Ligand: 5ID

Total number of chains: 22
Active chains: 8
Total number of genes: 6
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 22 100.0% 6G3AA

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
CK1 CSNK1G2 KC1G2_HUMAN 2C47A 2.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 44 - 338 0 None None Casein kinase I isoform gamma-2
CK1 CSNK1G2 KC1G2_HUMAN 2C47B 2.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 44 - 338 0 None None Casein kinase I isoform gamma-2
CK1 CSNK1G2 KC1G2_HUMAN 2C47C 2.4 None DFGin‑BLAminus in-none in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 46 - 337 0 None None Casein kinase I isoform gamma-2
CK1 CSNK1G2 KC1G2_HUMAN 2C47D 2.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 43 - 338 0 None None Casein kinase I isoform gamma-2
CMGC CLK1 CLK1_HUMAN 6G33A 2.05 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaino APEdist_oioo 5ID Type1 148 - 482 0 SEP341,TPO342 None Dual specificity protein kinase CLK1
CMGC CLK1 CLK1_HUMAN 6G33B 2.05 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiio APEdist_iioo 5ID Type1 148 - 482 0 None None Dual specificity protein kinase CLK1
CMGC CLK1 CLK1_HUMAN 6G33C 2.05 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaini APEdist_oioi 5ID Type1 148 - 482 0 None None Dual specificity protein kinase CLK1
CMGC CSNK2A1 CSK21_HUMAN 6JWAA 1.781 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_iiii 5ID Type1 2 - 328 0 None None Casein kinase II subunit alpha
CMGC MAPK1 MK01_HUMAN 8ZJVA 1.8 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 10 - 358 0 None None Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 5AX3A 2.984 Inactive DFGin‑BLAminus out-out in-out nonTYR APEdihe_aanii APEdist_iion 5ID Type1 10 - 358 0 None None Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 7W5OA 2.35 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_ioii 5ID Type1 11 - 360 0 None None Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 7XC1B 2.09 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_ioii 5ID Type1 12 - 357 0 None None Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 7XC1A 2.09 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_ioii 5ID, B8Z Type1, Allosteric 10 - 360 0 None None Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 7X4UA 1.98 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID, 8DK, BTB Type1, Allosteric, Allosteric 10 - 359 0 None None Mitogen-activated protein kinase 1
CMGC MAPK3 MK03_HUMAN 2ZOQA 2.39 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_oiii 5ID Type1 24 - 375 0 PTR204 None Mitogen-activated protein kinase 3
CMGC MAPK3 MK03_HUMAN 2ZOQB 2.39 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaoio APEdist_iiii 5ID Type1 24 - 375 0 PTR204 None Mitogen-activated protein kinase 3
OTHER HASPIN HASP_HUMAN 6G39A 1.45 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 471 - 798 0 None F605Y Serine/threonine-protein kinase haspin
OTHER HASPIN HASP_HUMAN 2VUWA 1.8 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 470 - 798 0 None None Serine/threonine-protein kinase haspin
OTHER HASPIN HASP_HUMAN 3IQ7A 2.0 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 471 - 798 0 None None Serine/threonine-protein kinase haspin
OTHER HASPIN HASP_HUMAN 4OUCA 1.9 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 470 - 798 0 None None Serine/threonine-protein kinase haspin
OTHER HASPIN HASP_HUMAN 6G34A 1.76 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 472 - 798 0 None None Serine/threonine-protein kinase haspin
OTHER HASPIN HASP_HUMAN 6G3AA 1.43 Inactive DFGin‑BLAminus in-out in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 471 - 798 0 None F605T Serine/threonine-protein kinase haspin

Ligand: 5ID

Total number of chains: 22
Active chains: 8
Total number of genes: 6
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 22 100.0% 6G3AA

