PDB: 4RIW — 2 kinases

Total number of chains: 4
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLBplus 2 50.0% 4RIWC
DFGin None 2 50.0% 4RIWD

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
TYR EGFR EGFR_HUMAN 4RIWB 3.1 Inactive DFGin‑None in-in in-none TYR APEdihe_nniai APEdist_aaai ADP ATPlike 688 - 984 0 None V948R,F997A,L1001A Epidermal growth factor receptor
TYR EGFR EGFR_HUMAN 4RIWD 3.1 Inactive DFGin‑None in-in in-in TYR APEdihe_iiiai APEdist_aaai ADP ATPlike 688 - 984 0 None V948R,F997A,L1001A Epidermal growth factor receptor
TYR ERBB3 ERBB3_HUMAN 4RIWA 3.1 Pseudo DFGin‑BLBplus out-na out-none TYR APEdihe_nnnai APEdist_aaan ANP ATPlike 699 - 979 0 None None Receptor tyrosine-protein kinase erbB-3
TYR ERBB3 ERBB3_HUMAN 4RIWC 3.1 Pseudo DFGin‑BLBplus out-na out-out TYR APEdihe_oioai APEdist_aaao ANP ATPlike 699 - 979 0 None None Receptor tyrosine-protein kinase erbB-3

PDB: 4RIW — 2 kinases

Total number of chains: 4
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLBplus 2 50.0% 4RIWC
DFGin None 2 50.0% 4RIWD

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TYR EGFR EGFR_HUMAN 4RIWB 3.1 Inactive DFGin‑None in-in in-none TYR APEdihe_nniai APEdist_aaai ADP ATPlike 688 - 984 0 None V948R,F997A,L1001A Epidermal growth factor receptor Homo sapiens
TYR EGFR EGFR_HUMAN 4RIWD 3.1 Inactive DFGin‑None in-in in-in TYR APEdihe_iiiai APEdist_aaai ADP ATPlike 688 - 984 0 None V948R,F997A,L1001A Epidermal growth factor receptor Homo sapiens
TYR ERBB3 ERBB3_HUMAN 4RIWA 3.1 Pseudo DFGin‑BLBplus out-na out-none TYR APEdihe_nnnai APEdist_aaan ANP ATPlike 699 - 979 0 None None Receptor tyrosine-protein kinase erbB-3 Homo sapiens
TYR ERBB3 ERBB3_HUMAN 4RIWC 3.1 Pseudo DFGin‑BLBplus out-na out-out TYR APEdihe_oioai APEdist_aaao ANP ATPlike 699 - 979 0 None None Receptor tyrosine-protein kinase erbB-3 Homo sapiens

PDB: 4RIW — 2 kinases

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism