| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | PIM1 | PIM1_HUMAN | 5O11A | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 34 - 305 | 0 | SEP261 | None | Serine/threonine-protein kinase pim-1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDC | 2.7 | Inactive | DFGin‑ABAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iioo | 3NG | Type1 | 150 - 479 | 0 | None | None | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDB | 2.7 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiio | APEdist_iiii | 3NG | Type1 | 149 - 482 | 0 | None | None | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDA | 2.7 | Inactive | DFGin‑None | in-in | in-out | nonTYR | APEdihe_aannn | APEdist_ioon | 3NG | Type1 | 149 - 481 | 0 | None | None | Dual specificity protein kinase CLK1 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYLA | 1.95 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 144 - 483 | 0 | None | None | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6KHEA | 2.8 | Inactive | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 144 - 485 | 0 | None | None | Dual specificity protein kinase CLK2 |
| CMGC | CLK3 | CLK3_HUMAN | 6FYPA | 2.29 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 482 | 0 | None | None | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 6KHFA | 2.598 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_oioi | 3NG | Type1 | 142 - 481 | 0 | None | None | Dual specificity protein kinase CLK3 |
| CMGC | CLK4 | CLK4_HUMAN | 6FYVA | 2.46 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 148 - 479 | 0 | None | None | Dual specificity protein kinase CLK4 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHA | 1.96 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | SY4, 3NG | Allosteric, Type1 | 2 - 333 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAA | 2.71 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAB | 2.71 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3PE1A | 1.6 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 3 - 329 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHB | 1.96 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, SY4 | Type1, Allosteric | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHA | 2.07 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, T9Y | Type1, Allosteric | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHB | 2.07 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, T9Y | Type1, Allosteric | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha |
| CMGC | CSNK2A2 | CSK22_HUMAN | 8QBUA | 1.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 42J, 3NG | Allosteric, Type1 | 6 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9IHIA | 1.23 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | SY4, 3NG | Allosteric, Type1 | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9BA | 1.84 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | VN9, 3NG | Allosteric, Type1 | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QB6A | 1.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | RDV, 3NG | Allosteric, Type1 | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QABA | 0.95 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | RA7, 3NG, RA7 | Allosteric, Type1, Allosteric | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 6HMBA | 1.04 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 7 - 334 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9HK5A | 1.491 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 7 - 334 | 0 | None | P32V,V83I,T101I,C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9AA | 1.03 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, A1I4V | Type1, Allosteric | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9DA | 0.89 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, R9G | Type1, Allosteric | 7 - 332 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QAGA | 1.01 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, RBJ | Type1, Allosteric | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NA | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NB | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NC | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 134 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5ND | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NE | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NF | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NG | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 137 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NH | 2.77 | None | DFGin‑BLAminus | in-in | in-none | nonTYR | APEdihe_aaini | APEdist_niii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FA | 3.0 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 28 - 383 | 0 | PTR216 | None | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FB | 3.0 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 38 - 382 | 0 | PTR216 | None | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1GA | 2.85 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 27 - 383 | 0 | None | None | Glycogen synthase kinase-3 beta |
| CMGC | HIPK2 | HIPK2_HUMAN | 6P5SA | 2.194 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 185 - 535 | 0 | PTR361,SEP441 | None | Homeodomain-interacting protein kinase 2 |
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CKA1 | J9VNH4_CRYN9 | 6K3LB | 2.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 5 - 333 | 0 | None | None | Casein kinase II subunit alpha | Cryptococcus neoformans |
