AGC_PKN1 (Serine/threonine-protein kinase N1)

Total number of chains: 6
Active chains: 2
Uniprot: PKN1_HUMAN
Kinase Domain Residues: 615 - 874
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 2 33.3% 4OTDA
DFGin BLAminus 2 33.3% AF-Q16512-K1A
DFGin BLAplus 2 33.3% 4OTHA

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PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
AF-Q16512-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 607 - 882 0 None None Serine/threonine-protein kinase N1
AF-Q16512-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 607 - 882 0 None None Serine/threonine-protein kinase N1
4OTDA 2.0 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 605 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1
4OTGA 2.6 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 2V9 Type1 605 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1
4OTHA 1.8 Inactive DFGin‑BLAplus in-in out-none nonTYR APEdihe_aannn APEdist_nnnn DRN Type1 606 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1
4OTIA 1.93 Inactive DFGin‑BLAplus in-in none-none nonTYR APEdihe_aannn APEdist_nnnn MI1 Type1 606 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1

AGC_PKN1 (Serine/threonine-protein kinase N1)

Total number of chains: 6
Active chains: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 2 33.3% 4OTDA
DFGin BLAminus 2 33.3% AF-Q16512-K1A
DFGin BLAplus 2 33.3% 4OTHA

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
PKN1_HUMAN AF-Q16512-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 607 - 882 0 None None Serine/threonine-protein kinase N1 Homo sapiens
PKN1_HUMAN AF-Q16512-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 607 - 882 0 None None Serine/threonine-protein kinase N1 Homo sapiens
PKN1_HUMAN 4OTDA 2.0 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 605 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1 Homo sapiens
PKN1_HUMAN 4OTGA 2.6 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 2V9 Type1 605 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1 Homo sapiens
PKN1_HUMAN 4OTHA 1.8 Inactive DFGin‑BLAplus in-in out-none nonTYR APEdihe_aannn APEdist_nnnn DRN Type1 606 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1 Homo sapiens
PKN1_HUMAN 4OTIA 1.93 Inactive DFGin‑BLAplus in-in none-none nonTYR APEdihe_aannn APEdist_nnnn MI1 Type1 606 - 940 0 TPO774,SEP916 None Serine/threonine-protein kinase N1 Homo sapiens

AGC_PKN1 (Serine/threonine-protein kinase N1)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism