CMGC_DYRK1A (Dual specificity tyrosine-phosphorylation-regulated kinase 1A)

Total number of chains: 228
Uniprot: DYR1A_HUMAN
Kinase Domain Residues: 159 - 479
Spatial label Dihedral label Number of Chains Representative
DFGin BLAminus 225 AF-Q13627-K1A
DFGin ABAminus 2 6UIPB
DFGin None 1 6UIPA

Database table as tsv

PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
6UIP 3.7 Inactive DFGin‑ABAminus in-in in-in Q8J Type1 136 - 478 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6UIP 3.7 Inactive DFGin‑ABAminus in-in none-out Q8J Type1 131 - 477 9 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
AF-Q13627-K1 -1.0 Active DFGin‑BLAminus in-in in-in No_ligand No_ligand 151 - 487 0 None None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
AF-Q13627-K3 -1.0 Active DFGin‑BLAminus in-in in-in No_ligand No_ligand 151 - 487 0 None None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6T6A 2.8 Active DFGin‑BLAminus in-in in-in No_ligand No_ligand 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIL 2.465 Inactive DFGin‑BLAminus in-in in-out No_ligand No_ligand 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6LN1 2.699 Active DFGin‑BLAminus in-in in-in EKU Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6LN1 2.699 Active DFGin‑BLAminus in-in in-in EKU Type1 140 - 479 4 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4R 1.8 Active DFGin‑BLAminus in-in in-in QY8 Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4R 1.8 Active DFGin‑BLAminus in-in in-in QY8 Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A52 2.1 Inactive DFGin‑BLAminus in-in in-out QYB Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A52 2.1 Active DFGin‑BLAminus in-in in-in QYB Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJM 2.4 Active DFGin‑BLAminus in-in in-in RKW Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJM 2.4 Active DFGin‑BLAminus in-in in-in RKW Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJS 2.15 Active DFGin‑BLAminus in-in in-in RKH Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJS 2.15 Active DFGin‑BLAminus in-in in-in RKH Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7OY6 2.38 Inactive DFGin‑BLAminus in-in in-out 39I Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4S 3.1 Active DFGin‑BLAminus in-in in-in QYE Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4Z 1.9 Active DFGin‑BLAminus in-in in-in 6SD Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A51 1.9 Active DFGin‑BLAminus in-in in-in QYK Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A53 2.2 Active DFGin‑BLAminus in-in in-in QYZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A53 2.2 Active DFGin‑BLAminus in-in in-in QYZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A5D 1.8 Active DFGin‑BLAminus in-in in-in QYW Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A5L 2.1 Active DFGin‑BLAminus in-in in-in QZW Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A5N 2.3 Active DFGin‑BLAminus in-in in-in R05 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A5N 2.3 Active DFGin‑BLAminus in-in in-in R05 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJ2 2.1 Active DFGin‑BLAminus in-in in-in RJ5 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJ4 2.0 Active DFGin‑BLAminus in-in in-in RHZ Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJ5 2.0 Active DFGin‑BLAminus in-in in-in RHW Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJ7 2.9 Active DFGin‑BLAminus in-in in-in RHT Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJ8 2.0 Active DFGin‑BLAminus in-in in-in RJ8 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJA 2.2 Active DFGin‑BLAminus in-in in-in RJ2 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJV 2.1 Inactive DFGin‑BLAminus in-in in-out RKK Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJV 2.1 Inactive DFGin‑BLAminus in-in in-out RKK Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJW 2.8 Active DFGin‑BLAminus in-in in-in RKQ Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJY 2.2 Inactive DFGin‑BLAminus in-in in-out RKZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AJY 2.2 Inactive DFGin‑BLAminus in-in in-out RKZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AK2 2.1 Inactive DFGin‑BLAminus in-in in-out RHH Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AK2 2.1 Inactive DFGin‑BLAminus in-in in-out RHH Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKA 1.9 Inactive DFGin‑BLAminus in-in in-out RK2 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKA 1.9 Inactive DFGin‑BLAminus in-in