| CAMK | PIM1 | PIM1_HUMAN | 5O11A | 2.4 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 34 - 305 | 0 | SEP261 | None | Serine/threonine-protein kinase pim-1 | Homo sapiens |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDC | 2.7 | Inactive | DFGin‑ABAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iioo | 3NG | Type1 | 150 - 479 | 0 | None | None | Dual specificity protein kinase CLK1 | Homo sapiens |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDB | 2.7 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiio | APEdist_iiii | 3NG | Type1 | 149 - 482 | 0 | None | None | Dual specificity protein kinase CLK1 | Homo sapiens |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDA | 2.7 | Inactive | DFGin‑None | in-in | in-out | nonTYR | APEdihe_aannn | APEdist_ioon | 3NG | Type1 | 149 - 481 | 0 | None | None | Dual specificity protein kinase CLK1 | Homo sapiens |
| CMGC | CLK2 | CLK2_HUMAN | 6FYLA | 1.95 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 144 - 483 | 0 | None | None | Dual specificity protein kinase CLK2 | Homo sapiens |
| CMGC | CLK2 | CLK2_HUMAN | 6KHEA | 2.8 | Inactive | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 144 - 485 | 0 | None | None | Dual specificity protein kinase CLK2 | Homo sapiens |
| CMGC | CLK3 | CLK3_HUMAN | 6FYPA | 2.29 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 482 | 0 | None | None | Dual specificity protein kinase CLK3 | Homo sapiens |
| CMGC | CLK3 | CLK3_HUMAN | 6KHFA | 2.598 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaiii | APEdist_oioi | 3NG | Type1 | 142 - 481 | 0 | None | None | Dual specificity protein kinase CLK3 | Homo sapiens |
| CMGC | CLK4 | CLK4_HUMAN | 6FYVA | 2.46 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 148 - 479 | 0 | None | None | Dual specificity protein kinase CLK4 | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHA | 1.96 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | SY4, 3NG | Allosteric, Type1 | 2 - 333 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAA | 2.71 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAB | 2.71 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3PE1A | 1.6 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 3 - 329 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHB | 1.96 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, SY4 | Type1, Allosteric | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHA | 2.07 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, T9Y | Type1, Allosteric | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHB | 2.07 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, T9Y | Type1, Allosteric | 2 - 332 | 0 | None | None | Casein kinase II subunit alpha | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 8QBUA | 1.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 42J, 3NG | Allosteric, Type1 | 6 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9IHIA | 1.23 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | SY4, 3NG | Allosteric, Type1 | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9BA | 1.84 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | VN9, 3NG | Allosteric, Type1 | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QB6A | 1.05 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | RDV, 3NG | Allosteric, Type1 | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QABA | 0.95 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | RA7, 3NG, RA7 | Allosteric, Type1, Allosteric | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 6HMBA | 1.04 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 7 - 334 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9HK5A | 1.491 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 7 - 334 | 0 | None | P32V,V83I,T101I,C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9AA | 1.03 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, A1I4V | Type1, Allosteric | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9DA | 0.89 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, R9G | Type1, Allosteric | 7 - 332 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QAGA | 1.01 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG, RBJ | Type1, Allosteric | 7 - 333 | 0 | None | C336S | Casein kinase II subunit alpha' | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NA | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NB | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NC | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 134 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5ND | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NE | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NF | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NG | 2.77 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 137 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NH | 2.77 | None | DFGin‑BLAminus | in-in | in-none | nonTYR | APEdihe_aaini | APEdist_niii | 3NG | Type1 | 135 - 480 | 0 | PTR321 | None | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FA | 3.0 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 28 - 383 | 0 | PTR216 | None | Glycogen synthase kinase-3 beta | Homo sapiens |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FB | 3.0 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 38 - 382 | 0 | PTR216 | None | Glycogen synthase kinase-3 beta | Homo sapiens |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1GA | 2.85 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | 3NG | Type1 | 27 - 383 | 0 | None | None | Glycogen synthase kinase-3 beta | Homo sapiens |
| CMGC | HIPK2 | HIPK2_HUMAN | 6P5SA | 2.194 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 185 - 535 | 0 | PTR361,SEP441 | None | Homeodomain-interacting protein kinase 2 | Homo sapiens |
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CKA1 | J9VNH4_CRYN9 | 6K3LB | 2.09 | Inactive | DFGin‑BLAminus | in-in | in-out | nonTYR | APEdihe_aaioi | APEdist_iiii | 3NG | Type1 | 5 - 333 | 0 | None | None | Casein kinase II subunit alpha | Cryptococcus neoformans |