
|
1.83 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ACP,
C15
|
ATPlike,
Allosteric
|
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4Z9LA
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ANP,
880
|
Allosteric,
Type1
|
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4KKGA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3FI2A
|
2.28 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
JK1 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3FV8A
|
2.28 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
JK3 |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2B1PA
|
1.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
AIZ |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2R9SA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
255 |
Type1 |
46 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2R9SB
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
255 |
Type1 |
46 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2EXCX
|
2.75 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
JNK |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3OY1A
|
1.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
589 |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3RTPA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
34I |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2O2UA
|
2.45 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
738 |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2WAJA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
SNB |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2ZDTA
|
2.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
46C |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2ZDUA
|
2.5 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
446 |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3FI3A
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
JK2 |
Type1 |
45 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3KVXA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
FMY |
Type1 |
46 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3V6RA
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
CQQ |
Type1 |
45 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3V6RB
|
2.6 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
CQQ |
Type1 |
45 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3V6SA
|
2.97 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0F0 |
Type1 |
45 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3V6SB
|
2.97 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnno |
0F0 |
Type1 |
45 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
1PMNA
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
984 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
1PMUA
|
2.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
9HP |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7ORFA
|
1.7 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
0G3 |
Type1 |
45 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2OK1A
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
33A |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2P33A
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
J07 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3CGFA
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
JNF |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3CGOA
|
3.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
JNO |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3G90X
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
J72 |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3G9LX
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
J67 |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3G9NA
|
2.8 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
J88 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4KKHA
|
2.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
1RQ |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4W4VA
|
2.01 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
3H8 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4W4WA
|
1.9 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
3HJ |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4W4XA
|
2.65 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
3HN |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4W4YA
|
2.3 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
3HQ |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4Y46A
|
2.04 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
4F2 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4Y5HA
|
2.055 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
519 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4X21A
|
1.95 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3WH |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4X21B
|
1.95 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3WH |
Type1 |
47 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EKDA
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
B9K |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EMHC
|
1.76 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
BGE |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EMHD
|
1.76 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
BGE |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4WHZA
|
1.79 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
3NL |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3TTIA
|
2.2 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
KBI |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3TTJA
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
JBI |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7KSIA
|
1.726 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X3S |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7KSJA
|
2.06 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X3Y |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7KSKA
|
1.84 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_onoo |
X3V |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7S1NA
|
2.11 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
86C |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7YL1A
|
2.48 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
J6F |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8ENJA
|
2.81 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
WNK |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8VNXA
|
2.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
WHQ |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8VO4A
|
2.07 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
WHE |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8VTFA
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
A1ACP |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8BZPA
|
1.86 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_onno |
SWM,
C15
|
Type1,
Allosteric
|
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EMHA
|
1.76 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
BGE,
C15
|
Type1,
Allosteric
|
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
6EMHB
|
1.76 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
BGE,
C15
|
Type1,
Allosteric
|
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
7OREA
|
2.18 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
0EI,
0EI
|
Type1,
Type1
|
44 - 402 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8BZPB
|
1.86 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
SWM,
C15,
C15
|
Type1,
Type1,
Allosteric
|
47 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
2O0UA
|
2.1 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
C0M |
Type1.5_Back |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3DA6A
|
2.0 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
BZ9 |
Type1.5_Front |
46 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4U79A
|
2.23 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3EL |
Type1.5_Front |
44 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4H39A
|
1.992 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnno |
No_ligand |
No_ligand |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4H36A
|
3.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4H3BA
|
2.08 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
4H3BC
|
2.08 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3OXIA
|
2.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
SYY |
Type1 |
46 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
