| Organism |
UniprotID |
PDB |
Resolution |
Activity Label |
Spatial Label |
Dihedral Label |
Chelix-SaltBridge |
ActLoopNT-ActLoopCT |
Ligand |
Type |
Residues in structure |
Mutation |
Phosphorylation |
Unresolved residues in A-loop |
| Homo sapiens |
CHK1_HUMAN |
3JVRA |
1.76 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AGX |
Allosteric |
2 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3JVSA |
1.9 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
AGY |
Allosteric |
2 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3F9NA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
38M |
Allosteric |
7 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
AF-O14757-K1A |
-1.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
1 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
1IA8A |
1.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7AKMB |
1.93 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
2 - 269 |
D10R |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
1ZYSA |
1.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
199 |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2E9VA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
85A |
Type1 |
2 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2E9VB |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
85A |
Type1 |
2 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2E9OA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A58 |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2E9PA |
2.6 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
77A |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2E9UA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A25 |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2GHGA |
3.5 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A53 |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YWPA |
2.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A42 |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3OT3A |
1.44 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
22K |
Type1 |
4 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3OT8A |
1.645 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
MI5 |
Type1 |
4 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3PA3A |
1.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
C70 |
Type1 |
4 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3PA4A |
1.59 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
C72 |
Type1 |
6 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3PA5A |
1.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
C73 |
Type1 |
3 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3U9NA |
1.85 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
09H |
Type1 |
7 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4JIKA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1KO |
Type1 |
4 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2X8EA |
2.5 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
X8E |
Type1 |
9 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YDJA |
1.85 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YDJ |
Type1 |
8 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YDJB |
1.85 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YDJ |
Type1 |
9 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YDKA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YDK |
Type1 |
3 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YERA |
1.83 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
TQ1 |
Type1 |
2 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YEXA |
1.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YEX |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
6FC8A |
1.61 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
D4Q |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
6FCFA |
1.85 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
D58 |
Type1 |
9 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
6FCKA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
D4Z |
Type1 |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSNA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A58 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSMA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK1 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSRA |
2.5 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HKC |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSWA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK6 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSYA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK7 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSZA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK8 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FT0A |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK9 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FT3A |
2.5 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H1K |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FT5A |
2.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H2K |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FT7A |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H3K |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FT9A |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H4K |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTAA |
2.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H5K |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTCA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H6K |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTIA |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H7K |
Type1 |
3 - 279 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTJA |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H8K |
Type1 |
3 - 279 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTOA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3HK |
Type1 |
3 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTQA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4HK |
Type1 |
3 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTRA |
2.25 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
5HK |
Type1 |
3 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTTA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
6HK |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTUA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
7HK |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4GH2A |
2.03 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK0 |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
1NVQA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
UCN |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
1NVRA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
STU |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
1NVSA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
UCM |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMQA |
2.48 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYQ |
Type1 |
7 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMRA |
2.43 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYR |
Type1 |
7 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMSA |
2.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYS |
Type1 |
7 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMTA |
2.55 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYT |
Type1 |
8 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMUA |
2.6 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYU |
Type1 |
9 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMVA |
2.009 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYV |
Type1 |
7 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMWA |
2.43 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZYW |
Type1 |
7 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2WMXA |
2.45 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZY6 |
Type1 |
7 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2X8DA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
X8D |
Type1 |
2 - 281 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2X8IA |
1.92 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
X8I |
Type1 |
2 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2XEYA |
2.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YVQ |
Type1 |
6 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2XEZA |
2.25 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XEZ |
Type1 |
7 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2XF0A |
2.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4UB |
Type1 |
4 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YDIA |
1.6 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YDI |
Type1 |
2 - 281 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YM3A |
2.007 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YM3 |
Type1 |
8 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YM4A |
2.35 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4YM |
Type1 |
4 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YM5A |
2.03 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
YM5 |
Type1 |
8 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YM6A |
2.01 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
YM6 |
Type1 |
7 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YM8A |
2.07 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YM8 |
Type1 |
8 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4HYHA |
1.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1AM |
Type1 |
4 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4HYIA |
1.399 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1AO |
Type1 |
3 - 274 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
1ZLTA |
1.74 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HYM |
Type1 |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2GDOA |
3.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
12C |
Type1 |
1 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BR1A |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
PFP |
Type1 |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BRBA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
PFQ |
Type1 |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BRGA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
DFY |
Type1 |
7 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BRHA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
DFW |
Type1 |
6 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BRMA |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
DFZ |
Type1 |
7 - 274 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BRNA |
2.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
DF1 |
Type1 |
6 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2BROA |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
DF2 |
Type1 |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2C3JA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
DBQ |
Type1 |
6 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2C3LA |
2.35 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
IDZ |
Type1 |
2 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2CGUA |
2.5 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3A3 |
Type1 |
6 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2CGVA |
2.6 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3B3 |
Type1 |
6 - 272 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2CGWA |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3C3 |
Type1 |
6 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2CGXA |
2.2 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3D3 |
Type1 |
6 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3NLBA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
5BE |
Type1 |
6 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5DLSA |
2.15 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
5CV |
Type1 |
6 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BKNA |
2.74 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADE |
Type1 |
7 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BKOA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
TVW |
Type1 |
7 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4QYEA |
2.05 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3DL |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4QYFA |
2.15 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3DV |
Type1 |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4QYGA |
1.75 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3DW |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4QYGB |
1.75 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3DW |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4QYHA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3DX |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4QYHB |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3DX |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4RVKA |
1.85 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3XK |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4RVLA |
1.85 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3XL |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4RVMA |
1.86 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3X7 |
Type1 |
3 - 273 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7AKMA |
1.93 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AGS |
Type1 |
2 - 271 |
D10R |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7AKOA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
STU |
Type1 |
2 - 271 |
D10R |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7AKOB |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
STU |
Type1 |
2 - 271 |
D10R |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2HOGA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
710 |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2HXLA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
422 |
Type1 |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2HXQA |
2.0 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
373 |
Type1 |
2 - 276 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2HY0A |
1.7 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
306 |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2QHMA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
7CS |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2QHNA |
1.7 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
582 |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2R0UA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
M54 |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3TKHA |
1.79 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
07S |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
3TKIA |
1.6 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
S25 |
Type1 |
2 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OQ5A |
1.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4K4 |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OQ7A |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A0Q |
Type1 |
8 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OQ7B |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A0Q |
Type1 |
8 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSUA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK5 |
Type1 |
4 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OQ6A |
1.95 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4K4 |
Type1 |
5 - 270 |
A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OQ8A |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A0Q |
Type1 |
4 - 270 |
A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
9CE4A |
1.31 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A1AV4 |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OOPA |
1.7 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
ANP |
Type1 |
5 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OORA |
1.9 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
3 - 283 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OOTA |
2.1 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4K4 |
Type1 |
4 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OP2A |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A0Q |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OP4A |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A0T |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OP5A |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3FE |
Type1 |
4 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OP7A |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A1K |
Type1 |
4 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OPBA |
1.55 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A1N |
Type1 |
5 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OPRA |
1.95 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A3E |
Type1 |
4 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OPSA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A3Q |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OPUA |
1.55 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A3K |
Type1 |
3 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5OPVA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A3H |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJDA |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
TVT |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJEA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADE |
Type1 |
4 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJHA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
42C |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJJA |
1.8 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
TVW |
Type1 |
3 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJMA |
2.3 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
TW2 |
Type1 |
5 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJOA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
TWK |
Type1 |
5 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJRA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
TWH |
Type1 |
5 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJXA |
2.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
U0Q |
Type1 |
8 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BJXB |
2.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
U0Q |
Type1 |
8 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BK1A |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
U0N |
Type1 |
8 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BK2A |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
U0K |
Type1 |
5 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7BK3A |
2.0 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
U0T |
Type1 |
5 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7MCKA |
1.65 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YXD |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7SUFA |
1.48 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BVI |
Type1 |
3 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7SUGA |
1.48 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BWI |
Type1 |
3 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7SUHA |
2.46 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BXI |
Type1 |
4 - 270 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7SUIA |
2.119 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L80 |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7SUJA |
2.299 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
BYL |
Type1 |
9 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
7SUJB |
2.299 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BYL |
Type1 |
9 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
8E80A |
1.49 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
UUF |
Type1 |
8 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
8E81A |
1.62 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
UU6 |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
8SIVA |
1.759 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZXH |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
8SIWA |
1.877 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZXL |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
8SIWB |
1.877 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZXL |
Type1 |
4 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
8SIXA |
1.55 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZXP |
Type1 |
8 - 271 |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
5F4NA |
1.91 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
5UY
5UY
|
Type1
Allosteric
|
5 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2YM7A |
1.81 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YM7
YM7
|
Type1
Type1
|
7 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2E9NA |
2.5 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
76A |
Type1.5_Back |
2 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSTA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK4 |
Type1.5_Back |
3 - 270 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2AYPA |
2.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
43A |
Type1.5_Back |
2 - 269 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FSQA |
2.4 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HK3 |
Type1.5_Back |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTKA |
2.3 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H9K |
Type1.5_Back |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTLA |
2.5 |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
H0K |
Type1.5_Back |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTMA |
1.9 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1HK |
Type1.5_Back |
3 - 280 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
4FTNA |
2.02 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
2HK |
Type1.5_Back |
3 - 271 |
None |
None |
0 |
| Homo sapiens |
CHK1_HUMAN |
2C3KA |
2.6 |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ABO |
Type1.5_Back |
6 - 270 |
None |
None |
0 |