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
CK1 CSNK1G2 KC1G2_HUMAN 2C47A 2.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 44 - 338 0 None None Casein kinase I isoform gamma-2 Homo sapiens
CK1 CSNK1G2 KC1G2_HUMAN 2C47B 2.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 44 - 338 0 None None Casein kinase I isoform gamma-2 Homo sapiens
CK1 CSNK1G2 KC1G2_HUMAN 2C47C 2.4 None DFGin‑BLAminus in-none in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 46 - 337 0 None None Casein kinase I isoform gamma-2 Homo sapiens
CK1 CSNK1G2 KC1G2_HUMAN 2C47D 2.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 43 - 338 0 None None Casein kinase I isoform gamma-2 Homo sapiens
CMGC CLK1 CLK1_HUMAN 6G33A 2.05 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaino APEdist_oioo 5ID Type1 148 - 482 0 SEP341,TPO342 None Dual specificity protein kinase CLK1 Homo sapiens
CMGC CLK1 CLK1_HUMAN 6G33B 2.05 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiio APEdist_iioo 5ID Type1 148 - 482 0 None None Dual specificity protein kinase CLK1 Homo sapiens
CMGC CLK1 CLK1_HUMAN 6G33C 2.05 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaini APEdist_oioi 5ID Type1 148 - 482 0 None None Dual specificity protein kinase CLK1 Homo sapiens
CMGC CSNK2A1 CSK21_HUMAN 6JWAA 1.781 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_iiii 5ID Type1 2 - 328 0 None None Casein kinase II subunit alpha Homo sapiens
CMGC MAPK1 MK01_HUMAN 8ZJVA 1.8 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID Type1 10 - 358 0 None None Mitogen-activated protein kinase 1 Homo sapiens
CMGC MAPK1 MK01_HUMAN 5AX3A 2.984 Inactive DFGin‑BLAminus out-out in-out nonTYR APEdihe_aanii APEdist_iion 5ID Type1 10 - 358 0 None None Mitogen-activated protein kinase 1 Homo sapiens
CMGC MAPK1 MK01_HUMAN 7W5OA 2.35 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_ioii 5ID Type1 11 - 360 0 None None Mitogen-activated protein kinase 1 Homo sapiens
CMGC MAPK1 MK01_HUMAN 7XC1B 2.09 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_ioii 5ID Type1 12 - 357 0 None None Mitogen-activated protein kinase 1 Homo sapiens
CMGC MAPK1 MK01_HUMAN 7XC1A 2.09 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_ioii 5ID, B8Z Type1, Allosteric 10 - 360 0 None None Mitogen-activated protein kinase 1 Homo sapiens
CMGC MAPK1 MK01_HUMAN 7X4UA 1.98 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii 5ID, 8DK, BTB Type1, Allosteric, Allosteric 10 - 359 0 None None Mitogen-activated protein kinase 1 Homo sapiens
CMGC MAPK3 MK03_HUMAN 2ZOQA 2.39 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_oiii 5ID Type1 24 - 375 0 PTR204 None Mitogen-activated protein kinase 3 Homo sapiens
CMGC MAPK3 MK03_HUMAN 2ZOQB 2.39 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaoio APEdist_iiii 5ID Type1 24 - 375 0 PTR204 None Mitogen-activated protein kinase 3 Homo sapiens
OTHER HASPIN HASP_HUMAN 6G39A 1.45 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 471 - 798 0 None F605Y Serine/threonine-protein kinase haspin Homo sapiens
OTHER HASPIN HASP_HUMAN 2VUWA 1.8 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 470 - 798 0 None None Serine/threonine-protein kinase haspin Homo sapiens
OTHER HASPIN HASP_HUMAN 3IQ7A 2.0 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 471 - 798 0 None None Serine/threonine-protein kinase haspin Homo sapiens
OTHER HASPIN HASP_HUMAN 4OUCA 1.9 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 470 - 798 0 None None Serine/threonine-protein kinase haspin Homo sapiens
OTHER HASPIN HASP_HUMAN 6G34A 1.76 Active DFGin‑BLAminus in-in in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 472 - 798 0 None None Serine/threonine-protein kinase haspin Homo sapiens
OTHER HASPIN HASP_HUMAN 6G3AA 1.43 Inactive DFGin‑BLAminus in-out in-na noAPE APEdihe_aaaaa APEdist_aaaa 5ID Type1 471 - 798 0 None F605T Serine/threonine-protein kinase haspin Homo sapiens

Ligand: 5ID

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism