All / Activity_Active / ATPlike

Total number of chains: 178
Active chains: 178
Total number of genes: 55
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 178 100.0% 8QCGB

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AGC AKT1 AKT1_HUMAN 4EKKA P31749 144 477 480.0 ANP:60501 ATPlike Active DFGin 6.048 13.113 BLAminus -112.5, -177.27 66.46, 90.66 -111.95, 23.34 296.26, 86.16 -69.26, -23.9 in-in in 8.651 Saltbr-in 2.978 HRD-in -63.51, -40.13 66.5, -18.58 in-in-in SNCiii in-in ActLoopNT-in 3.05 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.71, 172.01 APE9-dihe-na 121.09, -152.4 APE8-dihe-in -119.32, 125.09 APE8-rot-in 285.38 APE67-dihe-in -63.61, -25.53 -44.69, -42.52 APE12-dist-in 8.814 APE11-dist-in 11.718 APE10-dist-in 6.07 APE9-dist-in 4.069 S473D TPO308 TPO308 XRAY 2.8 0.22 0.28 A 341 319 0 0 0 0 [[150, 408]] 1.0 4ekk AGC_AKT1_HUMAN AGC 2.3e-99 337.7 1 260 260 291 292 293 295 297 179 198 202 271 273 272 274 331 319 314 313 312 311 310 309 308 228 RAC-alpha serine/threonine-protein kinase
AGC AKT1 AKT1_HUMAN 4EKKB P31749 144 477 480.0 ANP:60501 ATPlike Active DFGin 6.075 13.046 BLAminus -112.98, 175.61 60.18, 117.01 -127.72, 18.67 304.81, 92.19 -54.85, -36.32 in-in in 8.766 Saltbr-in 2.665 HRD-in -65.56, -47.0 73.75, -27.2 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.2, 164.76 APE9-dihe-na 136.6, -155.35 APE8-dihe-in -114.57, 129.15 APE8-rot-in 273.31 APE67-dihe-in -63.86, -22.96 -45.74, -46.48 APE12-dist-in 8.77 APE11-dist-in 11.686 APE10-dist-in 6.125 APE9-dist-in 4.285 S473D TPO308 TPO308 XRAY 2.8 0.22 0.28 B 341 319 0 0 0 0 [[150, 408]] 1.0 4ekk AGC_AKT1_HUMAN AGC 2.3e-99 337.7 1 260 260 291 292 293 295 297 179 198 202 271 273 272 274 331 319 314 313 312 311 310 309 308 228 RAC-alpha serine/threonine-protein kinase
AGC AKT2 AKT2_HUMAN 1O6KA P31751 146 479 481.0 ANP:1480 ATPlike Active DFGin 6.146 12.734 BLAminus -120.8, -176.05 56.87, 82.9 -98.82, 24.49 299.36, 92.56 -61.37, -25.29 in-in in 8.749 Saltbr-in 2.796 HRD-in -73.34, -45.79 65.54, -9.2 in-in-in SNCiii in-in ActLoopNT-in 3.027 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.85, 170.7 APE9-dihe-na 130.02, -155.15 APE8-dihe-in -119.36, 127.57 APE8-rot-in 291.96 APE67-dihe-in -68.55, -16.48 -36.55, -56.12 APE12-dist-in 8.193 APE11-dist-in 11.759 APE10-dist-in 6.119 APE9-dist-in 3.921 S474D TPO309 TPO309 XRAY 1.7 0.205 0.234 A 336 318 0 0 0 0 [[152, 409]] 1.0 1o6k AGC_AKT2_HUMAN AGC 1.7e-99 338.1 1 260 260 292 293 294 296 298 181 200 204 272 274 273 275 332 320 315 314 313 312 311 310 309 230 RAC-beta serine/threonine-protein kinase
AGC AKT2 AKT2_HUMAN 1O6LA P31751 146 477 481.0 ANP:61480 ATPlike Active DFGin 6.258 12.925 BLAminus -121.53, -178.18 58.41, 83.34 -98.83, 24.71 297.57, 89.85 -63.5, -19.94 in-in in 8.794 Saltbr-in 2.76 HRD-in -74.06, -43.29 62.88, -5.6 in-in-in SNCiii in-in ActLoopNT-in 3.006 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.79, 169.91 APE9-dihe-na 133.49, -153.33 APE8-dihe-in -120.8, 127.55 APE8-rot-in 289.07 APE67-dihe-in -68.04, -17.15 -37.13, -54.04 APE12-dist-in 8.173 APE11-dist-in 11.74 APE10-dist-in 6.122 APE9-dist-in 3.747 None TPO309 TPO309 XRAY 1.6 0.198 0.227 A 337 312 0 0 0 0 [[152, 409]] 1.0 1o6l AGC_AKT2_HUMAN AGC 1.8e-99 338.1 1 260 260 292 293 294 296 298 181 200 204 272 274 273 275 332 320 315 314 313 312 311 310 309 230 RAC-beta serine/threonine-protein kinase
AGC CDC42BPB MRCKB_HUMAN 4UAKA Q9Y5S2 2 417 1711.0 ADP:60501 ATPlike Active DFGin 6.536 13.389 BLAminus -126.67, 169.91 71.43, 81.15 -99.11, 14.11 300.02, 102.96 -73.12, -5.53 in-in in 8.635 Saltbr-in 2.748 HRD-in -78.82, -49.28 69.95, 4.01 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.28, 157.85 APE9-dihe-na 87.21, -164.86 APE8-dihe-in -127.15, 132.61 APE8-rot-in 302.21 APE67-dihe-in -64.23, -20.61 -57.86, -36.49 APE12-dist-in 10.511 APE11-dist-in 11.151 APE10-dist-in 6.313 APE9-dist-in 3.548 None None None XRAY 1.73 0.198 0.243 A 419 401 0 0 0 0 [[76, 342]] 1.0 4uak AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
AGC GRK4 GRK4_HUMAN 4YHJA P32298 25 525 578.0 AN2:601 ATPlike Active DFGin 6.129 13.374 BLAminus -118.16, -176.89 50.04, 69.58 -89.94, 31.88 285.36, 98.48 -66.46, -45.19 in-in in 9.266 Saltbr-in 3.026 HRD-in -63.35, -45.97 74.46, -21.42 in-in-in SNCiii in-in ActLoopNT-in 2.855 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.22, 157.81 APE9-dihe-na 113.97, -154.87 APE8-dihe-in -108.33, 139.74 APE8-rot-in 312.15 APE67-dihe-inflip 104.58, -18.92 -61.34, 124.85 APE12-dist-in 11.453 APE11-dist-in 12.888 APE10-dist-in 6.916 APE9-dist-in 4.145 C563S,C578S None None XRAY 2.6 0.2 0.248 A 584 501 0 0 0 0 [[187, 449]] 1.0 4yhj AGC_GRK4_HUMAN AGC 8.1e-84 286.9 1 260 260 329 330 331 333 335 216 235 239 309 311 310 312 368 356 351 350 349 348 347 346 345 265 G protein-coupled receptor kinase 4
AGC GRK4 GRK4_HUMAN 4YHJB P32298 25 527 578.0 AN2:601 ATPlike Active DFGin 6.038 13.172 BLAminus -128.85, 178.91 61.8, 67.7 -94.52, 28.72 287.39, 101.3 -65.66, -45.87 in-in in 9.016 Saltbr-in 3.179 HRD-in -66.59, -45.54 76.27, -17.2 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.9, 153.12 APE9-dihe-na 125.18, -147.1 APE8-dihe-in -118.5, 134.63 APE8-rot-in 298.66 APE67-dihe-inflip 107.33, -19.99 -54.96, 119.79 APE12-dist-in 11.128 APE11-dist-in 12.752 APE10-dist-in 6.774 APE9-dist-in 3.816 C563S,C578S None None XRAY 2.6 0.2 0.248 B 584 490 0 0 0 0 [[187, 449]] 1.0 4yhj AGC_GRK4_HUMAN AGC 8.1e-84 286.9 1 260 260 329 330 331 333 335 216 235 239 309 311 310 312 368 356 351 350 349 348 347 346 345 265 G protein-coupled receptor kinase 4
AGC GRK5 GRK5_HUMAN 4TNDA P34947 15 543 590.0 ANP:601 ATPlike Active DFGin 5.282 13.172 BLAminus -119.9, 173.82 59.88, 73.64 -89.53, 7.87 278.21, 112.8 -54.71, -33.69 in-in in 9.193 Saltbr-in 3.053 HRD-in -67.8, -56.87 74.64, -6.61 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.25, 150.21 APE9-dihe-na 143.02, -165.26 APE8-dihe-in -107.11, 142.28 APE8-rot-in 314.69 APE67-dihe-inflip 92.64, -22.22 -59.58, 132.94 APE12-dist-in 10.302 APE11-dist-in 12.056 APE10-dist-in 6.23 APE9-dist-in 4.255 None None None XRAY 1.802 0.174 0.205 A 590 529 0 0 0 0 [[186, 448]] 1.0 4tnd AGC_GRK5_HUMAN AGC 1.1e-83 286.4 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 5
AGC GRK5 GRK5_HUMAN 9CKRA P34947 25 542 590.0 ATP:603 ATPlike Active DFGin 6.172 12.867 BLAminus -123.04, 159.77 67.48, 80.75 -99.52, 5.04 278.7, 83.61 -52.63, -21.44 in-in in 8.589 Saltbr-in 3.447 HRD-in -94.88, -52.49 68.7, 5.59 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.66, 167.59 APE9-dihe-na 129.66, -152.54 APE8-dihe-in -119.66, 138.17 APE8-rot-in 320.31 APE67-dihe-inflip 80.19, -6.12 -54.38, 134.58 APE12-dist-in 9.872 APE11-dist-in 12.258 APE10-dist-in 6.529 APE9-dist-in 4.181 D311N None None XRAY 2.8 0.239 0.286 A 598 501 0 0 0 0 [[186, 448]] 1.0 9ckr AGC_GRK5_HUMAN AGC 7.6e-83 283.7 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 5
AGC GRK5 GRK5_HUMAN 9CKSA P34947 25 542 590.0 ATP:603 ATPlike Active DFGin 6.038 13.061 BLAminus -123.04, 167.6 79.98, 56.79 -87.17, 17.84 285.5, 62.72 -70.38, -31.79 in-in in 9.222 Saltbr-in 2.672 HRD-in -92.29, -53.7 68.73, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.24, 151.24 APE9-dihe-na 138.17, -158.29 APE8-dihe-in -117.35, 145.2 APE8-rot-in 310.61 APE67-dihe-inflip 85.98, -22.04 -53.6, 135.84 APE12-dist-in 10.616 APE11-dist-in 12.407 APE10-dist-in 6.563 APE9-dist-in 4.207 D311N None None XRAY 3.08 0.228 0.28 A 598 501 0 0 0 0 [[186, 448]] 1.0 9cks AGC_GRK5_HUMAN AGC 7.6e-83 283.7 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 5
AGC GRK6 GRK6_HUMAN 2ACXA P43250 14 532 576.0 ANP:577 ATPlike Active DFGin 6.207 13.284 BLAminus -133.82, 164.79 58.79, 76.03 -96.19, 24.41 281.42, 82.4 -59.68, -24.05 in-in in 9.341 Saltbr-in 3.219 HRD-in -78.26, -56.85 77.2, -1.95 in-in-in SNCiii in-in ActLoopNT-in 2.971 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.49, 157.4 APE9-dihe-na 123.02, -168.26 APE8-dihe-in -95.03, 140.31 APE8-rot-in 303.17 APE67-dihe-in -86.56, -0.13 -45.11, -52.69 APE12-dist-in 10.478 APE11-dist-in 11.834 APE10-dist-in 6.083 APE9-dist-in 3.906 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 A 576 495 0 0 0 0 [[186, 448]] 1.0 2acx AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC GRK6 GRK6_HUMAN 2ACXB P43250 14 535 576.0 ANP:577 ATPlike Active DFGin 6.09 13.146 BLAminus -128.37, 163.87 55.35, 87.14 -100.56, 21.26 285.61, 77.77 -55.4, -30.56 in-in in 9.231 Saltbr-in 2.439 HRD-in -77.3, -59.12 75.78, 1.97 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.83, 161.38 APE9-dihe-na 125.99, -167.44 APE8-dihe-in -95.89, 144.8 APE8-rot-in 307.19 APE67-dihe-in -70.72, -14.39 -48.06, -55.51 APE12-dist-in 10.477 APE11-dist-in 11.872 APE10-dist-in 6.167 APE9-dist-in 3.71 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 B 576 492 5 0 0 0 [[186, 448]] 1.0 2acx AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC GRK6 GRK6_HUMAN 3NYOA P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.423 12.986 BLAminus -150.32, 176.66 46.57, 93.99 -112.64, 27.92 269.12, 56.38 -53.19, -36.92 in-in in 8.492 Saltbr-in 3.133 HRD-in -67.42, -53.58 67.41, 17.23 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.58, 145.08 APE9-dihe-na 153.72, -154.4 APE8-dihe-in -119.63, 125.01 APE8-rot-in 309.24 APE67-dihe-inflip 99.19, -30.43 -48.0, 129.76 APE12-dist-in 10.102 APE11-dist-in 11.881 APE10-dist-in 6.152 APE9-dist-in 3.985 None None None XRAY 2.92 0.222 0.253 A 576 553 3 0 0 0 [[186, 448]] 1.0 3nyo AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC GRK6 GRK6_HUMAN 3NYOB P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.469 12.921 BLAminus -147.57, -176.88 49.48, 66.09 -89.42, 43.68 283.74, 78.16 -61.9, -48.01 in-in in 8.429 Saltbr-in 2.859 HRD-in -67.89, -44.49 63.77, 4.77 in-in-in SNCiii in-in ActLoopNT-in 2.959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.44, 138.67 APE9-dihe-na 143.94, 179.93 APE8-dihe-in -100.37, 135.53 APE8-rot-in 311.67 APE67-dihe-inflip 96.9, -39.59 -38.27, 126.0 APE12-dist-in 10.148 APE11-dist-in 11.731 APE10-dist-in 5.96 APE9-dist-in 3.734 None None None XRAY 2.92 0.222 0.253 B 576 553 3 0 0 0 [[186, 448]] 1.0 3nyo AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC PDPK1 PDPK1_HUMAN 2BIYA O15530 72 359 556.0 ATP:1373 ATPlike Active DFGin 6.619 15.095 BLAminus -141.33, -175.84 82.91, 67.67 -104.99, 1.58 283.05, 104.18 -61.63, -33.06 in-in in 8.673 Saltbr-in 2.575 HRD-in -63.52, -52.73 78.44, -11.09 in-in-in SNCiii in-in ActLoopNT-in 2.82 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.22, 130.12 APE9-dihe-na 106.71, 171.13 APE8-dihe-in -96.94, 126.07 APE8-rot-in 299.07 APE67-dihe-in -62.15, -19.51 -52.23, -44.36 APE12-dist-in 12.868 APE11-dist-in 12.869 APE10-dist-in 7.268 APE9-dist-in 4.745 S241A None None XRAY 1.95 0.186 0.23 A 310 288 0 0 0 0 [[82, 342]] 1.0 2biy AGC_PDPK1_HUMAN AGC 1.8e-84 288.8 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3HRCA O15530 76 359 556.0 ATP:1373 ATPlike Active DFGin 6.486 14.833 BLAminus -136.91, -178.17 71.81, 74.55 -104.54, 6.98 286.89, 102.51 -65.47, -24.41 in-in in 8.421 Saltbr-in 3.159 HRD-in -77.24, -54.93 76.93, -11.42 in-in-in SNCiii in-in ActLoopNT-in 2.87 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.25, 162.0 APE9-dihe-na 130.63, -171.63 APE8-dihe-in -125.01, 129.68 APE8-rot-in 292.48 APE67-dihe-in -58.92, -25.29 -45.32, -48.7 APE12-dist-in 7.409 APE11-dist-in 10.582 APE10-dist-in 4.926 APE9-dist-in 3.479 Y288G,Q292A SEP241 SEP241 XRAY 1.91 0.182 0.207 A 311 280 4 0 0 4 [[82, 342]] 1.0 3hrc AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 4RRVA O15530 76 359 556.0 ATP:60401 ATPlike Active DFGin 6.548 14.998 BLAminus -136.55, -175.99 74.63, 72.8 -106.52, 5.78 286.61, 100.18 -68.12, -17.88 in-in in 8.52 Saltbr-in 2.956 HRD-in -71.77, -54.29 78.75, -11.73 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.13, 162.83 APE9-dihe-na 132.08, -169.67 APE8-dihe-in -127.24, 132.02 APE8-rot-in 298.33 APE67-dihe-in -59.21, -24.3 -51.83, -46.04 APE12-dist-in 7.281 APE11-dist-in 10.502 APE10-dist-in 4.943 APE9-dist-in 3.569 Y288G,Q292A SEP241 SEP241 XRAY 1.412 0.135 0.163 A 311 284 0 0 0 0 [[82, 342]] 1.0 4rrv AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5ACKA O15530 73 359 556.0 ATP:500 ATPlike Active DFGin 6.615 14.861 BLAminus -135.34, 179.84 72.22, 79.01 -106.01, 4.14 287.93, 97.64 -67.02, -18.73 in-in in 8.418 Saltbr-in 2.583 HRD-in -74.68, -53.67 78.01, -12.73 in-in-in SNCiii in-in ActLoopNT-in 2.906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.4, 162.51 APE9-dihe-na 136.44, -168.07 APE8-dihe-in -132.35, 133.52 APE8-rot-in 296.36 APE67-dihe-in -62.96, -23.95 -54.34, -43.19 APE12-dist-in 7.326 APE11-dist-in 10.522 APE10-dist-in 4.978 APE9-dist-in 3.558 Y288G,Q292A SEP241 SEP241 XRAY 1.24 0.143 0.166 A 311 287 0 0 0 0 [[82, 342]] 1.0 5ack AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPA O15530 75 359 556.0 ATP:500 ATPlike Active DFGin 6.303 14.998 BLAminus -144.92, -168.82 66.06, 77.78 -108.23, 11.17 281.99, 93.22 -63.04, -32.41 in-in in 9.539 Saltbr-in 3.158 HRD-in -77.47, -51.83 79.92, -12.48 in-in-in SNCiii in-in ActLoopNT-in 2.848 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.64, 166.02 APE9-dihe-na 141.61, 177.5 APE8-dihe-in -123.02, 134.29 APE8-rot-in 296.02 APE67-dihe-in -68.65, -16.53 -46.89, -50.92 APE12-dist-in 7.907 APE11-dist-in 10.671 APE10-dist-in 5.166 APE9-dist-in 3.705 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 A 311 276 9 0 0 9 [[82, 342]] 1.0 5lvp AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPB O15530 74 359 556.0 ATP:401 ATPlike Active DFGin 6.328 14.55 BLAminus -137.23, -179.71 80.14, 74.16 -105.47, 15.38 295.0, 84.83 -59.91, -31.47 in-in in 9.274 Saltbr-in 3.302 HRD-in -80.68, -44.41 73.96, -16.23 in-in-in SNCiii in-in ActLoopNT-in 2.744 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.8, 152.43 APE9-dihe-na 134.43, -173.75 APE8-dihe-in -120.09, 128.28 APE8-rot-in 302.93 APE67-dihe-in -67.56, -25.72 -44.99, -47.55 APE12-dist-in 7.872 APE11-dist-in 11.011 APE10-dist-in 5.375 APE9-dist-in 3.787 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 B 311 277 9 0 0 9 [[82, 342]] 1.0 5lvp AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPC O15530 75 359 556.0 ATP:401 ATPlike Active DFGin 6.391 14.608 BLAminus -132.15, -176.81 71.98, 84.02 -116.53, 7.62 291.47, 90.46 -60.24, -24.5 in-in in 9.304 Saltbr-in 3.087 HRD-in -75.92, -52.06 78.45, -5.49 in-in-in SNCiii in-in ActLoopNT-in 2.823 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -113.81, 168.64 APE9-dihe-na 131.92, -176.79 APE8-dihe-in -126.79, 133.21 APE8-rot-in 299.13 APE67-dihe-in -67.64, -15.8 -51.62, -50.49 APE12-dist-in 7.652 APE11-dist-in 10.863 APE10-dist-in 5.123 APE9-dist-in 3.645 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 C 311 276 9 0 0 9 [[82, 342]] 1.0 5lvp AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPD O15530 74 359 556.0 ATP:500 ATPlike Active DFGin 6.334 14.433 BLAminus -146.99, -174.22 74.22, 81.56 -113.84, 4.02 287.97, 93.59 -56.11, -25.73 in-in in 9.304 Saltbr-in 3.252 HRD-in -82.38, -50.18 78.4, -12.51 in-in-in SNCiii in-in ActLoopNT-in 2.836 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.65, 165.17 APE9-dihe-na 129.1, -166.82 APE8-dihe-in -132.84, 129.79 APE8-rot-in 300.06 APE67-dihe-in -65.46, -17.03 -48.9, -48.47 APE12-dist-in 8.228 APE11-dist-in 10.891 APE10-dist-in 5.348 APE9-dist-in 3.646 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 D 311 277 9 0 0 9 [[82, 342]] 1.0 5lvp AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 4CT2A O15530 75 359 556.0 ATP:500 ATPlike Active DFGin 6.551 14.867 BLAminus -136.23, -174.98 70.54, 70.07 -102.02, 6.41 290.69, 95.78 -63.73, -21.59 in-in in 8.252 Saltbr-in 2.643 HRD-in -73.2, -54.84 77.37, -9.78 in-in-in SNCiii in-in ActLoopNT-in 2.965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.02, 163.59 APE9-dihe-na 137.39, -170.05 APE8-dihe-in -132.12, 131.72 APE8-rot-in 295.26 APE67-dihe-in -63.06, -17.27 -51.84, -45.87 APE12-dist-in 7.163 APE11-dist-in 10.524 APE10-dist-in 4.979 APE9-dist-in 3.527 L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A SEP241 SEP241 XRAY 1.25 0.194 0.226 A 311 280 5 0 0 0 [[82, 342]] 1.0 4ct2 AGC_PDPK1_HUMAN AGC 9.5e-84 286.4 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5MRDA O15530 76 359 556.0 ATP:405 ATPlike Active DFGin 6.429 14.7 BLAminus -133.69, -177.11 74.21, 73.9 -105.88, 9.0 289.39, 99.64 -68.32, -19.62 in-in in 8.346 Saltbr-in 2.667 HRD-in -74.32, -53.19 77.26, -10.58 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.86, 160.68 APE9-dihe-na 136.11, -166.87 APE8-dihe-in -131.1, 132.63 APE8-rot-in 296.36 APE67-dihe-in -62.36, -23.28 -53.02, -44.84 APE12-dist-in 7.352 APE11-dist-in 10.498 APE10-dist-in 4.91 APE9-dist-in 3.542 K76S,L113V,I118V,I119N,V124I,T128Q,R131K,T148C SEP241 SEP241 XRAY 1.41 0.142 0.174 A 310 284 0 0 0 0 [[82, 342]] 1.0 5mrd AGC_PDPK1_HUMAN AGC 1.7e-83 285.6 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PRKACA KAPCA_HUMAN 4WB8A P17612 16 351 351.0 ATP:60401 ATPlike Active DFGin 5.684 14.414 BLAminus -121.45, -177.2 62.67, 77.75 -91.98, 24.58 268.87, 53.09 -58.34, -31.51 in-in in 8.913 Saltbr-in 2.759 HRD-in -95.2, -52.32 70.44, 11.38 in-in-in SNCiii in-in ActLoopNT-in 2.912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.85, 164.58 APE9-dihe-na 131.46, -156.38 APE8-dihe-in -129.55, 139.43 APE8-rot-in 297.11 APE67-dihe-in -60.54, -22.69 -52.03, -49.04 APE12-dist-in 8.098 APE11-dist-in 11.392 APE10-dist-in 5.827 APE9-dist-in 3.498 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.164 0.184 A 337 336 0 0 0 0 [[44, 298]] 1.0 4wb8 AGC_PRKACA_HUMAN AGC 4e-95 323.8 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB5A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 5.6 14.452 BLAminus -123.05, 176.84 68.94, 80.02 -91.46, 24.86 270.2, 52.92 -60.74, -31.43 in-in in 9.03 Saltbr-in 2.715 HRD-in -92.12, -52.84 69.8, 13.37 in-in-in SNCiii in-in ActLoopNT-in 2.918 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.48, 163.75 APE9-dihe-na 132.31, -149.49 APE8-dihe-in -132.05, 134.14 APE8-rot-in 301.14 APE67-dihe-in -60.1, -21.12 -48.44, -50.23 APE12-dist-in 8.012 APE11-dist-in 11.4 APE10-dist-in 5.799 APE9-dist-in 3.567 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.641 0.165 0.196 A 350 338 0 0 0 0 [[44, 298]] 1.0 4wb5 AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB7A P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.445 14.649 BLAminus -119.06, -174.39 59.4, 77.28 -89.09, 26.42 267.74, 51.48 -60.48, -28.34 in-in in 8.87 Saltbr-in 2.769 HRD-in -93.55, -50.9 68.82, 8.95 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.63, 158.06 APE9-dihe-na 139.02, -156.91 APE8-dihe-in -126.94, 137.23 APE8-rot-in 299.54 APE67-dihe-in -64.26, -23.0 -50.4, -48.13 APE12-dist-in 8.18 APE11-dist-in 11.54 APE10-dist-in 5.955 APE9-dist-in 3.723 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 A 405 336 0 0 0 0 [[44, 298]] 1.0 4wb7 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB7B P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.38 14.712 BLAminus -115.93, -176.79 62.38, 75.33 -88.91, 25.18 264.71, 51.71 -56.9, -30.26 in-in in 8.962 Saltbr-in 2.773 HRD-in -94.01, -50.55 67.24, 10.48 in-in-in SNCiii in-in ActLoopNT-in 2.939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.07, 161.39 APE9-dihe-na 132.31, -156.17 APE8-dihe-in -127.2, 138.18 APE8-rot-in 298.14 APE67-dihe-in -59.62, -23.37 -52.63, -48.78 APE12-dist-in 8.198 APE11-dist-in 11.563 APE10-dist-in 5.97 APE9-dist-in 3.642 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 B 405 336 0 0 0 0 [[44, 298]] 1.0 4wb7 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 6BYRA P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.626 14.616 BLAminus -128.29, 177.03 62.06, 86.64 -97.54, 28.59 271.87, 66.62 -63.2, -33.23 in-in in 8.808 Saltbr-in 3.196 HRD-in -87.43, -52.47 67.28, 5.18 in-in-in SNCiii in-in ActLoopNT-in 3.193 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.51, 153.24 APE9-dihe-na 149.32, -133.8 APE8-dihe-in -139.35, 133.91 APE8-rot-in 312.31 APE67-dihe-in -68.4, -6.95 -52.73, -48.25 APE12-dist-in 8.734 APE11-dist-in 11.076 APE10-dist-in 5.63 APE9-dist-in 3.491 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 A 405 336 0 0 0 0 [[44, 298]] 1.0 6byr AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 6BYRC P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.679 14.34 BLAminus -129.89, 172.29 61.76, 74.25 -79.2, 34.93 281.69, 54.14 -61.8, -27.34 in-in in 8.733 Saltbr-in 2.498 HRD-in -93.13, -49.8 64.55, 7.44 in-in-in SNCiii in-in ActLoopNT-in 3.052 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.29, 161.94 APE9-dihe-na 130.51, -156.26 APE8-dihe-in -112.31, 134.09 APE8-rot-in 302.07 APE67-dihe-in -64.15, -16.52 -52.64, -41.39 APE12-dist-in 8.316 APE11-dist-in 11.106 APE10-dist-in 5.767 APE9-dist-in 3.618 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 C 405 336 0 0 0 0 [[44, 298]] 1.0 6byr AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 9EDCA P17612 14 351 351.0 ATP:60400 ATPlike Active DFGin 5.626 13.772 BLAminus -125.61, -173.52 60.53, 69.6 -81.59, 16.86 273.36, 51.23 -62.38, -30.28 in-in in 9.129 Saltbr-in 3.0 HRD-in -112.54, -46.7 65.17, 1.82 in-in-in SNCiii in-in ActLoopNT-in 3.14 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.87, 159.92 APE9-dihe-na 136.42, -156.18 APE8-dihe-in -101.13, 126.83 APE8-rot-in 299.98 APE67-dihe-in -84.76, -8.6 -60.74, -28.35 APE12-dist-in 7.999 APE11-dist-in 11.111 APE10-dist-in 5.797 APE9-dist-in 3.748 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 EM 4.18 999.0 999.0 A 350 338 0 0 0 0 [[44, 298]] 1.0 9edc AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB6A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 6.068 14.398 BLAminus -118.38, -169.49 51.77, 82.47 -95.61, 17.78 271.18, 55.73 -42.8, -37.29 in-in in 8.83 Saltbr-in 2.561 HRD-in -94.17, -52.18 74.17, 2.46 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.55, 166.68 APE9-dihe-na 116.18, 128.45 APE8-dihe-in -46.62, 128.74 APE8-rot-in 303.5 APE67-dihe-in -58.01, -23.74 -49.09, -50.89 APE12-dist-in 8.046 APE11-dist-in 11.764 APE10-dist-in 6.243 APE9-dist-in 3.767 L206R SEP11,SEP140,TPO198 SEP11,SEP140,TPO198 XRAY 2.1 0.19 0.237 A 350 338 0 0 0 0 [[44, 298]] 1.0 4wb6 AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB6B P17612 9 351 351.0 ATP:60401 ATPlike Active DFGin 5.872 14.073 BLAminus -117.82, -168.32 53.27, 78.35 -91.25, 29.34 274.97, 62.46 -60.26, -35.85 in-in in 8.687 Saltbr-in 2.75 HRD-in -101.62, -46.5 64.42, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.38, 164.15 APE9-dihe-na 120.83, 133.18 APE8-dihe-in -48.66, 125.41 APE8-rot-in 298.86 APE67-dihe-in -54.58, -37.6 -53.55, -42.52 APE12-dist-in 8.078 APE11-dist-in 11.617 APE10-dist-in 6.204 APE9-dist-in 3.822 L206R SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.19 0.237 B 350 343 0 0 0 0 [[44, 298]] 1.0 4wb6 AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKCB KPCB_HUMAN 8SE1A P05771 19 668 671.0 ANP:60706 ATPlike Active DFGin 6.007 12.839 BLAminus -130.5, -169.38 54.07, 70.37 -91.85, 35.76 301.77, 99.49 -89.35, 3.84 in-in in 8.337 Saltbr-in 2.524 HRD-in -91.65, -37.95 43.68, 28.8 in-in-in SNCiii in-in ActLoopNT-in 3.16 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.86, 170.42 APE9-dihe-na 126.28, -151.58 APE8-dihe-in -120.81, 128.88 APE8-rot-in 299.44 APE67-dihe-in -79.06, -41.06 -50.17, -27.42 APE12-dist-in 8.88 APE11-dist-in 12.178 APE10-dist-in 6.66 APE9-dist-in 3.611 None TPO500,TPO642,SEP661 TPO500,TPO642,SEP661 XRAY 3.32 0.202 0.256 A 674 607 0 0 0 0 [[342, 600]] 1.0 8se1 AGC_PRKCB_HUMAN AGC 1.5e-97 332.1 1 260 260 483 484 485 487 489 371 390 394 463 465 464 466 523 511 506 505 504 503 502 501 500 421 Protein kinase C beta type
AGC PRKCB KPCB_HUMAN 8SE1B P05771 19 668 671.0 ANP:60706 ATPlike Active DFGin 6.093 12.778 BLAminus -130.75, -169.0 53.85, 70.09 -92.15, 34.96 301.62, 99.67 -90.48, 2.45 in-in in 8.312 Saltbr-in 2.216 HRD-in -89.42, -35.84 47.27, 23.7 in-in-in SNCiii in-in ActLoopNT-in 3.284 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.83, 169.92 APE9-dihe-na 126.33, -152.59 APE8-dihe-in -121.43, 128.62 APE8-rot-in 299.3 APE67-dihe-in -78.67, -41.09 -50.34, -26.64 APE12-dist-in 8.722 APE11-dist-in 12.182 APE10-dist-in 6.709 APE9-dist-in 3.767 None TPO500,TPO642,SEP661 TPO500,TPO642,SEP661 XRAY 3.32 0.202 0.256 B 674 631 0 0 0 0 [[342, 600]] 1.0 8se1 AGC_PRKCB_HUMAN AGC 1.5e-97 332.1 1 260 260 483 484 485 487 489 371 390 394 463 465 464 466 523 511 506 505 504 503 502 501 500 421 Protein kinase C beta type
AGC PRKCB KPCB_HUMAN 8SE2B P05771 30 671 671.0 ANP:701 ATPlike Active DFGin 5.706 12.737 BLAminus -122.79, -175.57 50.54, 85.22 -103.07, 33.77 300.25, 95.58 -78.87, -5.25 in-in in 8.251 Saltbr-in 2.675 HRD-in -90.05, -48.77 75.62, -5.68 in-in-in SNCiii in-in ActLoopNT-in 3.126 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.22, 161.28 APE9-dihe-na 125.49, -179.08 APE8-dihe-in -100.09, 129.99 APE8-rot-in 297.02 APE67-dihe-in -66.56, -21.71 -49.98, -38.79 APE12-dist-in 8.634 APE11-dist-in 11.712 APE10-dist-in 6.223 APE9-dist-in 3.606 None TPO500,TPO642,SEP661 TPO500,TPO642,SEP661 XRAY 2.95 0.196 0.252 B 672 589 0 0 0 0 [[342, 600]] 1.0 8se2 AGC_PRKCB_HUMAN AGC 1.5e-97 332.1 1 260 260 483 484 485 487 489 371 390 394 463 465 464 466 523 511 506 505 504 503 502 501 500 421 Protein kinase C beta type
AGC PRKCI KPCI_HUMAN 5LIHA P41743 248 588 596.0 ADP:60601 ATPlike Active DFGin 5.403 11.863 BLAminus -129.58, 178.7 63.64, 84.98 -106.19, 67.5 320.36, 105.86 -96.86, -30.05 in-in in 9.178 Saltbr-in 3.031 HRD-in -49.42, -59.61 61.3, 24.72 in-in-in SNCiii in-in ActLoopNT-in 3.109 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.76, 169.43 APE9-dihe-na 122.35, -170.42 APE8-dihe-in -91.96, 136.55 APE8-rot-in 289.3 APE67-dihe-in -72.22, -23.04 -49.75, -40.52 APE12-dist-in 7.983 APE11-dist-in 10.986 APE10-dist-in 5.421 APE9-dist-in 3.56 None TPO412,TPO564 TPO412,TPO564 XRAY 3.25 0.258 0.284 A 349 326 15 0 0 0 [[254, 522]] 1.0 5lih AGC_PRKCI_HUMAN AGC 1.1e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKCI KPCI_HUMAN 5LIHB P41743 249 588 596.0 ADP:60601 ATPlike Active DFGin 5.31 11.876 BLAminus -129.18, 178.42 63.46, 84.62 -106.43, 67.35 320.63, 105.98 -96.29, -29.69 in-in in 8.72 Saltbr-in 2.545 HRD-in -49.62, -59.64 61.27, 24.64 in-in-in SNCiii in-in ActLoopNT-in 3.141 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.47, 168.99 APE9-dihe-na 122.16, -170.23 APE8-dihe-in -91.66, 136.86 APE8-rot-in 289.24 APE67-dihe-in -72.3, -22.91 -49.4, -40.32 APE12-dist-in 8.329 APE11-dist-in 11.256 APE10-dist-in 5.693 APE9-dist-in 3.742 None TPO412,TPO564 TPO412,TPO564 XRAY 3.25 0.258 0.284 B 349 320 20 0 0 0 [[254, 522]] 1.0 5lih AGC_PRKCI_HUMAN AGC 1.1e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKCI KPCI_HUMAN 5LI9A P41743 248 589 596.0 ACP:60601 ATPlike Active DFGin 5.635 12.633 BLAminus -139.17, 172.4 72.31, 78.11 -98.86, 1.23 304.03, 143.26 -64.9, -22.84 in-in in 8.361 Saltbr-in 2.614 HRD-in -73.79, -55.22 70.11, -1.11 in-in-in SNCiii in-in ActLoopNT-in 2.81 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.64, 169.55 APE9-dihe-na 127.72, -178.47 APE8-dihe-in -93.25, 127.56 APE8-rot-in 298.81 APE67-dihe-in -60.64, -20.02 -47.28, -45.36 APE12-dist-in 8.812 APE11-dist-in 11.949 APE10-dist-in 6.432 APE9-dist-in 3.836 None TPO412,TPO564 TPO412,TPO564 XRAY 1.79 0.19 0.231 A 350 330 12 0 0 0 [[254, 522]] 1.0 5li9 AGC_PRKCI_HUMAN AGC 1.2e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKCI KPCI_HUMAN 5LI1A P41743 248 589 596.0 ANP:60601 ATPlike Active DFGin 5.079 11.961 BLAminus -129.24, 176.98 73.22, 90.17 -103.83, 11.43 308.18, 130.49 -69.42, -18.98 in-in in 8.413 Saltbr-in 2.816 HRD-in -77.28, -52.44 73.77, 3.75 in-in-in SNCiii in-in ActLoopNT-in 2.975 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.65, 168.01 APE9-dihe-na 127.57, -168.6 APE8-dihe-in -111.48, 126.0 APE8-rot-in 296.01 APE67-dihe-in -54.62, -31.15 -46.95, -45.66 APE12-dist-in 8.752 APE11-dist-in 11.822 APE10-dist-in 6.31 APE9-dist-in 3.517 None TPO412,SEP484,TPO564 TPO412,SEP484,TPO564 XRAY 2.0 0.154 0.217 A 354 332 10 0 0 0 [[254, 522]] 1.0 5li1 AGC_PRKCI_HUMAN AGC 1.2e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKG1 KGP1_HUMAN 6BG2A Q13976 336 671 671.0 ANP:700 ATPlike Active DFGin 5.811 14.714 BLAminus -124.15, 169.14 66.07, 88.5 -100.57, 30.98 280.35, 66.41 -65.35, -25.12 in-in in 9.522 Saltbr-in 2.883 HRD-in -85.83, -52.95 73.29, 9.38 in-in-in SNCiii in-in ActLoopNT-in 2.851 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.93, 165.57 APE9-dihe-na 117.74, 172.78 APE8-dihe-in -83.6, 129.51 APE8-rot-in 307.46 APE67-dihe-in -66.9, -19.23 -49.63, -41.3 APE12-dist-in 8.235 APE11-dist-in 11.512 APE10-dist-in 6.041 APE9-dist-in 4.269 None TPO517 TPO517 XRAY 1.83 0.188 0.215 A 347 336 0 0 0 0 [[360, 619]] 1.0 6bg2 AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 6BG2B Q13976 346 671 671.0 ANP:700 ATPlike Active DFGin 6.001 13.81 BLAminus -122.67, 175.58 65.94, 84.43 -99.77, 30.78 285.96, 70.42 -64.93, -24.07 in-in in 8.944 Saltbr-in 2.743 HRD-in -86.95, -52.47 73.99, 7.96 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.61, 163.67 APE9-dihe-na 118.96, 172.39 APE8-dihe-in -86.94, 131.94 APE8-rot-in 306.51 APE67-dihe-in -68.79, -20.88 -48.58, -41.68 APE12-dist-in 7.826 APE11-dist-in 11.215 APE10-dist-in 5.769 APE9-dist-in 4.008 None TPO517 TPO517 XRAY 1.83 0.188 0.215 B 347 326 0 0 0 0 [[360, 619]] 1.0 6bg2 AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 6BG2C Q13976 337 671 671.0 ANP:700 ATPlike Active DFGin 5.746 14.057 BLAminus -122.99, 175.03 65.66, 84.22 -99.61, 30.7 281.62, 66.26 -64.81, -23.57 in-in in 8.742 Saltbr-in 2.723 HRD-in -85.99, -53.51 74.31, 7.4 in-in-in SNCiii in-in ActLoopNT-in 2.951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.66, 165.85 APE9-dihe-na 118.46, 173.18 APE8-dihe-in -87.41, 130.75 APE8-rot-in 306.63 APE67-dihe-in -67.71, -19.03 -48.39, -42.55 APE12-dist-in 7.972 APE11-dist-in 11.385 APE10-dist-in 5.857 APE9-dist-in 3.861 None TPO517 TPO517 XRAY 1.83 0.188 0.215 C 347 335 0 0 0 0 [[360, 619]] 1.0 6bg2 AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 6BG2D Q13976 344 671 671.0 ANP:700 ATPlike Active DFGin 5.71 14.012 BLAminus -124.49, 174.79 65.67, 84.87 -99.37, 30.45 283.38, 66.11 -64.13, -22.3 in-in in 8.754 Saltbr-in 2.644 HRD-in -85.68, -52.69 74.16, 8.99 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.92, 166.42 APE9-dihe-na 119.53, 169.97 APE8-dihe-in -84.81, 130.45 APE8-rot-in 305.19 APE67-dihe-in -66.29, -19.88 -48.13, -43.31 APE12-dist-in 7.988 APE11-dist-in 11.327 APE10-dist-in 5.784 APE9-dist-in 3.81 None TPO517 TPO517 XRAY 1.83 0.188 0.215 D 347 328 0 0 0 0 [[360, 619]] 1.0 6bg2 AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 7LV3A Q13976 57 671 671.0 ANP:60803 ATPlike Active DFGin 5.851 14.036 BLAminus -116.97, 177.04 63.26, 88.72 -106.87, 28.72 283.22, 63.7 -62.95, -24.33 in-in in 8.624 Saltbr-in 2.891 HRD-in -87.82, -54.22 74.26, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.911 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.28, 149.98 APE9-dihe-na 157.95, -145.59 APE8-dihe-in -124.73, 128.61 APE8-rot-in 299.79 APE67-dihe-in -58.37, -20.06 -47.89, -51.97 APE12-dist-in 7.972 APE11-dist-in 11.057 APE10-dist-in 5.469 APE9-dist-in 3.811 None TPO517 TPO517 XRAY 2.41 0.201 0.238 A 617 600 0 0 0 0 [[360, 619]] 1.0 7lv3 AGC_PRKG1_HUMAN AGC 1.3e-83 286.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 7LV3B Q13976 58 671 671.0 ANP:60803 ATPlike Active DFGin 5.634 13.962 BLAminus -116.52, 178.28 63.3, 90.17 -108.68, 29.08 283.48, 65.02 -62.88, -23.93 in-in in 8.883 Saltbr-in 2.824 HRD-in -86.48, -52.9 74.97, 7.4 in-in-in SNCiii in-in ActLoopNT-in 2.959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.28, 149.21 APE9-dihe-na 157.62, -145.94 APE8-dihe-in -123.75, 129.22 APE8-rot-in 300.73 APE67-dihe-in -59.05, -19.44 -46.41, -52.49 APE12-dist-in 8.134 APE11-dist-in 11.198 APE10-dist-in 5.604 APE9-dist-in 3.787 None TPO517 TPO517 XRAY 2.41 0.201 0.238 B 617 593 0 0 0 0 [[360, 619]] 1.0 7lv3 AGC_PRKG1_HUMAN AGC 1.3e-83 286.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC ROCK1 ROCK1_HUMAN 2V55A Q13464 6 404 1354.0 ANP:1480 ATPlike Active DFGin 5.88 13.604 BLAminus -137.29, -177.31 60.22, 109.9 -132.74, 24.25 290.89, 71.12 -53.92, -52.21 in-in in 9.076 Saltbr-in 2.708 HRD-in -79.75, -71.28 93.49, -31.37 in-in-in SNCiii in-in ActLoopNT-in 3.281 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.46, 139.75 APE9-dihe-na 103.51, 160.5 APE8-dihe-in -55.22, 144.8 APE8-rot-in 285.63 APE67-dihe-in -74.86, -38.79 -80.34, -13.24 APE12-dist-in 10.324 APE11-dist-in 11.278 APE10-dist-in 5.647 APE9-dist-in 4.131 None None None XRAY 3.705 0.238 0.269 A 406 393 0 0 0 0 [[76, 338]] 1.0 2v55 AGC_ROCK1_HUMAN AGC 3.3e-94 320.8 1 260 260 215 216 217 219 221 105 124 128 195 197 196 198 260 244 239 238 237 236 235 234 233 154 Rho-associated protein kinase 1
AGC ROCK1 ROCK1_HUMAN 2V55C Q13464 6 404 1354.0 ANP:1480 ATPlike Active DFGin 5.884 13.608 BLAminus -137.56, -177.44 62.15, 108.48 -130.26, 22.71 291.3, 72.92 -54.95, -50.69 in-in in 9.111 Saltbr-in 2.706 HRD-in -78.29, -71.79 95.11, -31.46 in-in-in SNCiii in-in ActLoopNT-in 3.247 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.41, 139.12 APE9-dihe-na 103.28, 159.31 APE8-dihe-in -53.48, 142.5 APE8-rot-in 287.35 APE67-dihe-in -76.24, -37.92 -78.8, -11.99 APE12-dist-in 10.28 APE11-dist-in 11.269 APE10-dist-in 5.623 APE9-dist-in 4.097 None None None XRAY 3.705 0.238 0.269 C 406 396 0 0 0 0 [[76, 338]] 1.0 2v55 AGC_ROCK1_HUMAN AGC 3.3e-94 320.8 1 260 260 215 216 217 219 221 105 124 128 195 197 196 198 260 244 239 238 237 236 235 234 233 154 Rho-associated protein kinase 1
CAMK AURKA AURKA_HUMAN 1OL5A O14965 123 388 403.0 ADP:1388 ATPlike Active DFGin 5.578 15.096 BLAminus -139.2, -172.08 52.22, 80.16 -90.83, 24.66 282.61, 72.55 -49.87, -44.18 in-in in 9.451 Saltbr-in 2.912 HRD-in -63.28, -60.88 73.6, 1.59 in-in-in SNCiii in-in ActLoopNT-in 2.928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.42, 162.5 APE9-dihe-na 119.45, -153.19 APE8-dihe-in -110.77, 140.24 APE8-rot-in 313.06 APE67-dihe-in -62.23, -14.3 -43.16, -62.5 APE12-dist-in 8.174 APE11-dist-in 10.957 APE10-dist-in 5.274 APE9-dist-in 3.683 None TPO287,TPO288 TPO287,TPO288 XRAY 2.5 0.194 0.252 A 282 266 0 0 0 0 [[133, 383]] 1.0 1ol5 CAMK_AURKA_HUMAN CAMK 7.4e-80 273.9 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK AURKA AURKA_HUMAN 6VPGA O14965 7 389 403.0 ANP:60401 ATPlike Active DFGin 5.318 15.07 BLAminus -133.54, 176.05 56.91, 81.54 -90.61, 23.9 286.39, 75.22 -62.73, -9.76 in-in in 9.884 Saltbr-in 2.954 HRD-in -72.51, -51.0 67.55, 11.3 in-in-in SNCiii in-in ActLoopNT-in 3.043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.96, 159.16 APE9-dihe-na 122.67, -152.53 APE8-dihe-in -117.94, 146.39 APE8-rot-in 309.68 APE67-dihe-in -61.83, -12.97 -52.19, -62.88 APE12-dist-in 8.517 APE11-dist-in 11.427 APE10-dist-in 5.724 APE9-dist-in 3.833 None TPO287,TPO288 TPO287,TPO288 XRAY 2.64 0.204 0.245 A 292 267 0 0 0 0 [[133, 383]] 1.0 6vpg CAMK_AURKA_HUMAN CAMK 8.4e-80 273.7 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK AURKA AURKA_HUMAN 5LXMA O14965 126 392 403.0 ADP:60501 ATPlike Active DFGin 5.391 14.976 BLAminus -135.45, -179.78 54.7, 80.97 -90.8, 30.12 283.16, 71.51 -72.4, -3.16 in-in in 9.247 Saltbr-in 2.724 HRD-in -74.23, -48.55 66.99, 5.01 in-in-in SNCiii in-in ActLoopNT-in 3.114 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.91, 137.37 APE9-dihe-na 128.62, -150.21 APE8-dihe-in -129.87, 142.81 APE8-rot-in 303.47 APE67-dihe-in -69.71, -10.62 -37.99, -61.07 APE12-dist-in 8.257 APE11-dist-in 10.692 APE10-dist-in 5.213 APE9-dist-in 3.298 C290A,C393A TPO288 TPO288 XRAY 2.08 0.202 0.243 A 283 267 0 0 0 0 [[133, 383]] 1.0 5lxm CAMK_AURKA_HUMAN CAMK 9.2e-79 270.3 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK AURKA AURKA_HUMAN 5G1XA O14965 126 389 403.0 ADP:1390 ATPlike Active DFGin 5.343 15.03 BLAminus -132.86, -170.57 52.68, 76.5 -90.96, 13.96 279.12, 78.43 -59.51, -20.51 in-in in 9.278 Saltbr-in 2.828 HRD-in -82.61, -50.12 70.7, 5.33 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.42, -179.26 APE9-dihe-na 65.74, -155.89 APE8-dihe-in -128.23, 121.78 APE8-rot-in 304.75 APE67-dihe-in -61.27, -19.7 -46.07, -47.67 APE12-dist-in 8.247 APE11-dist-in 10.799 APE10-dist-in 5.53 APE9-dist-in 3.699 C290A,C393A TPO288 TPO288 XRAY 1.72 0.177 0.195 A 285 264 0 0 0 0 [[133, 383]] 1.0 5g1x CAMK_AURKA_HUMAN CAMK 9.4e-79 270.3 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK CAMK2A KCC2A_HUMAN 7UJSA Q9UQM7 7 274 478.0 ADP:301 ATPlike Active DFGin 6.209 15.164 BLAminus -142.86, -173.92 52.2, 80.06 -100.62, 24.47 291.74, 81.6 -63.11, -26.23 in-in in 9.512 Saltbr-in 3.444 HRD-in -76.47, -52.69 80.52, -7.0 in-in-in SNCiii in-in ActLoopNT-in 2.952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.88, 140.41 APE9-dihe-na 133.49, -148.09 APE8-dihe-in -128.43, 117.33 APE8-rot-in 305.05 APE67-dihe-in -59.07, -26.67 -36.29, -54.08 APE12-dist-in 10.197 APE11-dist-in 11.505 APE10-dist-in 5.779 APE9-dist-in 3.683 Q223K None None XRAY 2.75 0.201 0.262 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujs CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UIRA Q9UQM7 7 274 478.0 ATP:302 ATPlike Active DFGin 6.045 15.107 BLAminus -137.0, 179.68 44.28, 101.28 -106.42, 24.78 295.79, 81.95 -53.14, -27.06 in-in in 9.85 Saltbr-in 3.466 HRD-in -74.22, -43.69 67.52, 3.92 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.48, 156.41 APE9-dihe-na 131.95, -156.1 APE8-dihe-in -122.09, 129.91 APE8-rot-in 298.28 APE67-dihe-in -55.12, -36.11 -51.43, -40.3 APE12-dist-in 10.333 APE11-dist-in 11.793 APE10-dist-in 6.056 APE9-dist-in 3.425 D135N,Q223K None None XRAY 3.1 0.234 0.274 A 268 268 0 0 0 0 [[13, 271]] 1.0 7uir CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UIRB Q9UQM7 7 273 478.0 ATP:301 ATPlike Active DFGin 6.093 14.463 BLAminus -136.84, -179.4 43.86, 99.82 -105.8, 24.57 296.99, 81.24 -56.04, -26.17 in-in in 9.403 Saltbr-in 3.027 HRD-in -74.93, -42.65 67.84, 3.24 in-in-in SNCiii in-in ActLoopNT-in 2.915 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.86, 157.92 APE9-dihe-na 132.59, -155.55 APE8-dihe-in -122.09, 129.05 APE8-rot-in 298.73 APE67-dihe-in -54.7, -35.97 -51.63, -40.47 APE12-dist-in 10.303 APE11-dist-in 11.733 APE10-dist-in 5.989 APE9-dist-in 3.504 D135N,Q223K None None XRAY 3.1 0.234 0.274 B 268 261 6 0 0 0 [[13, 271]] 1.0 7uir CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UJPA Q9UQM7 7 274 478.0 ADP:301 ATPlike Active DFGin 6.775 14.64 BLAminus -129.88, 174.11 65.35, 73.67 -96.28, 29.41 284.7, 81.79 -65.3, -26.47 in-in in 8.527 Saltbr-in 2.903 HRD-in -76.38, -51.72 77.74, -11.0 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.94, 142.69 APE9-dihe-na 139.08, -169.53 APE8-dihe-in -115.65, 123.25 APE8-rot-in 308.77 APE67-dihe-in -69.44, -15.11 -33.38, -56.34 APE12-dist-in 10.469 APE11-dist-in 11.397 APE10-dist-in 5.657 APE9-dist-in 3.521 D135N,Q223K None None XRAY 2.56 0.234 0.281 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujp CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UJPB Q9UQM7 7 273 478.0 ATP:301 ATPlike Active DFGin 6.942 14.313 BLAminus -133.64, 174.92 62.39, 75.15 -97.38, 27.07 283.14, 81.65 -64.42, -25.12 in-in in 8.558 Saltbr-in 2.783 HRD-in -76.01, -51.46 77.74, -9.31 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.94, 139.06 APE9-dihe-na 146.74, -166.31 APE8-dihe-in -115.05, 124.1 APE8-rot-in 308.42 APE67-dihe-in -69.31, -14.12 -35.51, -54.36 APE12-dist-in 10.25 APE11-dist-in 11.592 APE10-dist-in 5.843 APE9-dist-in 3.572 D135N,Q223K None None XRAY 2.56 0.234 0.281 B 268 267 0 0 0 0 [[13, 271]] 1.0 7ujp CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CHEK1 CHK1_HUMAN 7AKMA O14757 2 271 476.0 AGS:401 ATPlike Active DFGin 6.775 14.143 BLAminus -128.66, 150.55 71.15, 96.3 -103.32, 28.49 292.74, 82.8 -70.74, -21.81 in-in in 9.111 Saltbr-in 2.706 HRD-in -78.28, -45.32 76.75, -0.14 in-in-in SNCiii in-in ActLoopNT-in 3.011 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.43, 171.3 APE9-dihe-na 110.38, -147.97 APE8-dihe-in -135.73, 125.59 APE8-rot-in 300.71 APE67-dihe-in -62.97, -17.75 -56.42, -42.48 APE12-dist-in 9.309 APE11-dist-in 11.674 APE10-dist-in 6.171 APE9-dist-in 3.407 D10R None None XRAY 1.93 0.199 0.242 A 298 270 0 0 0 0 [[9, 265]] 1.0 7akm CAMK_CHEK1_HUMAN CAMK 3.4e-71 245.5 2 256 255 147 148 149 151 153 38 55 59 127 129 128 130 190 177 172 171 170 169 168 167 166 85 Serine/threonine-protein kinase Chk1
CAMK DAPK1 DAPK1_HUMAN 2W4KA P53355 2 302 1430.0 ADP:1303 ATPlike Active DFGin 6.672 14.178 BLAminus -119.76, -176.11 66.35, 79.87 -97.37, 22.41 282.66, 74.96 -63.58, -22.08 in-in in 9.11 Saltbr-in 2.829 HRD-in -72.34, -46.15 68.63, 4.94 in-in-in SNCiii in-in ActLoopNT-in 2.866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.51, 175.21 APE9-dihe-na 86.37, -178.83 APE8-dihe-in -92.32, 120.41 APE8-rot-in 301.2 APE67-dihe-in -65.94, -16.49 -43.92, -47.7 APE12-dist-in 9.204 APE11-dist-in 12.288 APE10-dist-in 6.82 APE9-dist-in 5.132 None None None XRAY 1.9 0.195 0.228 A 302 301 0 0 0 0 [[13, 275]] 1.0 2w4k CAMK_DAPK1_HUMAN CAMK 6.8e-95 323.2 1 256 256 160 161 162 164 166 42 64 68 136 138 137 139 199 187 182 181 180 179 178 177 176 94 Death-associated protein kinase 1
CAMK DAPK1 DAPK1_HUMAN 2XUUA P53355 2 302 1430.0 ADP:1303 ATPlike Active DFGin 6.814 14.3 BLAminus -117.01, 179.93 67.97, 81.82 -97.7, 27.63 286.42, 73.81 -75.99, -13.96 in-in in 9.047 Saltbr-in 2.623 HRD-in -76.48, -45.49 71.86, 3.84 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.39, 167.91 APE9-dihe-na 89.82, 178.63 APE8-dihe-in -101.18, 124.0 APE8-rot-in 296.23 APE67-dihe-in -60.21, -22.55 -44.54, -47.64 APE12-dist-in 8.87 APE11-dist-in 11.727 APE10-dist-in 6.406 APE9-dist-in 5.145 E182A None None XRAY 1.8 0.179 0.226 A 334 301 0 0 0 0 [[13, 275]] 1.0 2xuu CAMK_DAPK1_HUMAN CAMK 1.4e-94 322.3 1 256 256 160 161 162 164 166 42 64 68 136 138 137 139 199 187 182 181 180 179 178 177 176 94 Death-associated protein kinase 1
CAMK DCLK1 DCLK1_HUMAN 5JZJA O15075 374 648 740.0 AN2:703 ATPlike Active DFGin 6.559 14.457 BLAminus -124.73, -164.54 49.76, 81.39 -91.62, 27.77 280.9, 72.89 -62.64, -30.24 in-in in 9.264 Saltbr-in 2.961 HRD-in -80.29, -46.18 67.47, 2.65 in-in-in SNCiii in-in ActLoopNT-in 2.862 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.12, 159.65 APE9-dihe-na 123.02, -170.92 APE8-dihe-in -106.5, 129.13 APE8-rot-in 307.92 APE67-dihe-in -61.41, -36.29 -48.5, -40.56 APE12-dist-in 8.952 APE11-dist-in 12.325 APE10-dist-in 6.742 APE9-dist-in 4.306 None None None XRAY 1.71 0.178 0.208 A 297 271 4 0 0 0 [[390, 647]] 1.0 5jzj CAMK_DCLK1_HUMAN CAMK 7.6e-90 306.6 1 256 256 532 533 534 536 538 419 436 440 508 510 509 511 569 557 552 551 550 549 548 547 546 466 Serine/threonine-protein kinase DCLK1
CAMK DCLK1 DCLK1_HUMAN 5JZJB O15075 382 648 740.0 AN2:902 ATPlike Active DFGin 6.403 14.423 BLAminus -126.14, -167.19 53.32, 81.81 -94.99, 26.92 281.83, 75.21 -56.86, -35.14 in-in in 8.806 Saltbr-in 2.638 HRD-in -80.6, -45.11 67.98, 3.84 in-in-in SNCiii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.06, 162.17 APE9-dihe-na 120.91, -173.72 APE8-dihe-in -109.44, 126.03 APE8-rot-in 300.86 APE67-dihe-in -59.98, -31.53 -43.43, -44.7 APE12-dist-in 9.044 APE11-dist-in 12.358 APE10-dist-in 6.832 APE9-dist-in 4.274 None None None XRAY 1.71 0.178 0.208 B 297 261 6 0 0 0 [[390, 647]] 1.0 5jzj CAMK_DCLK1_HUMAN CAMK 7.6e-90 306.6 1 256 256 532 533 534 536 538 419 436 440 508 510 509 511 569 557 552 551 550 549 548 547 546 466 Serine/threonine-protein kinase DCLK1
CAMK PASK PASK_HUMAN 3DLSA Q96RG2 982 1266 1323.0 ADP:1 ATPlike Active DFGin 6.001 14.204 BLAminus -129.0, 178.94 63.52, 79.16 -100.96, 27.03 282.44, 72.76 -70.92, -15.42 in-in in 8.655 Saltbr-in 2.605 HRD-na-E -71.55, -40.2 72.7, 1.22 in-in-in SNCiii in-in ActLoopNT-in 2.993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -115.6, 5.88 APE9-dihe-na -96.65, -154.85 APE8-dihe-in -98.92, 122.93 APE8-rot-in 302.12 APE67-dihe-in -72.66, -14.95 -65.45, -19.89 APE12-dist-in 10.203 APE11-dist-in 10.574 APE10-dist-in 5.061 APE9-dist-in 3.451 None None None XRAY 2.3 0.244 0.297 A 335 285 0 0 0 0 [[999, 1251]] 1.0 3dls CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSB Q96RG2 982 1267 1323.0 ADP:2 ATPlike Active DFGin 6.1 14.087 BLAminus -126.55, 179.43 61.31, 80.64 -98.16, 22.24 284.4, 71.69 -72.83, -6.95 in-in in 8.346 Saltbr-in 2.677 HRD-na-E -67.25, -43.38 72.94, 0.56 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.86, 22.09 APE9-dihe-na -121.63, -155.86 APE8-dihe-in -97.56, 124.97 APE8-rot-in 306.83 APE67-dihe-in -68.7, -17.81 -61.84, -27.67 APE12-dist-in 10.243 APE11-dist-in 10.688 APE10-dist-in 5.149 APE9-dist-in 3.521 None None None XRAY 2.3 0.244 0.297 B 335 280 6 0 0 0 [[999, 1251]] 1.0 3dls CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSC Q96RG2 982 1267 1323.0 ADP:3 ATPlike Active DFGin 6.549 14.136 BLAminus -121.24, -178.98 61.8, 81.93 -100.03, 24.34 279.06, 77.86 -70.4, -24.84 in-in in 8.286 Saltbr-in 2.707 HRD-na-E -75.53, -39.96 73.3, -0.15 in-in-in SNCiii in-in ActLoopNT-in 2.808 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -109.16, 23.96 APE9-dihe-na -111.98, -161.37 APE8-dihe-in -95.46, 124.23 APE8-rot-in 302.16 APE67-dihe-in -72.29, -18.02 -57.94, -30.36 APE12-dist-in 9.98 APE11-dist-in 10.437 APE10-dist-in 4.962 APE9-dist-in 3.466 None None None XRAY 2.3 0.244 0.297 C 335 281 5 0 0 0 [[999, 1251]] 1.0 3dls CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSD Q96RG2 982 1266 1323.0 ADP:4 ATPlike Active DFGin 5.989 14.037 BLAminus -119.78, -174.43 57.15, 82.44 -96.61, 20.08 283.36, 68.59 -63.18, -13.75 in-in in 8.596 Saltbr-in 2.674 HRD-na-E -66.59, -43.13 75.45, -3.58 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.17, 8.76 APE9-dihe-na -100.36, -154.44 APE8-dihe-in -94.34, 129.8 APE8-rot-in 309.84 APE67-dihe-in -63.24, -17.05 -59.73, -34.41 APE12-dist-in 10.579 APE11-dist-in 10.601 APE10-dist-in 5.212 APE9-dist-in 3.318 None None None XRAY 2.3 0.244 0.297 D 335 284 1 0 0 0 [[999, 1251]] 1.0 3dls CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSE Q96RG2 982 1267 1323.0 ADP:5 ATPlike Active DFGin 6.351 14.113 BLAminus -115.03, 172.38 61.43, 82.92 -98.38, 26.76 287.19, 66.36 -61.94, -22.57 in-in in 8.272 Saltbr-in 3.015 HRD-na-E -64.64, -41.08 75.56, -14.47 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.8, 6.63 APE9-dihe-na -93.38, -160.98 APE8-dihe-in -92.63, 131.98 APE8-rot-in 304.09 APE67-dihe-in -71.09, -14.17 -58.49, -32.88 APE12-dist-in 10.767 APE11-dist-in 10.575 APE10-dist-in 5.072 APE9-dist-in 3.423 None None None XRAY 2.3 0.244 0.297 E 335 282 4 0 0 0 [[999, 1251]] 1.0 3dls CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSF Q96RG2 982 1266 1323.0 ADP:6 ATPlike Active DFGin 6.208 14.428 BLAminus -120.86, -179.45 54.8, 74.61 -87.61, 27.75 280.29, 66.66 -72.72, -14.22 in-in in 8.492 Saltbr-in 2.879 HRD-na-E -64.59, -48.9 86.1, -8.79 in-in-in SNCiii in-in ActLoopNT-in 2.704 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.3, 4.74 APE9-dihe-na -89.15, -152.34 APE8-dihe-in -104.88, 132.7 APE8-rot-in 302.97 APE67-dihe-in -72.03, -17.52 -62.59, -27.45 APE12-dist-in 10.486 APE11-dist-in 10.547 APE10-dist-in 5.101 APE9-dist-in 3.284 None None None XRAY 2.3 0.244 0.297 F 335 281 4 0 0 0 [[999, 1251]] 1.0 3dls CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PIM1 PIM1_HUMAN 1YXTA P11309 33 306 313.0 ANP:322 ATPlike Active DFGin 6.029 14.245 BLAminus -131.81, 176.98 66.39, 83.69 -99.64, 19.64 287.53, 80.25 -65.72, -15.35 in-in in 8.309 Saltbr-in 2.894 HRD-na-A -67.95, -50.18 66.45, 4.68 in-in-in SNCiii in-in ActLoopNT-in 2.809 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.69, 12.99 APE9-dihe-na -80.03, -158.46 APE8-dihe-in -83.46, 121.7 APE8-rot-in 308.53 APE67-dihe-in -70.36, -3.81 -49.69, -52.76 APE12-dist-in 9.729 APE11-dist-in 8.665 APE10-dist-in 5.279 APE9-dist-in 3.805 None None None XRAY 2.0 0.183 0.216 A 293 274 0 0 0 0 [[38, 290]] 1.0 1yxt CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUA P11309 33 305 313.0 AMP:550 ATPlike Active DFGin 6.045 14.58 BLAminus -128.48, 170.01 62.85, 77.77 -90.35, 20.24 287.6, 77.99 -74.7, 1.63 in-in in 8.513 Saltbr-in 2.486 HRD-na-A -60.24, -50.74 67.33, 4.52 in-in-in SNCiii in-in ActLoopNT-in 2.893 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.18, 25.46 APE9-dihe-na -90.91, -158.18 APE8-dihe-in -86.5, 120.86 APE8-rot-in 310.09 APE67-dihe-in -63.06, -9.2 -60.21, -45.83 APE12-dist-in 9.959 APE11-dist-in 8.835 APE10-dist-in 5.689 APE9-dist-in 3.869 None None None XRAY 2.24 0.231 0.276 A 293 273 0 0 0 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUB P11309 33 305 313.0 AMP:650 ATPlike Active DFGin 6.12 14.673 BLAminus -120.37, 167.93 65.74, 85.44 -95.36, 14.03 285.37, 78.45 -64.71, -9.22 in-in in 8.6 Saltbr-in 2.814 HRD-na-A -59.51, -51.25 68.06, 6.92 in-in-in SNCiii in-in ActLoopNT-in 2.999 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.12, 36.18 APE9-dihe-na -84.74, -152.35 APE8-dihe-in -93.27, 122.65 APE8-rot-in 302.12 APE67-dihe-in -68.21, -7.03 -55.31, -45.11 APE12-dist-in 9.8 APE11-dist-in 8.534 APE10-dist-in 5.457 APE9-dist-in 3.841 None None None XRAY 2.24 0.231 0.276 B 293 273 0 0 0 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUC P11309 34 305 313.0 AMP:750 ATPlike Active DFGin 6.11 14.741 BLAminus -134.94, 167.86 62.59, 83.1 -95.62, 21.45 280.06, 80.63 -81.83, 7.92 in-in in 8.716 Saltbr-in 2.612 HRD-na-A -67.31, -48.53 67.93, 5.85 in-in-in SNCiii in-in ActLoopNT-in 2.899 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.01, 44.98 APE9-dihe-na -103.92, -155.25 APE8-dihe-in -86.11, 117.99 APE8-rot-in 310.09 APE67-dihe-in -68.22, -9.23 -52.45, -45.39 APE12-dist-in 9.697 APE11-dist-in 8.654 APE10-dist-in 5.604 APE9-dist-in 3.847 None None None XRAY 2.24 0.231 0.276 C 293 272 0 0 0 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUD P11309 33 305 313.0 AMP:850 ATPlike Active DFGin 6.236 14.556 BLAminus -126.04, 169.08 67.7, 73.28 -88.52, 13.94 289.01, 78.99 -70.28, -2.85 in-in in 8.789 Saltbr-in 2.466 HRD-na-A -64.06, -51.29 66.47, 10.4 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.8, 31.82 APE9-dihe-na -93.66, -159.09 APE8-dihe-in -85.99, 118.35 APE8-rot-in 303.12 APE67-dihe-in -71.66, -13.36 -52.91, -39.75 APE12-dist-in 9.896 APE11-dist-in 8.645 APE10-dist-in 5.457 APE9-dist-in 3.827 None None None XRAY 2.24 0.231 0.276 D 293 273 0 0 0 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1XR1A P11309 32 308 313.0 ANP:501 ATPlike Active DFGin 5.888 14.214 BLAminus -138.05, 176.98 59.78, 85.31 -96.55, 16.88 287.93, 82.19 -61.38, -7.19 in-in in 8.717 Saltbr-in 2.833 HRD-na-A -59.95, -51.82 71.23, 5.72 in-in-in SNCiii in-in ActLoopNT-in 2.752 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.05, 45.66 APE9-dihe-na -114.17, -171.15 APE8-dihe-in -64.11, 112.97 APE8-rot-in 299.41 APE67-dihe-in -49.28, -12.21 -42.84, -67.53 APE12-dist-in 9.608 APE11-dist-in 8.695 APE10-dist-in 5.522 APE9-dist-in 4.07 None None None XRAY 2.1 0.267 0.301 A 300 277 0 0 0 0 [[38, 290]] 1.0 1xr1 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 3A99A P11309 33 305 313.0 ANP:501 ATPlike Active DFGin 5.934 14.254 BLAminus -128.38, 171.59 60.85, 87.29 -96.61, 22.08 288.57, 75.78 -65.84, -9.23 in-in in 8.754 Saltbr-in 2.604 HRD-na-A -66.86, -47.45 66.12, 8.26 in-in-in SNCiii in-in ActLoopNT-in 2.889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.19, 26.41 APE9-dihe-na -87.51, -159.07 APE8-dihe-in -85.64, 119.66 APE8-rot-in 305.41 APE67-dihe-in -70.7, -5.81 -56.65, -39.81 APE12-dist-in 9.612 APE11-dist-in 8.461 APE10-dist-in 5.29 APE9-dist-in 3.778 None None None XRAY 1.6 0.187 0.206 A 320 273 0 0 0 0 [[38, 290]] 1.0 3a99 CAMK_PIM1_HUMAN CAMK 4.3e-65 225.5 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 2BZKB P11309 33 305 313.0 ANP:1306 ATPlike Active DFGin 6.126 14.443 BLAminus -123.86, 174.78 64.57, 79.13 -87.5, 17.23 286.98, 86.61 -67.5, -17.62 in-in in 8.781 Saltbr-in 2.727 HRD-na-A -70.49, -48.81 68.36, 6.4 in-in-in SNCiii in-in ActLoopNT-in 2.813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.63, 10.91 APE9-dihe-na -77.79, -156.22 APE8-dihe-in -90.85, 124.06 APE8-rot-in 315.85 APE67-dihe-in -68.94, -10.63 -60.69, -42.64 APE12-dist-in 9.464 APE11-dist-in 8.478 APE10-dist-in 4.851 APE9-dist-in 3.782 R250G None None XRAY 2.45 0.191 0.225 B 313 268 5 0 0 0 [[38, 290]] 1.0 2bzk CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK STK11 STK11_HUMAN 2WTKC Q15831 47 342 433.0 ANP:2 ATPlike Active DFGin 6.192 13.745 BLAminus -119.65, -175.81 55.97, 66.27 -90.3, 25.87 311.18, 25.77 -80.53, -8.11 in-in in 9.443 Saltbr-in 3.361 HRD-in -68.47, -42.92 70.9, -7.9 in-in-in SNCiii in-in ActLoopNT-in 2.648 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na 69.85, 15.07 APE9-dihe-na -72.04, -171.91 APE8-dihe-in -90.01, 115.78 APE8-rot-in 306.68 APE67-dihe-in -55.63, -13.05 -36.08, -60.58 APE12-dist-in 7.784 APE11-dist-in 9.233 APE10-dist-in 5.395 APE9-dist-in 3.173 D194A None None XRAY 2.65 0.24 0.291 C 305 285 3 0 0 0 [[49, 309]] 1.0 2wtk CAMK_STK11_HUMAN CAMK 7.7e-66 228.0 1 256 256 193 194 195 197 199 78 98 102 173 175 174 176 237 223 218 217 216 215 214 213 212 130 Serine/threonine-protein kinase STK11
CAMK STK11 STK11_HUMAN 2WTKF Q15831 45 340 433.0 ANP:4 ATPlike Active DFGin 5.938 13.841 BLAminus -119.11, -173.26 54.53, 62.76 -80.33, 19.16 295.83, 69.09 -48.31, -46.43 in-in in 9.483 Saltbr-in 3.568 HRD-in -68.65, -42.45 72.6, -14.65 in-in-in SNCiii in-in ActLoopNT-in 2.922 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na 45.91, 2.58 APE9-dihe-na -73.83, 178.68 APE8-dihe-in -66.98, 134.68 APE8-rot-in 293.57 APE67-dihe-in -65.1, -33.79 -54.08, -45.39 APE12-dist-in 8.609 APE11-dist-in 9.659 APE10-dist-in 5.793 APE9-dist-in 3.313 D194A None None XRAY 2.65 0.24 0.291 F 305 268 16 0 0 0 [[49, 309]] 1.0 2wtk CAMK_STK11_HUMAN CAMK 7.7e-66 228.0 1 256 256 193 194 195 197 199 78 98 102 173 175 174 176 237 223 218 217 216 215 214 213 212 130 Serine/threonine-protein kinase STK11
CK1 CSNK1D KC1D_HUMAN 6RU6A P48730 3 294 415.0 ACP:60301 ATPlike Active DFGin 6.436 15.264 BLAminus -136.56, 176.84 69.53, 73.53 -93.66, 24.95 289.84, 81.36 -61.77, -30.96 in-in in 7.923 Saltbr-in 2.789 HRD-in -77.83, -55.12 76.08, 12.52 in-in-in SNCiii in-in ActLoopNT-in 2.85 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.64, 119.59 APE9-dihe-na 102.6, -136.74 APE8-dihe-in -117.46, 127.27 APE8-rot-in 311.09 APE67-dihe-in -57.82, -37.85 -53.66, -47.41 APE12-dist-in 12.315 APE11-dist-in 11.908 APE10-dist-in 6.481 APE9-dist-in 3.505 None None None XRAY 2.05 0.213 0.257 A 296 288 4 0 0 0 [[9, 275]] 1.0 6ru6 CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7FA P48730 3 294 415.0 AMP:305 ATPlike Active DFGin 6.386 14.989 BLAminus -135.41, 179.24 65.29, 82.6 -99.51, 20.86 287.48, 77.77 -56.63, -36.85 in-in in 8.099 Saltbr-in 2.591 HRD-in -82.17, -51.93 74.76, 11.47 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -100.01, 118.96 APE9-dihe-na 109.81, -163.5 APE8-dihe-in -91.97, 119.49 APE8-rot-in 320.94 APE67-dihe-in -55.9, -38.32 -51.55, -37.41 APE12-dist-in 13.114 APE11-dist-in 12.585 APE10-dist-in 6.845 APE9-dist-in 3.948 None TPO220 TPO220 XRAY 1.96 0.19 0.221 A 296 292 0 0 0 0 [[9, 275]] 1.0 7p7f CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7FB P48730 3 294 415.0 AMP:310 ATPlike Active DFGin 6.389 15.041 BLAminus -134.9, -178.65 62.6, 84.78 -99.93, 21.19 288.23, 78.97 -57.89, -34.16 in-in in 8.117 Saltbr-in 2.593 HRD-in -86.23, -54.05 76.65, 11.34 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.84, 118.88 APE9-dihe-na 108.83, -162.51 APE8-dihe-in -93.95, 118.29 APE8-rot-in 320.41 APE67-dihe-in -55.93, -38.53 -50.49, -37.42 APE12-dist-in 13.14 APE11-dist-in 12.546 APE10-dist-in 6.804 APE9-dist-in 4.014 None TPO220 TPO220 XRAY 1.96 0.19 0.221 B 296 292 0 0 0 0 [[9, 275]] 1.0 7p7f CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7HA P48730 3 294 415.0 AMP:301 ATPlike Active DFGin 5.85 14.904 BLAminus -131.69, 175.32 69.71, 86.46 -98.17, 29.2 291.07, 84.43 -61.3, -36.51 in-in in 8.328 Saltbr-in 2.869 HRD-in -85.02, -56.99 74.97, 14.35 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.26, -19.24 APE9-dihe-na -88.34, -159.24 APE8-dihe-in -92.63, 127.36 APE8-rot-in 313.8 APE67-dihe-in -57.88, -32.21 -74.29, -29.96 APE12-dist-in 10.816 APE11-dist-in 12.399 APE10-dist-in 6.988 APE9-dist-in 4.101 None None None XRAY 2.4 0.225 0.268 A 296 292 0 0 0 0 [[9, 275]] 1.0 7p7h CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7HB P48730 3 294 415.0 AMP:301 ATPlike Active DFGin 5.843 14.916 BLAminus -130.5, 174.9 69.57, 86.72 -100.58, 28.91 292.34, 82.14 -57.01, -35.01 in-in in 8.325 Saltbr-in 2.918 HRD-in -84.55, -57.9 81.6, 9.08 in-in-in SNCiii in-in ActLoopNT-in 2.946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.93, 49.41 APE9-dihe-na 140.08, -131.01 APE8-dihe-in -99.84, 119.2 APE8-rot-in 321.52 APE67-dihe-in -56.55, -33.9 -75.78, -27.7 APE12-dist-in 12.421 APE11-dist-in 12.165 APE10-dist-in 7.215 APE9-dist-in 4.736 None None None XRAY 2.4 0.225 0.268 B 296 292 0 0 0 0 [[9, 275]] 1.0 7p7h CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 TTBK1 TTBK1_HUMAN 4BTJA Q5TCY1 21 312 1321.0 ADP:61337 ATPlike Active DFGin 5.513 12.699 BLAminus -122.16, 167.53 65.74, 92.18 -107.62, 12.94 309.85, 113.04 -64.35, -28.29 in-in in 7.127 Saltbr-in 2.757 HRD-in -79.44, -52.71 73.3, -5.89 in-in-in SNCiii in-in ActLoopNT-in 2.821 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.78, 143.11 APE9-dihe-na 98.14, -168.76 APE8-dihe-in -84.14, 153.12 APE8-rot-in 322.08 APE67-dihe-in -60.57, -38.77 -75.21, -43.81 APE12-dist-in 11.388 APE11-dist-in 11.45 APE10-dist-in 5.945 APE9-dist-in 3.412 None None None XRAY 2.16 0.179 0.197 A 337 292 0 0 0 0 [[34, 295]] 1.0 4btj CK1_TTBK1_HUMAN CK1 5.7e-105 356.4 1 262 262 175 176 177 179 181 63 77 81 151 153 152 154 221 209 204 203 202 201 200 199 198 108 Tau-tubulin kinase 1
CK1 TTBK1 TTBK1_HUMAN 4BTJB Q5TCY1 21 313 1321.0 ATP:61338 ATPlike Active DFGin 5.352 12.718 BLAminus -122.53, 168.88 60.17, 88.3 -98.51, 13.52 307.1, 115.33 -64.8, -32.06 in-in in 7.148 Saltbr-in 2.816 HRD-in -78.94, -51.75 72.7, -0.47 in-in-in SNCiii in-in ActLoopNT-in 2.748 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -105.82, -14.94 APE9-dihe-na -62.51, -161.18 APE8-dihe-in -100.71, 125.28 APE8-rot-in 309.68 APE67-dihe-in -55.66, -43.07 -52.23, -50.62 APE12-dist-in 11.078 APE11-dist-in 10.816 APE10-dist-in 6.463 APE9-dist-in 4.328 None None None XRAY 2.16 0.179 0.197 B 337 293 0 0 0 0 [[34, 295]] 1.0 4btj CK1_TTBK1_HUMAN CK1 5.7e-105 356.4 1 262 262 175 176 177 179 181 63 77 81 151 153 152 154 221 209 204 203 202 201 200 199 198 108 Tau-tubulin kinase 1
CK1 TTBK2 TTBK2_HUMAN 6VRFA Q6IQ55 9 298 1244.0 ADP:301 ATPlike Active DFGin 5.354 13.116 BLAminus -121.29, 164.21 73.75, 82.24 -97.72, 13.38 304.67, 116.94 -64.06, -29.66 in-in in 7.214 Saltbr-in 2.751 HRD-in -77.1, -49.95 73.69, -4.56 in-in-in SNCiii in-in ActLoopNT-in 2.813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -108.12, -30.06 APE9-dihe-na -84.65, -146.34 APE8-dihe-in -107.58, 129.44 APE8-rot-in 302.21 APE67-dihe-in -59.13, -37.2 -56.28, -42.66 APE12-dist-in 11.197 APE11-dist-in 11.387 APE10-dist-in 5.48 APE9-dist-in 3.784 None None None XRAY 1.5 0.175 0.209 A 299 287 3 0 0 0 [[21, 282]] 1.0 6vrf CK1_TTBK2_HUMAN CK1 7.7e-104 352.6 1 262 262 162 163 164 166 168 50 64 68 138 140 139 141 208 196 191 190 189 188 187 186 185 95 Tau-tubulin kinase 2
CK1 TTBK2 TTBK2_HUMAN 6VRFB Q6IQ55 9 298 1244.0 ADP:301 ATPlike Active DFGin 5.431 12.695 BLAminus -121.38, 163.64 74.07, 85.5 -102.64, 12.86 306.76, 116.33 -62.94, -32.7 in-in in 7.346 Saltbr-in 2.891 HRD-in -78.31, -51.54 73.55, 1.77 in-in-in SNCiii in-in ActLoopNT-in 2.86 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -109.78, -23.36 APE9-dihe-na -86.88, -149.11 APE8-dihe-in -108.63, 128.02 APE8-rot-in 302.45 APE67-dihe-in -58.2, -36.14 -56.96, -43.7 APE12-dist-in 11.039 APE11-dist-in 11.244 APE10-dist-in 5.337 APE9-dist-in 3.712 None None None XRAY 1.5 0.175 0.209 B 299 287 3 0 0 0 [[21, 282]] 1.0 6vrf CK1_TTBK2_HUMAN CK1 7.7e-104 352.6 1 262 262 162 163 164 166 168 50 64 68 138 140 139 141 208 196 191 190 189 188 187 186 185 95 Tau-tubulin kinase 2
CMGC CDK2 CDK2_HUMAN 4I3ZA P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.408 15.148 BLAminus -137.57, -176.06 52.96, 75.44 -91.33, 19.91 280.72, 70.75 -64.88, -19.38 in-in in 8.599 Saltbr-in 2.988 HRD-in -80.76, -55.87 72.55, 4.85 in-in-in SNCiii in-in ActLoopNT-in 2.901 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.11, -96.25 APE9-dihe-na -51.92, 142.27 APE8-dihe-in -55.11, 135.08 APE8-rot-in 307.48 APE67-dihe-in -54.58, -26.51 -40.4, -56.95 APE12-dist-in 13.064 APE11-dist-in 10.585 APE10-dist-in 6.823 APE9-dist-in 3.305 None TPO160 TPO160 XRAY 2.05 0.199 0.228 A 296 296 0 0 0 0 [[4, 286]] 1.0 4i3z CMGC_CDK2_HUMAN CMGC 6.2e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 4I3ZC P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.367 15.146 BLAminus -139.14, -175.0 51.64, 79.19 -95.11, 18.85 278.6, 70.91 -64.63, -17.11 in-in in 8.653 Saltbr-in 2.979 HRD-in -79.85, -55.96 72.81, 4.84 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.52, -96.18 APE9-dihe-na -52.61, 142.23 APE8-dihe-in -53.61, 133.4 APE8-rot-in 308.84 APE67-dihe-in -53.33, -28.57 -37.02, -58.54 APE12-dist-in 13.081 APE11-dist-in 10.618 APE10-dist-in 6.861 APE9-dist-in 3.305 None TPO160 TPO160 XRAY 2.05 0.199 0.228 C 296 296 0 0 0 0 [[4, 286]] 1.0 4i3z CMGC_CDK2_HUMAN CMGC 6.2e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHRA P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.557 15.107 BLAminus -129.61, -176.27 55.27, 75.32 -97.07, 17.79 280.43, 72.68 -60.79, -23.59 in-in in 8.696 Saltbr-in 2.88 HRD-in -78.46, -57.59 71.9, 8.99 in-in-in SNCiii in-in ActLoopNT-in 2.877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.99, 139.5 APE9-dihe-na 85.76, 129.74 APE8-dihe-in -56.31, 140.07 APE8-rot-in 302.24 APE67-dihe-in -65.07, -20.31 -41.24, -52.35 APE12-dist-in 12.989 APE11-dist-in 10.171 APE10-dist-in 7.111 APE9-dist-in 3.341 None TPO160 TPO160 XRAY 2.17 0.18 0.21 A 298 296 0 0 0 0 [[4, 286]] 1.0 3qhr CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHRC P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.565 15.121 BLAminus -133.25, -174.75 53.96, 72.74 -93.36, 15.91 281.14, 71.23 -60.56, -21.49 in-in in 8.7 Saltbr-in 2.868 HRD-in -78.47, -57.15 72.13, 9.85 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.81, 147.52 APE9-dihe-na 81.05, 137.24 APE8-dihe-in -64.2, 137.48 APE8-rot-in 304.68 APE67-dihe-in -62.37, -22.27 -38.55, -53.11 APE12-dist-in 12.985 APE11-dist-in 10.232 APE10-dist-in 6.99 APE9-dist-in 3.293 None TPO160 TPO160 XRAY 2.17 0.18 0.21 C 298 296 0 0 0 0 [[4, 286]] 1.0 3qhr CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHWA P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.435 15.013 BLAminus -134.08, -174.07 54.44, 75.18 -91.31, 13.19 281.29, 72.4 -60.66, -23.16 in-in in 8.64 Saltbr-in 2.934 HRD-in -72.46, -52.11 70.84, 4.06 in-in-in SNCiii in-in ActLoopNT-in 2.903 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.61, -86.88 APE9-dihe-na -62.59, 147.47 APE8-dihe-in -61.56, 138.19 APE8-rot-in 297.56 APE67-dihe-in -60.69, -27.39 -44.54, -49.89 APE12-dist-in 12.995 APE11-dist-in 10.23 APE10-dist-in 6.782 APE9-dist-in 3.359 None TPO160 TPO160 XRAY 1.91 0.189 0.219 A 298 296 0 0 0 0 [[4, 286]] 1.0 3qhw CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHWC P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.453 15.083 BLAminus -135.33, -175.53 57.5, 71.73 -89.85, 9.67 280.79, 72.12 -55.86, -26.79 in-in in 8.617 Saltbr-in 2.896 HRD-in -73.76, -53.15 71.96, 3.16 in-in-in SNCiii in-in ActLoopNT-in 2.898 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.86, -80.28 APE9-dihe-na -65.52, 146.91 APE8-dihe-in -61.19, 139.69 APE8-rot-in 298.69 APE67-dihe-in -57.2, -28.53 -47.15, -50.79 APE12-dist-in 12.997 APE11-dist-in 10.133 APE10-dist-in 6.722 APE9-dist-in 3.361 None TPO160 TPO160 XRAY 1.91 0.189 0.219 C 298 296 0 0 0 0 [[4, 286]] 1.0 3qhw CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1JSTA P24941 1 298 298.0 ATP:300 ATPlike Active DFGin 6.427 15.464 BLAminus -139.88, 179.46 48.93, 78.76 -92.24, 30.29 284.11, 71.63 -70.08, -30.4 in-in in 8.717 Saltbr-in 2.757 HRD-in -78.76, -47.67 60.69, 17.81 in-in-in SNCiii in-in ActLoopNT-in 2.949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.53, 164.64 APE9-dihe-na 80.72, 135.16 APE8-dihe-in -62.71, 138.95 APE8-rot-in 293.52 APE67-dihe-in -51.22, -30.94 -33.79, -62.16 APE12-dist-in 13.121 APE11-dist-in 11.934 APE10-dist-in 7.067 APE9-dist-in 3.277 None TPO160 TPO160 XRAY 2.6 0.2 999.0 A 298 298 0 0 0 0 [[4, 286]] 1.0 1jst CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1JSTC P24941 1 298 298.0 ATP:300 ATPlike Active DFGin 6.225 15.133 BLAminus -133.76, 179.75 53.92, 86.29 -100.05, 15.63 279.16, 71.07 -59.91, -21.96 in-in in 8.679 Saltbr-in 2.947 HRD-in -76.84, -49.3 61.77, 13.04 in-in-in SNCiii in-in ActLoopNT-in 2.701 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.31, -163.7 APE9-dihe-na 66.67, 148.27 APE8-dihe-in -72.61, 126.34 APE8-rot-in 301.65 APE67-dihe-in -51.49, -27.24 -26.21, -64.21 APE12-dist-in 13.412 APE11-dist-in 12.741 APE10-dist-in 6.942 APE9-dist-in 3.204 None TPO160 TPO160 XRAY 2.6 0.2 999.0 C 298 298 0 0 0 0 [[4, 286]] 1.0 1jst CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CJMA P24941 1 292 298.0 ATP:1294 ATPlike Active DFGin 6.412 15.477 BLAminus -133.49, 174.28 59.08, 80.72 -93.05, 17.33 280.25, 71.88 -51.1, -37.87 in-in in 8.875 Saltbr-in 3.027 HRD-in -83.77, -55.33 74.52, 15.85 in-in-in SNCiii in-in ActLoopNT-in 2.796 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.97, -48.89 APE9-dihe-na -98.03, 148.0 APE8-dihe-in -53.4, 136.55 APE8-rot-in 296.67 APE67-dihe-in -56.28, -31.52 -52.78, -45.83 APE12-dist-in 13.329 APE11-dist-in 10.553 APE10-dist-in 7.18 APE9-dist-in 3.464 None PTR15,TPO160 PTR15,TPO160 XRAY 2.3 0.204 0.265 A 298 287 5 0 0 0 [[4, 286]] 1.0 2cjm CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CJMC P24941 1 297 298.0 ATP:1298 ATPlike Active DFGin 6.446 15.389 BLAminus -136.23, -173.15 48.46, 78.84 -90.01, 21.15 280.3, 74.36 -53.78, -24.47 in-in in 8.957 Saltbr-in 2.575 HRD-in -82.67, -49.67 67.53, 9.26 in-in-in SNCiii in-in ActLoopNT-in 2.979 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.3, -72.35 APE9-dihe-na -81.21, 139.76 APE8-dihe-in -48.67, 128.86 APE8-rot-in 299.02 APE67-dihe-in -54.58, -22.4 -47.31, -51.92 APE12-dist-in 13.068 APE11-dist-in 10.808 APE10-dist-in 7.009 APE9-dist-in 3.58 None PTR15,TPO160 PTR15,TPO160 XRAY 2.3 0.204 0.265 C 298 297 0 0 0 0 [[4, 286]] 1.0 2cjm CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 4II5A P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.295 15.275 BLAminus -136.76, -174.67 48.15, 75.69 -89.27, 15.07 281.74, 67.11 -54.49, -30.0 in-in in 8.675 Saltbr-in 2.898 HRD-in -77.95, -58.94 72.46, 5.93 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.58, 147.66 APE9-dihe-na 74.72, 130.64 APE8-dihe-in -63.5, 139.49 APE8-rot-in 303.89 APE67-dihe-in -59.35, -27.46 -47.25, -50.52 APE12-dist-in 13.127 APE11-dist-in 10.372 APE10-dist-in 7.034 APE9-dist-in 3.344 None TPO160 TPO160 XRAY 2.15 0.2 0.226 A 298 296 0 0 0 0 [[4, 286]] 1.0 4ii5 CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 4II5C P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.289 15.288 BLAminus -134.89, -171.63 44.93, 79.89 -96.21, 16.02 275.02, 74.95 -60.79, -24.87 in-in in 8.666 Saltbr-in 2.94 HRD-in -77.09, -52.7 69.17, 3.7 in-in-in SNCiii in-in ActLoopNT-in 2.858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.65, 138.88 APE9-dihe-na 85.57, 133.69 APE8-dihe-in -65.51, 139.86 APE8-rot-in 305.2 APE67-dihe-in -60.76, -27.54 -47.35, -49.81 APE12-dist-in 13.141 APE11-dist-in 10.382 APE10-dist-in 7.061 APE9-dist-in 3.387 None TPO160 TPO160 XRAY 2.15 0.2 0.226 C 298 296 0 0 0 0 [[4, 286]] 1.0 4ii5 CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1GY3A P24941 1 296 298.0 ATP:1297 ATPlike Active DFGin 6.711 15.739 BLAminus -148.85, -171.85 44.28, 78.14 -91.55, 12.53 280.84, 73.84 -49.56, -35.56 in-in in 8.826 Saltbr-in 2.87 HRD-in -78.88, -56.55 74.04, 15.78 in-in-in SNCiii in-in ActLoopNT-in 3.129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.01, 152.98 APE9-dihe-na 75.99, 139.26 APE8-dihe-in -71.28, 139.34 APE8-rot-in 297.69 APE67-dihe-in -59.44, -30.42 -47.65, -49.93 APE12-dist-in 13.156 APE11-dist-in 10.678 APE10-dist-in 7.643 APE9-dist-in 3.395 None TPO160 TPO160 XRAY 2.7 0.25 0.313 A 299 296 0 0 0 0 [[4, 286]] 1.0 1gy3 CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1GY3C P24941 1 296 298.0 ATP:1298 ATPlike Active DFGin 6.824 15.376 BLAminus -159.42, -172.39 46.56, 69.8 -88.25, 18.8 278.1, 68.22 -63.28, -3.45 in-in in 8.61 Saltbr-in 3.316 HRD-in -72.89, -69.46 86.12, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.794 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.99, 145.31 APE9-dihe-na 77.28, 144.74 APE8-dihe-in -75.96, 137.92 APE8-rot-in 277.1 APE67-dihe-in -64.24, -30.46 -41.97, -49.4 APE12-dist-in 13.195 APE11-dist-in 10.636 APE10-dist-in 7.772 APE9-dist-in 3.212 None TPO160 TPO160 XRAY 2.7 0.25 0.313 C 299 296 0 0 0 0 [[4, 286]] 1.0 1gy3 CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1QMZA P24941 1 296 298.0 ATP:60381 ATPlike Active DFGin 6.424 15.17 BLAminus -146.26, -172.65 47.53, 78.45 -93.94, 24.34 280.23, 76.95 -74.2, -4.32 in-in in 8.74 Saltbr-in 2.663 HRD-in -79.61, -61.2 70.52, 19.43 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.31, 152.76 APE9-dihe-na 72.53, 130.75 APE8-dihe-in -60.65, 130.8 APE8-rot-in 293.88 APE67-dihe-in -60.7, -26.37 -33.48, -54.72 APE12-dist-in 13.02 APE11-dist-in 10.095 APE10-dist-in 7.17 APE9-dist-in 3.235 None TPO160 TPO160 XRAY 2.2 0.22 0.28 A 299 296 0 0 0 0 [[4, 286]] 1.0 1qmz CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1QMZC P24941 1 296 298.0 ATP:60381 ATPlike Active DFGin 6.512 15.134 BLAminus -147.61, -169.98 41.15, 80.53 -95.52, 25.6 283.09, 73.82 -79.03, -0.31 in-in in 8.74 Saltbr-in 2.54 HRD-in -75.88, -57.22 71.34, 18.39 in-in-in SNCiii in-in ActLoopNT-in 2.993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.04, 148.92 APE9-dihe-na 73.46, 130.58 APE8-dihe-in -61.75, 132.61 APE8-rot-in 296.97 APE67-dihe-in -70.09, -17.52 -37.4, -48.3 APE12-dist-in 12.947 APE11-dist-in 10.103 APE10-dist-in 7.19 APE9-dist-in 3.234 None TPO160 TPO160 XRAY 2.2 0.22 0.28 C 299 296 0 0 0 0 [[4, 286]] 1.0 1qmz CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCHA P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.648 15.496 BLAminus -138.14, 178.31 65.58, 62.78 -86.23, 16.74 281.6, 70.81 -63.75, -23.41 in-in in 8.795 Saltbr-in 2.828 HRD-in -78.21, -56.44 71.04, 15.24 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.4, 152.64 APE9-dihe-na 69.68, 132.94 APE8-dihe-in -57.07, 137.05 APE8-rot-in 294.63 APE67-dihe-in -60.03, -20.02 -46.03, -52.89 APE12-dist-in 13.198 APE11-dist-in 10.36 APE10-dist-in 7.208 APE9-dist-in 3.286 None TPO160 TPO160 XRAY 1.7 0.15 0.182 A 299 296 0 0 0 0 [[4, 286]] 1.0 2cch CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCHC P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.477 15.382 BLAminus -137.71, -178.58 51.07, 78.61 -96.17, 22.01 279.1, 72.77 -65.43, -25.94 in-in in 8.653 Saltbr-in 2.719 HRD-in -81.45, -53.09 63.51, 17.55 in-in-in SNCiii in-in ActLoopNT-in 2.886 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.56, 136.55 APE9-dihe-na 76.27, 128.23 APE8-dihe-in -59.37, 134.24 APE8-rot-in 303.33 APE67-dihe-in -63.22, -26.6 -41.45, -49.27 APE12-dist-in 12.866 APE11-dist-in 10.056 APE10-dist-in 7.377 APE9-dist-in 3.26 None TPO160 TPO160 XRAY 1.7 0.15 0.182 C 299 296 0 0 0 0 [[4, 286]] 1.0 2cch CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCIA P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.459 15.372 BLAminus -128.71, -173.86 48.01, 81.43 -98.73, 25.24 282.02, 74.31 -66.86, -20.71 in-in in 8.902 Saltbr-in 3.076 HRD-in -75.27, -47.91 58.22, 13.15 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.39, 140.99 APE9-dihe-na 76.14, 131.3 APE8-dihe-in -63.2, 133.24 APE8-rot-in 305.53 APE67-dihe-in -53.35, -21.65 -35.23, -63.18 APE12-dist-in 12.958 APE11-dist-in 10.323 APE10-dist-in 7.246 APE9-dist-in 3.291 None TPO160 TPO160 XRAY 2.7 0.264 0.321 A 299 296 0 0 0 0 [[4, 286]] 1.0 2cci CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCIC P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.232 15.382 BLAminus -129.31, 167.15 64.1, 86.76 -100.18, 28.53 276.86, 72.85 -63.26, -37.36 in-in in 8.551 Saltbr-in 2.666 HRD-in -73.66, -47.99 63.69, 10.4 in-in-in SNCiii in-in ActLoopNT-in 3.064 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.2, 138.6 APE9-dihe-na 71.13, 137.9 APE8-dihe-in -63.98, 129.66 APE8-rot-in 301.4 APE67-dihe-in -61.96, -9.78 -29.15, -60.17 APE12-dist-in 12.753 APE11-dist-in 9.767 APE10-dist-in 7.42 APE9-dist-in 3.234 None TPO160 TPO160 XRAY 2.7 0.264 0.321 C 299 296 0 0 0 0 [[4, 286]] 1.0 2cci CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK7 CDK7_HUMAN 9HIYJ P50613 10 310 346.0 AGS:60401 ATPlike Active DFGin 6.727 15.718 BLAminus -144.39, -174.23 58.17, 64.72 -87.83, 23.91 281.92, 72.77 -77.85, -11.75 in-in in 8.542 Saltbr-in 3.5 HRD-in -67.31, -50.64 65.74, 8.28 in-in-in SNCiii in-in ActLoopNT-in 2.733 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.25, 164.09 APE9-dihe-na 67.64, 142.62 APE8-dihe-in -59.57, 146.87 APE8-rot-in 317.63 APE67-dihe-in -64.96, -18.05 -61.86, -38.17 APE12-dist-in 13.579 APE11-dist-in 11.322 APE10-dist-in 6.933 APE9-dist-in 3.352 D97N None None EM 2.3 999.0 999.0 J 349 287 14 0 0 3 [[12, 295]] 1.0 9hiy CMGC_CDK7_HUMAN CMGC 1.8e-78 271.6 1 301 301 154 155 156 158 160 41 62 66 134 136 135 137 195 182 177 176 175 174 173 172 171 92 Cyclin-dependent kinase 7
CMGC CDK9 CDK9_HUMAN 3BLQA P50750 7 325 372.0 ATP:332 ATPlike Active DFGin 6.983 15.235 BLAminus -137.33, 167.71 61.72, 82.78 -101.54, 27.58 292.13, 71.79 -68.35, -20.47 in-in in 9.514 Saltbr-in 3.257 HRD-in -70.77, -57.41 73.91, 6.35 in-in-in SNCiii in-in ActLoopNT-in 2.85 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.28, 155.2 APE9-dihe-na 75.14, 129.25 APE8-dihe-in -51.14, 147.2 APE8-rot-in 304.68 APE67-dihe-in -62.86, -25.73 -50.2, -49.1 APE12-dist-in 13.028 APE11-dist-in 11.03 APE10-dist-in 6.896 APE9-dist-in 3.154 None TPO186 TPO186 XRAY 2.9 0.174 0.234 A 331 296 23 0 0 7 [[19, 315]] 1.0 3blq CMGC_CDK9_HUMAN CMGC 4.1e-80 275.1 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CDK9 CDK9_HUMAN 4IMYC P50750 8 330 372.0 AMP:401 ATPlike Active DFGin 6.789 15.123 BLAminus -140.61, 175.84 60.41, 77.79 -97.02, 19.01 284.69, 80.72 -68.98, -8.54 in-in in 9.232 Saltbr-in 2.833 HRD-in -67.68, -50.97 65.16, 13.16 in-in-in SNCiii in-in ActLoopNT-in 2.928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.81, 161.81 APE9-dihe-na 73.71, 135.92 APE8-dihe-in -53.34, 141.57 APE8-rot-in 294.85 APE67-dihe-in -61.16, -25.06 -47.9, -50.46 APE12-dist-in 13.386 APE11-dist-in 11.431 APE10-dist-in 7.006 APE9-dist-in 3.279 None TPO186 TPO186 XRAY 2.94 0.209 0.245 C 332 311 12 0 0 0 [[19, 315]] 1.0 4imy CMGC_CDK9_HUMAN CMGC 4.1e-80 275.1 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CDK9 CDK9_HUMAN 4IMYE P50750 8 330 372.0 AMP:401 ATPlike Active DFGin 6.794 15.112 BLAminus -141.41, 175.75 59.75, 77.9 -96.66, 19.65 284.44, 80.03 -69.65, -8.18 in-in in 9.197 Saltbr-in 2.816 HRD-in -68.02, -51.11 68.06, 12.23 in-in-in SNCiii in-in ActLoopNT-in 2.919 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.97, 161.65 APE9-dihe-na 74.14, 135.63 APE8-dihe-in -53.23, 140.74 APE8-rot-in 294.81 APE67-dihe-in -59.86, -25.62 -47.7, -50.88 APE12-dist-in 13.405 APE11-dist-in 11.437 APE10-dist-in 7.01 APE9-dist-in 3.278 None TPO186 TPO186 XRAY 2.94 0.209 0.245 E 332 314 9 0 0 0 [[19, 315]] 1.0 4imy CMGC_CDK9_HUMAN CMGC 4.1e-80 275.1 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CDK9 CDK9_HUMAN 3MIAA P50750 8 340 372.0 ANP:352 ATPlike Active DFGin 6.803 15.077 BLAminus -137.71, 176.33 64.58, 74.97 -96.55, 26.44 284.7, 90.38 -67.18, -14.54 in-in in 9.313 Saltbr-in 2.689 HRD-in -70.81, -51.43 63.16, 28.9 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.04, 160.49 APE9-dihe-na 82.03, 127.94 APE8-dihe-in -49.75, 143.51 APE8-rot-in 280.63 APE67-dihe-in -52.26, -14.47 -51.96, -57.94 APE12-dist-in 13.258 APE11-dist-in 11.524 APE10-dist-in 6.949 APE9-dist-in 3.523 None TPO186 TPO186 XRAY 3.0 0.219 0.287 A 351 325 8 0 0 0 [[19, 315]] 1.0 3mia CMGC_CDK9_HUMAN CMGC 5.1e-80 274.8 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CSNK2A1 CSK21_HUMAN 3JUHA P68400 2 335 391.0 ANP:339 ATPlike Active DFGin 7.401 16.242 BLAminus -115.69, -178.29 60.62, 71.57 -93.06, 11.37 295.1, 82.09 -62.22, -22.13 in-in in 9.721 Saltbr-in 2.746 HRD-in -70.06, -49.94 64.15, 21.46 in-in-in SNCiii in-in ActLoopNT-in 2.862 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.98, 153.86 APE9-dihe-na 70.33, -177.46 APE8-dihe-in -104.19, 142.14 APE8-rot-in 291.28 APE67-dihe-in -67.33, -12.83 -40.87, -55.27 APE12-dist-in 12.316 APE11-dist-in 9.578 APE10-dist-in 6.044 APE9-dist-in 3.086 V66A,M163L None None XRAY 1.66 0.158 0.218 A 335 334 0 0 0 0 [[39, 324]] 1.0 3juh CMGC_CSNK2A1_HUMAN CMGC 1.1e-70 244.1 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 3JUHB P68400 2 335 391.0 ANP:339 ATPlike Active DFGin 7.492 16.356 BLAminus -124.69, -176.29 51.46, 71.26 -80.35, 23.48 299.01, 83.37 -80.68, -22.43 in-in in 9.852 Saltbr-in 2.699 HRD-in -76.38, -50.5 78.84, -1.13 in-in-in SNCiii in-in ActLoopNT-in 2.807 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.59, 175.23 APE9-dihe-na 56.07, 138.8 APE8-dihe-in -58.03, 149.04 APE8-rot-in 282.66 APE67-dihe-in -69.98, -19.52 -43.94, -46.02 APE12-dist-in 12.714 APE11-dist-in 9.541 APE10-dist-in 5.884 APE9-dist-in 3.411 V66A,M163L None None XRAY 1.66 0.158 0.218 B 335 334 0 0 0 0 [[39, 324]] 1.0 3juh CMGC_CSNK2A1_HUMAN CMGC 1.1e-70 244.1 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 6Z19B P68400 2 329 391.0 ADP:401 ATPlike Active DFGin 7.399 16.102 BLAminus -106.47, -175.56 60.6, 79.25 -100.03, 20.37 297.28, 82.12 -73.41, -21.13 in-in in 8.717 Saltbr-in 2.8 HRD-in -71.6, -55.48 75.88, 3.64 in-in-in SNCiii in-in ActLoopNT-in 2.928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.14, 153.25 APE9-dihe-na 78.4, 166.67 APE8-dihe-in -74.52, 152.52 APE8-rot-in 285.35 APE67-dihe-in -64.18, -23.8 -57.77, -45.77 APE12-dist-in 12.968 APE11-dist-in 10.993 APE10-dist-in 6.495 APE9-dist-in 3.591 None None None XRAY 1.47 0.19 0.221 B 328 328 0 0 0 0 [[39, 324]] 1.0 6z19 CMGC_CSNK2A1_HUMAN CMGC 1.2e-69 240.7 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 3NSZA P68400 2 328 391.0 ANP:1000 ATPlike Active DFGin 7.29 16.639 BLAminus -116.89, -174.28 57.53, 72.95 -91.24, 19.04 295.43, 81.74 -67.97, -19.44 in-in in 9.56 Saltbr-in 2.721 HRD-in -71.38, -46.87 68.1, 12.99 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.59, 174.99 APE9-dihe-na 61.7, -173.37 APE8-dihe-in -118.84, 140.8 APE8-rot-in 296.4 APE67-dihe-in -69.07, -13.11 -30.5, -60.15 APE12-dist-in 12.605 APE11-dist-in 10.316 APE10-dist-in 6.145 APE9-dist-in 2.961 None None None XRAY 1.3 0.169 0.187 A 330 327 0 0 0 0 [[39, 324]] 1.0 3nsz CMGC_CSNK2A1_HUMAN CMGC 1.3e-69 240.7 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 1PJKA P68400 2 332 391.0 ANP:340 ATPlike Active DFGin 7.44 16.238 BLAminus -115.92, -179.78 53.21, 80.99 -96.44, 28.53 295.64, 78.1 -72.28, -30.66 in-in in 8.93 Saltbr-in 2.81 HRD-in -80.54, -40.11 57.34, 9.1 in-in-in SNCiii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.58, 173.24 APE9-dihe-na 63.2, 174.94 APE8-dihe-in -93.15, 157.9 APE8-rot-in 277.8 APE67-dihe-in -66.77, -23.27 -54.74, -47.48 APE12-dist-in 13.026 APE11-dist-in 10.669 APE10-dist-in 6.368 APE9-dist-in 3.173 None None None XRAY 2.5 0.188 0.257 A 334 331 0 0 0 0 [[39, 324]] 1.0 1pjk CMGC_CSNK2A1_HUMAN CMGC 1.3e-69 240.6 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 2PVRA P68400 2 329 391.0 ANP:6004 ATPlike Active DFGin 7.492 16.497 BLAminus -121.67, -179.6 56.35, 70.32 -89.0, 17.49 296.64, 81.69 -72.81, -15.87 in-in in 9.284 Saltbr-in 2.7 HRD-in -75.03, -46.77 70.22, 6.37 in-in-in SNCiii in-in ActLoopNT-in 2.86 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.8, 175.01 APE9-dihe-na 60.61, 163.14 APE8-dihe-in -93.89, 147.69 APE8-rot-in 305.18 APE67-dihe-in -67.68, -15.16 -34.32, -58.13 APE12-dist-in 12.728 APE11-dist-in 10.346 APE10-dist-in 6.131 APE9-dist-in 3.189 None None None XRAY 1.605 0.187 0.241 A 334 328 0 0 0 0 [[39, 324]] 1.0 2pvr CMGC_CSNK2A1_HUMAN CMGC 1.3e-69 240.6 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 3U87B P68400 2 331 391.0 ANP:60401 ATPlike Active DFGin 7.471 16.335 BLAminus -123.33, -169.35 50.94, 85.5 -106.65, 24.88 299.58, 83.47 -72.97, -19.72 in-in in 9.505 Saltbr-in 2.848 HRD-in -72.0, -49.6 70.96, 8.41 in-in-in SNCiii in-in ActLoopNT-in 2.78 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.34, 168.89 APE9-dihe-na 66.61, 166.24 APE8-dihe-in -76.34, 153.62 APE8-rot-in 296.27 APE67-dihe-in -70.99, -10.83 -52.99, -46.79 APE12-dist-in 12.822 APE11-dist-in 10.801 APE10-dist-in 6.15 APE9-dist-in 3.577 None None None XRAY 2.9 0.187 0.218 B 349 324 0 0 0 0 [[39, 324]] 1.0 3u87 CMGC_CSNK2A1_HUMAN CMGC 1.5e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5OQUB P68400 4 327 391.0 ADP:401 ATPlike Active DFGin 7.324 16.392 BLAminus -107.74, -171.87 52.49, 78.62 -101.36, 19.11 291.9, 83.91 -71.23, -12.83 in-in in 9.496 Saltbr-in 2.901 HRD-in -65.86, -46.78 65.2, 13.55 in-in-in SNCiii in-in ActLoopNT-in 2.895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.87, 169.85 APE9-dihe-na 66.11, 165.52 APE8-dihe-in -87.57, 142.09 APE8-rot-in 294.71 APE67-dihe-in -65.28, -26.45 -36.1, -50.26 APE12-dist-in 12.592 APE11-dist-in 10.419 APE10-dist-in 6.089 APE9-dist-in 3.154 R21S None None XRAY 2.324 0.221 0.244 B 352 324 0 0 0 0 [[39, 324]] 1.0 5oqu CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5ORKB P68400 4 326 391.0 ADP:401 ATPlike Active DFGin 7.365 16.488 BLAminus -111.04, -174.54 54.53, 77.94 -96.47, 19.83 296.01, 82.36 -66.2, -23.13 in-in in 9.552 Saltbr-in 3.041 HRD-in -70.69, -49.04 67.52, 16.07 in-in-in SNCiii in-in ActLoopNT-in 2.862 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.56, 172.18 APE9-dihe-na 65.73, 167.16 APE8-dihe-in -89.89, 143.95 APE8-rot-in 298.57 APE67-dihe-in -64.35, -23.63 -31.56, -56.57 APE12-dist-in 12.614 APE11-dist-in 10.418 APE10-dist-in 6.062 APE9-dist-in 3.149 R21S None None XRAY 2.143 0.217 0.243 B 352 323 0 0 0 0 [[39, 324]] 1.0 5ork CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 7QUXA P68400 2 329 391.0 ADP:60401 ATPlike Active DFGin 7.585 16.194 BLAminus -111.52, -172.63 60.82, 80.19 -104.84, 23.49 298.85, 85.23 -72.93, -20.15 in-in in 8.958 Saltbr-in 2.838 HRD-in -72.19, -52.24 72.27, 9.35 in-in-in SNCiii in-in ActLoopNT-in 2.846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.66, 178.74 APE9-dihe-na 61.29, -172.26 APE8-dihe-in -113.53, 144.19 APE8-rot-in 304.18 APE67-dihe-in -65.08, -18.11 -36.49, -57.4 APE12-dist-in 12.723 APE11-dist-in 10.579 APE10-dist-in 6.214 APE9-dist-in 2.896 None SEP2 SEP2 XRAY 1.48 0.181 0.204 A 352 328 0 0 0 0 [[39, 324]] 1.0 7qux CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 6YZHA P68400 3 329 391.0 ADP:60403 ATPlike Active DFGin 7.386 16.31 BLAminus -108.01, -176.38 61.1, 79.34 -99.78, 17.26 297.37, 82.49 -78.41, -8.16 in-in in 9.131 Saltbr-in 2.829 HRD-in -74.51, -47.7 69.86, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.83, 175.48 APE9-dihe-na 62.95, -168.81 APE8-dihe-in -126.52, 135.38 APE8-rot-in 299.93 APE67-dihe-in -66.68, -18.66 -34.87, -54.46 APE12-dist-in 12.682 APE11-dist-in 10.343 APE10-dist-in 6.227 APE9-dist-in 3.084 None None None XRAY 1.19 0.173 0.19 A 398 327 0 0 0 0 [[39, 324]] 1.0 6yzh CMGC_CSNK2A1_HUMAN CMGC 2.4e-69 239.8 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU6A P68400 3 329 391.0 ATP:401 ATPlike Active DFGin 7.373 16.301 BLAminus -117.96, -176.97 52.74, 80.35 -94.88, 19.06 296.35, 83.62 -69.11, -18.98 in-in in 9.296 Saltbr-in 2.997 HRD-in -73.54, -48.21 69.17, 10.55 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.92, 173.11 APE9-dihe-na 58.61, 170.65 APE8-dihe-in -94.81, 150.1 APE8-rot-in 295.17 APE67-dihe-in -71.66, -13.32 -37.08, -56.84 APE12-dist-in 12.652 APE11-dist-in 10.334 APE10-dist-in 6.182 APE9-dist-in 3.146 R21S,K74A,K75A,K76A None None XRAY 1.36 0.188 0.209 A 328 327 0 0 0 0 [[39, 324]] 1.0 5cu6 CMGC_CSNK2A1_HUMAN CMGC 8.1e-69 238.0 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A2 CSK22_HUMAN 8QCGB P19784 7 333 350.0 ANP:401 ATPlike Active DFGin 7.314 16.209 BLAminus -113.91, -178.96 61.11, 75.42 -92.86, 17.98 298.38, 79.8 -69.62, -20.0 in-in in 9.436 Saltbr-in 2.83 HRD-in -72.51, -49.6 69.57, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.828 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.91, 170.94 APE9-dihe-na 61.2, 166.37 APE8-dihe-in -93.43, 149.98 APE8-rot-in 300.62 APE67-dihe-in -69.2, -15.18 -40.28, -54.89 APE12-dist-in 12.657 APE11-dist-in 10.295 APE10-dist-in 6.172 APE9-dist-in 3.11 C336S None None XRAY 1.04 0.151 0.17 B 364 327 0 0 0 0 [[40, 325]] 1.0 8qcg CMGC_CSNK2A2_HUMAN CMGC 1e-69 241.0 1 301 301 175 176 177 179 181 69 82 86 154 156 155 157 215 202 197 196 195 194 193 192 191 115 Casein kinase II subunit alpha'
CMGC DYRK1A DYR1A_HUMAN 7A4OA Q13627 136 481 763.0 ANP:501 ATPlike Active DFGin 7.404 15.034 BLAminus -121.6, 173.77 67.88, 73.96 -92.34, 22.26 284.87, 82.1 -70.26, -21.97 in-in in 8.684 Saltbr-in 2.793 HRD-in -65.03, -49.19 79.83, -0.94 in-in-in SNCiii in-in ActLoopNT-in 2.8 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.61, 174.39 APE9-dihe-na 70.74, 151.67 APE8-dihe-in -72.34, 134.57 APE8-rot-in 295.77 APE67-dihe-in -65.19, -24.46 -43.45, -47.13 APE12-dist-in 10.098 APE11-dist-in 12.237 APE10-dist-in 7.723 APE9-dist-in 3.156 None PTR321 PTR321 XRAY 1.9 0.18 0.203 A 382 341 5 0 0 0 [[159, 479]] 1.0 7a4o CMGC_DYRK1A_HUMAN CMGC 1e-90 310.0 1 301 301 306 307 308 310 312 188 203 207 284 286 285 287 343 331 326 325 324 323 322 321 320 239 Dual specificity tyrosine-phosphorylation-regulated kinase 1A
CMGC GSK3B GSK3B_HUMAN 4NM5A P49841 24 383 420.0 ADP:60401 ATPlike Active DFGin 6.55 14.006 BLAminus -136.16, -177.73 61.88, 88.47 -108.64, 28.76 287.87, 80.78 -73.66, -15.44 in-in in 8.619 Saltbr-in 2.673 HRD-in -65.83, -43.73 64.82, 15.23 in-in-in SNCiii in-in ActLoopNT-in 2.839 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.92, 173.97 APE9-dihe-na 66.26, 147.02 APE8-dihe-in -77.1, 152.8 APE8-rot-in 293.28 APE67-dihe-inflip 82.03, -25.76 -52.23, 150.7 APE12-dist-in 13.279 APE11-dist-in 11.599 APE10-dist-in 6.949 APE9-dist-in 3.238 None None None XRAY 2.3 0.185 0.232 A 377 360 0 0 0 0 [[56, 340]] 1.0 4nm5 CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 4NM7A P49841 25 383 420.0 ADP:60401 ATPlike Active DFGin 6.515 13.993 BLAminus -137.35, -178.06 62.82, 88.6 -107.3, 24.56 288.41, 80.2 -69.84, -12.63 in-in in 8.818 Saltbr-in 2.743 HRD-in -66.5, -46.64 67.84, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.829 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 172.54 APE9-dihe-na 68.99, 153.43 APE8-dihe-in -86.9, 151.79 APE8-rot-in 300.04 APE67-dihe-inflip 84.67, -25.93 -50.38, 146.2 APE12-dist-in 13.355 APE11-dist-in 11.678 APE10-dist-in 6.905 APE9-dist-in 3.21 None None None XRAY 2.3 0.185 0.234 A 377 354 2 0 0 0 [[56, 340]] 1.0 4nm7 CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 4NM3A P49841 6 383 420.0 ADP:60409 ATPlike Active DFGin 6.475 13.947 BLAminus -129.98, -178.05 63.17, 87.87 -103.96, 21.26 289.38, 80.04 -65.46, -16.35 in-in in 8.806 Saltbr-in 2.726 HRD-in -69.81, -46.77 71.59, 6.75 in-in-in SNCiii in-in ActLoopNT-in 2.75 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.34, 169.99 APE9-dihe-na 69.15, 146.37 APE8-dihe-in -83.47, 151.55 APE8-rot-in 296.54 APE67-dihe-inflip 86.0, -31.11 -49.79, 146.79 APE12-dist-in 13.269 APE11-dist-in 11.484 APE10-dist-in 6.907 APE9-dist-in 3.112 None SEP9 SEP9 XRAY 2.1 0.197 0.242 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nm3 CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1BA P49841 35 388 420.0 ANP:60430 ATPlike Active DFGin 6.767 13.788 BLAminus -136.8, -178.88 61.6, 83.12 -97.64, 25.1 286.09, 80.4 -68.7, -13.11 in-in in 8.566 Saltbr-in 2.59 HRD-in -71.16, -45.98 70.36, 3.88 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.52, 175.26 APE9-dihe-na 75.44, 133.64 APE8-dihe-in -75.76, 147.49 APE8-rot-in 306.57 APE67-dihe-inflip 98.15, -33.72 -56.43, 141.52 APE12-dist-in 13.056 APE11-dist-in 10.974 APE10-dist-in 5.893 APE9-dist-in 3.112 None None None XRAY 1.8 0.216 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1b CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1BB P49841 23 386 420.0 ANP:60930 ATPlike Active DFGin 6.609 13.669 BLAminus -136.4, -177.03 61.49, 81.88 -98.08, 27.2 288.49, 82.07 -71.33, -13.14 in-in in 8.457 Saltbr-in 2.713 HRD-in -67.51, -45.87 68.87, 6.43 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.88, 174.17 APE9-dihe-na 76.18, 138.08 APE8-dihe-in -76.12, 141.41 APE8-rot-in 301.11 APE67-dihe-inflip 98.0, -37.59 -54.78, 144.25 APE12-dist-in 12.978 APE11-dist-in 11.066 APE10-dist-in 6.011 APE9-dist-in 3.174 None None None XRAY 1.8 0.216 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1b CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1CA P49841 35 388 420.0 ADP:60430 ATPlike Active DFGin 6.812 13.93 BLAminus -139.24, -179.75 62.79, 82.17 -97.34, 25.19 286.68, 82.3 -65.83, -19.9 in-in in 8.601 Saltbr-in 2.647 HRD-in -68.65, -43.85 68.34, 7.36 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.05, 172.96 APE9-dihe-na 78.17, 130.85 APE8-dihe-in -73.54, 145.97 APE8-rot-in 310.16 APE67-dihe-inflip 99.09, -35.01 -54.43, 141.28 APE12-dist-in 13.077 APE11-dist-in 11.067 APE10-dist-in 5.926 APE9-dist-in 3.2 None None None XRAY 2.1 0.218 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1c CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1CB P49841 23 386 420.0 ADP:60930 ATPlike Active DFGin 6.694 13.709 BLAminus -138.27, -179.99 63.33, 82.68 -100.46, 28.2 289.88, 80.26 -70.45, -13.94 in-in in 8.52 Saltbr-in 2.738 HRD-in -67.92, -43.36 67.59, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.71, 170.27 APE9-dihe-na 78.71, 139.86 APE8-dihe-in -81.56, 140.05 APE8-rot-in 302.5 APE67-dihe-inflip 101.62, -36.53 -50.52, 137.44 APE12-dist-in 12.868 APE11-dist-in 11.128 APE10-dist-in 6.025 APE9-dist-in 3.208 None None None XRAY 2.1 0.218 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1c CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 8XN6A P49841 35 384 420.0 ANP:501 ATPlike Active DFGin 6.682 13.862 BLAminus -137.72, 173.39 67.73, 84.48 -99.84, 22.57 287.77, 80.54 -65.33, -24.58 in-in in 8.463 Saltbr-in 2.63 HRD-in -71.05, -47.88 67.82, 15.5 in-in-in SNCiii in-in ActLoopNT-in 3.054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.0, 164.43 APE9-dihe-na 85.44, 135.36 APE8-dihe-in -74.2, 151.55 APE8-rot-in 291.81 APE67-dihe-in -69.28, -17.83 -36.59, -67.98 APE12-dist-in 12.907 APE11-dist-in 10.787 APE10-dist-in 5.68 APE9-dist-in 3.182 None None None XRAY 2.4 0.194 0.242 A 421 350 0 0 0 0 [[56, 340]] 1.0 8xn6 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1PYXA P49841 35 386 420.0 ANP:1001 ATPlike Active DFGin 6.584 13.622 BLAminus -138.81, -178.07 65.18, 79.92 -98.83, 26.07 289.95, 78.27 -73.24, -7.6 in-in in 8.373 Saltbr-in 2.765 HRD-in -67.79, -47.84 71.28, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.12, 170.17 APE9-dihe-na 80.64, 129.74 APE8-dihe-in -63.79, 140.05 APE8-rot-in 299.48 APE67-dihe-in -56.43, -21.61 -20.65, -80.28 APE12-dist-in 12.903 APE11-dist-in 10.937 APE10-dist-in 5.784 APE9-dist-in 3.15 None None None XRAY 2.4 0.206 0.233 A 422 343 9 0 0 0 [[56, 340]] 1.0 1pyx CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1PYXB P49841 35 383 420.0 ANP:2001 ATPlike Active DFGin 6.593 13.718 BLAminus -140.94, -178.47 65.26, 79.98 -98.11, 22.32 290.75, 76.51 -68.32, -7.73 in-in in 8.488 Saltbr-in 2.666 HRD-in -69.98, -47.18 70.83, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.3, 169.41 APE9-dihe-na 81.27, 131.24 APE8-dihe-in -66.67, 140.79 APE8-rot-in 300.74 APE67-dihe-in -56.9, -22.2 -20.58, -79.9 APE12-dist-in 12.838 APE11-dist-in 10.861 APE10-dist-in 5.718 APE9-dist-in 3.132 None None None XRAY 2.4 0.206 0.233 B 422 338 11 0 0 0 [[56, 340]] 1.0 1pyx CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC MAPK1 MK01_HUMAN 6OPGA P28482 10 358 360.0 ANP:60401 ATPlike Active DFGin 6.535 14.668 BLAminus -130.49, -173.97 55.35, 72.85 -87.66, 25.26 285.94, 65.79 -65.31, -19.22 in-in in 9.066 Saltbr-in 2.695 HRD-in -72.87, -54.34 77.9, 3.87 in-in-in SNCiii in-in ActLoopNT-in 2.758 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -102.35, 163.88 APE9-dihe-na 79.13, 168.47 APE8-dihe-in -88.92, 138.85 APE8-rot-in 292.11 APE67-dihe-in -68.23, -14.82 -51.35, -45.86 APE12-dist-in 12.57 APE11-dist-in 11.134 APE10-dist-in 6.653 APE9-dist-in 2.942 None TPO185,PTR187 TPO185,PTR187 XRAY 2.9 0.16 0.239 A 354 349 0 0 0 0 [[25, 313]] 1.0 6opg CMGC_MAPK1_HUMAN CMGC 8.6e-86 293.8 1 301 301 166 167 168 170 172 54 71 75 146 148 147 149 210 197 192 191 190 189 188 187 186 106 Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 5V60A P28482 10 358 360.0 ACP:401 ATPlike Active DFGin 6.669 14.887 BLAminus -124.21, -175.27 60.56, 75.29 -91.11, 25.45 286.11, 68.09 -67.4, -23.76 in-in in 9.269 Saltbr-in 3.088 HRD-in -75.88, -52.24 69.24, 12.32 in-in-in SNCiii in-in ActLoopNT-in 2.951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.66, 171.23 APE9-dihe-na 66.7, 168.41 APE8-dihe-in -89.68, 141.19 APE8-rot-in 301.48 APE67-dihe-in -66.12, -19.67 -43.41, -50.15 APE12-dist-in 12.574 APE11-dist-in 11.086 APE10-dist-in 6.633 APE9-dist-in 2.987 None TPO185,PTR187 TPO185,PTR187 XRAY 2.18 0.193 0.226 A 356 349 0 0 0 0 [[25, 313]] 1.0 5v60 CMGC_MAPK1_HUMAN CMGC 8.8e-86 293.8 1 301 301 166 167 168 170 172 54 71 75 146 148 147 149 210 197 192 191 190 189 188 187 186 106 Mitogen-activated protein kinase 1
CMGC MAPK12 MK12_HUMAN 1CM8A P53778 8 353 367.0 ANP:60400 ATPlike Active DFGin 6.965 14.774 BLAminus -109.08, -177.81 49.88, 82.62 -94.66, 21.96 279.65, 74.31 -61.38, -21.21 in-in in 9.0 Saltbr-in 2.777 HRD-in -80.35, -48.18 64.34, 20.91 in-in-in SNCiii in-in ActLoopNT-in 2.793 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.88, 159.85 APE9-dihe-na 73.62, 141.22 APE8-dihe-in -70.32, 134.6 APE8-rot-in 295.09 APE67-dihe-in -62.17, -12.08 -34.13, -61.33 APE12-dist-in 11.604 APE11-dist-in 10.956 APE10-dist-in 6.991 APE9-dist-in 3.072 None TPO183,PTR185 TPO183,PTR185 XRAY 2.4 0.232 0.283 A 367 329 6 0 0 0 [[27, 311]] 1.0 1cm8 CMGC_MAPK12_HUMAN CMGC 5.6e-85 291.2 1 301 301 170 171 172 174 176 56 74 78 150 152 151 153 208 195 190 189 188 187 186 185 184 110 Mitogen-activated protein kinase 12
CMGC MAPK12 MK12_HUMAN 1CM8B P53778 8 353 367.0 ANP:61400 ATPlike Active DFGin 6.965 14.794 BLAminus -106.93, -177.79 50.51, 81.99 -94.3, 22.09 279.91, 74.94 -61.07, -21.75 in-in in 9.031 Saltbr-in 2.759 HRD-in -80.7, -47.04 63.03, 19.82 in-in-in SNCiii in-in ActLoopNT-in 2.817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.88, 160.62 APE9-dihe-na 73.12, 141.25 APE8-dihe-in -70.38, 133.34 APE8-rot-in 295.67 APE67-dihe-in -62.05, -11.85 -33.55, -61.0 APE12-dist-in 11.613 APE11-dist-in 10.95 APE10-dist-in 6.996 APE9-dist-in 3.048 None TPO183,PTR185 TPO183,PTR185 XRAY 2.4 0.232 0.283 B 367 329 6 0 0 0 [[27, 311]] 1.0 1cm8 CMGC_MAPK12_HUMAN CMGC 5.6e-85 291.2 1 301 301 170 171 172 174 176 56 74 78 150 152 151 153 208 195 190 189 188 187 186 185 184 110 Mitogen-activated protein kinase 12
CMGC SRPK1 SRPK1_HUMAN 1WBPA Q96SB4 67 655 655.0 ADP:60950 ATPlike Active DFGin 6.093 14.484 BLAminus -120.66, 177.09 55.57, 73.12 -93.78, 28.92 297.48, 63.42 -60.8, -41.52 in-in in 9.616 Saltbr-in 3.534 HRD-in -64.25, -33.37 61.64, -4.85 in-in-in SNCiii in-in ActLoopNT-in 2.855 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.23, 175.25 APE9-dihe-na 64.87, 133.49 APE8-dihe-in -68.33, 140.58 APE8-rot-in 294.72 APE67-dihe-in -48.4, -19.96 -25.96, -79.02 APE12-dist-in 12.421 APE11-dist-in 10.401 APE10-dist-in 7.455 APE9-dist-in 2.973 None None None XRAY 2.4 0.228 0.247 A 397 350 22 0 0 0 [[80, 653]] 1.0 1wbp CMGC_SRPK1_HUMAN CMGC 2e-139 469.9 1 301 301 496 497 498 500 502 109 124 128 210 212 211 213 533 521 516 515 514 513 512 511 510 166 SRSF protein kinase 1
OTHER HASPIN HASP_HUMAN 3DLZA Q8TF76 470 798 798.0 AMP:902 ATPlike Active DFGin 5.254 12.469 BLAminus -120.14, 174.05 73.32, 91.07 -105.92, 29.14 315.79, 130.04 -57.27, -36.15 in-in in 9.264 Saltbr-in 2.695 HRD-na-N -71.0, -49.07 68.99, 3.03 in-in-na SNCiia in-na ActLoopNT-in 2.821 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -122.28, 17.39 APE9-dihe-na -67.57, 157.85 APE8-dihe-na -149.51, 177.99 APE8-rot-na 58.52 APE67-dihe-na -159.03, 144.74 95.06, -6.22 APE12-dist-na 9.493 APE11-dist-na 13.466 APE10-dist-na 17.05 APE9-dist-na 12.819 None None None XRAY 1.85 0.167 0.216 A 357 329 0 0 0 0 [[484, 797]] 1.0 3dlz OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
OTHER TP53RK PRPK_HUMAN 6WQXC Q96S44 17 247 253.0 ANP:301 ATPlike Active DFGin 5.95 14.251 BLAminus -146.19, 177.42 55.9, 80.94 -109.82, 15.46 288.95, 83.65 -50.48, -21.92 in-in in 7.493 Saltbr-in 2.923 HRD-in -69.98, -47.0 96.04, -14.43 in-in-na SNCiia in-na ActLoopNT-in 2.804 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -67.54, -42.02 APE9-dihe-na -66.2, -40.19 APE8-dihe-na -55.79, -43.62 APE8-rot-na 183.14 APE67-dihe-na -65.72, -35.03 -54.78, -48.19 APE12-dist-na 16.724 APE11-dist-na 12.036 APE10-dist-na 14.577 APE9-dist-na 11.741 None None None XRAY 2.53 0.214 0.265 C 267 231 6 0 0 0 [[32, 253]] 1.0 6wqx OTHER_TP53RK_HUMAN TP53RK 1.2e-114 387.3 1 224 224 182 183 184 186 188 60 84 88 159 161 160 162 199 205 200 199 198 197 196 195 194 114 EKC/KEOPS complex subunit TP53RK
OTHER TP53RK PRPK_HUMAN 6WQXD Q96S44 18 247 253.0 ANP:301 ATPlike Active DFGin 6.043 14.258 BLAminus -133.24, 171.19 66.42, 73.64 -108.34, 16.47 289.91, 91.17 -66.2, -15.73 in-in in 7.377 Saltbr-in 2.505 HRD-in -60.03, -49.96 100.64, -20.8 in-in-na SNCiia in-na ActLoopNT-in 2.816 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -66.35, -39.45 APE9-dihe-na -58.51, -49.84 APE8-dihe-na -58.36, -37.8 APE8-rot-na 168.78 APE67-dihe-na -71.45, -37.84 -63.19, -40.46 APE12-dist-na 16.676 APE11-dist-na 12.07 APE10-dist-na 14.499 APE9-dist-na 11.469 None None None XRAY 2.53 0.214 0.265 D 267 230 6 0 0 0 [[32, 253]] 1.0 6wqx OTHER_TP53RK_HUMAN TP53RK 1.2e-114 387.3 1 224 224 182 183 184 186 188 60 84 88 159 161 160 162 199 205 200 199 198 197 196 195 194 114 EKC/KEOPS complex subunit TP53RK
OTHER WNK3 WNK3_HUMAN 5O26A Q9BYP7 135 414 1800.0 ANP:501 ATPlike Active DFGin 6.954 12.201 BLAminus -125.28, -164.72 58.79, 65.89 -88.2, 18.66 305.61, 176.73 -69.56, -20.03 na-na na 15.898 Saltbr-na 999.0 HRD-in -66.1, -48.87 66.45, 11.22 na-in-in SNCaii in-in ActLoopNT-in 3.021 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.2, 167.0 APE9-dihe-na 127.63, -163.54 APE8-dihe-in -104.53, 119.98 APE8-rot-in 309.3 APE67-dihe-in -64.09, -19.44 -52.49, -34.59 APE12-dist-in 8.873 APE11-dist-in 11.829 APE10-dist-in 6.326 APE9-dist-in 3.706 None SEP304,SEP308 SEP304,SEP308 XRAY 2.379 0.231 0.278 A 284 273 7 0 0 0 [[146, 405]] 1.0 5o26 OTHER_WNK3_HUMAN WNK 2.6e-178 596.6 1 260 260 293 294 295 297 299 176 194 198 272 274 273 275 330 319 314 313 312 311 310 309 308 228 Serine/threonine-protein kinase WNK3
OTHER WNK3 WNK3_HUMAN 5O26B Q9BYP7 136 413 1800.0 ANP:501 ATPlike Active DFGin 7.182 12.078 BLAminus -111.0, -167.63 57.49, 63.76 -86.7, 17.71 307.84, 173.05 -70.2, -27.96 na-na na 15.641 Saltbr-na 999.0 HRD-in -66.99, -53.82 74.22, 8.4 na-in-in SNCaii in-in ActLoopNT-in 3.073 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.41, 145.08 APE9-dihe-na 140.9, -162.45 APE8-dihe-in -99.46, 120.61 APE8-rot-in 305.94 APE67-dihe-in -65.71, -19.72 -54.06, -31.08 APE12-dist-in 8.136 APE11-dist-in 11.827 APE10-dist-in 6.044 APE9-dist-in 3.51 None SEP304,SEP308 SEP304,SEP308 XRAY 2.379 0.231 0.278 B 284 267 11 0 0 0 [[146, 405]] 1.0 5o26 OTHER_WNK3_HUMAN WNK 2.6e-178 596.6 1 260 260 293 294 295 297 299 176 194 198 272 274 273 275 330 319 314 313 312 311 310 309 308 228 Serine/threonine-protein kinase WNK3
STE PAK3 PAK3_HUMAN 6FD3A O75914 261 556 559.0 ADP:60603 ATPlike Active DFGin 5.952 14.149 BLAminus -133.62, -174.01 64.9, 77.07 -96.85, 18.52 289.09, 83.73 -72.71, -11.5 in-in in 8.938 Saltbr-in 2.761 HRD-in -71.32, -50.63 74.19, 1.63 in-in-in SNCiii in-in ActLoopNT-in 2.913 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.75, 147.44 APE9-dihe-na 132.72, -161.48 APE8-dihe-in -114.41, 121.22 APE8-rot-in 305.33 APE67-dihe-in -64.48, -19.99 -44.4, -48.2 APE12-dist-in 8.849 APE11-dist-in 11.358 APE10-dist-in 5.576 APE9-dist-in 3.34 A537D None T8L436 XRAY 1.52 0.176 0.19 A 300 296 0 0 0 0 [[283, 534]] 1.0 6fd3 STE_PAK3_HUMAN STE 1.1e-94 322.5 1 257 257 419 420 421 423 425 312 328 332 399 401 400 402 459 447 442 441 440 439 438 437 436 358 Serine/threonine-protein kinase PAK 3
STE PAK4 PAK4_HUMAN 4FIFA O96013 296 589 591.0 ANP:1000 ATPlike Active DFGin 6.132 13.879 BLAminus -134.27, -172.64 55.78, 65.69 -91.22, 11.11 299.57, 98.92 -61.37, -20.58 in-in in 7.046 Saltbr-in 3.112 HRD-in -73.18, -47.2 74.11, -8.39 in-in-in SNCiii in-in ActLoopNT-in 2.852 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.08, 134.89 APE9-dihe-na 136.18, -173.61 APE8-dihe-in -102.98, 119.55 APE8-rot-in 312.46 APE67-dihe-in -69.75, -26.2 -30.93, -52.34 APE12-dist-in 9.318 APE11-dist-in 11.709 APE10-dist-in 5.875 APE9-dist-in 3.299 None SEP474 SEP474 XRAY 2.6 0.207 0.227 A 346 294 0 0 0 0 [[321, 572]] 1.0 4fif STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 4FIFB O96013 297 589 591.0 ANP:1000 ATPlike Active DFGin 5.899 13.85 BLAminus -129.09, -170.37 52.27, 68.51 -93.51, 10.45 301.97, 96.23 -63.09, -15.01 in-in in 7.007 Saltbr-in 3.167 HRD-in -65.39, -48.9 75.1, -7.5 in-in-in SNCiii in-in ActLoopNT-in 2.801 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.88, 134.77 APE9-dihe-na 136.42, -174.06 APE8-dihe-in -101.96, 121.94 APE8-rot-in 314.36 APE67-dihe-in -72.79, -21.56 -33.03, -50.98 APE12-dist-in 9.238 APE11-dist-in 11.712 APE10-dist-in 5.886 APE9-dist-in 3.335 None SEP474 SEP474 XRAY 2.6 0.207 0.227 B 346 293 0 0 0 0 [[321, 572]] 1.0 4fif STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 4JDIA O96013 300 589 591.0 ANP:1000 ATPlike Active DFGin 6.291 14.47 BLAminus -134.26, 177.87 63.72, 71.58 -94.6, 13.78 289.77, 79.71 -54.15, -28.77 in-in in 6.959 Saltbr-in 2.737 HRD-in -72.82, -49.09 73.48, 2.76 in-in-in SNCiii in-in ActLoopNT-in 2.829 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.62, 145.0 APE9-dihe-na 130.41, -160.49 APE8-dihe-in -120.53, 123.45 APE8-rot-in 305.94 APE67-dihe-in -63.49, -22.51 -36.89, -56.07 APE12-dist-in 8.769 APE11-dist-in 11.535 APE10-dist-in 5.874 APE9-dist-in 3.327 None SEP474 SEP474 XRAY 1.85 0.194 0.233 A 346 290 0 0 0 0 [[321, 572]] 1.0 4jdi STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 5UPKB O96013 300 588 591.0 ANP:60600 ATPlike Active DFGin 6.272 14.139 BLAminus -132.3, -169.35 61.71, 61.5 -87.86, 7.28 293.59, 93.96 -55.36, -28.3 in-in in 7.077 Saltbr-in 3.329 HRD-in -65.35, -49.16 70.36, 11.54 in-in-in SNCiii in-in ActLoopNT-in 2.997 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.55, 149.52 APE9-dihe-na 120.09, -163.11 APE8-dihe-in -119.51, 121.87 APE8-rot-in 313.98 APE67-dihe-in -69.89, -18.98 -32.47, -57.41 APE12-dist-in 8.623 APE11-dist-in 11.267 APE10-dist-in 5.616 APE9-dist-in 3.426 None SEP474 SEP474 XRAY 2.4 0.22 0.264 B 346 289 0 0 0 0 [[321, 572]] 1.0 5upk STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 7S46A O96013 300 589 591.0 ANP:600 ATPlike Active DFGin 9.021 14.349 BLAminus -133.61, -177.07 54.75, 76.68 -92.18, 14.46 286.49, 80.35 -59.04, -19.55 in-in in 7.534 Saltbr-in 2.867 HRD-in -69.43, -50.5 76.76, 2.96 in-in-in SNCiii in-in ActLoopNT-in 2.922 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.73, 132.58 APE9-dihe-na 145.82, -167.86 APE8-dihe-in -110.13, 128.57 APE8-rot-in 305.26 APE67-dihe-in -70.79, -21.11 -38.41, -55.32 APE12-dist-in 9.02 APE11-dist-in 11.537 APE10-dist-in 5.793 APE9-dist-in 3.286 D440N,S474E None None XRAY 2.1 0.182 0.22 A 346 290 0 0 0 0 [[321, 572]] 1.0 7s46 STE_PAK4_HUMAN STE 5.5e-87 297.4 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 7S47A O96013 300 589 591.0 ANP:600 ATPlike Active DFGin 9.217 14.646 BLAminus -126.8, -179.34 54.51, 73.91 -89.97, 15.41 285.81, 78.05 -59.21, -18.99 in-in in 7.79 Saltbr-in 2.931 HRD-in -66.64, -48.47 70.7, 6.89 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.53, 138.41 APE9-dihe-na 140.72, -164.27 APE8-dihe-in -114.61, 124.35 APE8-rot-in 304.9 APE67-dihe-in -66.22, -20.32 -36.39, -56.83 APE12-dist-in 9.039 APE11-dist-in 11.45 APE10-dist-in 5.747 APE9-dist-in 3.401 D440N,S474E None None XRAY 2.0 0.196 0.237 A 383 290 0 0 0 0 [[321, 572]] 1.0 7s47 STE_PAK4_HUMAN STE 7.5e-87 297.0 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE STK24 STK24_HUMAN 3A7JA Q9Y6E0 25 311 443.0 ADP:60500 ATPlike Active DFGin 6.747 14.583 BLAminus -138.67, 168.25 71.5, 79.52 -101.19, 20.06 287.01, 95.64 -64.31, -27.68 in-in in 8.53 Saltbr-in 2.552 HRD-in -69.86, -43.49 67.32, -1.05 in-in-in SNCiii in-in ActLoopNT-in 2.741 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.28, 158.62 APE9-dihe-na 130.53, -164.99 APE8-dihe-in -116.23, 120.86 APE8-rot-in 304.02 APE67-dihe-in -60.63, -23.79 -34.15, -55.13 APE12-dist-in 8.296 APE11-dist-in 11.11 APE10-dist-in 5.251 APE9-dist-in 3.288 None TPO190 TPO190 XRAY 1.5 0.191 0.21 A 303 287 0 0 0 0 [[36, 286]] 1.0 3a7j STE_STK24_HUMAN STE 3.6e-100 340.5 1 257 257 173 174 175 177 179 65 82 86 153 155 154 156 213 201 196 195 194 193 192 191 190 112 Serine/threonine-protein kinase 24
STE STK24 STK24_HUMAN 4QMLA Q9Y6E0 30 310 443.0 ANP:60403 ATPlike Active DFGin 6.598 15.178 BLAminus -130.38, 172.22 70.9, 79.24 -104.53, 20.01 285.96, 83.16 -61.35, -25.21 in-in in 9.065 Saltbr-in 2.927 HRD-in -70.82, -51.82 74.23, -2.97 in-in-in SNCiii in-in ActLoopNT-in 2.848 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.04, 155.96 APE9-dihe-na 125.92, -168.67 APE8-dihe-in -115.63, 119.31 APE8-rot-in 310.36 APE67-dihe-in -60.1, -29.49 -47.33, -42.77 APE12-dist-in 8.276 APE11-dist-in 11.051 APE10-dist-in 5.558 APE9-dist-in 3.386 None TPO190 TPO190 XRAY 1.882 0.19 0.23 A 310 281 0 0 0 0 [[36, 286]] 1.0 4qml STE_STK24_HUMAN STE 3.9e-100 340.4 1 257 257 173 174 175 177 179 65 82 86 153 155 154 156 213 201 196 195 194 193 192 191 190 112 Serine/threonine-protein kinase 24
STE TAOK3 TAOK3_HUMAN 6BDNA Q9H2K8 8 314 898.0 ADP:404 ATPlike Active DFGin 6.771 13.825 BLAminus -136.73, -179.28 62.01, 80.15 -97.31, 23.85 293.38, 102.08 -68.85, -11.35 in-in in 8.485 Saltbr-in 2.682 HRD-in -74.02, -52.69 74.7, -5.2 in-in-in SNCiii in-in ActLoopNT-in 2.797 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.94, 158.28 APE9-dihe-na 130.64, -172.75 APE8-dihe-in -113.55, 120.19 APE8-rot-in 301.22 APE67-dihe-in -62.99, -26.26 -46.03, -46.8 APE12-dist-in 8.28 APE11-dist-in 11.04 APE10-dist-in 5.18 APE9-dist-in 3.383 R2A,K3A None None XRAY 1.5 0.187 0.214 A 320 307 0 0 0 0 [[24, 277]] 1.0 6bdn STE_TAOK3_HUMAN STE 6.3e-90 307.0 4 257 254 164 165 166 168 170 53 72 76 144 146 145 147 203 188 183 182 181 180 179 178 177 102 Serine/threonine-protein kinase TAO3
STE TNIK TNIK_HUMAN 7XZRB Q9UKE5 12 312 1360.0 ANP:1401 ATPlike Active DFGin 6.439 15.163 BLAminus -131.61, 176.54 70.33, 83.31 -101.27, 21.61 286.01, 77.74 -67.8, -30.96 in-in in 9.126 Saltbr-in 2.582 HRD-in -64.36, -58.64 76.74, 3.35 in-in-in SNCiii in-in ActLoopNT-in 2.931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.27, 150.43 APE9-dihe-na 126.35, -168.16 APE8-dihe-in -105.07, 123.33 APE8-rot-in 308.43 APE67-dihe-in -61.4, -25.19 -44.62, -54.45 APE12-dist-in 8.7 APE11-dist-in 11.705 APE10-dist-in 6.078 APE9-dist-in 3.705 None TPO181,TPO187 TPO181,TPO187 XRAY 2.26 0.184 0.226 B 306 301 0 0 0 0 [[25, 289]] 1.0 7xzr STE_TNIK_HUMAN STE 3e-105 357.1 1 257 257 170 171 172 174 176 54 69 73 150 152 151 153 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
TKL BMPR2 BMPR2_HUMAN 3G2FA Q13873 197 510 1038.0 ADP:900 ATPlike Active DFGin 6.957 13.944 BLAminus -131.62, -179.2 66.08, 79.87 -102.79, 27.43 304.26, 96.52 -59.99, -25.3 in-in in 8.107 Saltbr-in 2.757 HRD-in -69.81, -50.66 82.19, -10.63 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.1, -22.11 APE9-dihe-na -73.96, -168.61 APE8-dihe-in -80.16, 127.03 APE8-rot-in 308.56 APE67-dihe-in -65.91, -22.58 -59.75, -41.5 APE12-dist-in 11.403 APE11-dist-in 12.63 APE10-dist-in 7.026 APE9-dist-in 4.033 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 A 336 305 9 0 0 9 [[202, 503]] 1.0 3g2f TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2 266 265 350 351 352 354 356 230 243 247 330 332 331 333 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
TKL BMPR2 BMPR2_HUMAN 3G2FB Q13873 198 513 1038.0 ADP:900 ATPlike Active DFGin 6.968 14.008 BLAminus -149.7, 179.95 61.07, 87.18 -102.54, 11.93 293.8, 112.47 -56.7, -17.91 in-in in 8.065 Saltbr-in 2.732 HRD-in -73.22, -52.25 87.7, -10.0 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.94, -26.41 APE9-dihe-na -71.73, -175.39 APE8-dihe-in -71.07, 133.08 APE8-rot-in 315.55 APE67-dihe-in -68.07, -13.93 -56.75, -42.89 APE12-dist-in 11.194 APE11-dist-in 12.108 APE10-dist-in 6.494 APE9-dist-in 3.722 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 B 336 303 13 0 0 13 [[202, 503]] 1.0 3g2f TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2 266 265 350 351 352 354 356 230 243 247 330 332 331 333 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
TKL BMPR2 BMPR2_HUMAN 6UNPB Q13873 197 509 1038.0 ADP:601 ATPlike Active DFGin 6.917 14.051 BLAminus -140.56, 176.5 63.35, 76.41 -96.26, 25.8 302.12, 104.12 -61.08, -20.73 in-in in 7.904 Saltbr-in 2.865 HRD-in -75.95, -48.17 78.17, -6.91 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.29, -9.38 APE9-dihe-na -69.43, -161.26 APE8-dihe-in -89.59, 127.34 APE8-rot-in 301.19 APE67-dihe-in -48.39, -33.11 -62.11, -43.63 APE12-dist-in 12.009 APE11-dist-in 12.508 APE10-dist-in 7.099 APE9-dist-in 4.016 D485G None CAS288,CAS397,CAS496 XRAY 2.3 0.19 0.211 B 363 303 10 0 0 8 [[202, 503]] 1.0 6unp TKL_BMPR2_HUMAN TKL 1.1e-74 257.3 2 266 265 350 351 352 354 356 230 243 247 330 332 331 333 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
TKL IRAK4 IRAK4_HUMAN 2OIDD Q9NWZ3 164 459 460.0 ANP:4 ATPlike Active DFGin 6.56 13.972 BLAminus -129.12, -177.03 59.13, 109.88 -131.38, 17.54 304.54, 87.5 -68.37, -4.63 in-in in 8.15 Saltbr-in 3.52 HRD-in -75.54, -51.34 70.58, 2.03 in-in-in SNCiii in-in ActLoopNT-in 2.765 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.72, 147.52 APE9-dihe-na 139.0, -173.6 APE8-dihe-in -107.1, 118.58 APE8-rot-in 309.04 APE67-dihe-in -62.68, -15.82 -47.4, -49.91 APE12-dist-in 9.75 APE11-dist-in 11.44 APE10-dist-in 5.928 APE9-dist-in 3.97 None TPO342,TPO345,SEP346 TPO342,TPO345,SEP346 XRAY 2.3 0.244 0.295 D 301 277 19 0 0 3 [[183, 456]] 1.0 2oid TKL_IRAK4_HUMAN TKL 4.1e-84 288.2 5 266 262 328 329 330 332 334 213 233 237 308 310 309 311 369 358 353 352 351 350 349 348 347 263 Interleukin-1 receptor-associated kinase 4
TKL LIMK1 LIMK1_HUMAN 5L6WL P53667 330 633 647.0 AGS:60701 ATPlike Active DFGin 6.235 14.337 BLAminus -131.64, -166.52 46.75, 81.93 -92.83, 15.71 304.28, 98.92 -42.69, -49.84 in-in in 7.664 Saltbr-in 2.67 HRD-in -78.67, -47.86 69.62, -13.12 in-in-in SNCiii in-in ActLoopNT-in 3.066 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -134.6, 165.2 APE9-dihe-na 100.19, 162.86 APE8-dihe-in -63.5, 131.5 APE8-rot-na 185.1 APE67-dihe-in -61.44, -31.47 -69.46, -29.71 APE12-dist-in 9.116 APE11-dist-in 11.134 APE10-dist-in 5.438 APE9-dist-in 3.762 None None None XRAY 2.53 0.229 0.284 L 310 288 16 0 0 16 [[339, 606]] 1.0 5l6w TKL_LIMK1_HUMAN TKL 4.5e-77 265.1 3 266 264 477 478 479 481 483 368 384 388 457 459 458 460 531 519 514 513 512 511 510 509 508 414 LIM domain kinase 1
TKL LIMK1 LIMK1_HUMAN 5HVKA P53667 329 634 647.0 ANP:61001 ATPlike Active DFGin 6.405 13.646 BLAminus -145.46, 176.84 65.07, 82.49 -109.26, 24.73 304.62, 92.73 -71.79, -22.73 in-in in 7.795 Saltbr-in 3.159 HRD-in -70.8, -44.42 59.42, 18.52 in-in-in SNCiii in-in ActLoopNT-in 3.324 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -139.63, 151.17 APE9-dihe-na 143.88, 171.7 APE8-dihe-in -71.51, 120.27 APE8-rot-na 199.31 APE67-dihe-in -66.59, -36.22 -54.03, -34.34 APE12-dist-in 9.301 APE11-dist-in 11.081 APE10-dist-in 5.636 APE9-dist-in 3.574 D460N TPO508 TPO508 XRAY 3.5 0.275 0.31 A 315 293 13 0 0 13 [[339, 606]] 1.0 5hvk TKL_LIMK1_HUMAN TKL 3e-76 262.4 3 266 264 477 478 479 481 483 368 384 388 457 459 458 460 531 519 514 513 512 511 510 509 508 414 LIM domain kinase 1
TKL LRRK2 LRRK2_HUMAN 8FO9A Q5S007 1329 2527 2527.0 ATP:2602 ATPlike Active DFGin 6.273 13.41 BLAminus -138.23, -175.7 59.6, 64.71 -84.85, 53.99 305.84, 101.34 -78.49, -28.55 in-in in 7.88 Saltbr-in 2.735 HRD-in -107.83, -47.31 66.25, 1.81 in-in-in SNCiii in-in ActLoopNT-in 3.031 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.21, 156.34 APE9-dihe-na 139.24, 152.96 APE8-dihe-in -67.96, 127.7 APE8-rot-in 305.42 APE67-dihe-inflip 98.56, -16.69 -58.5, 136.92 APE12-dist-in 9.183 APE11-dist-in 11.487 APE10-dist-in 6.004 APE9-dist-in 3.816 None None None EM 3.48 999.0 999.0 A 2527 1173 0 0 0 0 [[1875, 2134]] 1.0 8fo9 TKL_LRRK2_HUMAN TKL 3.8e-57 200.3 5 266 262 2016 2017 2018 2020 2022 1906 1920 1924 1991 1993 1992 1994 2055 2042 2037 2036 2035 2034 2033 2032 2031 1948 Leucine-rich repeat serine/threonine-protein kinase 2
TKL LRRK2 LRRK2_HUMAN 8FO9C Q5S007 1329 2527 2527.0 ATP:2602 ATPlike Active DFGin 6.275 13.405 BLAminus -138.14, -175.77 59.5, 64.85 -84.95, 53.97 305.9, 101.31 -78.52, -28.52 in-in in 7.883 Saltbr-in 2.729 HRD-in -108.59, -47.2 66.33, 1.76 in-in-in SNCiii in-in ActLoopNT-in 3.008 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.94, 156.21 APE9-dihe-na 139.37, 152.96 APE8-dihe-in -67.92, 127.71 APE8-rot-in 305.58 APE67-dihe-inflip 98.46, -16.81 -58.61, 136.94 APE12-dist-in 9.177 APE11-dist-in 11.503 APE10-dist-in 6.012 APE9-dist-in 3.804 None None None EM 3.48 999.0 999.0 C 2527 1173 0 0 0 0 [[1875, 2134]] 1.0 8fo9 TKL_LRRK2_HUMAN TKL 3.8e-57 200.3 5 266 262 2016 2017 2018 2020 2022 1906 1920 1924 1991 1993 1992 1994 2055 2042 2037 2036 2035 2034 2033 2032 2031 1948 Leucine-rich repeat serine/threonine-protein kinase 2
TKL TGFBR2 TGFR2_HUMAN 5E92A P37173 240 543 567.0 ANP:601 ATPlike Active DFGin 7.396 13.303 BLAminus -134.93, 178.1 63.07, 87.04 -105.26, 16.76 300.78, 96.96 -60.58, -26.14 in-in in 7.67 Saltbr-in 2.752 HRD-in -64.87, -46.8 71.14, -4.53 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.21, 144.17 APE9-dihe-na 126.96, -149.92 APE8-dihe-in -116.55, 119.38 APE8-rot-in 300.41 APE67-dihe-in -54.91, -33.03 -42.96, -45.47 APE12-dist-in 11.788 APE11-dist-in 12.049 APE10-dist-in 6.089 APE9-dist-in 3.401 E431A,R433A,E485A,K488A,R493A,R495A None None XRAY 2.08 0.204 0.231 A 316 298 6 0 0 0 [[244, 540]] 1.0 5e92 TKL_TGFBR2_HUMAN TKL 1.9e-77 266.3 2 266 265 396 397 398 400 402 277 290 294 376 378 377 379 446 428 423 422 421 420 419 418 417 326 TGF-beta receptor type-2
TYR EGFR EGFR_HUMAN 2ITXA P00533 697 1019 1210.0 ANP:2020 ATPlike Active DFGin 5.874 15.737 BLAminus -136.31, -171.94 65.34, 93.22 -111.54, 18.75 298.27, 92.75 -59.44, 2.06 in-in in 9.241 Saltbr-in 3.583 HRD-in -62.41, -44.72 61.37, 7.79 in-in-in SNCiii in-in ActLoopNT-in 2.642 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -78.73, 124.39 APE9-dihe-in -125.4, 144.12 APE8-dihe-in -79.64, 94.32 APE8-rot-na 30.37 APE67-dihe-in -65.37, -0.17 -61.69, -47.61 APE12-dist-na 11.888 APE11-dist-na 10.151 APE10-dist-na 11.134 APE9-dist-in 7.058 None None None XRAY 2.98 0.191 0.261 A 327 307 4 0 0 4 [[712, 970]] 1.0 2itx TYR_EGFR_HUMAN TYR 1e-87 299.8 3 259 257 854 855 856 858 860 745 762 766 834 836 835 837 896 884 879 878 877 876 875 874 873 791 Epidermal growth factor receptor
TYR FGFR1 FGFR1_HUMAN 3GQIA P11362 464 770 822.0 ACP:775 ATPlike Active DFGin 6.466 13.946 BLAminus -126.61, -175.83 60.19, 72.36 -91.08, 18.42 288.73, 91.63 -64.67, -15.4 in-in in 7.751 Saltbr-in 2.69 HRD-in -77.5, -49.87 72.48, -2.68 in-in-in SNCiii in-in ActLoopNT-in 2.961 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -58.96, 135.34 APE9-dihe-in -149.19, 136.62 APE8-dihe-in -75.51, 66.48 APE8-rot-na 33.4 APE67-dihe-in -65.08, -11.82 -44.91, -41.18 APE12-dist-na 14.083 APE11-dist-na 11.258 APE10-dist-na 10.128 APE9-dist-in 7.137 C488A,Y583F,C584S,Y585F PTR653,PTR654,PTR766 PTR653,PTR654,PTR766 XRAY 2.5 0.249 0.289 A 326 307 0 0 0 0 [[478, 756]] 1.0 3gqi TYR_FGFR1_HUMAN TYR 1.7e-104 354.6 1 260 260 640 641 642 644 646 514 531 535 620 622 621 623 682 670 665 664 663 662 661 660 659 562 Fibroblast growth factor receptor 1
TYR FGFR2 FGFR2_HUMAN 2PVFA P21802 467 765 821.0 ACP:60300 ATPlike Active DFGin 6.048 13.821 BLAminus -138.88, -175.17 54.67, 80.46 -90.11, 24.33 291.08, 76.38 -54.38, -36.38 in-in in 7.913 Saltbr-in 2.769 HRD-in -85.37, -48.4 70.03, 0.26 in-in-in SNCiii in-in ActLoopNT-in 2.879 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -86.94, 115.27 APE9-dihe-in -125.87, 160.91 APE8-dihe-in -74.41, 68.1 APE8-rot-na 35.92 APE67-dihe-in -70.82, -9.54 -47.44, -41.99 APE12-dist-na 15.14 APE11-dist-na 11.649 APE10-dist-na 11.604 APE9-dist-in 7.168 C491A PTR586,PTR656,PTR657 PTR586,PTR656,PTR657 XRAY 1.8 0.251 0.265 A 334 288 11 0 0 0 [[481, 759]] 1.0 2pvf TYR_FGFR2_HUMAN TYR 2.2e-104 354.3 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 3CLYA P21802 468 772 821.0 ACP:61803 ATPlike Active DFGin 6.229 14.183 BLAminus -138.78, -172.76 51.4, 79.79 -91.29, 32.46 290.47, 75.81 -61.86, -29.26 in-in in 7.661 Saltbr-in 2.621 HRD-in -89.86, -45.92 68.93, -0.84 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -72.79, 139.96 APE9-dihe-in -131.36, 152.18 APE8-dihe-in -76.17, 66.16 APE8-rot-na 37.1 APE67-dihe-in -66.78, -6.73 -47.95, -40.48 APE12-dist-na 13.253 APE11-dist-na 10.402 APE10-dist-na 11.097 APE9-dist-in 6.913 C491A PTR656,PTR657 PTR656,PTR657 XRAY 2.0 0.216 0.247 A 334 291 14 0 0 0 [[481, 759]] 1.0 3cly TYR_FGFR2_HUMAN TYR 2.2e-104 354.3 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 5EG3A P21802 466 774 821.0 ACP:60801 ATPlike Active DFGin 6.034 13.825 BLAminus -138.71, -166.61 47.53, 87.44 -100.17, 28.73 285.85, 82.29 -77.8, -14.99 in-in in 8.045 Saltbr-in 2.941 HRD-in -83.82, -45.21 62.18, 9.75 in-in-in SNCiii in-in ActLoopNT-in 2.991 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -66.56, 121.06 APE9-dihe-in -128.9, 119.34 APE8-dihe-in -79.6, 67.11 APE8-rot-na 30.51 APE67-dihe-in -77.81, 0.08 -48.0, -39.27 APE12-dist-na 13.558 APE11-dist-na 10.078 APE10-dist-na 8.259 APE9-dist-in 7.021 Y466F,C491A,E565A,Y586L,Y588P,Y656F,Y657F,K659E PTR769 PTR769 XRAY 2.606 0.191 0.237 A 334 302 7 0 0 0 [[481, 759]] 1.0 5eg3 TYR_FGFR2_HUMAN TYR 2.3e-101 344.4 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR3 FGFR3_HUMAN 4K33A P22607 459 755 806.0 ACP:801 ATPlike Active DFGin 6.252 13.787 BLAminus -133.88, -173.58 58.49, 82.81 -96.43, 27.55 291.81, 80.95 -59.32, -31.32 in-in in 8.211 Saltbr-in 2.895 HRD-in -87.09, -47.34 67.06, 1.63 in-in-in SNCiii in-in ActLoopNT-in 2.99 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -55.89, 133.11 APE9-dihe-in -125.43, 130.21 APE8-dihe-in -78.76, 72.58 APE8-rot-na 29.71 APE67-dihe-in -71.45, -4.47 -50.14, -48.75 APE12-dist-na 13.31 APE11-dist-na 9.602 APE10-dist-na 8.305 APE9-dist-in 6.873 C482A,C582S,K650E None None XRAY 2.341 0.181 0.228 A 325 293 4 0 0 0 [[472, 750]] 1.0 4k33 TYR_FGFR3_HUMAN TYR 2.3e-104 354.2 1 260 260 634 635 636 638 640 508 525 529 614 616 615 617 676 664 659 658 657 656 655 654 653 556 Fibroblast growth factor receptor 3
TYR INSR INSR_HUMAN 3BU5A P06213 1014 1310 1382.0 ATP:60300 ATPlike Active DFGin 6.659 13.934 BLAminus -128.64, -166.6 44.54, 89.54 -102.81, 23.91 295.82, 99.34 -57.5, -34.18 in-in in 8.261 Saltbr-in 3.13 HRD-in -68.86, -51.91 77.02, -10.33 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -82.0, 102.51 APE9-dihe-in -127.85, 151.44 APE8-dihe-in -79.76, 69.1 APE8-rot-na 32.47 APE67-dihe-in -66.77, -8.03 -57.27, -41.89 APE12-dist-na 15.937 APE11-dist-na 11.724 APE10-dist-na 11.3 APE9-dist-in 7.401 C1008S PTR1185,PTR1189,PTR1190 PTR1185,PTR1189,PTR1190 XRAY 2.1 0.196 0.239 A 306 294 3 0 0 0 [[1023, 1292]] 1.0 3bu5 TYR_INSR_HUMAN TYR 1.3e-96 328.8 1 260 260 1176 1177 1178 1180 1182 1057 1074 1078 1156 1158 1157 1159 1218 1206 1201 1200 1199 1198 1197 1196 1195 1104 Insulin receptor
TYR INSR INSR_HUMAN 4XLVA P06213 1001 1310 1382.0 ACP:61301 ATPlike Active DFGin 6.357 13.404 BLAminus -129.47, -169.61 59.33, 81.3 -99.86, 10.75 301.2, 100.62 -50.37, -35.15 in-in in 8.175 Saltbr-in 2.441 HRD-in -74.09, -41.95 72.32, -7.69 in-in-in SNCiii in-in ActLoopNT-in 3.029 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -31.8, 98.01 APE9-dihe-in -128.43, 131.43 APE8-dihe-in -62.62, 111.75 APE8-rot-na 18.22 APE67-dihe-in -71.49, -19.39 -64.21, -23.54 APE12-dist-na 14.741 APE11-dist-na 10.551 APE10-dist-na 11.027 APE9-dist-in 6.615 Y992F,C1008S PTR999,PTR1185,PTR1189,PTR1190 PTR999,PTR1185,PTR1189,PTR1190 XRAY 2.3 0.207 0.266 A 328 310 0 0 0 0 [[1023, 1292]] 1.0 4xlv TYR_INSR_HUMAN TYR 1.7e-96 328.5 1 260 260 1176 1177 1178 1180 1182 1057 1074 1078 1156 1158 1157 1159 1218 1206 1201 1200 1199 1198 1197 1196 1195 1104 Insulin receptor
TYR JAK1-2 JAK1_HUMAN 6C7YA P23458 869 1153 1154.0 ADP:61201 ATPlike Active DFGin 6.032 13.967 BLAminus -134.15, -164.18 58.49, 84.96 -109.28, 28.04 298.78, 97.45 -66.39, -27.05 in-in in 8.311 Saltbr-in 2.732 HRD-in -67.59, -46.53 68.25, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -72.91, 151.36 APE9-dihe-in -137.76, 143.32 APE8-dihe-in -74.71, 81.76 APE8-rot-na 30.49 APE67-dihe-in -79.4, -2.38 -65.2, -24.66 APE12-dist-na 12.972 APE11-dist-na 8.02 APE10-dist-na 10.344 APE9-dist-in 6.316 None PTR1035 PTR1035 XRAY 2.499 0.21 0.241 A 286 273 12 0 0 0 [[583, 847], [875, 1151]] 2.0 6c7y TYR_JAK1-2_HUMAN TYR 1.8e-87 298.9 2 259 258 1020 1021 1022 1024 1026 908 925 929 1000 1002 1001 1003 1063 1051 1046 1045 1044 1043 1042 1041 1040 957 Tyrosine-protein kinase JAK1
TYR LCK LCK_HUMAN 1QPCA P06239 231 502 509.0 ANP:904 ATPlike Active DFGin 6.61 14.416 BLAminus -133.73, 179.02 58.4, 83.48 -97.79, 21.23 295.19, 99.8 -60.65, -35.99 in-in in 8.702 Saltbr-in 3.096 HRD-in -103.01, -49.32 74.3, -4.36 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -120.97, 142.08 APE9-dihe-in -126.79, 156.19 APE8-dihe-in -63.13, 117.89 APE8-rot-na 333.56 APE67-dihe-in -65.85, -20.96 -57.94, -43.39 APE12-dist-na 14.856 APE11-dist-na 10.005 APE10-dist-na 12.788 APE9-dist-in 6.784 None PTR394 PTR394 XRAY 1.6 0.2 0.23 A 279 272 0 0 0 0 [[245, 496]] 1.0 1qpc TYR_LCK_HUMAN TYR 1.4e-94 322.2 1 260 260 381 382 383 385 387 273 288 292 361 363 362 364 422 410 405 404 403 402 401 400 399 317 Tyrosine-protein kinase Lck
TYR SYK KSYK_HUMAN 4FL1A P43405 363 635 635.0 ANP:701 ATPlike Active DFGin 6.669 15.063 BLAminus -122.6, -175.53 56.16, 78.38 -92.62, 24.67 287.04, 93.75 -57.67, -38.36 in-in in 8.059 Saltbr-in 2.683 HRD-in -76.27, -50.57 71.77, 3.28 in-in-in SNCiii in-in ActLoopNT-in 2.976 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -89.55, 85.11 APE9-dihe-in -99.28, 138.37 APE8-dihe-in -79.64, 69.72 APE8-rot-na 29.68 APE67-dihe-in -60.65, -16.95 -44.16, -41.68 APE12-dist-na 13.816 APE11-dist-na 10.806 APE10-dist-na 10.412 APE9-dist-in 7.132 None None None XRAY 1.79 0.197 0.225 A 291 268 5 0 0 0 [[370, 628]] 1.0 4fl1 TYR_SYK_HUMAN TYR 5.5e-90 307.1 5 260 256 511 512 513 515 517 402 420 424 491 493 492 494 554 542 537 536 535 534 533 532 531 449 Tyrosine-protein kinase SYK
TYR TNK2 ACK1_HUMAN 1U54B Q07912 117 388 1038.0 ACP:400 ATPlike Active DFGin 6.615 13.378 BLAminus -120.4, -155.16 27.84, 85.75 -104.36, 38.7 310.01, 93.15 -67.71, -28.73 in-in in 7.966 Saltbr-in 3.021 HRD-in -109.84, -42.56 64.6, 13.11 in-in-in SNCiii in-in ActLoopNT-in 3.014 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -150.8, 133.1 APE9-dihe-in -126.86, 129.0 APE8-dihe-in -43.1, 130.27 APE8-rot-na 329.12 APE67-dihe-in -70.13, -6.6 -62.78, -39.45 APE12-dist-na 12.662 APE11-dist-na 7.646 APE10-dist-na 11.0 APE9-dist-in 5.878 None None None XRAY 2.8 0.226 0.322 B 291 261 11 0 0 0 [[126, 387]] 1.0 1u54 TYR_TNK2_HUMAN TYR 9e-86 293.3 1 259 259 269 270 271 273 275 158 177 181 249 251 250 252 312 300 295 294 293 292 291 290 289 206 Activated CDC42 kinase 1

All / Activity_Active / ATPlike

Total number of chains: 310
Active chains: 310
Total number of genes: 79
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 310 100.0% 8QCGB

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC CKA1 CSK21_ARATH 6XX7A Q08467 77 406 409.0 ANP:60401 ATPlike Active DFGin 7.522 16.054 BLAminus -117.69, -174.69 54.04, 89.21 -108.75, 22.96 298.46, 82.8 -72.45, -17.87 in-in in 9.197 Saltbr-in 3.111 HRD-in -78.14, -48.74 65.41, 21.05 in-in-in SNCiii in-in ActLoopNT-in 2.834 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.12, 170.49 APE9-dihe-na 62.76, -171.63 APE8-dihe-in -114.91, 151.01 APE8-rot-in 304.83 APE67-dihe-in -66.49, -17.41 -50.66, -50.22 APE12-dist-in 12.585 APE11-dist-in 10.283 APE10-dist-in 6.188 APE9-dist-in 3.134 None None None XRAY 2.4 0.198 0.246 A 342 330 0 0 0 0 [[110, 395]] 1.0 6xx7 Arabidopsis thaliana CMGC_CKA1_ARATH CMGC 2.6e-65 226.5 1 301 301 245 246 247 249 251 139 152 156 224 226 225 227 285 272 267 266 265 264 263 262 261 185 Casein kinase II subunit alpha-1
TKL BRI1 BRI1_ARATH 5LPBA O22476 867 1160 1196.0 ADP:1201 ATPlike Active DFGin 5.075 15.058 BLAminus -134.68, 179.03 63.17, 81.59 -99.15, 20.06 285.86, 73.26 -60.78, -23.17 in-in in 8.649 Saltbr-in 3.148 HRD-in -69.16, -46.8 71.42, -2.74 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -107.78, 147.47 APE9-dihe-na 145.38, -170.04 APE8-dihe-in -133.78, 133.64 APE8-rot-in 306.07 APE67-dihe-inflip 102.35, -15.45 -46.22, 126.04 APE12-dist-in 9.248 APE11-dist-in 11.275 APE10-dist-in 5.497 APE9-dist-in 3.743 T872A TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 1.98 0.184 0.203 A 296 284 10 0 0 0 [[882, 1157]] 1.0 5lpb Arabidopsis thaliana TKL_BRI1_ARATH TKL 2e-63 220.4 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 5LPVA O22476 867 1160 1196.0 ANP:1200 ATPlike Active DFGin 5.144 14.999 BLAminus -125.7, -177.27 57.44, 79.7 -100.2, 28.83 289.11, 69.34 -64.8, -27.23 in-in in 8.616 Saltbr-in 2.692 HRD-in -72.39, -48.96 69.78, 4.25 in-in-in SNCiii in-in ActLoopNT-in 2.973 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.4, 152.93 APE9-dihe-na 138.14, -175.87 APE8-dihe-in -122.84, 131.25 APE8-rot-in 310.37 APE67-dihe-inflip 103.25, -12.92 -53.02, 126.73 APE12-dist-in 9.499 APE11-dist-in 11.435 APE10-dist-in 5.667 APE9-dist-in 3.671 T872A TPO1039,SEP1042,SEP1044 TPO1039,SEP1042,SEP1044 XRAY 2.7 0.193 0.233 A 296 285 9 0 0 0 [[882, 1157]] 1.0 5lpv Arabidopsis thaliana TKL_BRI1_ARATH TKL 2e-63 220.4 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 5LPYA O22476 867 1160 1196.0 ATP:1200 ATPlike Active DFGin 5.175 15.203 BLAminus -134.16, 179.9 60.37, 82.56 -100.0, 17.51 285.92, 71.71 -57.07, -20.27 in-in in 8.892 Saltbr-in 3.152 HRD-in -70.7, -49.88 77.86, -1.82 in-in-in SNCiii in-in ActLoopNT-in 2.908 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.47, 151.76 APE9-dihe-na 140.48, 176.99 APE8-dihe-in -121.99, 138.13 APE8-rot-in 307.91 APE67-dihe-inflip 92.03, -10.16 -52.79, 133.04 APE12-dist-in 9.609 APE11-dist-in 11.524 APE10-dist-in 5.721 APE9-dist-in 3.885 T872A TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 2.3 0.203 0.248 A 296 286 8 0 0 0 [[882, 1157]] 1.0 5lpy Arabidopsis thaliana TKL_BRI1_ARATH TKL 2e-63 220.4 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 5LPZA O22476 866 1160 1196.0 ADP:1200 ATPlike Active DFGin 5.281 15.229 BLAminus -133.61, -178.19 59.45, 71.09 -88.15, 19.11 288.53, 76.38 -60.79, -23.86 in-in in 8.633 Saltbr-in 2.829 HRD-in -68.17, -37.55 64.9, -2.92 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -69.74, 170.98 APE9-dihe-na 106.33, 162.6 APE8-dihe-in -102.72, 137.46 APE8-rot-in 305.68 APE67-dihe-inflip 102.78, -18.56 -57.05, 134.59 APE12-dist-in 9.342 APE11-dist-in 11.755 APE10-dist-in 5.72 APE9-dist-in 3.579 T872A TPO1039,SEP1042,SEP1044 TPO1039,SEP1042,SEP1044 XRAY 2.48 0.226 0.253 A 332 286 9 0 0 0 [[882, 1157]] 1.0 5lpz Arabidopsis thaliana TKL_BRI1_ARATH TKL 3e-63 219.9 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4OH4A O22476 863 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.109 14.621 BLAminus -140.27, -170.9 60.42, 81.58 -96.75, 17.94 285.65, 72.49 -62.14, -24.45 in-in in 8.43 Saltbr-in 2.981 HRD-in -67.48, -45.07 71.79, 0.23 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.28, 137.25 APE9-dihe-na 143.97, 175.71 APE8-dihe-in -113.05, 131.41 APE8-rot-in 300.18 APE67-dihe-inflip 103.6, -22.59 -52.56, 134.8 APE12-dist-in 10.688 APE11-dist-in 12.06 APE10-dist-in 6.328 APE9-dist-in 4.124 None TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 2.25 0.203 0.236 A 333 292 6 0 0 0 [[882, 1157]] 1.0 4oh4 Arabidopsis thaliana TKL_BRI1_ARATH TKL 3e-63 219.8 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4OH4B O22476 867 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.028 14.866 BLAminus -128.92, -179.57 66.05, 81.1 -97.08, 13.19 285.07, 69.22 -52.61, -27.46 in-in in 8.604 Saltbr-in 2.585 HRD-in -68.96, -46.37 73.67, -10.15 in-in-in SNCiii in-in ActLoopNT-in 2.87 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.43, 142.85 APE9-dihe-na 162.33, 170.81 APE8-dihe-in -132.62, 128.73 APE8-rot-in 297.7 APE67-dihe-inflip 104.71, -30.59 -48.41, 132.44 APE12-dist-in 9.471 APE11-dist-in 10.311 APE10-dist-in 5.146 APE9-dist-in 4.053 None TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 2.25 0.203 0.236 B 333 283 11 0 0 0 [[882, 1157]] 1.0 4oh4 Arabidopsis thaliana TKL_BRI1_ARATH TKL 3e-63 219.8 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4Q5JA O22476 863 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.066 14.74 BLAminus -137.9, 174.67 63.19, 85.3 -100.14, 20.42 284.87, 74.71 -62.5, -33.31 in-in in 8.354 Saltbr-in 3.257 HRD-in -68.22, -43.45 65.77, 3.93 in-in-in SNCiii in-in ActLoopNT-in 2.662 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -108.48, 139.01 APE9-dihe-na 175.24, 173.84 APE8-dihe-in -115.42, 129.74 APE8-rot-in 289.59 APE67-dihe-inflip 96.87, -1.52 -53.59, 124.31 APE12-dist-in 10.51 APE11-dist-in 12.065 APE10-dist-in 6.236 APE9-dist-in 4.467 None TPO1039,SEP1042,SEP1044,SEP1060 MSE925,MSE928,MSE959,MSE1010,MSE1030,MSE1034,MSE1037,TPO1039,SEP1042,SEP1044,SEP1060,MSE1117,MSE1148,MSE1152,MSE1154 XRAY 2.772 0.203 0.259 A 341 287 11 0 0 0 [[882, 1157]] 1.0 4q5j Arabidopsis thaliana TKL_BRI1_ARATH TKL 3.2e-63 219.7 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4Q5JB O22476 867 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.259 14.8 BLAminus -126.47, -178.56 58.45, 93.89 -112.89, 22.9 283.23, 71.66 -57.4, -19.56 in-in in 8.732 Saltbr-in 3.184 HRD-in -81.55, -35.96 67.72, -5.15 in-in-in SNCiii in-in ActLoopNT-in 2.775 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.14, 134.16 APE9-dihe-na 157.62, 164.27 APE8-dihe-in -126.08, 123.8 APE8-rot-in 304.99 APE67-dihe-inflip 120.44, -28.11 -46.98, 122.06 APE12-dist-in 9.403 APE11-dist-in 10.636 APE10-dist-in 5.512 APE9-dist-in 4.081 None TPO1039,SEP1042,SEP1044,SEP1060 MSE925,MSE928,MSE959,MSE1010,MSE1030,MSE1034,MSE1037,TPO1039,SEP1042,SEP1044,SEP1060,MSE1117,MSE1148,MSE1152,MSE1154 XRAY 2.772 0.203 0.259 B 341 283 11 0 0 0 [[882, 1157]] 1.0 4q5j Arabidopsis thaliana TKL_BRI1_ARATH TKL 3.2e-63 219.7 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
AGC GRK1 GRK1_BOVIN 3T8OA P28327 30 532 561.0 ATP:562 ATPlike Active DFGin 6.784 13.652 BLAminus -147.61, 176.5 66.51, 86.5 -106.39, 20.07 278.45, 121.96 -78.51, -8.51 in-in in 9.131 Saltbr-in 2.946 HRD-in -72.08, -59.57 74.93, 15.13 in-in-in SNCiii in-in ActLoopNT-in 3.034 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.6, 145.4 APE9-dihe-na 140.82, -165.62 APE8-dihe-in -114.33, 123.31 APE8-rot-in 302.45 APE67-dihe-inflip 90.49, -9.25 -48.36, 136.06 APE12-dist-in 10.419 APE11-dist-in 11.645 APE10-dist-in 5.795 APE9-dist-in 4.276 L166K None None XRAY 2.5 0.209 0.245 A 543 493 0 0 0 0 [[187, 452]] 1.0 3t8o Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4WA P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 6.587 13.314 BLAminus -157.51, 175.0 67.79, 80.23 -106.97, 21.1 277.77, 138.55 -72.95, -18.52 in-in in 8.671 Saltbr-in 2.659 HRD-in -67.86, -51.97 60.46, 12.85 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.73, 153.77 APE9-dihe-na 125.45, -175.95 APE8-dihe-in -101.44, 127.92 APE8-rot-in 301.93 APE67-dihe-inflip 97.46, -21.92 -46.81, 133.28 APE12-dist-in 10.007 APE11-dist-in 11.248 APE10-dist-in 5.534 APE9-dist-in 3.508 None TPO8 TPO8 XRAY 2.7 0.192 999.0 A 543 494 0 0 0 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4WB P28327 5 533 561.0 ATP:562 ATPlike Active DFGin 5.963 13.111 BLAminus -155.04, 178.49 64.64, 79.84 -103.28, 19.03 277.57, 109.21 -72.3, -19.68 in-in in 8.548 Saltbr-in 2.84 HRD-in -67.79, -54.67 64.69, 11.83 in-in-in SNCiii in-in ActLoopNT-in 2.958 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.45, 154.48 APE9-dihe-na 126.08, -175.35 APE8-dihe-in -101.18, 126.91 APE8-rot-in 300.91 APE67-dihe-inflip 94.23, -17.08 -47.18, 130.86 APE12-dist-in 10.103 APE11-dist-in 11.254 APE10-dist-in 5.545 APE9-dist-in 3.534 None TPO8 TPO8 XRAY 2.7 0.192 999.0 B 543 519 0 0 0 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4XA P28327 30 533 561.0 ATP:562 ATPlike Active DFGin 6.392 13.294 BLAminus -153.36, -178.73 56.38, 83.66 -101.23, 19.01 282.86, 141.85 -58.01, -33.04 in-in in 8.623 Saltbr-in 2.825 HRD-in -65.41, -52.58 62.44, 13.36 in-in-in SNCiii in-in ActLoopNT-in 2.96 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.48, 144.22 APE9-dihe-na 128.55, -174.69 APE8-dihe-in -103.7, 129.98 APE8-rot-in 314.1 APE67-dihe-inflip 101.04, -22.84 -50.28, 132.61 APE12-dist-in 10.283 APE11-dist-in 11.237 APE10-dist-in 5.726 APE9-dist-in 3.827 None None None XRAY 2.9 0.193 999.0 A 543 496 0 0 0 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4XB P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 5.903 13.063 BLAminus -149.62, 174.69 57.3, 76.73 -95.24, 8.98 282.05, 96.12 -51.11, -35.54 in-in in 8.642 Saltbr-in 2.675 HRD-in -62.32, -48.48 63.55, 4.44 in-in-in SNCiii in-in ActLoopNT-in 3.043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.42, 143.72 APE9-dihe-na 129.46, -175.16 APE8-dihe-in -98.28, 125.3 APE8-rot-in 312.69 APE67-dihe-inflip 98.15, -18.1 -45.11, 129.51 APE12-dist-in 10.201 APE11-dist-in 11.247 APE10-dist-in 5.61 APE9-dist-in 3.639 None None None XRAY 2.9 0.193 999.0 B 543 475 0 0 0 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4ZA P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.913 13.235 BLAminus -149.46, 171.26 70.91, 78.39 -108.02, 16.47 270.55, 111.24 -69.43, -16.01 in-in in 8.736 Saltbr-in 2.716 HRD-in -71.08, -53.07 69.31, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.878 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.53, 147.45 APE9-dihe-na 134.96, -165.72 APE8-dihe-in -111.39, 128.56 APE8-rot-in 296.58 APE67-dihe-inflip 96.79, -17.75 -54.96, 131.39 APE12-dist-in 10.43 APE11-dist-in 11.113 APE10-dist-in 5.49 APE9-dist-in 3.542 None None None XRAY 1.84 0.193 999.0 A 543 493 0 0 0 0 [[187, 452]] 1.0 3c4z Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C50A P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.075 13.034 BLAminus -142.59, 172.43 68.85, 78.38 -104.12, 14.36 280.99, 104.76 -67.57, -15.07 in-in in 8.602 Saltbr-in 2.925 HRD-in -76.21, -52.36 64.46, 15.62 in-in-in SNCiii in-in ActLoopNT-in 2.795 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.66, 144.27 APE9-dihe-na 130.37, -165.26 APE8-dihe-in -104.68, 131.22 APE8-rot-in 300.48 APE67-dihe-inflip 92.29, -6.18 -56.88, 135.03 APE12-dist-in 10.685 APE11-dist-in 11.469 APE10-dist-in 5.876 APE9-dist-in 3.473 None None None XRAY 2.6 0.19 999.0 A 543 499 0 0 0 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C50B P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.078 13.068 BLAminus -140.52, 175.4 66.53, 77.05 -104.14, 18.55 279.39, 103.87 -67.23, -21.39 in-in in 8.532 Saltbr-in 2.721 HRD-in -71.74, -52.34 63.89, 11.32 in-in-in SNCiii in-in ActLoopNT-in 2.89 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.47, 143.37 APE9-dihe-na 137.53, -168.17 APE8-dihe-in -105.39, 125.32 APE8-rot-in 297.12 APE67-dihe-inflip 95.82, -17.57 -51.32, 135.4 APE12-dist-in 10.129 APE11-dist-in 11.115 APE10-dist-in 5.538 APE9-dist-in 3.418 None None None XRAY 2.6 0.19 999.0 B 543 496 0 0 0 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C51A P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.735 13.235 BLAminus -156.28, 178.74 57.85, 73.51 -84.14, -2.01 283.03, 106.57 -47.35, -22.99 in-in in 8.798 Saltbr-in 2.687 HRD-in -64.41, -45.82 69.5, -19.46 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.64, 142.5 APE9-dihe-na 155.52, -169.52 APE8-dihe-in -101.5, 135.25 APE8-rot-in 300.99 APE67-dihe-inflip 84.91, 4.53 -59.96, 128.0 APE12-dist-in 10.573 APE11-dist-in 11.541 APE10-dist-in 6.152 APE9-dist-in 3.937 None None None XRAY 3.55 0.281 999.0 A 543 487 0 0 0 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C51B P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.785 13.187 BLAminus -156.29, 175.57 58.57, 74.43 -85.29, -1.69 285.99, 107.07 -47.38, -22.91 in-in in 8.696 Saltbr-in 2.792 HRD-in -66.67, -42.5 63.68, -15.39 in-in-in SNCiii in-in ActLoopNT-in 2.969 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.05, 141.93 APE9-dihe-na 155.26, -171.96 APE8-dihe-in -101.33, 138.35 APE8-rot-in 299.85 APE67-dihe-inflip 84.6, 5.24 -64.39, 128.67 APE12-dist-in 10.537 APE11-dist-in 11.598 APE10-dist-in 6.156 APE9-dist-in 3.94 None None None XRAY 3.55 0.281 999.0 B 543 461 20 0 0 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9A P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.852 13.484 BLAminus -151.04, 174.48 70.22, 99.25 -129.57, 18.73 275.22, 99.19 -61.63, -18.96 in-in in 8.961 Saltbr-in 3.127 HRD-in -61.98, -58.15 73.37, -3.42 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.32, 133.82 APE9-dihe-na 142.48, -169.15 APE8-dihe-in -104.33, 125.71 APE8-rot-in 302.67 APE67-dihe-inflip 104.42, -3.83 -50.74, 122.55 APE12-dist-in 10.356 APE11-dist-in 11.014 APE10-dist-in 5.5 APE9-dist-in 3.664 T8C,N480C None None XRAY 2.7 0.194 0.229 A 543 486 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9B P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.899 13.504 BLAminus -154.17, 173.67 70.5, 100.81 -132.54, 18.75 276.87, 97.69 -56.57, -24.02 in-in in 8.931 Saltbr-in 3.099 HRD-in -65.24, -58.34 73.4, -2.88 in-in-in SNCiii in-in ActLoopNT-in 2.934 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -166.53, 132.45 APE9-dihe-na 145.72, -169.79 APE8-dihe-in -103.09, 126.5 APE8-rot-in 303.38 APE67-dihe-inflip 99.94, -4.73 -52.12, 123.93 APE12-dist-in 10.368 APE11-dist-in 11.038 APE10-dist-in 5.525 APE9-dist-in 3.677 T8C,N480C None None XRAY 2.7 0.194 0.229 B 543 481 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9C P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.868 13.481 BLAminus -151.87, 172.48 72.03, 98.62 -128.19, 19.72 276.34, 98.38 -59.47, -19.79 in-in in 8.951 Saltbr-in 3.107 HRD-in -62.09, -58.44 72.04, -1.68 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.26, 134.05 APE9-dihe-na 142.83, -170.11 APE8-dihe-in -104.04, 126.58 APE8-rot-in 301.36 APE67-dihe-inflip 105.14, -2.81 -49.9, 120.73 APE12-dist-in 10.384 APE11-dist-in 11.018 APE10-dist-in 5.508 APE9-dist-in 3.673 T8C,N480C None None XRAY 2.7 0.194 0.229 C 543 482 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9D P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.923 13.517 BLAminus -151.29, 174.11 71.25, 99.27 -130.54, 20.81 276.77, 98.72 -58.99, -24.3 in-in in 8.931 Saltbr-in 3.091 HRD-in -63.44, -57.63 71.87, -0.43 in-in-in SNCiii in-in ActLoopNT-in 2.927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.95, 134.69 APE9-dihe-na 141.2, -168.54 APE8-dihe-in -103.28, 126.55 APE8-rot-in 303.76 APE67-dihe-inflip 102.49, -2.5 -51.29, 121.62 APE12-dist-in 10.397 APE11-dist-in 11.044 APE10-dist-in 5.513 APE9-dist-in 3.693 T8C,N480C None None XRAY 2.7 0.194 0.229 D 543 486 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC PRKACA KAPCA_BOVIN 9DW9G P00517 13 351 351.0 ATP:401 ATPlike Active DFGin 6.569 15.126 BLAminus -133.9, -169.96 59.46, 64.31 -83.85, 33.99 275.29, 73.58 -66.33, -24.36 in-in in 9.499 Saltbr-in 3.217 HRD-in -92.3, -53.34 68.25, 14.14 in-in-in SNCiii in-in ActLoopNT-in 3.08 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.91, 151.76 APE9-dihe-na 126.66, -174.62 APE8-dihe-in -92.84, 130.69 APE8-rot-in 299.41 APE67-dihe-in -68.55, -23.13 -58.33, -34.44 APE12-dist-in 8.703 APE11-dist-in 11.563 APE10-dist-in 6.17 APE9-dist-in 4.568 None TPO198 TPO198 EM 2.8 999.0 999.0 G 351 328 0 0 0 0 [[44, 298]] 1.0 9dw9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_BOVIN 1Q24A P00517 15 351 351.0 ATP:60400 ATPlike Active DFGin 5.983 14.319 BLAminus -113.95, 178.0 66.86, 85.15 -103.99, 32.82 274.7, 64.8 -65.44, -25.66 in-in in 8.779 Saltbr-in 2.742 HRD-in -93.22, -55.61 73.46, 14.95 in-in-in SNCiii in-in ActLoopNT-in 3.09 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.66, 162.77 APE9-dihe-na 133.15, -143.39 APE8-dihe-in -135.22, 127.61 APE8-rot-in 301.89 APE67-dihe-in -67.43, -30.61 -42.63, -46.05 APE12-dist-in 8.036 APE11-dist-in 11.447 APE10-dist-in 6.024 APE9-dist-in 3.486 V124A,L174M TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.202 0.25 A 350 337 0 0 0 0 [[44, 298]] 1.0 1q24 Bos taurus AGC_PRKACA_BOVIN AGC 4.8e-94 320.4 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CMGC CKA1 A0A1D8PUA2_CANAL 6O6QA A0A1D8PUA2 4 333 335.0 AMP:401 ATPlike Active DFGin 7.386 16.256 BLAminus -114.24, -174.82 59.27, 62.07 -85.23, 23.85 304.56, 80.46 -69.03, -20.65 in-in in 9.001 Saltbr-in 2.88 HRD-in -68.75, -45.06 62.13, 23.87 in-in-in SNCiii in-in ActLoopNT-in 3.222 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.59, 173.17 APE9-dihe-na 57.84, -166.47 APE8-dihe-in -122.64, 160.2 APE8-rot-in 318.49 APE67-dihe-in -66.36, -14.81 -53.74, -47.77 APE12-dist-in 12.507 APE11-dist-in 10.219 APE10-dist-in 6.094 APE9-dist-in 3.225 None None None XRAY 2.7 0.236 0.287 A 335 326 4 0 0 0 [[43, 327]] 1.0 6o6q Candida albicans CMGC_CKA1_CANAL CMGC 1.1e-62 217.9 1 301 301 178 179 180 182 184 72 85 89 157 159 158 160 218 205 200 199 198 197 196 195 194 118 Casein kinase II subunit alpha
CMGC CKA1 A0A1D8PUA2_CANAL 6O6QB A0A1D8PUA2 5 333 335.0 AMP:401 ATPlike Active DFGin 7.292 15.98 BLAminus -125.13, -179.74 57.94, 64.68 -85.91, 27.32 303.1, 76.17 -70.46, -30.29 in-in in 9.011 Saltbr-in 2.813 HRD-in -81.71, -46.62 63.63, 27.36 in-in-in SNCiii in-in ActLoopNT-in 2.902 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.56, 167.57 APE9-dihe-na 58.76, -171.72 APE8-dihe-in -113.79, 160.74 APE8-rot-in 318.5 APE67-dihe-in -64.2, -12.3 -53.09, -54.06 APE12-dist-in 12.689 APE11-dist-in 10.132 APE10-dist-in 6.255 APE9-dist-in 3.214 None None None XRAY 2.7 0.236 0.287 B 335 325 4 0 0 0 [[43, 327]] 1.0 6o6q Candida albicans CMGC_CKA1_CANAL CMGC 1.1e-62 217.9 1 301 301 178 179 180 182 184 72 85 89 157 159 158 160 218 205 200 199 198 197 196 195 194 118 Casein kinase II subunit alpha
AGC PRKACA KAPCA_CRIGR 6EM7A P25321 11 351 351.0 ADP:60403 ATPlike Active DFGin 5.924 14.338 BLAminus -118.71, 173.1 68.53, 85.06 -96.18, 23.36 270.78, 55.34 -59.75, -28.55 in-in in 8.741 Saltbr-in 2.711 HRD-in -88.33, -53.93 74.88, 10.19 in-in-in SNCiii in-in ActLoopNT-in 2.967 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.73, 159.92 APE9-dihe-na 127.98, -160.75 APE8-dihe-in -119.5, 137.47 APE8-rot-in 298.57 APE67-dihe-in -59.39, -22.73 -49.47, -50.59 APE12-dist-in 8.05 APE11-dist-in 11.429 APE10-dist-in 5.809 APE9-dist-in 3.674 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.238 0.139 0.157 A 353 341 0 0 0 0 [[44, 298]] 1.0 6em7 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_CRIGR 6EMAA P25321 12 351 351.0 ATP:60401 ATPlike Active DFGin 6.847 14.028 BLAminus -121.3, 163.01 76.03, 95.19 -107.48, 29.41 285.05, 72.84 -63.27, -23.25 in-in in 8.581 Saltbr-in 2.912 HRD-in -88.06, -51.23 73.05, 9.34 in-in-in SNCiii in-in ActLoopNT-in 2.843 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.85, 162.03 APE9-dihe-na 127.51, -167.2 APE8-dihe-in -113.51, 133.85 APE8-rot-in 299.54 APE67-dihe-in -58.99, -24.47 -49.7, -50.19 APE12-dist-in 8.208 APE11-dist-in 11.434 APE10-dist-in 5.777 APE9-dist-in 3.585 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.88 0.184 0.213 A 353 340 0 0 0 0 [[44, 298]] 1.0 6ema Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_CRIGR 6ESAA P25321 11 351 351.0 AMP:60401 ATPlike Active DFGin 6.139 14.365 BLAminus -120.63, 169.73 70.22, 89.96 -100.72, 24.5 270.85, 56.09 -58.05, -28.66 in-in in 8.691 Saltbr-in 2.873 HRD-in -93.01, -53.86 73.79, 10.3 in-in-in SNCiii in-in ActLoopNT-in 2.964 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.44, 160.95 APE9-dihe-na 124.73, -163.46 APE8-dihe-in -117.05, 136.25 APE8-rot-in 299.26 APE67-dihe-in -59.89, -22.61 -49.24, -49.61 APE12-dist-in 8.091 APE11-dist-in 11.499 APE10-dist-in 5.822 APE9-dist-in 3.66 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.307 0.132 0.147 A 353 341 0 0 0 0 [[44, 298]] 1.0 6esa Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_CRIGR 6Y8CA P25321 13 351 351.0 ATP:60402 ATPlike Active DFGin 5.727 14.302 BLAminus -123.99, 172.57 69.5, 82.73 -92.15, 25.74 279.44, 63.0 -58.78, -31.82 in-in in 9.166 Saltbr-in 2.638 HRD-in -96.49, -52.39 69.1, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.28, 160.42 APE9-dihe-na 122.78, -169.96 APE8-dihe-in -106.17, 134.07 APE8-rot-in 304.81 APE67-dihe-in -60.24, -22.7 -48.33, -48.43 APE12-dist-in 8.044 APE11-dist-in 11.517 APE10-dist-in 5.939 APE9-dist-in 3.895 None TPO198,SEP339 TPO198,SEP339 XRAY 1.76 0.162 0.19 A 353 339 0 0 0 0 [[44, 298]] 1.0 6y8c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CMGC CK2 Q5KF69_CRYD1 6ISEA Q5KF69 5 331 336.0 ANP:403 ATPlike Active DFGin 7.339 16.208 BLAminus -129.3, -170.99 44.36, 71.77 -91.05, 22.67 299.01, 82.29 -66.02, -23.99 in-in in 9.482 Saltbr-in 3.336 HRD-in -65.48, -54.09 76.82, 9.27 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.0, -19.23 APE9-dihe-na -99.69, -172.72 APE8-dihe-in -80.09, 147.5 APE8-rot-in 301.93 APE67-dihe-in -61.24, -16.59 -47.75, -58.81 APE12-dist-in 12.687 APE11-dist-in 10.631 APE10-dist-in 6.144 APE9-dist-in 3.609 None None None XRAY 2.8 0.198 0.23 A 338 327 0 0 0 0 [[38, 323]] 1.0 6ise Cryptococcus deneoformans CMGC_CK2_CRYD1 CMGC 6e-64 222.0 1 301 301 173 174 175 177 179 67 80 84 152 154 153 155 213 200 195 194 193 192 191 190 189 113 Casein kinase II subunit alpha
CMGC CK2 Q5KF69_CRYD1 6ISEB Q5KF69 5 331 336.0 ANP:403 ATPlike Active DFGin 7.308 16.238 BLAminus -133.11, -171.48 44.36, 73.35 -91.98, 23.51 299.28, 79.86 -68.68, -21.78 in-in in 9.591 Saltbr-in 3.496 HRD-in -67.7, -51.8 75.87, 7.92 in-in-in SNCiii in-in ActLoopNT-in 2.976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.38, 168.0 APE9-dihe-na 74.76, -173.48 APE8-dihe-in -110.86, 148.66 APE8-rot-in 271.82 APE67-dihe-in -65.62, -23.31 -54.68, -45.78 APE12-dist-in 12.576 APE11-dist-in 10.311 APE10-dist-in 6.266 APE9-dist-in 3.367 None None None XRAY 2.8 0.198 0.23 B 338 327 0 0 0 0 [[38, 323]] 1.0 6ise Cryptococcus deneoformans CMGC_CK2_CRYD1 CMGC 6e-64 222.0 1 301 301 173 174 175 177 179 67 80 84 152 154 153 155 213 200 195 194 193 192 191 190 189 113 Casein kinase II subunit alpha
CMGC CKA1 J9VNH4_CRYN9 6KO6B J9VNH4 5 334 338.0 ANP:401 ATPlike Active DFGin 7.298 16.236 BLAminus -115.02, -165.9 52.87, 72.55 -94.97, 21.12 299.2, 77.23 -71.99, -18.35 in-in in 9.324 Saltbr-in 3.151 HRD-in -64.53, -49.64 63.27, 19.41 in-in-in SNCiii in-in ActLoopNT-in 3.055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.45, 156.98 APE9-dihe-na 76.83, -179.82 APE8-dihe-in -92.38, 159.35 APE8-rot-in 277.62 APE67-dihe-in -71.62, -13.46 -53.06, -52.26 APE12-dist-in 12.792 APE11-dist-in 10.474 APE10-dist-in 6.177 APE9-dist-in 3.249 None None None XRAY 2.4 0.238 0.268 B 338 330 0 0 0 0 [[38, 323]] 1.0 6ko6 Cryptococcus neoformans CMGC_CKA1_CRYN9 CMGC 6e-64 222.0 1 301 301 173 174 175 177 179 67 80 84 152 154 153 155 213 200 195 194 193 192 191 190 189 113 Casein kinase II subunit alpha
OTHER PK1 A0A097P1P8_GVCP 6VVGA A0A097P1P8 3 279 279.0 AMP:301 ATPlike Active DFGin 9.47 12.504 BLAminus -139.45, 174.39 59.11, 72.82 -82.01, 20.88 324.49, 136.4 -73.16, -16.8 na-na na 15.471 Saltbr-na 12.976 HRD-in -69.17, -49.37 73.82, 3.86 na-in-in SNCaii in-in ActLoopNT-in 2.866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.58, 157.03 APE9-dihe-na 90.57, -158.23 APE8-dihe-in -103.25, 120.97 APE8-rot-in 311.05 APE67-dihe-in -75.71, -2.76 -55.41, -39.8 APE12-dist-in 10.799 APE11-dist-in 12.039 APE10-dist-in 6.083 APE9-dist-in 4.885 None None None XRAY 2.01 0.195 0.225 A 279 267 10 0 0 0 [[17, 277]] 1.0 6vvg Cydia pomonella granulosis virus OTHER_PK1_GVCP CAMK 1.9e-45 161.2 8 256 249 159 160 161 163 165 49 62 66 138 140 139 141 195 183 178 177 176 175 174 173 172 92 PK-1
OTHER PK1 A0A097P1P8_GVCP 6VVGB A0A097P1P8 3 278 279.0 AMP:301 ATPlike Active DFGin 9.485 12.665 BLAminus -138.4, 172.21 59.64, 73.0 -83.58, 22.42 324.54, 137.78 -67.63, -19.86 na-na na 15.282 Saltbr-na 13.214 HRD-in -58.02, -51.7 78.84, -1.77 na-in-in SNCaii in-in ActLoopNT-in 2.858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.97, 161.51 APE9-dihe-na 88.81, -151.71 APE8-dihe-in -109.06, 113.8 APE8-rot-in 308.85 APE67-dihe-in -72.96, -2.91 -51.95, -43.87 APE12-dist-in 10.828 APE11-dist-in 12.169 APE10-dist-in 6.178 APE9-dist-in 4.697 None None None XRAY 2.01 0.195 0.225 B 279 264 12 0 0 0 [[17, 277]] 1.0 6vvg Cydia pomonella granulosis virus OTHER_PK1_GVCP CAMK 1.9e-45 161.2 8 256 249 159 160 161 163 165 49 62 66 138 140 139 141 195 183 178 177 176 175 174 173 172 92 PK-1
CAMK CAMKII KCC2A_DROME 5FG8A Q00168 7 275 530.0 ADP:301 ATPlike Active DFGin 5.883 14.23 BLAminus -120.35, -179.38 64.2, 77.37 -92.62, 22.59 287.14, 78.3 -59.18, -27.49 in-in in 8.996 Saltbr-in 2.798 HRD-in -79.26, -45.5 78.31, -3.25 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.29, 153.59 APE9-dihe-na 138.39, -158.82 APE8-dihe-in -123.15, 126.57 APE8-rot-in 291.32 APE67-dihe-in -61.12, -15.42 -38.96, -61.46 APE12-dist-in 10.208 APE11-dist-in 11.816 APE10-dist-in 6.289 APE9-dist-in 3.479 None None None XRAY 1.955 0.192 0.221 A 285 269 0 0 0 0 [[14, 272]] 1.0 5fg8 Drosophila melanogaster CAMK_CAMKII_DROME CAMK 6.3e-98 333.1 1 256 256 156 157 158 160 162 43 61 65 133 135 134 136 196 184 179 178 177 176 175 174 173 91 Calcium/calmodulin-dependent protein kinase type II alpha chain
CAMK CAMKII KCC2A_DROME 5H9BA Q00168 7 275 530.0 AN2:301 ATPlike Active DFGin 5.687 14.14 BLAminus -121.83, -177.58 63.45, 84.2 -103.14, 25.35 292.56, 80.33 -62.44, -18.79 in-in in 9.014 Saltbr-in 2.65 HRD-in -79.17, -42.13 69.98, 5.32 in-in-in SNCiii in-in ActLoopNT-in 3.047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.23, 154.68 APE9-dihe-na 138.91, -156.64 APE8-dihe-in -125.98, 126.82 APE8-rot-in 298.36 APE67-dihe-in -64.57, -17.97 -35.44, -64.1 APE12-dist-in 10.217 APE11-dist-in 11.689 APE10-dist-in 6.016 APE9-dist-in 3.419 None None None XRAY 2.25 0.204 0.222 A 285 269 0 0 0 0 [[14, 272]] 1.0 5h9b Drosophila melanogaster CAMK_CAMKII_DROME CAMK 6.3e-98 333.1 1 256 256 156 157 158 160 162 43 61 65 133 135 134 136 196 184 179 178 177 176 175 174 173 91 Calcium/calmodulin-dependent protein kinase type II alpha chain
CAMK CAMKII KCC2A_DROME 5HU3A Q00168 7 272 530.0 ADP:301 ATPlike Active DFGin 5.625 14.217 BLAminus -125.3, -175.54 57.54, 73.58 -90.7, 26.83 289.37, 84.29 -62.44, -29.23 in-in in 8.952 Saltbr-in 2.671 HRD-in -75.88, -45.31 74.57, -1.26 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.12, 157.18 APE9-dihe-na 139.99, -158.88 APE8-dihe-in -121.63, 130.83 APE8-rot-in 294.31 APE67-dihe-in -66.75, -12.95 -42.37, -59.45 APE12-dist-in 10.059 APE11-dist-in 11.766 APE10-dist-in 6.277 APE9-dist-in 3.564 D136N None None XRAY 1.885 0.194 0.228 A 285 266 0 0 0 0 [[14, 272]] 1.0 5hu3 Drosophila melanogaster CAMK_CAMKII_DROME CAMK 5.7e-97 329.9 1 256 256 156 157 158 160 162 43 61 65 133 135 134 136 196 184 179 178 177 176 175 174 173 91 Calcium/calmodulin-dependent protein kinase type II alpha chain
CAMK CDPK Q3HNM4_EIMTE 4YSJA Q3HNM4 26 499 505.0 ADP:60506 ATPlike Active DFGin 6.651 14.005 BLAminus -140.39, -165.72 52.75, 66.63 -84.34, 22.0 285.15, 82.54 -78.31, -16.63 in-in in 8.319 Saltbr-in 3.482 HRD-in -81.29, -53.0 84.02, -6.2 in-in-in SNCiii in-in ActLoopNT-in 2.898 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.58, 142.92 APE9-dihe-na 138.88, -163.22 APE8-dihe-in -136.98, 140.82 APE8-rot-in 303.29 APE67-dihe-in -62.88, -33.46 -45.59, -53.66 APE12-dist-in 9.144 APE11-dist-in 11.564 APE10-dist-in 5.99 APE9-dist-in 3.493 None None None XRAY 2.7 0.249 0.292 A 491 459 10 0 0 0 [[46, 303]] 1.0 4ysj Eimeria tenella CAMK_CDPK_EIMTE CAMK 6.1e-90 307.2 1 256 256 189 190 191 193 195 75 94 98 166 168 167 169 227 216 211 210 209 208 207 206 205 124 non-specific serine/threonine protein kinase
CAMK CDPK Q3HNM4_EIMTE 4YSJB Q3HNM4 26 499 505.0 ADP:60506 ATPlike Active DFGin 6.595 13.993 BLAminus -140.54, -165.92 54.1, 65.38 -84.49, 22.28 285.29, 82.38 -78.18, -16.85 in-in in 8.3 Saltbr-in 3.494 HRD-in -81.3, -52.72 84.55, -6.86 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.46, 142.21 APE9-dihe-na 137.64, -162.65 APE8-dihe-in -138.56, 141.54 APE8-rot-in 303.24 APE67-dihe-in -62.83, -32.98 -44.74, -55.37 APE12-dist-in 8.901 APE11-dist-in 11.534 APE10-dist-in 5.979 APE9-dist-in 3.505 None None None XRAY 2.7 0.249 0.292 B 491 462 10 0 0 0 [[46, 303]] 1.0 4ysj Eimeria tenella CAMK_CDPK_EIMTE CAMK 6.1e-90 307.2 1 256 256 189 190 191 193 195 75 94 98 166 168 167 169 227 216 211 210 209 208 207 206 205 124 non-specific serine/threonine protein kinase
TYR PTK2 FAK1_CHICK 6TY4A Q00944 34 686 1053.0 ANP:702 ATPlike Active DFGin 7.546 15.951 BLAminus -124.05, -151.88 51.86, 82.13 -107.99, 32.9 286.39, 85.0 -72.01, -36.58 in-in in 8.437 Saltbr-in 3.562 HRD-in -70.16, -30.0 74.19, -18.38 in-in-in SNCiii in-in ActLoopNT-in 2.815 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -86.31, 66.54 APE9-dihe-in -63.31, 139.75 APE8-dihe-in -64.41, 127.23 APE8-rot-na 22.65 APE67-dihe-in -56.19, -42.03 -70.19, -41.73 APE12-dist-na 11.489 APE11-dist-na 10.184 APE10-dist-na 13.636 APE9-dist-in 7.205 None None None EM 5.96 999.0 999.0 A 658 621 0 0 0 0 [[422, 678]] 1.0 6ty4 Gallus gallus TYR_PTK2_CHICK TYR 1.5e-91 312.7 1 260 260 563 564 565 567 569 454 471 475 543 545 544 546 604 592 587 586 585 584 583 582 581 500 Focal adhesion kinase 1
TYR PTK2 FAK1_CHICK 6TY4B Q00944 34 686 1053.0 ANP:702 ATPlike Active DFGin 7.546 15.95 BLAminus -124.03, -151.9 51.82, 82.14 -107.99, 32.89 286.33, 85.06 -71.97, -36.56 in-in in 8.436 Saltbr-in 3.562 HRD-in -70.15, -30.0 74.26, -18.38 in-in-in SNCiii in-in ActLoopNT-in 2.815 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -86.3, 66.56 APE9-dihe-in -63.34, 139.79 APE8-dihe-in -64.42, 127.23 APE8-rot-na 22.65 APE67-dihe-in -56.21, -42.01 -70.19, -41.71 APE12-dist-na 11.489 APE11-dist-na 10.183 APE10-dist-na 13.636 APE9-dist-in 7.205 None None None EM 5.96 999.0 999.0 B 658 621 0 0 0 0 [[422, 678]] 1.0 6ty4 Gallus gallus TYR_PTK2_CHICK TYR 1.5e-91 312.7 1 260 260 563 564 565 567 569 454 471 475 543 545 544 546 604 592 587 586 585 584 583 582 581 500 Focal adhesion kinase 1
TYR SRC SRC_CHICK 3DQWA P00523 255 533 533.0 AGS:534 ATPlike Active DFGin 6.357 14.133 BLAminus -133.72, -176.8 56.69, 80.14 -98.42, 17.02 297.52, 87.02 -49.14, -41.19 in-in in 7.931 Saltbr-in 2.687 HRD-in -86.31, -48.96 78.42, -4.92 in-in-in SNCiii in-in ActLoopNT-in 3.014 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -125.37, 137.46 APE9-dihe-in -129.59, 150.85 APE8-dihe-in -68.35, 111.94 APE8-rot-na 22.98 APE67-dihe-in -63.37, -24.29 -54.33, -47.45 APE12-dist-na 14.454 APE11-dist-na 9.918 APE10-dist-na 12.726 APE9-dist-in 6.835 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 A 286 279 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQWB P00523 255 533 533.0 AGS:534 ATPlike Active DFGin 6.515 14.112 BLAminus -130.32, -179.28 59.57, 78.46 -98.37, 14.52 296.04, 88.38 -51.47, -39.24 in-in in 7.861 Saltbr-in 2.594 HRD-in -92.73, -49.37 74.2, -0.04 in-in-in SNCiii in-in ActLoopNT-in 2.955 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -118.73, 138.44 APE9-dihe-in -131.19, 150.2 APE8-dihe-in -68.24, 113.76 APE8-rot-na 20.72 APE67-dihe-in -68.02, -21.16 -58.05, -42.12 APE12-dist-na 14.577 APE11-dist-na 10.068 APE10-dist-na 12.667 APE9-dist-in 6.835 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 B 286 279 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQWC P00523 258 533 533.0 AGS:534 ATPlike Active DFGin 7.23 15.586 BLAminus -138.39, -169.49 49.44, 64.48 -88.87, 22.55 279.28, 86.64 -59.44, -34.1 in-in in 7.666 Saltbr-in 3.046 HRD-in -87.18, -49.68 80.05, -15.46 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -114.69, 105.75 APE9-dihe-in -126.06, 131.23 APE8-dihe-in -49.28, 106.82 APE8-rot-na 333.72 APE67-dihe-in -71.67, -16.03 -52.29, -42.49 APE12-dist-na 14.071 APE11-dist-na 9.851 APE10-dist-na 10.947 APE9-dist-in 6.124 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 C 286 276 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQWD P00523 257 533 533.0 AGS:534 ATPlike Active DFGin 7.183 15.5 BLAminus -135.25, -176.07 62.11, 64.12 -89.05, 15.75 281.43, 79.51 -51.86, -37.09 in-in in 7.529 Saltbr-in 3.018 HRD-in -81.74, -56.17 86.4, -15.46 in-in-in SNCiii in-in ActLoopNT-in 2.971 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -120.41, 149.47 APE9-dihe-in -128.09, 155.96 APE8-dihe-in -55.17, 98.07 APE8-rot-na 334.76 APE67-dihe-in -67.99, -16.44 -49.1, -40.45 APE12-dist-na 15.071 APE11-dist-na 10.305 APE10-dist-na 13.293 APE9-dist-in 6.675 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 D 286 277 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQXB P00523 259 533 533.0 AMP:2 ATPlike Active DFGin 6.808 14.815 BLAminus -123.08, -167.74 51.93, 60.88 -81.23, 10.84 295.11, 95.49 -43.33, -48.19 in-in in 7.906 Saltbr-in 3.425 HRD-in -73.53, -53.77 83.73, -6.08 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -120.36, 128.73 APE9-dihe-in -122.57, 114.22 APE8-dihe-in -63.43, 112.38 APE8-rot-na 23.41 APE67-dihe-in -72.31, -17.76 -46.16, -42.59 APE12-dist-na 10.885 APE11-dist-na 6.755 APE10-dist-na 9.999 APE9-dist-in 5.75 None None None XRAY 2.3 0.194 0.241 B 286 268 7 0 0 7 [[267, 518]] 1.0 3dqx Gallus gallus TYR_SRC_CHICK TYR 3.4e-94 320.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
AGC AKT1 AKT1_HUMAN 4EKKA P31749 144 477 480.0 ANP:60501 ATPlike Active DFGin 6.048 13.113 BLAminus -112.5, -177.27 66.46, 90.66 -111.95, 23.34 296.26, 86.16 -69.26, -23.9 in-in in 8.651 Saltbr-in 2.978 HRD-in -63.51, -40.13 66.5, -18.58 in-in-in SNCiii in-in ActLoopNT-in 3.05 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.71, 172.01 APE9-dihe-na 121.09, -152.4 APE8-dihe-in -119.32, 125.09 APE8-rot-in 285.38 APE67-dihe-in -63.61, -25.53 -44.69, -42.52 APE12-dist-in 8.814 APE11-dist-in 11.718 APE10-dist-in 6.07 APE9-dist-in 4.069 S473D TPO308 TPO308 XRAY 2.8 0.22 0.28 A 341 319 0 0 0 0 [[150, 408]] 1.0 4ekk Homo sapiens AGC_AKT1_HUMAN AGC 2.3e-99 337.7 1 260 260 291 292 293 295 297 179 198 202 271 273 272 274 331 319 314 313 312 311 310 309 308 228 RAC-alpha serine/threonine-protein kinase
AGC AKT1 AKT1_HUMAN 4EKKB P31749 144 477 480.0 ANP:60501 ATPlike Active DFGin 6.075 13.046 BLAminus -112.98, 175.61 60.18, 117.01 -127.72, 18.67 304.81, 92.19 -54.85, -36.32 in-in in 8.766 Saltbr-in 2.665 HRD-in -65.56, -47.0 73.75, -27.2 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.2, 164.76 APE9-dihe-na 136.6, -155.35 APE8-dihe-in -114.57, 129.15 APE8-rot-in 273.31 APE67-dihe-in -63.86, -22.96 -45.74, -46.48 APE12-dist-in 8.77 APE11-dist-in 11.686 APE10-dist-in 6.125 APE9-dist-in 4.285 S473D TPO308 TPO308 XRAY 2.8 0.22 0.28 B 341 319 0 0 0 0 [[150, 408]] 1.0 4ekk Homo sapiens AGC_AKT1_HUMAN AGC 2.3e-99 337.7 1 260 260 291 292 293 295 297 179 198 202 271 273 272 274 331 319 314 313 312 311 310 309 308 228 RAC-alpha serine/threonine-protein kinase
AGC AKT2 AKT2_HUMAN 1O6KA P31751 146 479 481.0 ANP:1480 ATPlike Active DFGin 6.146 12.734 BLAminus -120.8, -176.05 56.87, 82.9 -98.82, 24.49 299.36, 92.56 -61.37, -25.29 in-in in 8.749 Saltbr-in 2.796 HRD-in -73.34, -45.79 65.54, -9.2 in-in-in SNCiii in-in ActLoopNT-in 3.027 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.85, 170.7 APE9-dihe-na 130.02, -155.15 APE8-dihe-in -119.36, 127.57 APE8-rot-in 291.96 APE67-dihe-in -68.55, -16.48 -36.55, -56.12 APE12-dist-in 8.193 APE11-dist-in 11.759 APE10-dist-in 6.119 APE9-dist-in 3.921 S474D TPO309 TPO309 XRAY 1.7 0.205 0.234 A 336 318 0 0 0 0 [[152, 409]] 1.0 1o6k Homo sapiens AGC_AKT2_HUMAN AGC 1.7e-99 338.1 1 260 260 292 293 294 296 298 181 200 204 272 274 273 275 332 320 315 314 313 312 311 310 309 230 RAC-beta serine/threonine-protein kinase
AGC AKT2 AKT2_HUMAN 1O6LA P31751 146 477 481.0 ANP:61480 ATPlike Active DFGin 6.258 12.925 BLAminus -121.53, -178.18 58.41, 83.34 -98.83, 24.71 297.57, 89.85 -63.5, -19.94 in-in in 8.794 Saltbr-in 2.76 HRD-in -74.06, -43.29 62.88, -5.6 in-in-in SNCiii in-in ActLoopNT-in 3.006 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.79, 169.91 APE9-dihe-na 133.49, -153.33 APE8-dihe-in -120.8, 127.55 APE8-rot-in 289.07 APE67-dihe-in -68.04, -17.15 -37.13, -54.04 APE12-dist-in 8.173 APE11-dist-in 11.74 APE10-dist-in 6.122 APE9-dist-in 3.747 None TPO309 TPO309 XRAY 1.6 0.198 0.227 A 337 312 0 0 0 0 [[152, 409]] 1.0 1o6l Homo sapiens AGC_AKT2_HUMAN AGC 1.8e-99 338.1 1 260 260 292 293 294 296 298 181 200 204 272 274 273 275 332 320 315 314 313 312 311 310 309 230 RAC-beta serine/threonine-protein kinase
AGC CDC42BPB MRCKB_HUMAN 4UAKA Q9Y5S2 2 417 1711.0 ADP:60501 ATPlike Active DFGin 6.536 13.389 BLAminus -126.67, 169.91 71.43, 81.15 -99.11, 14.11 300.02, 102.96 -73.12, -5.53 in-in in 8.635 Saltbr-in 2.748 HRD-in -78.82, -49.28 69.95, 4.01 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.28, 157.85 APE9-dihe-na 87.21, -164.86 APE8-dihe-in -127.15, 132.61 APE8-rot-in 302.21 APE67-dihe-in -64.23, -20.61 -57.86, -36.49 APE12-dist-in 10.511 APE11-dist-in 11.151 APE10-dist-in 6.313 APE9-dist-in 3.548 None None None XRAY 1.73 0.198 0.243 A 419 401 0 0 0 0 [[76, 342]] 1.0 4uak Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
AGC GRK4 GRK4_HUMAN 4YHJA P32298 25 525 578.0 AN2:601 ATPlike Active DFGin 6.129 13.374 BLAminus -118.16, -176.89 50.04, 69.58 -89.94, 31.88 285.36, 98.48 -66.46, -45.19 in-in in 9.266 Saltbr-in 3.026 HRD-in -63.35, -45.97 74.46, -21.42 in-in-in SNCiii in-in ActLoopNT-in 2.855 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.22, 157.81 APE9-dihe-na 113.97, -154.87 APE8-dihe-in -108.33, 139.74 APE8-rot-in 312.15 APE67-dihe-inflip 104.58, -18.92 -61.34, 124.85 APE12-dist-in 11.453 APE11-dist-in 12.888 APE10-dist-in 6.916 APE9-dist-in 4.145 C563S,C578S None None XRAY 2.6 0.2 0.248 A 584 501 0 0 0 0 [[187, 449]] 1.0 4yhj Homo sapiens AGC_GRK4_HUMAN AGC 8.1e-84 286.9 1 260 260 329 330 331 333 335 216 235 239 309 311 310 312 368 356 351 350 349 348 347 346 345 265 G protein-coupled receptor kinase 4
AGC GRK4 GRK4_HUMAN 4YHJB P32298 25 527 578.0 AN2:601 ATPlike Active DFGin 6.038 13.172 BLAminus -128.85, 178.91 61.8, 67.7 -94.52, 28.72 287.39, 101.3 -65.66, -45.87 in-in in 9.016 Saltbr-in 3.179 HRD-in -66.59, -45.54 76.27, -17.2 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.9, 153.12 APE9-dihe-na 125.18, -147.1 APE8-dihe-in -118.5, 134.63 APE8-rot-in 298.66 APE67-dihe-inflip 107.33, -19.99 -54.96, 119.79 APE12-dist-in 11.128 APE11-dist-in 12.752 APE10-dist-in 6.774 APE9-dist-in 3.816 C563S,C578S None None XRAY 2.6 0.2 0.248 B 584 490 0 0 0 0 [[187, 449]] 1.0 4yhj Homo sapiens AGC_GRK4_HUMAN AGC 8.1e-84 286.9 1 260 260 329 330 331 333 335 216 235 239 309 311 310 312 368 356 351 350 349 348 347 346 345 265 G protein-coupled receptor kinase 4
AGC GRK5 GRK5_HUMAN 4TNDA P34947 15 543 590.0 ANP:601 ATPlike Active DFGin 5.282 13.172 BLAminus -119.9, 173.82 59.88, 73.64 -89.53, 7.87 278.21, 112.8 -54.71, -33.69 in-in in 9.193 Saltbr-in 3.053 HRD-in -67.8, -56.87 74.64, -6.61 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.25, 150.21 APE9-dihe-na 143.02, -165.26 APE8-dihe-in -107.11, 142.28 APE8-rot-in 314.69 APE67-dihe-inflip 92.64, -22.22 -59.58, 132.94 APE12-dist-in 10.302 APE11-dist-in 12.056 APE10-dist-in 6.23 APE9-dist-in 4.255 None None None XRAY 1.802 0.174 0.205 A 590 529 0 0 0 0 [[186, 448]] 1.0 4tnd Homo sapiens AGC_GRK5_HUMAN AGC 1.1e-83 286.4 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 5
AGC GRK5 GRK5_HUMAN 9CKRA P34947 25 542 590.0 ATP:603 ATPlike Active DFGin 6.172 12.867 BLAminus -123.04, 159.77 67.48, 80.75 -99.52, 5.04 278.7, 83.61 -52.63, -21.44 in-in in 8.589 Saltbr-in 3.447 HRD-in -94.88, -52.49 68.7, 5.59 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.66, 167.59 APE9-dihe-na 129.66, -152.54 APE8-dihe-in -119.66, 138.17 APE8-rot-in 320.31 APE67-dihe-inflip 80.19, -6.12 -54.38, 134.58 APE12-dist-in 9.872 APE11-dist-in 12.258 APE10-dist-in 6.529 APE9-dist-in 4.181 D311N None None XRAY 2.8 0.239 0.286 A 598 501 0 0 0 0 [[186, 448]] 1.0 9ckr Homo sapiens AGC_GRK5_HUMAN AGC 7.6e-83 283.7 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 5
AGC GRK5 GRK5_HUMAN 9CKSA P34947 25 542 590.0 ATP:603 ATPlike Active DFGin 6.038 13.061 BLAminus -123.04, 167.6 79.98, 56.79 -87.17, 17.84 285.5, 62.72 -70.38, -31.79 in-in in 9.222 Saltbr-in 2.672 HRD-in -92.29, -53.7 68.73, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.24, 151.24 APE9-dihe-na 138.17, -158.29 APE8-dihe-in -117.35, 145.2 APE8-rot-in 310.61 APE67-dihe-inflip 85.98, -22.04 -53.6, 135.84 APE12-dist-in 10.616 APE11-dist-in 12.407 APE10-dist-in 6.563 APE9-dist-in 4.207 D311N None None XRAY 3.08 0.228 0.28 A 598 501 0 0 0 0 [[186, 448]] 1.0 9cks Homo sapiens AGC_GRK5_HUMAN AGC 7.6e-83 283.7 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 5
