Ligand: T5L

Total number of chains: 8
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 8 100.0% 8C14A

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
CAMK AURKA AURKA_HUMAN 8C14A 1.93 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_iioo ADP, T5L, T0L ATPlike, Allosteric, Allosteric 126 - 389 0 TPO288 None Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C15A 2.41 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno ADP, T4C, T5L ATPlike, Allosteric, Allosteric 126 - 388 0 None C290A Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C1FA 1.924 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno ADP, T5L, T2O ATPlike, Allosteric, Allosteric 126 - 388 0 None C290A Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C1IA 2.81 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno ADP, T1L, T5L ATPlike, Allosteric, Allosteric 126 - 388 0 None C290A Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C1DA 2.115 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno T2F, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C1GA 1.96 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno T3I, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C1HA 2.233 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno T3U, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A
CAMK AURKA AURKA_HUMAN 8C1KA 2.43 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_iioo T4O, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A

Ligand: T5L

Total number of chains: 8
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 8 100.0% 8C14A

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
CAMK AURKA AURKA_HUMAN 8C14A 1.93 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_iioo ADP, T5L, T0L ATPlike, Allosteric, Allosteric 126 - 389 0 TPO288 None Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C15A 2.41 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno ADP, T4C, T5L ATPlike, Allosteric, Allosteric 126 - 388 0 None C290A Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C1FA 1.924 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno ADP, T5L, T2O ATPlike, Allosteric, Allosteric 126 - 388 0 None C290A Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C1IA 2.81 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno ADP, T1L, T5L ATPlike, Allosteric, Allosteric 126 - 388 0 None C290A Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C1DA 2.115 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno T2F, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C1GA 1.96 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno T3I, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C1HA 2.233 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_nnno T3U, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A Homo sapiens
CAMK AURKA AURKA_HUMAN 8C1KA 2.43 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_iioo T4O, ADP, T5L Allosteric, ATPlike, Allosteric 127 - 388 0 None C290A Aurora kinase A Homo sapiens

Ligand: T5L

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism