Ligand: STI (Imatinib)

Total number of chains: 26
Active chains: 1
Total number of genes: 9
Spatial label Dihedral label Number of Chains Percent Representative
DFGout BBAminus 21 80.8% 8S16A
DFGin BLAminus 2 7.7% 7N9GB
DFGinter None 2 7.7% 7N9GA
DFGout None 1 3.8% 3HECA

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
CMGC MAPK14 MK14_HUMAN 3HECA 2.5 Inactive DFGout‑None in-in none-out nonTYR APEdihe_aaoii APEdist_nnno STI Type2 5 - 352 0 None None Mitogen-activated protein kinase 14
TYR ABL1 ABL1_HUMAN 7N9GB 2.2 Active DFGin‑BLAminus in-in in-in TYR APEdihe_iiiai APEdist_aaai STI, 1N1 Allosteric, Type1 233 - 498 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 7N9GA 2.2 Inactive DFGinter‑None in-out out-none TYR APEdihe_nniai APEdist_aaai STI, 1N1 Allosteric, Type1 233 - 498 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 7N9GC 2.2 Inactive DFGinter‑None in-none out-none TYR APEdihe_nniai APEdist_aaai STI, 1N1 Allosteric, Type1 234 - 499 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 2HYYA 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 235 - 498 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 2HYYB 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 233 - 498 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 2HYYC 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 233 - 498 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 2HYYD 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 233 - 498 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 3PYYA 1.85 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, 3YY Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 3PYYB 1.85 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_iiiai APEdist_aaao STI, 3YY Type2, Allosteric 233 - 510 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 6NPEA 2.15 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, KWD Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 6NPEB 2.15 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nniai APEdist_aaai STI, KWD Type2, Allosteric 233 - 511 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 6NPUA 2.33 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, KWV Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 6NPUB 2.33 Inactive DFGout‑BBAminus in-in none-in TYR APEdihe_iiiai APEdist_aaai STI, KWV Type2, Allosteric 233 - 510 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 6NPVA 1.86 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, KWP Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1
TYR ABL1 ABL1_HUMAN 6NPVB 1.86 Inactive DFGout‑BBAminus in-in none-in TYR APEdihe_iiiai APEdist_aaai STI, KWP Type2, Allosteric 233 - 510 0 None None Tyrosine-protein kinase ABL1
TYR ABL2 ABL2_HUMAN 3GVUA 2.05 Inactive DFGout‑BBAminus in-in out-none TYR APEdihe_niiai APEdist_aaai STI, STI Type2, Allosteric 279 - 546 0 None None Tyrosine-protein kinase ABL2
TYR CSF1R CSF1R_HUMAN 4R7IA 2.75 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 567 - 914 0 None C667T,C830S,C907T Macrophage colony-stimulating factor 1 receptor
TYR DDR1 DDR1_HUMAN 4BKJA 1.7 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 601 - 913 0 None None Epithelial discoidin domain-containing receptor 1
TYR DDR1 DDR1_HUMAN 4BKJB 1.7 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 601 - 913 0 None None Epithelial discoidin domain-containing receptor 1
TYR KIT KIT_HUMAN 8S16A 1.85 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 566 - 932 0 None I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D Mast/stem cell growth factor receptor Kit
TYR KIT KIT_HUMAN 8S16B 1.85 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 578 - 931 0 None I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D Mast/stem cell growth factor receptor Kit
TYR KIT KIT_HUMAN 1T46A 1.6 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 565 - 933 0 None None Mast/stem cell growth factor receptor Kit
TYR LCK LCK_HUMAN 2PL0A 2.8 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 231 - 498 0 None None Tyrosine-protein kinase Lck
TYR PDGFRA PGFRA_HUMAN 6JOLA 1.9 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 583 - 957 0 None None Platelet-derived growth factor receptor alpha
TYR SYK KSYK_HUMAN 1XBBA 1.57 None DFGin‑BLAminus in-in in-none TYR APEdihe_niiai APEdist_aaai STI Type1 363 - 635 0 None None Tyrosine-protein kinase SYK

Ligand: STI (Imatinib)

Total number of chains: 45
Active chains: 1
Total number of genes: 10
Spatial label Dihedral label Number of Chains Percent Representative
DFGout BBAminus 40 88.9% 1OPJA
DFGin BLAminus 2 4.4% 7N9GB
DFGinter None 2 4.4% 7N9GA
DFGout None 1 2.2% 3HECA

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TYR SRC SRC_CHICK 3OEZA 2.4 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao STI Type2 257 - 533 0 None L317I Proto-oncogene tyrosine-protein kinase Src Gallus gallus
TYR SRC SRC_CHICK 3OEZB 2.4 Inactive DFGout‑BBAminus in-out none-out TYR APEdihe_nnoai APEdist_aaao STI Type2 256 - 533 0 None L317I Proto-oncogene tyrosine-protein kinase Src Gallus gallus
TYR SRC SRC_CHICK 2OIQA 2.07 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_iiiai APEdist_aaao STI Type2 256 - 533 0 None None Proto-oncogene tyrosine-protein kinase Src Gallus gallus
CMGC MAPK14 MK14_HUMAN 3HECA 2.5 Inactive DFGout‑None in-in none-out nonTYR APEdihe_aaoii APEdist_nnno STI Type2 5 - 352 0 None None Mitogen-activated protein kinase 14 Homo sapiens
TYR ABL1 ABL1_HUMAN 7N9GB 2.2 Active DFGin‑BLAminus in-in in-in TYR APEdihe_iiiai APEdist_aaai STI, 1N1 Allosteric, Type1 233 - 498 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 7N9GA 2.2 Inactive DFGinter‑None in-out out-none TYR APEdihe_nniai APEdist_aaai STI, 1N1 Allosteric, Type1 233 - 498 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 7N9GC 2.2 Inactive DFGinter‑None in-none out-none TYR APEdihe_nniai APEdist_aaai STI, 1N1 Allosteric, Type1 234 - 499 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 2HYYA 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 235 - 498 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 2HYYB 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 233 - 498 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 2HYYC 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 233 - 498 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 2HYYD 2.4 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 233 - 498 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 3PYYA 1.85 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, 3YY Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 3PYYB 1.85 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_iiiai APEdist_aaao STI, 3YY Type2, Allosteric 233 - 510 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 6NPEA 2.15 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, KWD Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 6NPEB 2.15 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nniai APEdist_aaai STI, KWD Type2, Allosteric 233 - 511 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 6NPUA 2.33 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, KWV Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 6NPUB 2.33 Inactive DFGout‑BBAminus in-in none-in TYR APEdihe_iiiai APEdist_aaai STI, KWV Type2, Allosteric 233 - 510 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 6NPVA 1.86 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, KWP Type2, Allosteric 232 - 500 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL1 ABL1_HUMAN 6NPVB 1.86 Inactive DFGout‑BBAminus in-in none-in TYR APEdihe_iiiai APEdist_aaai STI, KWP Type2, Allosteric 233 - 510 0 None None Tyrosine-protein kinase ABL1 Homo sapiens
TYR ABL2 ABL2_HUMAN 3GVUA 2.05 Inactive DFGout‑BBAminus in-in out-none TYR APEdihe_niiai APEdist_aaai STI, STI Type2, Allosteric 279 - 546 0 None None Tyrosine-protein kinase ABL2 Homo sapiens
TYR CSF1R CSF1R_HUMAN 4R7IA 2.75 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 567 - 914 0 None C667T,C830S,C907T Macrophage colony-stimulating factor 1 receptor Homo sapiens
TYR DDR1 DDR1_HUMAN 4BKJA 1.7 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 601 - 913 0 None None Epithelial discoidin domain-containing receptor 1 Homo sapiens
TYR DDR1 DDR1_HUMAN 4BKJB 1.7 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 601 - 913 0 None None Epithelial discoidin domain-containing receptor 1 Homo sapiens
TYR KIT KIT_HUMAN 8S16A 1.85 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 566 - 932 0 None I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D Mast/stem cell growth factor receptor Kit Homo sapiens
TYR KIT KIT_HUMAN 8S16B 1.85 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 578 - 931 0 None I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D Mast/stem cell growth factor receptor Kit Homo sapiens
TYR KIT KIT_HUMAN 1T46A 1.6 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 565 - 933 0 None None Mast/stem cell growth factor receptor Kit Homo sapiens
TYR LCK LCK_HUMAN 2PL0A 2.8 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 231 - 498 0 None None Tyrosine-protein kinase Lck Homo sapiens
TYR PDGFRA PGFRA_HUMAN 6JOLA 1.9 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 583 - 957 0 None None Platelet-derived growth factor receptor alpha Homo sapiens
TYR SYK KSYK_HUMAN 1XBBA 1.57 None DFGin‑BLAminus in-in in-none TYR APEdihe_niiai APEdist_aaai STI Type1 363 - 635 0 None None Tyrosine-protein kinase SYK Homo sapiens
TYR ABL1 ABL1_MOUSE 3K5VA 1.74 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STJ, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3K5VB 1.74 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STJ, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD4A 2.03 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai FYW, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD4B 2.03 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai FYW, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD6A 2.3 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai FYH, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1IEPA 2.1 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1IEPB 2.1 Inactive DFGout‑BBAminus in-out out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1OPJA 1.75 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao STI Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1OPJB 1.75 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 512 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD6B 2.3 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MS9A 1.8 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS9 Type2, Allosteric 230 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MS9B 1.8 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS9 Type2, Allosteric 229 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSA 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSB 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSC 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSD 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus

Ligand: STI (Imatinib)

Total number of chains: 19
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGout BBAminus 19 100.0% 1OPJA

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TYR SRC SRC_CHICK 3OEZA 2.4 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao STI Type2 257 - 533 0 None L317I Proto-oncogene tyrosine-protein kinase Src Gallus gallus
TYR SRC SRC_CHICK 3OEZB 2.4 Inactive DFGout‑BBAminus in-out none-out TYR APEdihe_nnoai APEdist_aaao STI Type2 256 - 533 0 None L317I Proto-oncogene tyrosine-protein kinase Src Gallus gallus
TYR SRC SRC_CHICK 2OIQA 2.07 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_iiiai APEdist_aaao STI Type2 256 - 533 0 None None Proto-oncogene tyrosine-protein kinase Src Gallus gallus
TYR ABL1 ABL1_MOUSE 3K5VA 1.74 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STJ, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3K5VB 1.74 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STJ, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD4A 2.03 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai FYW, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD4B 2.03 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai FYW, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD6A 2.3 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai FYH, STI Allosteric, Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1IEPA 2.1 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1IEPB 2.1 Inactive DFGout‑BBAminus in-out out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1OPJA 1.75 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao STI Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 1OPJB 1.75 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 512 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 6HD6B 2.3 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI Type2 229 - 510 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MS9A 1.8 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS9 Type2, Allosteric 230 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MS9B 1.8 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS9 Type2, Allosteric 229 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSA 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSB 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSC 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus
TYR ABL1 ABL1_MOUSE 3MSSD 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai STI, MS7 Type2, Allosteric 232 - 498 0 None None Tyrosine-protein kinase ABL1 Mus musculus