|
AGC
|
GRK1
|
GRK1_BOVIN
|
3T8OA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
30 - 532 |
0 |
None |
L166K |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4WA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
31 - 533 |
0 |
TPO8 |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4WB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
5 - 533 |
0 |
TPO8 |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4XA
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
30 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4XB
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
31 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4ZA
|
1.84 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C50A
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
30 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C50B
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
30 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C51A
|
3.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C51B
|
3.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3QC9A
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
T8C,N480C |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3QC9B
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
T8C,N480C |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3QC9C
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
T8C,N480C |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3QC9D
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
31 - 533 |
0 |
None |
T8C,N480C |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4YA
|
7.509 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 532 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4L9IA
|
2.32 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PR |
Type1 |
30 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4L9IB
|
2.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PR |
Type1 |
31 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4WBOA
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANW |
Type1 |
28 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4WBOB
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANW |
Type1 |
30 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4WBOC
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANW |
Type1 |
31 - 531 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4WBOD
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANW |
Type1 |
30 - 531 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
4PNIA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
KQQ |
Type1 |
30 - 533 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
7MT9G
|
7.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
SGV,
SGV,
SGV,
SGV,
SGV,
SGV
|
Type1,
Type1,
Type1,
Type1,
Type1,
Type1
|
6 - 508 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
7MT8G
|
5.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
SGV,
SGV,
SGV,
SGV,
SGV,
SGV
|
Type1,
Type1,
Type1,
Type1,
Type1,
Type1
|
6 - 508 |
0 |
None |
S5E,S488E,T489E |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
7MTAG
|
4.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV,
SGV,
SGV,
SGV,
SGV,
SGV
|
Type1,
Type1,
Type1,
Type1,
Type1,
Type1
|
6 - 508 |
0 |
None |
S5E,S488E,T489E |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
7MTBG
|
4.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV,
SGV,
SGV,
SGV,
SGV,
SGV
|
Type1,
Type1,
Type1,
Type1,
Type1,
Type1
|
6 - 508 |
0 |
None |
S5E,S488E,T489E |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK1
|
GRK1_BOVIN
|
3C4YB
|
7.509 |
Inactive |
DFGinter‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 532 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
1YM7B
|
4.5 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 656 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
8JPBG
|
3.07 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
2 - 659 |
0 |
None |
A292P,R295I,S455D |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
8JPCG
|
3.07 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
2 - 659 |
0 |
None |
A292P,R295I,S455D |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
8JPDG
|
2.81 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
2 - 659 |
0 |
None |
A292P,R295I,S455D |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
5HE0A
|
2.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
453 |
Type1 |
30 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
5HE2A
|
2.79 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F0S |
Type1 |
30 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
5HE3A
|
2.74 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FF1 |
Type1 |
30 - 670 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
5UKMA
|
3.03 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T0E |
Type1 |
31 - 669 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
1OMWA
|
2.5 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
1YM7A
|
4.5 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 656 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
1YM7C
|
4.5 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 656 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
1YM7D
|
4.5 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 656 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
2BCJA
|
3.061 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
28 - 667 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
3UZSA
|
4.52 |
Inactive |
DFGin‑None |
in-out |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 671 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
3UZTA
|
3.51 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 656 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
3PSCA
|
2.67 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
3PVUA
|
2.48 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QRW |
Type1 |
30 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK2
|
ARBK1_BOVIN
|
3PVWA
|
2.49 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QRX |
Type1 |
29 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Bos taurus |
|
AGC
|
GRK5
|
GRK5_BOVIN
|
4WNKA
|
2.42 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
453 |
Type1.5_Front |
24 - 541 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GNIA
|
2.27 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
L50I,V124M,E128D,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1STCE
|
2.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
16 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3ZO2A
|
1.98 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
15I |
Type1 |
8 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3ZO3A
|
2.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QNI |
Type1 |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
5VI9A
|
1.95 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9D4 |
Type1 |
15 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
5VIBA
|
2.37 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9D1 |
Type1 |
19 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1SZMB
|
2.5 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI4 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4AXAA
|
1.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RKD |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4C34A
|
1.78 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
11 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
F55Y,M121L,V124L,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4C37A
|
1.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Z21 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
F55Y,M121L,V124L,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GNHA
|
2.05 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H52,
H52
|
Type1,
Allosteric
|
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
L50I,V124M,E128D,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9DW5G
|
3.8 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
13 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9DW8G
|
3.5 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 329 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9DW9G
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1Q24A
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
15 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2VO7A
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M05,
M05
|
Allosteric,
Type1
|
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GNGA
|
1.87 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
L50I,V124M,E128D,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GFCA
|
1.87 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3AG9A
|
2.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9FQRXT
|
5.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
26 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1Q61A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1SMHA
|
2.044 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
TPO198,SEP339 |
Q85E,V124A,L174M,F188L |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1Q62A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4C33A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
F55Y,M121L,V124L,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GNFA
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y27 |
Type1 |
11 - 351 |
0 |
TPO198,SEP339 |
L50I,V124M,E128D,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GNJA
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y27 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
L50I,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2GNLA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H52 |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
L50I,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UZTA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SS3 |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UZUE
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L20 |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UZVA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SS5 |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UZWE
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SS4 |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1Q8TA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y27 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1Q8WA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1SVEA
|
2.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I01 |
Type1 |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1SVGA
|
2.02 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I04 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1VEBA
|
2.89 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I05 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XH4A
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R69 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XH5A
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R68 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XH6A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R94 |
Type1 |
19 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XH7A
|
2.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R96 |
Type1 |
11 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XH8A
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R55 |
Type1 |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3KKVA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B99 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4IJ9A
|
2.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PTV |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2C1AA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I5S |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2C1BA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQP |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2F7EE
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2EA |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2F7XE
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4EA |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2F7ZE
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6EA |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2JDSA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L20 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2OH0E
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2PY |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2OJFE
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4PY |
Type1 |
16 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3AG9B
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A02 |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3ZO1A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SIJ |
Type1 |
10 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3ZO4A
|
1.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QWI |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4IE9A
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZX |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
5VHBA
|
1.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9CY |
Type1 |
19 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
6E99A
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0G |
Type1 |
19 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
6E9LA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0P |
Type1 |
18 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
8SF8A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZWG |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3DNDA
|
2.26 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LL2 |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3DNEA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LL1 |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4YXRA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0RW |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4YXSA
|
2.11 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EMU |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1YDRE
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQP |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1YDSE
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQS |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1YDTE
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQB |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1SZMA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI4 |
Type1 |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4Z84A
|
1.554 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVX |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XHAA
|
2.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R68 |
Type1 |
2 - 351 |
0 |
TPO198,SEP339 |
Q85E,V124A,L174M,F188L |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2JDTA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I5S |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2JDVA
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L20 |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UVXA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVH |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UVYA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVI |
Type1 |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UVZA
|
1.94 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVJ |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW0A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVK |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW3A
|
2.19 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVG |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW4A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L15 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW5A
|
2.14 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVN |
Type1 |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW6A
|
2.23 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVO |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW7A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVP |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2UW8A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVQ |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2VNWA
|
2.09 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M01 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2VNYA
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M02 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2VO3A
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M04 |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2VO6A
|
1.97 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M05 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4C36A
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZO9 |
Type1 |
14 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
F55Y,M121L,V124L,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4C38A
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VUP |
Type1 |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
F55Y,M121L,V124L,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1Q8UA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H52,
H52
|
Type1,
Allosteric
|
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3BWJA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ARX,
ARX
|
Type1,
Allosteric
|
11 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4Z83E
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4L7,
4L7
|
Type1,
Allosteric
|
15 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
2VO0A
|
1.94 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M03,
M03
|
Type1,
Allosteric
|
9 - 351 |
0 |
SEP11,TPO198,SEP339 |
V105T,V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8CA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8CB
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8CC
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8CD
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8CE
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
14 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8CF
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8EA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8EB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
13 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8EE
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8EI
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
4 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8EL
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
14 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
3E8EP
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
8 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1XH9A
|
1.64 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R69 |
Type1.5_Front |
14 - 351 |
0 |
TPO198,SEP339 |
Q85E,V124A,L174M,Q182K,F188L |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
1SVHA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I08 |
Type1.5_Front |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
4C35A
|
2.19 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NU3 |
Type1.5_Back |
11 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
F55Y,M121L,V124L,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9DW7G
|
6.0 |
Inactive |
None‑None |
out-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iiio |
ANP |
ATPlike |
13 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9DW4K
|
9.0 |
Inactive |
None‑None |
in-none |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
PRKACA
|
KAPCA_BOVIN
|
9DW7K
|
6.0 |
Inactive |
None‑None |
in-none |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Bos taurus |
|
AGC
|
ROCK2
|
ROCK2_BOVIN
|
2F2UA
|
2.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
M77 |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Bos taurus |
|
AGC
|
ROCK2
|
ROCK2_BOVIN
|
2H9VA
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y27 |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Bos taurus |
|
AGC
|
ROCK2
|
ROCK2_BOVIN
|
2F2UB
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
M77 |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Bos taurus |
|
AGC
|
PKH2
|
PKH2_CANAL
|
4C0TA
|
3.16 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioo |
No_ligand |
No_ligand |
233 - 523 |
0 |
SEP407 |
None |
Serine/threonine-protein kinase PKH2 |
Candida albicans |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OUAA
|
1.67 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OUSA
|
2.21 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5NW8A
|
2.086 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5LCPA
|
1.433 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5LCRA
|
1.565 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6TX |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5LCTA
|
1.615 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6TY |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5LCUA
|
1.579 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQP |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M6VA
|
1.418 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H52 |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M6YA
|
1.367 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7KB |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M71A
|
1.488 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7K7 |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M75A
|
1.538 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9K6 |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1DA
|
1.609 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8FZ |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3DA
|
1.77 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8NE |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5O0EA
|
1.5 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5O5MA
|
1.583 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9LQ |
Type1 |
10 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OK3A
|
1.588 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OL3A
|
1.58 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9LQ |
Type1 |
11 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OT3A
|
2.04 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9LQ |
Type1 |
13 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OTGA
|
1.73 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AO8 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5OUCA
|
1.46 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AO8 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EGWA
|
1.74 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9LQ |
Type1 |
14 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EH3A
|
1.95 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4Z |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6ERTA
|
1.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BVZ |
Type1 |
14 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6ERWA
|
1.89 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6I2AA
|
1.75 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6I2CA
|
1.82 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6I2DA
|
1.91 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9LQ |
Type1 |
9 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6I2HA
|
1.68 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AO8 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Y0BA
|
1.71 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1LQ |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Y2UA
|
1.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LRT |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7AXWA
|
1.69 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1SQ |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7BAQA
|
1.54 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T82 |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7PIDA
|
1.496 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7QI |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7PIEA
|
1.427 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7QF |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7PIFA
|
1.395 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7QL |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7PIGA
|
1.553 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7QR |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7PNSA
|
1.855 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7W8 |
Type1 |
10 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6I2BA
|
1.97 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9LQ,
9LQ
|
Type1,
Allosteric
|
5 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REKA
|
1.38 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D8P,
D8P,
D8P,
D8P
|
Type1,
Allosteric,
Allosteric,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EH2A
|
1.76 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EM6A
|
1.64 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EM7A
|
1.238 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
11 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EMAA
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6ESAA
|
1.307 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
11 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Y8CA
|
1.76 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3NA
|
1.224 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
152 |
Allosteric |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1GA
|
1.14 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8G5 |
Allosteric |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1NA
|
1.405 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8G8 |
Allosteric |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3IA
|
1.14 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BJQ |
Allosteric |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3KA
|
1.33 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GGB |
Allosteric |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3RA
|
1.36 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CDT |
Allosteric |
13 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Z08A
|
1.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NPO |
Allosteric |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE2A
|
1.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JE1 |
Allosteric |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REHA
|
1.33 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JEO |
Allosteric |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REMA
|
1.43 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEL |
Allosteric |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RESA
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEG |
Allosteric |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RETA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEF |
Allosteric |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N37A
|
1.589 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8JT,
8JT
|
Allosteric,
Allosteric
|
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3GA
|
1.16 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8KB,
8KB
|
Allosteric,
Allosteric
|
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3TA
|
1.209 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8K2,
8K2
|
Allosteric,
Allosteric
|
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RDZA
|
1.64 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JE9,
A1JE9
|
Allosteric,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REDA
|
1.31 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JEV,
A1JEV
|
Allosteric,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REEA
|
1.34 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEW,
A1JEW
|
Allosteric,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RELA
|
1.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D8V,
D8V
|
Allosteric,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REPA
|
1.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JFA,
A1JFA,
A1JFA
|
Allosteric,
Allosteric,
Type1
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REOA
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEJ,
A1JEJ,
A1JEJ,
A1JEJ,
A1JEJ
|
Allosteric,
Allosteric,
Type1,
Type1,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7AXVA
|
1.79 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S95,
S95
|
Allosteric,
Type1
|
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RDWA
|
1.44 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JE6,
A1JE6
|
Allosteric,
Type1
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE3A
|
1.57 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JE0,
A1JE0
|
Allosteric,
Type1
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3OA
|
1.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5AO,
5AO,
5AO
|
Allosteric,
Type1,
Allosteric
|
14 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REJA
|
1.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JEM,
A1JEM,
A1JEM
|
Allosteric,
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
4WIHA
|
1.139 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M0UA
|
1.667 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3MA
|
1.229 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5NTJA
|
1.56 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EH0A
|
1.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6ERUA
|
2.15 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6ERVA
|
2.06 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Z44A
|
1.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6F14A
|
1.867 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ISQ |
Type1 |
9 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SNNA
|
1.817 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
BEZ |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5LCQA
|
1.423 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6TV |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M0BA
|
1.506 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQU |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M0CA
|
1.734 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7CB |
Type1 |
14 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1EA
|
1.529 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9NT |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1FA
|
1.12 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8ET |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1HA
|
1.18 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8G2 |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1LA
|
1.489 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
47V |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1MA
|
1.436 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BJK |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1OA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8GB |
Type1 |
8 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N33A
|
1.434 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8JW |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N36A
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F05 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N39A
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8LZ |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3AA
|
1.404 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
46P |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3BA
|
1.64 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BJN |
Type1 |
5 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3CA
|
1.772 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8M2 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3EA
|
1.529 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
46L |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3HA
|
1.36 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NCA |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3JA
|
1.12 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4NB |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3LA
|
1.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E5E |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3PA
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5H1 |
Type1 |
13 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3SA
|
1.14 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
HBD |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N7PA
|
1.501 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E9Q |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N7UA
|
1.371 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PQ |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6EM2A
|
1.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
12 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SOXA
|
1.38 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
LQ2 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SPMA
|
1.37 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3AE |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SPSA
|
1.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LR5 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SPUA
|
1.39 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
GAB |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SPYA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LR8 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SQ1A
|
1.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LRT |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Y05A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADE |
Type1 |
8 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Y2OA
|
2.01 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
O72 |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6Y89A
|
1.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
OGB |
Type1 |
11 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YNAA
|
1.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YNBA
|
1.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQU |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YNCA
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7CT |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YNRA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
O72 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YNTA
|
1.52 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LRT |
Type1 |
6 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YOUA
|
1.73 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
P4Q |
Type1 |
14 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YPPA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ISQ |
