| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47A | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 44 - 338 | 0 | None | None | Casein kinase I isoform gamma-2 |
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47B | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 44 - 338 | 0 | None | None | Casein kinase I isoform gamma-2 |
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47C | 2.4 | None | DFGin‑BLAminus | in-none | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 46 - 337 | 0 | None | None | Casein kinase I isoform gamma-2 |
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47D | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 43 - 338 | 0 | None | None | Casein kinase I isoform gamma-2 |
| CMGC | CLK1 | CLK1_HUMAN | 6G33A | 2.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaino | APEdist_oioo | 5ID | Type1 | 148 - 482 | 0 | SEP341,TPO342 | None | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6G33B | 2.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiio | APEdist_iioo | 5ID | Type1 | 148 - 482 | 0 | None | None | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6G33C | 2.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaini | APEdist_oioi | 5ID | Type1 | 148 - 482 | 0 | None | None | Dual specificity protein kinase CLK1 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 6JWAA | 1.781 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 5ID | Type1 | 2 - 328 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | MAPK1 | MK01_HUMAN | 8ZJVA | 1.8 | Inactive | DFGin‑BLAminus | in-out | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 10 - 358 | 0 | None | None | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 5AX3A | 2.984 | Inactive | DFGin‑BLAminus | out-out | in-out | nonTYR | APEdihe_aanii | APEdist_iion | 5ID | Type1 | 10 - 358 | 0 | None | None | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 7W5OA | 2.35 | Inactive | DFGin‑BLAminus | in-out | in-out | nonTYR | APEdihe_aaiii | APEdist_ioii | 5ID | Type1 | 11 - 360 | 0 | None | None | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 7XC1B | 2.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_ioii | 5ID | Type1 | 12 - 357 | 0 | None | None | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 7XC1A | 2.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_ioii | 5ID, B8Z | Type1, Allosteric | 10 - 360 | 0 | None | None | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 7X4UA | 1.98 | Inactive | DFGin‑BLAminus | in-out | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID, 8DK, BTB | Type1, Allosteric, Allosteric | 10 - 359 | 0 | None | None | Mitogen-activated protein kinase 1 |
| CMGC | MAPK3 | MK03_HUMAN | 2ZOQA | 2.39 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_oiii | 5ID | Type1 | 24 - 375 | 0 | PTR204 | None | Mitogen-activated protein kinase 3 |
| CMGC | MAPK3 | MK03_HUMAN | 2ZOQB | 2.39 | Inactive | DFGin‑BLAminus | in-out | in-out | nonTYR | APEdihe_aaoio | APEdist_iiii | 5ID | Type1 | 24 - 375 | 0 | PTR204 | None | Mitogen-activated protein kinase 3 |
| OTHER | HASPIN | HASP_HUMAN | 6G39A | 1.45 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 471 - 798 | 0 | None | F605Y | Serine/threonine-protein kinase haspin |
| OTHER | HASPIN | HASP_HUMAN | 2VUWA | 1.8 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 470 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin |
| OTHER | HASPIN | HASP_HUMAN | 3IQ7A | 2.0 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 471 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin |
| OTHER | HASPIN | HASP_HUMAN | 4OUCA | 1.9 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 470 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin |
| OTHER | HASPIN | HASP_HUMAN | 6G34A | 1.76 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 472 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin |
| OTHER | HASPIN | HASP_HUMAN | 6G3AA | 1.43 | Inactive | DFGin‑BLAminus | in-out | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 471 - 798 | 0 | None | F605T | Serine/threonine-protein kinase haspin |
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47A | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 44 - 338 | 0 | None | None | Casein kinase I isoform gamma-2 | Homo sapiens |
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47B | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 44 - 338 | 0 | None | None | Casein kinase I isoform gamma-2 | Homo sapiens |
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47C | 2.4 | None | DFGin‑BLAminus | in-none | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 46 - 337 | 0 | None | None | Casein kinase I isoform gamma-2 | Homo sapiens |
| CK1 | CSNK1G2 | KC1G2_HUMAN | 2C47D | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 43 - 338 | 0 | None | None | Casein kinase I isoform gamma-2 | Homo sapiens |
| CMGC | CLK1 | CLK1_HUMAN | 6G33A | 2.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaino | APEdist_oioo | 5ID | Type1 | 148 - 482 | 0 | SEP341,TPO342 | None | Dual specificity protein kinase CLK1 | Homo sapiens |
| CMGC | CLK1 | CLK1_HUMAN | 6G33B | 2.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiio | APEdist_iioo | 5ID | Type1 | 148 - 482 | 0 | None | None | Dual specificity protein kinase CLK1 | Homo sapiens |
| CMGC | CLK1 | CLK1_HUMAN | 6G33C | 2.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaini | APEdist_oioi | 5ID | Type1 | 148 - 482 | 0 | None | None | Dual specificity protein kinase CLK1 | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 6JWAA | 1.781 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 5ID | Type1 | 2 - 328 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | MAPK1 | MK01_HUMAN | 8ZJVA | 1.8 | Inactive | DFGin‑BLAminus | in-out | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID | Type1 | 10 - 358 | 0 | None | None | Mitogen-activated protein kinase 1 | Homo sapiens |
| CMGC | MAPK1 | MK01_HUMAN | 5AX3A | 2.984 | Inactive | DFGin‑BLAminus | out-out | in-out | nonTYR | APEdihe_aanii | APEdist_iion | 5ID | Type1 | 10 - 358 | 0 | None | None | Mitogen-activated protein kinase 1 | Homo sapiens |
| CMGC | MAPK1 | MK01_HUMAN | 7W5OA | 2.35 | Inactive | DFGin‑BLAminus | in-out | in-out | nonTYR | APEdihe_aaiii | APEdist_ioii | 5ID | Type1 | 11 - 360 | 0 | None | None | Mitogen-activated protein kinase 1 | Homo sapiens |
| CMGC | MAPK1 | MK01_HUMAN | 7XC1B | 2.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_ioii | 5ID | Type1 | 12 - 357 | 0 | None | None | Mitogen-activated protein kinase 1 | Homo sapiens |
| CMGC | MAPK1 | MK01_HUMAN | 7XC1A | 2.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_ioii | 5ID, B8Z | Type1, Allosteric | 10 - 360 | 0 | None | None | Mitogen-activated protein kinase 1 | Homo sapiens |
| CMGC | MAPK1 | MK01_HUMAN | 7X4UA | 1.98 | Inactive | DFGin‑BLAminus | in-out | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 5ID, 8DK, BTB | Type1, Allosteric, Allosteric | 10 - 359 | 0 | None | None | Mitogen-activated protein kinase 1 | Homo sapiens |
| CMGC | MAPK3 | MK03_HUMAN | 2ZOQA | 2.39 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_oiii | 5ID | Type1 | 24 - 375 | 0 | PTR204 | None | Mitogen-activated protein kinase 3 | Homo sapiens |
| CMGC | MAPK3 | MK03_HUMAN | 2ZOQB | 2.39 | Inactive | DFGin‑BLAminus | in-out | in-out | nonTYR | APEdihe_aaoio | APEdist_iiii | 5ID | Type1 | 24 - 375 | 0 | PTR204 | None | Mitogen-activated protein kinase 3 | Homo sapiens |
| OTHER | HASPIN | HASP_HUMAN | 6G39A | 1.45 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 471 - 798 | 0 | None | F605Y | Serine/threonine-protein kinase haspin | Homo sapiens |
| OTHER | HASPIN | HASP_HUMAN | 2VUWA | 1.8 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 470 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin | Homo sapiens |
| OTHER | HASPIN | HASP_HUMAN | 3IQ7A | 2.0 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 471 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin | Homo sapiens |
| OTHER | HASPIN | HASP_HUMAN | 4OUCA | 1.9 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 470 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin | Homo sapiens |
| OTHER | HASPIN | HASP_HUMAN | 6G34A | 1.76 | Active | DFGin‑BLAminus | in-in | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 472 - 798 | 0 | None | None | Serine/threonine-protein kinase haspin | Homo sapiens |
| OTHER | HASPIN | HASP_HUMAN | 6G3AA | 1.43 | Inactive | DFGin‑BLAminus | in-out | in-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | 5ID | Type1 | 471 - 798 | 0 | None | F605T | Serine/threonine-protein kinase haspin | Homo sapiens |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|