|
OTHER
|
BSK8
|
BSK8_ARATH
|
4I94A
|
1.8 |
Pseudo |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioo |
ANP |
ATPlike |
40 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase BSK8 |
Arabidopsis thaliana |
|
OTHER
|
BSK8
|
BSK8_ARATH
|
4I94B
|
1.8 |
Pseudo |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioo |
ANP |
ATPlike |
40 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase BSK8 |
Arabidopsis thaliana |
|
OTHER
|
BSK8
|
BSK8_ARATH
|
4I92A
|
1.6 |
Pseudo |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iooo |
No_ligand |
No_ligand |
40 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase BSK8 |
Arabidopsis thaliana |
|
OTHER
|
BSK8
|
BSK8_ARATH
|
4I93A
|
1.5 |
Pseudo |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioo |
No_ligand |
No_ligand |
40 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase BSK8 |
Arabidopsis thaliana |
|
OTHER
|
BSK8
|
BSK8_ARATH
|
4I93B
|
1.5 |
Pseudo |
DFGout‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
40 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase BSK8 |
Arabidopsis thaliana |
|
TKL
|
CTR1
|
CTR1_ARATH
|
3P86A
|
2.496 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
STU |
Type1 |
544 - 810 |
0 |
None |
D676N |
Serine/threonine-protein kinase CTR1 |
Arabidopsis thaliana |
|
TYR
|
SRC
|
SRC_CHICK
|
7D57A
|
2.104 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
37O |
Type1 |
258 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3WA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
1BU |
Type2 |
257 - 533 |
0 |
None |
T338M,S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3WB
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
1BU |
Type2 |
258 - 533 |
0 |
None |
T338M,S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3G6HB
|
2.35 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
G6H |
Type2 |
258 - 533 |
0 |
None |
T338I |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3OEZA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
STI |
Type2 |
257 - 533 |
0 |
None |
L317I |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3OEZB
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
STI |
Type2 |
256 - 533 |
0 |
None |
L317I |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
2OIQA
|
2.07 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
STI |
Type2 |
256 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3G6GA
|
2.31 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
G6G |
Type2 |
256 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
4YBJA
|
2.61 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
4A9 |
Type2 |
259 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
4YBJB
|
2.61 |
Inactive |
DFGout‑BBAminus |
in-none |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
4A9 |
Type2 |
259 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
7WF5A
|
1.798 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
0LI |
Type2 |
257 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
7WF5B
|
1.798 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
0LI |
Type2 |
254 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3VA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
1BU |
Type2 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3VB
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
1BU |
Type2 |
256 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3TZ7A
|
3.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
AQB |
Type2 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3TZ7B
|
3.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
AQB |
Type2 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3TZ8A
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
AQM |
Type2 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3TZ8B
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nioai |
APEdist_aaao |
AQM |
Type2 |
256 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3TZ9A
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
AQU |
Type2 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
5SYSA
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
72F |
Type2 |
258 - 533 |
0 |
None |
V281C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
5SYSB
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
72F |
Type2 |
258 - 533 |
0 |
None |
V281C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3UB
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
1AW |
Type3 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3TA
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
1AU,
1AU
|
Type3,
Type1
|
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3F3UA
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
1AW,
1AW
|
Type3,
Type1
|
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3D7TB
|
2.899 |
Inactive |
DFGout‑None |
in-in |
out-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
STU |
Type1 |
258 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
5K9IB
|
2.5 |
Inactive |
DFGout‑None |
out-out |
in-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
O44 |
Type1 |
259 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
7D5OB
|
2.69 |
Inactive |
DFGout‑None |
out-out |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
TZ0 |
Type1 |
258 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3EL7A
|
2.8 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
PD3 |
Type2 |
257 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3EL8A
|
2.3 |
Inactive |
DFGout‑None |
in-in |
in-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
PD5 |
Type2 |
258 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3G6GB
|
2.31 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
G6G |
Type2 |
256 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
4AGWA
|
2.6 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
NG7 |
Type2 |
257 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
4AGWB
|
2.6 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
NG7 |
Type2 |
258 - 533 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
TYR
|
SRC
|
SRC_CHICK
|
3TZ9B
|
3.1 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
AQU |
Type2 |
257 - 533 |
0 |
None |
S345C |
Proto-oncogene tyrosine-protein kinase Src |
Gallus gallus |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UVYA
|
2.11 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XOO |
Allosteric |
3 - 439 |
0 |
None |
E17K |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW2A
|
2.2 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
XOO |
Allosteric |
4 - 437 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW9A
|
1.9 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XQ2 |
Allosteric |
3 - 428 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW7A
|
1.972 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 439 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3O96A
|
2.7 |
Inactive |
DFGout‑BBAminus |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
IQO |
Allosteric |
2 - 429 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHHA
|
2.7 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
G4Q |
Allosteric |
2 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHJA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4H |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9WA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
L1Z |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EJNA
|
2.19 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
0R4 |
Type1 |
4 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
5KCVA
|
2.7 |
Inactive |
DFGout‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
6S1 |
Allosteric |
6 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7APJA
|
2.05 |
Inactive |
DFGout‑None |
none-none |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
3 - 439 |
0 |
None |
S2N |
RAC-alpha serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
9C1WA
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 440 |
0 |
None |
P115A,G116A |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
8Q61A
|
2.32 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
K06 |
Type3 |
1 - 435 |
0 |
None |
N2D |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZKA
|
2.3 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 441 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZOA
|
2.75 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZNA
|
2.5 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRVA
|
2.8 |
Inactive |
DFGout‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
147 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRYA
|
2.8 |
Inactive |
DFGout‑None |
none-none |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnio |
No_ligand |
No_ligand |
146 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAXA
|
1.75 |
Inactive |
DFGout‑BBAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MP7 |
Type2 |
76 - 360 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4A
|
1.8 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
76 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4B
|
1.8 |
Inactive |
DFGout‑None |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
51 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25A
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
86G |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25B
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
86G |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25C
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86G |
Type1 |
13 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUA
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUC
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSA
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSB
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSC
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSD
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
Z8O |
Type1.5_Front |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUB
|
3.02 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUD
|
3.02 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8EQ5A
|
1.8 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
QCT |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8R58A
|
2.31 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
QCT |
Type1 |
49 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYA
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
58 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYB
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
59 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYC
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
61 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYD
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYE
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
64 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYF
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 345 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYG
|
3.2 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYH
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYI
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYJ
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
65 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NUSA
|
2.39 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2NK |
Type1 |
53 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9LA
|
2.15 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
583 |
Type1 |
49 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KA
|
2.55 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KB
|
2.55 |
Inactive |
DFGout‑None |
in-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Homo sapiens |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
7PUEA
|
2.506 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
86H |
Type1 |
82 - 376 |
0 |
None |
R192A,S422D |
Serine/threonine-protein kinase Sgk1 |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6EA
|
2.1 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
HPM |
Type1.5_Back |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPJA
|
2.1 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
ANP |
ATPlike |
104 - 389 |
0 |
None |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPHA
|
2.14 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
ANP |
ATPlike |
7 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JAIA
|
3.2 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
XU2 |
Type1 |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7AYHA
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
S9H |
Type1 |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7O2VA
|
3.1 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
V0K |
Type1 |
117 - 390 |
0 |
None |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O51A
|
3.2 |
Inactive |
DFGout‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
LJF |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6HJKA
|
2.4 |
Inactive |
DFGout‑None |
out-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
G7W |
Type1.5_Front |
127 - 391 |
0 |
None |
L210C,C290A,C393A |
Aurora kinase A |
Homo sapiens |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5K00A
|
1.77 |
Inactive |
DFGout‑None |
out-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6PV |
Type2 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
Homo sapiens |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
2HW6A
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
39 - 376 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
2HW6B
|
2.5 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
40 - 375 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
5WVDA
|
3.0 |
Inactive |
DFGout‑None |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7UX |
Type1 |
41 - 375 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
5WVDB
|
3.0 |
Inactive |
DFGout‑None |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7UX |
Type1 |
41 - 374 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2AC3A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
No_ligand |
No_ligand |
72 - 369 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6JLRA
|
2.901 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BV9 |
Type1 |
72 - 369 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
2H6DA
|
1.85 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
10 - 278 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
Homo sapiens |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
2YZAA
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
10 - 278 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
Homo sapiens |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HNIA
|
2.74 |
Inactive |
DFGout‑BBAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
Homo sapiens |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HNIB
|
2.74 |
Inactive |
DFGout‑BBAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
Homo sapiens |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
5G6VA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
919 |
Type2 |
163 - 474 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
Homo sapiens |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
3MTLA
|
2.4 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FEF |
Type1 |
163 - 473 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
Homo sapiens |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
5G6VB
|
2.2 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
919 |
Type2 |
163 - 475 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
Homo sapiens |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5A14A
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LQ5,
LQ5
|
Type2,
Allosteric
|
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
Homo sapiens |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1G3NA
|
2.9 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
Homo sapiens |
|
CMGC
|
CDK6
|
CDK6_HUMAN
|
1G3NE
|
2.9 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 301 |
0 |
None |
None |
Cyclin-dependent kinase 6 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
3RGFA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BAX |
Type2 |
1 - 353 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F6UA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
0SR |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F6WA
|
2.39 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
0SS |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7LA
|
2.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
0SO |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7NA
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
0SV |
Type2 |
1 - 361 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
5HVYA
|
2.39 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
66X |
Type2 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
6TPAA
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
NZ8,
NZ5,
NZ5,
NZ5
|
Type2,
Allosteric,
Allosteric,
Allosteric
|
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F6SA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0SQ |
Type3 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CDK8
|
CDK8_HUMAN
|
4F7JA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0SU |
Type3 |
1 - 359 |
0 |
None |
None |
Cyclin-dependent kinase 8 |
Homo sapiens |
|
CMGC
|
CLK3
|
CLK3_HUMAN
|
9EZ3A
|
2.7 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
A1H74 |
Type2 |
136 - 481 |
0 |
None |
None |
Dual specificity protein kinase CLK3 |
Homo sapiens |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
3GP0A
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
NIL |
Type2 |
5 - 348 |
0 |
None |
None |
Mitogen-activated protein kinase 11 |
Homo sapiens |
|
CMGC
|
MAPK11
|
MK11_HUMAN
|
8YGWA
|
3.301 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
B96 |
Type2 |
5 - 348 |
0 |
None |
None |
Mitogen-activated protein kinase 11 |
Homo sapiens |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
4EYJA
|
2.102 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
N61 |
Type2 |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
Homo sapiens |
|
CMGC
|
MAPK13
|
MK13_HUMAN
|
5EKNA
|
2.594 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
N58 |
Type2 |
2 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 13 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9CJ3A
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
PDO,
A1AWV
|
Allosteric,
Type2
|
4 - 352 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6QDZA
|
1.73 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
I46,
HYK
|
Allosteric,
Type2
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6QE1A
|
1.85 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
I46,
HYW
|
Allosteric,
Type2
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GCQA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
1BU |
Type2 |
4 - 355 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GCSA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
BAX |
Type2 |
5 - 352 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GCVA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
SS6 |
Type2 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV3A
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
R49 |
Type2 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3LFEA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
Z84 |
Type2 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3LFFA
|
1.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
Z83 |
Type2 |
5 - 352 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3PG3A
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
DG7 |
Type2 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6SFIA
|
1.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LB5 |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6SFJA
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
LBB |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6SFOA
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
LBE |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6ZWPA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
OE8 |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3CTQA
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
337 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5MZ3A
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
8EN |
Type2 |
4 - 353 |
0 |
None |
C162S |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HEGA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
BAX |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1W83A
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
L11 |
Type2 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WBNA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
L09 |
Type2 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3D83A
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
GK6 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9CJ4A
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
B96 |
Type2 |
5 - 352 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GCUA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
R48 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GCUB
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
R48 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV4A
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
L51 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV4B
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
L51 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV5A
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
R24 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV5B
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
R24 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV6A
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
R39 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2BAKA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
AQZ |
Type2 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4A9YA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
AQZ |
Type2 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4AA0A
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
AA0 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3E93A
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
19B |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3KQ7A
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
KQ7 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3GI3A
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
B10 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3IW8A
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
HIZ |
Type3 |
4 - 352 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3LFBA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
Z87 |
Type3 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3LFCA
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
Z86 |
Type3 |
4 - 354 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3NNVA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
437 |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3NNXA
|
2.28 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nioo |
EDD |
Type3 |
5 - 352 |
0 |
PTR182 |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1W82A
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
L10 |
Type3 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WBVA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
LI3 |
Type3 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HV7A
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
1AU |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2BAJA
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
1PP |
Type3 |
2 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3O8UA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
BMU |
Type3 |
5 - 352 |
0 |
None |
F169Y |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3OBJA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
BMU |
Type3 |
5 - 352 |
0 |
None |
F169R |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3K3IA
|
1.7 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
JZJ,
I46,
I46
|
Type3,
Allosteric,
Allosteric
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5N64A
|
2.4 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
8OH |
Allosteric |
5 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
5N66A
|
2.4 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
BW1,
B96
|
Allosteric,
Type2
|
6 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4EH8A
|
2.2 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
IRG,
0OP,
0OP
|
Allosteric,
Type3,
Type1
|
4 - 354 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2FSMX
|
1.86 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
No_ligand |
No_ligand |
4 - 352 |
0 |
None |
D176A,F327S |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2NPQA
|
1.8 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
No_ligand |
No_ligand |
4 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4GEOA
|
1.66 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
No_ligand |
No_ligand |
5 - 351 |
0 |
None |
M194A,L195A,H228A,I229A,Y258A |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MH3A
|
2.2 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
F169R |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3MH1A
|
2.2 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
No_ligand |
No_ligand |
5 - 352 |
0 |
None |
F169G |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3IW5A
|
2.5 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
DF3 |
Type1 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3L8SA
|
2.35 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
BFF |
Type1 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
6SFKA
|
1.8 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
LB8 |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3HECA
|
2.5 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
STI |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3NNUA
|
2.4 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
EDB |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3NNWA
|
1.89 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
EDD |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1KV2A
|
2.8 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
B96 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WBSA
|
1.8 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
LI2 |
Type2 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1WBTA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
WBT |
Type2 |
4 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9CJ1A
|
1.8 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
NIL |
Type2 |
5 - 351 |
0 |
TPO180,PTR182 |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3UVRA
|
2.1 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
06F |
Type2 |
5 - 351 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
4L8MA
|
2.1 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
F46 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3BV3A
|
2.59 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nioo |
P39 |
Type2 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2YISA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
YIS,
I46
|
Type2,
Allosteric
|
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
2YIWA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
YIW,
I46
|
Type2,
Allosteric
|
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
9CJ5A
|
3.3 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
A1AWV,
PDO
|
Type2,
Allosteric
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3K3JA
|
1.995 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4C,
I46
|
Type2,
Allosteric
|
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3LFDA
|
3.4 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
Z85 |
Type3 |
4 - 353 |
0 |
None |
C119S,C162S,A172C,F327L |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
1KV1A
|
2.5 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
BMU |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3O8TA
|
2.0 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
BMU |
Type3 |
5 - 352 |
0 |
None |
F169A |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK14
|
MK14_HUMAN
|
3OC1A
|
2.59 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
BMU |
Type3 |
5 - 352 |
0 |
None |
F169G |
Mitogen-activated protein kinase 14 |
Homo sapiens |
|
CMGC
|
MAPK6
|
MK06_HUMAN
|
6YLCA
|
2.43 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
OXW |
Type1 |
15 - 320 |
0 |
None |
L290V |
Mitogen-activated protein kinase 6 |
Homo sapiens |
|
CMGC
|
MAPK9
|
MK09_HUMAN
|
3NPCA
|
2.35 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
B96 |
Type2 |
7 - 363 |
0 |
None |
D3K,C6V,S8N,Q14E,K203A,E204A,K250A,K251A |
Mitogen-activated protein kinase 9 |
Homo sapiens |
|
CMGC
|
MAPK9
|
MK09_HUMAN
|
3NPCB
|
2.35 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
B96 |
Type2 |
8 - 363 |
0 |
None |
D3K,C6V,S8N,Q14E,K203A,E204A,K250A,K251A |
Mitogen-activated protein kinase 9 |
Homo sapiens |
|
CMGC
|
PRP4K
|
PRP4K_HUMAN
|
6CNHA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
919 |
Type2 |
657 - 1005 |
0 |
None |
None |
Serine/threonine-protein kinase PRP4 homolog |
Homo sapiens |
|
NEK
|
NEK2
|
NEK2_HUMAN
|
2XK3A
|
2.2 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnno |
XK3 |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Nek2 |
Homo sapiens |
|
NEK
|
NEK2
|
NEK2_HUMAN
|
2XK4A
|
2.1 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nooo |
OL2 |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Nek2 |
Homo sapiens |
|
NEK
|
NEK2
|
NEK2_HUMAN
|
2XK8A
|
2.001 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnno |
5R1 |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Nek2 |
Homo sapiens |
|
NEK
|
NEK2
|
NEK2_HUMAN
|
2XNPA
|
1.98 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nooo |
WCX |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Nek2 |
Homo sapiens |
|
NEK
|
NEK2
|
NEK2_HUMAN
|
4AFEA
|
2.597 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnoo |
GGY |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Nek2 |
Homo sapiens |
|
NEK
|
NEK2
|
NEK2_HUMAN
|
4A4XA
|
2.4 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnoo |
JUP |
Type1 |
3 - 271 |
0 |
None |
T170E,S171D,T175E |
Serine/threonine-protein kinase Nek2 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
8WS0B
|
2.12 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
No_ligand |
No_ligand |
19 - 299 |
0 |
None |
S195D |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
8WS1B
|
2.4 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
No_ligand |
No_ligand |
20 - 300 |
0 |
None |
D161N |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
5DE2A
|
2.78 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnno |
No_ligand |
No_ligand |
20 - 300 |
0 |
None |
Y97F |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
6S75D
|
3.3 |
Inactive |
DFGout‑None |
out-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
28 - 299 |
0 |
None |
None |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
8WS0A
|
2.12 |
Inactive |
DFGout‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
20 - 300 |
0 |
None |
S195D |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
8SXNA
|
4.04 |
Inactive |
DFGout‑None |
out-na |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oiio |
No_ligand |
No_ligand |
19 - 302 |
0 |
None |
None |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
8SXNB
|
4.04 |
Inactive |
DFGout‑None |
out-na |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oiio |
No_ligand |
No_ligand |
19 - 302 |
0 |
None |
None |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
8WS1A
|
2.4 |
Inactive |
DFGout‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
20 - 300 |
0 |
None |
D161N |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
NEK
|
NEK7
|
NEK7_HUMAN
|
6S75A
|
3.3 |
Inactive |
DFGout‑None |
out-none |
none-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
F9N |
Type1 |
19 - 300 |
0 |
None |
None |
Serine/threonine-protein kinase Nek7 |
Homo sapiens |
|
OTHER
|
EIF2AK3
|
E2AK3_HUMAN
|
4X7JA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
3Z1 |
Type1 |
585 - 1086 |
0 |
None |
D937N |
Eukaryotic translation initiation factor 2-alpha kinase 3 |
Homo sapiens |
|
OTHER
|
EIF2AK3
|
E2AK3_HUMAN
|
4X7KA
|
1.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
3Z3 |
Type2 |
585 - 1087 |
0 |
None |
D937N |
Eukaryotic translation initiation factor 2-alpha kinase 3 |
Homo sapiens |
|
OTHER
|
EIF2AK3
|
E2AK3_HUMAN
|
4X7LA
|
1.9 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
3Z4 |
Type2 |
585 - 1087 |
0 |
None |
D937N |
Eukaryotic translation initiation factor 2-alpha kinase 3 |
Homo sapiens |
|
OTHER
|
EIF2AK3
|
E2AK3_HUMAN
|
4X7NA
|
2.35 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
3Z5 |
Type2 |
585 - 1087 |
0 |
None |
D937N |
Eukaryotic translation initiation factor 2-alpha kinase 3 |
Homo sapiens |
|
OTHER
|
EIF2AK3
|
E2AK3_HUMAN
|
4X7HA
|
2.0 |
Inactive |
DFGout‑None |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
3Z2 |
Type2 |
585 - 1086 |
0 |
None |
D937N |
Eukaryotic translation initiation factor 2-alpha kinase 3 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
7QWKA
|
2.3 |
Inactive |
DFGout‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
G41 |
Type1 |
583 - 998 |
0 |
None |
D848N |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
7QWKB
|
2.3 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
G41 |
Type1 |
583 - 998 |
0 |
None |
D848N |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
7QWKC
|
2.3 |
Inactive |
DFGout‑None |
out-out |
out-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
G41 |
Type1 |
583 - 1004 |
0 |
None |
D848N |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
7QWKD
|
2.3 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
G41 |
Type1 |
583 - 1003 |
0 |
None |
D848N |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
7QWKE
|
2.3 |
Inactive |
DFGout‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
G41 |
Type1 |
584 - 1004 |
0 |
None |
D848N |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
7QWKG
|
2.3 |
Inactive |
DFGout‑None |
out-out |
out-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
G41 |
Type1 |
584 - 1007 |
0 |
None |
D848N |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
6N3LA
|
2.61 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
KAV |
Type2 |
584 - 1002 |
0 |
None |
K807A,D848N,T899A,T904A |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
EIF2AK4-2
|
E2AK4_HUMAN
|
6N3LB
|
2.61 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
KAV |
Type2 |
584 - 1002 |
0 |
None |
K807A,D848N,T899A,T904A |
eIF-2-alpha kinase GCN2 |
Homo sapiens |
|
OTHER
|
ERN1
|
ERN1_HUMAN
|
4YZ9A
|
2.463 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
4K7 |
Type3 |
562 - 964 |
0 |
None |
None |
Serine/threonine-protein kinase/endoribonuclease IRE1 |
Homo sapiens |
|
OTHER
|
ERN1
|
ERN1_HUMAN
|
4YZ9B
|
2.463 |
Inactive |
DFGout‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
4K7 |
Type3 |
563 - 963 |
0 |
None |
None |
Serine/threonine-protein kinase/endoribonuclease IRE1 |
Homo sapiens |
|
OTHER
|
ERN1
|
ERN1_HUMAN
|
4YZ9C
|
2.463 |
Inactive |
DFGout‑None |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
4K7 |
Type3 |
562 - 964 |
0 |
None |
None |
Serine/threonine-protein kinase/endoribonuclease IRE1 |
Homo sapiens |
|
OTHER
|
MLKL
|
MLKL_HUMAN
|
6O5ZB
|
2.285 |
Pseudo |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
LN4 |
Type2 |
190 - 467 |
0 |
None |
None |
Mixed lineage kinase domain-like protein |
Homo sapiens |
|
OTHER
|
ULK3
|
ULK3_HUMAN
|
6FDZU
|
2.55 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
C87 |
Type1 |
8 - 274 |
0 |
None |
None |
Serine/threonine-protein kinase ULK3 |
Homo sapiens |
|
STE
|
MAP2K1
|
MP2K1_HUMAN
|
5HZEA
|
2.4 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
E62 |
Type1 |
43 - 382 |
0 |
None |
S298N,S299K,Y300F |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP2K1
|
MP2K1_HUMAN
|
8YP4B
|
2.35 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
WNT |
Type1 |
43 - 383 |
0 |
None |
T286A,T292A,S298A |
Dual specificity mitogen-activated protein kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP2K6
|
MP2K6_HUMAN
|
8P7JA
|
2.4 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
X3K |
Type1 |
47 - 333 |
0 |
None |
S207D,T211D |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
|
STE
|
MAP2K6
|
MP2K6_HUMAN
|
8P7JB
|
2.4 |
Inactive |
DFGout‑None |
out-na |
out-out |
nonTYR |
APEdihe_aanao |
APEdist_nnnn |
X3K |
Type1 |
47 - 333 |
0 |
None |
S207D,T211D |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
|
STE
|
MAP2K6
|
MP2K6_HUMAN
|
8PM3A
|
2.0 |
Inactive |
DFGout‑None |
out-na |
out-out |
nonTYR |
APEdihe_aanao |
APEdist_nnnn |
ZLE |
Type1 |
47 - 333 |
0 |
None |
S207D,T211D |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
|
STE
|
MAP2K6
|
MP2K6_HUMAN
|
8PM3B
|
2.0 |
Inactive |
DFGout‑None |
out-na |
out-out |
nonTYR |
APEdihe_aanao |
APEdist_nnnn |
ZLE |
Type1 |
47 - 333 |
0 |
None |
S207D,T211D |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
|
STE
|
MAP2K6
|
MP2K6_HUMAN
|
8PM3C
|
2.0 |
Inactive |
DFGout‑None |
out-na |
out-out |
nonTYR |
APEdihe_aanao |
APEdist_nnnn |
ZLE |
Type1 |
47 - 333 |
0 |
None |
S207D,T211D |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
|
STE
|
MAP2K6
|
MP2K6_HUMAN
|
8PM3D
|
2.0 |
Inactive |
DFGout‑None |
out-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ZLE |
Type1 |
47 - 333 |
0 |
None |
S207D,T211D |
Dual specificity mitogen-activated protein kinase kinase 6 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG7A
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-na |
none-out |
nonTYR |
APEdihe_aanao |
APEdist_nnnn |
OQ2 |
Type2 |
102 - 403 |
0 |
None |
S271D,T275D |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG7B
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-na |
none-out |
nonTYR |
APEdihe_aaiao |
APEdist_nnno |
OQ2 |
Type2 |
103 - 403 |
0 |
None |
S271D,T275D |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YZ4A
|
1.7 |
Inactive |
DFGout‑None |
in-na |
out-out |
nonTYR |
APEdihe_aaoai |
APEdist_nnno |
1E8 |
Allosteric |
101 - 404 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
5Y8UA
|
2.92 |
Inactive |
DFGout‑None |
out-na |
none-out |
nonTYR |
APEdihe_aaiao |
APEdist_nnoo |
No_ligand |
No_ligand |
103 - 402 |
0 |
None |
C260S |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
5Y90A
|
1.3 |
Inactive |
DFGout‑None |
in-na |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnoi |
No_ligand |
No_ligand |
103 - 419 |
0 |
None |
C202S |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
5B2LA
|
2.1 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aaiai |
APEdist_nnni |
No_ligand |
No_ligand |
104 - 403 |
0 |
None |
C202S |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YFZA
|
1.9 |
Inactive |
DFGout‑None |
in-na |
out-out |
nonTYR |
APEdihe_aaoai |
APEdist_nnno |
No_ligand |
No_ligand |
100 - 405 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6QFRA
|
2.3 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
102 - 402 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
5B2KA
|
2.75 |
Inactive |
DFGout‑None |
out-na |
none-out |
nonTYR |
APEdihe_aaoai |
APEdist_nnno |
No_ligand |
No_ligand |
104 - 400 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG0A
|
2.0 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
102 - 402 |
0 |
None |
S271D,T275D |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
7CBXA
|
2.061 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
FU6 |
Type1 |
103 - 402 |
0 |
None |
C202S |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
5Z1EA
|
2.3 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aaiai |
APEdist_nnni |
95U |
Type1 |
103 - 419 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG4A
|
2.3 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
SU9 |
Type1 |
103 - 401 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG5A
|
2.4 |
Inactive |
DFGout‑None |
in-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
IHH |
Type1 |
101 - 403 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
3WZUA
|
3.01 |
Inactive |
DFGout‑None |
none-na |
none-out |
nonTYR |
APEdihe_aaoai |
APEdist_nnno |
1FM |
Type1 |
104 - 402 |
0 |
None |
None |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG6A
|
2.15 |
Inactive |
DFGout‑None |
out-na |
none-out |
nonTYR |
APEdihe_aaiao |
APEdist_nnno |
OQ8 |
Type2 |
103 - 403 |
0 |
None |
S271D,T275D |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP2K7
|
MP2K7_HUMAN
|
6YG6B
|
2.15 |
Inactive |
DFGout‑None |
out-na |
none-out |
nonTYR |
APEdihe_aaiao |
APEdist_nnno |
OQ8 |
Type2 |
104 - 403 |
0 |
None |
S271D,T275D |
Dual specificity mitogen-activated protein kinase kinase 7 |
Homo sapiens |
|
STE
|
MAP3K2
|
M3K2_HUMAN
|
9P6AA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
0LI |
Type2 |
351 - 617 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 2 |
Homo sapiens |
|
STE
|
MAP3K2
|
M3K2_HUMAN
|
9P6AB
|
2.4 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
0LI |
Type2 |
347 - 618 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 2 |
Homo sapiens |
|
STE
|
MAP3K5
|
M3K5_HUMAN
|
8QGYA
|
3.71 |
Inactive |
DFGout‑None |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
95 - 940 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 5 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0KA
|
2.01 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK7 |
Type1 |
6 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0KB
|
2.01 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK7 |
Type1 |
8 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0KC
|
2.01 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK7 |
Type1 |
8 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0KD
|
2.01 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK7 |
Type1 |
6 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0LA
|
2.43 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK4 |
Type1 |
6 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0LB
|
2.43 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK4 |
Type1 |
7 - 291 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0LC
|
2.43 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK4 |
Type1 |
5 - 293 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
7M0LD
|
2.43 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YK4 |
Type1 |
6 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8XN7A
|
2.65 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
A1LVT |
Type1 |
6 - 292 |
0 |
None |
T165E,S171E |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8XN7B
|
2.65 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
A1LVT |
Type1 |
6 - 293 |
0 |
None |
T165E,S171E |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
6NG0B
|
2.05 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
B49 |
Type1 |
7 - 293 |
0 |
None |
T165E,S171E |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
9BIKA
|
2.25 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A1APO |
Type1 |
6 - 293 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
9N7RB
|
2.13 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A1BWC |
Type1 |
8 - 293 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
9N7RA
|
2.13 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
A1BWC,
A1BWC,
A1BWC,
A1BWC
|
Allosteric,
Allosteric,
Type1,
Type3
|
6 - 293 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8PAUA
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
XOR |
Type1 |
7 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8PAUB
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
XOR |
Type1 |
7 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8PASA
|
2.7 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
XOH |
Type1 |
8 - 295 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8PASB
|
2.7 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
XOH |
Type1 |
7 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8CDWA
|
1.941 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
UES |
Type1 |
7 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8CIJA
|
2.821 |
Inactive |
DFGout‑None |
out-out |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
USF |
Type1 |
14 - 294 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K1
|
M4K1_HUMAN
|
8PARA
|
2.0 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XON |
Type1 |
7 - 294 |
0 |
None |
T165E,S171E |
Mitogen-activated protein kinase kinase kinase kinase 1 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U3YB
|
1.45 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
8 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U3ZB
|
2.09 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
14 - 311 |
0 |
None |
T181E |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4ZP5B
|
2.29 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
10 - 309 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
5DI1B
|
2.9 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
10 - 309 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
5J95B
|
2.5 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
10 - 309 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
8V5IB
|
2.18 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
16 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4RVTB
|
2.4 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4OBOB
|
2.1 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
12 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4OBPB
|
2.27 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
14 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4OBQB
|
2.19 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U40B
|
2.3 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U41B
|
2.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
12 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U43B
|
2.18 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
10 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U44B
|
2.43 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
14 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4U45B
|
2.58 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
4ZK5B
|
2.89 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
MAP4K4
|
M4K4_HUMAN
|
5W5QB
|
2.33 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
13 - 311 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase kinase 4 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJIA
|
1.99 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4OQ |
Type3 |
254 - 542 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJIB
|
1.99 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4OQ |
Type3 |
254 - 540 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJIC
|
1.99 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
4OQ |
Type3 |
250 - 541 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJID
|
1.99 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
4OQ |
Type3 |
253 - 541 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJJA
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4OR |
Type3 |
249 - 539 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJJB
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
4OR |
Type3 |
251 - 539 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJJC
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
4OR |
Type3 |
251 - 542 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZJJD
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
4OR |
Type3 |
252 - 541 |
0 |
None |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK1
|
PAK1_HUMAN
|
4ZLOA
|
2.5 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
4PV |
Type3 |
250 - 543 |
0 |
TPO423 |
None |
Serine/threonine-protein kinase PAK 1 |
Homo sapiens |
|
STE
|
PAK2
|
PAK2_HUMAN
|
9M41A
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
No_ligand |
No_ligand |
85 - 520 |
0 |
None |
K278R,D368N |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
|
STE
|
PAK2
|
PAK2_HUMAN
|
9M41B
|
3.02 |
Inactive |
DFGout‑None |
out-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnno |
No_ligand |
No_ligand |
83 - 521 |
0 |
None |
K278R,D368N |
Serine/threonine-protein kinase PAK 2 |
Homo sapiens |
|
STE
|
SLK
|
SLK_HUMAN
|
8BEMD
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
AV9 |
Type1 |
19 - 310 |
0 |
None |
None |
STE20-like serine/threonine-protein kinase |
Homo sapiens |
|
STE
|
SLK
|
SLK_HUMAN
|
8BEMG
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
AV9 |
Type1 |
19 - 309 |
0 |
None |
None |
STE20-like serine/threonine-protein kinase |
Homo sapiens |
|
STE
|
SLK
|
SLK_HUMAN
|
8BEMA
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
AV9 |
Type1.5_Front |
19 - 309 |
0 |
None |
None |
STE20-like serine/threonine-protein kinase |
Homo sapiens |
|
STE
|
SLK
|
SLK_HUMAN
|
8BEMB
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
AV9 |
Type1.5_Front |
19 - 310 |
0 |
None |
None |
STE20-like serine/threonine-protein kinase |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
6GTTA
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
B96 |
Type2 |
18 - 316 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
6EIMA
|
1.43 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
B6E |
Type2 |
26 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
6EIMB
|
1.43 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
B6E |
Type2 |
23 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
4AOTA
|
2.33 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnno |
GW8 |
Type1 |
18 - 314 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
4AOTB
|
2.33 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnoo |
GW8 |
Type1 |
18 - 314 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
4USDA
|
3.05 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnno |
R09 |
Type1 |
24 - 314 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
4USDB
|
3.05 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiio |
APEdist_nnno |
R09 |
Type1 |
24 - 314 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
4EQUA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
G6I |
Type2 |
24 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
4EQUB
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
G6I |
Type2 |
24 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
6I2YA
|
2.56 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
88Z |
Type2 |
24 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK10
|
STK10_HUMAN
|
6I2YB
|
2.56 |
Inactive |
DFGout‑None |
out-none |
out-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoo |
88Z |
Type2 |
24 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase 10 |
Homo sapiens |
|
STE
|
STK26
|
STK26_HUMAN
|
4FZAB
|
3.15 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
18 - 297 |
0 |
None |
D162A |
Serine/threonine-protein kinase 26 |
Homo sapiens |
|
STE
|
STK26
|
STK26_HUMAN
|
4FZDB
|
3.25 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
18 - 297 |
0 |
None |
D162A |
Serine/threonine-protein kinase 26 |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4H58C
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
No_ligand |
No_ligand |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4G9RB
|
3.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B1E |
Type1 |
448 - 721 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5CSXA
|
2.51 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
54J |
Type1.5_Back |
448 - 720 |
0 |
None |
R443P,I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8C7YA
|
1.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
TXV |
Type2 |
448 - 721 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8C7YB
|
1.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
TXV |
Type2 |
449 - 721 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6V34A
|
3.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
QOP |
Type2 |
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6V34B
|
3.15 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QOP |
Type2 |
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4R5YA
|
3.5 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
3K3 |
Type2 |
449 - 720 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4R5YB
|
3.5 |
Inactive |
DFGout‑BBAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
3K3 |
Type2 |
449 - 720 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6XFPA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
V1Y |
Type2 |
449 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6XLOA
|
2.493 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
V5J |
Type2 |
449 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6XLOB
|
2.493 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
V5J |
Type2 |
450 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
7K0VA
|
1.93 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
VQP |
Type2 |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
7K0VB
|
1.93 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
VQP |
Type2 |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
7K0VC
|
1.93 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
VQP |
Type2 |
448 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
7K0VD
|
1.93 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
VQP |
Type2 |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6P3DA
|
2.11 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
0LI |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6P7GA
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
E7M |
Type2 |
449 - 720 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6P7GC
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
E7M |
Type2 |
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6P7GD
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
E7M |
Type2 |
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8F7OA
|
3.54 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
QOP |
Type2 |
449 - 723 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8F7OB
|
3.54 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
QOP |
Type2 |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8F7PA
|
2.74 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
K81 |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8F7PB
|
2.74 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
K81 |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4JVGA
|
3.09 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
B96 |
Type2 |
448 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4JVGB
|
3.09 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
B96 |
Type2 |
448 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4JVGC
|
3.09 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
B96 |
Type2 |
448 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4JVGD
|
3.09 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
B96 |
Type2 |
448 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6CADA
|
2.55 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
EU4 |
Type2 |
449 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6NSQA
|
3.05 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
KZP |
Type2 |
448 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8C7XA
|
1.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
TXV |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8C7XB
|
1.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
TXV |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4XV9A
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
1OO |
Type2 |
448 - 705 |
0 |
None |
R443S,I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5HI2A
|
2.512 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
BAX |
Type2 |
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5HIDA
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
B1E |
Type2 |
449 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5HIDB
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
B1E |
Type2 |
449 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
1UWJA
|
3.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BAX |
Type2 |
448 - 723 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
1UWJB
|
3.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BAX |
Type2 |
448 - 723 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6N0PA
|
2.37 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
K81 |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6N0PB
|
2.37 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
K81 |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8QQGB
|
2.979 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
WJ9 |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8QQGC
|
2.979 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
WJ9 |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5CT7A
|
3.17 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
55J |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5VALA
|
2.26 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
92D |
Type2 |
446 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5VALB
|
2.26 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
92D |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5VAMA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
92J |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5VAMB
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
92J |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6B8UA
|
2.68 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
8EN |
Type2 |
449 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6B8UB
|
2.68 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
8EN |
Type2 |
447 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6N0QA
|
2.04 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
K7S |
Type2 |
446 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6N0QB
|
2.04 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
K7S |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3Q96A
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
0NF |
Type2 |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3Q96B
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0NF |
Type2 |
449 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4DBNA
|
3.15 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0JA |
Type2 |
448 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4DBNB
|
3.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0JA |
Type2 |
448 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4FC0A
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0T2 |
Type2 |
448 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4FC0B
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0T2 |
Type2 |
448 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4KSPA
|
2.93 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
1SU |
Type2 |
448 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4KSPB
|
2.93 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
1SU |
Type2 |
448 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4KSQA
|
3.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1SW |
Type2 |
448 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4KSQB
|
3.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
1SW |
Type2 |
449 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3IDPA
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
L1E |
Type2 |
449 - 720 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3IDPB
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
L1E |
Type2 |
449 - 720 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4G9RA
|
3.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
B1E |
Type2 |
448 - 721 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5C9CA
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
4Z5 |
Type2 |
449 - 720 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5C9CB
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
4Z5 |
Type2 |
449 - 720 |
0 |
None |
V600E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
1UWHA
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nioo |
BAX |
Type2 |
448 - 723 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
1UWHB
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nioo |
BAX |
Type2 |
448 - 723 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3II5A
|
2.79 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
831 |
Type2 |
448 - 720 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3II5B
|
2.79 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
831 |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4G9CA
|
3.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
0WP |
Type2 |
448 - 723 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4G9CB
|
3.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
0WP |
Type2 |
448 - 723 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6P7GB
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
E7M,
NHE
|
Type2,
Allosteric
|
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4RZWA
|
3.493 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B1E |
Type1 |
448 - 720 |
0 |
None |
R509H,I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
3C4CB
|
2.57 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
324 |
Type1.5_Back |
448 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
4RZWB
|
3.493 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B1E |
Type2 |
448 - 721 |
0 |
None |
R509H,I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6CADB
|
2.55 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
EU4 |
Type2 |
449 - 721 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
6NSQB
|
3.05 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
KZP |
Type2 |
447 - 722 |
0 |
None |
I543A,I544S,I551K,Q562R,L588N,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
8QQGA
|
2.979 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
WJ9 |
Type2 |
449 - 722 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
BRAF
|
BRAF_HUMAN
|
5CT7B
|
3.17 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
55J |
Type2 |
449 - 721 |
0 |
None |
None |
Serine/threonine-protein kinase B-raf |
Homo sapiens |
|
TKL
|
IRAK4
|
IRAK4_HUMAN
|
6EG9A
|
2.414 |
Inactive |
DFGout‑None |
in-out |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
0LI |
Type2 |
164 - 459 |
0 |
None |
None |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
|
TKL
|
IRAK4
|
IRAK4_HUMAN
|
6EG9B
|
2.414 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
0LI |
Type2 |
165 - 459 |
0 |
None |
None |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
|
TKL
|
IRAK4
|
IRAK4_HUMAN
|
6EGAA
|
2.512 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnni |
J8A |
Type2 |
166 - 459 |
0 |
None |
None |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
|
TKL
|
IRAK4
|
IRAK4_HUMAN
|
6EGAB
|
2.512 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
J8A |
Type2 |
164 - 459 |
0 |
None |
None |
Interleukin-1 receptor-associated kinase 4 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7B8WA
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
T3B |
Type2 |
330 - 633 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7B8WB
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
T3B |
Type2 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7B8WC
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
T3B |
Type2 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7B8WD
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
T3B |
Type2 |
331 - 632 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7ATUA
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioo |
RXN |
Type3 |
330 - 634 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7ATUB
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioo |
RXN |
Type3 |
330 - 636 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7ATUC
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-none |
out-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
RXN |
Type3 |
350 - 632 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK1
|
LIMK1_HUMAN
|
7ATUD
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-none |
out-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
RXN |
Type3 |
354 - 632 |
0 |
None |
None |
LIM domain kinase 1 |
Homo sapiens |
|
TKL
|
LIMK2
|
LIMK2_HUMAN
|
7QHGA
|
1.45 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_oooo |
T3B |
Type2 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 2 |
Homo sapiens |
|
TKL
|
LIMK2
|
LIMK2_HUMAN
|
7QHGB
|
1.45 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaoao |
APEdist_iooo |
T3B |
Type2 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 2 |
Homo sapiens |
|
TKL
|
LIMK2
|
LIMK2_HUMAN
|
4TPTA
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iooi |
35H |
Type3 |
330 - 631 |
0 |
None |
None |
LIM domain kinase 2 |
Homo sapiens |
|
TKL
|
LIMK2
|
LIMK2_HUMAN
|
4TPTB
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiai |
APEdist_iooi |
35H |
Type3 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 2 |
Homo sapiens |
|
TKL
|
LIMK2
|
LIMK2_HUMAN
|
5NXDB
|
1.9 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
9D8 |
Type3 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 2 |
Homo sapiens |
|
TKL
|
LIMK2
|
LIMK2_HUMAN
|
5NXDA
|
1.9 |
Inactive |
DFGout‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
9D8 |
Type3 |
330 - 632 |
0 |
None |
None |
LIM domain kinase 2 |
Homo sapiens |
|
TKL
|
LRRK1
|
LRRK1_HUMAN
|
8E04A
|
3.8 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
381 - 2007 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
LRRK1
|
LRRK1_HUMAN
|
8E05A
|
4.6 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
51 - 2007 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
LRRK1
|
LRRK1_HUMAN
|
8E05B
|
4.6 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
51 - 2007 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
LRRK1
|
LRRK1_HUMAN
|
8E06A
|
4.3 |
Inactive |
DFGout‑None |
in-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
51 - 2007 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
LRRK1
|
LRRK1_HUMAN
|
8FACA
|
3.92 |
Inactive |
DFGout‑None |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
341 - 2013 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8TZBA
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
T3X |
Type2 |
1334 - 2522 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8U7LA
|
3.6 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
T3X |
Type2 |
558 - 2526 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8U7LB
|
3.6 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
T3X |
Type2 |
558 - 2526 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8U8AB
|
3.4 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0LI |
Type2 |
558 - 2526 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8U8AC
|
3.4 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
0LI |
Type2 |
558 - 2526 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8U8BA
|
3.7 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
919 |
Type2 |
558 - 2527 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8U8BB
|
3.7 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
919 |
Type2 |
558 - 2527 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8TYQA
|
2.99 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
T3X |
Type2 |
1335 - 2525 |
0 |
None |
G2019S |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8FO9E
|
3.48 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
ATP |
ATPlike |
12 - 2527 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
9DMIA
|
3.35 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
A1A7Q |
Type2 |
1334 - 2526 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8TZEA
|
2.9 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
T3X |
Type2 |
1624 - 2522 |
0 |
None |
None |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
LRRK2
|
LRRK2_HUMAN
|
8TZFA
|
3.4 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
T3X |
Type2 |
587 - 2522 |
0 |
None |
I2020T |
Leucine-rich repeat serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
5E7RA
|
2.11 |
Inactive |
DFGout‑BBAminus |
none-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
5KW |
Type1 |
31 - 496 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
2YIYA
|
2.49 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
YIY |
Type2 |
31 - 496 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
4O91A
|
2.393 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
NG2 |
Type2 |
31 - 496 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
5GJDA
|
2.79 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
6V3 |
Type2 |
31 - 495 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
5J9LA
|
2.752 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
6HF |
Type1 |
31 - 496 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
5J7SA
|
2.368 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
6H3 |
Type1 |
31 - 496 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
MAP3K7
|
M3K7_HUMAN
|
5GJFA
|
2.89 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiio |
6V4 |
Type2 |
31 - 496 |
0 |
None |
None |
Mitogen-activated protein kinase kinase kinase 7 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9Q31B
|
2.05 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
TME,
A1CNU
|
Allosteric,
Type3
|
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9MZZA
|
2.68 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1BU5 |
Type1 |
7 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6C3EB
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
EJY |
Type1 |
10 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7XMKA
|
2.376 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
GO4 |
Type1 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7XMKB
|
2.376 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
GO4 |
Type1 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7YDXB
|
2.642 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3CI |
Type1 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
8I2NA
|
2.29 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
O4U |
Type1 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
5HX6B
|
2.23 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
65U |
Type1 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
5TX5B
|
2.56 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
7MJ |
Type1 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6OCQA
|
2.793 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
M5J |
Type1 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6RLNB
|
2.87 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
K8K |
Type1 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9GTGB
|
2.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1IPG,
RCM
|
Type1,
Type3
|
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4ITJA
|
1.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1HX |
Type2 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4ITJB
|
1.8 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
1HX |
Type2 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7YDXA
|
2.642 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3CI |
Type2 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
8I2NB
|
2.29 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
O4U |
Type2 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7FD0A
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
3IU |
Type2 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7FD0B
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
3IU |
Type2 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4NEUA
|
2.57 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
Q1A |
Type2 |
6 - 313 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4NEUB
|
2.57 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
Q1A |
Type2 |
7 - 310 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9MZYA
|
2.32 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1BU6 |
Type3 |
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9MZYB
|
2.32 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
A1BU6 |
Type3 |
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9MZZB
|
2.68 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1BU5 |
Type3 |
7 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9MZXA
|
2.53 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1BU4 |
Type3 |
6 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9MZXB
|
2.53 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1BU4 |
Type3 |
6 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6C3EA
|
2.6 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
EJY |
Type3 |
9 - 293 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4ITHA
|
2.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
RCM |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4ITHB
|
2.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
RCM |
Type3 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4ITIA
|
2.86 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
1HW |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
4ITIB
|
2.86 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
1HW |
Type3 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6NYHA
|
2.1 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L8D |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6NYHB
|
2.1 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L8D |
Type3 |
11 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9Q31A
|
2.05 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1CNU |
Type3 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9Q32A
|
2.49 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1CNV |
Type3 |
6 - 293 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9Q32B
|
2.49 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1CNV |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9Q32C
|
2.49 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1CNV |
Type3 |
6 - 293 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9Q32D
|
2.49 |
Inactive |
DFGout‑BBAminus |
out-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1CNV |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7FCZA
|
2.21 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
3IF |
Type3 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
7FCZB
|
2.21 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3IF |
Type3 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9HY8A
|
2.98 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1IX7 |
Type3 |
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9HY8B
|
2.98 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1HX |
Type3 |
7 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9HY9A
|
2.29 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
A1IX9 |
Type3 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9HY9B
|
2.29 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
A1IX9 |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6C4DA
|
2.52 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
EJP |
Type3 |
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6C4DB
|
2.52 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
EJP |
Type3 |
7 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6C4DC
|
2.52 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
EJP |
Type3 |
10 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6C4DD
|
2.52 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
EJP |
Type3 |
5 - 293 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
5HX6A
|
2.23 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
65U |
Type3 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
5TX5A
|
2.56 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
7MJ |
Type3 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6HHOA
|
3.49 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
G4W |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6HHOB
|
3.49 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
G4W |
Type3 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6OCQB
|
2.793 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
M5J |
Type3 |
7 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6R5FA
|
3.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
JSW |
Type3 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6R5FB
|
3.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
JSW |
Type3 |
10 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6R5FC
|
3.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
JSW |
Type3 |
9 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6R5FD
|
3.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
JSW |
Type3 |
11 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6RLNA
|
2.87 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
K8K |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6NW2A
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
L4Y |
Type3 |
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
6NW2B
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
L4Y |
Type3 |
11 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9GTYA
|
2.145 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
RCM |
Type3 |
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9GTGA
|
2.25 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
RCM,
A1IPG
|
Type3,
Type1
|
8 - 294 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK1
|
RIPK1_HUMAN
|
9GTYB
|
2.145 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
RCM,
A1IKX
|
Type3,
Type1
|
8 - 294 |
0 |
None |
C34A,C127A,C233A,C240A |
Receptor-interacting serine/threonine-protein kinase 1 |
Homo sapiens |
|
TKL
|
RIPK2
|
RIPK2_HUMAN
|
6ES0A
|
2.38 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
BW8 |
Type2 |
5 - 316 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
RIPK2
|
RIPK2_HUMAN
|
6ES0B
|
2.38 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BW8 |
Type2 |
5 - 315 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
RIPK2
|
RIPK2_HUMAN
|
5AR7B
|
2.71 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
SR8 |
Type2 |
6 - 310 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
RIPK2
|
RIPK2_HUMAN
|
4C8BA
|
2.75 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
0LI |
Type2 |
8 - 316 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
RIPK2
|
RIPK2_HUMAN
|
4C8BB
|
2.75 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
0LI |
Type2 |
9 - 316 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
RIPK2
|
RIPK2_HUMAN
|
5AR7A
|
2.71 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
SR8 |
Type2 |
6 - 310 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 2 |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGKA
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnno |
ZGD |
Type2 |
444 - 726 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGKB
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnno |
ZGD |
Type2 |
444 - 727 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGKC
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
ZGD |
Type2 |
445 - 726 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGKD
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnoo |
ZGD |
Type2 |
444 - 727 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGJA
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnno |
ZFS |
Type2 |
445 - 726 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGJB
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnoo |
ZFS |
Type2 |
445 - 726 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGJC
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
nonTYR |
APEdihe_aanai |
APEdist_nnnn |
ZFS |
Type2 |
445 - 726 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TKL
|
TNNI3K
|
TNI3K_HUMAN
|
7MGJD
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaiai |
APEdist_nnoo |
ZFS |
Type2 |
445 - 726 |
0 |
None |
None |
Serine/threonine-protein kinase TNNI3K |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6XRGA
|
999.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oiiai |
APEdist_aaai |
No_ligand |
No_ligand |
229 - 515 |
0 |
None |
G250E,M290L,T389Y |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3QRJA
|
1.82 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
919 |
Type2 |
234 - 496 |
0 |
None |
T315I |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3QRJB
|
1.82 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
919 |
Type2 |
233 - 497 |
0 |
None |
T315I |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HZ0A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
GIN |
Type2 |
233 - 497 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HZ0B
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
GIN |
Type2 |
228 - 497 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HYYA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
235 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HYYB
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
233 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HYYC
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
233 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HYYD
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
233 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3CS9A
|
2.21 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
NIL |
Type2 |
233 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3CS9B
|
2.21 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
NIL |
Type2 |
233 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3CS9C
|
2.21 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
NIL |
Type2 |
232 - 497 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3CS9D
|
2.21 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
NIL |
Type2 |
233 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3QRIA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
919 |
Type2 |
229 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3QRIB
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
919 |
Type2 |
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HIWA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
7MP |
Type2 |
230 - 499 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HIWB
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
7MP |
Type2 |
230 - 499 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2E2BA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
406 |
Type2 |
229 - 502 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2E2BB
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
406 |
Type2 |
229 - 497 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
5HU9A
|
1.529 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oiiai |
APEdist_aaao |
66K,
66K
|
Type2,
Allosteric
|
229 - 499 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3PYYA
|
1.85 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
3YY
|
Type2,
Allosteric
|
232 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3PYYB
|
1.85 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
STI,
3YY
|
Type2,
Allosteric
|
233 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6NPEA
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
KWD
|
Type2,
Allosteric
|
232 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6NPEB
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
STI,
KWD
|
Type2,
Allosteric
|
233 - 511 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6NPUA
|
2.33 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
KWV
|
Type2,
Allosteric
|
232 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6NPUB
|
2.33 |
Inactive |
DFGout‑BBAminus |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
KWV
|
Type2,
Allosteric
|
233 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6NPVA
|
1.86 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
KWP
|
Type2,
Allosteric
|
232 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6NPVB
|
1.86 |
Inactive |
DFGout‑BBAminus |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
KWP
|
Type2,
Allosteric
|
233 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3QRKA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
9DP |
Type3 |
229 - 496 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2G2FB
|
2.7 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AGS |
ATPlike |
234 - 502 |
0 |
None |
H396P |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
6XR7A
|
999.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
TYR |
APEdihe_ooiai |
APEdist_aaai |
No_ligand |
No_ligand |
229 - 515 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
8I7TB
|
2.8 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6I5 |
Type1 |
232 - 500 |
0 |
PTR393 |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HZIA
|
1.7 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
JIN |
Type1 |
233 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
4ZOGB
|
2.3 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
VX6 |
Type1 |
234 - 503 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
4WA9B
|
2.2 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AXI |
Type1 |
246 - 508 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3UE4A
|
2.424 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DB8 |
Type1 |
233 - 502 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
3UE4B
|
2.424 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DB8 |
Type1 |
233 - 502 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
8I7TA
|
2.8 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6I5 |
Type1.5_Back |
232 - 500 |
0 |
PTR393 |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2HZIB
|
1.7 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
JIN |
Type1.5_Back |
233 - 500 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2G2HB
|
2.0 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P16 |
Type1.5_Back |
233 - 504 |
0 |
None |
H396P |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
2FO0A
|
2.27 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P16 |
Type1.5_Back |
46 - 511 |
0 |
SEP50 |
D363N |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
1OPLA
|
3.42 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P16 |
Type1.5_Back |
62 - 512 |
0 |
None |
K12R,D363N |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
1OPLB
|
3.42 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P16 |
Type1.5_Back |
121 - 499 |
0 |
None |
K12R,D363N |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL1
|
ABL1_HUMAN
|
5MO4A
|
2.17 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
NIL,
AY7
|
Type2,
Allosteric
|
64 - 512 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Homo sapiens |
|
TYR
|
ABL2
|
ABL2_HUMAN
|
3GVUA
|
2.05 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
STI,
STI
|
Type2,
Allosteric
|
279 - 546 |
0 |
None |
None |
Tyrosine-protein kinase ABL2 |
Homo sapiens |
|
TYR
|
ALK
|
ALK_HUMAN
|
5IUGA
|
1.93 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_oiiai |
APEdist_aaao |
729 |
Type2 |
1093 - 1404 |
0 |
None |
C1097S |
ALK tyrosine kinase receptor |
Homo sapiens |
|
TYR
|
ALK
|
ALK_HUMAN
|
5IUHA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_oiiai |
APEdist_aaao |
34Y |
Type2 |
1093 - 1404 |
0 |
None |
C1097S |
ALK tyrosine kinase receptor |
Homo sapiens |
|
TYR
|
ALK
|
ALK_HUMAN
|
4FNYA
|
2.45 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_oiiai |
APEdist_aaao |
I3K |
Type2 |
1103 - 1404 |
0 |
None |
C1097S,R1275Q |
ALK tyrosine kinase receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
8CGCA
|
1.925 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
LMR,
UIK
|
Allosteric,
Type1
|
547 - 919 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
3BEAA
|
2.02 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
IXH |
Type1 |
547 - 921 |
0 |
None |
A933L |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
2I1MA
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5CN |
Type1 |
547 - 921 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
8JOTA
|
1.69 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
UKI |
Type1 |
543 - 914 |
0 |
None |
C667T,C830S,C907T |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
8W1LA
|
2.26 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A1AE3 |
Type1 |
563 - 914 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
2I0VA
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6C3 |
Type1 |
544 - 916 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
2I0YA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5CN |
Type1 |
548 - 916 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
3KRJA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
KRJ |
Type1 |
544 - 914 |
0 |
None |
S686S |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
3KRLA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
KRL |
Type1 |
545 - 912 |
0 |
None |
S686S |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
7TNHA
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
I9W |
Type1 |
445 - 912 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
6T2WA
|
1.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
M9T |
Type1 |
547 - 916 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
3DPKA
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
8C5 |
Type1.5_Back |
548 - 912 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
4HW7A
|
2.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
64M |
Type2 |
566 - 914 |
0 |
None |
C667T,C830S,C907T |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
4R7HA
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P31 |
Type2 |
544 - 915 |
0 |
None |
C667T,C830S,C907T |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
4R7IA
|
2.75 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
567 - 914 |
0 |
None |
C667T,C830S,C907T |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
6N33A
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
622 |
Type2 |
566 - 915 |
0 |
None |
C667T,C830S,C907T |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
7MFCA
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
Z6V |
Type2 |
567 - 913 |
0 |
None |
C667T,C830S,C907T |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
6WXJA
|
2.62 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
UF4 |
Type2 |
559 - 917 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
3LCOA
|
3.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
LC0 |
Type2 |
551 - 915 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
6IG8A
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A7O |
Type2 |
550 - 916 |
0 |
None |
S688A |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
CSF1R
|
CSF1R_HUMAN
|
2OGVA
|
2.7 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
543 - 918 |
0 |
None |
None |
Macrophage colony-stimulating factor 1 receptor |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAUA
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IF |
Type2 |
604 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAVA
|
1.76 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IJ |
Type2 |
602 - 909 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAWA
|
1.601 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IM |
Type2 |
603 - 907 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAXA
|
1.902 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IM |
Type2 |
601 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAYA
|
2.19 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IJ |
Type2 |
602 - 907 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAYB
|
2.19 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IJ |
Type2 |
602 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SAZA
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IW |
Type2 |
603 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SB0A
|
1.97 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1IZ |
Type2 |
604 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SB1A
|
1.53 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1JI |
Type2 |
604 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6FEWA
|
1.44 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6W |
Type2 |
603 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6FEXA
|
1.291 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Z |
Type2 |
602 - 908 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6FILA
|
1.73 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6W |
Type2 |
604 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6FINA
|
1.67 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DJQ |
Type2 |
603 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6FIOA
|
1.99 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DJH |
Type2 |
598 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6FIQA
|
1.79 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oiiai |
APEdist_aaai |
DJW |
Type2 |
601 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
3ZOSB
|
1.92 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI |
Type2 |
601 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
4BKJA
|
1.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
601 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
4BKJB
|
1.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
601 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
4CKRA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
DI1 |
Type2 |
601 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6GWRA
|
2.07 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FEW |
Type2 |
601 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6GWRB
|
2.07 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FEW |
Type2 |
602 - 908 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6HP9A
|
1.96 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
GKB |
Type2 |
601 - 909 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
6HP9B
|
1.96 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
GKB |
Type2 |
603 - 909 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
7BCMA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
TBK |
Type2 |
604 - 909 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
7BCMB
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
TBK |
Type2 |
604 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
7BE6A
|
1.871 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
TJW |
Type2 |
601 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5BVNA
|
2.21 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
4VD |
Type2 |
604 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5BVOA
|
1.98 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
4VE |
Type2 |
604 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5FDPA
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5WR |
Type2 |
604 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5FDXA
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5X1 |
Type2 |
604 - 909 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5FDXB
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5X1 |
Type2 |
605 - 907 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
3ZOSA
|
1.92 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI,
0LI
|
Type2,
Allosteric
|
602 - 913 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
7FEHA
|
1.61 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
3UI |
Type3 |
603 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5BVWA
|
1.94 |
Inactive |
DFGout‑None |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1N1 |
Type1 |
604 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5SB2A
|
1.6 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
1K2 |
Type2 |
603 - 912 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR1
|
DDR1_HUMAN
|
5BVKA
|
2.29 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
4VC |
Type3 |
604 - 911 |
0 |
None |
None |
Epithelial discoidin domain-containing receptor 1 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERD
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type1 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERI
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type1 |
555 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERA
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERB
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERC
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERE
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERF
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERG
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERH
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERJ
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
553 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERK
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
555 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
6FERL
|
2.87 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
D6Q |
Type2 |
554 - 851 |
0 |
None |
None |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
DDR2
|
DDR2_HUMAN
|
7AYMA
|
2.12 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
4VD |
Type2 |
558 - 849 |
0 |
None |
K826E,L847R |
Discoidin domain-containing receptor 2 |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
2RF9A
|
3.5 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
TYR |
APEdihe_ooiai |
APEdist_aaai |
No_ligand |
No_ligand |
699 - 983 |
0 |
None |
None |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
4ZJVA
|
2.7 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
703 - 985 |
0 |
None |
None |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
4ZJVB
|
2.7 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
703 - 982 |
0 |
None |
None |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5HG5A
|
1.52 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
633 |
Type1 |
700 - 1001 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5HG7A
|
1.85 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
630 |
Type1 |
702 - 984 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5HG8A
|
1.42 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
634 |
Type1 |
700 - 999 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5HG9A
|
2.15 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
63A |
Type1 |
702 - 985 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5U8LA
|
1.6 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O44 |
Type1 |
702 - 990 |
0 |
None |
None |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5UG8A
|
1.46 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
8BP |
Type1 |
702 - 985 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5UG9A
|
1.33 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
8AM |
Type1 |
702 - 985 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5UGAA
|
1.82 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
8BM |
Type1 |
703 - 985 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
5UGCA
|
1.58 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
8BS |
Type1 |
702 - 985 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
4I1ZA
|
3.0 |
Inactive |
DFGout‑None |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
701 - 987 |
0 |
None |
T790M,L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
4I21A
|
3.37 |
Inactive |
DFGout‑None |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
703 - 1019 |
0 |
None |
T790M,L858R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
4I21B
|
3.37 |
Inactive |
DFGout‑None |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
703 - 1020 |
0 |
None |
T790M,L858R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
2RF9B
|
3.5 |
Inactive |
DFGout‑None |
out-none |
in-out |
TYR |
APEdihe_ioiai |
APEdist_aaao |
No_ligand |
No_ligand |
701 - 985 |
0 |
None |
None |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EGFR
|
EGFR_HUMAN
|
4I20A
|
3.34 |
Inactive |
DFGout‑None |
out-out |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
701 - 987 |
0 |
None |
L858R,V948R |
Epidermal growth factor receptor |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8XPVA
|
1.55 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
4Z5 |
Type2 |
604 - 895 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6FNFA
|
1.556 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
DXH |
Type2 |
606 - 894 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6FNGA
|
1.038 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
DWT |
Type2 |
599 - 897 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HESA
|
1.128 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
G0H |
Type2 |
599 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HETA
|
1.208 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
G0Q |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HEUA
|
1.719 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
G0N |
Type2 |
600 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HEVA
|
1.28 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
G0K |
Type2 |
600 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HEWA
|
1.268 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
G0E |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HEXA
|
1.413 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
G02 |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6HEYA
|
1.367 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_niiai |
APEdist_aaao |
FZW |
Type2 |
600 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6Q7BA
|
1.009 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
HO5 |
Type2 |
599 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6Q7CA
|
1.049 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
HOK |
Type2 |
599 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6Q7DA
|
0.978 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
HOT |
Type2 |
600 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6Q7EA
|
1.059 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
HMW |
Type2 |
601 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6Q7GA
|
1.047 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
HO8 |
Type2 |
601 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BM8A
|
1.68 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
QT1 |
Type2 |
605 - 895 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOCA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
QUF |
Type2 |
605 - 888 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BODA
|
1.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
QTX |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOGA
|
1.47 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
QUU |
Type2 |
600 - 895 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOHA
|
1.42 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
R0T |
Type2 |
604 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOIA
|
1.63 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
R0O |
Type2 |
604 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOKA
|
2.02 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
R0X |
Type2 |
605 - 890 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOMA
|
1.12 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
QU6 |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
5IA4A
|
1.797 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
88Z |
Type2 |
605 - 877 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
5IA5A
|
1.776 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
GV0 |
Type2 |
605 - 880 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
6Q7FA
|
1.204 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
HNZ |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA2
|
EPHA2_HUMAN
|
8BOFA
|
1.82 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
R3L |
Type2 |
605 - 896 |
0 |
None |
None |
Ephrin type-A receptor 2 |
Homo sapiens |
|
TYR
|
EPHA3
|
EPHA3_HUMAN
|
3DZQA
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
IFC |
Type2 |
609 - 904 |
0 |
None |
None |
Ephrin type-A receptor 3 |
Homo sapiens |
|
TYR
|
EPHA3
|
EPHA3_HUMAN
|
4P5ZA
|
2.002 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
Q7M |
Type2 |
609 - 903 |
0 |
None |
None |
Ephrin type-A receptor 3 |
Homo sapiens |
|
TYR
|
EPHA3
|
EPHA3_HUMAN
|
4TWNA
|
1.706 |
Inactive |
DFGout‑None |
in-in |
out-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
B96 |
Type2 |
609 - 904 |
0 |
None |
None |
Ephrin type-A receptor 3 |
Homo sapiens |
|
TYR
|
EPHA7
|
EPHA7_HUMAN
|
3DKOA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
IHZ |
Type2 |
607 - 899 |
0 |
None |
None |
Ephrin type-A receptor 7 |
Homo sapiens |
|
TYR
|
EPHB4
|
EPHB4_HUMAN
|
6FNIA
|
1.468 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
DXH |
Type2 |
607 - 889 |
0 |
None |
Y774E,A803V,V870I |
Ephrin type-B receptor 4 |
Homo sapiens |
|
TYR
|
EPHB4
|
EPHB4_HUMAN
|
6FNJA
|
1.239 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
DWT |
Type2 |
607 - 888 |
0 |
None |
Y774E,A803V,V870I |
Ephrin type-B receptor 4 |
Homo sapiens |
|
TYR
|
EPHB4
|
EPHB4_HUMAN
|
6FNJB
|
1.239 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
DWT |
Type2 |
607 - 888 |
0 |
None |
Y774E,A803V,V870I |
Ephrin type-B receptor 4 |
Homo sapiens |
|
TYR
|
ERBB2
|
ERBB2_HUMAN
|
8U8XA
|
1.69 |
Inactive |
DFGout‑None |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
W9N |
Type1 |
712 - 1024 |
0 |
None |
None |
Receptor tyrosine-protein kinase erbB-2 |
Homo sapiens |
|
TYR
|
FGFR1
|
FGFR1_HUMAN
|
4V04B
|
2.12 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
0LI |
Type2 |
458 - 765 |
0 |
None |
C488A,C584S |
Fibroblast growth factor receptor 1 |
Homo sapiens |
|
TYR
|
FGFR1
|
FGFR1_HUMAN
|
4V01A
|
2.33 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
0LI |
Type2 |
465 - 765 |
0 |
None |
C488A,C584S |
Fibroblast growth factor receptor 1 |
Homo sapiens |
|
TYR
|
FGFR1
|
FGFR1_HUMAN
|
4V01B
|
2.33 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
0LI |
Type2 |
461 - 763 |
0 |
None |
C488A,C584S |
Fibroblast growth factor receptor 1 |
Homo sapiens |
|
TYR
|
FGFR1
|
FGFR1_HUMAN
|
4V04A
|
2.12 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
0LI |
Type2 |
463 - 765 |
0 |
None |
C488A,C584S |
Fibroblast growth factor receptor 1 |
Homo sapiens |
|
TYR
|
FGFR4
|
FGFR4_HUMAN
|
4QQ5A
|
2.203 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
37O |
Type1.5_Back |
445 - 750 |
0 |
None |
V550L,R664E |
Fibroblast growth factor receptor 4 |
Homo sapiens |
|
TYR
|
FGFR4
|
FGFR4_HUMAN
|
4R6VA
|
2.353 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
FI3 |
Type1.5_Back |
445 - 750 |
0 |
None |
V550L,R664E |
Fibroblast growth factor receptor 4 |
Homo sapiens |
|
TYR
|
FGFR4
|
FGFR4_HUMAN
|
4UXQA
|
1.85 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
0LI |
Type2 |
452 - 750 |
0 |
None |
C477A |
Fibroblast growth factor receptor 4 |
Homo sapiens |
|
TYR
|
FGFR4
|
FGFR4_HUMAN
|
4TYJA
|
2.45 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
0LI |
Type2 |
447 - 753 |
0 |
None |
None |
Fibroblast growth factor receptor 4 |
Homo sapiens |
|
TYR
|
FGFR4
|
FGFR4_HUMAN
|
4QRCA
|
1.901 |
Inactive |
DFGout‑None |
in-in |
out-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
0LI |
Type2 |
454 - 750 |
0 |
None |
C477A,R664E |
Fibroblast growth factor receptor 4 |
Homo sapiens |
|
TYR
|
FGR
|
FGR_HUMAN
|
7UY3A
|
2.99 |
Inactive |
DFGout‑None |
in-in |
out-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
OJL |
Type2 |
135 - 527 |
0 |
PTR523 |
Q524E,P525E,G526I,D527P |
Tyrosine-protein kinase Fgr |
Homo sapiens |
|
TYR
|
FLT1
|
VGFR1_HUMAN
|
3HNGA
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
8ST |
Type2 |
803 - 1158 |
0 |
None |
None |
Vascular endothelial growth factor receptor 1 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
4XUFA
|
3.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P30 |
Type2 |
600 - 947 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
4XUFB
|
3.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P30 |
Type2 |
600 - 946 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
4RT7A
|
3.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P30 |
Type2 |
599 - 950 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
1RJBA
|
2.1 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
572 - 947 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
6JQRA
|
2.2 |
Inactive |
DFGout‑None |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
C6F |
Type1 |
571 - 951 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
8XB1A
|
2.85 |
Inactive |
DFGout‑None |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
ZX3 |
Type1 |
573 - 950 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
5X02A
|
2.401 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F6M |
Type1 |
573 - 947 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
FLT3
|
FLT3_HUMAN
|
6IL3A
|
2.5 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A9R |
Type1 |
569 - 947 |
0 |
None |
None |
Receptor-type tyrosine-protein kinase FLT3 |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
3LW0A
|
1.79 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
CCX,
CCX
|
Type3,
Allosteric
|
983 - 1286 |
0 |
None |
E1097A,E1099A |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
3LW0B
|
1.79 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
CCX,
CCX
|
Type3,
Allosteric
|
983 - 1286 |
0 |
None |
E1097A,E1099A |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
3LW0C
|
1.79 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
CCX,
CCX
|
Type3,
Allosteric
|
983 - 1286 |
0 |
None |
E1097A,E1099A |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
3O23A
|
2.1 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
MQY |
Type2 |
991 - 1283 |
0 |
None |
Y987F |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
8PYJAAA
|
2.702 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
IEA |
Type2 |
986 - 1270 |
0 |
None |
None |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
8PYKAAA
|
2.23 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
IC2 |
Type2 |
986 - 1270 |
0 |
None |
None |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
8PYLAAA
|
2.93 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
IE0 |
Type2 |
986 - 1270 |
0 |
None |
None |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
8PYMAAA
|
2.652 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
IED |
Type2 |
984 - 1270 |
0 |
None |
None |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
8PYNAAA
|
1.71 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
ICV |
Type2 |
986 - 1270 |
0 |
None |
None |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
IGF1R
|
IGF1R_HUMAN
|
3LW0D
|
1.79 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
CCX,
CCX
|
Type3,
Allosteric
|
983 - 1286 |
0 |
None |
E1097A,E1099A |
Insulin-like growth factor 1 receptor |
Homo sapiens |
|
TYR
|
INSR
|
INSR_HUMAN
|
1IRKA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
1008 - 1310 |
0 |
None |
None |
Insulin receptor |
Homo sapiens |
|
TYR
|
INSR
|
INSR_HUMAN
|
3ETAA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
351 |
Type2 |
1017 - 1310 |
0 |
None |
None |
Insulin receptor |
Homo sapiens |
|
TYR
|
INSR
|
INSR_HUMAN
|
3ETAB
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
351 |
Type2 |
1017 - 1310 |
0 |
None |
None |
Insulin receptor |
Homo sapiens |
|
TYR
|
JAK2-2
|
JAK2_HUMAN
|
7RN6A
|
1.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nioai |
APEdist_aaao |
046 |
Type2 |
839 - 1130 |
0 |
PTR1007 |
None |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
|
TYR
|
JAK2-2
|
JAK2_HUMAN
|
3UGCA
|
1.34 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oioai |
APEdist_aaao |
046 |
Type2 |
843 - 1129 |
0 |
None |
Y1007F,Y1008F |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
|
TYR
|
JAK2-2
|
JAK2_HUMAN
|
7TEUA
|
1.45 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oioai |
APEdist_aaao |
I6C |
Type2 |
843 - 1131 |
0 |
None |
Y1007F,Y1008F |
Tyrosine-protein kinase JAK2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
4AG8A
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AXI |
Type1 |
816 - 1168 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
4AGDA
|
2.81 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B49 |
Type1 |
802 - 1169 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3CPBB
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
C92 |
Type1 |
820 - 1165 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2XIRA
|
1.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
00J |
Type1.5_Back |
816 - 1168 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
4AGCA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AXI |
Type1.5_Back |
801 - 1169 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3WZEA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
BAX |
Type2 |
815 - 1167 |
0 |
None |
T940V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2OH4A
|
2.05 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
GIG |
Type2 |
816 - 1171 |
0 |
PTR1054,PTR1059 |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2P2IA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
608 |
Type2 |
817 - 1172 |
0 |
PTR1054,PTR1059 |
C817A,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3EFLA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
706 |
Type2 |
817 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3EFLB
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
706 |
Type2 |
821 - 1165 |
0 |
PTR1054,PTR1059 |
C817A,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
5EW3A
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
5T2 |
Type2 |
821 - 1168 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
5EW3B
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
5T2 |
Type2 |
820 - 1165 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
6GQOA
|
1.87 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F82 |
Type2 |
811 - 1168 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
6GQPA
|
2.09 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
F88 |
Type2 |
821 - 1168 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
6GQQA
|
1.52 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
F8B |
Type2 |
813 - 1167 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
6XVJA
|
1.78 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O35 |
Type2 |
813 - 1167 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
6XVKA
|
1.99 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O3E |
Type2 |
821 - 1168 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
4ASDA
|
2.03 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
BAX |
Type2 |
807 - 1168 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
4ASEA
|
1.83 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AV9 |
Type2 |
807 - 1169 |
0 |
None |
E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3VHEA
|
1.55 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
42Q |
Type2 |
811 - 1169 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3VHKA
|
2.49 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
BPK |
Type2 |
814 - 1168 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2QU5A
|
2.95 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_oooai |
APEdist_aaao |
276 |
Type2 |
816 - 1170 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2QU6A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
857 |
Type2 |
817 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2RL5A
|
2.65 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_oooai |
APEdist_aaao |
2RL |
Type2 |
815 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3B8QB
|
2.75 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
900 |
Type2 |
820 - 1166 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3BE2A
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
RAJ |
Type2 |
815 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3CP9A
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
C19 |
Type2 |
817 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3CP9B
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
C19 |
Type2 |
819 - 1165 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3CPCB
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
C52 |
Type2 |
820 - 1165 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3DTWB
|
2.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nooai |
APEdist_aaao |
A96 |
Type2 |
820 - 1166 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3EWHA
|
1.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
K11 |
Type2 |
815 - 1171 |
0 |
None |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3U6JA
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
03X |
Type2 |
815 - 1171 |
0 |
None |
V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3C7QA
|
2.1 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
XIN |
Type1 |
819 - 1171 |
0 |
PTR1054,PTR1059 |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2P2IB
|
2.4 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
608 |
Type1 |
820 - 1168 |
0 |
PTR1054,PTR1059 |
C817A,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3VNTA
|
1.64 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0JA |
Type2 |
812 - 1168 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3VO3A
|
1.52 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0KF |
Type2 |
812 - 1168 |
0 |
None |
None |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
2QU6B
|
2.1 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
857 |
Type2 |
822 - 1165 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3B8QA
|
2.75 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
900 |
Type2 |
818 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3CPBA
|
2.7 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
C92 |
Type2 |
819 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3CPCA
|
2.4 |
Inactive |
DFGout‑None |
in-out |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
C52 |
Type2 |
820 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KDR
|
VGFR2_HUMAN
|
3DTWA
|
2.9 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
A96 |
Type2 |
818 - 1171 |
0 |
PTR1054,PTR1059 |
C817A,V916T,E990V |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S13A
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
554 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S14A
|
1.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B49 |
Type1 |
554 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S15A
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
XIN |
Type1 |
554 - 929 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
3G0FA
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B49 |
Type1 |
566 - 930 |
0 |
None |
D816H |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
3G0FB
|
2.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B49 |
Type1 |
564 - 930 |
0 |
None |
D816H |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
7ZW8A
|
2.119 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
K3R |
Type1 |
554 - 932 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6KLAA
|
2.109 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DJX |
Type1 |
554 - 931 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
4HVSA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
647 |
Type2 |
551 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,I690H,C691S,K693D,Q694T,E695S,I756S,L762N,V825D,C844S,L890S,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
7KHGA
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P31 |
Type2 |
547 - 931 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S16A
|
1.85 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
566 - 932 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S16B
|
1.85 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
578 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S17A
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI |
Type2 |
567 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S17B
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI |
Type2 |
578 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S18A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A1H4U |
Type2 |
568 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S18B
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A1H4U |
Type2 |
578 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQJA
|
2.33 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F82 |
Type2 |
567 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQJB
|
2.33 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F82 |
Type2 |
572 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQKA
|
2.31 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
F88 |
Type2 |
567 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQKB
|
2.31 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
F88 |
Type2 |
572 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQLA
|
2.01 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F8B |
Type2 |
568 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQLB
|
2.01 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
F8B |
Type2 |
577 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQMA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F8H |
Type2 |
569 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6GQMB
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
F8H |
Type2 |
577 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6XV9A
|
3.38 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O35 |
Type2 |
566 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6XV9B
|
3.38 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O35 |
Type2 |
572 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6XVAA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O2K |
Type2 |
569 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6XVAB
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O2K |
Type2 |
577 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6XVBA
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O2H |
Type2 |
569 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6XVBB
|
2.15 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
O2H |
Type2 |
577 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6HH1A
|
2.25 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_iiiai |
APEdist_aaan |
G4E |
Type2 |
565 - 929 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6MOBA
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
JWY |
Type2 |
567 - 930 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
1T46A
|
1.6 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
565 - 933 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
4U0IA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI |
Type2 |
565 - 933 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
7ZY6A
|
3.09 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
KCI |
Type2 |
557 - 932 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6ITTA
|
2.103 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AWO |
Type2 |
563 - 932 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6ITTB
|
2.103 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AWO |
Type2 |
566 - 932 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
6ITVA
|
1.881 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AWO |
Type2 |
569 - 935 |
0 |
PTR570 |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S1BB
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
K3R,
K3R,
K3R
|
Type2,
Allosteric,
Allosteric
|
565 - 930 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
1T45A
|
1.9 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
547 - 935 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
3G0EA
|
1.6 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B49 |
Type1 |
544 - 931 |
0 |
None |
None |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
KIT
|
KIT_HUMAN
|
8S1BA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
K3R |
Type2 |
565 - 931 |
0 |
None |
I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D |
Mast/stem cell growth factor receptor Kit |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
6PDJA
|
1.81 |
Inactive |
DFGout‑BBAminus |
out-none |
in-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
ODJ |
Type1.5_Front |
225 - 500 |
0 |
PTR394 |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
2OG8A
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
1N8 |
Type2 |
237 - 499 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
2OG8B
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
1N8 |
Type2 |
237 - 499 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
3BYSA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnnao |
APEdist_aaan |
AM5 |
Type2 |
230 - 501 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
3BYUA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nioao |
APEdist_aaai |
AM6 |
Type2 |
231 - 501 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
2PL0A
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
231 - 498 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
2OFVA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnan |
APEdist_aaan |
242 |
Type2 |
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LCK
|
LCK_HUMAN
|
2OFVB
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
242 |
Type2 |
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase Lck |
Homo sapiens |
|
TYR
|
LMTK3
|
LMTK3_HUMAN
|
6SEQA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
130 - 413 |
0 |
None |
None |
Serine/threonine-protein kinase LMTK3 |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
9KS9B
|
2.8 |
Inactive |
DFGout‑BBAminus |
out-none |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1L6L |
Type1 |
577 - 863 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7XHYA
|
2.16 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
E0X |
Type1 |
571 - 862 |
0 |
None |
K591R,K693R,K702R,K856R |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7AAYA
|
1.87 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nnoai |
APEdist_aaao |
L1X |
Type2 |
571 - 862 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
9KRYB
|
2.25 |
Inactive |
DFGout‑BBAminus |
out-none |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1L6J |
Type2 |
580 - 863 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7AW4A
|
1.98 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
S5E |
Type3 |
576 - 862 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7AW4B
|
1.98 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
S5E |
Type3 |
574 - 862 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7AVXB
|
2.44 |
Inactive |
DFGout‑None |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
S4K |
Type1 |
577 - 862 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
9KRZA
|
2.6 |
Inactive |
DFGout‑None |
out-none |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1L6K |
Type1.5_Front |
577 - 864 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
9KRZB
|
2.6 |
Inactive |
DFGout‑None |
out-none |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1L6K |
Type1.5_Front |
575 - 863 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
9KRYA
|
2.25 |
Inactive |
DFGout‑None |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1L6J |
Type2 |
580 - 863 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
9KS9A
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1L6L |
Type2 |
576 - 862 |
0 |
None |
None |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7AAXA
|
1.762 |
Inactive |
DFGout‑None |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
R6H |
Type2 |
571 - 862 |
0 |
None |
K591R,K693R,K702R,K856R |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MERTK
|
MERTK_HUMAN
|
7AW1A
|
1.98 |
Inactive |
DFGout‑None |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
S4T |
Type2 |
571 - 862 |
0 |
None |
K591R,K693R,K702R,K856R |
Tyrosine-protein kinase Mer |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3RHKB
|
1.94 |
Inactive |
DFGout‑BBAminus |
out-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
M97 |
Type1 |
1046 - 1344 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8ANSA
|
2.01 |
Inactive |
DFGout‑BBAminus |
out-none |
in-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
MDI |
Type1.5_Front |
1052 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8VI1A
|
3.11 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
A1AB1 |
Type1.5_Front |
1053 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8VI1B
|
3.11 |
Inactive |
DFGout‑BBAminus |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A1AB1 |
Type1.5_Front |
1050 - 1345 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8AN8A
|
2.394 |
Inactive |
DFGout‑BBAminus |
out-out |
in-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
MDI |
Type1.5_Front |
1073 - 1345 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8AN8B
|
2.394 |
Inactive |
DFGout‑BBAminus |
out-out |
in-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
MDI |
Type1.5_Front |
1058 - 1345 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
6SDCA
|
1.67 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
88Z |
Type2 |
1052 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
6SDDA
|
1.93 |
Inactive |
DFGout‑BBAminus |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
353 |
Type2 |
1062 - 1344 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
9C1RA
|
1.59 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
A1ATS |
Type2 |
1048 - 1348 |
0 |
None |
D1228N |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3LQ8A
|
2.02 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
88Z |
Type2 |
1053 - 1345 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
6SD9A
|
2.35 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
88Z |
Type2 |
1062 - 1345 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
4EEVA
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
L1X |
Type2 |
1045 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
4MXCA
|
1.632 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DWF |
Type2 |
1052 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
5HTIA
|
1.66 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
66L |
Type2 |
1052 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
7V3SA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5I9 |
Type2 |
1053 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3VW8A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DF6 |
Type2 |
1024 - 1352 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3CE3A
|
2.4 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
TYR |
APEdihe_oiiai |
APEdist_aaai |
1FN |
Type2 |
1054 - 1360 |
0 |
None |
Y1194F,Y1234F,Y1235D,L1272L |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3CTHA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
TYR |
APEdihe_oiiai |
APEdist_aaai |
319 |
Type2 |
1052 - 1360 |
0 |
None |
Y1194F,Y1234F,Y1235D |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3F82A
|
2.5 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
353 |
Type2 |
1055 - 1360 |
0 |
None |
Y1194F,Y1234F,Y1235D |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3L8VA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
TYR |
APEdihe_oiiai |
APEdist_aaai |
L8V |
Type2 |
1054 - 1360 |
0 |
None |
Y1194F,Y1234F,Y1235D |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OUUA
|
1.77 |
Inactive |
DFGout‑BBAminus |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
W49 |
Type3 |
1059 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OUUB
|
1.77 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
W49 |
Type3 |
1057 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OUVA
|
1.783 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
W3R |
Type3 |
1053 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OUVB
|
1.783 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
W3R |
Type3 |
1057 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OV7A
|
1.95 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iioai |
APEdist_aaao |
W3W |
Type3 |
1051 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OVZA
|
2.206 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
W3N |
Type3 |
1061 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OVZB
|
2.206 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
W3N |
Type3 |
1057 - 1346 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OWGA
|
2.631 |
Inactive |
DFGout‑BBAminus |
out-none |
out-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
W40 |
Type3 |
1060 - 1344 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OWGB
|
2.631 |
Inactive |
DFGout‑BBAminus |
out-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
W40 |
Type3 |
1060 - 1343 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OWGC
|
2.631 |
Inactive |
DFGout‑BBAminus |
out-none |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
W40 |
Type3 |
1060 - 1343 |
0 |
None |
D1228V |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
8OW3A
|
2.27 |
Inactive |
DFGout‑BBAminus |
out-none |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
W40 |
Type3 |
1058 - 1345 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3RHKA
|
1.94 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
M97 |
Type1 |
1049 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3EFJA
|
2.6 |
Inactive |
DFGout‑None |
out-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
MT3 |
Type1.5_Front |
1054 - 1351 |
0 |
None |
L1272L |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
5DG5A
|
2.6 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5B4 |
Type2 |
1050 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
5DG5B
|
2.6 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
5B4 |
Type2 |
1050 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
7V3RA
|
1.7 |
Inactive |
DFGout‑None |
in-out |
out-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
5IE |
Type2 |
1053 - 1346 |
0 |
None |
None |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3CTJA
|
2.5 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
320 |
Type2 |
1051 - 1360 |
0 |
None |
Y1194F,Y1234F,Y1235D |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
MET
|
MET_HUMAN
|
3C1XA
|
2.17 |
Inactive |
DFGout‑None |
in-out |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
CKK |
Type2 |
1050 - 1360 |
0 |
None |
Y1194F,Y1234F,Y1235D,L1272L |
Hepatocyte growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6DKGA
|
2.53 |
Inactive |
DFGout‑BBAminus |
in-out |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
22L,
GO7
|
Allosteric,
Type2
|
500 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6DKIA
|
2.11 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
22L,
GOD
|
Allosteric,
Type2
|
500 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6D1ZA
|
1.87 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FQD,
FQM
|
Allosteric,
Type3
|
483 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
7VKMA
|
2.55 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
502 - 795 |
0 |
None |
G595R |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
4PMPA
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
31W |
Type1 |
501 - 787 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5H3QA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
7HF |
Type1 |
484 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
4PMMA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
31V |
Type2 |
501 - 787 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5JFSA
|
2.07 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
6K0 |
Type2 |
502 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5JFVA
|
1.59 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
6K1 |
Type2 |
502 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5JFWA
|
1.52 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
6K2 |
Type2 |
502 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5JFXA
|
1.63 |
Inactive |
DFGout‑BBAminus |
out-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
6K4 |
Type2 |
502 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6DKWA
|
2.91 |
Inactive |
DFGout‑BBAminus |
out-out |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
GXA |
Type2 |
502 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6DKWB
|
2.91 |
Inactive |
DFGout‑BBAminus |
in-out |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
GXA |
Type2 |
502 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PL2A
|
2.59 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OOM |
Type2 |
499 - 795 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
7XBIA
|
2.16 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
CVY |
Type2 |
497 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
8J5XA
|
2.092 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A4U |
Type2 |
500 - 795 |
0 |
None |
G595R |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PL4A
|
2.06 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OO7 |
Type3 |
485 - 795 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6D20A
|
1.94 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FQD,
FQG
|
Allosteric,
Type3
|
482 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
4F0IA
|
2.302 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
501 - 790 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
4F0IB
|
2.302 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
501 - 794 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
4GT5A
|
2.398 |
Inactive |
DFGout‑None |
in-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
498 - 793 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6D22A
|
2.46 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
502 - 794 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6DKBA
|
2.68 |
Inactive |
DFGout‑None |
out-in |
none-none |
TYR |
APEdihe_niiai |
APEdist_aaai |
FKY |
Type1 |
501 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMOA
|
2.67 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UM |
Type1 |
500 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
4PMSA
|
2.8 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
31X |
Type1.5_Back |
501 - 787 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
8J5WA
|
2.28 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A4U |
Type2 |
485 - 795 |
0 |
None |
F589L |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
8J61A
|
3.051 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A0X |
Type2 |
499 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
8J63A
|
3.001 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A6X |
Type2 |
500 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5WR7A
|
2.76 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
RCH |
Type2 |
489 - 792 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PL1A
|
2.03 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OOJ |
Type2 |
500 - 795 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PL3A
|
3.0 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OOD |
Type2 |
500 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PMAA
|
2.53 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OQS |
Type2 |
500 - 795 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PMBA
|
2.81 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OQM |
Type2 |
500 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6PMCA
|
2.19 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
OQJ |
Type2 |
500 - 795 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6NSPA
|
2.31 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
L0P |
Type3 |
500 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6NPTA
|
2.19 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
KWY |
Type3 |
491 - 795 |
0 |
SEP677 |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6NSSA
|
1.97 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
L0M |
Type3 |
485 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
6D1YA
|
1.93 |
Inactive |
DFGout‑None |
out-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FQJ |
Type3 |
481 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMIA
|
1.87 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UE |
Type3 |
486 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMJA
|
2.04 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UF |
Type3 |
486 - 795 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMKA
|
2.24 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UG |
Type3 |
484 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMMA
|
2.12 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UJ |
Type3 |
484 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMLA
|
2.01 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UH |
Type3 |
474 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK1
|
NTRK1_HUMAN
|
5KMNA
|
2.14 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
6UK |
Type3 |
474 - 796 |
0 |
None |
None |
High affinity nerve growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK2
|
NTRK2_HUMAN
|
4AT4A
|
2.36 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
T6E |
Type2 |
527 - 822 |
0 |
None |
None |
BDNF/NT-3 growth factors receptor |
Homo sapiens |
|
TYR
|
NTRK2
|
NTRK2_HUMAN
|
4ASZA
|
1.7 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
527 - 822 |
0 |
None |
None |
BDNF/NT-3 growth factors receptor |
Homo sapiens |
|
TYR
|
NTRK2
|
NTRK2_HUMAN
|
4AT5A
|
1.71 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
MUJ |
Type2 |
527 - 822 |
0 |
None |
None |
BDNF/NT-3 growth factors receptor |
Homo sapiens |
|
TYR
|
NTRK3
|
NTRK3_HUMAN
|
3V5QA
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-out |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0F4 |
Type2 |
530 - 832 |
0 |
None |
None |
NT-3 growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK3
|
NTRK3_HUMAN
|
3V5QB
|
2.2 |
Inactive |
DFGout‑BBAminus |
out-out |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0F4 |
Type2 |
530 - 832 |
0 |
None |
None |
NT-3 growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK3
|
NTRK3_HUMAN
|
6KZCA
|
2.0 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DZC |
Type2 |
528 - 837 |
0 |
None |
None |
NT-3 growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK3
|
NTRK3_HUMAN
|
6KZDA
|
1.708 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
DZ6 |
Type2 |
528 - 837 |
0 |
None |
None |
NT-3 growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK3
|
NTRK3_HUMAN
|
4YMJA
|
2.0 |
Inactive |
DFGout‑None |
out-out |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
4EJ |
Type1 |
530 - 831 |
0 |
SEP706 |
None |
NT-3 growth factor receptor |
Homo sapiens |
|
TYR
|
NTRK3
|
NTRK3_HUMAN
|
4YMJB
|
2.0 |
Inactive |
DFGout‑None |
out-none |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
4EJ |
Type1 |
530 - 834 |
0 |
SEP706 |
None |
NT-3 growth factor receptor |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
9GZHA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
A1IRC |
Type2 |
583 - 958 |
0 |
None |
T674I |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
5GRNA
|
1.77 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
748 |
Type2 |
583 - 958 |
0 |
None |
None |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
6JOLA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
583 - 957 |
0 |
None |
None |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
8PQKA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
554 - 973 |
0 |
None |
T674I |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
6A32A
|
1.87 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
554 - 973 |
0 |
None |
T674I |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
8PQJA
|
1.82 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
553 - 973 |
0 |
None |
None |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
5K5XA
|
2.168 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
554 - 973 |
0 |
None |
None |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PDGFRA
|
PGFRA_HUMAN
|
6JOKA
|
3.8 |
Inactive |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B49 |
Type1 |
556 - 973 |
0 |
None |
None |
Platelet-derived growth factor receptor alpha |
Homo sapiens |
|
TYR
|
PTK2
|
FAK1_HUMAN
|
4KAOA
|
2.39 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
KAO |
Type2 |
415 - 686 |
0 |
None |
P410G |
Focal adhesion kinase 1 |
Homo sapiens |
|
TYR
|
PTK2
|
FAK1_HUMAN
|
4KAOB
|
2.39 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
KAO |
Type2 |
414 - 686 |
0 |
None |
P410G |
Focal adhesion kinase 1 |
Homo sapiens |
|
TYR
|
PTK2
|
FAK1_HUMAN
|
4EBVA
|
1.67 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_niiai |
APEdist_aaao |
0O7 |
Type1 |
411 - 686 |
0 |
None |
None |
Focal adhesion kinase 1 |
Homo sapiens |
|
TYR
|
PTK2
|
FAK1_HUMAN
|
4K9YA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
TYR |
APEdihe_oiiai |
APEdist_aaao |
K9Y |
Type2 |
415 - 685 |
0 |
None |
None |
Focal adhesion kinase 1 |
Homo sapiens |
|
TYR
|
PTK2
|
FAK1_HUMAN
|
4I4FA
|
1.75 |
Inactive |
DFGout‑None |
out-out |
none-out |
TYR |
APEdihe_niiai |
APEdist_aaao |
1BR |
Type3 |
415 - 686 |
0 |
None |
None |
Focal adhesion kinase 1 |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
3FZSA
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
B96 |
Type2 |
420 - 690 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
4H1MA
|
1.99 |
Inactive |
DFGout‑BBAminus |
in-in |
none-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
0YJ |
Type2 |
420 - 690 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
3FZPA
|
2.1 |
Inactive |
DFGout‑None |
in-out |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
AGS |
ATPlike |
419 - 692 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
3ET7A
|
2.7 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
349 |
Type1 |
419 - 691 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
3FZRA
|
2.7 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
3JZ |
Type1 |
419 - 691 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
5TO8A
|
1.985 |
Inactive |
DFGout‑None |
in-none |
out-none |
TYR |
APEdihe_nnnan |
APEdist_aaan |
7FM |
Type1 |
420 - 691 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
3FZTA
|
1.95 |
Inactive |
DFGout‑None |
in-in |
out-none |
TYR |
APEdihe_nniai |
APEdist_aaai |
4JZ |
Type2 |
420 - 690 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK2B
|
FAK2_HUMAN
|
4H1JA
|
2.0 |
Inactive |
DFGout‑None |
in-in |
out-out |
TYR |
APEdihe_oiiai |
APEdist_aaai |
0YH |
Type2 |
419 - 690 |
0 |
None |
None |
Protein-tyrosine kinase 2-beta |
Homo sapiens |
|
TYR
|
PTK6
|
PTK6_HUMAN
|
6CZ4A
|
1.5 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
FKY |
Type2 |
183 - 443 |
0 |
None |
None |
Protein-tyrosine kinase 6 |
Homo sapiens |
|
TYR
|
PTK7
|
PTK7_HUMAN
|
6VG3A
|
1.95 |
Pseudo |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
788 - 1064 |
0 |
None |
None |
Inactive tyrosine-protein kinase 7 |
Homo sapiens |
|
TYR
|
PTK7
|
PTK7_HUMAN
|
6VG3B
|
1.95 |
Pseudo |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
788 - 1066 |
0 |
None |
None |
Inactive tyrosine-protein kinase 7 |
Homo sapiens |
|
TYR
|
PTK7
|
PTK7_HUMAN
|
6VG3C
|
1.95 |
Pseudo |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
789 - 1063 |
0 |
None |
None |
Inactive tyrosine-protein kinase 7 |
Homo sapiens |
|
TYR
|
ROR2
|
ROR2_HUMAN
|
3ZZWB
|
2.9 |
Pseudo |
DFGout‑None |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
No_ligand |
No_ligand |
466 - 750 |
0 |
None |
None |
Tyrosine-protein kinase transmembrane receptor ROR2 |
Homo sapiens |
|
TYR
|
SRC
|
SRC_HUMAN
|
7OTEA
|
2.49 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
0LI |
Type2 |
261 - 536 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Homo sapiens |
|
TYR
|
SRC
|
SRC_HUMAN
|
7OTEB
|
2.49 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
0LI |
Type2 |
261 - 536 |
0 |
None |
None |
Proto-oncogene tyrosine-protein kinase Src |
Homo sapiens |
|
TYR
|
SYK
|
KSYK_HUMAN
|
3TUBA
|
2.23 |
Inactive |
DFGout‑BBAminus |
in-out |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
FPU |
Type2 |
362 - 633 |
0 |
None |
None |
Tyrosine-protein kinase SYK |
Homo sapiens |
|
TYR
|
SYK
|
KSYK_HUMAN
|
3TUDA
|
2.33 |
Inactive |
DFGout‑None |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FPX |
Type2 |
363 - 635 |
0 |
None |
None |
Tyrosine-protein kinase SYK |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
2OO8X
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
RAJ |
Type2 |
836 - 1117 |
0 |
None |
None |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
2OSCA
|
2.8 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
MUH |
Type2 |
837 - 1116 |
0 |
None |
None |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
2P4IA
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
MR9 |
Type2 |
838 - 1117 |
0 |
None |
None |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
6MWEA
|
2.05 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oooai |
APEdist_aaao |
919 |
Type2 |
816 - 1122 |
0 |
None |
None |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
6MWEB
|
2.05 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_oooai |
APEdist_aaao |
919 |
Type2 |
816 - 1122 |
0 |
None |
None |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
2WQBA
|
2.95 |
Inactive |
DFGout‑None |
none-none |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
QQ1 |
Type1 |
816 - 1120 |
0 |
None |
D964N |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
2P4IB
|
2.5 |
Inactive |
DFGout‑None |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
MR9 |
Type2 |
836 - 1117 |
0 |
None |
None |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TEK
|
TIE2_HUMAN
|
4X3JA
|
2.5 |
Inactive |
DFGout‑None |
in-out |
none-out |
TYR |
APEdihe_nniai |
APEdist_aaao |
3WR |
Type2 |
838 - 1117 |
0 |
None |
D964N |
Angiopoietin-1 receptor |
Homo sapiens |
|
TYR
|
TNK2
|
ACK1_HUMAN
|
5ZXBA
|
2.198 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
9KO |
Type2 |
117 - 389 |
0 |
None |
None |
Activated CDC42 kinase 1 |
Homo sapiens |
|
TYR
|
TNK2
|
ACK1_HUMAN
|
5ZXBB
|
2.198 |
Inactive |
DFGout‑None |
in-in |
none-none |
TYR |
APEdihe_nnnai |
APEdist_aaan |
9KO |
Type2 |
117 - 389 |
0 |
None |
None |
Activated CDC42 kinase 1 |
Homo sapiens |
|
CMGC
|
MPK3
|
A0A3S7WR45_LEIDO
|
4O2ZA
|
2.71 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
046 |
Type2 |
5 - 363 |
0 |
None |
None |
Mitogen-activated protein kinase |
Leishmania donovani |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
3UBDA
|
1.53 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
SL0 |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
4EL9A
|
1.55 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
AFE |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
AGC
|
RPS6KA3-1
|
KS6A3_MOUSE
|
4GUEA
|
1.8 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
QCT |
Type1 |
48 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
5LARA
|
1.5 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
6SH |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6Y4TA
|
1.98 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
O8W |
Type2 |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6Y4UA
|
1.86 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
O98 |
Type2 |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6Y4VA
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
O8Z |
Type2 |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6Y4WA
|
1.86 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
O8T |
Type2 |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6Y4XA
|
1.6 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
O8Q |
Type2 |
1 - 360 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6Y6VA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
OE5 |
Type2 |
4 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6YJCA
|
1.741 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
OSZ |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6YK7A
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nioo |
OU2 |
Type2 |
5 - 355 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
6ZWRA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
OEB |
Type2 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
7BDQA
|
2.75 |
Inactive |
DFGout‑BBAminus |
in-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
TJZ |
Type2 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
7BE4A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
TK5 |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
7BE5A
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
TKB |
Type2 |
4 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
2PUUA
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
G2G |
Type2 |
5 - 352 |
0 |
None |
N14A |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
3P5KA
|
2.09 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
P5K |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
3P78A
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
P78 |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
3P79A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
P79 |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
3P7AA
|
2.31 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
P7A |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
3P7BA
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
P7B |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
3P7CA
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
P7C |
Type3 |
5 - 352 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
CMGC
|
MAPK14
|
MK14_MOUSE
|
7BDOA
|
2.7 |
Inactive |
DFGout‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
TBK |
Type2 |
5 - 353 |
0 |
None |
None |
Mitogen-activated protein kinase 14 |
Mus musculus |
|
TKL
|
RIPK3
|
RIPK3_MOUSE
|
6OKOA
|
2.1 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
1FN |
Type2 |
14 - 311 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 3 |
Mus musculus |
|
TKL
|
RIPK3
|
RIPK3_MOUSE
|
6OKOB
|
2.1 |
Inactive |
DFGout‑None |
in-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
1FN |
Type2 |
13 - 311 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 3 |
Mus musculus |
|
TKL
|
RIPK3
|
RIPK3_MOUSE
|
9IX2A
|
2.39 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1SU |
Type2 |
15 - 311 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 3 |
Mus musculus |
|
TKL
|
RIPK3
|
RIPK3_MOUSE
|
9IX3A
|
2.07 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1EAA |
Type2 |
15 - 311 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 3 |
Mus musculus |
|
TKL
|
RIPK3
|
RIPK3_MOUSE
|
9IX3B
|
2.07 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1EAA |
Type2 |
15 - 310 |
0 |
None |
None |
Receptor-interacting serine/threonine-protein kinase 3 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3K5VA
|
1.74 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STJ,
STI
|
Allosteric,
Type2
|
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3K5VB
|
1.74 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STJ,
STI
|
Allosteric,
Type2
|
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
6HD4A
|
2.03 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FYW,
STI
|
Allosteric,
Type2
|
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
6HD4B
|
2.03 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FYW,
STI
|
Allosteric,
Type2
|
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
6HD6A
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
FYH,
STI
|
Allosteric,
Type2
|
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3OY3A
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
XY3 |
Type2 |
229 - 511 |
0 |
None |
T315I |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3OY3B
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
XY3 |
Type2 |
229 - 511 |
0 |
None |
T315I |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3IK3A
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
none-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI |
Type2 |
229 - 513 |
0 |
None |
T315I |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3IK3B
|
1.9 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
0LI |
Type2 |
229 - 513 |
0 |
None |
T315I |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3OXZA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
none-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
0LI |
Type2 |
229 - 511 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3KFAA
|
1.22 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B91 |
Type2 |
229 - 511 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3KFAB
|
1.22 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
B91 |
Type2 |
229 - 511 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1FPUA
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
PRC |
Type2 |
229 - 499 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1FPUB
|
2.4 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
PRC |
Type2 |
229 - 499 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1IEPA
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
229 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1IEPB
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-out |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
229 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1OPJA
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
TYR |
APEdihe_iiiai |
APEdist_aaao |
STI |
Type2 |
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1OPJB
|
1.75 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
229 - 512 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
2HZNA
|
2.7 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
KIN |
Type2 |
229 - 502 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
6HD6B
|
2.3 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI |
Type2 |
229 - 510 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3MS9A
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
MS9
|
Type2,
Allosteric
|
230 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3MS9B
|
1.8 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
MS9
|
Type2,
Allosteric
|
229 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3MSSA
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
MS7
|
Type2,
Allosteric
|
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3MSSB
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
MS7
|
Type2,
Allosteric
|
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3MSSC
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
MS7
|
Type2,
Allosteric
|
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
3MSSD
|
1.95 |
Inactive |
DFGout‑BBAminus |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
STI,
MS7
|
Type2,
Allosteric
|
232 - 498 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1M52A
|
2.6 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P17 |
Type1.5_Back |
232 - 502 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1M52B
|
2.6 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P17 |
Type1.5_Back |
232 - 503 |
0 |
None |
None |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
TYR
|
ABL1
|
ABL1_MOUSE
|
1OPKA
|
1.8 |
Inactive |
DFGout‑None |
in-in |
out-in |
TYR |
APEdihe_iiiai |
APEdist_aaai |
P16 |
Type1.5_Back |
64 - 512 |
0 |
None |
D363N |
Tyrosine-protein kinase ABL1 |
Mus musculus |
|
OTHER
|
PKNE
|
PKNE_MYCTU
|
2H34A
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
14 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase PknE |
Mycobacterium tuberculosis |
|
OTHER
|
PKNE
|
PKNE_MYCTU
|
2H34B
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
14 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase PknE |
Mycobacterium tuberculosis |
|
CMGC
|
MAPK1
|
MK01_RAT
|
4I5HA
|
1.9 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
G17 |
Type2 |
9 - 356 |
0 |
None |
Q103A,C164L |
Mitogen-activated protein kinase 1 |
Rattus norvegicus |
|
CMGC
|
P38A
|
A9UJZ9_SALSA
|
3OHTA
|
2.7 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
1N1,
1N1
|
Type1.5_Back,
Allosteric
|
5 - 352 |
0 |
None |
None |
mitogen-activated protein kinase |
Salmo salar |
|
CMGC
|
P38A
|
A9UJZ9_SALSA
|
3OHTB
|
2.7 |
Inactive |
DFGout‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
1N1,
1N1
|
Type1.5_Back,
Allosteric
|
5 - 352 |
0 |
None |
None |
mitogen-activated protein kinase |
Salmo salar |
|
OTHER
|
TCUR0376
|
D1A2F7_THECD
|
8CAVA
|
2.87 |
Inactive |
DFGout‑None |
out-na |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
Allosteric |
6 - 865 |
0 |
None |
None |
Serine/threonine protein kinase |
Thermomonospora curvata |
|
OTHER
|
TCUR0376
|
D1A2F7_THECD
|
8CAVB
|
2.87 |
Inactive |
DFGout‑None |
out-na |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
Allosteric |
6 - 863 |
0 |
None |
None |
Serine/threonine protein kinase |
Thermomonospora curvata |
|
CMGC
|
PRP4K
|
S7UT92_TOXGG
|
7Q4AA
|
2.31 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
A9I |
Type2 |
547 - 894 |
0 |
PTR729 |
None |
non-specific serine/threonine protein kinase |
Toxoplasma gondii |
|
CMGC
|
PRP4K
|
S7UT92_TOXGG
|
7Q4AB
|
2.31 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
A9I |
Type2 |
546 - 891 |
0 |
PTR729 |
None |
non-specific serine/threonine protein kinase |
Toxoplasma gondii |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8A
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 650 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8B
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 650 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8C
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 650 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8D
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 650 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8E
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 650 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8F
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 650 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8G
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 621 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
IKBKBL
|
Q6INT1_XENLA
|
3QA8H
|
3.6 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 621 |
0 |
None |
S161E,S165E |
IkappaB kinase |
Xenopus laevis |
|
OTHER
|
DRIK1
|
C0P4K9_MAIZE
|
6CPYA
|
1.7 |
Pseudo |
DFGout‑BBAminus |
in-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
187 - 492 |
0 |
None |
None |
Protein kinase superfamily protein |
Zea mays |
|
OTHER
|
DRIK1
|
C0P4K9_MAIZE
|
6CPYB
|
1.7 |
Pseudo |
DFGout‑BBAminus |
out-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
209 - 492 |
0 |
None |
None |
Protein kinase superfamily protein |
Zea mays |
|
OTHER
|
DRIK1
|
C0P4K9_MAIZE
|
6EASA
|
2.0 |
Pseudo |
DFGout‑BBAminus |
out-na |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
J3A |
Type1 |
208 - 492 |
0 |
None |
None |
Protein kinase superfamily protein |
Zea mays |