Type1 |
13 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YPSA
|
1.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
P72 |
Type1 |
14 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YQIA
|
1.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6TV |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YQJA
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6TX |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YQKA
|
1.67 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7KB |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7AXTA
|
1.86 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S9B |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7BARA
|
1.37 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T82 |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7BB0A
|
1.75 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T7W |
Type1 |
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
7PIHA
|
1.374 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7QW |
Type1 |
1 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RDXA
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JE5 |
Type1 |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RDYA
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JE4 |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE6A
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEX |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REBA
|
1.39 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JET |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RECA
|
1.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JEU |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REFA
|
1.42 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D8J |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RENA
|
1.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEK |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REQA
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEI |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RERA
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEH |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5M0LA
|
1.465 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7CT,
7CT
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5MHIA
|
1.489 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7N9,
7N9
|
Type1,
Allosteric
|
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N1KA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
489,
489
|
Type1,
Allosteric
|
7 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N32A
|
1.833 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8K5,
8K5
|
Type1,
Allosteric
|
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3FA
|
1.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
463,
463
|
Type1,
Allosteric
|
8 - 334 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
5N3QA
|
1.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3AB,
3AB
|
Type1,
Allosteric
|
13 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6SNXA
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UNU,
UNU
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6YOTA
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
P4W,
P4W
|
Type1,
Allosteric
|
1 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
6ZN0A
|
1.59 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NTN,
NTN
|
Type1,
Allosteric
|
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RDVA
|
1.32 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JE7,
A1JE7
|
Type1,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE0A
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JE3,
A1JE3
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE1A
|
1.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JE2,
A1JE2
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE5A
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JEY,
A1JEY
|
Type1,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE8A
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEQ,
A1JEQ
|
Type1,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE9A
|
1.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JER,
A1JER
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REAA
|
1.52 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JES,
A1JES
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REGA
|
1.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JEP,
A1JEP
|
Type1,
Allosteric
|
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RDUA
|
1.42 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1JE8,
A1JE8,
A1JE8
|
Type1,
Allosteric,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE4A
|
1.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEZ,
A1JEZ,
A1JEZ
|
Type1,
Allosteric,
Allosteric
|
11 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9RE7A
|
1.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D6V,
D6V,
D6V,
D6V
|
Type1,
Allosteric,
Allosteric,
Allosteric
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
PRKACA
|
KAPCA_CRIGR
|
9REIA
|
1.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1JEN,
A1JEN
|
Type1,
Type1
|
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Cricetulus griseus |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EKKA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EKKB
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
AF-P31749-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 416 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
AF-P31749-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 416 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6BUUA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 478 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6BUUB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 477 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6NPZA
|
2.12 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 478 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6NPZB
|
2.12 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
141 - 477 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4GV1A
|
1.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0XZ |
Type1 |
144 - 477 |
0 |
TPO308 |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OCBA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XM1 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OCBB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XM1 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OW4A
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMY |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OW4B
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMY |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKLA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMR |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKMA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SM9 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EKLA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0RF |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3CQUA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQU |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3CQWA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQW |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3MV5A
|
2.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3MVHA
|
2.01 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WFE |
Type1 |
145 - 476 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6CCYA
|
2.18 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX4 |
Type1 |
144 - 983 |
0 |
TPO308 |
N199S,S396P,E397S,T433V |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKKA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMH |
Type1.5_Front |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UVYA
|
2.11 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XOO |
Allosteric |
3 - 439 |
0 |
None |
E17K |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW2A
|
2.2 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
XOO |
Allosteric |
4 - 437 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW9A
|
1.9 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XQ2 |
Allosteric |
3 - 428 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW7A
|
1.972 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 439 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3O96A
|
2.7 |
Inactive |
DFGout‑BBAminus |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
IQO |
Allosteric |
2 - 429 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHHA
|
2.7 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
G4Q |
Allosteric |
2 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHJA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4H |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9WA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
L1Z |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EJNA
|
2.19 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
0R4 |
Type1 |
4 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
5KCVA
|
2.7 |
Inactive |
DFGout‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
6S1 |
Allosteric |
6 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7APJA
|
2.05 |
Inactive |
DFGout‑None |
none-none |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
3 - 439 |
0 |
None |
S2N |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHFA
|
2.9 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
G4K |
Allosteric |
3 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHGA
|
2.3 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4T |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHIA
|
2.7 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4N |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9XA
|
2.6 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
L1W |
Allosteric |
3 - 443 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7NH4A
|
2.3 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
UCE |
Allosteric |
4 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7NH5A
|
1.9 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
UC8 |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1O6KA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
146 - 479 |
0 |
TPO309 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1O6LA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
AF-P31751-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 417 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
AF-P31751-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 417 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E87A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G95 |
Type1 |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E87B
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G95 |
Type1 |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2JDOA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I5S |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2JDRA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L20 |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2UW9A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVP |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2X39A
|
1.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X39 |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2XH5A
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X37 |
Type1 |
146 - 479 |
0 |
TPO309 |
R467Q,T468E,H469M,P471E,Q472D,S474D,S476I,S478D,I479W |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3D0EA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G93 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3D0EB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G93 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E88A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E88B
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E8DA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E8DB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
9C1WA
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 440 |
0 |
None |
P115A,G116A |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
8Q61A
|
2.32 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
K06 |
Type3 |
1 - 435 |
0 |
None |
N2D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZKA
|
2.3 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 441 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZOA
|
2.75 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZNA
|
2.5 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRVA
|
2.8 |
Inactive |
DFGout‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
147 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRYA
|
2.8 |
Inactive |
DFGout‑None |
none-none |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnio |
No_ligand |
No_ligand |
146 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT3
|
AKT3_HUMAN
|
AF-Q9Y243-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
140 - 413 |
0 |
None |
None |
RAC-gamma serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT3
|
AKT3_HUMAN
|
AF-Q9Y243-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
140 - 413 |
0 |
None |
None |
RAC-gamma serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
CDC42BPA
|
MRCKA_HUMAN
|
AF-Q5VT25-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
69 - 351 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK alpha |
Homo sapiens |
|
AGC
|
CDC42BPA
|
MRCKA_HUMAN
|
AF-Q5VT25-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
69 - 351 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK alpha |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
4UAKA
|
1.73 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
AF-Q9Y5S2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 350 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
AF-Q9Y5S2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 350 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3QFVA
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NM7 |
Type1 |
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3QFVB
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NM7 |
Type1 |
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
4UALA
|
1.71 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3FV |
Type1 |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
5OTEA
|
1.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AQE |
Type1 |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
5OTFA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AQ5 |
Type1 |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3TKUA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77,
M77
|
Type1,
Allosteric
|
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3TKUB
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77,
M77
|
Type1,
Allosteric
|
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
Homo sapiens |
|
AGC
|
CDC42BPG
|
MRCKG_HUMAN
|
AF-Q6DT37-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 345 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK gamma |
Homo sapiens |
|
AGC
|
CDC42BPG
|
MRCKG_HUMAN
|
AF-Q6DT37-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 345 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK gamma |
Homo sapiens |
|
AGC
|
CIT
|
CTRO_HUMAN
|
AF-O14578-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
89 - 368 |
0 |
None |
None |
Citron Rho-interacting kinase |
Homo sapiens |
|
AGC
|
CIT
|
CTRO_HUMAN
|
AF-O14578-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
89 - 368 |
0 |
None |
None |
Citron Rho-interacting kinase |
Homo sapiens |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
AF-Q09013-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 347 |
0 |
None |
None |
Myotonin-protein kinase |
Homo sapiens |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
AF-Q09013-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 347 |
0 |
None |
None |
Myotonin-protein kinase |
Homo sapiens |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
2VD5A
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI8 |
Type1 |
11 - 416 |
0 |
None |
None |
Myotonin-protein kinase |
Homo sapiens |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
2VD5B
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI8 |
Type1 |
11 - 416 |
0 |
None |
None |
Myotonin-protein kinase |
Homo sapiens |
|
AGC
|
GRK1
|
GRK1_HUMAN
|
AF-Q15835-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
182 - 463 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Homo sapiens |
|
AGC
|
GRK1
|
GRK1_HUMAN
|
AF-Q15835-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
182 - 463 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
AF-P25098-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
AF-P25098-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UVCA
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PV |
Type1 |
30 - 536 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UKLA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SIX |
Type1 |
31 - 671 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5HE1A
|
3.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZS2 |
Type1 |
29 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
6C2YA
|
2.74 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EJS |
Type1 |
30 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
4MK0A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
29X |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7K7LA
|
2.539 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W4D |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7K7ZA
|
2.606 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W4G |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3V5WA
|
2.07 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PR |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
4PNKA
|
2.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
KZQ |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG3A
|
2.896 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFM |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG4A
|
2.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFV |
Type1 |
31 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG5A
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZSO |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UUUA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QRW |
Type1.5_Front |
31 - 538 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UKKA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8DJ |
Type1.5_Front |
30 - 667 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
6U7CA
|
2.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q1Y |
Type1.5_Front |
30 - 669 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3CIKA
|
2.75 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 669 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7PWDA
|
2.6 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8DS |
Type1 |
27 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3KRWA
|
2.9 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
30 - 671 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3KRXA
|
3.1 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
30 - 671 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
Homo sapiens |
|
AGC
|
GRK3
|
ARBK2_HUMAN
|
AF-P35626-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
G protein-coupled receptor kinase 3 |
Homo sapiens |
|
AGC
|
GRK3
|
ARBK2_HUMAN
|
AF-P35626-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
G protein-coupled receptor kinase 3 |
Homo sapiens |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
4YHJA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
25 - 525 |
0 |
None |
C563S,C578S |
G protein-coupled receptor kinase 4 |
Homo sapiens |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
4YHJB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
25 - 527 |
0 |
None |
C563S,C578S |
G protein-coupled receptor kinase 4 |
Homo sapiens |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
AF-P32298-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
179 - 457 |
0 |
None |
None |
G protein-coupled receptor kinase 4 |
Homo sapiens |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
AF-P32298-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
179 - 457 |
0 |
None |
None |
G protein-coupled receptor kinase 4 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKOA
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRKA
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARA |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRLA
|
2.73 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARB |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRPA
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARF |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
4TNDA
|
1.802 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 543 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKRA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKSA
|
3.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
AF-P34947-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
AF-P34947-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKQA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
4TNBA
|
2.113 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
15 - 543 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
8UAPA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W2T |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BREA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3F |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRGA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ6 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRHA
|
3.69 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ7 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRMA
|
2.73 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARC |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRNA
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARD |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BROA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARE |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKPA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9MX2A
|
3.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
6PJXA
|
1.96 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
E104K,R304H,G438E |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
8UAQA
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3F |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRFA
|
2.84 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ5 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRIA
|
2.9 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ8 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRJA
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ9 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
2ACXA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 532 |
0 |
None |
C561S,C562S,C565S |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
2ACXB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 535 |
0 |
None |
C561S,C562S,C565S |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYOA
|
2.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYOB
|
2.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
AF-P43250-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
AF-P43250-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYNA
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYNB
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
Homo sapiens |
|
AGC
|
GRK7
|
GRK7_HUMAN
|
AF-Q8WTQ7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 462 |
0 |
None |
None |
Rhodopsin kinase GRK7 |
Homo sapiens |
|
AGC
|
GRK7
|
GRK7_HUMAN
|
AF-Q8WTQ7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 462 |
0 |
None |
None |
Rhodopsin kinase GRK7 |
Homo sapiens |
|
AGC
|
LATS1
|
LATS1_HUMAN
|
AF-O95835-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
697 - 1018 |
0 |
None |
None |
Serine/threonine-protein kinase LATS1 |
Homo sapiens |
|
AGC
|
LATS1
|
LATS1_HUMAN
|
AF-O95835-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
697 - 1018 |
0 |
None |
None |
Serine/threonine-protein kinase LATS1 |
Homo sapiens |
|
AGC
|
LATS2
|
LATS2_HUMAN
|
AF-Q9NRM7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
660 - 981 |
0 |
None |
None |
Serine/threonine-protein kinase LATS2 |
Homo sapiens |
|
AGC
|
LATS2
|
LATS2_HUMAN
|
AF-Q9NRM7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
660 - 981 |
0 |
None |
None |
Serine/threonine-protein kinase LATS2 |
Homo sapiens |
|
AGC
|
MAST1
|
MAST1_HUMAN
|
AF-Q9Y2H9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
366 - 655 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 1 |
Homo sapiens |
|
AGC
|
MAST1
|
MAST1_HUMAN
|
AF-Q9Y2H9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
366 - 655 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 1 |
Homo sapiens |
|
AGC
|
MAST2
|
MAST2_HUMAN
|
AF-Q6P0Q8-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
504 - 793 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 2 |
Homo sapiens |
|
AGC
|
MAST2
|
MAST2_HUMAN
|
AF-Q6P0Q8-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
504 - 793 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 2 |
Homo sapiens |
|
AGC
|
MAST3
|
MAST3_HUMAN
|
AF-O60307-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
359 - 648 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 3 |
Homo sapiens |
|
AGC
|
MAST3
|
MAST3_HUMAN
|
AF-O60307-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
359 - 648 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 3 |
Homo sapiens |
|
AGC
|
MAST4
|
MAST4_HUMAN
|
AF-O15021-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
562 - 851 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 4 |
Homo sapiens |
|
AGC
|
MAST4
|
MAST4_HUMAN
|
AF-O15021-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
562 - 851 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 4 |
Homo sapiens |
|
AGC
|
MASTL
|
GWL_HUMAN
|
AF-Q96GX5-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 843 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
Homo sapiens |
|
AGC
|
MASTL
|
GWL_HUMAN
|
AF-Q96GX5-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 843 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
Homo sapiens |
|
AGC
|
MASTL
|
GWL_HUMAN
|
8V5HA
|
2.74 |
Inactive |
DFGin‑BLAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
A1AAE |
Type1 |
29 - 847 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
Homo sapiens |
|
AGC
|
MASTL
|
GWL_HUMAN
|
5LOHA
|
3.1 |
Inactive |
DFGin‑BLAplus |
none-none |
out-out |
nonTYR |
APEdihe_aanon |
APEdist_nnno |
STU |
Type1 |
30 - 854 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
Homo sapiens |
|
AGC
|
MASTL
|
GWL_HUMAN
|
5LOHB
|
3.1 |
Inactive |
None‑None |
none-none |
none-out |
nonTYR |
APEdihe_aannn |
APEdist_nnno |
STU |
Type1 |
30 - 854 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1H1WA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2BIYA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
72 - 359 |
0 |
None |
S241A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3HRCA
|
1.91 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
76 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4RRVA
|
1.412 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
76 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5ACKA
|
1.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
73 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPB
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPC
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPD
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4CT2A
|
1.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
75 - 359 |
0 |
SEP241 |
L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5MRDA
|
1.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
76 - 359 |
0 |
SEP241 |
K76S,L113V,I118V,I119N,V124I,T128Q,R131K,T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3HRFA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
P47
|
ATPlike,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4A06A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
A06
|
ATPlike,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4AW0A
|
1.43 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
MJF
|
ATPlike,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4AW1A
|
1.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
21O
|
ATPlike,
Allosteric
|
66 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4RQKA
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
R1S
|
ATPlike,
Allosteric
|
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4RQVA
|
1.502 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
R2S
|
ATPlike,
Allosteric
|
71 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVOA
|
1.09 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
78W
|
ATPlike,
Allosteric
|
73 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4CT1A
|
1.85 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
31S
|
ATPlike,
Allosteric
|
76 - 359 |
0 |
SEP241 |
L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4XX9A
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
RF4,
RF4
|
ATPlike,
Allosteric,
Allosteric
|
71 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4A07A
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
AZ7,
AZ7
|
ATPlike,
Allosteric,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXA
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXB
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
77 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXC
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXD
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
76 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXE
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
1F8 |
Allosteric |
76 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXF
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXG
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXH
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
8DQTA
|
1.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U35,
U35,
U35
|
Allosteric,
Allosteric,
Allosteric
|
70 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
74 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZB
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
73 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
74 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZD
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
73 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3OTUA
|
2.101 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J30,
BI4
|
Allosteric,
Type1.5_Front
|
77 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
AF-O15530-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
74 - 350 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
AF-O15530-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
74 - 350 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1Z5MA
|
2.17 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LI8 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE0A
|
2.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
39Z |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE1A
|
2.14 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
517 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE2A
|
2.13 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
464 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JNZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUUA
|
1.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JOZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUYA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JPZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU9A
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI3 |
Type1 |
72 - 357 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UVRA
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI8 |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUNA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JMZ |
Type1 |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2XCHA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
CKG |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HKMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
61Y |
Type1 |
76 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HNGA
|
3.01 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
62O |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HO7A
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
63L |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HO8A
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
63E |
Type1 |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1OKYA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STU |
Type1 |
72 - 360 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1OKZA
|
2.51 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
UCN |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU3A
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LY4 |
Type1 |
73 - 360 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU7A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI2 |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU8A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI1 |
Type1 |
72 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAYA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MP6 |
Type1 |
76 - 362 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAYB
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MP6 |
Type1 |
76 - 362 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RWPA
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ABQ |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RWQA
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3RW |
Type1 |
72 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3SC1A
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3S1 |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3H9OA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
9BD |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2R7BA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
253 |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3IONA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
8H1 |
Type1 |
75 - 359 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3IOPA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8I1 |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCQA
|
2.501 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q0 |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCSA
|
