| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | MELK | MELK_HUMAN | 4IXPA | 2.749 | Inactive | DFGinter‑BABtrans | out-none | out-out | nonTYR | APEdihe_aaoii | APEdist_oooo | No_ligand | No_ligand | 2 - 335 | 0 | None | K40R,D150A | Maternal embryonic leucine zipper kinase |
| NEK | NEK1 | NEK1_HUMAN | 4APCA | 2.1 | Inactive | DFGinter‑BABtrans | out-none | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | No_ligand | No_ligand | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 |
| NEK | NEK1 | NEK1_HUMAN | 4APCB | 2.1 | Inactive | DFGinter‑BABtrans | out-out | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | No_ligand | No_ligand | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 |
| NEK | NEK1 | NEK1_HUMAN | 4B9DA | 1.9 | Inactive | DFGinter‑BABtrans | out-none | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | CK7 | Type1 | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 |
| NEK | NEK1 | NEK1_HUMAN | 4B9DB | 1.9 | Inactive | DFGinter‑BABtrans | out-out | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | CK7 | Type1 | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 |
| OTHER | EIF2AK4-2 | E2AK4_HUMAN | 7QWKH | 2.3 | Inactive | DFGinter‑BABtrans | out-out | out-out | nonTYR | APEdihe_aaoni | APEdist_oooo | G41 | Type1 | 584 - 1006 | 0 | None | D848N | eIF-2-alpha kinase GCN2 |
| STE | MAP3K5 | M3K5_HUMAN | 2CLQA | 2.3 | Inactive | DFGinter‑BABtrans | out-out | in-out | nonTYR | APEdihe_aaiii | APEdist_iooi | STU | Type1 | 670 - 940 | 0 | None | None | Mitogen-activated protein kinase kinase kinase 5 |
| STE | MAP3K5 | M3K5_HUMAN | 2CLQB | 2.3 | Inactive | DFGinter‑BABtrans | in-none | in-out | nonTYR | APEdihe_aaiii | APEdist_nooi | STU | Type1 | 670 - 940 | 0 | None | None | Mitogen-activated protein kinase kinase kinase 5 |
| TYR | ABL1 | ABL1_HUMAN | 7W7XA | 2.0 | Inactive | DFGinter‑BABtrans | in-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | 8DW | Type1 | 232 - 500 | 0 | PTR393 | None | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 7W7XB | 2.0 | Inactive | DFGinter‑BABtrans | in-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | 8DW | Type1 | 232 - 500 | 0 | PTR393 | None | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 4XEYB | 2.891 | Inactive | DFGinter‑BABtrans | in-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | 1N1 | Type1 | 122 - 504 | 0 | None | None | Tyrosine-protein kinase ABL1 |
| TYR | BMX | BMX_HUMAN | 3SXRA | 2.4 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | 1N1 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 3SXRB | 2.4 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | 1N1 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 3SXSA | 1.89 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | PP2 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 6I99A | 2.001 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | H88 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 6I99B | 2.001 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | H88 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BTK | BTK_HUMAN | 5XYZA | 2.64 | Inactive | DFGinter‑BABtrans | out-out | out-none | TYR | APEdihe_nniai | APEdist_aaai | GYL | Type1 | 394 - 656 | 0 | None | None | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 5XYZB | 2.64 | Inactive | DFGinter‑BABtrans | out-out | out-none | TYR | APEdihe_nniai | APEdist_aaai | GYL | Type1 | 394 - 656 | 0 | None | None | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 7YC9A | 1.4 | Inactive | DFGinter‑BABtrans | out-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | IS4 | Type1 | 395 - 658 | 0 | None | None | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 3OCTA | 1.95 | Inactive | DFGinter‑BABtrans | in-out | out-none | TYR | APEdihe_nniai | APEdist_aaai | 1N1 | Type1 | 394 - 656 | 0 | None | V555R | Tyrosine-protein kinase BTK |
| TYR | CSK | CSK_HUMAN | 1BYGA | 2.4 | Inactive | DFGinter‑BABtrans | out-out | none-none | TYR | APEdihe_nniai | APEdist_aaai | STU | Type1 | 187 - 448 | 0 | None | None | Tyrosine-protein kinase CSK |
| TYR | SRC | SRC_HUMAN | 4MXXB | 2.6 | Inactive | DFGinter‑BABtrans | out-out | none-none | TYR | APEdihe_nniai | APEdist_aaai | DB8 | Type1 | 261 - 536 | 0 | None | A406T | Proto-oncogene tyrosine-protein kinase Src |
| TYR | TEK | TIE2_HUMAN | 1FVRA | 2.2 | Inactive | DFGinter‑BABtrans | out-out | out-out | TYR | APEdihe_nniai | APEdist_aaao | No_ligand | No_ligand | 813 - 1121 | 0 | None | None | Angiopoietin-1 receptor |
| TYR | TEK | TIE2_HUMAN | 1FVRB | 2.2 | Inactive | DFGinter‑BABtrans | out-out | out-out | TYR | APEdihe_niiai | APEdist_aaao | No_ligand | No_ligand | 813 - 1121 | 0 | None | None | Angiopoietin-1 receptor |
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | MELK | MELK_HUMAN | 4IXPA | 2.749 | Inactive | DFGinter‑BABtrans | out-none | out-out | nonTYR | APEdihe_aaoii | APEdist_oooo | No_ligand | No_ligand | 2 - 335 | 0 | None | K40R,D150A | Maternal embryonic leucine zipper kinase | Homo sapiens |
| NEK | NEK1 | NEK1_HUMAN | 4APCA | 2.1 | Inactive | DFGinter‑BABtrans | out-none | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | No_ligand | No_ligand | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 | Homo sapiens |
| NEK | NEK1 | NEK1_HUMAN | 4APCB | 2.1 | Inactive | DFGinter‑BABtrans | out-out | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | No_ligand | No_ligand | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 | Homo sapiens |
| NEK | NEK1 | NEK1_HUMAN | 4B9DA | 1.9 | Inactive | DFGinter‑BABtrans | out-none | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | CK7 | Type1 | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 | Homo sapiens |
| NEK | NEK1 | NEK1_HUMAN | 4B9DB | 1.9 | Inactive | DFGinter‑BABtrans | out-out | out-out | nonTYR | APEdihe_aaiii | APEdist_oooo | CK7 | Type1 | 1 - 284 | 0 | None | T162A | Serine/threonine-protein kinase Nek1 | Homo sapiens |
| OTHER | EIF2AK4-2 | E2AK4_HUMAN | 7QWKH | 2.3 | Inactive | DFGinter‑BABtrans | out-out | out-out | nonTYR | APEdihe_aaoni | APEdist_oooo | G41 | Type1 | 584 - 1006 | 0 | None | D848N | eIF-2-alpha kinase GCN2 | Homo sapiens |
| STE | MAP3K5 | M3K5_HUMAN | 2CLQA | 2.3 | Inactive | DFGinter‑BABtrans | out-out | in-out | nonTYR | APEdihe_aaiii | APEdist_iooi | STU | Type1 | 670 - 940 | 0 | None | None | Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens |
| STE | MAP3K5 | M3K5_HUMAN | 2CLQB | 2.3 | Inactive | DFGinter‑BABtrans | in-none | in-out | nonTYR | APEdihe_aaiii | APEdist_nooi | STU | Type1 | 670 - 940 | 0 | None | None | Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens |
| TYR | ABL1 | ABL1_HUMAN | 7W7XA | 2.0 | Inactive | DFGinter‑BABtrans | in-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | 8DW | Type1 | 232 - 500 | 0 | PTR393 | None | Tyrosine-protein kinase ABL1 | Homo sapiens |
| TYR | ABL1 | ABL1_HUMAN | 7W7XB | 2.0 | Inactive | DFGinter‑BABtrans | in-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | 8DW | Type1 | 232 - 500 | 0 | PTR393 | None | Tyrosine-protein kinase ABL1 | Homo sapiens |
| TYR | ABL1 | ABL1_HUMAN | 4XEYB | 2.891 | Inactive | DFGinter‑BABtrans | in-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | 1N1 | Type1 | 122 - 504 | 0 | None | None | Tyrosine-protein kinase ABL1 | Homo sapiens |
| TYR | BMX | BMX_HUMAN | 3SXRA | 2.4 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | 1N1 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens |
| TYR | BMX | BMX_HUMAN | 3SXRB | 2.4 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | 1N1 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens |
| TYR | BMX | BMX_HUMAN | 3SXSA | 1.89 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | PP2 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens |
| TYR | BMX | BMX_HUMAN | 6I99A | 2.001 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | H88 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens |
| TYR | BMX | BMX_HUMAN | 6I99B | 2.001 | Inactive | DFGinter‑BABtrans | out-out | in-in | TYR | APEdihe_iiiai | APEdist_aaai | H88 | Type1 | 411 - 671 | 0 | None | Q432K,Q611M,D617T,Q620E | Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens |
| TYR | BTK | BTK_HUMAN | 5XYZA | 2.64 | Inactive | DFGinter‑BABtrans | out-out | out-none | TYR | APEdihe_nniai | APEdist_aaai | GYL | Type1 | 394 - 656 | 0 | None | None | Tyrosine-protein kinase BTK | Homo sapiens |
| TYR | BTK | BTK_HUMAN | 5XYZB | 2.64 | Inactive | DFGinter‑BABtrans | out-out | out-none | TYR | APEdihe_nniai | APEdist_aaai | GYL | Type1 | 394 - 656 | 0 | None | None | Tyrosine-protein kinase BTK | Homo sapiens |
| TYR | BTK | BTK_HUMAN | 7YC9A | 1.4 | Inactive | DFGinter‑BABtrans | out-out | out-in | TYR | APEdihe_iiiai | APEdist_aaai | IS4 | Type1 | 395 - 658 | 0 | None | None | Tyrosine-protein kinase BTK | Homo sapiens |
| TYR | BTK | BTK_HUMAN | 3OCTA | 1.95 | Inactive | DFGinter‑BABtrans | in-out | out-none | TYR | APEdihe_nniai | APEdist_aaai | 1N1 | Type1 | 394 - 656 | 0 | None | V555R | Tyrosine-protein kinase BTK | Homo sapiens |
| TYR | CSK | CSK_HUMAN | 1BYGA | 2.4 | Inactive | DFGinter‑BABtrans | out-out | none-none | TYR | APEdihe_nniai | APEdist_aaai | STU | Type1 | 187 - 448 | 0 | None | None | Tyrosine-protein kinase CSK | Homo sapiens |
| TYR | SRC | SRC_HUMAN | 4MXXB | 2.6 | Inactive | DFGinter‑BABtrans | out-out | none-none | TYR | APEdihe_nniai | APEdist_aaai | DB8 | Type1 | 261 - 536 | 0 | None | A406T | Proto-oncogene tyrosine-protein kinase Src | Homo sapiens |
| TYR | TEK | TIE2_HUMAN | 1FVRA | 2.2 | Inactive | DFGinter‑BABtrans | out-out | out-out | TYR | APEdihe_nniai | APEdist_aaao | No_ligand | No_ligand | 813 - 1121 | 0 | None | None | Angiopoietin-1 receptor | Homo sapiens |
| TYR | TEK | TIE2_HUMAN | 1FVRB | 2.2 | Inactive | DFGinter‑BABtrans | out-out | out-out | TYR | APEdihe_niiai | APEdist_aaao | No_ligand | No_ligand | 813 - 1121 | 0 | None | None | Angiopoietin-1 receptor | Homo sapiens |
| TYR | BTK | BTK_MOUSE | 8S9FA | 2.6 | Inactive | DFGinter‑BABtrans | out-out | out-none | TYR | APEdihe_nnnai | APEdist_aaan | 1N1 | Type1 | 392 - 659 | 0 | None | L390G,Y551E,Y617P | Tyrosine-protein kinase BTK | Mus musculus |
| TYR | BTK | BTK_MOUSE | 8S9FB | 2.6 | Inactive | DFGinter‑BABtrans | out-out | out-out | TYR | APEdihe_niiai | APEdist_aaao | 1N1 | Type1 | 392 - 659 | 0 | None | L390G,Y551E,Y617P | Tyrosine-protein kinase BTK | Mus musculus |
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | BTK | BTK_MOUSE | 8S9FA | 2.6 | Inactive | DFGinter‑BABtrans | out-out | out-none | TYR | APEdihe_nnnai | APEdist_aaan | 1N1 | Type1 | 392 - 659 | 0 | None | L390G,Y551E,Y617P | Tyrosine-protein kinase BTK | Mus musculus |
| TYR | BTK | BTK_MOUSE | 8S9FB | 2.6 | Inactive | DFGinter‑BABtrans | out-out | out-out | TYR | APEdihe_niiai | APEdist_aaao | 1N1 | Type1 | 392 - 659 | 0 | None | L390G,Y551E,Y617P | Tyrosine-protein kinase BTK | Mus musculus |