in-out RK2 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKB 2.8 Inactive DFGin‑BLAminus in-in in-out RJZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKB 2.8 Inactive DFGin‑BLAminus in-in in-out RJZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKE 2.3 Inactive DFGin‑BLAminus in-in in-out RK8 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKE 2.3 Inactive DFGin‑BLAminus in-in in-out RK8 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7AKL 2.0 Active DFGin‑BLAminus in-in in-in RK5 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6A1F 1.5 Active DFGin‑BLAminus in-in in-in 9OF Type1 134 - 483 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6A1G 2.15 Active DFGin‑BLAminus in-in in-in 9OL Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6A1G 2.15 Active DFGin‑BLAminus in-in in-in 9OL Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8YEV 2.252 Active DFGin‑BLAminus in-in in-in CUE Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8YEV 2.252 Active DFGin‑BLAminus in-in in-in CUE Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ2 2.8 Active DFGin‑BLAminus in-in in-in 2C4 Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ2 2.8 Active DFGin‑BLAminus in-in in-in 2C4 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ2 2.8 Active DFGin‑BLAminus in-in in-in 2C4 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4MQ2 2.8 Inactive DFGin‑BLAminus in-in in-out 2C4 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YLK 1.4 Active DFGin‑BLAminus in-in in-in 4E2 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YLL 1.4 Active DFGin‑BLAminus in-in in-in 4E3 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S11 2.445 Active DFGin‑BLAminus in-in in-in KQE Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S11 2.445 None DFGin‑BLAminus in-in in-none KQE Type1 136 - 480 3 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S14 1.05 Active DFGin‑BLAminus in-in in-in KQW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S17 1.1 Active DFGin‑BLAminus in-in in-in KQK Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1B 1.3 Active DFGin‑BLAminus in-in in-in KRQ Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1H 1.05 Active DFGin‑BLAminus in-in in-in KQZ Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 1 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 1 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6S1J 1.408 Active DFGin‑BLAminus in-in in-in KRK Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6T6A 2.8 Active DFGin‑BLAminus in-in in-in MLW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6T6A 2.8 Active DFGin‑BLAminus in-in in-in MLW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6T6A 2.8 Active DFGin‑BLAminus in-in in-in MLW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8R8E 2.22 Inactive DFGin‑BLAminus in-in in-out YOX Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8R8E 2.22 Active DFGin‑BLAminus in-in in-in YOX Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8R8E 2.22 Active DFGin‑BLAminus in-in in-in YOX Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8R8E 2.22 Active DFGin‑BLAminus in-in in-in YOX Type1 135 - 480 0 None None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHS 2.42 Inactive DFGin‑BLAminus in-in in-out 4VZ Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHS 2.42 Active DFGin‑BLAminus in-in in-in 4VZ Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHS 2.42 Inactive DFGin‑BLAminus in-in in-out 4VZ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHS 2.42 Inactive DFGin‑BLAminus in-in in-out 4VZ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8T2H 1.85 Active DFGin‑BLAminus in-in in-in XIR Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8T2H 1.85 Active DFGin‑BLAminus in-in in-in XIR Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
9CY5 2.49 Active DFGin‑BLAminus in-in in-in A1A04 Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
9CY5 2.49 Active DFGin‑BLAminus in-in in-in A1A04 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 136 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANR 2.6 Active DFGin‑BLAminus in-in in-in HRM Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANR 2.6 Inactive DFGin‑BLAminus in-in in-out HRM Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANR 2.6 Inactive DFGin‑BLAminus in-in in-out HRM Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
3ANR 2.6 Inactive DFGin‑BLAminus in-in in-out HRM Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 134 - 479 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4E 2.68 Active DFGin‑BLAminus in-in in-in 7QQ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4E 2.68 Active DFGin‑BLAminus in-in in-in 7QQ Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4E 2.68 Inactive DFGin‑BLAminus in-out in-out 7QQ Type1 134 - 473 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4E 2.68 Active DFGin‑BLAminus in-in in-in 7QQ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4L 2.73 Active DFGin‑BLAminus in-in in-in ZC3 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4L 2.73 Inactive DFGin‑BLAminus in-in in-out ZC3 Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4L 2.73 Inactive DFGin‑BLAminus in-in out-out ZC3 Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4L 2.73 Active DFGin‑BLAminus in-in in-in ZC3 Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4Q 2.37 Inactive DFGin‑BLAminus in-in in-out Y3L Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4Q 2.37 Active DFGin‑BLAminus in-in in-in Y3L Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4Q 2.37 Inactive DFGin‑BLAminus in-in in-out Y3L Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4Q 2.37 Active DFGin‑BLAminus in-in in-in Y3L Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4T 2.15 Active DFGin‑BLAminus in-in in-in AJG Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4T 2.15 Active DFGin‑BLAminus in-in in-in AJG Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4T 2.15 Inactive DFGin‑BLAminus in-in in-out AJG Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A4T 2.15 Active DFGin‑BLAminus in-in in-in AJG Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A54 2.63 Active DFGin‑BLAminus in-in in-in 5PW Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A54 2.63 Active DFGin‑BLAminus in-in in-in 5PW Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A54 2.63 Inactive DFGin‑BLAminus in-in in-out 5PW Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5A54 2.63 Active DFGin‑BLAminus in-in in-in 5PW Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIF 2.22 Active DFGin‑BLAminus in-in in-in B5T Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIF 2.22 Inactive DFGin‑BLAminus in-in in-out B5T Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIF 2.22 Inactive DFGin‑BLAminus in-in in-out B5T Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIF 2.22 Inactive DFGin‑BLAminus in-in in-out B5T Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIJ 2.42 Inactive DFGin‑BLAminus in-out in-in B5Z Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIJ 2.42 Active DFGin‑BLAminus in-in in-in B5Z Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIJ 2.42 Active DFGin‑BLAminus in-in in-in B5Z Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIL 2.465 Active DFGin‑BLAminus in-in in-in B6B Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIL 2.465 Inactive DFGin‑BLAminus in-in in-out B6B Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIL 2.465 Inactive DFGin‑BLAminus in-in in-out B6B Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIP 2.56 Inactive DFGin‑BLAminus in-out in-in B7B Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIP 2.56 Active DFGin‑BLAminus in-in in-in B7B Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIP 2.56 Inactive DFGin‑BLAminus in-in in-out B7B Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIP 2.56 Active DFGin‑BLAminus in-in in-in B7B Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIQ 2.3 Inactive DFGin‑BLAminus in-in in-out B6Z Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIQ 2.3 Inactive DFGin‑BLAminus in-in in-out B6Z Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIQ 2.3 Inactive DFGin‑BLAminus in-in in-out B6Z Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIQ 2.3 Active DFGin‑BLAminus in-in in-in B6Z Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIS 2.36 Inactive DFGin‑BLAminus in-in in-out B6N Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIS 2.36 Active DFGin‑BLAminus in-in in-in B6N Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIS 2.36 Inactive DFGin‑BLAminus in-in in-out B6N Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIS 2.36 Active DFGin‑BLAminus in-in in-in B6N Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EJ4 2.88 Inactive DFGin‑BLAminus in-out in-out B7W Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EJ4 2.88 Inactive DFGin‑BLAminus in-in in-out B7W Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EJ4 2.88 Active DFGin‑BLAminus in-in in-in B7W Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EJ4 2.88 Inactive DFGin‑BLAminus in-in in-out B7W Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6YF8 3.198 Active DFGin‑BLAminus in-in in-in OPW Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6YF8 3.198 Active DFGin‑BLAminus in-in in-in OPW Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6YF8 3.198 Inactive DFGin‑BLAminus in-in in-out OPW Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6YF8 3.198 Active DFGin‑BLAminus in-in in-in OPW Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 137 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7Z5N 2.77 None DFGin‑BLAminus in-in in-none 3NG Type1 135 - 480 4 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3R 2.06 Active DFGin‑BLAminus in-in in-in R7O Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3R 2.06 Active DFGin‑BLAminus in-in in-in R7O Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
9FPX 2.69 Active DFGin‑BLAminus in-in in-in CC9 Type1 136 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
9FPX 2.69 Active DFGin‑BLAminus in-in in-in CC9 Type1 143 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2WO6 2.5 Active DFGin‑BLAminus in-in in-in D15 Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2WO6 2.5 Active DFGin‑BLAminus in-in in-in D15 Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4AZE 3.15 Active DFGin‑BLAminus in-in in-in 3RA Type1 132 - 481 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4AZE 3.15 Active DFGin‑BLAminus in-in in-in 3RA Type1 135 - 481 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
4AZE 3.15 Active DFGin‑BLAminus in-in in-in 3RA Type1 132 - 481 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4O 1.9 Active DFGin‑BLAminus in-in in-in ANP Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4O 1.9 Inactive DFGin‑BLAminus in-in in-out ANP Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4W 2.7 Active DFGin‑BLAminus in-in in-in QYH Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A4W 2.7 Inactive DFGin‑BLAminus in-in in-out QYH Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A55 2.2 Active DFGin‑BLAminus in-in in-in QZ2 Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A55 2.2 Inactive DFGin‑BLAminus in-in in-out QZ2 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A5B 2.6 Active DFGin‑BLAminus in-in in-in MFR Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7A5B 2.6 Inactive DFGin‑BLAminus in-in in-out MFR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7O7K 1.82 Inactive DFGin‑BLAminus in-in in-out 6ZV, LI Type1, Allosteric 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7O7K 1.82 Inactive DFGin‑BLAminus in-in in-out 6ZV, LI Type1, Allosteric 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 135 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3Q 2.32 Active DFGin‑BLAminus in-in in-in RUT Type1.5_Back 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
8C3Q 2.32 Active DFGin‑BLAminus in-in in-in RUT Type1.5_Back 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6EIJ 2.42 Inactive DFGin‑BLAminus in-in in-out B5Z Type1.5_Front 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A
6UIP 3.7 Inactive DFGin‑None in-in in-in Q8J Type1 131 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A

CMGC_DYRK1A (Dual specificity tyrosine-phosphorylation-regulated kinase 1A)

Total number of chains: 230
Spatial label Dihedral label Number of Chains Representative
DFGin BLAminus 226 AF-Q13627-K1A
DFGin ABAminus 3 9KRJA
DFGin None 1 6UIPA

Database table as tsv

UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
DYR1A_HUMAN 6UIP 3.7 Inactive DFGin‑ABAminus in-in in-in Q8J Type1 136 - 478 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6UIP 3.7 Inactive DFGin‑ABAminus in-in none-out Q8J Type1 131 - 477 9 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN AF-Q13627-K1 -1.0 Active DFGin‑BLAminus in-in in-in No_ligand No_ligand 151 - 487 0 None None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN AF-Q13627-K3 -1.0 Active DFGin‑BLAminus in-in in-in No_ligand No_ligand 151 - 487 0 None None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6T6A 2.8 Active DFGin‑BLAminus in-in in-in No_ligand No_ligand 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIL 2.465 Inactive DFGin‑BLAminus in-in in-out No_ligand No_ligand 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6LN1 2.699 Active DFGin‑BLAminus in-in in-in EKU Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6LN1 2.699 Active DFGin‑BLAminus in-in in-in EKU Type1 140 - 479 4 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4R 1.8 Active DFGin‑BLAminus in-in in-in QY8 Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4R 1.8 Active DFGin‑BLAminus in-in in-in QY8 Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A52 2.1 Inactive DFGin‑BLAminus in-in in-out QYB Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A52 2.1 Active DFGin‑BLAminus in-in in-in QYB Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJM 2.4 Active DFGin‑BLAminus in-in in-in RKW Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJM 2.4 Active DFGin‑BLAminus in-in in-in RKW Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJS 2.15 Active DFGin‑BLAminus in-in in-in RKH Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJS 2.15 Active DFGin‑BLAminus in-in in-in RKH Type1 148 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7OY6 2.38 Inactive DFGin‑BLAminus in-in in-out 39I Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4S 3.1 Active DFGin‑BLAminus in-in in-in QYE Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4Z 1.9 Active DFGin‑BLAminus in-in in-in 6SD Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A51 1.9 Active DFGin‑BLAminus in-in in-in QYK Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A53 2.2 Active DFGin‑BLAminus in-in in-in QYZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A53 2.2 Active DFGin‑BLAminus in-in in-in QYZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A5D 1.8 Active DFGin‑BLAminus in-in in-in QYW Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A5L 2.1 Active DFGin‑BLAminus in-in in-in QZW Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A5N 2.3 Active DFGin‑BLAminus in-in in-in R05 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A5N 2.3 Active DFGin‑BLAminus in-in in-in R05 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJ2 2.1 Active DFGin‑BLAminus in-in in-in RJ5 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJ4 2.0 Active DFGin‑BLAminus in-in in-in RHZ Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJ5 2.0 Active DFGin‑BLAminus in-in in-in RHW Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJ7 2.9 Active DFGin‑BLAminus in-in in-in RHT Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJ8 2.0 Active DFGin‑BLAminus in-in in-in RJ8 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJA 2.2 Active DFGin‑BLAminus in-in in-in RJ2 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJV 2.1 Inactive DFGin‑BLAminus in-in in-out RKK Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJV 2.1 Inactive DFGin‑BLAminus in-in in-out RKK Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJW 2.8 Active DFGin‑BLAminus in-in in-in RKQ Type1 149 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJY 2.2 Inactive DFGin‑BLAminus in-in in-out RKZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AJY 2.2 Inactive DFGin‑BLAminus in-in in-out RKZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AK2 2.1 Inactive DFGin‑BLAminus in-in in-out RHH Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AK2 2.1 Inactive DFGin‑BLAminus in-in in-out RHH Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKA 1.9 Inactive DFGin‑BLAminus in-in in-out RK2 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKA 1.9 Inactive DFGin‑BLAminus in-in in-out RK2 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKB 2.8 Inactive DFGin‑BLAminus in-in in-out RJZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKB 2.8 Inactive DFGin‑BLAminus in-in in-out RJZ Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKE 2.3 Inactive DFGin‑BLAminus in-in in-out RK8 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKE 2.3 Inactive DFGin‑BLAminus in-in in-out RK8 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7AKL 2.0 Active DFGin‑BLAminus in-in in-in RK5 Type1 148 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6A1F 1.5 Active DFGin‑BLAminus in-in in-in 9OF Type1 134 - 483 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6A1G 2.15 Active DFGin‑BLAminus in-in in-in 9OL Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6A1G 2.15 Active DFGin‑BLAminus in-in in-in 9OL Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8YEV 2.252 Active DFGin‑BLAminus in-in in-in CUE Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8YEV 2.252 Active DFGin‑BLAminus in-in in-in CUE Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ1 2.35 Active DFGin‑BLAminus in-in in-in 2C3 Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ2 2.8 Active DFGin‑BLAminus in-in in-in 2C4 Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ2 2.8 Active DFGin‑BLAminus in-in in-in 2C4 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ2 2.8 Active DFGin‑BLAminus in-in in-in 2C4 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4MQ2 2.8 Inactive DFGin‑BLAminus in-in in-out 2C4 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YLJ 2.58 Active DFGin‑BLAminus in-in in-in 4E1 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YLK 1.4 Active DFGin‑BLAminus in-in in-in 4E2 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YLL 1.4 Active DFGin‑BLAminus in-in in-in 4E3 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4YU2 2.9 Active DFGin‑BLAminus in-in in-in 4H5 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6QU2 2.9 Active DFGin‑BLAminus in-in in-in JHW Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S11 2.445 Active DFGin‑BLAminus in-in in-in KQE Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S11 2.445 None DFGin‑BLAminus in-in in-none KQE Type1 136 - 480 3 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S14 1.05 Active DFGin‑BLAminus in-in in-in KQW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S17 1.1 Active DFGin‑BLAminus in-in in-in KQK Type1 134 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1B 1.3 Active DFGin‑BLAminus in-in in-in KRQ Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1H 1.05 Active DFGin‑BLAminus in-in in-in KQZ Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 1 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1I 2.38 Active DFGin‑BLAminus in-in in-in KR8 Type1 135 - 481 1 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6S1J 1.408 Active DFGin‑BLAminus in-in in-in KRK Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6T6A 2.8 Active DFGin‑BLAminus in-in in-in MLW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6T6A 2.8 Active DFGin‑BLAminus in-in in-in MLW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6T6A 2.8 Active DFGin‑BLAminus in-in in-in MLW Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6UWY 2.95 Active DFGin‑BLAminus in-in in-in QKG Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8R8E 2.22 Inactive DFGin‑BLAminus in-in in-out YOX Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8R8E 2.22 Active DFGin‑BLAminus in-in in-in YOX Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8R8E 2.22 Active DFGin‑BLAminus in-in in-in YOX Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8R8E 2.22 Active DFGin‑BLAminus in-in in-in YOX Type1 135 - 480 0 None None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHS 2.42 Inactive DFGin‑BLAminus in-in in-out 4VZ Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHS 2.42 Active DFGin‑BLAminus in-in in-in 4VZ Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHS 2.42 Inactive DFGin‑BLAminus in-in in-out 4VZ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHS 2.42 Inactive DFGin‑BLAminus in-in in-out 4VZ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7FHT 2.68 Inactive DFGin‑BLAminus in-in in-out 4WD Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8T2H 1.85 Active DFGin‑BLAminus in-in in-in XIR Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8T2H 1.85 Active DFGin‑BLAminus in-in in-in XIR Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 9CY5 2.49 Active DFGin‑BLAminus in-in in-in A1A04 Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 9CY5 2.49 Active DFGin‑BLAminus in-in in-in A1A04 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANQ 2.6 Inactive DFGin‑BLAminus in-in in-out EHB Type1 136 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANR 2.6 Active DFGin‑BLAminus in-in in-in HRM Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANR 2.6 Inactive DFGin‑BLAminus in-in in-out HRM Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANR 2.6 Inactive DFGin‑BLAminus in-in in-out HRM Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 3ANR 2.6 Inactive DFGin‑BLAminus in-in in-out HRM Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 134 - 479 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4NCT 2.597 Inactive DFGin‑BLAminus in-in in-out 2K2 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A3X 2.26 Inactive DFGin‑BLAminus in-in in-out QIV Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4E 2.68 Active DFGin‑BLAminus in-in in-in 7QQ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4E 2.68 Active DFGin‑BLAminus in-in in-in 7QQ Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4E 2.68 Inactive DFGin‑BLAminus in-out in-out 7QQ Type1 134 - 473 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4E 2.68 Active DFGin‑BLAminus in-in in-in 7QQ Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4L 2.73 Active DFGin‑BLAminus in-in in-in ZC3 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4L 2.73 Inactive DFGin‑BLAminus in-in in-out ZC3 Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4L 2.73 Inactive DFGin‑BLAminus in-in out-out ZC3 Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4L 2.73 Active DFGin‑BLAminus in-in in-in ZC3 Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4Q 2.37 Inactive DFGin‑BLAminus in-in in-out Y3L Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4Q 2.37 Active DFGin‑BLAminus in-in in-in Y3L Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4Q 2.37 Inactive DFGin‑BLAminus in-in in-out Y3L Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4Q 2.37 Active DFGin‑BLAminus in-in in-in Y3L Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4T 2.15 Active DFGin‑BLAminus in-in in-in AJG Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4T 2.15 Active DFGin‑BLAminus in-in in-in AJG Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4T 2.15 Inactive DFGin‑BLAminus in-in in-out AJG Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A4T 2.15 Active DFGin‑BLAminus in-in in-in AJG Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A54 2.63 Active DFGin‑BLAminus in-in in-in 5PW Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A54 2.63 Active DFGin‑BLAminus in-in in-in 5PW Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A54 2.63 Inactive DFGin‑BLAminus in-in in-out 5PW Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5A54 2.63 Active DFGin‑BLAminus in-in in-in 5PW Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIF 2.22 Active DFGin‑BLAminus in-in in-in B5T Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIF 2.22 Inactive DFGin‑BLAminus in-in in-out B5T Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIF 2.22 Inactive DFGin‑BLAminus in-in in-out B5T Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIF 2.22 Inactive DFGin‑BLAminus in-in in-out B5T Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIJ 2.42 Inactive DFGin‑BLAminus in-out in-in B5Z Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIJ 2.42 Active DFGin‑BLAminus in-in in-in B5Z Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIJ 2.42 Active DFGin‑BLAminus in-in in-in B5Z Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIL 2.465 Active DFGin‑BLAminus in-in in-in B6B Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIL 2.465 Inactive DFGin‑BLAminus in-in in-out B6B Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIL 2.465 Inactive DFGin‑BLAminus in-in in-out B6B Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIP 2.56 Inactive DFGin‑BLAminus in-out in-in B7B Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIP 2.56 Active DFGin‑BLAminus in-in in-in B7B Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIP 2.56 Inactive DFGin‑BLAminus in-in in-out B7B Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIP 2.56 Active DFGin‑BLAminus in-in in-in B7B Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIQ 2.3 Inactive DFGin‑BLAminus in-in in-out B6Z Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIQ 2.3 Inactive DFGin‑BLAminus in-in in-out B6Z Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIQ 2.3 Inactive DFGin‑BLAminus in-in in-out B6Z Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIQ 2.3 Active DFGin‑BLAminus in-in in-in B6Z Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIR 2.4 Inactive DFGin‑BLAminus in-in in-out B6H Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIS 2.36 Inactive DFGin‑BLAminus in-in in-out B6N Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIS 2.36 Active DFGin‑BLAminus in-in in-in B6N Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIS 2.36 Inactive DFGin‑BLAminus in-in in-out B6N Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIS 2.36 Active DFGin‑BLAminus in-in in-in B6N Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIV 2.68 Inactive DFGin‑BLAminus in-in in-out B6Q Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EJ4 2.88 Inactive DFGin‑BLAminus in-out in-out B7W Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EJ4 2.88 Inactive DFGin‑BLAminus in-in in-out B7W Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EJ4 2.88 Active DFGin‑BLAminus in-in in-in B7W Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EJ4 2.88 Inactive DFGin‑BLAminus in-in in-out B7W Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6YF8 3.198 Active DFGin‑BLAminus in-in in-in OPW Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6YF8 3.198 Active DFGin‑BLAminus in-in in-in OPW Type1 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6YF8 3.198 Inactive DFGin‑BLAminus in-in in-out OPW Type1 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6YF8 3.198 Active DFGin‑BLAminus in-in in-in OPW Type1 134 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 Active DFGin‑BLAminus in-in in-in 3NG Type1 137 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7Z5N 2.77 None DFGin‑BLAminus in-in in-none 3NG Type1 135 - 480 4 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3R 2.06 Active DFGin‑BLAminus in-in in-in R7O Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3R 2.06 Active DFGin‑BLAminus in-in in-in R7O Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3G 2.08 Active DFGin‑BLAminus in-in in-in QS0 Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 9FPX 2.69 Active DFGin‑BLAminus in-in in-in CC9 Type1 136 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 9FPX 2.69 Active DFGin‑BLAminus in-in in-in CC9 Type1 143 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 2VX3 2.4 Active DFGin‑BLAminus in-in in-in D15 Type1 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 2WO6 2.5 Active DFGin‑BLAminus in-in in-in D15 Type1 133 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 2WO6 2.5 Active DFGin‑BLAminus in-in in-in D15 Type1 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4AZE 3.15 Active DFGin‑BLAminus in-in in-in 3RA Type1 132 - 481 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4AZE 3.15 Active DFGin‑BLAminus in-in in-in 3RA Type1 135 - 481 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 4AZE 3.15 Active DFGin‑BLAminus in-in in-in 3RA Type1 132 - 481 0 X301,X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 5AIK 2.7 Active DFGin‑BLAminus in-in in-in AWR Type1 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4O 1.9 Active DFGin‑BLAminus in-in in-in ANP Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4O 1.9 Inactive DFGin‑BLAminus in-in in-out ANP Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4W 2.7 Active DFGin‑BLAminus in-in in-in QYH Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A4W 2.7 Inactive DFGin‑BLAminus in-in in-out QYH Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A55 2.2 Active DFGin‑BLAminus in-in in-in QZ2 Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A55 2.2 Inactive DFGin‑BLAminus in-in in-out QZ2 Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A5B 2.6 Active DFGin‑BLAminus in-in in-in MFR Type1 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7A5B 2.6 Inactive DFGin‑BLAminus in-in in-out MFR Type1 134 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7O7K 1.82 Inactive DFGin‑BLAminus in-in in-out 6ZV, LI Type1, Allosteric 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7O7K 1.82 Inactive DFGin‑BLAminus in-in in-out 6ZV, LI Type1, Allosteric 133 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 135 - 482 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 135 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 136 - 481 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 7ZH8 2.3 Active DFGin‑BLAminus in-in in-in IWU, IWU Type1, Allosteric 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3Q 2.32 Active DFGin‑BLAminus in-in in-in RUT Type1.5_Back 134 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 8C3Q 2.32 Active DFGin‑BLAminus in-in in-in RUT Type1.5_Back 136 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6EIJ 2.42 Inactive DFGin‑BLAminus in-in in-out B5Z Type1.5_Front 135 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_HUMAN 6UIP 3.7 Inactive DFGin‑None in-in in-in Q8J Type1 131 - 479 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Homo sapiens
DYR1A_MOUSE 9KRJ 3.0 Inactive DFGin‑ABAminus in-in in-in No_ligand No_ligand 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Mus musculus
DYR1A_MOUSE 9KRJ 3.0 Inactive DFGin‑BLAminus in-in in-out No_ligand No_ligand 136 - 480 2 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Mus musculus

CMGC_DYRK1A (Dual specificity tyrosine-phosphorylation-regulated kinase 1A)

Total number of chains: 2
Spatial label Dihedral label Number of Chains Representative
DFGin BLAminus 1 9KRJB
DFGin ABAminus 1 9KRJA

Database table as tsv

UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
DYR1A_MOUSE 9KRJ 3.0 Inactive DFGin‑ABAminus in-in in-in No_ligand No_ligand 135 - 480 0 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Mus musculus
DYR1A_MOUSE 9KRJ 3.0 Inactive DFGin‑BLAminus in-in in-out No_ligand No_ligand 136 - 480 2 X321 None Dual specificity tyrosine-phosphorylation-regulated kinase 1A Mus musculus