2.487 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q1 |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RCJA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3RC |
Type1 |
77 - 358 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVLA
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
537 |
Type1 |
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVMA
|
1.26 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADE |
Type1 |
76 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVNA
|
1.379 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3PWYA
|
3.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
SYP |
Type1 |
71 - 359 |
0 |
None |
E166C,C260S |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2XCKA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MH4 |
Type1 |
76 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCXA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q2 |
Type1.5_Back |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCYA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
3Q3 |
Type1.5_Front |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD0A
|
1.99 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
3Q4 |
Type1.5_Front |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD3A
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q5 |
Type1.5_Front |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD4A
|
2.3 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
3Q6 |
Type1.5_Front |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAXA
|
1.75 |
Inactive |
DFGout‑BBAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MP7 |
Type2 |
76 - 360 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4A
|
1.8 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
76 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4B
|
1.8 |
Inactive |
DFGout‑None |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
51 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTDA
|
2.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
605 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
Homo sapiens |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTGA
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2V9 |
Type1 |
605 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
Homo sapiens |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
AF-Q16512-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
607 - 882 |
0 |
None |
None |
Serine/threonine-protein kinase N1 |
Homo sapiens |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
AF-Q16512-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
607 - 882 |
0 |
None |
None |
Serine/threonine-protein kinase N1 |
Homo sapiens |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTHA
|
1.8 |
Inactive |
DFGin‑BLAplus |
in-in |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
DRN |
Type1 |
606 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
Homo sapiens |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTIA
|
1.93 |
Inactive |
DFGin‑BLAplus |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MI1 |
Type1 |
606 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
Homo sapiens |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
4CRSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
AGS |
ATPlike |
646 - 984 |
0 |
SEP755,TPO816,TPO958 |
None |
Serine/threonine-protein kinase N2 |
Homo sapiens |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
AF-Q16513-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
649 - 924 |
0 |
None |
None |
Serine/threonine-protein kinase N2 |
Homo sapiens |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
AF-Q16513-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
649 - 924 |
0 |
None |
None |
Serine/threonine-protein kinase N2 |
Homo sapiens |
|
AGC
|
PKN3
|
PKN3_HUMAN
|
AF-Q6P5Z2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
551 - 826 |
0 |
None |
None |
Serine/threonine-protein kinase N3 |
Homo sapiens |
|
AGC
|
PKN3
|
PKN3_HUMAN
|
AF-Q6P5Z2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
551 - 826 |
0 |
None |
None |
Serine/threonine-protein kinase N3 |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE6A
|
2.1 |
Inactive |
DFGin‑ABAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE6B
|
2.1 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE9A
|
2.3 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE9B
|
2.3 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
7Y1GB
|
2.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I5G |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DC6A
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3I |
Type1 |
16 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DC6B
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3I |
Type1 |
16 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AMBA
|
2.25 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
4 - 351 |
0 |
SEP11,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8X5LA
|
2.75 |
Inactive |
DFGin‑ABAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
RKD |
Type1 |
17 - 351 |
0 |
SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8X5LB
|
2.75 |
Inactive |
DFGin‑ABAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
RKD |
Type1 |
17 - 334 |
0 |
SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB8A
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB5A
|
1.641 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7E
|
3.55 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7G
|
3.55 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB7A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB7B
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYRA
|
3.661 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYRC
|
3.661 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDCA
|
4.18 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDDA
|
6.3 |
Inactive |
DFGin‑BLAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDEA
|
5.9 |
Inactive |
DFGin‑BLAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB6A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
SEP11,SEP140,TPO198 |
L206R |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB6B
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
9 - 351 |
0 |
SEP11,TPO198,SEP339 |
L206R |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZJA
|
1.85 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6J9 |
Allosteric |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZJB
|
1.85 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6J9 |
Allosteric |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5J5XA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6J9 |
Allosteric |
10 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
AF-P17612-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
AF-P17612-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSA
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSC
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSE
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSG
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7A
|
3.55 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7C
|
3.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AGMA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZFA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJB
|
2.49 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3NX8A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJFA
|
7.5 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJFB
|
7.5 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJGA
|
6.2 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJGB
|
6.2 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DCDA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3J |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AGLA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A03 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AGLB
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A03 |
Type1 |
15 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9LA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9L |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9LB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9L |
Type1 |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OOGA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YTP |
Type1 |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OVVA
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1SB |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OWPA
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2SB |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OXTA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SB |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3P0MA
|
2.03 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SB |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3POOA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S69 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3VQHA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQB |
Type1 |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ1A
|
1.768 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVX |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ2A
|
2.019 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVV |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ9A
|
1.87 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S3N |
Type1 |
11 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJAA
|
1.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4L7 |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJBA
|
1.949 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8BQ |
Type1 |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5BX6A
|
1.89 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
495 |
Type1 |
6 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5BX7A
|
1.89 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4W1 |
Type1 |
6 - 350 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5UZKA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
504 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6QJ7A
|
1.69 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J4B |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
7Y1GA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I5G |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6C0UA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EE4 |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJA
|
2.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJE
|
2.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9MA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9M |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9MB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9M |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9NA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9N |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE2A
|
2.34 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTI |
Type1 |
4 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE2B
|
2.34 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTI |
Type1 |
4 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE5A
|
2.51 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTT |
Type1 |
3 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE5B
|
2.51 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTT |
Type1 |
4 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FECA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XU0 |
Type1 |
3 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FECB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XU0 |
Type1 |
3 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
2GU8A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
796 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5N23A
|
2.088 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
35R |
Type1 |
9 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AMAA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SKE |
Type1 |
2 - 351 |
0 |
SEP11,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6FRXA
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E3Z |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Homo sapiens |
|
AGC
|
PRKACB
|
KAPCB_HUMAN
|
AF-P22694-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit beta |
Homo sapiens |
|
AGC
|
PRKACB
|
KAPCB_HUMAN
|
AF-P22694-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit beta |
Homo sapiens |
|
AGC
|
PRKACG
|
KAPCG_HUMAN
|
AF-P22612-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit gamma |
Homo sapiens |
|
AGC
|
PRKACG
|
KAPCG_HUMAN
|
AF-P22612-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit gamma |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
AF-P17252-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
331 - 605 |
0 |
None |
None |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
AF-P17252-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
331 - 605 |
0 |
None |
None |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
4RA4A
|
2.63 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3KZ |
Type1 |
332 - 666 |
0 |
TPO497,TPO638,SEP657 |
C619S |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
3IW4A
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LW4 |
Type1 |
331 - 669 |
0 |
TPO638,SEP657 |
T497E |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
3IW4B
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LW4 |
Type1 |
332 - 666 |
0 |
TPO638,SEP657 |
T497E |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
3IW4C
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LW4 |
Type1 |
330 - 670 |
0 |
TPO638,SEP657 |
T497E |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
8U37A
|
2.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V5U |
Type1 |
332 - 666 |
0 |
TPO497,TPO638 |
D463N,V568I,S657E |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
8UAKA
|
2.82 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W39 |
Type1 |
332 - 666 |
0 |
TPO497,TPO638 |
D463N,V568I,S657E |
Protein kinase C alpha type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE2A
|
2.95 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE3A
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE4A
|
2.68 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE4B
|
2.68 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE1A
|
3.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
19 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE1B
|
3.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
19 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE2B
|
2.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
AF-P05771-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
334 - 608 |
0 |
None |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
AF-P05771-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
334 - 608 |
0 |
None |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
2I0EA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
PDS |
Type1 |
339 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
2I0EB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PDS |
Type1 |
339 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
9S9TA
|
3.425 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LY4 |
Type1 |
340 - 667 |
0 |
TPO500,TPO642,SEP661 |
D427N |
Protein kinase C beta type |
Homo sapiens |
|
AGC
|
PRKCD
|
KPCD_HUMAN
|
AF-Q05655-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
341 - 611 |
0 |
None |
None |
Protein kinase C delta type |
Homo sapiens |
|
AGC
|
PRKCD
|
KPCD_HUMAN
|
AF-Q05655-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
341 - 611 |
0 |
None |
None |
Protein kinase C delta type |
Homo sapiens |
|
AGC
|
PRKCE
|
KPCE_HUMAN
|
AF-Q02156-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
400 - 676 |
0 |
None |
None |
Protein kinase C epsilon type |
Homo sapiens |
|
AGC
|
PRKCE
|
KPCE_HUMAN
|
AF-Q02156-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
400 - 676 |
0 |
None |
None |
Protein kinase C epsilon type |
Homo sapiens |
|
AGC
|
PRKCG
|
KPCG_HUMAN
|
AF-P05129-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
343 - 622 |
0 |
None |
None |
Protein kinase C gamma type |
Homo sapiens |
|
AGC
|
PRKCG
|
KPCG_HUMAN
|
AF-P05129-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
343 - 622 |
0 |
None |
None |
Protein kinase C gamma type |
Homo sapiens |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
AF-P24723-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
347 - 622 |
0 |
None |
None |
Protein kinase C eta type |
Homo sapiens |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
AF-P24723-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
347 - 622 |
0 |
None |
None |
Protein kinase C eta type |
Homo sapiens |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
8FP1A
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XXF |
Type1 |
349 - 676 |
0 |
TPO513,TPO656 |
S675E |
Protein kinase C eta type |
Homo sapiens |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
8FP3A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y3I |
Type1 |
349 - 679 |
0 |
TPO513,TPO656 |
S675E |
Protein kinase C eta type |
Homo sapiens |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
3TXOA
|
2.05 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
07U |
Type1 |
353 - 679 |
0 |
TPO656 |
S675E |
Protein kinase C eta type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3YI
|
3.68 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
248 - 585 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3XA
|
2.591 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3XB
|
2.591 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZA
|
3.261 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8WA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8WB
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LIHA
|
3.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
248 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LIHB
|
3.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LI9A
|
1.79 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ACP |
ATPlike |
248 - 589 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LI1A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
248 - 589 |
0 |
TPO412,SEP484,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
9EJMB
|
3.33 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
AF-P41743-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
246 - 530 |
0 |
None |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
AF-P41743-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
246 - 530 |
0 |
None |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8XA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8XB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
9EJKB
|
3.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
9EJLB
|
3.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZC
|
3.261 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZE
|
3.261 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
255 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZG
|
3.261 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3ZH8A
|
2.739 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C58 |
Type1 |
248 - 590 |
0 |
TPO412,TPO564 |
C595S |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3ZH8B
|
2.739 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C58 |
Type1 |
248 - 589 |
0 |
TPO412,TPO564 |
C595S |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3ZH8C
|
2.739 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C58 |
Type1 |
248 - 588 |
0 |
TPO412,TPO564 |
C595S |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
1ZRZA
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI1 |
Type1 |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
AF-Q04759-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
372 - 642 |
0 |
None |
None |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
AF-Q04759-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
372 - 642 |
0 |
None |
None |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4Q9ZA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZW |
Type1 |
375 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4Q9ZB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZW |
Type1 |
374 - 704 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4RA5A
|
2.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3L0 |
Type1 |
374 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4RA5B
|
2.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3L0 |
Type1 |
375 - 701 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
2JEDA
|
2.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LG8 |
Type1 |
375 - 700 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
2JEDB
|
2.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LG8 |
Type1 |
375 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
5F9EA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5VS |
Type1 |
374 - 706 |
0 |
SEP676,SEP695 |
None |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
5F9EB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5VS |
Type1 |
375 - 700 |
0 |
SEP676,SEP695 |
None |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
1XJDA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
377 - 696 |
0 |
TPO538,SEP695 |
None |
Protein kinase C theta type |
Homo sapiens |
|
AGC
|
PRKCZ
|
KPCZ_HUMAN
|
AF-Q05513-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
244 - 526 |
0 |
None |
None |
Protein kinase C zeta type |
Homo sapiens |
|
AGC
|
PRKCZ
|
KPCZ_HUMAN
|
AF-Q05513-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
244 - 526 |
0 |
None |
None |
Protein kinase C zeta type |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4UA
|
1.99 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX6 |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4UB
|
1.99 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX6 |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4WA
|
2.23 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZJ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4WB
|
2.23 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZJ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4TA
|
2.08 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PCG,
ATP
|
Allosteric,
ATPlike
|
204 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4TB
|
2.08 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PCG,
ATP
|
Allosteric,
ATPlike
|
204 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2A
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
336 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2B
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
346 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2C
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2D
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
344 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7LV3A
|
2.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
57 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7LV3B
|
2.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
58 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4VA
|
2.28 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
EXZ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4VB
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EXZ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
AF-Q13976-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
352 - 627 |
0 |
None |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
AF-Q13976-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
352 - 627 |
0 |
None |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BDLA
|
1.96 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iiio |
No_ligand |
No_ligand |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BDLB
|
1.96 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_iiii |
No_ligand |
No_ligand |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6C0TA
|
1.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EE4 |
Type1.5_Front |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PRKG2
|
KGP2_HUMAN
|
AF-Q13237-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
445 - 719 |
0 |
None |
None |
cGMP-dependent protein kinase 2 |
Homo sapiens |
|
AGC
|
PRKG2
|
KGP2_HUMAN
|
AF-Q13237-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
445 - 719 |
0 |
None |
None |
cGMP-dependent protein kinase 2 |
Homo sapiens |
|
AGC
|
PRKX
|
PRKX_HUMAN
|
AF-P51817-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 311 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit PRKX |
Homo sapiens |
|
AGC
|
PRKX
|
PRKX_HUMAN
|
AF-P51817-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 311 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit PRKX |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMA
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZA
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZB
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZC
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZD
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMB
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3ND |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMC
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
3ND |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMD
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3ND |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFA
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4V |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFB
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
B4V |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFC
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4V |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFD
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4V |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGA
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4Y |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGB
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
B4Y |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGC
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4Y |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGD
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4Y |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHA
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5G |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHB
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHC
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHD
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
6E9WA
|
2.96 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0P |
Type1 |
9 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
6E9WB
|
2.96 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
J0P |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2V55A
|
3.705 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2V55C
|
3.705 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
AF-Q13464-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 346 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
AF-Q13464-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 346 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26D
|
2.744 |
Inactive |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
6 - 399 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
8ZH5A
|
3.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26A
|
2.744 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86K |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26B
|
2.744 |
None |
DFGin‑BLAminus |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
86K |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7A
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiio |
07Q |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7B
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
07Q |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7C
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
07Q |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7D
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
07Q |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SA
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0HD |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SB
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
0HD |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SC
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0HD |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SD
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
0HD |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PB
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PC
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PD
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 403 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7JOUA
|
3.318 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ESMA
|
3.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ESMB
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
M77 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETKA
|
2.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HFS |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETKB
|
2.96 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
HFS |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETRA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y27 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETRB
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
Y27 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3D9VA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H52 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3D9VB
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
H52 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVCA
|
3.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4KH |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVCB
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
4KH |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVEA
|
3.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4KK |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVEB
|
3.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
4KK |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5BMLA
|
2.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4TW |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5BMLB
|
2.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
4TW |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKSA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6U1 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKTA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6U2 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5UZJA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8UV |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5UZJB
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
8UV |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
07R |
Type1.5_Back |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5HVUA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
65R |
Type1.5_Front |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5HVUB
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
65R |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKSB
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
6U1 |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKTB
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
6U2 |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNEA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4J |
Type1.5_Front |
14 - 400 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNEB
|
2.6 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B4J |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNEC
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4J |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNED
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4J |
Type1.5_Front |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26C
|
2.744 |
Inactive |
DFGin‑BLBminus |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86K |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJC
|
2.9 |
Inactive |
DFGin‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oiio |
07R |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJB
|
2.9 |
Inactive |
DFGinter‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJD
|
2.9 |
Inactive |
DFGinter‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25A
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
86G |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25B
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
86G |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25C
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86G |
Type1 |
13 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25D
|
2.337 |
Inactive |
None‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
9 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MC
|
2.65 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MD
|
2.65 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QA
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QB
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
No_ligand |
No_ligand |
28 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QC
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QD
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RA
|
3.33 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RC
|
3.33 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PA
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O1V |
Type1 |
27 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PB
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnio |
O1V |
Type1 |
27 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PC
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O1V |
Type1 |
28 - 416 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PD
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
O1V |
Type1 |
26 - 416 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8YB
|
3.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
YEA |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8ZA
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEI |
Type1 |
31 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8ZB
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
YEI |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X92A
|
2.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEW |
Type1 |
29 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X92B
|
2.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_noio |
YEW |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTA
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTB
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTC
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTD
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
3SG |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9HFPA
|
2.92 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IUI |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4L6QA
|
2.79 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1WU |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4L6QB
|
2.79 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1WU |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
AF-O75116-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
84 - 362 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
AF-O75116-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
84 - 362 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RB
|
3.33 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
O1S |
Type1 |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MB
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
O1S |
Type1 |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8XA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDW |
Type1 |
32 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8XB
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
YDW |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8YA
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
YEA |
Type1 |
31 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVA
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVB
|
2.586 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVC
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_onno |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVD
|
2.586 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVE
|
2.586 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_innn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVF
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVG
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_innn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVH
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTA
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTB
|
2.214 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTC
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTD
|
2.214 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTE
|
2.214 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTF
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTG
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_innn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTH
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NA
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_niio |
5YS |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NB
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NC
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6ND
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NE
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NF
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NG
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NH
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
5YK |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OB
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OD
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_inii |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OE
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OF
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PA
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_onoo |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PB
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PC
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PD
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QA
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QB
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QC
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QD
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8A
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
A1H6L |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8B
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H6L |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8C
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H6L |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8D
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
A1H6L |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6ED6A
|
2.86 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0P |
Type1 |
27 - 415 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OC
|
2.75 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YK |
Type1.5_Front |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OG
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1.5_Front |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OH
|
2.75 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YK |
Type1.5_Front |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6ED6B
|
2.86 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
J0P |
Type1.5_Front |
28 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RD
|
3.33 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_onno |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUA
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUC
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSA
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSB
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSC
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSD
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
Z8O |
Type1.5_Front |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUB
|
3.02 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUD
|
3.02 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
AF-Q15418-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 329 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
Homo sapiens |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
AF-Q15418-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 329 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
Homo sapiens |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
8XOVA
|
2.55 |
Inactive |
DFGin‑BLAplus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
ANP |
ATPlike |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
Homo sapiens |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7QA
|
2.0 |
Inactive |
DFGin‑BLBplus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ACP |
ATPlike |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
Homo sapiens |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7RA
|
2.0 |
Inactive |
DFGin‑BLBplus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
STU |
Type1 |
53 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
Homo sapiens |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7SA
|
2.1 |
Inactive |
DFGin‑BLBplus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
P01 |
Type1 |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
Homo sapiens |
|
AGC
|
RPS6KA2-1
|
KS6A2_HUMAN
|
AF-Q15349-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-2 |
Homo sapiens |
|
AGC
|
RPS6KA2-1
|
KS6A2_HUMAN
|
AF-Q15349-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-2 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NW5A
|
1.94 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2NR |
Type1 |
51 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NW6A
|
1.74 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2NS |
Type1 |
51 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
AF-P51812-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
60 - 335 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
AF-P51812-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
60 - 335 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOA
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
45 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOE
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOI
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_onnn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOK
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOC
|
2.75 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
46 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOG
|
2.75 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanni |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8EQ5A
|
1.8 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
QCT |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8R58A
|
2.31 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
QCT |
Type1 |
49 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYA
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
58 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYB
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
59 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYC
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
61 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYD
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYE
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
64 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYF
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 345 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYG
|
3.2 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYH
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYI
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYJ
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
65 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NUSA
|
2.39 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2NK |
Type1 |
53 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9LA
|
2.15 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
583 |
Type1 |
49 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KA
|
2.55 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KB
|
2.55 |
Inactive |
DFGout‑None |
in-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA4-1
|
KS6A4_HUMAN
|
AF-O75676-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 309 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-4 |
Homo sapiens |
|
AGC
|
RPS6KA4-1
|
KS6A4_HUMAN
|
AF-O75676-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 309 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-4 |
Homo sapiens |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
AF-O75582-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
Homo sapiens |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
AF-O75582-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
Homo sapiens |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
1VZOA
|
1.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
24 - 345 |
0 |
None |
S212D |
Ribosomal protein S6 kinase alpha-5 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
AF-Q9UK32-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
65 - 338 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
AF-Q9UK32-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
65 - 338 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G77A
|
2.499 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
Allosteric,
ATPlike
|
51 - 349 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G77B
|
2.499 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
Allosteric,
ATPlike
|
51 - 349 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G76B
|
3.0 |
Inactive |
DFGinter‑None |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
51 - 349 |
0 |
SEP232 |
None |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G78A
|
2.5 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ANP |
ATPlike |
51 - 349 |
0 |
None |
S232E |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G78B
|
2.5 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ANP |
ATPlike |
51 - 349 |
0 |
None |
S232E |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G76A
|
3.0 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
ATPlike,
Allosteric
|
51 - 349 |
0 |
SEP232 |
None |
Ribosomal protein S6 kinase alpha-6 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLPA
|
2.79 |
Inactive |
DFGin‑ABAminus |
none-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
72B |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L3JA
|
2.1 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 375 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L3LA
|
2.1 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 375 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N91A
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1RJ |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N91B
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1RJ |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N93A
|
2.74 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
1SK |
Type1 |
87 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N93B
|
2.74 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1SK |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A62A
|
2.35 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
STU |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WE4A
|
1.995 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF5A
|
2.099 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FZ8 |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF6A
|
2.031 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FZ9 |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L45A
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412E |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L42A
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
5FI |
Type1 |
84 - 417 |
0 |
None |
S403E,A404E,N405Q,Q406E,V407M,L409R,G410D,T412E,V414I,P416D,S417W |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L46A
|
3.01 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
80 - 417 |
0 |
TPO412 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
AF-P23443-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
83 - 360 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
AF-P23443-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
83 - 360 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF8A
|
1.975 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
F76 |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF9A
|
2.035 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FS7 |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L43A
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412A |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L44A
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412A |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLOA
|
2.527 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3T3 |
Type1 |
85 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A60A
|
2.8 |
Inactive |
DFGin‑None |
in-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
STU |
Type1 |
85 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A61A
|
3.43 |
Inactive |
DFGin‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
STU |
Type1 |
87 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF7A
|
1.85 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
FS9 |
Type1 |
83 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLOB
|
2.527 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
STU |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A60B
|
2.8 |
Inactive |
None‑None |
none-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
STU |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
Homo sapiens |
|
AGC
|
RPS6KB2
|
KS6B2_HUMAN
|
AF-Q9UBS0-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
59 - 336 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-2 |
Homo sapiens |
|
AGC
|
RPS6KB2
|
KS6B2_HUMAN
|
AF-Q9UBS0-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
59 - 336 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-2 |
Homo sapiens |
|
AGC
|
RSKR
|
KS6R_HUMAN
|
AF-Q96LW2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
99 - 367 |
0 |
None |
None |
Ribosomal protein S6 kinase-related protein |
Homo sapiens |
|
AGC
|
RSKR
|
KS6R_HUMAN
|
AF-Q96LW2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
99 - 367 |
0 |
None |
None |
Ribosomal protein S6 kinase-related protein |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
AF-O00141-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
90 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
AF-O00141-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
90 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
2R5TA
|
1.9 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
ANP |
ATPlike |
82 - 378 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
3HDMA
|
2.6 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
MMG |
Type1 |
81 - 378 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
3HDNA
|
3.1 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
GMG |
Type1 |
82 - 374 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
7PUEA
|
2.506 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
86H |
Type1 |
82 - 376 |
0 |
None |
R192A,S422D |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
AGC
|
SGK2
|
SGK2_HUMAN
|
AF-Q9HBY8-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 300 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
|
AGC
|
SGK2
|
SGK2_HUMAN
|
AF-Q9HBY8-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 300 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk2 |
Homo sapiens |
|
AGC
|
SGK3
|
SGK3_HUMAN
|
AF-Q96BR1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
154 - 427 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
|
AGC
|
SGK3
|
SGK3_HUMAN
|
AF-Q96BR1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
154 - 427 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk3 |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
AF-Q8WU08-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 289 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
AF-Q8WU08-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 289 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4A
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4B
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4C
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4D
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4E
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 372 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4F
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
Homo sapiens |
|
AGC
|
STK32B
|
ST32B_HUMAN
|
AF-Q9NY57-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 291 |
0 |
None |
None |
Serine/threonine-protein kinase 32B |
Homo sapiens |
|
AGC
|
STK32B
|
ST32B_HUMAN
|
AF-Q9NY57-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 291 |
0 |
None |
None |
Serine/threonine-protein kinase 32B |
Homo sapiens |
|
AGC
|
STK32C
|
ST32C_HUMAN
|
AF-Q86UX6-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
No_ligand |
No_ligand |
85 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase 32C |
Homo sapiens |
|
AGC
|
STK32C
|
ST32C_HUMAN
|
AF-Q86UX6-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
85 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase 32C |
Homo sapiens |
|
AGC
|
STK38
|
STK38_HUMAN
|
AF-Q15208-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
81 - 390 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
Homo sapiens |
|
AGC
|
STK38
|
STK38_HUMAN
|
AF-Q15208-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
81 - 390 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
Homo sapiens |
|
AGC
|
STK38
|
STK38_HUMAN
|
6BXIA
|
2.2 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
82 - 414 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
Homo sapiens |
|
AGC
|
STK38
|
STK38_HUMAN
|
6BXIB
|
2.2 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
83 - 414 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
Homo sapiens |
|
AGC
|
STK38L
|
ST38L_HUMAN
|
AF-Q9Y2H1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
82 - 391 |
0 |
None |
None |
Serine/threonine-protein kinase 38-like |
Homo sapiens |
|
AGC
|
STK38L
|
ST38L_HUMAN
|
AF-Q9Y2H1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
82 - 391 |
0 |
None |
None |
Serine/threonine-protein kinase 38-like |
Homo sapiens |
|
AGC
|
GRK3
|
ARBK2_MOUSE
|
9IJJ4Z
|
7.7 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
No_ligand |
No_ligand |
31 - 666 |
0 |
None |
None |
G protein-coupled receptor kinase 3 |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6MM6C
|
2.39 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
19 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6MM6E
|
2.39 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
19 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6MM7A
|
1.85 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6MM7D
|
1.85 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6MM8C
|
1.85 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
8UKND
|
2.75 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
8UKOE
|
2.89 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
8UKPE
|
2.85 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
17 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4NTTB
|
3.5 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
11 - 351 |
0 |
TPO198,SEP339 |
K8C |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
8UKNC
|
2.75 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
8UKNF
|
2.75 |
Inactive |
DFGin‑ABAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
8UKNH
|
2.75 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3TNPC
|
2.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3TNPF
|
2.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4WBBB
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4X6QC
|
2.52 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4NTSA
|
2.9 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 351 |
0 |
TPO198,SEP339 |
K8C |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4NTSB
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 351 |
0 |
TPO198,SEP339 |
K8C |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
5X3FB
|
3.38 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 317 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4O21A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
7E11A
|
3.43 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6MM5E
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3PVBA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
7 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1ATPE
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1BKXA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
13 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1L3RE
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
2 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
2QCSA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3FJQE
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3IDBA
|
1.62 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
9 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3IDCA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
9 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DG0E
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
11 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DH1A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DH3A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DH5A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DH7A
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DH8A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DINA
|
3.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
10 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4HPTE
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4HPUE
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
5JR7A
|
3.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
5JR7C
|
3.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
7UJXE
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
7V0GE
|
1.63 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
17 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DFXE
|
1.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
K8C |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4X6RA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
K8C |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3X2UA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3X2VA
|
1.77 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
18 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3X2WA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IACA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ACP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IADA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IAFA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IAIA
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IAKA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IAYA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IAZA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IB0A
|
1.87 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IB1A
|
1.63 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4IB3A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4XW4A
|
1.82 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4XW5A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4XW6A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
6E21A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
7E0ZA
|
2.162 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
7E12A
|
2.796 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
19 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1JBPE
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
10 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DG3E
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198 |
R337A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3O7LB
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
18 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3FHIA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
C200A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3QAME
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
TPO198,SEP339 |
E209A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3QALE
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
TPO198,SEP339 |
R281A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1RDQE
|
1.26 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP,
ATP
|
ATPlike,
ATPlike
|
2 - 351 |
0 |
TPO198,SEP339 |
Y205A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4O22A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1J3HA
|
2.9 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1J3HB
|
2.9 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1JLUE
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
2CPKE
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
2QVSE
|
2.5 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3O7LD
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DG2E
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
9O7VA
|
3.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3J4QD
|
35.0 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3J4QE
|
35.0 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3J4RD
|
35.0 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3J4RE
|
35.0 |
None |
DFGin‑BLAminus |
out-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DFZE
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
K8C |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1APME
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
S140A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
2QURA
|
2.5 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 351 |
0 |
TPO198,SEP339 |
K286P,F328A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1BX6A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
13 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1FMOE
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1RE8A
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BD2 |
Type1 |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1REJA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B1L |
Type1 |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
3OW3A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMY |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
2ERZE
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HFS |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1REKA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B8L,
PTL
|
Type1,
Allosteric
|
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4NTTA
|
3.5 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
11 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1SYKA
|
2.8 |
Inactive |
DFGin‑None |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
TPO198,SEP339 |
E231Q |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
1SYKB
|
2.8 |
Inactive |
DFGin‑None |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
TPO198,SEP339 |
E231Q |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DFYA
|
2.997 |
Inactive |
None‑None |
in-none |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
No_ligand |
No_ligand |
15 - 351 |
0 |
SEP339 |
R195A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKACA
|
KAPCA_MOUSE
|
4DFYE
|
2.997 |
Inactive |
None‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
No_ligand |
No_ligand |
15 - 351 |
0 |
SEP339 |
R195A |
cAMP-dependent protein kinase catalytic subunit alpha |
Mus musculus |
|
AGC
|
PRKCI
|
KPCI_MOUSE
|
4DC2A
|
2.4 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADE |
Type1 |
248 - 586 |
0 |
TPO563 |
None |
Protein kinase C iota type |
Mus musculus |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
3G51A
|
1.8 |
Inactive |
DFGin‑None |
none-none |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ANP |
ATPlike |
47 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
3UBDA
|
1.53 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
SL0 |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
4EL9A
|
1.55 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
AFE |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
4GUEA
|
1.8 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
QCT |
Type1 |
48 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
AGC
|
PKG
|
KGP_PLAF7
|
8EM8A
|
2.54 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WLK |
Type1 |
28 - 817 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium falciparum |
|
AGC
|
PKG
|
KGP_PLAF7
|
5DYKA
|
2.45 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 853 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium falciparum |
|
AGC
|
PKG
|
KGP_PLAVS
|
4RZ7A
|
2.351 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1E8 |
Type1 |
1 - 815 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium vivax |
|
AGC
|
PKG
|
KGP_PLAVS
|
5FETA
|
3.07 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1TR |
Type1 |
2 - 816 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium vivax |
|
AGC
|
PKG
|
KGP_PLAVS
|
5DZCA
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
1 - 843 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium vivax |
|
AGC
|
PKG
|
KGP_PLAVS
|
5DYLA
|
2.4 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 816 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium vivax |
|
AGC
|
PKG
|
KGP_PLAVS
|
5F0AA
|
2.6 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1FB |
Type1 |
1 - 846 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium vivax |
|
AGC
|
PKG
|
KGP_PLAVS
|
5EZRA
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4ZS |
Type1.5_Back |
2 - 815 |
0 |
None |
None |
cGMP-dependent protein kinase |
Plasmodium vivax |
|
AGC
|
CDC42BPA
|
MRCKA_RAT
|
4AW2A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
22E |
Allosteric |
2 - 417 |
0 |
None |
D254G |
Serine/threonine-protein kinase MRCK alpha |
Rattus norvegicus |
|
AGC
|
PRKACA
|
KAPCA_RAT
|
3TNQB
|
3.097 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
18 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Rattus norvegicus |
|
AGC
|
PRKCB
|
KPCB_RAT
|
3PFQA
|
4.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
101 - 668 |
0 |
TPO500,TPO642,SEP661 |
C71S,C217S,R622S |
Protein kinase C beta type |
Rattus norvegicus |
|
AGC
|
CBK1
|
CBK1_YEAST
|
4LQSA
|
3.3 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
ANP |
ATPlike |
294 - 749 |
0 |
None |
D475A |
Serine/threonine-protein kinase CBK1 |
Saccharomyces cerevisiae |
|
AGC
|
CBK1
|
CBK1_YEAST
|
5NCLA
|
3.15 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
ANP |
ATPlike |
266 - 756 |
0 |
None |
D475A |
Serine/threonine-protein kinase CBK1 |
Saccharomyces cerevisiae |
|
AGC
|
CBK1
|
CBK1_YEAST
|
4LQPA
|
4.5 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
ANP |
ATPlike |
282 - 749 |
0 |
None |
D475A,T743E |
Serine/threonine-protein kinase CBK1 |
Saccharomyces cerevisiae |
|
AGC
|
CBK1
|
CBK1_YEAST
|
4LQQA
|
3.6 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
ANP |
ATPlike |
282 - 749 |
0 |
None |
D475A,T743E |
Serine/threonine-protein kinase CBK1 |
Saccharomyces cerevisiae |
|
AGC
|
CBK1
|
CBK1_YEAST
|
4LQQD
|
3.6 |
Inactive |
None‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
294 - 749 |
0 |
None |
D475A,T743E |
Serine/threonine-protein kinase CBK1 |
Saccharomyces cerevisiae |
|
AGC
|
TPK1
|
KAPA_YEAST
|
1FOTA
|
2.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
82 - 397 |
0 |
TPO241 |
None |
cAMP-dependent protein kinase type 1 |
Saccharomyces cerevisiae |
|
AGC
|
PRKACA
|
KAPCA_PIG
|
1CDKA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
9 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Sus scrofa |
|
AGC
|
PRKACA
|
KAPCA_PIG
|
1CDKB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
9 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Sus scrofa |
|
AGC
|
PRKACA
|
KAPCA_PIG
|
1CTPE
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 351 |
0 |
TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Sus scrofa |
|
AGC
|
PRKACA
|
KAPCA_PIG
|
1CMKE
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
Sus scrofa |
|
AGC
|
TB0348O8470
|
Q582V7_TRYB2
|
9Z8KA
|
2.05 |
Inactive |
DFGin‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
54 - 348 |
0 |
SEP71 |
None |
Serine/threonine-protein kinase, putative |
Trypanosoma brucei brucei |
|
AGC
|
TB0348O8470
|
Q582V7_TRYB2
|
9Z8KB
|
2.05 |
Inactive |
DFGinter‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
54 - 347 |
0 |
None |
None |
Serine/threonine-protein kinase, putative |
Trypanosoma brucei brucei |