| PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 4YHJA | 2.6 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | AN2 | ATPlike | 25 - 525 | 0 | None | C563S,C578S | G protein-coupled receptor kinase 4 |
| 4YHJB | 2.6 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | AN2 | ATPlike | 25 - 527 | 0 | None | C563S,C578S | G protein-coupled receptor kinase 4 |
| AF-P32298-K1A | -1.0 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | No_ligand | No_ligand | 179 - 457 | 0 | None | None | G protein-coupled receptor kinase 4 |
| AF-P32298-K3A | -1.0 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | No_ligand | No_ligand | 179 - 457 | 0 | None | None | G protein-coupled receptor kinase 4 |
| UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK4_HUMAN | 4YHJA | 2.6 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | AN2 | ATPlike | 25 - 525 | 0 | None | C563S,C578S | G protein-coupled receptor kinase 4 | Homo sapiens |
| GRK4_HUMAN | 4YHJB | 2.6 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | AN2 | ATPlike | 25 - 527 | 0 | None | C563S,C578S | G protein-coupled receptor kinase 4 | Homo sapiens |
| GRK4_HUMAN | AF-P32298-K1A | -1.0 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | No_ligand | No_ligand | 179 - 457 | 0 | None | None | G protein-coupled receptor kinase 4 | Homo sapiens |
| GRK4_HUMAN | AF-P32298-K3A | -1.0 | Active | DFGin‑BLAminus | in-in | in-in | nonTYR | APEdihe_aaiii | APEdist_iiii | No_ligand | No_ligand | 179 - 457 | 0 | None | None | G protein-coupled receptor kinase 4 | Homo sapiens |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|