3PTGA
|
2.43 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
932 |
Type1 |
46 - 401 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
1PMVA
|
2.5 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
537 |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK10
|
MK10_HUMAN
|
8VS0A
|
2.46 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
A1ACT |
Type1 |
45 - 400 |
0 |
None |
None |
Mitogen-activated protein kinase 10 |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
3GC9B
|
2.05 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
B45 |
Type1 |
2 - 349 |
0 |
None |
C119S,C162S |
Mitogen-activated protein kinase 11 |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
3GC8A
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
B45 |
Type1 |
3 - 349 |
0 |
None |
C162S |
Mitogen-activated protein kinase 11 |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
3GC8B
|
2.4 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
B45 |
Type1 |
4 - 349 |
0 |
None |
C162S |
Mitogen-activated protein kinase 11 |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
3GC9A
|
2.05 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
B45 |
Type1 |
3 - 348 |
0 |
None |
C119S,C162S |
Mitogen-activated protein kinase 11 |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
3GP0A
|
1.9 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
NIL |
Type2 |
5 - 348 |
0 |
None |
None |
Mitogen-activated protein kinase 11 |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
8YGWA
|
3.301 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
B96 |
Type2 |
5 - 348 |
0 |
None |
None |
Mitogen-activated protein kinase 11 |
|
CMGC
|
MAPK12
|
MK12_HUMAN
|
7CGAB
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
No_ligand |
No_ligand |
9 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 12 |
|
CMGC
|
MAPK12
|
MK12_HUMAN
|
7CGAC
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
No_ligand |
No_ligand |
9 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 12 |
|
CMGC
|
MAPK12
|
MK12_HUMAN
|
7CGAD
|
3.15 |
Inactive |
DFGin‑ABAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
No_ligand |
No_ligand |
9 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 12 |
|
CMGC
|
MAPK12
|
MK12_HUMAN
|
7CGAA
|
3.15 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
No_ligand |
No_ligand |
9 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 12 |
|
CMGC
|
MAPK12
|
MK12_HUMAN
|
6UNAA
|
2.554 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
10 - 351 |
0 |
None |
Q31R |
Mitogen-activated protein kinase 12 |
|
CMGC
|
MAPK12
|
MK12_HUMAN
|
6UNAB
|
2.554 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
9 - 351 |
0 |
None |
Q31R |
Mitogen-activated protein kinase 12 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
8X23A
|
1.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
4YNOA
|
1.7 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
3COIA
|
2.09 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnoo |
No_ligand |
No_ligand |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
4EYMA
|
2.353 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
0RX |
Type1 |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
5EKOA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
N17 |
Type1 |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
4EYJA
|
2.102 |
Inactive |
DFGout‑BBAminus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
N61 |
Type2 |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
5EKNA
|
2.594 |
Inactive |
DFGout‑None |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
N58 |
Type2 |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HVCA
|
2.1 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WBWA
|
2.41 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
LI4 |
Type1 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6ZQSA
|
1.95 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3FF |
Type1 |
4 - 353 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6TCAB
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
39G |
Type1.5_Back |
6 - 354 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6TCAD
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioi |
39G |
Type1.5_Back |
4 - 353 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6TCAF
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
39G |
Type1.5_Back |
6 - 353 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6TCAH
|
3.7 |
Inactive |
DFGin‑BLAminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
39G |
Type1.5_Back |
4 - 353 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HUBA
|
2.25 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
469 |
Type1 |
4 - 352 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3UVPA
|
2.4 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
048 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3UVQA
|
2.2 |
Inactive |
DFGin‑BLAplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FS8 |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5N68A
|
1.85 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
8OK |
Allosteric |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
8YD9A
|
1.66 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
6GI |
Allosteric |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2Y8OA
|
1.95 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 353 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1R3CA
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
4 - 352 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2LGCA
|
999.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
2 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5ETAA
|
2.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5ETAB
|
2.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9CJ2B
|
2.83 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 352 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1R39A
|
2.3 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2OKRA
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
No_ligand |
No_ligand |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2OKRD
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2ONLA
|
4.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2ONLB
|
4.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
No_ligand |
No_ligand |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5ETFA
|
2.4 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
out-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1BMKA
|
2.4 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
SB5 |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MW1A
|
2.8 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
MIH |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1DI9A
|
2.6 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
MSQ |
Type1 |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1W7HA
|
2.214 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
3IP |
Type1 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1W84A
|
2.2 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
L12 |
Type1 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2ZB0A
|
2.1 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
GK3 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1M7QA
|
2.4 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
DQO |
Type1 |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1OUKA
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
084 |
Type1 |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1OUYA
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
094 |
Type1 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1YQJA
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
6NP |
Type1 |
2 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3ZYAA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
out-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
2A8 |
Type1 |
1 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1OZ1A
|
2.1 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FPH |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FLQA
|
1.9 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
891 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FMJA
|
2.0 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FMJ |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FSFA
|
2.1 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FSS |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1A9UA
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
SB2 |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1BL6A
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
SB6 |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1BL7A
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
SB4 |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MPAA
|
2.1 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-none |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
SB2 |
Type1 |
5 - 352 |
0 |
None |
D168G |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2ZB1A
|
2.5 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
GK4 |
Type1.5_Back |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5XYXA
|
2.61 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FTZ |
Type1.5_Back |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5XYYA
|
1.7 |
Inactive |
DFGin‑BLBminus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
P0F |
Type1.5_Back |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3NEWA
|
2.51 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
3NE |
Allosteric |
5 - 352 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4EH2A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
IRG,
0OK
|
Allosteric,
Type1
|
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MH2A
|
2.3 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
F169Y |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5ETIA
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
out-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FI4A
|
2.2 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FI4 |
Type1 |
4 - 352 |
0 |
None |
R57K |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FKOA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FKO |
Type1 |
5 - 352 |
0 |
None |
R57K |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FLNC
|
1.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
3FN |
Type1 |
3 - 352 |
0 |
None |
R57K |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6OHDA
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
MKP |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1OVEA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
358 |
Type1 |
4 - 352 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GC7A
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
B45 |
Type1 |
4 - 352 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3S3IA
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
CQ0 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1ZZLA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
TZY |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2YIXA
|
2.3 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
YIX |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HRBA
|
2.2 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
I39 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1ZYJA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
BI5 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1ZZ2A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
B11 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2ZAZA
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
GK1 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3D7ZA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
GK5 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3IPHA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
G11 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3KF7A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
L9G |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3RINA
|
2.2 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
I2O |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5MTXA
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FJI |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5MTYA
|
2.31 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
HB9 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5TBEA
|
2.44 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
78L |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9D8GA
|
2.13 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
A1IKC |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9Y8BA
|
1.97 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
A1CTD |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5TCOA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
79Q |
Type1 |
6 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9Q5BA
|
2.05 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1CRZ |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6M9LA
|
2.45 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
J9G |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3DS6A
|
2.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
A17 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3DS6B
|
2.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
A17 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3DS6C
|
2.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
A17 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3DS6D
|
2.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A17 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GFEA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
P37 |
Type1 |
1 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3ITZA
|
2.25 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
P66 |
Type1 |
1 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3LHJA
|
3.31 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
LHJ |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3U8WA
|
2.15 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
09J |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2BALA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
PQA |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4AA4A
|
2.3 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
QC0 |
Type1 |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4AA5A
|
2.38 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
NQB |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4AACA
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
AAV |
Type1 |
5 - 359 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2QD9A
|
1.7 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
LGF |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MVLA
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
38P |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MVLB
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
38P |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MVMA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
39P |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MVMB
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
39P |
Type1 |
5 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3NWWA
|
2.09 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
3NW |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3S4QA
|
2.27 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
NK0 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KINA
|
1.97 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_nooo |
1M8 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KINB
|
1.97 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
1M8 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KINC
|
1.97 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1M8 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIND
|
1.97 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1M8 |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIPA
|
2.27 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
1R9 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIPB
|
2.27 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
1R9 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIQA
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
1RA |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIQB
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaino |
APEdist_nnno |
1RA |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIQC
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
1RA |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4KIQD
|
2.5 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaino |
APEdist_nnno |
1RA |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FKLA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FKL |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FKNA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FKN |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FL4A
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FL4 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FLSA
|
2.3 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-in |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FLS |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FLWA
|
2.1 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FLW |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FLYA
|
1.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FLY |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FLZA
|
2.23 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FLZ |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FMHA
|
1.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
533 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FMKA
|
1.7 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FMK |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FMMA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
XI2 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FMNA
|
1.9 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
530 |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3E92A
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
G6A |
Type1 |
3 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MPTA
|
1.89 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
1GK |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3DT1A
|
2.8 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
P40 |
Type1 |
1 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4F9YA
|
1.85 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
LM3 |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HL7A
|
1.88 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
I47,
I46
|
Type1,
Allosteric
|
6 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3ROCA
|
1.7 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
29A,
29B
|
Type1,
Allosteric
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HLLA
|
1.95 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
I45,
I46,
PO2
|
Type1,
Allosteric,
Allosteric
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2I0HA
|
2.0 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
222,
222
|
Type1,
Type1
|
4 - 352 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2RG5A
|
2.4 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
279 |
Type1.5_Back |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3BX5A
|
2.4 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
304 |
Type1.5_Back |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3L8XA
|
2.4 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
N4D |
Type1.5_Back |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2RG6A
|
1.72 |
Inactive |
DFGin‑BLBplus |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
287,
287
|
Type1.5_Back,
Allosteric
|
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4E6AA
|
2.09 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
0O9 |
Allosteric |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4E6CA
|
2.39 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
0O8 |
Allosteric |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5N67A
|
1.9 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
8ON |
Allosteric |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
8X3MA
|
1.85 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
B8Z |
Allosteric |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4DLIA
|
1.91 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
IRG,
IRG
|
Allosteric,
Allosteric
|
5 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4EH4A
|
2.5 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
IRG,
0OL
|
Allosteric,
Type1
|
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3C5UA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnoo |
P41,
P41
|
Allosteric,
Type1
|
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4E5AX
|
1.87 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
3 - 353 |
0 |
None |
W197A |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3OD6X
|
2.682 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
4 - 352 |
0 |
None |
Y323T |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3OEFX
|
1.6 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
Y323F |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3ODYX
|
2.2 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
No_ligand |
No_ligand |
4 - 353 |
0 |
None |
Y323Q |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MGYA
|
2.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-none |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4E5BA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3ODZX
|
2.3 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
No_ligand |
No_ligand |
4 - 353 |
0 |
None |
Y323R |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5ETCA
|
2.422 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WFCA
|
2.3 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
5 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MH0A
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
F169A |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3IW6A
|
2.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
PP0 |
Type1 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3IW7A
|
2.4 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
IPK |
Type1 |
4 - 352 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2BAQA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
PQB |
Type1 |
5 - 351 |
0 |
None |
V30I |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WBOA
|
2.16 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
2CH |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5OMGA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
9Y8 |
Type1 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9YTYA
|
2.25 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
A1BB6 |
Type1 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3QUDA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
N3F |
Type1 |
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3QUEA
|
2.7 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
3FF |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3ZSIA
|
2.4 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
52P |
Type1 |
6 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9MHBA
|
1.65 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
A1BLA |
Type1 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FC1X
|
2.4 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
52P |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3BV2A
|
2.4 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
P38 |
Type1 |
5 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3OCGA
|
2.21 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
OCG |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2GFSA
|
1.752 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
PQB |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FMLA
|
2.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
FML |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3FSKA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
RO6 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HA8A
|
2.48 |
Inactive |
DFGin‑None |
DFGAsp-rot-in |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
5JZ |
Type1 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4F9WA
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
LM4 |
Type1 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4FA2A
|
2.0 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
SB0 |
Type1 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4ZTHA
|
2.15 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
VVT |
Type1 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9O4LA
|
2.27 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
A1B8B |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3O8PA
|
2.1 |
Inactive |
DFGin‑None |
DFGAsp-rot-none |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
BMU |
Type1 |
5 - 351 |
0 |
None |
D168G |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3OBGA
|
2.8 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
SB2 |
Type1 |
5 - 352 |
0 |
None |
F169G |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9D6PA
|
2.13 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1IKD |
Type1 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9D75A
|
2.13 |
Inactive |
DFGin‑None |
DFGAsp-rot-out |
in-in |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
|