AGC GRK6 GRK6_HUMAN 2ACXA P43250 14 532 576.0 ANP:577 ATPlike Active DFGin 6.207 13.284 BLAminus -133.82, 164.79 58.79, 76.03 -96.19, 24.41 281.42, 82.4 -59.68, -24.05 in-in in 9.341 Saltbr-in 3.219 HRD-in -78.26, -56.85 77.2, -1.95 in-in-in SNCiii in-in ActLoopNT-in 2.971 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.49, 157.4 APE9-dihe-na 123.02, -168.26 APE8-dihe-in -95.03, 140.31 APE8-rot-in 303.17 APE67-dihe-in -86.56, -0.13 -45.11, -52.69 APE12-dist-in 10.478 APE11-dist-in 11.834 APE10-dist-in 6.083 APE9-dist-in 3.906 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 A 576 495 0 0 0 0 [[186, 448]] 1.0 2acx Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC GRK6 GRK6_HUMAN 2ACXB P43250 14 535 576.0 ANP:577 ATPlike Active DFGin 6.09 13.146 BLAminus -128.37, 163.87 55.35, 87.14 -100.56, 21.26 285.61, 77.77 -55.4, -30.56 in-in in 9.231 Saltbr-in 2.439 HRD-in -77.3, -59.12 75.78, 1.97 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.83, 161.38 APE9-dihe-na 125.99, -167.44 APE8-dihe-in -95.89, 144.8 APE8-rot-in 307.19 APE67-dihe-in -70.72, -14.39 -48.06, -55.51 APE12-dist-in 10.477 APE11-dist-in 11.872 APE10-dist-in 6.167 APE9-dist-in 3.71 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 B 576 492 5 0 0 0 [[186, 448]] 1.0 2acx Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC GRK6 GRK6_HUMAN 3NYOA P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.423 12.986 BLAminus -150.32, 176.66 46.57, 93.99 -112.64, 27.92 269.12, 56.38 -53.19, -36.92 in-in in 8.492 Saltbr-in 3.133 HRD-in -67.42, -53.58 67.41, 17.23 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.58, 145.08 APE9-dihe-na 153.72, -154.4 APE8-dihe-in -119.63, 125.01 APE8-rot-in 309.24 APE67-dihe-inflip 99.19, -30.43 -48.0, 129.76 APE12-dist-in 10.102 APE11-dist-in 11.881 APE10-dist-in 6.152 APE9-dist-in 3.985 None None None XRAY 2.92 0.222 0.253 A 576 553 3 0 0 0 [[186, 448]] 1.0 3nyo Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC GRK6 GRK6_HUMAN 3NYOB P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.469 12.921 BLAminus -147.57, -176.88 49.48, 66.09 -89.42, 43.68 283.74, 78.16 -61.9, -48.01 in-in in 8.429 Saltbr-in 2.859 HRD-in -67.89, -44.49 63.77, 4.77 in-in-in SNCiii in-in ActLoopNT-in 2.959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.44, 138.67 APE9-dihe-na 143.94, 179.93 APE8-dihe-in -100.37, 135.53 APE8-rot-in 311.67 APE67-dihe-inflip 96.9, -39.59 -38.27, 126.0 APE12-dist-in 10.148 APE11-dist-in 11.731 APE10-dist-in 5.96 APE9-dist-in 3.734 None None None XRAY 2.92 0.222 0.253 B 576 553 3 0 0 0 [[186, 448]] 1.0 3nyo Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1 260 260 328 329 330 332 334 215 234 238 308 310 309 311 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
AGC PDPK1 PDPK1_HUMAN 2BIYA O15530 72 359 556.0 ATP:1373 ATPlike Active DFGin 6.619 15.095 BLAminus -141.33, -175.84 82.91, 67.67 -104.99, 1.58 283.05, 104.18 -61.63, -33.06 in-in in 8.673 Saltbr-in 2.575 HRD-in -63.52, -52.73 78.44, -11.09 in-in-in SNCiii in-in ActLoopNT-in 2.82 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.22, 130.12 APE9-dihe-na 106.71, 171.13 APE8-dihe-in -96.94, 126.07 APE8-rot-in 299.07 APE67-dihe-in -62.15, -19.51 -52.23, -44.36 APE12-dist-in 12.868 APE11-dist-in 12.869 APE10-dist-in 7.268 APE9-dist-in 4.745 S241A None None XRAY 1.95 0.186 0.23 A 310 288 0 0 0 0 [[82, 342]] 1.0 2biy Homo sapiens AGC_PDPK1_HUMAN AGC 1.8e-84 288.8 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3HRCA O15530 76 359 556.0 ATP:1373 ATPlike Active DFGin 6.486 14.833 BLAminus -136.91, -178.17 71.81, 74.55 -104.54, 6.98 286.89, 102.51 -65.47, -24.41 in-in in 8.421 Saltbr-in 3.159 HRD-in -77.24, -54.93 76.93, -11.42 in-in-in SNCiii in-in ActLoopNT-in 2.87 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.25, 162.0 APE9-dihe-na 130.63, -171.63 APE8-dihe-in -125.01, 129.68 APE8-rot-in 292.48 APE67-dihe-in -58.92, -25.29 -45.32, -48.7 APE12-dist-in 7.409 APE11-dist-in 10.582 APE10-dist-in 4.926 APE9-dist-in 3.479 Y288G,Q292A SEP241 SEP241 XRAY 1.91 0.182 0.207 A 311 280 4 0 0 4 [[82, 342]] 1.0 3hrc Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 4RRVA O15530 76 359 556.0 ATP:60401 ATPlike Active DFGin 6.548 14.998 BLAminus -136.55, -175.99 74.63, 72.8 -106.52, 5.78 286.61, 100.18 -68.12, -17.88 in-in in 8.52 Saltbr-in 2.956 HRD-in -71.77, -54.29 78.75, -11.73 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.13, 162.83 APE9-dihe-na 132.08, -169.67 APE8-dihe-in -127.24, 132.02 APE8-rot-in 298.33 APE67-dihe-in -59.21, -24.3 -51.83, -46.04 APE12-dist-in 7.281 APE11-dist-in 10.502 APE10-dist-in 4.943 APE9-dist-in 3.569 Y288G,Q292A SEP241 SEP241 XRAY 1.412 0.135 0.163 A 311 284 0 0 0 0 [[82, 342]] 1.0 4rrv Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5ACKA O15530 73 359 556.0 ATP:500 ATPlike Active DFGin 6.615 14.861 BLAminus -135.34, 179.84 72.22, 79.01 -106.01, 4.14 287.93, 97.64 -67.02, -18.73 in-in in 8.418 Saltbr-in 2.583 HRD-in -74.68, -53.67 78.01, -12.73 in-in-in SNCiii in-in ActLoopNT-in 2.906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.4, 162.51 APE9-dihe-na 136.44, -168.07 APE8-dihe-in -132.35, 133.52 APE8-rot-in 296.36 APE67-dihe-in -62.96, -23.95 -54.34, -43.19 APE12-dist-in 7.326 APE11-dist-in 10.522 APE10-dist-in 4.978 APE9-dist-in 3.558 Y288G,Q292A SEP241 SEP241 XRAY 1.24 0.143 0.166 A 311 287 0 0 0 0 [[82, 342]] 1.0 5ack Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPA O15530 75 359 556.0 ATP:500 ATPlike Active DFGin 6.303 14.998 BLAminus -144.92, -168.82 66.06, 77.78 -108.23, 11.17 281.99, 93.22 -63.04, -32.41 in-in in 9.539 Saltbr-in 3.158 HRD-in -77.47, -51.83 79.92, -12.48 in-in-in SNCiii in-in ActLoopNT-in 2.848 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.64, 166.02 APE9-dihe-na 141.61, 177.5 APE8-dihe-in -123.02, 134.29 APE8-rot-in 296.02 APE67-dihe-in -68.65, -16.53 -46.89, -50.92 APE12-dist-in 7.907 APE11-dist-in 10.671 APE10-dist-in 5.166 APE9-dist-in 3.705 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 A 311 276 9 0 0 9 [[82, 342]] 1.0 5lvp Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPB O15530 74 359 556.0 ATP:401 ATPlike Active DFGin 6.328 14.55 BLAminus -137.23, -179.71 80.14, 74.16 -105.47, 15.38 295.0, 84.83 -59.91, -31.47 in-in in 9.274 Saltbr-in 3.302 HRD-in -80.68, -44.41 73.96, -16.23 in-in-in SNCiii in-in ActLoopNT-in 2.744 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.8, 152.43 APE9-dihe-na 134.43, -173.75 APE8-dihe-in -120.09, 128.28 APE8-rot-in 302.93 APE67-dihe-in -67.56, -25.72 -44.99, -47.55 APE12-dist-in 7.872 APE11-dist-in 11.011 APE10-dist-in 5.375 APE9-dist-in 3.787 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 B 311 277 9 0 0 9 [[82, 342]] 1.0 5lvp Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPC O15530 75 359 556.0 ATP:401 ATPlike Active DFGin 6.391 14.608 BLAminus -132.15, -176.81 71.98, 84.02 -116.53, 7.62 291.47, 90.46 -60.24, -24.5 in-in in 9.304 Saltbr-in 3.087 HRD-in -75.92, -52.06 78.45, -5.49 in-in-in SNCiii in-in ActLoopNT-in 2.823 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -113.81, 168.64 APE9-dihe-na 131.92, -176.79 APE8-dihe-in -126.79, 133.21 APE8-rot-in 299.13 APE67-dihe-in -67.64, -15.8 -51.62, -50.49 APE12-dist-in 7.652 APE11-dist-in 10.863 APE10-dist-in 5.123 APE9-dist-in 3.645 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 C 311 276 9 0 0 9 [[82, 342]] 1.0 5lvp Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5LVPD O15530 74 359 556.0 ATP:500 ATPlike Active DFGin 6.334 14.433 BLAminus -146.99, -174.22 74.22, 81.56 -113.84, 4.02 287.97, 93.59 -56.11, -25.73 in-in in 9.304 Saltbr-in 3.252 HRD-in -82.38, -50.18 78.4, -12.51 in-in-in SNCiii in-in ActLoopNT-in 2.836 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.65, 165.17 APE9-dihe-na 129.1, -166.82 APE8-dihe-in -132.84, 129.79 APE8-rot-in 300.06 APE67-dihe-in -65.46, -17.03 -48.9, -48.47 APE12-dist-in 8.228 APE11-dist-in 10.891 APE10-dist-in 5.348 APE9-dist-in 3.646 Y288G,Q292A SEP241 SEP241 XRAY 2.5 0.176 0.226 D 311 277 9 0 0 9 [[82, 342]] 1.0 5lvp Homo sapiens AGC_PDPK1_HUMAN AGC 6.9e-84 286.9 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 4CT2A O15530 75 359 556.0 ATP:500 ATPlike Active DFGin 6.551 14.867 BLAminus -136.23, -174.98 70.54, 70.07 -102.02, 6.41 290.69, 95.78 -63.73, -21.59 in-in in 8.252 Saltbr-in 2.643 HRD-in -73.2, -54.84 77.37, -9.78 in-in-in SNCiii in-in ActLoopNT-in 2.965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.02, 163.59 APE9-dihe-na 137.39, -170.05 APE8-dihe-in -132.12, 131.72 APE8-rot-in 295.26 APE67-dihe-in -63.06, -17.27 -51.84, -45.87 APE12-dist-in 7.163 APE11-dist-in 10.524 APE10-dist-in 4.979 APE9-dist-in 3.527 L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A SEP241 SEP241 XRAY 1.25 0.194 0.226 A 311 280 5 0 0 0 [[82, 342]] 1.0 4ct2 Homo sapiens AGC_PDPK1_HUMAN AGC 9.5e-84 286.4 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 5MRDA O15530 76 359 556.0 ATP:405 ATPlike Active DFGin 6.429 14.7 BLAminus -133.69, -177.11 74.21, 73.9 -105.88, 9.0 289.39, 99.64 -68.32, -19.62 in-in in 8.346 Saltbr-in 2.667 HRD-in -74.32, -53.19 77.26, -10.58 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.86, 160.68 APE9-dihe-na 136.11, -166.87 APE8-dihe-in -131.1, 132.63 APE8-rot-in 296.36 APE67-dihe-in -62.36, -23.28 -53.02, -44.84 APE12-dist-in 7.352 APE11-dist-in 10.498 APE10-dist-in 4.91 APE9-dist-in 3.542 K76S,L113V,I118V,I119N,V124I,T128Q,R131K,T148C SEP241 SEP241 XRAY 1.41 0.142 0.174 A 310 284 0 0 0 0 [[82, 342]] 1.0 5mrd Homo sapiens AGC_PDPK1_HUMAN AGC 1.7e-83 285.6 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PRKACA KAPCA_HUMAN 4WB8A P17612 16 351 351.0 ATP:60401 ATPlike Active DFGin 5.684 14.414 BLAminus -121.45, -177.2 62.67, 77.75 -91.98, 24.58 268.87, 53.09 -58.34, -31.51 in-in in 8.913 Saltbr-in 2.759 HRD-in -95.2, -52.32 70.44, 11.38 in-in-in SNCiii in-in ActLoopNT-in 2.912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.85, 164.58 APE9-dihe-na 131.46, -156.38 APE8-dihe-in -129.55, 139.43 APE8-rot-in 297.11 APE67-dihe-in -60.54, -22.69 -52.03, -49.04 APE12-dist-in 8.098 APE11-dist-in 11.392 APE10-dist-in 5.827 APE9-dist-in 3.498 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.164 0.184 A 337 336 0 0 0 0 [[44, 298]] 1.0 4wb8 Homo sapiens AGC_PRKACA_HUMAN AGC 4e-95 323.8 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB5A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 5.6 14.452 BLAminus -123.05, 176.84 68.94, 80.02 -91.46, 24.86 270.2, 52.92 -60.74, -31.43 in-in in 9.03 Saltbr-in 2.715 HRD-in -92.12, -52.84 69.8, 13.37 in-in-in SNCiii in-in ActLoopNT-in 2.918 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.48, 163.75 APE9-dihe-na 132.31, -149.49 APE8-dihe-in -132.05, 134.14 APE8-rot-in 301.14 APE67-dihe-in -60.1, -21.12 -48.44, -50.23 APE12-dist-in 8.012 APE11-dist-in 11.4 APE10-dist-in 5.799 APE9-dist-in 3.567 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.641 0.165 0.196 A 350 338 0 0 0 0 [[44, 298]] 1.0 4wb5 Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB7A P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.445 14.649 BLAminus -119.06, -174.39 59.4, 77.28 -89.09, 26.42 267.74, 51.48 -60.48, -28.34 in-in in 8.87 Saltbr-in 2.769 HRD-in -93.55, -50.9 68.82, 8.95 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.63, 158.06 APE9-dihe-na 139.02, -156.91 APE8-dihe-in -126.94, 137.23 APE8-rot-in 299.54 APE67-dihe-in -64.26, -23.0 -50.4, -48.13 APE12-dist-in 8.18 APE11-dist-in 11.54 APE10-dist-in 5.955 APE9-dist-in 3.723 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 A 405 336 0 0 0 0 [[44, 298]] 1.0 4wb7 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB7B P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.38 14.712 BLAminus -115.93, -176.79 62.38, 75.33 -88.91, 25.18 264.71, 51.71 -56.9, -30.26 in-in in 8.962 Saltbr-in 2.773 HRD-in -94.01, -50.55 67.24, 10.48 in-in-in SNCiii in-in ActLoopNT-in 2.939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.07, 161.39 APE9-dihe-na 132.31, -156.17 APE8-dihe-in -127.2, 138.18 APE8-rot-in 298.14 APE67-dihe-in -59.62, -23.37 -52.63, -48.78 APE12-dist-in 8.198 APE11-dist-in 11.563 APE10-dist-in 5.97 APE9-dist-in 3.642 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 B 405 336 0 0 0 0 [[44, 298]] 1.0 4wb7 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 6BYRA P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.626 14.616 BLAminus -128.29, 177.03 62.06, 86.64 -97.54, 28.59 271.87, 66.62 -63.2, -33.23 in-in in 8.808 Saltbr-in 3.196 HRD-in -87.43, -52.47 67.28, 5.18 in-in-in SNCiii in-in ActLoopNT-in 3.193 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.51, 153.24 APE9-dihe-na 149.32, -133.8 APE8-dihe-in -139.35, 133.91 APE8-rot-in 312.31 APE67-dihe-in -68.4, -6.95 -52.73, -48.25 APE12-dist-in 8.734 APE11-dist-in 11.076 APE10-dist-in 5.63 APE9-dist-in 3.491 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 A 405 336 0 0 0 0 [[44, 298]] 1.0 6byr Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 6BYRC P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.679 14.34 BLAminus -129.89, 172.29 61.76, 74.25 -79.2, 34.93 281.69, 54.14 -61.8, -27.34 in-in in 8.733 Saltbr-in 2.498 HRD-in -93.13, -49.8 64.55, 7.44 in-in-in SNCiii in-in ActLoopNT-in 3.052 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.29, 161.94 APE9-dihe-na 130.51, -156.26 APE8-dihe-in -112.31, 134.09 APE8-rot-in 302.07 APE67-dihe-in -64.15, -16.52 -52.64, -41.39 APE12-dist-in 8.316 APE11-dist-in 11.106 APE10-dist-in 5.767 APE9-dist-in 3.618 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 C 405 336 0 0 0 0 [[44, 298]] 1.0 6byr Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 9EDCA P17612 14 351 351.0 ATP:60400 ATPlike Active DFGin 5.626 13.772 BLAminus -125.61, -173.52 60.53, 69.6 -81.59, 16.86 273.36, 51.23 -62.38, -30.28 in-in in 9.129 Saltbr-in 3.0 HRD-in -112.54, -46.7 65.17, 1.82 in-in-in SNCiii in-in ActLoopNT-in 3.14 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.87, 159.92 APE9-dihe-na 136.42, -156.18 APE8-dihe-in -101.13, 126.83 APE8-rot-in 299.98 APE67-dihe-in -84.76, -8.6 -60.74, -28.35 APE12-dist-in 7.999 APE11-dist-in 11.111 APE10-dist-in 5.797 APE9-dist-in 3.748 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 EM 4.18 999.0 999.0 A 350 338 0 0 0 0 [[44, 298]] 1.0 9edc Homo sapiens AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB6A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 6.068 14.398 BLAminus -118.38, -169.49 51.77, 82.47 -95.61, 17.78 271.18, 55.73 -42.8, -37.29 in-in in 8.83 Saltbr-in 2.561 HRD-in -94.17, -52.18 74.17, 2.46 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.55, 166.68 APE9-dihe-na 116.18, 128.45 APE8-dihe-in -46.62, 128.74 APE8-rot-in 303.5 APE67-dihe-in -58.01, -23.74 -49.09, -50.89 APE12-dist-in 8.046 APE11-dist-in 11.764 APE10-dist-in 6.243 APE9-dist-in 3.767 L206R SEP11,SEP140,TPO198 SEP11,SEP140,TPO198 XRAY 2.1 0.19 0.237 A 350 338 0 0 0 0 [[44, 298]] 1.0 4wb6 Homo sapiens AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_HUMAN 4WB6B P17612 9 351 351.0 ATP:60401 ATPlike Active DFGin 5.872 14.073 BLAminus -117.82, -168.32 53.27, 78.35 -91.25, 29.34 274.97, 62.46 -60.26, -35.85 in-in in 8.687 Saltbr-in 2.75 HRD-in -101.62, -46.5 64.42, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.38, 164.15 APE9-dihe-na 120.83, 133.18 APE8-dihe-in -48.66, 125.41 APE8-rot-in 298.86 APE67-dihe-in -54.58, -37.6 -53.55, -42.52 APE12-dist-in 8.078 APE11-dist-in 11.617 APE10-dist-in 6.204 APE9-dist-in 3.822 L206R SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.19 0.237 B 350 343 0 0 0 0 [[44, 298]] 1.0 4wb6 Homo sapiens AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKCB KPCB_HUMAN 8SE1A P05771 19 668 671.0 ANP:60706 ATPlike Active DFGin 6.007 12.839 BLAminus -130.5, -169.38 54.07, 70.37 -91.85, 35.76 301.77, 99.49 -89.35, 3.84 in-in in 8.337 Saltbr-in 2.524 HRD-in -91.65, -37.95 43.68, 28.8 in-in-in SNCiii in-in ActLoopNT-in 3.16 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.86, 170.42 APE9-dihe-na 126.28, -151.58 APE8-dihe-in -120.81, 128.88 APE8-rot-in 299.44 APE67-dihe-in -79.06, -41.06 -50.17, -27.42 APE12-dist-in 8.88 APE11-dist-in 12.178 APE10-dist-in 6.66 APE9-dist-in 3.611 None TPO500,TPO642,SEP661 TPO500,TPO642,SEP661 XRAY 3.32 0.202 0.256 A 674 607 0 0 0 0 [[342, 600]] 1.0 8se1 Homo sapiens AGC_PRKCB_HUMAN AGC 1.5e-97 332.1 1 260 260 483 484 485 487 489 371 390 394 463 465 464 466 523 511 506 505 504 503 502 501 500 421 Protein kinase C beta type
AGC PRKCB KPCB_HUMAN 8SE1B P05771 19 668 671.0 ANP:60706 ATPlike Active DFGin 6.093 12.778 BLAminus -130.75, -169.0 53.85, 70.09 -92.15, 34.96 301.62, 99.67 -90.48, 2.45 in-in in 8.312 Saltbr-in 2.216 HRD-in -89.42, -35.84 47.27, 23.7 in-in-in SNCiii in-in ActLoopNT-in 3.284 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.83, 169.92 APE9-dihe-na 126.33, -152.59 APE8-dihe-in -121.43, 128.62 APE8-rot-in 299.3 APE67-dihe-in -78.67, -41.09 -50.34, -26.64 APE12-dist-in 8.722 APE11-dist-in 12.182 APE10-dist-in 6.709 APE9-dist-in 3.767 None TPO500,TPO642,SEP661 TPO500,TPO642,SEP661 XRAY 3.32 0.202 0.256 B 674 631 0 0 0 0 [[342, 600]] 1.0 8se1 Homo sapiens AGC_PRKCB_HUMAN AGC 1.5e-97 332.1 1 260 260 483 484 485 487 489 371 390 394 463 465 464 466 523 511 506 505 504 503 502 501 500 421 Protein kinase C beta type
AGC PRKCB KPCB_HUMAN 8SE2B P05771 30 671 671.0 ANP:701 ATPlike Active DFGin 5.706 12.737 BLAminus -122.79, -175.57 50.54, 85.22 -103.07, 33.77 300.25, 95.58 -78.87, -5.25 in-in in 8.251 Saltbr-in 2.675 HRD-in -90.05, -48.77 75.62, -5.68 in-in-in SNCiii in-in ActLoopNT-in 3.126 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.22, 161.28 APE9-dihe-na 125.49, -179.08 APE8-dihe-in -100.09, 129.99 APE8-rot-in 297.02 APE67-dihe-in -66.56, -21.71 -49.98, -38.79 APE12-dist-in 8.634 APE11-dist-in 11.712 APE10-dist-in 6.223 APE9-dist-in 3.606 None TPO500,TPO642,SEP661 TPO500,TPO642,SEP661 XRAY 2.95 0.196 0.252 B 672 589 0 0 0 0 [[342, 600]] 1.0 8se2 Homo sapiens AGC_PRKCB_HUMAN AGC 1.5e-97 332.1 1 260 260 483 484 485 487 489 371 390 394 463 465 464 466 523 511 506 505 504 503 502 501 500 421 Protein kinase C beta type
AGC PRKCI KPCI_HUMAN 5LIHA P41743 248 588 596.0 ADP:60601 ATPlike Active DFGin 5.403 11.863 BLAminus -129.58, 178.7 63.64, 84.98 -106.19, 67.5 320.36, 105.86 -96.86, -30.05 in-in in 9.178 Saltbr-in 3.031 HRD-in -49.42, -59.61 61.3, 24.72 in-in-in SNCiii in-in ActLoopNT-in 3.109 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.76, 169.43 APE9-dihe-na 122.35, -170.42 APE8-dihe-in -91.96, 136.55 APE8-rot-in 289.3 APE67-dihe-in -72.22, -23.04 -49.75, -40.52 APE12-dist-in 7.983 APE11-dist-in 10.986 APE10-dist-in 5.421 APE9-dist-in 3.56 None TPO412,TPO564 TPO412,TPO564 XRAY 3.25 0.258 0.284 A 349 326 15 0 0 0 [[254, 522]] 1.0 5lih Homo sapiens AGC_PRKCI_HUMAN AGC 1.1e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKCI KPCI_HUMAN 5LIHB P41743 249 588 596.0 ADP:60601 ATPlike Active DFGin 5.31 11.876 BLAminus -129.18, 178.42 63.46, 84.62 -106.43, 67.35 320.63, 105.98 -96.29, -29.69 in-in in 8.72 Saltbr-in 2.545 HRD-in -49.62, -59.64 61.27, 24.64 in-in-in SNCiii in-in ActLoopNT-in 3.141 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.47, 168.99 APE9-dihe-na 122.16, -170.23 APE8-dihe-in -91.66, 136.86 APE8-rot-in 289.24 APE67-dihe-in -72.3, -22.91 -49.4, -40.32 APE12-dist-in 8.329 APE11-dist-in 11.256 APE10-dist-in 5.693 APE9-dist-in 3.742 None TPO412,TPO564 TPO412,TPO564 XRAY 3.25 0.258 0.284 B 349 320 20 0 0 0 [[254, 522]] 1.0 5lih Homo sapiens AGC_PRKCI_HUMAN AGC 1.1e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKCI KPCI_HUMAN 5LI9A P41743 248 589 596.0 ACP:60601 ATPlike Active DFGin 5.635 12.633 BLAminus -139.17, 172.4 72.31, 78.11 -98.86, 1.23 304.03, 143.26 -64.9, -22.84 in-in in 8.361 Saltbr-in 2.614 HRD-in -73.79, -55.22 70.11, -1.11 in-in-in SNCiii in-in ActLoopNT-in 2.81 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.64, 169.55 APE9-dihe-na 127.72, -178.47 APE8-dihe-in -93.25, 127.56 APE8-rot-in 298.81 APE67-dihe-in -60.64, -20.02 -47.28, -45.36 APE12-dist-in 8.812 APE11-dist-in 11.949 APE10-dist-in 6.432 APE9-dist-in 3.836 None TPO412,TPO564 TPO412,TPO564 XRAY 1.79 0.19 0.231 A 350 330 12 0 0 0 [[254, 522]] 1.0 5li9 Homo sapiens AGC_PRKCI_HUMAN AGC 1.2e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKCI KPCI_HUMAN 5LI1A P41743 248 589 596.0 ANP:60601 ATPlike Active DFGin 5.079 11.961 BLAminus -129.24, 176.98 73.22, 90.17 -103.83, 11.43 308.18, 130.49 -69.42, -18.98 in-in in 8.413 Saltbr-in 2.816 HRD-in -77.28, -52.44 73.77, 3.75 in-in-in SNCiii in-in ActLoopNT-in 2.975 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.65, 168.01 APE9-dihe-na 127.57, -168.6 APE8-dihe-in -111.48, 126.0 APE8-rot-in 296.01 APE67-dihe-in -54.62, -31.15 -46.95, -45.66 APE12-dist-in 8.752 APE11-dist-in 11.822 APE10-dist-in 6.31 APE9-dist-in 3.517 None TPO412,SEP484,TPO564 TPO412,SEP484,TPO564 XRAY 2.0 0.154 0.217 A 354 332 10 0 0 0 [[254, 522]] 1.0 5li1 Homo sapiens AGC_PRKCI_HUMAN AGC 1.2e-95 325.5 1 260 260 395 396 397 399 401 283 302 306 375 377 376 378 435 423 418 417 416 415 414 413 412 333 Protein kinase C iota type
AGC PRKG1 KGP1_HUMAN 6BG2A Q13976 336 671 671.0 ANP:700 ATPlike Active DFGin 5.811 14.714 BLAminus -124.15, 169.14 66.07, 88.5 -100.57, 30.98 280.35, 66.41 -65.35, -25.12 in-in in 9.522 Saltbr-in 2.883 HRD-in -85.83, -52.95 73.29, 9.38 in-in-in SNCiii in-in ActLoopNT-in 2.851 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.93, 165.57 APE9-dihe-na 117.74, 172.78 APE8-dihe-in -83.6, 129.51 APE8-rot-in 307.46 APE67-dihe-in -66.9, -19.23 -49.63, -41.3 APE12-dist-in 8.235 APE11-dist-in 11.512 APE10-dist-in 6.041 APE9-dist-in 4.269 None TPO517 TPO517 XRAY 1.83 0.188 0.215 A 347 336 0 0 0 0 [[360, 619]] 1.0 6bg2 Homo sapiens AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 6BG2B Q13976 346 671 671.0 ANP:700 ATPlike Active DFGin 6.001 13.81 BLAminus -122.67, 175.58 65.94, 84.43 -99.77, 30.78 285.96, 70.42 -64.93, -24.07 in-in in 8.944 Saltbr-in 2.743 HRD-in -86.95, -52.47 73.99, 7.96 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.61, 163.67 APE9-dihe-na 118.96, 172.39 APE8-dihe-in -86.94, 131.94 APE8-rot-in 306.51 APE67-dihe-in -68.79, -20.88 -48.58, -41.68 APE12-dist-in 7.826 APE11-dist-in 11.215 APE10-dist-in 5.769 APE9-dist-in 4.008 None TPO517 TPO517 XRAY 1.83 0.188 0.215 B 347 326 0 0 0 0 [[360, 619]] 1.0 6bg2 Homo sapiens AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 6BG2C Q13976 337 671 671.0 ANP:700 ATPlike Active DFGin 5.746 14.057 BLAminus -122.99, 175.03 65.66, 84.22 -99.61, 30.7 281.62, 66.26 -64.81, -23.57 in-in in 8.742 Saltbr-in 2.723 HRD-in -85.99, -53.51 74.31, 7.4 in-in-in SNCiii in-in ActLoopNT-in 2.951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.66, 165.85 APE9-dihe-na 118.46, 173.18 APE8-dihe-in -87.41, 130.75 APE8-rot-in 306.63 APE67-dihe-in -67.71, -19.03 -48.39, -42.55 APE12-dist-in 7.972 APE11-dist-in 11.385 APE10-dist-in 5.857 APE9-dist-in 3.861 None TPO517 TPO517 XRAY 1.83 0.188 0.215 C 347 335 0 0 0 0 [[360, 619]] 1.0 6bg2 Homo sapiens AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 6BG2D Q13976 344 671 671.0 ANP:700 ATPlike Active DFGin 5.71 14.012 BLAminus -124.49, 174.79 65.67, 84.87 -99.37, 30.45 283.38, 66.11 -64.13, -22.3 in-in in 8.754 Saltbr-in 2.644 HRD-in -85.68, -52.69 74.16, 8.99 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.92, 166.42 APE9-dihe-na 119.53, 169.97 APE8-dihe-in -84.81, 130.45 APE8-rot-in 305.19 APE67-dihe-in -66.29, -19.88 -48.13, -43.31 APE12-dist-in 7.988 APE11-dist-in 11.327 APE10-dist-in 5.784 APE9-dist-in 3.81 None TPO517 TPO517 XRAY 1.83 0.188 0.215 D 347 328 0 0 0 0 [[360, 619]] 1.0 6bg2 Homo sapiens AGC_PRKG1_HUMAN AGC 2.6e-84 288.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 7LV3A Q13976 57 671 671.0 ANP:60803 ATPlike Active DFGin 5.851 14.036 BLAminus -116.97, 177.04 63.26, 88.72 -106.87, 28.72 283.22, 63.7 -62.95, -24.33 in-in in 8.624 Saltbr-in 2.891 HRD-in -87.82, -54.22 74.26, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.911 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.28, 149.98 APE9-dihe-na 157.95, -145.59 APE8-dihe-in -124.73, 128.61 APE8-rot-in 299.79 APE67-dihe-in -58.37, -20.06 -47.89, -51.97 APE12-dist-in 7.972 APE11-dist-in 11.057 APE10-dist-in 5.469 APE9-dist-in 3.811 None TPO517 TPO517 XRAY 2.41 0.201 0.238 A 617 600 0 0 0 0 [[360, 619]] 1.0 7lv3 Homo sapiens AGC_PRKG1_HUMAN AGC 1.3e-83 286.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC PRKG1 KGP1_HUMAN 7LV3B Q13976 58 671 671.0 ANP:60803 ATPlike Active DFGin 5.634 13.962 BLAminus -116.52, 178.28 63.3, 90.17 -108.68, 29.08 283.48, 65.02 -62.88, -23.93 in-in in 8.883 Saltbr-in 2.824 HRD-in -86.48, -52.9 74.97, 7.4 in-in-in SNCiii in-in ActLoopNT-in 2.959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.28, 149.21 APE9-dihe-na 157.62, -145.94 APE8-dihe-in -123.75, 129.22 APE8-rot-in 300.73 APE67-dihe-in -59.05, -19.44 -46.41, -52.49 APE12-dist-in 8.134 APE11-dist-in 11.198 APE10-dist-in 5.604 APE9-dist-in 3.787 None TPO517 TPO517 XRAY 2.41 0.201 0.238 B 617 593 0 0 0 0 [[360, 619]] 1.0 7lv3 Homo sapiens AGC_PRKG1_HUMAN AGC 1.3e-83 286.3 1 260 260 501 502 503 505 507 390 409 413 481 483 482 484 540 528 523 522 521 520 519 518 517 439 cGMP-dependent protein kinase 1
AGC ROCK1 ROCK1_HUMAN 2V55A Q13464 6 404 1354.0 ANP:1480 ATPlike Active DFGin 5.88 13.604 BLAminus -137.29, -177.31 60.22, 109.9 -132.74, 24.25 290.89, 71.12 -53.92, -52.21 in-in in 9.076 Saltbr-in 2.708 HRD-in -79.75, -71.28 93.49, -31.37 in-in-in SNCiii in-in ActLoopNT-in 3.281 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.46, 139.75 APE9-dihe-na 103.51, 160.5 APE8-dihe-in -55.22, 144.8 APE8-rot-in 285.63 APE67-dihe-in -74.86, -38.79 -80.34, -13.24 APE12-dist-in 10.324 APE11-dist-in 11.278 APE10-dist-in 5.647 APE9-dist-in 4.131 None None None XRAY 3.705 0.238 0.269 A 406 393 0 0 0 0 [[76, 338]] 1.0 2v55 Homo sapiens AGC_ROCK1_HUMAN AGC 3.3e-94 320.8 1 260 260 215 216 217 219 221 105 124 128 195 197 196 198 260 244 239 238 237 236 235 234 233 154 Rho-associated protein kinase 1
AGC ROCK1 ROCK1_HUMAN 2V55C Q13464 6 404 1354.0 ANP:1480 ATPlike Active DFGin 5.884 13.608 BLAminus -137.56, -177.44 62.15, 108.48 -130.26, 22.71 291.3, 72.92 -54.95, -50.69 in-in in 9.111 Saltbr-in 2.706 HRD-in -78.29, -71.79 95.11, -31.46 in-in-in SNCiii in-in ActLoopNT-in 3.247 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.41, 139.12 APE9-dihe-na 103.28, 159.31 APE8-dihe-in -53.48, 142.5 APE8-rot-in 287.35 APE67-dihe-in -76.24, -37.92 -78.8, -11.99 APE12-dist-in 10.28 APE11-dist-in 11.269 APE10-dist-in 5.623 APE9-dist-in 4.097 None None None XRAY 3.705 0.238 0.269 C 406 396 0 0 0 0 [[76, 338]] 1.0 2v55 Homo sapiens AGC_ROCK1_HUMAN AGC 3.3e-94 320.8 1 260 260 215 216 217 219 221 105 124 128 195 197 196 198 260 244 239 238 237 236 235 234 233 154 Rho-associated protein kinase 1
CAMK AURKA AURKA_HUMAN 1OL5A O14965 123 388 403.0 ADP:1388 ATPlike Active DFGin 5.578 15.096 BLAminus -139.2, -172.08 52.22, 80.16 -90.83, 24.66 282.61, 72.55 -49.87, -44.18 in-in in 9.451 Saltbr-in 2.912 HRD-in -63.28, -60.88 73.6, 1.59 in-in-in SNCiii in-in ActLoopNT-in 2.928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.42, 162.5 APE9-dihe-na 119.45, -153.19 APE8-dihe-in -110.77, 140.24 APE8-rot-in 313.06 APE67-dihe-in -62.23, -14.3 -43.16, -62.5 APE12-dist-in 8.174 APE11-dist-in 10.957 APE10-dist-in 5.274 APE9-dist-in 3.683 None TPO287,TPO288 TPO287,TPO288 XRAY 2.5 0.194 0.252 A 282 266 0 0 0 0 [[133, 383]] 1.0 1ol5 Homo sapiens CAMK_AURKA_HUMAN CAMK 7.4e-80 273.9 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK AURKA AURKA_HUMAN 6VPGA O14965 7 389 403.0 ANP:60401 ATPlike Active DFGin 5.318 15.07 BLAminus -133.54, 176.05 56.91, 81.54 -90.61, 23.9 286.39, 75.22 -62.73, -9.76 in-in in 9.884 Saltbr-in 2.954 HRD-in -72.51, -51.0 67.55, 11.3 in-in-in SNCiii in-in ActLoopNT-in 3.043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.96, 159.16 APE9-dihe-na 122.67, -152.53 APE8-dihe-in -117.94, 146.39 APE8-rot-in 309.68 APE67-dihe-in -61.83, -12.97 -52.19, -62.88 APE12-dist-in 8.517 APE11-dist-in 11.427 APE10-dist-in 5.724 APE9-dist-in 3.833 None TPO287,TPO288 TPO287,TPO288 XRAY 2.64 0.204 0.245 A 292 267 0 0 0 0 [[133, 383]] 1.0 6vpg Homo sapiens CAMK_AURKA_HUMAN CAMK 8.4e-80 273.7 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK AURKA AURKA_HUMAN 5LXMA O14965 126 392 403.0 ADP:60501 ATPlike Active DFGin 5.391 14.976 BLAminus -135.45, -179.78 54.7, 80.97 -90.8, 30.12 283.16, 71.51 -72.4, -3.16 in-in in 9.247 Saltbr-in 2.724 HRD-in -74.23, -48.55 66.99, 5.01 in-in-in SNCiii in-in ActLoopNT-in 3.114 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.91, 137.37 APE9-dihe-na 128.62, -150.21 APE8-dihe-in -129.87, 142.81 APE8-rot-in 303.47 APE67-dihe-in -69.71, -10.62 -37.99, -61.07 APE12-dist-in 8.257 APE11-dist-in 10.692 APE10-dist-in 5.213 APE9-dist-in 3.298 C290A,C393A TPO288 TPO288 XRAY 2.08 0.202 0.243 A 283 267 0 0 0 0 [[133, 383]] 1.0 5lxm Homo sapiens CAMK_AURKA_HUMAN CAMK 9.2e-79 270.3 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK AURKA AURKA_HUMAN 5G1XA O14965 126 389 403.0 ADP:1390 ATPlike Active DFGin 5.343 15.03 BLAminus -132.86, -170.57 52.68, 76.5 -90.96, 13.96 279.12, 78.43 -59.51, -20.51 in-in in 9.278 Saltbr-in 2.828 HRD-in -82.61, -50.12 70.7, 5.33 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.42, -179.26 APE9-dihe-na 65.74, -155.89 APE8-dihe-in -128.23, 121.78 APE8-rot-in 304.75 APE67-dihe-in -61.27, -19.7 -46.07, -47.67 APE12-dist-in 8.247 APE11-dist-in 10.799 APE10-dist-in 5.53 APE9-dist-in 3.699 C290A,C393A TPO288 TPO288 XRAY 1.72 0.177 0.195 A 285 264 0 0 0 0 [[133, 383]] 1.0 5g1x Homo sapiens CAMK_AURKA_HUMAN CAMK 9.4e-79 270.3 1 256 256 273 274 275 277 279 162 181 185 253 255 254 256 311 299 294 293 292 291 290 289 288 211 Aurora kinase A
CAMK CAMK2A KCC2A_HUMAN 7UJSA Q9UQM7 7 274 478.0 ADP:301 ATPlike Active DFGin 6.209 15.164 BLAminus -142.86, -173.92 52.2, 80.06 -100.62, 24.47 291.74, 81.6 -63.11, -26.23 in-in in 9.512 Saltbr-in 3.444 HRD-in -76.47, -52.69 80.52, -7.0 in-in-in SNCiii in-in ActLoopNT-in 2.952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.88, 140.41 APE9-dihe-na 133.49, -148.09 APE8-dihe-in -128.43, 117.33 APE8-rot-in 305.05 APE67-dihe-in -59.07, -26.67 -36.29, -54.08 APE12-dist-in 10.197 APE11-dist-in 11.505 APE10-dist-in 5.779 APE9-dist-in 3.683 Q223K None None XRAY 2.75 0.201 0.262 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujs Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UIRA Q9UQM7 7 274 478.0 ATP:302 ATPlike Active DFGin 6.045 15.107 BLAminus -137.0, 179.68 44.28, 101.28 -106.42, 24.78 295.79, 81.95 -53.14, -27.06 in-in in 9.85 Saltbr-in 3.466 HRD-in -74.22, -43.69 67.52, 3.92 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.48, 156.41 APE9-dihe-na 131.95, -156.1 APE8-dihe-in -122.09, 129.91 APE8-rot-in 298.28 APE67-dihe-in -55.12, -36.11 -51.43, -40.3 APE12-dist-in 10.333 APE11-dist-in 11.793 APE10-dist-in 6.056 APE9-dist-in 3.425 D135N,Q223K None None XRAY 3.1 0.234 0.274 A 268 268 0 0 0 0 [[13, 271]] 1.0 7uir Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UIRB Q9UQM7 7 273 478.0 ATP:301 ATPlike Active DFGin 6.093 14.463 BLAminus -136.84, -179.4 43.86, 99.82 -105.8, 24.57 296.99, 81.24 -56.04, -26.17 in-in in 9.403 Saltbr-in 3.027 HRD-in -74.93, -42.65 67.84, 3.24 in-in-in SNCiii in-in ActLoopNT-in 2.915 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.86, 157.92 APE9-dihe-na 132.59, -155.55 APE8-dihe-in -122.09, 129.05 APE8-rot-in 298.73 APE67-dihe-in -54.7, -35.97 -51.63, -40.47 APE12-dist-in 10.303 APE11-dist-in 11.733 APE10-dist-in 5.989 APE9-dist-in 3.504 D135N,Q223K None None XRAY 3.1 0.234 0.274 B 268 261 6 0 0 0 [[13, 271]] 1.0 7uir Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UJPA Q9UQM7 7 274 478.0 ADP:301 ATPlike Active DFGin 6.775 14.64 BLAminus -129.88, 174.11 65.35, 73.67 -96.28, 29.41 284.7, 81.79 -65.3, -26.47 in-in in 8.527 Saltbr-in 2.903 HRD-in -76.38, -51.72 77.74, -11.0 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.94, 142.69 APE9-dihe-na 139.08, -169.53 APE8-dihe-in -115.65, 123.25 APE8-rot-in 308.77 APE67-dihe-in -69.44, -15.11 -33.38, -56.34 APE12-dist-in 10.469 APE11-dist-in 11.397 APE10-dist-in 5.657 APE9-dist-in 3.521 D135N,Q223K None None XRAY 2.56 0.234 0.281 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujp Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_HUMAN 7UJPB Q9UQM7 7 273 478.0 ATP:301 ATPlike Active DFGin 6.942 14.313 BLAminus -133.64, 174.92 62.39, 75.15 -97.38, 27.07 283.14, 81.65 -64.42, -25.12 in-in in 8.558 Saltbr-in 2.783 HRD-in -76.01, -51.46 77.74, -9.31 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.94, 139.06 APE9-dihe-na 146.74, -166.31 APE8-dihe-in -115.05, 124.1 APE8-rot-in 308.42 APE67-dihe-in -69.31, -14.12 -35.51, -54.36 APE12-dist-in 10.25 APE11-dist-in 11.592 APE10-dist-in 5.843 APE9-dist-in 3.572 D135N,Q223K None None XRAY 2.56 0.234 0.281 B 268 267 0 0 0 0 [[13, 271]] 1.0 7ujp Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CHEK1 CHK1_HUMAN 7AKMA O14757 2 271 476.0 AGS:401 ATPlike Active DFGin 6.775 14.143 BLAminus -128.66, 150.55 71.15, 96.3 -103.32, 28.49 292.74, 82.8 -70.74, -21.81 in-in in 9.111 Saltbr-in 2.706 HRD-in -78.28, -45.32 76.75, -0.14 in-in-in SNCiii in-in ActLoopNT-in 3.011 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.43, 171.3 APE9-dihe-na 110.38, -147.97 APE8-dihe-in -135.73, 125.59 APE8-rot-in 300.71 APE67-dihe-in -62.97, -17.75 -56.42, -42.48 APE12-dist-in 9.309 APE11-dist-in 11.674 APE10-dist-in 6.171 APE9-dist-in 3.407 D10R None None XRAY 1.93 0.199 0.242 A 298 270 0 0 0 0 [[9, 265]] 1.0 7akm Homo sapiens CAMK_CHEK1_HUMAN CAMK 3.4e-71 245.5 2 256 255 147 148 149 151 153 38 55 59 127 129 128 130 190 177 172 171 170 169 168 167 166 85 Serine/threonine-protein kinase Chk1
CAMK DAPK1 DAPK1_HUMAN 2W4KA P53355 2 302 1430.0 ADP:1303 ATPlike Active DFGin 6.672 14.178 BLAminus -119.76, -176.11 66.35, 79.87 -97.37, 22.41 282.66, 74.96 -63.58, -22.08 in-in in 9.11 Saltbr-in 2.829 HRD-in -72.34, -46.15 68.63, 4.94 in-in-in SNCiii in-in ActLoopNT-in 2.866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.51, 175.21 APE9-dihe-na 86.37, -178.83 APE8-dihe-in -92.32, 120.41 APE8-rot-in 301.2 APE67-dihe-in -65.94, -16.49 -43.92, -47.7 APE12-dist-in 9.204 APE11-dist-in 12.288 APE10-dist-in 6.82 APE9-dist-in 5.132 None None None XRAY 1.9 0.195 0.228 A 302 301 0 0 0 0 [[13, 275]] 1.0 2w4k Homo sapiens CAMK_DAPK1_HUMAN CAMK 6.8e-95 323.2 1 256 256 160 161 162 164 166 42 64 68 136 138 137 139 199 187 182 181 180 179 178 177 176 94 Death-associated protein kinase 1
CAMK DAPK1 DAPK1_HUMAN 2XUUA P53355 2 302 1430.0 ADP:1303 ATPlike Active DFGin 6.814 14.3 BLAminus -117.01, 179.93 67.97, 81.82 -97.7, 27.63 286.42, 73.81 -75.99, -13.96 in-in in 9.047 Saltbr-in 2.623 HRD-in -76.48, -45.49 71.86, 3.84 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.39, 167.91 APE9-dihe-na 89.82, 178.63 APE8-dihe-in -101.18, 124.0 APE8-rot-in 296.23 APE67-dihe-in -60.21, -22.55 -44.54, -47.64 APE12-dist-in 8.87 APE11-dist-in 11.727 APE10-dist-in 6.406 APE9-dist-in 5.145 E182A None None XRAY 1.8 0.179 0.226 A 334 301 0 0 0 0 [[13, 275]] 1.0 2xuu Homo sapiens CAMK_DAPK1_HUMAN CAMK 1.4e-94 322.3 1 256 256 160 161 162 164 166 42 64 68 136 138 137 139 199 187 182 181 180 179 178 177 176 94 Death-associated protein kinase 1
CAMK DCLK1 DCLK1_HUMAN 5JZJA O15075 374 648 740.0 AN2:703 ATPlike Active DFGin 6.559 14.457 BLAminus -124.73, -164.54 49.76, 81.39 -91.62, 27.77 280.9, 72.89 -62.64, -30.24 in-in in 9.264 Saltbr-in 2.961 HRD-in -80.29, -46.18 67.47, 2.65 in-in-in SNCiii in-in ActLoopNT-in 2.862 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.12, 159.65 APE9-dihe-na 123.02, -170.92 APE8-dihe-in -106.5, 129.13 APE8-rot-in 307.92 APE67-dihe-in -61.41, -36.29 -48.5, -40.56 APE12-dist-in 8.952 APE11-dist-in 12.325 APE10-dist-in 6.742 APE9-dist-in 4.306 None None None XRAY 1.71 0.178 0.208 A 297 271 4 0 0 0 [[390, 647]] 1.0 5jzj Homo sapiens CAMK_DCLK1_HUMAN CAMK 7.6e-90 306.6 1 256 256 532 533 534 536 538 419 436 440 508 510 509 511 569 557 552 551 550 549 548 547 546 466 Serine/threonine-protein kinase DCLK1
CAMK DCLK1 DCLK1_HUMAN 5JZJB O15075 382 648 740.0 AN2:902 ATPlike Active DFGin 6.403 14.423 BLAminus -126.14, -167.19 53.32, 81.81 -94.99, 26.92 281.83, 75.21 -56.86, -35.14 in-in in 8.806 Saltbr-in 2.638 HRD-in -80.6, -45.11 67.98, 3.84 in-in-in SNCiii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.06, 162.17 APE9-dihe-na 120.91, -173.72 APE8-dihe-in -109.44, 126.03 APE8-rot-in 300.86 APE67-dihe-in -59.98, -31.53 -43.43, -44.7 APE12-dist-in 9.044 APE11-dist-in 12.358 APE10-dist-in 6.832 APE9-dist-in 4.274 None None None XRAY 1.71 0.178 0.208 B 297 261 6 0 0 0 [[390, 647]] 1.0 5jzj Homo sapiens CAMK_DCLK1_HUMAN CAMK 7.6e-90 306.6 1 256 256 532 533 534 536 538 419 436 440 508 510 509 511 569 557 552 551 550 549 548 547 546 466 Serine/threonine-protein kinase DCLK1
CAMK PASK PASK_HUMAN 3DLSA Q96RG2 982 1266 1323.0 ADP:1 ATPlike Active DFGin 6.001 14.204 BLAminus -129.0, 178.94 63.52, 79.16 -100.96, 27.03 282.44, 72.76 -70.92, -15.42 in-in in 8.655 Saltbr-in 2.605 HRD-na-E -71.55, -40.2 72.7, 1.22 in-in-in SNCiii in-in ActLoopNT-in 2.993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -115.6, 5.88 APE9-dihe-na -96.65, -154.85 APE8-dihe-in -98.92, 122.93 APE8-rot-in 302.12 APE67-dihe-in -72.66, -14.95 -65.45, -19.89 APE12-dist-in 10.203 APE11-dist-in 10.574 APE10-dist-in 5.061 APE9-dist-in 3.451 None None None XRAY 2.3 0.244 0.297 A 335 285 0 0 0 0 [[999, 1251]] 1.0 3dls Homo sapiens CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSB Q96RG2 982 1267 1323.0 ADP:2 ATPlike Active DFGin 6.1 14.087 BLAminus -126.55, 179.43 61.31, 80.64 -98.16, 22.24 284.4, 71.69 -72.83, -6.95 in-in in 8.346 Saltbr-in 2.677 HRD-na-E -67.25, -43.38 72.94, 0.56 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.86, 22.09 APE9-dihe-na -121.63, -155.86 APE8-dihe-in -97.56, 124.97 APE8-rot-in 306.83 APE67-dihe-in -68.7, -17.81 -61.84, -27.67 APE12-dist-in 10.243 APE11-dist-in 10.688 APE10-dist-in 5.149 APE9-dist-in 3.521 None None None XRAY 2.3 0.244 0.297 B 335 280 6 0 0 0 [[999, 1251]] 1.0 3dls Homo sapiens CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSC Q96RG2 982 1267 1323.0 ADP:3 ATPlike Active DFGin 6.549 14.136 BLAminus -121.24, -178.98 61.8, 81.93 -100.03, 24.34 279.06, 77.86 -70.4, -24.84 in-in in 8.286 Saltbr-in 2.707 HRD-na-E -75.53, -39.96 73.3, -0.15 in-in-in SNCiii in-in ActLoopNT-in 2.808 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -109.16, 23.96 APE9-dihe-na -111.98, -161.37 APE8-dihe-in -95.46, 124.23 APE8-rot-in 302.16 APE67-dihe-in -72.29, -18.02 -57.94, -30.36 APE12-dist-in 9.98 APE11-dist-in 10.437 APE10-dist-in 4.962 APE9-dist-in 3.466 None None None XRAY 2.3 0.244 0.297 C 335 281 5 0 0 0 [[999, 1251]] 1.0 3dls Homo sapiens CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSD Q96RG2 982 1266 1323.0 ADP:4 ATPlike Active DFGin 5.989 14.037 BLAminus -119.78, -174.43 57.15, 82.44 -96.61, 20.08 283.36, 68.59 -63.18, -13.75 in-in in 8.596 Saltbr-in 2.674 HRD-na-E -66.59, -43.13 75.45, -3.58 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.17, 8.76 APE9-dihe-na -100.36, -154.44 APE8-dihe-in -94.34, 129.8 APE8-rot-in 309.84 APE67-dihe-in -63.24, -17.05 -59.73, -34.41 APE12-dist-in 10.579 APE11-dist-in 10.601 APE10-dist-in 5.212 APE9-dist-in 3.318 None None None XRAY 2.3 0.244 0.297 D 335 284 1 0 0 0 [[999, 1251]] 1.0 3dls Homo sapiens CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSE Q96RG2 982 1267 1323.0 ADP:5 ATPlike Active DFGin 6.351 14.113 BLAminus -115.03, 172.38 61.43, 82.92 -98.38, 26.76 287.19, 66.36 -61.94, -22.57 in-in in 8.272 Saltbr-in 3.015 HRD-na-E -64.64, -41.08 75.56, -14.47 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.8, 6.63 APE9-dihe-na -93.38, -160.98 APE8-dihe-in -92.63, 131.98 APE8-rot-in 304.09 APE67-dihe-in -71.09, -14.17 -58.49, -32.88 APE12-dist-in 10.767 APE11-dist-in 10.575 APE10-dist-in 5.072 APE9-dist-in 3.423 None None None XRAY 2.3 0.244 0.297 E 335 282 4 0 0 0 [[999, 1251]] 1.0 3dls Homo sapiens CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PASK PASK_HUMAN 3DLSF Q96RG2 982 1266 1323.0 ADP:6 ATPlike Active DFGin 6.208 14.428 BLAminus -120.86, -179.45 54.8, 74.61 -87.61, 27.75 280.29, 66.66 -72.72, -14.22 in-in in 8.492 Saltbr-in 2.879 HRD-na-E -64.59, -48.9 86.1, -8.79 in-in-in SNCiii in-in ActLoopNT-in 2.704 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.3, 4.74 APE9-dihe-na -89.15, -152.34 APE8-dihe-in -104.88, 132.7 APE8-rot-in 302.97 APE67-dihe-in -72.03, -17.52 -62.59, -27.45 APE12-dist-in 10.486 APE11-dist-in 10.547 APE10-dist-in 5.101 APE9-dist-in 3.284 None None None XRAY 2.3 0.244 0.297 F 335 281 4 0 0 0 [[999, 1251]] 1.0 3dls Homo sapiens CAMK_PASK_HUMAN CAMK 2.7e-67 232.8 1 256 256 1145 1146 1147 1149 1151 1028 1052 1056 1125 1127 1126 1128 1185 1172 1167 1166 1165 1164 1163 1162 1161 1082 PAS domain-containing serine/threonine-protein kinase
CAMK PIM1 PIM1_HUMAN 1YXTA P11309 33 306 313.0 ANP:322 ATPlike Active DFGin 6.029 14.245 BLAminus -131.81, 176.98 66.39, 83.69 -99.64, 19.64 287.53, 80.25 -65.72, -15.35 in-in in 8.309 Saltbr-in 2.894 HRD-na-A -67.95, -50.18 66.45, 4.68 in-in-in SNCiii in-in ActLoopNT-in 2.809 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.69, 12.99 APE9-dihe-na -80.03, -158.46 APE8-dihe-in -83.46, 121.7 APE8-rot-in 308.53 APE67-dihe-in -70.36, -3.81 -49.69, -52.76 APE12-dist-in 9.729 APE11-dist-in 8.665 APE10-dist-in 5.279 APE9-dist-in 3.805 None None None XRAY 2.0 0.183 0.216 A 293 274 0 0 0 0 [[38, 290]] 1.0 1yxt Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUA P11309 33 305 313.0 AMP:550 ATPlike Active DFGin 6.045 14.58 BLAminus -128.48, 170.01 62.85, 77.77 -90.35, 20.24 287.6, 77.99 -74.7, 1.63 in-in in 8.513 Saltbr-in 2.486 HRD-na-A -60.24, -50.74 67.33, 4.52 in-in-in SNCiii in-in ActLoopNT-in 2.893 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.18, 25.46 APE9-dihe-na -90.91, -158.18 APE8-dihe-in -86.5, 120.86 APE8-rot-in 310.09 APE67-dihe-in -63.06, -9.2 -60.21, -45.83 APE12-dist-in 9.959 APE11-dist-in 8.835 APE10-dist-in 5.689 APE9-dist-in 3.869 None None None XRAY 2.24 0.231 0.276 A 293 273 0 0 0 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUB P11309 33 305 313.0 AMP:650 ATPlike Active DFGin 6.12 14.673 BLAminus -120.37, 167.93 65.74, 85.44 -95.36, 14.03 285.37, 78.45 -64.71, -9.22 in-in in 8.6 Saltbr-in 2.814 HRD-na-A -59.51, -51.25 68.06, 6.92 in-in-in SNCiii in-in ActLoopNT-in 2.999 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.12, 36.18 APE9-dihe-na -84.74, -152.35 APE8-dihe-in -93.27, 122.65 APE8-rot-in 302.12 APE67-dihe-in -68.21, -7.03 -55.31, -45.11 APE12-dist-in 9.8 APE11-dist-in 8.534 APE10-dist-in 5.457 APE9-dist-in 3.841 None None None XRAY 2.24 0.231 0.276 B 293 273 0 0 0 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUC P11309 34 305 313.0 AMP:750 ATPlike Active DFGin 6.11 14.741 BLAminus -134.94, 167.86 62.59, 83.1 -95.62, 21.45 280.06, 80.63 -81.83, 7.92 in-in in 8.716 Saltbr-in 2.612 HRD-na-A -67.31, -48.53 67.93, 5.85 in-in-in SNCiii in-in ActLoopNT-in 2.899 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.01, 44.98 APE9-dihe-na -103.92, -155.25 APE8-dihe-in -86.11, 117.99 APE8-rot-in 310.09 APE67-dihe-in -68.22, -9.23 -52.45, -45.39 APE12-dist-in 9.697 APE11-dist-in 8.654 APE10-dist-in 5.604 APE9-dist-in 3.847 None None None XRAY 2.24 0.231 0.276 C 293 272 0 0 0 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1YXUD P11309 33 305 313.0 AMP:850 ATPlike Active DFGin 6.236 14.556 BLAminus -126.04, 169.08 67.7, 73.28 -88.52, 13.94 289.01, 78.99 -70.28, -2.85 in-in in 8.789 Saltbr-in 2.466 HRD-na-A -64.06, -51.29 66.47, 10.4 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.8, 31.82 APE9-dihe-na -93.66, -159.09 APE8-dihe-in -85.99, 118.35 APE8-rot-in 303.12 APE67-dihe-in -71.66, -13.36 -52.91, -39.75 APE12-dist-in 9.896 APE11-dist-in 8.645 APE10-dist-in 5.457 APE9-dist-in 3.827 None None None XRAY 2.24 0.231 0.276 D 293 273 0 0 0 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 1XR1A P11309 32 308 313.0 ANP:501 ATPlike Active DFGin 5.888 14.214 BLAminus -138.05, 176.98 59.78, 85.31 -96.55, 16.88 287.93, 82.19 -61.38, -7.19 in-in in 8.717 Saltbr-in 2.833 HRD-na-A -59.95, -51.82 71.23, 5.72 in-in-in SNCiii in-in ActLoopNT-in 2.752 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.05, 45.66 APE9-dihe-na -114.17, -171.15 APE8-dihe-in -64.11, 112.97 APE8-rot-in 299.41 APE67-dihe-in -49.28, -12.21 -42.84, -67.53 APE12-dist-in 9.608 APE11-dist-in 8.695 APE10-dist-in 5.522 APE9-dist-in 4.07 None None None XRAY 2.1 0.267 0.301 A 300 277 0 0 0 0 [[38, 290]] 1.0 1xr1 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 3A99A P11309 33 305 313.0 ANP:501 ATPlike Active DFGin 5.934 14.254 BLAminus -128.38, 171.59 60.85, 87.29 -96.61, 22.08 288.57, 75.78 -65.84, -9.23 in-in in 8.754 Saltbr-in 2.604 HRD-na-A -66.86, -47.45 66.12, 8.26 in-in-in SNCiii in-in ActLoopNT-in 2.889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.19, 26.41 APE9-dihe-na -87.51, -159.07 APE8-dihe-in -85.64, 119.66 APE8-rot-in 305.41 APE67-dihe-in -70.7, -5.81 -56.65, -39.81 APE12-dist-in 9.612 APE11-dist-in 8.461 APE10-dist-in 5.29 APE9-dist-in 3.778 None None None XRAY 1.6 0.187 0.206 A 320 273 0 0 0 0 [[38, 290]] 1.0 3a99 Homo sapiens CAMK_PIM1_HUMAN CAMK 4.3e-65 225.5 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK PIM1 PIM1_HUMAN 2BZKB P11309 33 305 313.0 ANP:1306 ATPlike Active DFGin 6.126 14.443 BLAminus -123.86, 174.78 64.57, 79.13 -87.5, 17.23 286.98, 86.61 -67.5, -17.62 in-in in 8.781 Saltbr-in 2.727 HRD-na-A -70.49, -48.81 68.36, 6.4 in-in-in SNCiii in-in ActLoopNT-in 2.813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.63, 10.91 APE9-dihe-na -77.79, -156.22 APE8-dihe-in -90.85, 124.06 APE8-rot-in 315.85 APE67-dihe-in -68.94, -10.63 -60.69, -42.64 APE12-dist-in 9.464 APE11-dist-in 8.478 APE10-dist-in 4.851 APE9-dist-in 3.782 R250G None None XRAY 2.45 0.191 0.225 B 313 268 5 0 0 0 [[38, 290]] 1.0 2bzk Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1 256 256 185 186 187 189 191 67 89 93 164 166 165 167 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
CAMK STK11 STK11_HUMAN 2WTKC Q15831 47 342 433.0 ANP:2 ATPlike Active DFGin 6.192 13.745 BLAminus -119.65, -175.81 55.97, 66.27 -90.3, 25.87 311.18, 25.77 -80.53, -8.11 in-in in 9.443 Saltbr-in 3.361 HRD-in -68.47, -42.92 70.9, -7.9 in-in-in SNCiii in-in ActLoopNT-in 2.648 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na 69.85, 15.07 APE9-dihe-na -72.04, -171.91 APE8-dihe-in -90.01, 115.78 APE8-rot-in 306.68 APE67-dihe-in -55.63, -13.05 -36.08, -60.58 APE12-dist-in 7.784 APE11-dist-in 9.233 APE10-dist-in 5.395 APE9-dist-in 3.173 D194A None None XRAY 2.65 0.24 0.291 C 305 285 3 0 0 0 [[49, 309]] 1.0 2wtk Homo sapiens CAMK_STK11_HUMAN CAMK 7.7e-66 228.0 1 256 256 193 194 195 197 199 78 98 102 173 175 174 176 237 223 218 217 216 215 214 213 212 130 Serine/threonine-protein kinase STK11
CAMK STK11 STK11_HUMAN 2WTKF Q15831 45 340 433.0 ANP:4 ATPlike Active DFGin 5.938 13.841 BLAminus -119.11, -173.26 54.53, 62.76 -80.33, 19.16 295.83, 69.09 -48.31, -46.43 in-in in 9.483 Saltbr-in 3.568 HRD-in -68.65, -42.45 72.6, -14.65 in-in-in SNCiii in-in ActLoopNT-in 2.922 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na 45.91, 2.58 APE9-dihe-na -73.83, 178.68 APE8-dihe-in -66.98, 134.68 APE8-rot-in 293.57 APE67-dihe-in -65.1, -33.79 -54.08, -45.39 APE12-dist-in 8.609 APE11-dist-in 9.659 APE10-dist-in 5.793 APE9-dist-in 3.313 D194A None None XRAY 2.65 0.24 0.291 F 305 268 16 0 0 0 [[49, 309]] 1.0 2wtk Homo sapiens CAMK_STK11_HUMAN CAMK 7.7e-66 228.0 1 256 256 193 194 195 197 199 78 98 102 173 175 174 176 237 223 218 217 216 215 214 213 212 130 Serine/threonine-protein kinase STK11
CK1 CSNK1D KC1D_HUMAN 6RU6A P48730 3 294 415.0 ACP:60301 ATPlike Active DFGin 6.436 15.264 BLAminus -136.56, 176.84 69.53, 73.53 -93.66, 24.95 289.84, 81.36 -61.77, -30.96 in-in in 7.923 Saltbr-in 2.789 HRD-in -77.83, -55.12 76.08, 12.52 in-in-in SNCiii in-in ActLoopNT-in 2.85 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.64, 119.59 APE9-dihe-na 102.6, -136.74 APE8-dihe-in -117.46, 127.27 APE8-rot-in 311.09 APE67-dihe-in -57.82, -37.85 -53.66, -47.41 APE12-dist-in 12.315 APE11-dist-in 11.908 APE10-dist-in 6.481 APE9-dist-in 3.505 None None None XRAY 2.05 0.213 0.257 A 296 288 4 0 0 0 [[9, 275]] 1.0 6ru6 Homo sapiens CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7FA P48730 3 294 415.0 AMP:305 ATPlike Active DFGin 6.386 14.989 BLAminus -135.41, 179.24 65.29, 82.6 -99.51, 20.86 287.48, 77.77 -56.63, -36.85 in-in in 8.099 Saltbr-in 2.591 HRD-in -82.17, -51.93 74.76, 11.47 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -100.01, 118.96 APE9-dihe-na 109.81, -163.5 APE8-dihe-in -91.97, 119.49 APE8-rot-in 320.94 APE67-dihe-in -55.9, -38.32 -51.55, -37.41 APE12-dist-in 13.114 APE11-dist-in 12.585 APE10-dist-in 6.845 APE9-dist-in 3.948 None TPO220 TPO220 XRAY 1.96 0.19 0.221 A 296 292 0 0 0 0 [[9, 275]] 1.0 7p7f Homo sapiens CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7FB P48730 3 294 415.0 AMP:310 ATPlike Active DFGin 6.389 15.041 BLAminus -134.9, -178.65 62.6, 84.78 -99.93, 21.19 288.23, 78.97 -57.89, -34.16 in-in in 8.117 Saltbr-in 2.593 HRD-in -86.23, -54.05 76.65, 11.34 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.84, 118.88 APE9-dihe-na 108.83, -162.51 APE8-dihe-in -93.95, 118.29 APE8-rot-in 320.41 APE67-dihe-in -55.93, -38.53 -50.49, -37.42 APE12-dist-in 13.14 APE11-dist-in 12.546 APE10-dist-in 6.804 APE9-dist-in 4.014 None TPO220 TPO220 XRAY 1.96 0.19 0.221 B 296 292 0 0 0 0 [[9, 275]] 1.0 7p7f Homo sapiens CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7HA P48730 3 294 415.0 AMP:301 ATPlike Active DFGin 5.85 14.904 BLAminus -131.69, 175.32 69.71, 86.46 -98.17, 29.2 291.07, 84.43 -61.3, -36.51 in-in in 8.328 Saltbr-in 2.869 HRD-in -85.02, -56.99 74.97, 14.35 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.26, -19.24 APE9-dihe-na -88.34, -159.24 APE8-dihe-in -92.63, 127.36 APE8-rot-in 313.8 APE67-dihe-in -57.88, -32.21 -74.29, -29.96 APE12-dist-in 10.816 APE11-dist-in 12.399 APE10-dist-in 6.988 APE9-dist-in 4.101 None None None XRAY 2.4 0.225 0.268 A 296 292 0 0 0 0 [[9, 275]] 1.0 7p7h Homo sapiens CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 CSNK1D KC1D_HUMAN 7P7HB P48730 3 294 415.0 AMP:301 ATPlike Active DFGin 5.843 14.916 BLAminus -130.5, 174.9 69.57, 86.72 -100.58, 28.91 292.34, 82.14 -57.01, -35.01 in-in in 8.325 Saltbr-in 2.918 HRD-in -84.55, -57.9 81.6, 9.08 in-in-in SNCiii in-in ActLoopNT-in 2.946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.93, 49.41 APE9-dihe-na 140.08, -131.01 APE8-dihe-in -99.84, 119.2 APE8-rot-in 321.52 APE67-dihe-in -56.55, -33.9 -75.78, -27.7 APE12-dist-in 12.421 APE11-dist-in 12.165 APE10-dist-in 7.215 APE9-dist-in 4.736 None None None XRAY 2.4 0.225 0.268 B 296 292 0 0 0 0 [[9, 275]] 1.0 7p7h Homo sapiens CK1_CSNK1D_HUMAN CK1 1.6e-122 413.9 1 262 262 148 149 150 152 154 38 52 56 125 127 126 128 195 183 178 177 176 175 174 173 172 83 Casein kinase I isoform delta
CK1 TTBK1 TTBK1_HUMAN 4BTJA Q5TCY1 21 312 1321.0 ADP:61337 ATPlike Active DFGin 5.513 12.699 BLAminus -122.16, 167.53 65.74, 92.18 -107.62, 12.94 309.85, 113.04 -64.35, -28.29 in-in in 7.127 Saltbr-in 2.757 HRD-in -79.44, -52.71 73.3, -5.89 in-in-in SNCiii in-in ActLoopNT-in 2.821 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.78, 143.11 APE9-dihe-na 98.14, -168.76 APE8-dihe-in -84.14, 153.12 APE8-rot-in 322.08 APE67-dihe-in -60.57, -38.77 -75.21, -43.81 APE12-dist-in 11.388 APE11-dist-in 11.45 APE10-dist-in 5.945 APE9-dist-in 3.412 None None None XRAY 2.16 0.179 0.197 A 337 292 0 0 0 0 [[34, 295]] 1.0 4btj Homo sapiens CK1_TTBK1_HUMAN CK1 5.7e-105 356.4 1 262 262 175 176 177 179 181 63 77 81 151 153 152 154 221 209 204 203 202 201 200 199 198 108 Tau-tubulin kinase 1
CK1 TTBK1 TTBK1_HUMAN 4BTJB Q5TCY1 21 313 1321.0 ATP:61338 ATPlike Active DFGin 5.352 12.718 BLAminus -122.53, 168.88 60.17, 88.3 -98.51, 13.52 307.1, 115.33 -64.8, -32.06 in-in in 7.148 Saltbr-in 2.816 HRD-in -78.94, -51.75 72.7, -0.47 in-in-in SNCiii in-in ActLoopNT-in 2.748 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -105.82, -14.94 APE9-dihe-na -62.51, -161.18 APE8-dihe-in -100.71, 125.28 APE8-rot-in 309.68 APE67-dihe-in -55.66, -43.07 -52.23, -50.62 APE12-dist-in 11.078 APE11-dist-in 10.816 APE10-dist-in 6.463 APE9-dist-in 4.328 None None None XRAY 2.16 0.179 0.197 B 337 293 0 0 0 0 [[34, 295]] 1.0 4btj Homo sapiens CK1_TTBK1_HUMAN CK1 5.7e-105 356.4 1 262 262 175 176 177 179 181 63 77 81 151 153 152 154 221 209 204 203 202 201 200 199 198 108 Tau-tubulin kinase 1
CK1 TTBK2 TTBK2_HUMAN 6VRFA Q6IQ55 9 298 1244.0 ADP:301 ATPlike Active DFGin 5.354 13.116 BLAminus -121.29, 164.21 73.75, 82.24 -97.72, 13.38 304.67, 116.94 -64.06, -29.66 in-in in 7.214 Saltbr-in 2.751 HRD-in -77.1, -49.95 73.69, -4.56 in-in-in SNCiii in-in ActLoopNT-in 2.813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -108.12, -30.06 APE9-dihe-na -84.65, -146.34 APE8-dihe-in -107.58, 129.44 APE8-rot-in 302.21 APE67-dihe-in -59.13, -37.2 -56.28, -42.66 APE12-dist-in 11.197 APE11-dist-in 11.387 APE10-dist-in 5.48 APE9-dist-in 3.784 None None None XRAY 1.5 0.175 0.209 A 299 287 3 0 0 0 [[21, 282]] 1.0 6vrf Homo sapiens CK1_TTBK2_HUMAN CK1 7.7e-104 352.6 1 262 262 162 163 164 166 168 50 64 68 138 140 139 141 208 196 191 190 189 188 187 186 185 95 Tau-tubulin kinase 2
CK1 TTBK2 TTBK2_HUMAN 6VRFB Q6IQ55 9 298 1244.0 ADP:301 ATPlike Active DFGin 5.431 12.695 BLAminus -121.38, 163.64 74.07, 85.5 -102.64, 12.86 306.76, 116.33 -62.94, -32.7 in-in in 7.346 Saltbr-in 2.891 HRD-in -78.31, -51.54 73.55, 1.77 in-in-in SNCiii in-in ActLoopNT-in 2.86 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -109.78, -23.36 APE9-dihe-na -86.88, -149.11 APE8-dihe-in -108.63, 128.02 APE8-rot-in 302.45 APE67-dihe-in -58.2, -36.14 -56.96, -43.7 APE12-dist-in 11.039 APE11-dist-in 11.244 APE10-dist-in 5.337 APE9-dist-in 3.712 None None None XRAY 1.5 0.175 0.209 B 299 287 3 0 0 0 [[21, 282]] 1.0 6vrf Homo sapiens CK1_TTBK2_HUMAN CK1 7.7e-104 352.6 1 262 262 162 163 164 166 168 50 64 68 138 140 139 141 208 196 191 190 189 188 187 186 185 95 Tau-tubulin kinase 2
CMGC CDK2 CDK2_HUMAN 4I3ZA P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.408 15.148 BLAminus -137.57, -176.06 52.96, 75.44 -91.33, 19.91 280.72, 70.75 -64.88, -19.38 in-in in 8.599 Saltbr-in 2.988 HRD-in -80.76, -55.87 72.55, 4.85 in-in-in SNCiii in-in ActLoopNT-in 2.901 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.11, -96.25 APE9-dihe-na -51.92, 142.27 APE8-dihe-in -55.11, 135.08 APE8-rot-in 307.48 APE67-dihe-in -54.58, -26.51 -40.4, -56.95 APE12-dist-in 13.064 APE11-dist-in 10.585 APE10-dist-in 6.823 APE9-dist-in 3.305 None TPO160 TPO160 XRAY 2.05 0.199 0.228 A 296 296 0 0 0 0 [[4, 286]] 1.0 4i3z Homo sapiens CMGC_CDK2_HUMAN CMGC 6.2e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 4I3ZC P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.367 15.146 BLAminus -139.14, -175.0 51.64, 79.19 -95.11, 18.85 278.6, 70.91 -64.63, -17.11 in-in in 8.653 Saltbr-in 2.979 HRD-in -79.85, -55.96 72.81, 4.84 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.52, -96.18 APE9-dihe-na -52.61, 142.23 APE8-dihe-in -53.61, 133.4 APE8-rot-in 308.84 APE67-dihe-in -53.33, -28.57 -37.02, -58.54 APE12-dist-in 13.081 APE11-dist-in 10.618 APE10-dist-in 6.861 APE9-dist-in 3.305 None TPO160 TPO160 XRAY 2.05 0.199 0.228 C 296 296 0 0 0 0 [[4, 286]] 1.0 4i3z Homo sapiens CMGC_CDK2_HUMAN CMGC 6.2e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHRA P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.557 15.107 BLAminus -129.61, -176.27 55.27, 75.32 -97.07, 17.79 280.43, 72.68 -60.79, -23.59 in-in in 8.696 Saltbr-in 2.88 HRD-in -78.46, -57.59 71.9, 8.99 in-in-in SNCiii in-in ActLoopNT-in 2.877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.99, 139.5 APE9-dihe-na 85.76, 129.74 APE8-dihe-in -56.31, 140.07 APE8-rot-in 302.24 APE67-dihe-in -65.07, -20.31 -41.24, -52.35 APE12-dist-in 12.989 APE11-dist-in 10.171 APE10-dist-in 7.111 APE9-dist-in 3.341 None TPO160 TPO160 XRAY 2.17 0.18 0.21 A 298 296 0 0 0 0 [[4, 286]] 1.0 3qhr Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHRC P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.565 15.121 BLAminus -133.25, -174.75 53.96, 72.74 -93.36, 15.91 281.14, 71.23 -60.56, -21.49 in-in in 8.7 Saltbr-in 2.868 HRD-in -78.47, -57.15 72.13, 9.85 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.81, 147.52 APE9-dihe-na 81.05, 137.24 APE8-dihe-in -64.2, 137.48 APE8-rot-in 304.68 APE67-dihe-in -62.37, -22.27 -38.55, -53.11 APE12-dist-in 12.985 APE11-dist-in 10.232 APE10-dist-in 6.99 APE9-dist-in 3.293 None TPO160 TPO160 XRAY 2.17 0.18 0.21 C 298 296 0 0 0 0 [[4, 286]] 1.0 3qhr Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHWA P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.435 15.013 BLAminus -134.08, -174.07 54.44, 75.18 -91.31, 13.19 281.29, 72.4 -60.66, -23.16 in-in in 8.64 Saltbr-in 2.934 HRD-in -72.46, -52.11 70.84, 4.06 in-in-in SNCiii in-in ActLoopNT-in 2.903 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.61, -86.88 APE9-dihe-na -62.59, 147.47 APE8-dihe-in -61.56, 138.19 APE8-rot-in 297.56 APE67-dihe-in -60.69, -27.39 -44.54, -49.89 APE12-dist-in 12.995 APE11-dist-in 10.23 APE10-dist-in 6.782 APE9-dist-in 3.359 None TPO160 TPO160 XRAY 1.91 0.189 0.219 A 298 296 0 0 0 0 [[4, 286]] 1.0 3qhw Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 3QHWC P24941 1 296 298.0 ADP:60297 ATPlike Active DFGin 6.453 15.083 BLAminus -135.33, -175.53 57.5, 71.73 -89.85, 9.67 280.79, 72.12 -55.86, -26.79 in-in in 8.617 Saltbr-in 2.896 HRD-in -73.76, -53.15 71.96, 3.16 in-in-in SNCiii in-in ActLoopNT-in 2.898 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.86, -80.28 APE9-dihe-na -65.52, 146.91 APE8-dihe-in -61.19, 139.69 APE8-rot-in 298.69 APE67-dihe-in -57.2, -28.53 -47.15, -50.79 APE12-dist-in 12.997 APE11-dist-in 10.133 APE10-dist-in 6.722 APE9-dist-in 3.361 None TPO160 TPO160 XRAY 1.91 0.189 0.219 C 298 296 0 0 0 0 [[4, 286]] 1.0 3qhw Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1JSTA P24941 1 298 298.0 ATP:300 ATPlike Active DFGin 6.427 15.464 BLAminus -139.88, 179.46 48.93, 78.76 -92.24, 30.29 284.11, 71.63 -70.08, -30.4 in-in in 8.717 Saltbr-in 2.757 HRD-in -78.76, -47.67 60.69, 17.81 in-in-in SNCiii in-in ActLoopNT-in 2.949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.53, 164.64 APE9-dihe-na 80.72, 135.16 APE8-dihe-in -62.71, 138.95 APE8-rot-in 293.52 APE67-dihe-in -51.22, -30.94 -33.79, -62.16 APE12-dist-in 13.121 APE11-dist-in 11.934 APE10-dist-in 7.067 APE9-dist-in 3.277 None TPO160 TPO160 XRAY 2.6 0.2 999.0 A 298 298 0 0 0 0 [[4, 286]] 1.0 1jst Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1JSTC P24941 1 298 298.0 ATP:300 ATPlike Active DFGin 6.225 15.133 BLAminus -133.76, 179.75 53.92, 86.29 -100.05, 15.63 279.16, 71.07 -59.91, -21.96 in-in in 8.679 Saltbr-in 2.947 HRD-in -76.84, -49.3 61.77, 13.04 in-in-in SNCiii in-in ActLoopNT-in 2.701 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.31, -163.7 APE9-dihe-na 66.67, 148.27 APE8-dihe-in -72.61, 126.34 APE8-rot-in 301.65 APE67-dihe-in -51.49, -27.24 -26.21, -64.21 APE12-dist-in 13.412 APE11-dist-in 12.741 APE10-dist-in 6.942 APE9-dist-in 3.204 None TPO160 TPO160 XRAY 2.6 0.2 999.0 C 298 298 0 0 0 0 [[4, 286]] 1.0 1jst Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CJMA P24941 1 292 298.0 ATP:1294 ATPlike Active DFGin 6.412 15.477 BLAminus -133.49, 174.28 59.08, 80.72 -93.05, 17.33 280.25, 71.88 -51.1, -37.87 in-in in 8.875 Saltbr-in 3.027 HRD-in -83.77, -55.33 74.52, 15.85 in-in-in SNCiii in-in ActLoopNT-in 2.796 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.97, -48.89 APE9-dihe-na -98.03, 148.0 APE8-dihe-in -53.4, 136.55 APE8-rot-in 296.67 APE67-dihe-in -56.28, -31.52 -52.78, -45.83 APE12-dist-in 13.329 APE11-dist-in 10.553 APE10-dist-in 7.18 APE9-dist-in 3.464 None PTR15,TPO160 PTR15,TPO160 XRAY 2.3 0.204 0.265 A 298 287 5 0 0 0 [[4, 286]] 1.0 2cjm Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CJMC P24941 1 297 298.0 ATP:1298 ATPlike Active DFGin 6.446 15.389 BLAminus -136.23, -173.15 48.46, 78.84 -90.01, 21.15 280.3, 74.36 -53.78, -24.47 in-in in 8.957 Saltbr-in 2.575 HRD-in -82.67, -49.67 67.53, 9.26 in-in-in SNCiii in-in ActLoopNT-in 2.979 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.3, -72.35 APE9-dihe-na -81.21, 139.76 APE8-dihe-in -48.67, 128.86 APE8-rot-in 299.02 APE67-dihe-in -54.58, -22.4 -47.31, -51.92 APE12-dist-in 13.068 APE11-dist-in 10.808 APE10-dist-in 7.009 APE9-dist-in 3.58 None PTR15,TPO160 PTR15,TPO160 XRAY 2.3 0.204 0.265 C 298 297 0 0 0 0 [[4, 286]] 1.0 2cjm Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 4II5A P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.295 15.275 BLAminus -136.76, -174.67 48.15, 75.69 -89.27, 15.07 281.74, 67.11 -54.49, -30.0 in-in in 8.675 Saltbr-in 2.898 HRD-in -77.95, -58.94 72.46, 5.93 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.58, 147.66 APE9-dihe-na 74.72, 130.64 APE8-dihe-in -63.5, 139.49 APE8-rot-in 303.89 APE67-dihe-in -59.35, -27.46 -47.25, -50.52 APE12-dist-in 13.127 APE11-dist-in 10.372 APE10-dist-in 7.034 APE9-dist-in 3.344 None TPO160 TPO160 XRAY 2.15 0.2 0.226 A 298 296 0 0 0 0 [[4, 286]] 1.0 4ii5 Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 4II5C P24941 1 296 298.0 ADP:60301 ATPlike Active DFGin 6.289 15.288 BLAminus -134.89, -171.63 44.93, 79.89 -96.21, 16.02 275.02, 74.95 -60.79, -24.87 in-in in 8.666 Saltbr-in 2.94 HRD-in -77.09, -52.7 69.17, 3.7 in-in-in SNCiii in-in ActLoopNT-in 2.858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.65, 138.88 APE9-dihe-na 85.57, 133.69 APE8-dihe-in -65.51, 139.86 APE8-rot-in 305.2 APE67-dihe-in -60.76, -27.54 -47.35, -49.81 APE12-dist-in 13.141 APE11-dist-in 10.382 APE10-dist-in 7.061 APE9-dist-in 3.387 None TPO160 TPO160 XRAY 2.15 0.2 0.226 C 298 296 0 0 0 0 [[4, 286]] 1.0 4ii5 Homo sapiens CMGC_CDK2_HUMAN CMGC 6.3e-90 307.9 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1GY3A P24941 1 296 298.0 ATP:1297 ATPlike Active DFGin 6.711 15.739 BLAminus -148.85, -171.85 44.28, 78.14 -91.55, 12.53 280.84, 73.84 -49.56, -35.56 in-in in 8.826 Saltbr-in 2.87 HRD-in -78.88, -56.55 74.04, 15.78 in-in-in SNCiii in-in ActLoopNT-in 3.129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.01, 152.98 APE9-dihe-na 75.99, 139.26 APE8-dihe-in -71.28, 139.34 APE8-rot-in 297.69 APE67-dihe-in -59.44, -30.42 -47.65, -49.93 APE12-dist-in 13.156 APE11-dist-in 10.678 APE10-dist-in 7.643 APE9-dist-in 3.395 None TPO160 TPO160 XRAY 2.7 0.25 0.313 A 299 296 0 0 0 0 [[4, 286]] 1.0 1gy3 Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1GY3C P24941 1 296 298.0 ATP:1298 ATPlike Active DFGin 6.824 15.376 BLAminus -159.42, -172.39 46.56, 69.8 -88.25, 18.8 278.1, 68.22 -63.28, -3.45 in-in in 8.61 Saltbr-in 3.316 HRD-in -72.89, -69.46 86.12, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.794 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.99, 145.31 APE9-dihe-na 77.28, 144.74 APE8-dihe-in -75.96, 137.92 APE8-rot-in 277.1 APE67-dihe-in -64.24, -30.46 -41.97, -49.4 APE12-dist-in 13.195 APE11-dist-in 10.636 APE10-dist-in 7.772 APE9-dist-in 3.212 None TPO160 TPO160 XRAY 2.7 0.25 0.313 C 299 296 0 0 0 0 [[4, 286]] 1.0 1gy3 Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1QMZA P24941 1 296 298.0 ATP:60381 ATPlike Active DFGin 6.424 15.17 BLAminus -146.26, -172.65 47.53, 78.45 -93.94, 24.34 280.23, 76.95 -74.2, -4.32 in-in in 8.74 Saltbr-in 2.663 HRD-in -79.61, -61.2 70.52, 19.43 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.31, 152.76 APE9-dihe-na 72.53, 130.75 APE8-dihe-in -60.65, 130.8 APE8-rot-in 293.88 APE67-dihe-in -60.7, -26.37 -33.48, -54.72 APE12-dist-in 13.02 APE11-dist-in 10.095 APE10-dist-in 7.17 APE9-dist-in 3.235 None TPO160 TPO160 XRAY 2.2 0.22 0.28 A 299 296 0 0 0 0 [[4, 286]] 1.0 1qmz Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 1QMZC P24941 1 296 298.0 ATP:60381 ATPlike Active DFGin 6.512 15.134 BLAminus -147.61, -169.98 41.15, 80.53 -95.52, 25.6 283.09, 73.82 -79.03, -0.31 in-in in 8.74 Saltbr-in 2.54 HRD-in -75.88, -57.22 71.34, 18.39 in-in-in SNCiii in-in ActLoopNT-in 2.993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.04, 148.92 APE9-dihe-na 73.46, 130.58 APE8-dihe-in -61.75, 132.61 APE8-rot-in 296.97 APE67-dihe-in -70.09, -17.52 -37.4, -48.3 APE12-dist-in 12.947 APE11-dist-in 10.103 APE10-dist-in 7.19 APE9-dist-in 3.234 None TPO160 TPO160 XRAY 2.2 0.22 0.28 C 299 296 0 0 0 0 [[4, 286]] 1.0 1qmz Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCHA P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.648 15.496 BLAminus -138.14, 178.31 65.58, 62.78 -86.23, 16.74 281.6, 70.81 -63.75, -23.41 in-in in 8.795 Saltbr-in 2.828 HRD-in -78.21, -56.44 71.04, 15.24 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.4, 152.64 APE9-dihe-na 69.68, 132.94 APE8-dihe-in -57.07, 137.05 APE8-rot-in 294.63 APE67-dihe-in -60.03, -20.02 -46.03, -52.89 APE12-dist-in 13.198 APE11-dist-in 10.36 APE10-dist-in 7.208 APE9-dist-in 3.286 None TPO160 TPO160 XRAY 1.7 0.15 0.182 A 299 296 0 0 0 0 [[4, 286]] 1.0 2cch Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCHC P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.477 15.382 BLAminus -137.71, -178.58 51.07, 78.61 -96.17, 22.01 279.1, 72.77 -65.43, -25.94 in-in in 8.653 Saltbr-in 2.719 HRD-in -81.45, -53.09 63.51, 17.55 in-in-in SNCiii in-in ActLoopNT-in 2.886 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.56, 136.55 APE9-dihe-na 76.27, 128.23 APE8-dihe-in -59.37, 134.24 APE8-rot-in 303.33 APE67-dihe-in -63.22, -26.6 -41.45, -49.27 APE12-dist-in 12.866 APE11-dist-in 10.056 APE10-dist-in 7.377 APE9-dist-in 3.26 None TPO160 TPO160 XRAY 1.7 0.15 0.182 C 299 296 0 0 0 0 [[4, 286]] 1.0 2cch Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCIA P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.459 15.372 BLAminus -128.71, -173.86 48.01, 81.43 -98.73, 25.24 282.02, 74.31 -66.86, -20.71 in-in in 8.902 Saltbr-in 3.076 HRD-in -75.27, -47.91 58.22, 13.15 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.39, 140.99 APE9-dihe-na 76.14, 131.3 APE8-dihe-in -63.2, 133.24 APE8-rot-in 305.53 APE67-dihe-in -53.35, -21.65 -35.23, -63.18 APE12-dist-in 12.958 APE11-dist-in 10.323 APE10-dist-in 7.246 APE9-dist-in 3.291 None TPO160 TPO160 XRAY 2.7 0.264 0.321 A 299 296 0 0 0 0 [[4, 286]] 1.0 2cci Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK2 CDK2_HUMAN 2CCIC P24941 1 296 298.0 ATP:61297 ATPlike Active DFGin 6.232 15.382 BLAminus -129.31, 167.15 64.1, 86.76 -100.18, 28.53 276.86, 72.85 -63.26, -37.36 in-in in 8.551 Saltbr-in 2.666 HRD-in -73.66, -47.99 63.69, 10.4 in-in-in SNCiii in-in ActLoopNT-in 3.064 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.2, 138.6 APE9-dihe-na 71.13, 137.9 APE8-dihe-in -63.98, 129.66 APE8-rot-in 301.4 APE67-dihe-in -61.96, -9.78 -29.15, -60.17 APE12-dist-in 12.753 APE11-dist-in 9.767 APE10-dist-in 7.42 APE9-dist-in 3.234 None TPO160 TPO160 XRAY 2.7 0.264 0.321 C 299 296 0 0 0 0 [[4, 286]] 1.0 2cci Homo sapiens CMGC_CDK2_HUMAN CMGC 6.4e-90 307.8 1 301 301 144 145 146 148 150 33 51 55 124 126 125 127 185 172 167 166 165 164 163 162 161 81 Cyclin-dependent kinase 2
CMGC CDK7 CDK7_HUMAN 9HIYJ P50613 10 310 346.0 AGS:60401 ATPlike Active DFGin 6.727 15.718 BLAminus -144.39, -174.23 58.17, 64.72 -87.83, 23.91 281.92, 72.77 -77.85, -11.75 in-in in 8.542 Saltbr-in 3.5 HRD-in -67.31, -50.64 65.74, 8.28 in-in-in SNCiii in-in ActLoopNT-in 2.733 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.25, 164.09 APE9-dihe-na 67.64, 142.62 APE8-dihe-in -59.57, 146.87 APE8-rot-in 317.63 APE67-dihe-in -64.96, -18.05 -61.86, -38.17 APE12-dist-in 13.579 APE11-dist-in 11.322 APE10-dist-in 6.933 APE9-dist-in 3.352 D97N None None EM 2.3 999.0 999.0 J 349 287 14 0 0 3 [[12, 295]] 1.0 9hiy Homo sapiens CMGC_CDK7_HUMAN CMGC 1.8e-78 271.6 1 301 301 154 155 156 158 160 41 62 66 134 136 135 137 195 182 177 176 175 174 173 172 171 92 Cyclin-dependent kinase 7
CMGC CDK9 CDK9_HUMAN 3BLQA P50750 7 325 372.0 ATP:332 ATPlike Active DFGin 6.983 15.235 BLAminus -137.33, 167.71 61.72, 82.78 -101.54, 27.58 292.13, 71.79 -68.35, -20.47 in-in in 9.514 Saltbr-in 3.257 HRD-in -70.77, -57.41 73.91, 6.35 in-in-in SNCiii in-in ActLoopNT-in 2.85 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.28, 155.2 APE9-dihe-na 75.14, 129.25 APE8-dihe-in -51.14, 147.2 APE8-rot-in 304.68 APE67-dihe-in -62.86, -25.73 -50.2, -49.1 APE12-dist-in 13.028 APE11-dist-in 11.03 APE10-dist-in 6.896 APE9-dist-in 3.154 None TPO186 TPO186 XRAY 2.9 0.174 0.234 A 331 296 23 0 0 7 [[19, 315]] 1.0 3blq Homo sapiens CMGC_CDK9_HUMAN CMGC 4.1e-80 275.1 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CDK9 CDK9_HUMAN 4IMYC P50750 8 330 372.0 AMP:401 ATPlike Active DFGin 6.789 15.123 BLAminus -140.61, 175.84 60.41, 77.79 -97.02, 19.01 284.69, 80.72 -68.98, -8.54 in-in in 9.232 Saltbr-in 2.833 HRD-in -67.68, -50.97 65.16, 13.16 in-in-in SNCiii in-in ActLoopNT-in 2.928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.81, 161.81 APE9-dihe-na 73.71, 135.92 APE8-dihe-in -53.34, 141.57 APE8-rot-in 294.85 APE67-dihe-in -61.16, -25.06 -47.9, -50.46 APE12-dist-in 13.386 APE11-dist-in 11.431 APE10-dist-in 7.006 APE9-dist-in 3.279 None TPO186 TPO186 XRAY 2.94 0.209 0.245 C 332 311 12 0 0 0 [[19, 315]] 1.0 4imy Homo sapiens CMGC_CDK9_HUMAN CMGC 4.1e-80 275.1 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CDK9 CDK9_HUMAN 4IMYE P50750 8 330 372.0 AMP:401 ATPlike Active DFGin 6.794 15.112 BLAminus -141.41, 175.75 59.75, 77.9 -96.66, 19.65 284.44, 80.03 -69.65, -8.18 in-in in 9.197 Saltbr-in 2.816 HRD-in -68.02, -51.11 68.06, 12.23 in-in-in SNCiii in-in ActLoopNT-in 2.919 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.97, 161.65 APE9-dihe-na 74.14, 135.63 APE8-dihe-in -53.23, 140.74 APE8-rot-in 294.81 APE67-dihe-in -59.86, -25.62 -47.7, -50.88 APE12-dist-in 13.405 APE11-dist-in 11.437 APE10-dist-in 7.01 APE9-dist-in 3.278 None TPO186 TPO186 XRAY 2.94 0.209 0.245 E 332 314 9 0 0 0 [[19, 315]] 1.0 4imy Homo sapiens CMGC_CDK9_HUMAN CMGC 4.1e-80 275.1 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CDK9 CDK9_HUMAN 3MIAA P50750 8 340 372.0 ANP:352 ATPlike Active DFGin 6.803 15.077 BLAminus -137.71, 176.33 64.58, 74.97 -96.55, 26.44 284.7, 90.38 -67.18, -14.54 in-in in 9.313 Saltbr-in 2.689 HRD-in -70.81, -51.43 63.16, 28.9 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.04, 160.49 APE9-dihe-na 82.03, 127.94 APE8-dihe-in -49.75, 143.51 APE8-rot-in 280.63 APE67-dihe-in -52.26, -14.47 -51.96, -57.94 APE12-dist-in 13.258 APE11-dist-in 11.524 APE10-dist-in 6.949 APE9-dist-in 3.523 None TPO186 TPO186 XRAY 3.0 0.219 0.287 A 351 325 8 0 0 0 [[19, 315]] 1.0 3mia Homo sapiens CMGC_CDK9_HUMAN CMGC 5.1e-80 274.8 1 301 301 166 167 168 170 172 48 66 70 146 148 147 149 211 198 193 192 191 190 189 188 187 104 Cyclin-dependent kinase 9
CMGC CSNK2A1 CSK21_HUMAN 3JUHA P68400 2 335 391.0 ANP:339 ATPlike Active DFGin 7.401 16.242 BLAminus -115.69, -178.29 60.62, 71.57 -93.06, 11.37 295.1, 82.09 -62.22, -22.13 in-in in 9.721 Saltbr-in 2.746 HRD-in -70.06, -49.94 64.15, 21.46 in-in-in SNCiii in-in ActLoopNT-in 2.862 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.98, 153.86 APE9-dihe-na 70.33, -177.46 APE8-dihe-in -104.19, 142.14 APE8-rot-in 291.28 APE67-dihe-in -67.33, -12.83 -40.87, -55.27 APE12-dist-in 12.316 APE11-dist-in 9.578 APE10-dist-in 6.044 APE9-dist-in 3.086 V66A,M163L None None XRAY 1.66 0.158 0.218 A 335 334 0 0 0 0 [[39, 324]] 1.0 3juh Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.1e-70 244.1 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 3JUHB P68400 2 335 391.0 ANP:339 ATPlike Active DFGin 7.492 16.356 BLAminus -124.69, -176.29 51.46, 71.26 -80.35, 23.48 299.01, 83.37 -80.68, -22.43 in-in in 9.852 Saltbr-in 2.699 HRD-in -76.38, -50.5 78.84, -1.13 in-in-in SNCiii in-in ActLoopNT-in 2.807 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.59, 175.23 APE9-dihe-na 56.07, 138.8 APE8-dihe-in -58.03, 149.04 APE8-rot-in 282.66 APE67-dihe-in -69.98, -19.52 -43.94, -46.02 APE12-dist-in 12.714 APE11-dist-in 9.541 APE10-dist-in 5.884 APE9-dist-in 3.411 V66A,M163L None None XRAY 1.66 0.158 0.218 B 335 334 0 0 0 0 [[39, 324]] 1.0 3juh Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.1e-70 244.1 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 6Z19B P68400 2 329 391.0 ADP:401 ATPlike Active DFGin 7.399 16.102 BLAminus -106.47, -175.56 60.6, 79.25 -100.03, 20.37 297.28, 82.12 -73.41, -21.13 in-in in 8.717 Saltbr-in 2.8 HRD-in -71.6, -55.48 75.88, 3.64 in-in-in SNCiii in-in ActLoopNT-in 2.928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.14, 153.25 APE9-dihe-na 78.4, 166.67 APE8-dihe-in -74.52, 152.52 APE8-rot-in 285.35 APE67-dihe-in -64.18, -23.8 -57.77, -45.77 APE12-dist-in 12.968 APE11-dist-in 10.993 APE10-dist-in 6.495 APE9-dist-in 3.591 None None None XRAY 1.47 0.19 0.221 B 328 328 0 0 0 0 [[39, 324]] 1.0 6z19 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.2e-69 240.7 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 3NSZA P68400 2 328 391.0 ANP:1000 ATPlike Active DFGin 7.29 16.639 BLAminus -116.89, -174.28 57.53, 72.95 -91.24, 19.04 295.43, 81.74 -67.97, -19.44 in-in in 9.56 Saltbr-in 2.721 HRD-in -71.38, -46.87 68.1, 12.99 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.59, 174.99 APE9-dihe-na 61.7, -173.37 APE8-dihe-in -118.84, 140.8 APE8-rot-in 296.4 APE67-dihe-in -69.07, -13.11 -30.5, -60.15 APE12-dist-in 12.605 APE11-dist-in 10.316 APE10-dist-in 6.145 APE9-dist-in 2.961 None None None XRAY 1.3 0.169 0.187 A 330 327 0 0 0 0 [[39, 324]] 1.0 3nsz Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.3e-69 240.7 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 1PJKA P68400 2 332 391.0 ANP:340 ATPlike Active DFGin 7.44 16.238 BLAminus -115.92, -179.78 53.21, 80.99 -96.44, 28.53 295.64, 78.1 -72.28, -30.66 in-in in 8.93 Saltbr-in 2.81 HRD-in -80.54, -40.11 57.34, 9.1 in-in-in SNCiii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.58, 173.24 APE9-dihe-na 63.2, 174.94 APE8-dihe-in -93.15, 157.9 APE8-rot-in 277.8 APE67-dihe-in -66.77, -23.27 -54.74, -47.48 APE12-dist-in 13.026 APE11-dist-in 10.669 APE10-dist-in 6.368 APE9-dist-in 3.173 None None None XRAY 2.5 0.188 0.257 A 334 331 0 0 0 0 [[39, 324]] 1.0 1pjk Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.3e-69 240.6 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 2PVRA P68400 2 329 391.0 ANP:6004 ATPlike Active DFGin 7.492 16.497 BLAminus -121.67, -179.6 56.35, 70.32 -89.0, 17.49 296.64, 81.69 -72.81, -15.87 in-in in 9.284 Saltbr-in 2.7 HRD-in -75.03, -46.77 70.22, 6.37 in-in-in SNCiii in-in ActLoopNT-in 2.86 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.8, 175.01 APE9-dihe-na 60.61, 163.14 APE8-dihe-in -93.89, 147.69 APE8-rot-in 305.18 APE67-dihe-in -67.68, -15.16 -34.32, -58.13 APE12-dist-in 12.728 APE11-dist-in 10.346 APE10-dist-in 6.131 APE9-dist-in 3.189 None None None XRAY 1.605 0.187 0.241 A 334 328 0 0 0 0 [[39, 324]] 1.0 2pvr Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.3e-69 240.6 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 3U87B P68400 2 331 391.0 ANP:60401 ATPlike Active DFGin 7.471 16.335 BLAminus -123.33, -169.35 50.94, 85.5 -106.65, 24.88 299.58, 83.47 -72.97, -19.72 in-in in 9.505 Saltbr-in 2.848 HRD-in -72.0, -49.6 70.96, 8.41 in-in-in SNCiii in-in ActLoopNT-in 2.78 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.34, 168.89 APE9-dihe-na 66.61, 166.24 APE8-dihe-in -76.34, 153.62 APE8-rot-in 296.27 APE67-dihe-in -70.99, -10.83 -52.99, -46.79 APE12-dist-in 12.822 APE11-dist-in 10.801 APE10-dist-in 6.15 APE9-dist-in 3.577 None None None XRAY 2.9 0.187 0.218 B 349 324 0 0 0 0 [[39, 324]] 1.0 3u87 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.5e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5OQUB P68400 4 327 391.0 ADP:401 ATPlike Active DFGin 7.324 16.392 BLAminus -107.74, -171.87 52.49, 78.62 -101.36, 19.11 291.9, 83.91 -71.23, -12.83 in-in in 9.496 Saltbr-in 2.901 HRD-in -65.86, -46.78 65.2, 13.55 in-in-in SNCiii in-in ActLoopNT-in 2.895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.87, 169.85 APE9-dihe-na 66.11, 165.52 APE8-dihe-in -87.57, 142.09 APE8-rot-in 294.71 APE67-dihe-in -65.28, -26.45 -36.1, -50.26 APE12-dist-in 12.592 APE11-dist-in 10.419 APE10-dist-in 6.089 APE9-dist-in 3.154 R21S None None XRAY 2.324 0.221 0.244 B 352 324 0 0 0 0 [[39, 324]] 1.0 5oqu Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5ORKB P68400 4 326 391.0 ADP:401 ATPlike Active DFGin 7.365 16.488 BLAminus -111.04, -174.54 54.53, 77.94 -96.47, 19.83 296.01, 82.36 -66.2, -23.13 in-in in 9.552 Saltbr-in 3.041 HRD-in -70.69, -49.04 67.52, 16.07 in-in-in SNCiii in-in ActLoopNT-in 2.862 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.56, 172.18 APE9-dihe-na 65.73, 167.16 APE8-dihe-in -89.89, 143.95 APE8-rot-in 298.57 APE67-dihe-in -64.35, -23.63 -31.56, -56.57 APE12-dist-in 12.614 APE11-dist-in 10.418 APE10-dist-in 6.062 APE9-dist-in 3.149 R21S None None XRAY 2.143 0.217 0.243 B 352 323 0 0 0 0 [[39, 324]] 1.0 5ork Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 7QUXA P68400 2 329 391.0 ADP:60401 ATPlike Active DFGin 7.585 16.194 BLAminus -111.52, -172.63 60.82, 80.19 -104.84, 23.49 298.85, 85.23 -72.93, -20.15 in-in in 8.958 Saltbr-in 2.838 HRD-in -72.19, -52.24 72.27, 9.35 in-in-in SNCiii in-in ActLoopNT-in 2.846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.66, 178.74 APE9-dihe-na 61.29, -172.26 APE8-dihe-in -113.53, 144.19 APE8-rot-in 304.18 APE67-dihe-in -65.08, -18.11 -36.49, -57.4 APE12-dist-in 12.723 APE11-dist-in 10.579 APE10-dist-in 6.214 APE9-dist-in 2.896 None SEP2 SEP2 XRAY 1.48 0.181 0.204 A 352 328 0 0 0 0 [[39, 324]] 1.0 7qux Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 6YZHA P68400 3 329 391.0 ADP:60403 ATPlike Active DFGin 7.386 16.31 BLAminus -108.01, -176.38 61.1, 79.34 -99.78, 17.26 297.37, 82.49 -78.41, -8.16 in-in in 9.131 Saltbr-in 2.829 HRD-in -74.51, -47.7 69.86, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.83, 175.48 APE9-dihe-na 62.95, -168.81 APE8-dihe-in -126.52, 135.38 APE8-rot-in 299.93 APE67-dihe-in -66.68, -18.66 -34.87, -54.46 APE12-dist-in 12.682 APE11-dist-in 10.343 APE10-dist-in 6.227 APE9-dist-in 3.084 None None None XRAY 1.19 0.173 0.19 A 398 327 0 0 0 0 [[39, 324]] 1.0 6yzh Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 2.4e-69 239.8 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU6A P68400 3 329 391.0 ATP:401 ATPlike Active DFGin 7.373 16.301 BLAminus -117.96, -176.97 52.74, 80.35 -94.88, 19.06 296.35, 83.62 -69.11, -18.98 in-in in 9.296 Saltbr-in 2.997 HRD-in -73.54, -48.21 69.17, 10.55 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.92, 173.11 APE9-dihe-na 58.61, 170.65 APE8-dihe-in -94.81, 150.1 APE8-rot-in 295.17 APE67-dihe-in -71.66, -13.32 -37.08, -56.84 APE12-dist-in 12.652 APE11-dist-in 10.334 APE10-dist-in 6.182 APE9-dist-in 3.146 R21S,K74A,K75A,K76A None None XRAY 1.36 0.188 0.209 A 328 327 0 0 0 0 [[39, 324]] 1.0 5cu6 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 8.1e-69 238.0 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A2 CSK22_HUMAN 8QCGB P19784 7 333 350.0 ANP:401 ATPlike Active DFGin 7.314 16.209 BLAminus -113.91, -178.96 61.11, 75.42 -92.86, 17.98 298.38, 79.8 -69.62, -20.0 in-in in 9.436 Saltbr-in 2.83 HRD-in -72.51, -49.6 69.57, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.828 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.91, 170.94 APE9-dihe-na 61.2, 166.37 APE8-dihe-in -93.43, 149.98 APE8-rot-in 300.62 APE67-dihe-in -69.2, -15.18 -40.28, -54.89 APE12-dist-in 12.657 APE11-dist-in 10.295 APE10-dist-in 6.172 APE9-dist-in 3.11 C336S None None XRAY 1.04 0.151 0.17 B 364 327 0 0 0 0 [[40, 325]] 1.0 8qcg Homo sapiens CMGC_CSNK2A2_HUMAN CMGC 1e-69 241.0 1 301 301 175 176 177 179 181 69 82 86 154 156 155 157 215 202 197 196 195 194 193 192 191 115 Casein kinase II subunit alpha'
CMGC DYRK1A DYR1A_HUMAN 7A4OA Q13627 136 481 763.0 ANP:501 ATPlike Active DFGin 7.404 15.034 BLAminus -121.6, 173.77 67.88, 73.96 -92.34, 22.26 284.87, 82.1 -70.26, -21.97 in-in in 8.684 Saltbr-in 2.793 HRD-in -65.03, -49.19 79.83, -0.94 in-in-in SNCiii in-in ActLoopNT-in 2.8 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.61, 174.39 APE9-dihe-na 70.74, 151.67 APE8-dihe-in -72.34, 134.57 APE8-rot-in 295.77 APE67-dihe-in -65.19, -24.46 -43.45, -47.13 APE12-dist-in 10.098 APE11-dist-in 12.237 APE10-dist-in 7.723 APE9-dist-in 3.156 None PTR321 PTR321 XRAY 1.9 0.18 0.203 A 382 341 5 0 0 0 [[159, 479]] 1.0 7a4o Homo sapiens CMGC_DYRK1A_HUMAN CMGC 1e-90 310.0 1 301 301 306 307 308 310 312 188 203 207 284 286 285 287 343 331 326 325 324 323 322 321 320 239 Dual specificity tyrosine-phosphorylation-regulated kinase 1A
CMGC GSK3B GSK3B_HUMAN 4NM5A P49841 24 383 420.0 ADP:60401 ATPlike Active DFGin 6.55 14.006 BLAminus -136.16, -177.73 61.88, 88.47 -108.64, 28.76 287.87, 80.78 -73.66, -15.44 in-in in 8.619 Saltbr-in 2.673 HRD-in -65.83, -43.73 64.82, 15.23 in-in-in SNCiii in-in ActLoopNT-in 2.839 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.92, 173.97 APE9-dihe-na 66.26, 147.02 APE8-dihe-in -77.1, 152.8 APE8-rot-in 293.28 APE67-dihe-inflip 82.03, -25.76 -52.23, 150.7 APE12-dist-in 13.279 APE11-dist-in 11.599 APE10-dist-in 6.949 APE9-dist-in 3.238 None None None XRAY 2.3 0.185 0.232 A 377 360 0 0 0 0 [[56, 340]] 1.0 4nm5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 4NM7A P49841 25 383 420.0 ADP:60401 ATPlike Active DFGin 6.515 13.993 BLAminus -137.35, -178.06 62.82, 88.6 -107.3, 24.56 288.41, 80.2 -69.84, -12.63 in-in in 8.818 Saltbr-in 2.743 HRD-in -66.5, -46.64 67.84, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.829 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 172.54 APE9-dihe-na 68.99, 153.43 APE8-dihe-in -86.9, 151.79 APE8-rot-in 300.04 APE67-dihe-inflip 84.67, -25.93 -50.38, 146.2 APE12-dist-in 13.355 APE11-dist-in 11.678 APE10-dist-in 6.905 APE9-dist-in 3.21 None None None XRAY 2.3 0.185 0.234 A 377 354 2 0 0 0 [[56, 340]] 1.0 4nm7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 4NM3A P49841 6 383 420.0 ADP:60409 ATPlike Active DFGin 6.475 13.947 BLAminus -129.98, -178.05 63.17, 87.87 -103.96, 21.26 289.38, 80.04 -65.46, -16.35 in-in in 8.806 Saltbr-in 2.726 HRD-in -69.81, -46.77 71.59, 6.75 in-in-in SNCiii in-in ActLoopNT-in 2.75 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.34, 169.99 APE9-dihe-na 69.15, 146.37 APE8-dihe-in -83.47, 151.55 APE8-rot-in 296.54 APE67-dihe-inflip 86.0, -31.11 -49.79, 146.79 APE12-dist-in 13.269 APE11-dist-in 11.484 APE10-dist-in 6.907 APE9-dist-in 3.112 None SEP9 SEP9 XRAY 2.1 0.197 0.242 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nm3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1BA P49841 35 388 420.0 ANP:60430 ATPlike Active DFGin 6.767 13.788 BLAminus -136.8, -178.88 61.6, 83.12 -97.64, 25.1 286.09, 80.4 -68.7, -13.11 in-in in 8.566 Saltbr-in 2.59 HRD-in -71.16, -45.98 70.36, 3.88 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.52, 175.26 APE9-dihe-na 75.44, 133.64 APE8-dihe-in -75.76, 147.49 APE8-rot-in 306.57 APE67-dihe-inflip 98.15, -33.72 -56.43, 141.52 APE12-dist-in 13.056 APE11-dist-in 10.974 APE10-dist-in 5.893 APE9-dist-in 3.112 None None None XRAY 1.8 0.216 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1BB P49841 23 386 420.0 ANP:60930 ATPlike Active DFGin 6.609 13.669 BLAminus -136.4, -177.03 61.49, 81.88 -98.08, 27.2 288.49, 82.07 -71.33, -13.14 in-in in 8.457 Saltbr-in 2.713 HRD-in -67.51, -45.87 68.87, 6.43 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.88, 174.17 APE9-dihe-na 76.18, 138.08 APE8-dihe-in -76.12, 141.41 APE8-rot-in 301.11 APE67-dihe-inflip 98.0, -37.59 -54.78, 144.25 APE12-dist-in 12.978 APE11-dist-in 11.066 APE10-dist-in 6.011 APE9-dist-in 3.174 None None None XRAY 1.8 0.216 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1CA P49841 35 388 420.0 ADP:60430 ATPlike Active DFGin 6.812 13.93 BLAminus -139.24, -179.75 62.79, 82.17 -97.34, 25.19 286.68, 82.3 -65.83, -19.9 in-in in 8.601 Saltbr-in 2.647 HRD-in -68.65, -43.85 68.34, 7.36 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.05, 172.96 APE9-dihe-na 78.17, 130.85 APE8-dihe-in -73.54, 145.97 APE8-rot-in 310.16 APE67-dihe-inflip 99.09, -35.01 -54.43, 141.28 APE12-dist-in 13.077 APE11-dist-in 11.067 APE10-dist-in 5.926 APE9-dist-in 3.2 None None None XRAY 2.1 0.218 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1c Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1J1CB P49841 23 386 420.0 ADP:60930 ATPlike Active DFGin 6.694 13.709 BLAminus -138.27, -179.99 63.33, 82.68 -100.46, 28.2 289.88, 80.26 -70.45, -13.94 in-in in 8.52 Saltbr-in 2.738 HRD-in -67.92, -43.36 67.59, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.71, 170.27 APE9-dihe-na 78.71, 139.86 APE8-dihe-in -81.56, 140.05 APE8-rot-in 302.5 APE67-dihe-inflip 101.62, -36.53 -50.52, 137.44 APE12-dist-in 12.868 APE11-dist-in 11.128 APE10-dist-in 6.025 APE9-dist-in 3.208 None None None XRAY 2.1 0.218 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1c Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 8XN6A P49841 35 384 420.0 ANP:501 ATPlike Active DFGin 6.682 13.862 BLAminus -137.72, 173.39 67.73, 84.48 -99.84, 22.57 287.77, 80.54 -65.33, -24.58 in-in in 8.463 Saltbr-in 2.63 HRD-in -71.05, -47.88 67.82, 15.5 in-in-in SNCiii in-in ActLoopNT-in 3.054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.0, 164.43 APE9-dihe-na 85.44, 135.36 APE8-dihe-in -74.2, 151.55 APE8-rot-in 291.81 APE67-dihe-in -69.28, -17.83 -36.59, -67.98 APE12-dist-in 12.907 APE11-dist-in 10.787 APE10-dist-in 5.68 APE9-dist-in 3.182 None None None XRAY 2.4 0.194 0.242 A 421 350 0 0 0 0 [[56, 340]] 1.0 8xn6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1PYXA P49841 35 386 420.0 ANP:1001 ATPlike Active DFGin 6.584 13.622 BLAminus -138.81, -178.07 65.18, 79.92 -98.83, 26.07 289.95, 78.27 -73.24, -7.6 in-in in 8.373 Saltbr-in 2.765 HRD-in -67.79, -47.84 71.28, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.12, 170.17 APE9-dihe-na 80.64, 129.74 APE8-dihe-in -63.79, 140.05 APE8-rot-in 299.48 APE67-dihe-in -56.43, -21.61 -20.65, -80.28 APE12-dist-in 12.903 APE11-dist-in 10.937 APE10-dist-in 5.784 APE9-dist-in 3.15 None None None XRAY 2.4 0.206 0.233 A 422 343 9 0 0 0 [[56, 340]] 1.0 1pyx Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_HUMAN 1PYXB P49841 35 383 420.0 ANP:2001 ATPlike Active DFGin 6.593 13.718 BLAminus -140.94, -178.47 65.26, 79.98 -98.11, 22.32 290.75, 76.51 -68.32, -7.73 in-in in 8.488 Saltbr-in 2.666 HRD-in -69.98, -47.18 70.83, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.3, 169.41 APE9-dihe-na 81.27, 131.24 APE8-dihe-in -66.67, 140.79 APE8-rot-in 300.74 APE67-dihe-in -56.9, -22.2 -20.58, -79.9 APE12-dist-in 12.838 APE11-dist-in 10.861 APE10-dist-in 5.718 APE9-dist-in 3.132 None None None XRAY 2.4 0.206 0.233 B 422 338 11 0 0 0 [[56, 340]] 1.0 1pyx Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC MAPK1 MK01_HUMAN 6OPGA P28482 10 358 360.0 ANP:60401 ATPlike Active DFGin 6.535 14.668 BLAminus -130.49, -173.97 55.35, 72.85 -87.66, 25.26 285.94, 65.79 -65.31, -19.22 in-in in 9.066 Saltbr-in 2.695 HRD-in -72.87, -54.34 77.9, 3.87 in-in-in SNCiii in-in ActLoopNT-in 2.758 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -102.35, 163.88 APE9-dihe-na 79.13, 168.47 APE8-dihe-in -88.92, 138.85 APE8-rot-in 292.11 APE67-dihe-in -68.23, -14.82 -51.35, -45.86 APE12-dist-in 12.57 APE11-dist-in 11.134 APE10-dist-in 6.653 APE9-dist-in 2.942 None TPO185,PTR187 TPO185,PTR187 XRAY 2.9 0.16 0.239 A 354 349 0 0 0 0 [[25, 313]] 1.0 6opg Homo sapiens CMGC_MAPK1_HUMAN CMGC 8.6e-86 293.8 1 301 301 166 167 168 170 172 54 71 75 146 148 147 149 210 197 192 191 190 189 188 187 186 106 Mitogen-activated protein kinase 1
CMGC MAPK1 MK01_HUMAN 5V60A P28482 10 358 360.0 ACP:401 ATPlike Active DFGin 6.669 14.887 BLAminus -124.21, -175.27 60.56, 75.29 -91.11, 25.45 286.11, 68.09 -67.4, -23.76 in-in in 9.269 Saltbr-in 3.088 HRD-in -75.88, -52.24 69.24, 12.32 in-in-in SNCiii in-in ActLoopNT-in 2.951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.66, 171.23 APE9-dihe-na 66.7, 168.41 APE8-dihe-in -89.68, 141.19 APE8-rot-in 301.48 APE67-dihe-in -66.12, -19.67 -43.41, -50.15 APE12-dist-in 12.574 APE11-dist-in 11.086 APE10-dist-in 6.633 APE9-dist-in 2.987 None TPO185,PTR187 TPO185,PTR187 XRAY 2.18 0.193 0.226 A 356 349 0 0 0 0 [[25, 313]] 1.0 5v60 Homo sapiens CMGC_MAPK1_HUMAN CMGC 8.8e-86 293.8 1 301 301 166 167 168 170 172 54 71 75 146 148 147 149 210 197 192 191 190 189 188 187 186 106 Mitogen-activated protein kinase 1
CMGC MAPK12 MK12_HUMAN 1CM8A P53778 8 353 367.0 ANP:60400 ATPlike Active DFGin 6.965 14.774 BLAminus -109.08, -177.81 49.88, 82.62 -94.66, 21.96 279.65, 74.31 -61.38, -21.21 in-in in 9.0 Saltbr-in 2.777 HRD-in -80.35, -48.18 64.34, 20.91 in-in-in SNCiii in-in ActLoopNT-in 2.793 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.88, 159.85 APE9-dihe-na 73.62, 141.22 APE8-dihe-in -70.32, 134.6 APE8-rot-in 295.09 APE67-dihe-in -62.17, -12.08 -34.13, -61.33 APE12-dist-in 11.604 APE11-dist-in 10.956 APE10-dist-in 6.991 APE9-dist-in 3.072 None TPO183,PTR185 TPO183,PTR185 XRAY 2.4 0.232 0.283 A 367 329 6 0 0 0 [[27, 311]] 1.0 1cm8 Homo sapiens CMGC_MAPK12_HUMAN CMGC 5.6e-85 291.2 1 301 301 170 171 172 174 176 56 74 78 150 152 151 153 208 195 190 189 188 187 186 185 184 110 Mitogen-activated protein kinase 12
CMGC MAPK12 MK12_HUMAN 1CM8B P53778 8 353 367.0 ANP:61400 ATPlike Active DFGin 6.965 14.794 BLAminus -106.93, -177.79 50.51, 81.99 -94.3, 22.09 279.91, 74.94 -61.07, -21.75 in-in in 9.031 Saltbr-in 2.759 HRD-in -80.7, -47.04 63.03, 19.82 in-in-in SNCiii in-in ActLoopNT-in 2.817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.88, 160.62 APE9-dihe-na 73.12, 141.25 APE8-dihe-in -70.38, 133.34 APE8-rot-in 295.67 APE67-dihe-in -62.05, -11.85 -33.55, -61.0 APE12-dist-in 11.613 APE11-dist-in 10.95 APE10-dist-in 6.996 APE9-dist-in 3.048 None TPO183,PTR185 TPO183,PTR185 XRAY 2.4 0.232 0.283 B 367 329 6 0 0 0 [[27, 311]] 1.0 1cm8 Homo sapiens CMGC_MAPK12_HUMAN CMGC 5.6e-85 291.2 1 301 301 170 171 172 174 176 56 74 78 150 152 151 153 208 195 190 189 188 187 186 185 184 110 Mitogen-activated protein kinase 12
CMGC SRPK1 SRPK1_HUMAN 1WBPA Q96SB4 67 655 655.0 ADP:60950 ATPlike Active DFGin 6.093 14.484 BLAminus -120.66, 177.09 55.57, 73.12 -93.78, 28.92 297.48, 63.42 -60.8, -41.52 in-in in 9.616 Saltbr-in 3.534 HRD-in -64.25, -33.37 61.64, -4.85 in-in-in SNCiii in-in ActLoopNT-in 2.855 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.23, 175.25 APE9-dihe-na 64.87, 133.49 APE8-dihe-in -68.33, 140.58 APE8-rot-in 294.72 APE67-dihe-in -48.4, -19.96 -25.96, -79.02 APE12-dist-in 12.421 APE11-dist-in 10.401 APE10-dist-in 7.455 APE9-dist-in 2.973 None None None XRAY 2.4 0.228 0.247 A 397 350 22 0 0 0 [[80, 653]] 1.0 1wbp Homo sapiens CMGC_SRPK1_HUMAN CMGC 2e-139 469.9 1 301 301 496 497 498 500 502 109 124 128 210 212 211 213 533 521 516 515 514 513 512 511 510 166 SRSF protein kinase 1
OTHER HASPIN HASP_HUMAN 3DLZA Q8TF76 470 798 798.0 AMP:902 ATPlike Active DFGin 5.254 12.469 BLAminus -120.14, 174.05 73.32, 91.07 -105.92, 29.14 315.79, 130.04 -57.27, -36.15 in-in in 9.264 Saltbr-in 2.695 HRD-na-N -71.0, -49.07 68.99, 3.03 in-in-na SNCiia in-na ActLoopNT-in 2.821 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -122.28, 17.39 APE9-dihe-na -67.57, 157.85 APE8-dihe-na -149.51, 177.99 APE8-rot-na 58.52 APE67-dihe-na -159.03, 144.74 95.06, -6.22 APE12-dist-na 9.493 APE11-dist-na 13.466 APE10-dist-na 17.05 APE9-dist-na 12.819 None None None XRAY 1.85 0.167 0.216 A 357 329 0 0 0 0 [[484, 797]] 1.0 3dlz Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
OTHER TP53RK PRPK_HUMAN 6WQXC Q96S44 17 247 253.0 ANP:301 ATPlike Active DFGin 5.95 14.251 BLAminus -146.19, 177.42 55.9, 80.94 -109.82, 15.46 288.95, 83.65 -50.48, -21.92 in-in in 7.493 Saltbr-in 2.923 HRD-in -69.98, -47.0 96.04, -14.43 in-in-na SNCiia in-na ActLoopNT-in 2.804 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -67.54, -42.02 APE9-dihe-na -66.2, -40.19 APE8-dihe-na -55.79, -43.62 APE8-rot-na 183.14 APE67-dihe-na -65.72, -35.03 -54.78, -48.19 APE12-dist-na 16.724 APE11-dist-na 12.036 APE10-dist-na 14.577 APE9-dist-na 11.741 None None None XRAY 2.53 0.214 0.265 C 267 231 6 0 0 0 [[32, 253]] 1.0 6wqx Homo sapiens OTHER_TP53RK_HUMAN TP53RK 1.2e-114 387.3 1 224 224 182 183 184 186 188 60 84 88 159 161 160 162 199 205 200 199 198 197 196 195 194 114 EKC/KEOPS complex subunit TP53RK
OTHER TP53RK PRPK_HUMAN 6WQXD Q96S44 18 247 253.0 ANP:301 ATPlike Active DFGin 6.043 14.258 BLAminus -133.24, 171.19 66.42, 73.64 -108.34, 16.47 289.91, 91.17 -66.2, -15.73 in-in in 7.377 Saltbr-in 2.505 HRD-in -60.03, -49.96 100.64, -20.8 in-in-na SNCiia in-na ActLoopNT-in 2.816 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -66.35, -39.45 APE9-dihe-na -58.51, -49.84 APE8-dihe-na -58.36, -37.8 APE8-rot-na 168.78 APE67-dihe-na -71.45, -37.84 -63.19, -40.46 APE12-dist-na 16.676 APE11-dist-na 12.07 APE10-dist-na 14.499 APE9-dist-na 11.469 None None None XRAY 2.53 0.214 0.265 D 267 230 6 0 0 0 [[32, 253]] 1.0 6wqx Homo sapiens OTHER_TP53RK_HUMAN TP53RK 1.2e-114 387.3 1 224 224 182 183 184 186 188 60 84 88 159 161 160 162 199 205 200 199 198 197 196 195 194 114 EKC/KEOPS complex subunit TP53RK
OTHER WNK3 WNK3_HUMAN 5O26A Q9BYP7 135 414 1800.0 ANP:501 ATPlike Active DFGin 6.954 12.201 BLAminus -125.28, -164.72 58.79, 65.89 -88.2, 18.66 305.61, 176.73 -69.56, -20.03 na-na na 15.898 Saltbr-na 999.0 HRD-in -66.1, -48.87 66.45, 11.22 na-in-in SNCaii in-in ActLoopNT-in 3.021 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.2, 167.0 APE9-dihe-na 127.63, -163.54 APE8-dihe-in -104.53, 119.98 APE8-rot-in 309.3 APE67-dihe-in -64.09, -19.44 -52.49, -34.59 APE12-dist-in 8.873 APE11-dist-in 11.829 APE10-dist-in 6.326 APE9-dist-in 3.706 None SEP304,SEP308 SEP304,SEP308 XRAY 2.379 0.231 0.278 A 284 273 7 0 0 0 [[146, 405]] 1.0 5o26 Homo sapiens OTHER_WNK3_HUMAN WNK 2.6e-178 596.6 1 260 260 293 294 295 297 299 176 194 198 272 274 273 275 330 319 314 313 312 311 310 309 308 228 Serine/threonine-protein kinase WNK3
OTHER WNK3 WNK3_HUMAN 5O26B Q9BYP7 136 413 1800.0 ANP:501 ATPlike Active DFGin 7.182 12.078 BLAminus -111.0, -167.63 57.49, 63.76 -86.7, 17.71 307.84, 173.05 -70.2, -27.96 na-na na 15.641 Saltbr-na 999.0 HRD-in -66.99, -53.82 74.22, 8.4 na-in-in SNCaii in-in ActLoopNT-in 3.073 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.41, 145.08 APE9-dihe-na 140.9, -162.45 APE8-dihe-in -99.46, 120.61 APE8-rot-in 305.94 APE67-dihe-in -65.71, -19.72 -54.06, -31.08 APE12-dist-in 8.136 APE11-dist-in 11.827 APE10-dist-in 6.044 APE9-dist-in 3.51 None SEP304,SEP308 SEP304,SEP308 XRAY 2.379 0.231 0.278 B 284 267 11 0 0 0 [[146, 405]] 1.0 5o26 Homo sapiens OTHER_WNK3_HUMAN WNK 2.6e-178 596.6 1 260 260 293 294 295 297 299 176 194 198 272 274 273 275 330 319 314 313 312 311 310 309 308 228 Serine/threonine-protein kinase WNK3
STE PAK3 PAK3_HUMAN 6FD3A O75914 261 556 559.0 ADP:60603 ATPlike Active DFGin 5.952 14.149 BLAminus -133.62, -174.01 64.9, 77.07 -96.85, 18.52 289.09, 83.73 -72.71, -11.5 in-in in 8.938 Saltbr-in 2.761 HRD-in -71.32, -50.63 74.19, 1.63 in-in-in SNCiii in-in ActLoopNT-in 2.913 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.75, 147.44 APE9-dihe-na 132.72, -161.48 APE8-dihe-in -114.41, 121.22 APE8-rot-in 305.33 APE67-dihe-in -64.48, -19.99 -44.4, -48.2 APE12-dist-in 8.849 APE11-dist-in 11.358 APE10-dist-in 5.576 APE9-dist-in 3.34 A537D None T8L436 XRAY 1.52 0.176 0.19 A 300 296 0 0 0 0 [[283, 534]] 1.0 6fd3 Homo sapiens STE_PAK3_HUMAN STE 1.1e-94 322.5 1 257 257 419 420 421 423 425 312 328 332 399 401 400 402 459 447 442 441 440 439 438 437 436 358 Serine/threonine-protein kinase PAK 3
STE PAK4 PAK4_HUMAN 4FIFA O96013 296 589 591.0 ANP:1000 ATPlike Active DFGin 6.132 13.879 BLAminus -134.27, -172.64 55.78, 65.69 -91.22, 11.11 299.57, 98.92 -61.37, -20.58 in-in in 7.046 Saltbr-in 3.112 HRD-in -73.18, -47.2 74.11, -8.39 in-in-in SNCiii in-in ActLoopNT-in 2.852 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.08, 134.89 APE9-dihe-na 136.18, -173.61 APE8-dihe-in -102.98, 119.55 APE8-rot-in 312.46 APE67-dihe-in -69.75, -26.2 -30.93, -52.34 APE12-dist-in 9.318 APE11-dist-in 11.709 APE10-dist-in 5.875 APE9-dist-in 3.299 None SEP474 SEP474 XRAY 2.6 0.207 0.227 A 346 294 0 0 0 0 [[321, 572]] 1.0 4fif Homo sapiens STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 4FIFB O96013 297 589 591.0 ANP:1000 ATPlike Active DFGin 5.899 13.85 BLAminus -129.09, -170.37 52.27, 68.51 -93.51, 10.45 301.97, 96.23 -63.09, -15.01 in-in in 7.007 Saltbr-in 3.167 HRD-in -65.39, -48.9 75.1, -7.5 in-in-in SNCiii in-in ActLoopNT-in 2.801 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.88, 134.77 APE9-dihe-na 136.42, -174.06 APE8-dihe-in -101.96, 121.94 APE8-rot-in 314.36 APE67-dihe-in -72.79, -21.56 -33.03, -50.98 APE12-dist-in 9.238 APE11-dist-in 11.712 APE10-dist-in 5.886 APE9-dist-in 3.335 None SEP474 SEP474 XRAY 2.6 0.207 0.227 B 346 293 0 0 0 0 [[321, 572]] 1.0 4fif Homo sapiens STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 4JDIA O96013 300 589 591.0 ANP:1000 ATPlike Active DFGin 6.291 14.47 BLAminus -134.26, 177.87 63.72, 71.58 -94.6, 13.78 289.77, 79.71 -54.15, -28.77 in-in in 6.959 Saltbr-in 2.737 HRD-in -72.82, -49.09 73.48, 2.76 in-in-in SNCiii in-in ActLoopNT-in 2.829 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.62, 145.0 APE9-dihe-na 130.41, -160.49 APE8-dihe-in -120.53, 123.45 APE8-rot-in 305.94 APE67-dihe-in -63.49, -22.51 -36.89, -56.07 APE12-dist-in 8.769 APE11-dist-in 11.535 APE10-dist-in 5.874 APE9-dist-in 3.327 None SEP474 SEP474 XRAY 1.85 0.194 0.233 A 346 290 0 0 0 0 [[321, 572]] 1.0 4jdi Homo sapiens STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 5UPKB O96013 300 588 591.0 ANP:60600 ATPlike Active DFGin 6.272 14.139 BLAminus -132.3, -169.35 61.71, 61.5 -87.86, 7.28 293.59, 93.96 -55.36, -28.3 in-in in 7.077 Saltbr-in 3.329 HRD-in -65.35, -49.16 70.36, 11.54 in-in-in SNCiii in-in ActLoopNT-in 2.997 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.55, 149.52 APE9-dihe-na 120.09, -163.11 APE8-dihe-in -119.51, 121.87 APE8-rot-in 313.98 APE67-dihe-in -69.89, -18.98 -32.47, -57.41 APE12-dist-in 8.623 APE11-dist-in 11.267 APE10-dist-in 5.616 APE9-dist-in 3.426 None SEP474 SEP474 XRAY 2.4 0.22 0.264 B 346 289 0 0 0 0 [[321, 572]] 1.0 5upk Homo sapiens STE_PAK4_HUMAN STE 3.1e-88 301.5 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 7S46A O96013 300 589 591.0 ANP:600 ATPlike Active DFGin 9.021 14.349 BLAminus -133.61, -177.07 54.75, 76.68 -92.18, 14.46 286.49, 80.35 -59.04, -19.55 in-in in 7.534 Saltbr-in 2.867 HRD-in -69.43, -50.5 76.76, 2.96 in-in-in SNCiii in-in ActLoopNT-in 2.922 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.73, 132.58 APE9-dihe-na 145.82, -167.86 APE8-dihe-in -110.13, 128.57 APE8-rot-in 305.26 APE67-dihe-in -70.79, -21.11 -38.41, -55.32 APE12-dist-in 9.02 APE11-dist-in 11.537 APE10-dist-in 5.793 APE9-dist-in 3.286 D440N,S474E None None XRAY 2.1 0.182 0.22 A 346 290 0 0 0 0 [[321, 572]] 1.0 7s46 Homo sapiens STE_PAK4_HUMAN STE 5.5e-87 297.4 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE PAK4 PAK4_HUMAN 7S47A O96013 300 589 591.0 ANP:600 ATPlike Active DFGin 9.217 14.646 BLAminus -126.8, -179.34 54.51, 73.91 -89.97, 15.41 285.81, 78.05 -59.21, -18.99 in-in in 7.79 Saltbr-in 2.931 HRD-in -66.64, -48.47 70.7, 6.89 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.53, 138.41 APE9-dihe-na 140.72, -164.27 APE8-dihe-in -114.61, 124.35 APE8-rot-in 304.9 APE67-dihe-in -66.22, -20.32 -36.39, -56.83 APE12-dist-in 9.039 APE11-dist-in 11.45 APE10-dist-in 5.747 APE9-dist-in 3.401 D440N,S474E None None XRAY 2.0 0.196 0.237 A 383 290 0 0 0 0 [[321, 572]] 1.0 7s47 Homo sapiens STE_PAK4_HUMAN STE 7.5e-87 297.0 5 257 253 457 458 459 461 463 350 366 370 437 439 438 440 497 485 480 479 478 477 476 475 474 396 Serine/threonine-protein kinase PAK 4
STE STK24 STK24_HUMAN 3A7JA Q9Y6E0 25 311 443.0 ADP:60500 ATPlike Active DFGin 6.747 14.583 BLAminus -138.67, 168.25 71.5, 79.52 -101.19, 20.06 287.01, 95.64 -64.31, -27.68 in-in in 8.53 Saltbr-in 2.552 HRD-in -69.86, -43.49 67.32, -1.05 in-in-in SNCiii in-in ActLoopNT-in 2.741 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.28, 158.62 APE9-dihe-na 130.53, -164.99 APE8-dihe-in -116.23, 120.86 APE8-rot-in 304.02 APE67-dihe-in -60.63, -23.79 -34.15, -55.13 APE12-dist-in 8.296 APE11-dist-in 11.11 APE10-dist-in 5.251 APE9-dist-in 3.288 None TPO190 TPO190 XRAY 1.5 0.191 0.21 A 303 287 0 0 0 0 [[36, 286]] 1.0 3a7j Homo sapiens STE_STK24_HUMAN STE 3.6e-100 340.5 1 257 257 173 174 175 177 179 65 82 86 153 155 154 156 213 201 196 195 194 193 192 191 190 112 Serine/threonine-protein kinase 24
STE STK24 STK24_HUMAN 4QMLA Q9Y6E0 30 310 443.0 ANP:60403 ATPlike Active DFGin 6.598 15.178 BLAminus -130.38, 172.22 70.9, 79.24 -104.53, 20.01 285.96, 83.16 -61.35, -25.21 in-in in 9.065 Saltbr-in 2.927 HRD-in -70.82, -51.82 74.23, -2.97 in-in-in SNCiii in-in ActLoopNT-in 2.848 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.04, 155.96 APE9-dihe-na 125.92, -168.67 APE8-dihe-in -115.63, 119.31 APE8-rot-in 310.36 APE67-dihe-in -60.1, -29.49 -47.33, -42.77 APE12-dist-in 8.276 APE11-dist-in 11.051 APE10-dist-in 5.558 APE9-dist-in 3.386 None TPO190 TPO190 XRAY 1.882 0.19 0.23 A 310 281 0 0 0 0 [[36, 286]] 1.0 4qml Homo sapiens STE_STK24_HUMAN STE 3.9e-100 340.4 1 257 257 173 174 175 177 179 65 82 86 153 155 154 156 213 201 196 195 194 193 192 191 190 112 Serine/threonine-protein kinase 24
STE TAOK3 TAOK3_HUMAN 6BDNA Q9H2K8 8 314 898.0 ADP:404 ATPlike Active DFGin 6.771 13.825 BLAminus -136.73, -179.28 62.01, 80.15 -97.31, 23.85 293.38, 102.08 -68.85, -11.35 in-in in 8.485 Saltbr-in 2.682 HRD-in -74.02, -52.69 74.7, -5.2 in-in-in SNCiii in-in ActLoopNT-in 2.797 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.94, 158.28 APE9-dihe-na 130.64, -172.75 APE8-dihe-in -113.55, 120.19 APE8-rot-in 301.22 APE67-dihe-in -62.99, -26.26 -46.03, -46.8 APE12-dist-in 8.28 APE11-dist-in 11.04 APE10-dist-in 5.18 APE9-dist-in 3.383 R2A,K3A None None XRAY 1.5 0.187 0.214 A 320 307 0 0 0 0 [[24, 277]] 1.0 6bdn Homo sapiens STE_TAOK3_HUMAN STE 6.3e-90 307.0 4 257 254 164 165 166 168 170 53 72 76 144 146 145 147 203 188 183 182 181 180 179 178 177 102 Serine/threonine-protein kinase TAO3
STE TNIK TNIK_HUMAN 7XZRB Q9UKE5 12 312 1360.0 ANP:1401 ATPlike Active DFGin 6.439 15.163 BLAminus -131.61, 176.54 70.33, 83.31 -101.27, 21.61 286.01, 77.74 -67.8, -30.96 in-in in 9.126 Saltbr-in 2.582 HRD-in -64.36, -58.64 76.74, 3.35 in-in-in SNCiii in-in ActLoopNT-in 2.931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.27, 150.43 APE9-dihe-na 126.35, -168.16 APE8-dihe-in -105.07, 123.33 APE8-rot-in 308.43 APE67-dihe-in -61.4, -25.19 -44.62, -54.45 APE12-dist-in 8.7 APE11-dist-in 11.705 APE10-dist-in 6.078 APE9-dist-in 3.705 None TPO181,TPO187 TPO181,TPO187 XRAY 2.26 0.184 0.226 B 306 301 0 0 0 0 [[25, 289]] 1.0 7xzr Homo sapiens STE_TNIK_HUMAN STE 3e-105 357.1 1 257 257 170 171 172 174 176 54 69 73 150 152 151 153 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
TKL BMPR2 BMPR2_HUMAN 3G2FA Q13873 197 510 1038.0 ADP:900 ATPlike Active DFGin 6.957 13.944 BLAminus -131.62, -179.2 66.08, 79.87 -102.79, 27.43 304.26, 96.52 -59.99, -25.3 in-in in 8.107 Saltbr-in 2.757 HRD-in -69.81, -50.66 82.19, -10.63 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.1, -22.11 APE9-dihe-na -73.96, -168.61 APE8-dihe-in -80.16, 127.03 APE8-rot-in 308.56 APE67-dihe-in -65.91, -22.58 -59.75, -41.5 APE12-dist-in 11.403 APE11-dist-in 12.63 APE10-dist-in 7.026 APE9-dist-in 4.033 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 A 336 305 9 0 0 9 [[202, 503]] 1.0 3g2f Homo sapiens TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2 266 265 350 351 352 354 356 230 243 247 330 332 331 333 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
TKL BMPR2 BMPR2_HUMAN 3G2FB Q13873 198 513 1038.0 ADP:900 ATPlike Active DFGin 6.968 14.008 BLAminus -149.7, 179.95 61.07, 87.18 -102.54, 11.93 293.8, 112.47 -56.7, -17.91 in-in in 8.065 Saltbr-in 2.732 HRD-in -73.22, -52.25 87.7, -10.0 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.94, -26.41 APE9-dihe-na -71.73, -175.39 APE8-dihe-in -71.07, 133.08 APE8-rot-in 315.55 APE67-dihe-in -68.07, -13.93 -56.75, -42.89 APE12-dist-in 11.194 APE11-dist-in 12.108 APE10-dist-in 6.494 APE9-dist-in 3.722 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 B 336 303 13 0 0 13 [[202, 503]] 1.0 3g2f Homo sapiens TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2 266 265 350 351 352 354 356 230 243 247 330 332 331 333 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
TKL BMPR2 BMPR2_HUMAN 6UNPB Q13873 197 509 1038.0 ADP:601 ATPlike Active DFGin 6.917 14.051 BLAminus -140.56, 176.5 63.35, 76.41 -96.26, 25.8 302.12, 104.12 -61.08, -20.73 in-in in 7.904 Saltbr-in 2.865 HRD-in -75.95, -48.17 78.17, -6.91 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.29, -9.38 APE9-dihe-na -69.43, -161.26 APE8-dihe-in -89.59, 127.34 APE8-rot-in 301.19 APE67-dihe-in -48.39, -33.11 -62.11, -43.63 APE12-dist-in 12.009 APE11-dist-in 12.508 APE10-dist-in 7.099 APE9-dist-in 4.016 D485G None CAS288,CAS397,CAS496 XRAY 2.3 0.19 0.211 B 363 303 10 0 0 8 [[202, 503]] 1.0 6unp Homo sapiens TKL_BMPR2_HUMAN TKL 1.1e-74 257.3 2 266 265 350 351 352 354 356 230 243 247 330 332 331 333 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
TKL IRAK4 IRAK4_HUMAN 2OIDD Q9NWZ3 164 459 460.0 ANP:4 ATPlike Active DFGin 6.56 13.972 BLAminus -129.12, -177.03 59.13, 109.88 -131.38, 17.54 304.54, 87.5 -68.37, -4.63 in-in in 8.15 Saltbr-in 3.52 HRD-in -75.54, -51.34 70.58, 2.03 in-in-in SNCiii in-in ActLoopNT-in 2.765 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.72, 147.52 APE9-dihe-na 139.0, -173.6 APE8-dihe-in -107.1, 118.58 APE8-rot-in 309.04 APE67-dihe-in -62.68, -15.82 -47.4, -49.91 APE12-dist-in 9.75 APE11-dist-in 11.44 APE10-dist-in 5.928 APE9-dist-in 3.97 None TPO342,TPO345,SEP346 TPO342,TPO345,SEP346 XRAY 2.3 0.244 0.295 D 301 277 19 0 0 3 [[183, 456]] 1.0 2oid Homo sapiens TKL_IRAK4_HUMAN TKL 4.1e-84 288.2 5 266 262 328 329 330 332 334 213 233 237 308 310 309 311 369 358 353 352 351 350 349 348 347 263 Interleukin-1 receptor-associated kinase 4
TKL LIMK1 LIMK1_HUMAN 5L6WL P53667 330 633 647.0 AGS:60701 ATPlike Active DFGin 6.235 14.337 BLAminus -131.64, -166.52 46.75, 81.93 -92.83, 15.71 304.28, 98.92 -42.69, -49.84 in-in in 7.664 Saltbr-in 2.67 HRD-in -78.67, -47.86 69.62, -13.12 in-in-in SNCiii in-in ActLoopNT-in 3.066 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -134.6, 165.2 APE9-dihe-na 100.19, 162.86 APE8-dihe-in -63.5, 131.5 APE8-rot-na 185.1 APE67-dihe-in -61.44, -31.47 -69.46, -29.71 APE12-dist-in 9.116 APE11-dist-in 11.134 APE10-dist-in 5.438 APE9-dist-in 3.762 None None None XRAY 2.53 0.229 0.284 L 310 288 16 0 0 16 [[339, 606]] 1.0 5l6w Homo sapiens TKL_LIMK1_HUMAN TKL 4.5e-77 265.1 3 266 264 477 478 479 481 483 368 384 388 457 459 458 460 531 519 514 513 512 511 510 509 508 414 LIM domain kinase 1
TKL LIMK1 LIMK1_HUMAN 5HVKA P53667 329 634 647.0 ANP:61001 ATPlike Active DFGin 6.405 13.646 BLAminus -145.46, 176.84 65.07, 82.49 -109.26, 24.73 304.62, 92.73 -71.79, -22.73 in-in in 7.795 Saltbr-in 3.159 HRD-in -70.8, -44.42 59.42, 18.52 in-in-in SNCiii in-in ActLoopNT-in 3.324 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -139.63, 151.17 APE9-dihe-na 143.88, 171.7 APE8-dihe-in -71.51, 120.27 APE8-rot-na 199.31 APE67-dihe-in -66.59, -36.22 -54.03, -34.34 APE12-dist-in 9.301 APE11-dist-in 11.081 APE10-dist-in 5.636 APE9-dist-in 3.574 D460N TPO508 TPO508 XRAY 3.5 0.275 0.31 A 315 293 13 0 0 13 [[339, 606]] 1.0 5hvk Homo sapiens TKL_LIMK1_HUMAN TKL 3e-76 262.4 3 266 264 477 478 479 481 483 368 384 388 457 459 458 460 531 519 514 513 512 511 510 509 508 414 LIM domain kinase 1
TKL LRRK2 LRRK2_HUMAN 8FO9A Q5S007 1329 2527 2527.0 ATP:2602 ATPlike Active DFGin 6.273 13.41 BLAminus -138.23, -175.7 59.6, 64.71 -84.85, 53.99 305.84, 101.34 -78.49, -28.55 in-in in 7.88 Saltbr-in 2.735 HRD-in -107.83, -47.31 66.25, 1.81 in-in-in SNCiii in-in ActLoopNT-in 3.031 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.21, 156.34 APE9-dihe-na 139.24, 152.96 APE8-dihe-in -67.96, 127.7 APE8-rot-in 305.42 APE67-dihe-inflip 98.56, -16.69 -58.5, 136.92 APE12-dist-in 9.183 APE11-dist-in 11.487 APE10-dist-in 6.004 APE9-dist-in 3.816 None None None EM 3.48 999.0 999.0 A 2527 1173 0 0 0 0 [[1875, 2134]] 1.0 8fo9 Homo sapiens TKL_LRRK2_HUMAN TKL 3.8e-57 200.3 5 266 262 2016 2017 2018 2020 2022 1906 1920 1924 1991 1993 1992 1994 2055 2042 2037 2036 2035 2034 2033 2032 2031 1948 Leucine-rich repeat serine/threonine-protein kinase 2
TKL LRRK2 LRRK2_HUMAN 8FO9C Q5S007 1329 2527 2527.0 ATP:2602 ATPlike Active DFGin 6.275 13.405 BLAminus -138.14, -175.77 59.5, 64.85 -84.95, 53.97 305.9, 101.31 -78.52, -28.52 in-in in 7.883 Saltbr-in 2.729 HRD-in -108.59, -47.2 66.33, 1.76 in-in-in SNCiii in-in ActLoopNT-in 3.008 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.94, 156.21 APE9-dihe-na 139.37, 152.96 APE8-dihe-in -67.92, 127.71 APE8-rot-in 305.58 APE67-dihe-inflip 98.46, -16.81 -58.61, 136.94 APE12-dist-in 9.177 APE11-dist-in 11.503 APE10-dist-in 6.012 APE9-dist-in 3.804 None None None EM 3.48 999.0 999.0 C 2527 1173 0 0 0 0 [[1875, 2134]] 1.0 8fo9 Homo sapiens TKL_LRRK2_HUMAN TKL 3.8e-57 200.3 5 266 262 2016 2017 2018 2020 2022 1906 1920 1924 1991 1993 1992 1994 2055 2042 2037 2036 2035 2034 2033 2032 2031 1948 Leucine-rich repeat serine/threonine-protein kinase 2
TKL TGFBR2 TGFR2_HUMAN 5E92A P37173 240 543 567.0 ANP:601 ATPlike Active DFGin 7.396 13.303 BLAminus -134.93, 178.1 63.07, 87.04 -105.26, 16.76 300.78, 96.96 -60.58, -26.14 in-in in 7.67 Saltbr-in 2.752 HRD-in -64.87, -46.8 71.14, -4.53 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.21, 144.17 APE9-dihe-na 126.96, -149.92 APE8-dihe-in -116.55, 119.38 APE8-rot-in 300.41 APE67-dihe-in -54.91, -33.03 -42.96, -45.47 APE12-dist-in 11.788 APE11-dist-in 12.049 APE10-dist-in 6.089 APE9-dist-in 3.401 E431A,R433A,E485A,K488A,R493A,R495A None None XRAY 2.08 0.204 0.231 A 316 298 6 0 0 0 [[244, 540]] 1.0 5e92 Homo sapiens TKL_TGFBR2_HUMAN TKL 1.9e-77 266.3 2 266 265 396 397 398 400 402 277 290 294 376 378 377 379 446 428 423 422 421 420 419 418 417 326 TGF-beta receptor type-2
TYR EGFR EGFR_HUMAN 2ITXA P00533 697 1019 1210.0 ANP:2020 ATPlike Active DFGin 5.874 15.737 BLAminus -136.31, -171.94 65.34, 93.22 -111.54, 18.75 298.27, 92.75 -59.44, 2.06 in-in in 9.241 Saltbr-in 3.583 HRD-in -62.41, -44.72 61.37, 7.79 in-in-in SNCiii in-in ActLoopNT-in 2.642 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -78.73, 124.39 APE9-dihe-in -125.4, 144.12 APE8-dihe-in -79.64, 94.32 APE8-rot-na 30.37 APE67-dihe-in -65.37, -0.17 -61.69, -47.61 APE12-dist-na 11.888 APE11-dist-na 10.151 APE10-dist-na 11.134 APE9-dist-in 7.058 None None None XRAY 2.98 0.191 0.261 A 327 307 4 0 0 4 [[712, 970]] 1.0 2itx Homo sapiens TYR_EGFR_HUMAN TYR 1e-87 299.8 3 259 257 854 855 856 858 860 745 762 766 834 836 835 837 896 884 879 878 877 876 875 874 873 791 Epidermal growth factor receptor
TYR FGFR1 FGFR1_HUMAN 3GQIA P11362 464 770 822.0 ACP:775 ATPlike Active DFGin 6.466 13.946 BLAminus -126.61, -175.83 60.19, 72.36 -91.08, 18.42 288.73, 91.63 -64.67, -15.4 in-in in 7.751 Saltbr-in 2.69 HRD-in -77.5, -49.87 72.48, -2.68 in-in-in SNCiii in-in ActLoopNT-in 2.961 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -58.96, 135.34 APE9-dihe-in -149.19, 136.62 APE8-dihe-in -75.51, 66.48 APE8-rot-na 33.4 APE67-dihe-in -65.08, -11.82 -44.91, -41.18 APE12-dist-na 14.083 APE11-dist-na 11.258 APE10-dist-na 10.128 APE9-dist-in 7.137 C488A,Y583F,C584S,Y585F PTR653,PTR654,PTR766 PTR653,PTR654,PTR766 XRAY 2.5 0.249 0.289 A 326 307 0 0 0 0 [[478, 756]] 1.0 3gqi Homo sapiens TYR_FGFR1_HUMAN TYR 1.7e-104 354.6 1 260 260 640 641 642 644 646 514 531 535 620 622 621 623 682 670 665 664 663 662 661 660 659 562 Fibroblast growth factor receptor 1
TYR FGFR2 FGFR2_HUMAN 2PVFA P21802 467 765 821.0 ACP:60300 ATPlike Active DFGin 6.048 13.821 BLAminus -138.88, -175.17 54.67, 80.46 -90.11, 24.33 291.08, 76.38 -54.38, -36.38 in-in in 7.913 Saltbr-in 2.769 HRD-in -85.37, -48.4 70.03, 0.26 in-in-in SNCiii in-in ActLoopNT-in 2.879 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -86.94, 115.27 APE9-dihe-in -125.87, 160.91 APE8-dihe-in -74.41, 68.1 APE8-rot-na 35.92 APE67-dihe-in -70.82, -9.54 -47.44, -41.99 APE12-dist-na 15.14 APE11-dist-na 11.649 APE10-dist-na 11.604 APE9-dist-in 7.168 C491A PTR586,PTR656,PTR657 PTR586,PTR656,PTR657 XRAY 1.8 0.251 0.265 A 334 288 11 0 0 0 [[481, 759]] 1.0 2pvf Homo sapiens TYR_FGFR2_HUMAN TYR 2.2e-104 354.3 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 3CLYA P21802 468 772 821.0 ACP:61803 ATPlike Active DFGin 6.229 14.183 BLAminus -138.78, -172.76 51.4, 79.79 -91.29, 32.46 290.47, 75.81 -61.86, -29.26 in-in in 7.661 Saltbr-in 2.621 HRD-in -89.86, -45.92 68.93, -0.84 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -72.79, 139.96 APE9-dihe-in -131.36, 152.18 APE8-dihe-in -76.17, 66.16 APE8-rot-na 37.1 APE67-dihe-in -66.78, -6.73 -47.95, -40.48 APE12-dist-na 13.253 APE11-dist-na 10.402 APE10-dist-na 11.097 APE9-dist-in 6.913 C491A PTR656,PTR657 PTR656,PTR657 XRAY 2.0 0.216 0.247 A 334 291 14 0 0 0 [[481, 759]] 1.0 3cly Homo sapiens TYR_FGFR2_HUMAN TYR 2.2e-104 354.3 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 5EG3A P21802 466 774 821.0 ACP:60801 ATPlike Active DFGin 6.034 13.825 BLAminus -138.71, -166.61 47.53, 87.44 -100.17, 28.73 285.85, 82.29 -77.8, -14.99 in-in in 8.045 Saltbr-in 2.941 HRD-in -83.82, -45.21 62.18, 9.75 in-in-in SNCiii in-in ActLoopNT-in 2.991 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -66.56, 121.06 APE9-dihe-in -128.9, 119.34 APE8-dihe-in -79.6, 67.11 APE8-rot-na 30.51 APE67-dihe-in -77.81, 0.08 -48.0, -39.27 APE12-dist-na 13.558 APE11-dist-na 10.078 APE10-dist-na 8.259 APE9-dist-in 7.021 Y466F,C491A,E565A,Y586L,Y588P,Y656F,Y657F,K659E PTR769 PTR769 XRAY 2.606 0.191 0.237 A 334 302 7 0 0 0 [[481, 759]] 1.0 5eg3 Homo sapiens TYR_FGFR2_HUMAN TYR 2.3e-101 344.4 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR3 FGFR3_HUMAN 4K33A P22607 459 755 806.0 ACP:801 ATPlike Active DFGin 6.252 13.787 BLAminus -133.88, -173.58 58.49, 82.81 -96.43, 27.55 291.81, 80.95 -59.32, -31.32 in-in in 8.211 Saltbr-in 2.895 HRD-in -87.09, -47.34 67.06, 1.63 in-in-in SNCiii in-in ActLoopNT-in 2.99 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -55.89, 133.11 APE9-dihe-in -125.43, 130.21 APE8-dihe-in -78.76, 72.58 APE8-rot-na 29.71 APE67-dihe-in -71.45, -4.47 -50.14, -48.75 APE12-dist-na 13.31 APE11-dist-na 9.602 APE10-dist-na 8.305 APE9-dist-in 6.873 C482A,C582S,K650E None None XRAY 2.341 0.181 0.228 A 325 293 4 0 0 0 [[472, 750]] 1.0 4k33 Homo sapiens TYR_FGFR3_HUMAN TYR 2.3e-104 354.2 1 260 260 634 635 636 638 640 508 525 529 614 616 615 617 676 664 659 658 657 656 655 654 653 556 Fibroblast growth factor receptor 3
TYR INSR INSR_HUMAN 3BU5A P06213 1014 1310 1382.0 ATP:60300 ATPlike Active DFGin 6.659 13.934 BLAminus -128.64, -166.6 44.54, 89.54 -102.81, 23.91 295.82, 99.34 -57.5, -34.18 in-in in 8.261 Saltbr-in 3.13 HRD-in -68.86, -51.91 77.02, -10.33 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -82.0, 102.51 APE9-dihe-in -127.85, 151.44 APE8-dihe-in -79.76, 69.1 APE8-rot-na 32.47 APE67-dihe-in -66.77, -8.03 -57.27, -41.89 APE12-dist-na 15.937 APE11-dist-na 11.724 APE10-dist-na 11.3 APE9-dist-in 7.401 C1008S PTR1185,PTR1189,PTR1190 PTR1185,PTR1189,PTR1190 XRAY 2.1 0.196 0.239 A 306 294 3 0 0 0 [[1023, 1292]] 1.0 3bu5 Homo sapiens TYR_INSR_HUMAN TYR 1.3e-96 328.8 1 260 260 1176 1177 1178 1180 1182 1057 1074 1078 1156 1158 1157 1159 1218 1206 1201 1200 1199 1198 1197 1196 1195 1104 Insulin receptor
TYR INSR INSR_HUMAN 4XLVA P06213 1001 1310 1382.0 ACP:61301 ATPlike Active DFGin 6.357 13.404 BLAminus -129.47, -169.61 59.33, 81.3 -99.86, 10.75 301.2, 100.62 -50.37, -35.15 in-in in 8.175 Saltbr-in 2.441 HRD-in -74.09, -41.95 72.32, -7.69 in-in-in SNCiii in-in ActLoopNT-in 3.029 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -31.8, 98.01 APE9-dihe-in -128.43, 131.43 APE8-dihe-in -62.62, 111.75 APE8-rot-na 18.22 APE67-dihe-in -71.49, -19.39 -64.21, -23.54 APE12-dist-na 14.741 APE11-dist-na 10.551 APE10-dist-na 11.027 APE9-dist-in 6.615 Y992F,C1008S PTR999,PTR1185,PTR1189,PTR1190 PTR999,PTR1185,PTR1189,PTR1190 XRAY 2.3 0.207 0.266 A 328 310 0 0 0 0 [[1023, 1292]] 1.0 4xlv Homo sapiens TYR_INSR_HUMAN TYR 1.7e-96 328.5 1 260 260 1176 1177 1178 1180 1182 1057 1074 1078 1156 1158 1157 1159 1218 1206 1201 1200 1199 1198 1197 1196 1195 1104 Insulin receptor
TYR JAK1-2 JAK1_HUMAN 6C7YA P23458 869 1153 1154.0 ADP:61201 ATPlike Active DFGin 6.032 13.967 BLAminus -134.15, -164.18 58.49, 84.96 -109.28, 28.04 298.78, 97.45 -66.39, -27.05 in-in in 8.311 Saltbr-in 2.732 HRD-in -67.59, -46.53 68.25, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -72.91, 151.36 APE9-dihe-in -137.76, 143.32 APE8-dihe-in -74.71, 81.76 APE8-rot-na 30.49 APE67-dihe-in -79.4, -2.38 -65.2, -24.66 APE12-dist-na 12.972 APE11-dist-na 8.02 APE10-dist-na 10.344 APE9-dist-in 6.316 None PTR1035 PTR1035 XRAY 2.499 0.21 0.241 A 286 273 12 0 0 0 [[583, 847], [875, 1151]] 2.0 6c7y Homo sapiens TYR_JAK1-2_HUMAN TYR 1.8e-87 298.9 2 259 258 1020 1021 1022 1024 1026 908 925 929 1000 1002 1001 1003 1063 1051 1046 1045 1044 1043 1042 1041 1040 957 Tyrosine-protein kinase JAK1
TYR LCK LCK_HUMAN 1QPCA P06239 231 502 509.0 ANP:904 ATPlike Active DFGin 6.61 14.416 BLAminus -133.73, 179.02 58.4, 83.48 -97.79, 21.23 295.19, 99.8 -60.65, -35.99 in-in in 8.702 Saltbr-in 3.096 HRD-in -103.01, -49.32 74.3, -4.36 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -120.97, 142.08 APE9-dihe-in -126.79, 156.19 APE8-dihe-in -63.13, 117.89 APE8-rot-na 333.56 APE67-dihe-in -65.85, -20.96 -57.94, -43.39 APE12-dist-na 14.856 APE11-dist-na 10.005 APE10-dist-na 12.788 APE9-dist-in 6.784 None PTR394 PTR394 XRAY 1.6 0.2 0.23 A 279 272 0 0 0 0 [[245, 496]] 1.0 1qpc Homo sapiens TYR_LCK_HUMAN TYR 1.4e-94 322.2 1 260 260 381 382 383 385 387 273 288 292 361 363 362 364 422 410 405 404 403 402 401 400 399 317 Tyrosine-protein kinase Lck
TYR SYK KSYK_HUMAN 4FL1A P43405 363 635 635.0 ANP:701 ATPlike Active DFGin 6.669 15.063 BLAminus -122.6, -175.53 56.16, 78.38 -92.62, 24.67 287.04, 93.75 -57.67, -38.36 in-in in 8.059 Saltbr-in 2.683 HRD-in -76.27, -50.57 71.77, 3.28 in-in-in SNCiii in-in ActLoopNT-in 2.976 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -89.55, 85.11 APE9-dihe-in -99.28, 138.37 APE8-dihe-in -79.64, 69.72 APE8-rot-na 29.68 APE67-dihe-in -60.65, -16.95 -44.16, -41.68 APE12-dist-na 13.816 APE11-dist-na 10.806 APE10-dist-na 10.412 APE9-dist-in 7.132 None None None XRAY 1.79 0.197 0.225 A 291 268 5 0 0 0 [[370, 628]] 1.0 4fl1 Homo sapiens TYR_SYK_HUMAN TYR 5.5e-90 307.1 5 260 256 511 512 513 515 517 402 420 424 491 493 492 494 554 542 537 536 535 534 533 532 531 449 Tyrosine-protein kinase SYK
TYR TNK2 ACK1_HUMAN 1U54B Q07912 117 388 1038.0 ACP:400 ATPlike Active DFGin 6.615 13.378 BLAminus -120.4, -155.16 27.84, 85.75 -104.36, 38.7 310.01, 93.15 -67.71, -28.73 in-in in 7.966 Saltbr-in 3.021 HRD-in -109.84, -42.56 64.6, 13.11 in-in-in SNCiii in-in ActLoopNT-in 3.014 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -150.8, 133.1 APE9-dihe-in -126.86, 129.0 APE8-dihe-in -43.1, 130.27 APE8-rot-na 329.12 APE67-dihe-in -70.13, -6.6 -62.78, -39.45 APE12-dist-na 12.662 APE11-dist-na 7.646 APE10-dist-na 11.0 APE9-dist-in 5.878 None None None XRAY 2.8 0.226 0.322 B 291 261 11 0 0 0 [[126, 387]] 1.0 1u54 Homo sapiens TYR_TNK2_HUMAN TYR 9e-86 293.3 1 259 259 269 270 271 273 275 158 177 181 249 251 250 252 312 300 295 294 293 292 291 290 289 206 Activated CDC42 kinase 1
OTHER LPL0262 Q5WZW9_LEGPL 5CKWA Q5WZW9 15 404 961.0 ANP:60501 ATPlike Active DFGin 5.948 12.719 BLAminus -133.44, 169.43 70.28, 94.79 -117.83, 12.87 299.33, 117.8 -55.88, -8.97 in-in in 6.71 Saltbr-in 2.716 HRD-na-Q -80.53, -48.66 73.11, 5.26 in-in-in SNCiii in-in ActLoopNT-in 2.927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -69.26, -22.18 APE9-dihe-na -101.55, 179.41 APE8-dihe-in -117.11, 122.15 APE8-rot-in 302.21 APE67-dihe-in -64.67, -9.61 -57.44, -37.84 APE12-dist-in 11.762 APE11-dist-in 9.709 APE10-dist-in 4.647 APE9-dist-in 3.347 None None None XRAY 2.49 0.207 0.258 A 451 378 5 0 0 0 [[75, 309]] 1.0 5ckw Legionella pneumophila OTHER_LPL0262_LEGPL NEK 4.8e-15 62.8 10 222 213 212 213 214 216 218 104 119 123 192 194 193 195 249 237 232 231 230 229 228 227 226 146 non-specific serine/threonine protein kinase
OTHER LPL0262 Q5WZW9_LEGPL 5CKWB Q5WZW9 1 404 961.0 ANP:60501 ATPlike Active DFGin 6.189 12.674 BLAminus -144.06, 165.73 65.65, 85.18 -109.61, 21.73 306.46, 113.14 -57.87, -17.2 in-in in 6.769 Saltbr-in 2.882 HRD-na-Q -82.05, -45.94 73.24, -7.24 in-in-in SNCiii in-in ActLoopNT-in 2.976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -76.56, -19.65 APE9-dihe-na -103.71, -175.8 APE8-dihe-in -130.62, 116.65 APE8-rot-in 293.03 APE67-dihe-in -65.48, -28.87 -48.06, -39.07 APE12-dist-in 11.529 APE11-dist-in 9.586 APE10-dist-in 4.483 APE9-dist-in 3.458 None None None XRAY 2.49 0.207 0.258 B 451 399 5 0 0 0 [[75, 309]] 1.0 5ckw Legionella pneumophila OTHER_LPL0262_LEGPL NEK 4.8e-15 62.8 10 222 213 212 213 214 216 218 104 119 123 192 194 193 195 249 237 232 231 230 229 228 227 226 146 non-specific serine/threonine protein kinase
AGC PRKACA KAPCA_MOUSE 4O21A P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 6.037 14.439 BLAminus -125.27, 173.53 70.53, 83.75 -96.26, 25.58 272.04, 54.28 -57.91, -27.19 in-in in 8.953 Saltbr-in 2.716 HRD-in -83.95, -57.84 75.15, 8.54 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.15, 164.3 APE9-dihe-na 125.14, -151.92 APE8-dihe-in -125.51, 129.66 APE8-rot-in 308.07 APE67-dihe-in -63.53, -19.17 -43.91, -48.76 APE12-dist-in 8.04 APE11-dist-in 11.46 APE10-dist-in 5.911 APE9-dist-in 3.451 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.17 0.215 A 342 336 0 0 0 0 [[44, 298]] 1.0 4o21 Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7E11A P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 6.205 14.451 BLAminus -127.38, -169.19 58.28, 74.22 -96.53, 30.74 276.22, 81.09 -66.46, -21.72 in-in in 9.053 Saltbr-in 2.551 HRD-in -91.79, -53.23 62.57, 24.02 in-in-in SNCiii in-in ActLoopNT-in 3.129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.39, 155.98 APE9-dihe-na 134.96, -158.62 APE8-dihe-in -113.95, 132.34 APE8-rot-in 301.67 APE67-dihe-in -76.79, -1.28 -53.37, -39.68 APE12-dist-in 8.309 APE11-dist-in 11.135 APE10-dist-in 5.71 APE9-dist-in 3.659 None TPO198,SEP339 TPO198,SEP339 XRAY 3.43 0.262 0.317 A 338 337 0 0 0 0 [[44, 298]] 1.0 7e11 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3PVBA P05132 7 351 351.0 ANP:60400 ATPlike Active DFGin 5.261 14.107 BLAminus -138.85, 171.16 63.11, 82.89 -89.43, -59.95 273.17, 54.43 27.14, -66.26 in-in in 8.685 Saltbr-in 3.476 HRD-in -84.36, -35.8 62.24, -18.82 in-in-in SNCiii in-in ActLoopNT-in 3.217 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -177.84, 157.88 APE9-dihe-na 132.55, -154.74 APE8-dihe-in -122.19, 108.01 APE8-rot-in 318.81 APE67-dihe-in -60.75, -2.24 -13.41, -60.33 APE12-dist-in 7.733 APE11-dist-in 10.579 APE10-dist-in 5.511 APE9-dist-in 4.042 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 3.3 0.242 0.29 A 345 345 0 0 0 0 [[44, 298]] 1.0 3pvb Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 1BKXA P05132 13 351 351.0 AMP:60351 ATPlike Active DFGin 6.16 13.915 BLAminus -117.09, 179.26 61.99, 75.16 -83.18, 21.65 286.96, 82.43 -60.51, -17.53 in-in in 8.724 Saltbr-in 2.658 HRD-in -99.39, -38.31 69.2, -9.22 in-in-in SNCiii in-in ActLoopNT-in 3.468 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.44, 150.62 APE9-dihe-na 113.99, 166.84 APE8-dihe-in -65.88, 134.1 APE8-rot-in 334.22 APE67-dihe-in -70.66, -34.65 -48.92, -27.08 APE12-dist-in 8.284 APE11-dist-in 11.351 APE10-dist-in 5.704 APE9-dist-in 4.285 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.6 0.219 0.34 A 350 339 0 0 0 0 [[44, 298]] 1.0 1bkx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 1L3RE P05132 2 351 351.0 ADP:60381 ATPlike Active DFGin 5.754 14.44 BLAminus -119.14, -174.46 57.18, 81.19 -93.77, 20.31 270.88, 52.04 -50.0, -37.57 in-in in 9.023 Saltbr-in 2.792 HRD-in -82.45, -54.36 70.16, 7.26 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.84, 161.06 APE9-dihe-na 132.7, -149.01 APE8-dihe-in -131.06, 132.91 APE8-rot-in 298.56 APE67-dihe-in -55.27, -27.25 -33.24, -62.94 APE12-dist-in 8.198 APE11-dist-in 11.233 APE10-dist-in 5.825 APE9-dist-in 3.368 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.0 0.205 0.232 E 350 341 0 0 0 0 [[44, 298]] 1.0 1l3r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 2QCSA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.648 14.291 BLAminus -119.78, 176.88 65.56, 77.31 -85.05, 19.39 273.35, 51.28 -44.32, -42.51 in-in in 8.784 Saltbr-in 2.638 HRD-in -93.14, -54.78 73.52, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.735 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.52, 149.74 APE9-dihe-na 148.64, -142.53 APE8-dihe-in -132.36, 132.12 APE8-rot-in 297.18 APE67-dihe-in -64.67, -25.45 -36.74, -53.73 APE12-dist-in 8.133 APE11-dist-in 11.321 APE10-dist-in 5.851 APE9-dist-in 3.573 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.194 0.225 A 350 338 0 0 0 0 [[44, 298]] 1.0 2qcs Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3FJQE P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.671 14.459 BLAminus -119.42, 178.78 63.28, 80.04 -91.81, 23.31 270.73, 57.82 -56.09, -30.86 in-in in 9.149 Saltbr-in 2.834 HRD-in -91.33, -52.39 67.42, 13.87 in-in-in SNCiii in-in ActLoopNT-in 2.906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.19, 160.44 APE9-dihe-na 133.42, -155.21 APE8-dihe-in -125.75, 136.86 APE8-rot-in 304.0 APE67-dihe-in -61.0, -22.29 -48.87, -49.39 APE12-dist-in 8.086 APE11-dist-in 11.408 APE10-dist-in 5.838 APE9-dist-in 3.518 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.179 0.205 E 350 336 0 0 0 0 [[44, 298]] 1.0 3fjq Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3IDBA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.346 14.413 BLAminus -121.17, -175.1 59.7, 79.28 -94.34, 24.01 267.69, 48.22 -48.56, -33.02 in-in in 8.845 Saltbr-in 2.694 HRD-in -80.07, -50.75 69.18, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.99 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.99, 160.5 APE9-dihe-na 138.4, -150.07 APE8-dihe-in -124.64, 132.33 APE8-rot-in 296.41 APE67-dihe-in -59.26, -21.93 -30.94, -63.4 APE12-dist-in 8.102 APE11-dist-in 11.573 APE10-dist-in 6.068 APE9-dist-in 3.445 None TPO198,SEP339 TPO198,SEP339 XRAY 1.62 0.206 0.23 A 350 343 0 0 0 0 [[44, 298]] 1.0 3idb Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3IDCA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.079 14.472 BLAminus -127.31, 174.57 68.22, 96.34 -111.15, 30.11 265.57, 49.45 -62.75, -22.0 in-in in 8.642 Saltbr-in 3.031 HRD-in -69.04, -44.03 64.09, 13.38 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.35, 157.69 APE9-dihe-na 142.7, -132.16 APE8-dihe-in -139.58, 115.88 APE8-rot-in 293.03 APE67-dihe-in -54.66, -5.54 -16.73, -78.3 APE12-dist-in 7.844 APE11-dist-in 11.373 APE10-dist-in 6.164 APE9-dist-in 3.675 None TPO198,SEP339 TPO198,SEP339 XRAY 2.7 0.241 0.319 A 350 343 0 0 0 0 [[44, 298]] 1.0 3idc Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DG0E P05132 11 351 351.0 ANP:60402 ATPlike Active DFGin 5.583 14.342 BLAminus -118.87, 179.66 65.44, 79.89 -93.34, 25.25 272.35, 58.42 -52.71, -36.39 in-in in 8.955 Saltbr-in 2.699 HRD-in -84.35, -52.45 74.02, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.07, 161.1 APE9-dihe-na 130.81, -146.6 APE8-dihe-in -130.07, 130.32 APE8-rot-in 303.85 APE67-dihe-in -61.09, -22.5 -44.14, -49.24 APE12-dist-in 8.008 APE11-dist-in 11.498 APE10-dist-in 5.9 APE9-dist-in 3.389 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.196 0.228 E 350 341 0 0 0 0 [[44, 298]] 1.0 4dg0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH1A P05132 16 351 351.0 ATP:60402 ATPlike Active DFGin 6.234 14.38 BLAminus -130.7, 167.11 69.97, 89.08 -103.01, 26.92 273.93, 57.95 -52.62, -33.38 in-in in 8.931 Saltbr-in 3.01 HRD-in -75.69, -51.31 65.95, 10.85 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.97, 163.54 APE9-dihe-na 128.87, -151.55 APE8-dihe-in -123.52, 135.53 APE8-rot-in 304.09 APE67-dihe-in -55.69, -26.94 -40.23, -59.36 APE12-dist-in 8.169 APE11-dist-in 11.557 APE10-dist-in 5.95 APE9-dist-in 3.545 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.199 0.234 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH3A P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.984 14.379 BLAminus -125.47, 176.75 61.82, 79.89 -92.16, 24.39 276.69, 54.39 -43.39, -47.09 in-in in 9.021 Saltbr-in 2.723 HRD-in -82.56, -48.22 66.04, -2.33 in-in-in SNCiii in-in ActLoopNT-in 2.931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 165.55 APE9-dihe-na 126.96, -149.27 APE8-dihe-in -125.58, 130.88 APE8-rot-in 307.35 APE67-dihe-in -57.88, -25.54 -37.95, -56.15 APE12-dist-in 8.225 APE11-dist-in 11.592 APE10-dist-in 6.104 APE9-dist-in 3.74 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.203 0.233 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH5A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 6.121 14.339 BLAminus -125.12, -179.76 61.4, 85.13 -97.61, 27.77 279.05, 62.21 -46.99, -44.52 in-in in 9.043 Saltbr-in 2.552 HRD-in -77.92, -53.51 67.68, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.88, 153.17 APE9-dihe-na 132.88, -161.89 APE8-dihe-in -112.07, 131.8 APE8-rot-in 304.21 APE67-dihe-in -57.01, -23.17 -41.47, -55.69 APE12-dist-in 8.219 APE11-dist-in 11.602 APE10-dist-in 6.071 APE9-dist-in 3.87 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.187 0.222 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH7A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.574 14.349 BLAminus -124.43, -175.45 59.33, 78.79 -93.54, 24.71 270.97, 54.79 -50.12, -38.03 in-in in 9.025 Saltbr-in 2.724 HRD-in -76.49, -50.79 66.5, 11.01 in-in-in SNCiii in-in ActLoopNT-in 2.961 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.18, 162.39 APE9-dihe-na 131.3, -151.54 APE8-dihe-in -126.44, 134.15 APE8-rot-in 300.19 APE67-dihe-in -56.38, -25.77 -37.48, -60.34 APE12-dist-in 8.093 APE11-dist-in 11.455 APE10-dist-in 5.87 APE9-dist-in 3.417 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.8 0.179 0.194 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH8A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.901 14.014 BLAminus -123.95, -176.77 59.01, 85.18 -98.8, 24.84 279.52, 63.26 -51.76, -30.5 in-in in 8.8 Saltbr-in 2.713 HRD-in -77.99, -56.65 70.43, 3.78 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.95, 158.57 APE9-dihe-na 135.16, -154.79 APE8-dihe-in -124.8, 132.89 APE8-rot-in 296.53 APE67-dihe-in -58.95, -25.2 -38.46, -56.52 APE12-dist-in 8.145 APE11-dist-in 11.475 APE10-dist-in 5.904 APE9-dist-in 3.511 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.155 0.188 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh8 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4HPTE P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.748 14.424 BLAminus -115.4, 178.03 67.73, 81.09 -92.11, 21.69 273.09, 55.37 -58.71, -29.4 in-in in 9.053 Saltbr-in 2.66 HRD-in -90.64, -54.09 71.81, 9.39 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.27, 162.98 APE9-dihe-na 129.56, -147.32 APE8-dihe-in -127.39, 129.92 APE8-rot-in 299.02 APE67-dihe-in -63.31, -27.9 -40.61, -49.36 APE12-dist-in 8.069 APE11-dist-in 11.385 APE10-dist-in 5.825 APE9-dist-in 3.573 None TPO198,SEP339 TPO198,SEP339 XRAY 2.15 0.189 0.228 E 350 337 0 0 0 0 [[44, 298]] 1.0 4hpt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4HPUE P05132 13 351 351.0 ANP:60402 ATPlike Active DFGin 5.551 14.407 BLAminus -117.63, -178.61 63.83, 78.8 -92.22, 24.46 271.46, 55.23 -53.69, -32.94 in-in in 9.031 Saltbr-in 2.692 HRD-in -87.73, -52.35 74.85, 8.01 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.41, 162.17 APE9-dihe-na 134.1, -149.11 APE8-dihe-in -128.69, 136.04 APE8-rot-in 297.56 APE67-dihe-in -58.67, -24.48 -48.3, -49.81 APE12-dist-in 8.063 APE11-dist-in 11.507 APE10-dist-in 5.886 APE9-dist-in 3.403 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.173 0.194 E 350 339 0 0 0 0 [[44, 298]] 1.0 4hpu Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 5JR7A P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.739 13.691 BLAminus -145.14, 176.28 64.37, 76.68 -85.75, 18.89 294.14, 59.99 -43.66, -41.86 in-in in 8.674 Saltbr-in 2.709 HRD-in -93.38, -54.67 74.91, 7.39 in-in-in SNCiii in-in ActLoopNT-in 2.945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.46, 148.2 APE9-dihe-na 147.95, -159.28 APE8-dihe-in -109.66, 131.32 APE8-rot-in 258.88 APE67-dihe-in -65.5, -25.8 -38.64, -53.47 APE12-dist-in 8.014 APE11-dist-in 10.772 APE10-dist-in 5.528 APE9-dist-in 3.878 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 A 350 338 0 0 0 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 5JR7C P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.899 13.164 BLAminus -138.79, 176.44 54.89, 86.07 -89.1, 7.67 290.95, 62.79 -41.83, -37.01 in-in in 8.185 Saltbr-in 3.195 HRD-in -79.11, -50.37 72.48, -21.93 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.28, 123.46 APE9-dihe-na 160.31, -160.86 APE8-dihe-in -110.49, 124.04 APE8-rot-in 311.35 APE67-dihe-in -70.47, -24.34 -45.9, -42.95 APE12-dist-in 8.163 APE11-dist-in 10.628 APE10-dist-in 5.002 APE9-dist-in 4.262 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 C 350 338 0 0 0 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7UJXE P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 5.731 14.357 BLAminus -121.93, 179.51 64.92, 83.56 -91.91, 29.5 277.22, 63.03 -64.62, -28.12 in-in in 9.103 Saltbr-in 2.812 HRD-in -86.19, -57.72 74.11, 16.74 in-in-in SNCiii in-in ActLoopNT-in 2.931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.48, 155.47 APE9-dihe-na 127.23, -161.98 APE8-dihe-in -111.77, 133.52 APE8-rot-in 302.04 APE67-dihe-in -65.07, -18.97 -50.87, -44.77 APE12-dist-in 8.191 APE11-dist-in 11.5 APE10-dist-in 5.961 APE9-dist-in 4.008 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.133 0.176 E 350 336 0 0 0 0 [[44, 298]] 1.0 7ujx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7V0GE P05132 17 351 351.0 ADP:60401 ATPlike Active DFGin 5.739 14.319 BLAminus -119.5, 177.58 67.43, 82.74 -91.45, 25.21 276.8, 64.92 -62.46, -26.34 in-in in 9.07 Saltbr-in 2.802 HRD-in -88.93, -50.41 71.3, 15.33 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.52, 156.77 APE9-dihe-na 130.04, -162.37 APE8-dihe-in -114.97, 131.2 APE8-rot-in 299.52 APE67-dihe-in -60.0, -22.75 -47.18, -49.61 APE12-dist-in 8.174 APE11-dist-in 11.542 APE10-dist-in 6.037 APE9-dist-in 3.965 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.118 0.163 E 350 335 0 0 0 0 [[44, 298]] 1.0 7v0g Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DFXE P05132 2 351 351.0 ANP:60402 ATPlike Active DFGin 5.524 14.286 BLAminus -116.71, -179.39 66.13, 78.01 -91.08, 23.34 272.63, 51.46 -56.59, -32.27 in-in in 8.873 Saltbr-in 2.729 HRD-in -88.99, -54.58 73.79, 11.03 in-in-in SNCiii in-in ActLoopNT-in 2.934 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.69, 159.64 APE9-dihe-na 138.16, -148.52 APE8-dihe-in -130.4, 136.32 APE8-rot-in 296.63 APE67-dihe-in -59.91, -24.0 -47.38, -49.37 APE12-dist-in 8.046 APE11-dist-in 11.41 APE10-dist-in 5.819 APE9-dist-in 3.392 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.35 0.157 0.179 E 350 350 0 0 0 0 [[44, 298]] 1.0 4dfx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4X6RA P05132 2 351 351.0 ATP:60402 ATPlike Active DFGin 6.133 14.232 BLAminus -118.92, 178.27 64.18, 79.91 -89.21, 11.01 274.1, 55.74 -49.19, -34.95 in-in in 8.804 Saltbr-in 2.729 HRD-in -85.13, -60.38 77.67, -7.87 in-in-in SNCiii in-in ActLoopNT-in 2.718 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.34, 156.01 APE9-dihe-na 147.33, -149.7 APE8-dihe-in -130.56, 138.51 APE8-rot-in 291.09 APE67-dihe-in -61.2, -24.8 -52.44, -47.95 APE12-dist-in 8.281 APE11-dist-in 11.246 APE10-dist-in 5.836 APE9-dist-in 3.663 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.186 0.234 A 350 350 0 0 0 0 [[44, 298]] 1.0 4x6r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3X2UA P05132 13 351 351.0 ATP:60501 ATPlike Active DFGin 6.127 14.507 BLAminus -122.24, 178.58 59.36, 87.7 -101.54, 25.28 272.61, 50.83 -59.45, -24.26 in-in in 9.272 Saltbr-in 2.788 HRD-in -89.58, -50.62 64.84, 17.58 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.25, 158.3 APE9-dihe-na 134.88, -147.54 APE8-dihe-in -130.4, 131.58 APE8-rot-in 300.12 APE67-dihe-in -61.26, -14.4 -40.08, -55.22 APE12-dist-in 7.912 APE11-dist-in 11.137 APE10-dist-in 5.686 APE9-dist-in 3.427 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.202 0.239 A 357 339 0 0 0 0 [[44, 298]] 1.0 3x2u Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3X2VA P05132 18 351 351.0 ATP:60403 ATPlike Active DFGin 5.517 14.152 BLAminus -116.69, -175.94 62.92, 80.3 -91.77, 26.26 271.42, 55.44 -51.78, -39.79 in-in in 8.755 Saltbr-in 2.654 HRD-in -92.08, -50.84 67.69, 17.07 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.85, 164.45 APE9-dihe-na 134.14, -152.5 APE8-dihe-in -130.83, 133.42 APE8-rot-in 299.77 APE67-dihe-in -58.82, -21.18 -48.96, -48.11 APE12-dist-in 7.998 APE11-dist-in 11.346 APE10-dist-in 5.796 APE9-dist-in 3.415 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.77 0.185 0.23 A 357 334 0 0 0 0 [[44, 298]] 1.0 3x2v Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3X2WA P05132 13 351 351.0 ATP:60403 ATPlike Active DFGin 5.66 14.39 BLAminus -121.01, -177.68 63.51, 77.56 -90.4, 24.79 270.4, 59.29 -61.83, -28.06 in-in in 8.822 Saltbr-in 2.632 HRD-in -81.34, -52.24 70.22, 11.48 in-in-in SNCiii in-in ActLoopNT-in 2.906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.19, 162.39 APE9-dihe-na 132.4, -151.44 APE8-dihe-in -129.91, 133.08 APE8-rot-in 300.2 APE67-dihe-in -60.45, -20.83 -45.18, -51.38 APE12-dist-in 8.001 APE11-dist-in 11.44 APE10-dist-in 5.911 APE9-dist-in 3.45 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.165 0.198 A 357 339 0 0 0 0 [[44, 298]] 1.0 3x2w Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IACA P05132 16 351 351.0 ACP:60403 ATPlike Active DFGin 5.755 14.312 BLAminus -125.73, -177.16 59.8, 78.08 -94.31, 23.06 273.35, 54.81 -46.36, -37.92 in-in in 8.885 Saltbr-in 2.721 HRD-in -73.57, -53.97 72.67, 5.23 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.57, 156.93 APE9-dihe-na 137.19, -153.99 APE8-dihe-in -123.03, 128.21 APE8-rot-in 300.87 APE67-dihe-in -59.06, -23.99 -31.47, -61.7 APE12-dist-in 8.157 APE11-dist-in 11.515 APE10-dist-in 5.985 APE9-dist-in 3.502 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.15 0.181 0.212 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iac Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IADA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.658 14.362 BLAminus -130.04, -179.13 63.0, 77.66 -87.34, 22.78 276.11, 53.54 -55.12, -31.28 in-in in 9.085 Saltbr-in 2.83 HRD-in -93.22, -52.19 70.15, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.935 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.54, 160.6 APE9-dihe-na 133.65, -143.98 APE8-dihe-in -130.05, 134.5 APE8-rot-in 298.49 APE67-dihe-in -67.08, -22.74 -48.94, -44.54 APE12-dist-in 8.051 APE11-dist-in 11.55 APE10-dist-in 6.087 APE9-dist-in 3.521 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.189 0.243 A 356 337 0 0 0 0 [[44, 298]] 1.0 4iad Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAFA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.943 14.13 BLAminus -121.29, 178.82 64.06, 84.8 -98.0, 27.2 281.56, 65.38 -51.93, -33.25 in-in in 8.871 Saltbr-in 2.669 HRD-in -76.48, -53.65 65.3, 9.94 in-in-in SNCiii in-in ActLoopNT-in 2.974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.4, 160.11 APE9-dihe-na 128.66, -151.44 APE8-dihe-in -123.86, 135.06 APE8-rot-in 298.27 APE67-dihe-in -57.84, -25.84 -42.55, -55.44 APE12-dist-in 8.163 APE11-dist-in 11.523 APE10-dist-in 5.973 APE9-dist-in 3.563 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.16 0.192 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iaf Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAIA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.465 14.503 BLAminus -125.1, 176.4 64.24, 81.88 -90.74, 22.64 269.91, 49.4 -55.45, -35.99 in-in in 9.101 Saltbr-in 2.714 HRD-in -91.06, -49.32 68.79, 15.16 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.75, 156.86 APE9-dihe-na 141.29, -148.36 APE8-dihe-in -128.24, 130.8 APE8-rot-in 300.02 APE67-dihe-in -62.27, -23.0 -47.39, -47.75 APE12-dist-in 7.945 APE11-dist-in 11.458 APE10-dist-in 5.867 APE9-dist-in 3.608 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.171 0.209 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iai Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAKA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.705 14.569 BLAminus -126.92, 179.61 63.08, 81.74 -90.27, 23.65 270.26, 53.44 -59.05, -31.45 in-in in 8.985 Saltbr-in 2.747 HRD-in -94.54, -49.89 67.85, 16.15 in-in-in SNCiii in-in ActLoopNT-in 2.91 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.92, 164.74 APE9-dihe-na 131.87, -148.57 APE8-dihe-in -130.85, 127.67 APE8-rot-in 297.68 APE67-dihe-in -61.28, -21.91 -43.91, -50.7 APE12-dist-in 7.962 APE11-dist-in 11.443 APE10-dist-in 5.979 APE9-dist-in 3.545 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.6 0.185 0.222 A 356 337 0 0 0 0 [[44, 298]] 1.0 4iak Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAYA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.806 14.257 BLAminus -131.74, 174.05 67.76, 85.89 -95.28, 20.31 273.12, 61.73 -48.17, -36.05 in-in in 9.039 Saltbr-in 2.941 HRD-in -89.87, -50.65 68.98, 10.01 in-in-in SNCiii in-in ActLoopNT-in 3.055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.39, 159.46 APE9-dihe-na 132.54, -148.24 APE8-dihe-in -127.91, 130.95 APE8-rot-in 300.76 APE67-dihe-in -63.09, -19.35 -45.58, -49.88 APE12-dist-in 8.089 APE11-dist-in 11.466 APE10-dist-in 5.991 APE9-dist-in 3.823 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.182 0.227 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iay Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAZA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 6.144 14.635 BLAminus -132.33, 171.23 62.84, 84.78 -94.94, 21.85 278.49, 61.31 -54.74, -28.93 in-in in 9.219 Saltbr-in 2.747 HRD-in -95.03, -54.93 73.76, 14.73 in-in-in SNCiii in-in ActLoopNT-in 3.017 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.57, 164.74 APE9-dihe-na 127.12, -150.82 APE8-dihe-in -127.02, 138.46 APE8-rot-in 303.51 APE67-dihe-in -63.11, -25.72 -51.71, -47.83 APE12-dist-in 7.963 APE11-dist-in 11.514 APE10-dist-in 5.979 APE9-dist-in 3.574 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.85 0.201 0.248 A 356 337 0 0 0 0 [[44, 298]] 1.0 4iaz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IB0A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.713 14.439 BLAminus -123.68, 176.86 65.62, 82.22 -94.42, 18.76 272.15, 51.12 -47.84, -35.86 in-in in 9.065 Saltbr-in 3.023 HRD-in -84.67, -55.05 71.31, 12.11 in-in-in SNCiii in-in ActLoopNT-in 2.886 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.67, 157.49 APE9-dihe-na 139.08, -144.95 APE8-dihe-in -131.16, 131.55 APE8-rot-in 306.17 APE67-dihe-in -61.31, -24.54 -46.0, -48.78 APE12-dist-in 8.059 APE11-dist-in 11.516 APE10-dist-in 5.969 APE9-dist-in 3.692 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.87 0.219 0.287 A 356 337 0 0 0 0 [[44, 298]] 1.0 4ib0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IB1A P05132 14 351 351.0 ADP:60403 ATPlike Active DFGin 5.656 14.443 BLAminus -126.58, 171.72 66.62, 80.69 -90.79, 23.58 274.18, 53.88 -53.03, -31.34 in-in in 9.121 Saltbr-in 2.691 HRD-in -82.93, -51.49 69.93, 14.85 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.64, 163.58 APE9-dihe-na 133.1, -151.37 APE8-dihe-in -125.38, 138.08 APE8-rot-in 304.1 APE67-dihe-in -60.15, -23.69 -50.01, -49.7 APE12-dist-in 7.96 APE11-dist-in 11.404 APE10-dist-in 5.961 APE9-dist-in 3.635 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.196 0.223 A 356 338 0 0 0 0 [[44, 298]] 1.0 4ib1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IB3A P05132 13 351 351.0 ADP:60401 ATPlike Active DFGin 5.973 14.215 BLAminus -125.69, 173.12 66.37, 84.97 -98.59, 21.41 276.57, 60.51 -51.27, -29.52 in-in in 8.99 Saltbr-in 2.76 HRD-in -77.27, -49.79 61.58, 13.48 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.06, 160.46 APE9-dihe-na 127.6, -161.57 APE8-dihe-in -110.98, 129.89 APE8-rot-in 305.68 APE67-dihe-in -58.89, -23.07 -39.61, -54.94 APE12-dist-in 8.078 APE11-dist-in 11.522 APE10-dist-in 5.923 APE9-dist-in 3.568 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.182 0.228 A 356 339 0 0 0 0 [[44, 298]] 1.0 4ib3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4XW4A P05132 15 351 351.0 ANP:60403 ATPlike Active DFGin 5.673 14.562 BLAminus -117.82, -177.44 65.15, 79.34 -92.69, 26.58 269.45, 57.64 -61.99, -28.36 in-in in 8.931 Saltbr-in 2.858 HRD-in -86.05, -50.94 67.2, 15.72 in-in-in SNCiii in-in ActLoopNT-in 3.014 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.62, 159.69 APE9-dihe-na 135.12, -140.29 APE8-dihe-in -136.84, 125.12 APE8-rot-in 301.75 APE67-dihe-in -61.52, -26.6 -45.5, -44.66 APE12-dist-in 7.961 APE11-dist-in 11.419 APE10-dist-in 5.935 APE9-dist-in 3.664 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.82 0.183 0.24 A 356 337 0 0 0 0 [[44, 298]] 1.0 4xw4 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4XW5A P05132 15 351 351.0 ATP:60403 ATPlike Active DFGin 5.971 14.222 BLAminus -131.24, 177.82 59.66, 87.19 -93.08, 25.08 282.37, 63.43 -53.77, -29.24 in-in in 9.213 Saltbr-in 2.673 HRD-in -90.87, -48.94 63.52, 13.92 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.24, 155.03 APE9-dihe-na 137.47, -160.98 APE8-dihe-in -110.31, 133.6 APE8-rot-in 304.05 APE67-dihe-in -58.14, -25.36 -48.87, -50.12 APE12-dist-in 8.026 APE11-dist-in 11.601 APE10-dist-in 6.1 APE9-dist-in 3.922 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.185 0.252 A 356 337 0 0 0 0 [[44, 298]] 1.0 4xw5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4XW6A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.982 14.431 BLAminus -130.68, 178.48 65.03, 84.15 -99.24, 23.41 276.01, 56.03 -60.45, -23.49 in-in in 9.15 Saltbr-in 2.735 HRD-in -94.59, -52.61 68.2, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.791 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.91, 154.59 APE9-dihe-na 136.7, -154.91 APE8-dihe-in -121.39, 127.95 APE8-rot-in 293.9 APE67-dihe-in -62.75, -24.38 -45.59, -46.76 APE12-dist-in 8.051 APE11-dist-in 11.632 APE10-dist-in 6.051 APE9-dist-in 3.787 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.186 0.265 A 356 337 0 0 0 0 [[44, 298]] 1.0 4xw6 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 6E21A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.594 14.055 BLAminus -122.61, 176.37 63.02, 83.41 -94.2, 28.27 284.3, 46.09 -48.88, -41.13 in-in in 9.029 Saltbr-in 2.607 HRD-in -74.35, -56.8 67.48, 11.51 in-in-in SNCiii in-in ActLoopNT-in 2.907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.7, 159.01 APE9-dihe-na 131.41, -152.84 APE8-dihe-in -125.29, 130.56 APE8-rot-in 303.23 APE67-dihe-in -58.42, -25.04 -35.36, -60.06 APE12-dist-in 8.043 APE11-dist-in 11.584 APE10-dist-in 6.022 APE9-dist-in 3.58 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.187 0.217 A 356 336 0 0 0 0 [[44, 298]] 1.0 6e21 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7E0ZA P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 5.566 13.884 BLAminus -118.85, -174.47 59.93, 79.47 -94.43, 25.89 275.59, 63.85 -59.78, -31.6 in-in in 8.624 Saltbr-in 2.978 HRD-in -96.8, -56.38 78.26, 13.74 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.91, 162.74 APE9-dihe-na 131.67, -149.57 APE8-dihe-in -131.04, 130.65 APE8-rot-in 294.41 APE67-dihe-in -63.42, -12.5 -45.48, -52.1 APE12-dist-in 7.9 APE11-dist-in 11.182 APE10-dist-in 5.721 APE9-dist-in 3.4 None TPO198,SEP339 TPO198,SEP339 XRAY 2.162 0.184 0.228 A 358 337 0 0 0 0 [[44, 298]] 1.0 7e0z Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DG3E P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.481 14.342 BLAminus -115.99, -176.62 61.62, 77.98 -90.25, 24.84 270.29, 54.4 -55.44, -35.73 in-in in 8.842 Saltbr-in 2.695 HRD-in -87.1, -53.93 73.82, 10.76 in-in-in SNCiii in-in ActLoopNT-in 2.882 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.46, 161.61 APE9-dihe-na 135.41, -150.07 APE8-dihe-in -129.52, 135.22 APE8-rot-in 300.3 APE67-dihe-in -58.11, -23.91 -46.28, -51.67 APE12-dist-in 8.143 APE11-dist-in 11.482 APE10-dist-in 5.886 APE9-dist-in 3.405 R337A SEP140,TPO198 SEP140,TPO198 XRAY 1.8 0.185 0.217 E 371 337 0 0 0 0 [[44, 298]] 1.0 4dg3 Mus musculus AGC_PRKACA_MOUSE AGC 1.8e-94 321.8 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3FHIA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.463 14.263 BLAminus -118.0, -179.45 64.04, 75.7 -86.07, 24.14 267.17, 53.33 -59.82, -32.06 in-in in 8.887 Saltbr-in 2.79 HRD-in -94.84, -53.37 68.02, 7.49 in-in-in SNCiii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.67, 136.88 APE9-dihe-na 156.84, -158.52 APE8-dihe-in -126.08, 132.83 APE8-rot-in 296.09 APE67-dihe-in -67.08, -19.88 -42.62, -50.01 APE12-dist-in 8.233 APE11-dist-in 11.12 APE10-dist-in 5.402 APE9-dist-in 3.564 C200A TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.199 0.226 A 350 338 0 0 0 0 [[44, 298]] 1.0 3fhi Mus musculus AGC_PRKACA_MOUSE AGC 1e-93 319.3 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3QAME P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.559 14.19 BLAminus -125.2, -173.2 57.82, 79.24 -94.32, 24.42 273.28, 56.46 -52.36, -33.22 in-in in 8.98 Saltbr-in 2.804 HRD-in -80.54, -55.75 67.52, 12.49 in-in-in SNCiii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.45, 157.56 APE9-dihe-na 134.84, -152.56 APE8-dihe-in -129.9, 127.65 APE8-rot-in 298.13 APE67-dihe-in -57.31, -20.14 -26.19, -66.74 APE12-dist-in 8.094 APE11-dist-in 11.277 APE10-dist-in 5.806 APE9-dist-in 3.475 E209A TPO198,SEP339 TPO198,SEP339 XRAY 1.92 0.195 0.228 E 350 350 0 0 0 0 [[44, 298]] 1.0 3qam Mus musculus AGC_PRKACA_MOUSE AGC 2.2e-93 318.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3QALE P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.64 14.401 BLAminus -123.21, -177.09 59.31, 80.89 -94.71, 25.93 269.1, 56.43 -54.28, -32.32 in-in in 9.05 Saltbr-in 2.658 HRD-in -84.64, -51.07 65.64, 14.74 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.61, 159.73 APE9-dihe-na 131.58, -155.18 APE8-dihe-in -126.66, 132.34 APE8-rot-in 301.51 APE67-dihe-in -57.77, -23.32 -31.31, -63.36 APE12-dist-in 8.062 APE11-dist-in 11.309 APE10-dist-in 5.744 APE9-dist-in 3.531 R281A TPO198,SEP339 TPO198,SEP339 XRAY 1.7 0.176 0.194 E 350 341 0 0 0 0 [[44, 298]] 1.0 3qal Mus musculus AGC_PRKACA_MOUSE AGC 4.5e-93 317.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CAMK CAMK2A KCC2A_MOUSE 7B56B P11798 5 307 478.0 ANP:60401 ATPlike Active DFGin 6.729 14.232 BLAminus -127.69, 175.68 61.5, 79.97 -89.44, 23.96 289.95, 77.46 -66.33, -24.14 in-in in 8.963 Saltbr-in 2.797 HRD-in -75.83, -42.64 71.61, -6.11 in-in-in SNCiii in-in ActLoopNT-in 2.891 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.35, 145.48 APE9-dihe-na 136.45, -166.63 APE8-dihe-in -115.36, 130.21 APE8-rot-in 297.52 APE67-dihe-in -66.37, -13.84 -48.36, -50.63 APE12-dist-in 10.406 APE11-dist-in 11.67 APE10-dist-in 5.883 APE9-dist-in 3.799 T305A,T306A None None XRAY 1.45 0.191 0.215 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b56 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_MOUSE 7B57B P11798 5 307 478.0 ADP:603 ATPlike Active DFGin 6.612 14.081 BLAminus -127.42, 175.73 58.47, 86.34 -93.82, 26.41 288.57, 77.62 -63.18, -29.51 in-in in 8.79 Saltbr-in 2.799 HRD-in -66.41, -49.66 65.98, 1.57 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.13, 142.7 APE9-dihe-na 131.67, 177.43 APE8-dihe-in -91.43, 131.98 APE8-rot-in 302.75 APE67-dihe-in -62.31, -16.39 -48.04, -47.99 APE12-dist-in 10.368 APE11-dist-in 11.44 APE10-dist-in 5.743 APE9-dist-in 3.998 T305A,T306A None None XRAY 1.95 0.206 0.247 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b57 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK DAPK2 DAPK2_MOUSE 2YAAA Q8VDF3 12 311 370.0 ATP:61302 ATPlike Active DFGin 6.531 14.282 BLAminus -119.44, -173.75 61.63, 82.55 -100.44, 26.82 279.23, 73.82 -61.71, -30.38 in-in in 9.437 Saltbr-in 2.945 HRD-in -69.91, -51.35 70.12, 4.4 in-in-in SNCiii in-in ActLoopNT-in 2.83 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.66, 179.02 APE9-dihe-na 88.17, 165.82 APE8-dihe-in -83.03, 124.75 APE8-rot-in 307.34 APE67-dihe-in -54.24, -28.42 -45.93, -43.89 APE12-dist-in 8.679 APE11-dist-in 11.592 APE10-dist-in 6.391 APE9-dist-in 4.926 None None None XRAY 2.3 0.219 0.271 A 361 300 0 0 0 0 [[23, 285]] 1.0 2yaa Mus musculus CAMK_DAPK2_MOUSE CAMK 1.1e-93 319.4 1 256 256 170 171 172 174 176 52 74 78 146 148 147 149 209 197 192 191 190 189 188 187 186 104 Death-associated protein kinase 2
CAMK DAPK2 DAPK2_MOUSE 2YABA Q8VDF3 13 311 370.0 AMP:61302 ATPlike Active DFGin 6.504 14.098 BLAminus -124.73, -175.5 61.61, 83.44 -98.66, 29.53 280.86, 70.25 -68.26, -23.3 in-in in 9.084 Saltbr-in 2.894 HRD-in -75.19, -47.84 69.74, 6.94 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.38, -177.82 APE9-dihe-na 87.95, 171.12 APE8-dihe-in -92.08, 123.94 APE8-rot-in 301.03 APE67-dihe-in -53.06, -29.06 -44.13, -47.2 APE12-dist-in 8.535 APE11-dist-in 11.604 APE10-dist-in 6.372 APE9-dist-in 4.88 None None None XRAY 1.9 0.174 0.215 A 361 299 0 0 0 0 [[23, 285]] 1.0 2yab Mus musculus CAMK_DAPK2_MOUSE CAMK 1.1e-93 319.4 1 256 256 170 171 172 174 176 52 74 78 146 148 147 149 209 197 192 191 190 189 188 187 186 104 Death-associated protein kinase 2
CMGC GSK3B GSK3B_MOUSE 8VMFA Q9WV60 27 383 420.0 ADP:60504 ATPlike Active DFGin 6.612 14.1 BLAminus -148.4, -167.57 58.53, 66.72 -90.57, 24.21 287.49, 78.37 -75.04, -7.89 in-in in 8.66 Saltbr-in 2.678 HRD-in -67.34, -47.3 70.6, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.84 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.01, -20.74 APE9-dihe-na -93.16, -168.14 APE8-dihe-in -112.8, 164.36 APE8-rot-in 304.6 APE67-dihe-inflip 78.98, -8.38 -56.8, 140.56 APE12-dist-in 13.183 APE11-dist-in 10.949 APE10-dist-in 6.514 APE9-dist-in 3.308 None None None XRAY 2.5 0.21 0.251 A 364 354 0 0 0 0 [[56, 340]] 1.0 8vmf Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_MOUSE 8VMGA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 7.0 13.999 BLAminus -139.67, -176.86 60.44, 73.06 -89.27, 27.07 283.1, 81.19 -73.23, -12.63 in-in in 8.478 Saltbr-in 2.688 HRD-in -67.64, -48.38 72.75, 3.36 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.26, 164.63 APE9-dihe-na 72.45, 142.8 APE8-dihe-in -66.41, 146.08 APE8-rot-in 307.07 APE67-dihe-in -64.3, -22.81 -57.43, -46.54 APE12-dist-in 13.278 APE11-dist-in 11.627 APE10-dist-in 6.941 APE9-dist-in 2.984 None None None XRAY 2.45 0.195 0.23 A 364 358 0 0 0 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_MOUSE 8VMEA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 6.469 13.844 BLAminus -131.0, -171.33 63.41, 73.0 -92.56, 22.88 289.27, 83.61 -79.03, -1.02 in-in in 8.753 Saltbr-in 2.78 HRD-in -67.9, -47.67 70.4, 7.52 in-in-in SNCiii in-in ActLoopNT-in 2.731 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.18, 168.01 APE9-dihe-na 68.83, 161.19 APE8-dihe-in -90.7, 152.54 APE8-rot-in 290.93 APE67-dihe-inflip 82.32, -22.26 -51.38, 150.9 APE12-dist-in 13.288 APE11-dist-in 12.071 APE10-dist-in 6.934 APE9-dist-in 3.292 None None None XRAY 2.3 0.183 0.23 A 365 355 0 0 0 0 [[56, 340]] 1.0 8vme Mus musculus CMGC_GSK3B_MOUSE CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_MOUSE 4NU1A Q9WV60 6 383 420.0 ADP:405 ATPlike Active DFGin 6.109 13.677 BLAminus -140.27, -172.8 60.29, 88.19 -108.14, 24.39 289.57, 88.21 -68.01, -14.99 in-in in 8.691 Saltbr-in 2.793 HRD-in -66.76, -45.51 62.96, 19.85 in-in-in SNCiii in-in ActLoopNT-in 2.682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.38, 172.68 APE9-dihe-na 66.76, 153.81 APE8-dihe-in -82.08, 156.46 APE8-rot-in 299.93 APE67-dihe-inflip 76.53, -25.22 -54.39, 158.45 APE12-dist-in 13.51 APE11-dist-in 11.621 APE10-dist-in 7.126 APE9-dist-in 3.15 None SEP9 SEP9 XRAY 2.5 0.194 0.245 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nu1 Mus musculus CMGC_GSK3B_MOUSE CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC MAPK14 MK14_MOUSE 5NZZE P47811 4 353 360.0 AGS:60401 ATPlike Active DFGin 6.514 14.981 BLAminus -122.06, 164.78 72.33, 78.3 -82.97, 27.83 284.83, 92.09 -68.73, -16.77 in-in in 9.475 Saltbr-in 3.566 HRD-in -92.47, -52.47 76.16, -3.26 in-in-in SNCiii in-in ActLoopNT-in 2.855 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.62, 176.88 APE9-dihe-na 58.43, 166.45 APE8-dihe-in -84.96, 144.19 APE8-rot-in 316.3 APE67-dihe-in -61.16, -25.49 -55.46, -53.03 APE12-dist-in 11.933 APE11-dist-in 11.395 APE10-dist-in 7.236 APE9-dist-in 3.126 None TPO180,PTR182 TPO180,PTR182 XRAY 2.6 0.221 0.271 E 360 345 5 0 0 0 [[24, 308]] 1.0 5nzz Mus musculus CMGC_MAPK14_MOUSE CMGC 1.9e-85 292.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_MOUSE 5NZZF P47811 5 353 360.0 AGS:60401 ATPlike Active DFGin 6.581 14.746 BLAminus -104.46, 169.41 67.42, 93.44 -106.87, 21.93 284.61, 82.38 -60.31, -14.32 in-in in 9.318 Saltbr-in 2.692 HRD-in -84.83, -58.57 70.0, 21.45 in-in-in SNCiii in-in ActLoopNT-in 3.066 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.79, 145.31 APE9-dihe-na 83.88, 162.38 APE8-dihe-in -79.27, 130.51 APE8-rot-in 303.15 APE67-dihe-in -54.1, -23.47 -46.06, -59.5 APE12-dist-in 11.925 APE11-dist-in 11.532 APE10-dist-in 7.245 APE9-dist-in 3.334 None TPO180,PTR182 TPO180,PTR182 XRAY 2.6 0.221 0.271 F 360 343 6 0 0 0 [[24, 308]] 1.0 5nzz Mus musculus CMGC_MAPK14_MOUSE CMGC 1.9e-85 292.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
TYR LYN LYN_MOUSE 2ZV8A P25911 239 501 512.0 ANP:60001 ATPlike Active DFGin 6.207 14.166 BLAminus -127.46, 176.54 66.14, 76.26 -98.89, 34.27 306.37, 82.39 -66.23, -26.52 in-in in 8.182 Saltbr-in 2.888 HRD-na-N -93.92, -49.32 76.02, -10.27 in-in-in SNCiii in-in ActLoopNT-in 2.954 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -123.91, 116.52 APE9-dihe-in -60.43, 148.58 APE8-dihe-in -80.52, 92.26 APE8-rot-na 28.17 APE67-dihe-in -68.44, -3.54 -43.41, -52.9 APE12-dist-na 9.634 APE11-dist-na 5.923 APE10-dist-na 9.729 APE9-dist-in 5.004 None None None XRAY 2.7 0.201 0.245 A 279 256 7 0 0 7 [[247, 499]] 1.0 2zv8 Mus musculus TYR_LYN_MOUSE TYR 4.1e-95 323.9 1 260 260 384 385 386 388 390 275 290 294 364 366 365 367 425 413 408 407 406 405 404 403 402 320 Tyrosine-protein kinase Lyn
CAMK PHKG1 PHKG1_RABIT 2PHKA P00518 15 291 387.0 ATP:60381 ATPlike Active DFGin 6.355 14.931 BLAminus -137.29, -164.32 48.12, 82.5 -104.58, 35.29 286.95, 71.57 -66.18, -30.51 in-in in 9.223 Saltbr-in 2.867 HRD-in -75.14, -51.03 75.46, 17.9 in-in-in SNCiii in-in ActLoopNT-in 2.885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.02, 157.52 APE9-dihe-na 142.39, -153.7 APE8-dihe-in -119.73, 129.29 APE8-rot-in 312.14 APE67-dihe-in -75.97, -3.06 -46.22, -51.97 APE12-dist-in 9.188 APE11-dist-in 12.037 APE10-dist-in 6.565 APE9-dist-in 4.187 None None None XRAY 2.6 0.253 0.3 A 277 277 0 0 0 0 [[20, 288]] 1.0 2phk Oryctolagus cuniculus CAMK_PHKG1_RABIT CAMK 3e-86 294.8 1 256 256 167 168 169 171 173 49 74 78 147 149 148 150 212 194 189 188 187 186 185 184 183 105 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
CAMK PHKG1 PHKG1_RABIT 1QL6A P00518 12 292 387.0 ATP:60301 ATPlike Active DFGin 6.367 14.614 BLAminus -136.63, -170.42 53.21, 74.77 -97.04, 26.39 287.52, 75.09 -70.06, -14.72 in-in in 9.205 Saltbr-in 3.1 HRD-in -59.97, -49.78 67.92, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.896 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.76, 155.97 APE9-dihe-na 109.55, 169.96 APE8-dihe-in -76.43, 127.92 APE8-rot-in 308.32 APE67-dihe-in -67.24, -23.63 -51.61, -34.62 APE12-dist-in 9.259 APE11-dist-in 11.445 APE10-dist-in 6.11 APE9-dist-in 4.369 E183S None None XRAY 2.4 0.24 0.33 A 298 281 0 0 0 0 [[20, 288]] 1.0 1ql6 Oryctolagus cuniculus CAMK_PHKG1_RABIT CAMK 5.1e-86 294.1 1 256 256 167 168 169 171 173 49 74 78 147 149 148 150 212 194 189 188 187 186 185 184 183 105 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
CAMK PHKG1 PHKG1_RABIT 1PHKA P00518 16 292 387.0 ATP:60381 ATPlike Active DFGin 6.147 14.336 BLAminus -126.89, -173.45 56.12, 79.25 -99.09, 29.57 290.92, 76.23 -67.63, -19.58 in-in in 8.993 Saltbr-in 2.825 HRD-in -77.33, -46.36 68.03, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.41, 147.14 APE9-dihe-na 116.4, 168.87 APE8-dihe-in -72.55, 120.48 APE8-rot-in 295.05 APE67-dihe-in -62.26, -27.58 -41.92, -42.38 APE12-dist-in 8.836 APE11-dist-in 11.43 APE10-dist-in 6.157 APE9-dist-in 4.492 None None None XRAY 2.2 0.21 0.288 A 298 277 0 0 0 0 [[20, 288]] 1.0 1phk Oryctolagus cuniculus CAMK_PHKG1_RABIT CAMK 4e-86 294.4 1 256 256 167 168 169 171 173 49 74 78 147 149 148 150 212 194 189 188 187 186 185 184 183 105 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
OTHER PINK1 PINK1_PEDHC 8UYHA E0W1I1 115 574 575.0 ANP:601 ATPlike Active DFGin 9.322 14.819 BLAminus -130.08, -169.42 57.7, 62.71 -86.71, 26.39 286.61, 80.23 -66.61, -35.48 in-in in 7.967 Saltbr-in 3.27 HRD-in -73.02, -43.12 61.9, 7.28 in-in-in SNCiii in-in ActLoopNT-in 2.764 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 161.16, -131.74 APE9-dihe-na -112.83, -108.55 APE8-dihe-in -69.42, 145.98 APE8-rot-na 76.98 APE67-dihe-in -73.97, -39.08 -95.26, -9.75 APE12-dist-in 8.048 APE11-dist-in 10.262 APE10-dist-in 5.834 APE9-dist-in 3.572 None TPO305 TPO305 EM 2.84 999.0 999.0 A 463 375 49 0 0 0 [[64, 514]] 1.0 8uyh Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
OTHER PINK1 PINK1_PEDHC 8UYHB E0W1I1 121 574 575.0 ANP:601 ATPlike Active DFGin 9.449 14.871 BLAminus -129.89, -169.12 59.53, 64.83 -87.85, 20.05 283.99, 82.98 -70.23, -23.56 in-in in 7.846 Saltbr-in 2.387 HRD-in -70.23, -41.92 63.21, 0.58 in-in-in SNCiii in-in ActLoopNT-in 2.932 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 144.56, -157.47 APE9-dihe-na -105.64, -99.0 APE8-dihe-in -70.54, 139.11 APE8-rot-na 52.17 APE67-dihe-in -71.03, -46.42 -78.22, -15.68 APE12-dist-in 7.74 APE11-dist-in 10.385 APE10-dist-in 6.127 APE9-dist-in 3.781 None TPO305 TPO305 EM 2.84 999.0 999.0 B 463 370 50 0 0 0 [[64, 514]] 1.0 8uyh Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
OTHER PINK1 PINK1_PEDHC 8UYIA E0W1I1 120 572 575.0 ADP:601 ATPlike Active DFGin 9.472 14.492 BLAminus -126.54, -170.24 58.08, 66.04 -87.71, 25.91 289.34, 85.25 -66.89, -21.8 in-in in 7.734 Saltbr-in 2.489 HRD-in -72.82, -45.28 62.7, 4.34 in-in-in SNCiii in-in ActLoopNT-in 2.793 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 149.48, -127.57 APE9-dihe-na -109.63, -105.35 APE8-dihe-in -70.24, 160.24 APE8-rot-na 51.46 APE67-dihe-in -90.34, -42.74 -107.64, 8.21 APE12-dist-in 8.485 APE11-dist-in 10.413 APE10-dist-in 5.828 APE9-dist-in 3.643 None SEP202,TPO305 SEP202,TPO305 EM 3.13 999.0 999.0 A 463 369 49 0 0 0 [[64, 514]] 1.0 8uyi Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
OTHER PINK1 PINK1_PEDHC 8UYIB E0W1I1 122 574 575.0 ADP:601 ATPlike Active DFGin 9.37 14.767 BLAminus -128.32, -168.79 58.11, 64.54 -83.54, 12.33 278.78, 92.3 -66.63, -13.93 in-in in 8.001 Saltbr-in 2.363 HRD-in -66.42, -44.15 62.85, 2.17 in-in-in SNCiii in-in ActLoopNT-in 2.974 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 143.29, -143.85 APE9-dihe-na -111.19, -100.88 APE8-dihe-in -71.36, 134.31 APE8-rot-na 50.34 APE67-dihe-in -67.38, -41.28 -74.79, -24.08 APE12-dist-in 8.473 APE11-dist-in 10.806 APE10-dist-in 6.227 APE9-dist-in 3.553 None SEP202,TPO305 SEP202,TPO305 EM 3.13 999.0 999.0 B 463 369 51 0 0 0 [[64, 514]] 1.0 8uyi Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
CAMK CDPK1 CDPK1_PLABA 3Q5IA A0A509AHB6 38 518 523.0 ANP:61634 ATPlike Active DFGin 6.767 14.466 BLAminus -128.23, -176.48 60.5, 79.46 -95.96, 19.56 285.65, 75.94 -57.69, -30.19 in-in in 9.237 Saltbr-in 3.124 HRD-in -79.9, -50.9 74.57, -2.92 in-in-in SNCiii in-in ActLoopNT-in 2.988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.44, 148.94 APE9-dihe-na 143.23, -165.03 APE8-dihe-in -126.86, 133.51 APE8-rot-in 304.61 APE67-dihe-in -56.9, -32.89 -45.51, -52.84 APE12-dist-in 8.589 APE11-dist-in 11.465 APE10-dist-in 5.667 APE9-dist-in 3.634 None None None XRAY 2.1 0.197 0.25 A 504 461 18 0 0 0 [[57, 324]] 1.0 3q5i Plasmodium berghei CAMK_CDPK1_PLABA CAMK 4e-85 291.5 4 256 253 210 211 212 214 216 86 115 119 187 189 188 190 248 237 232 231 230 229 228 227 226 145 Calcium-dependent protein kinase 1
CMGC PSTK1 Q8IL19_PLAF7 3LLTA Q8IL19 535 875 881.0 ANP:877 ATPlike Active DFGin 7.143 15.216 BLAminus -123.92, -179.42 67.73, 65.46 -96.96, 21.34 280.85, 86.26 -60.95, -43.39 in-in in 9.013 Saltbr-in 2.621 HRD-in -67.76, -41.54 71.0, -10.38 in-in-in SNCiii in-in ActLoopNT-in 2.854 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.91, 173.39 APE9-dihe-na 75.57, 154.71 APE8-dihe-in -70.15, 136.15 APE8-rot-in 300.24 APE67-dihe-in -71.32, -17.13 -39.04, -49.24 APE12-dist-in 13.205 APE11-dist-in 11.39 APE10-dist-in 7.514 APE9-dist-in 2.941 None None None XRAY 2.5 0.225 0.267 A 360 341 0 0 0 0 [[552, 874]] 1.0 3llt Plasmodium falciparum CMGC_PSTK1_PLAF7 CMGC 8.3e-71 244.6 2 301 300 719 720 721 723 725 581 596 600 674 676 675 677 756 744 739 738 737 736 735 734 733 631 Protein serine/threonine kinase-1
STE TAOK2 TAOK2_RAT 1U5RA Q9JLS3 12 320 1235.0 ATP:411 ATPlike Active DFGin 6.99 14.24 BLAminus -128.27, -174.18 56.24, 80.49 -99.99, 21.83 293.09, 83.93 -60.11, -26.41 in-in in 8.687 Saltbr-in 2.887 HRD-in -75.95, -53.43 76.2, -2.14 in-in-in SNCiii in-in ActLoopNT-in 2.767 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.19, 153.0 APE9-dihe-na 135.08, -166.49 APE8-dihe-in -116.65, 119.51 APE8-rot-in 301.53 APE67-dihe-in -56.87, -24.9 -27.41, -63.55 APE12-dist-in 8.446 APE11-dist-in 11.391 APE10-dist-in 5.507 APE9-dist-in 3.279 None SEP181 SEP181 XRAY 2.1 0.211 0.244 A 348 309 0 0 0 0 [[28, 281]] 1.0 1u5r Rattus norvegicus STE_TAOK2_RAT STE 1.4e-89 305.8 2 257 256 168 169 170 172 174 57 76 80 148 150 149 151 207 192 187 186 185 184 183 182 181 106 Serine/threonine-protein kinase TAO2
STE TAOK2 TAOK2_RAT 1U5RB Q9JLS3 12 320 1235.0 ATP:412 ATPlike Active DFGin 6.763 13.896 BLAminus -129.03, -178.62 56.08, 82.23 -96.99, 22.88 295.53, 83.61 -63.46, -23.11 in-in in 8.772 Saltbr-in 2.623 HRD-in -71.62, -50.86 71.95, 2.83 in-in-in SNCiii in-in ActLoopNT-in 2.776 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.4, 155.39 APE9-dihe-na 130.83, -165.29 APE8-dihe-in -116.7, 116.24 APE8-rot-in 302.47 APE67-dihe-in -61.68, -22.51 -24.84, -62.59 APE12-dist-in 8.905 APE11-dist-in 11.02 APE10-dist-in 5.282 APE9-dist-in 3.304 None SEP181 SEP181 XRAY 2.1 0.211 0.244 B 348 309 0 0 0 0 [[28, 281]] 1.0 1u5r Rattus norvegicus STE_TAOK2_RAT STE 1.4e-89 305.8 2 257 256 168 169 170 172 174 57 76 80 148 150 149 151 207 192 187 186 185 184 183 182 181 106 Serine/threonine-protein kinase TAO2
CMGC SKY1 SKY1_YEAST 1Q8YA Q03656 144 737 742.0 ADP:60810 ATPlike Active DFGin 5.554 12.776 BLAminus -120.8, -179.55 50.32, 80.87 -92.72, 24.06 294.38, 19.86 -63.4, -18.16 in-in in 8.712 Saltbr-in 2.74 HRD-in -75.73, -45.78 71.18, -6.61 in-in-in SNCiii in-in ActLoopNT-in 2.965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.41, 175.98 APE9-dihe-na 63.08, 152.12 APE8-dihe-in -90.87, 131.26 APE8-rot-in 290.95 APE67-dihe-in -56.18, -26.85 -9.03, -76.03 APE12-dist-in 12.534 APE11-dist-in 10.496 APE10-dist-in 7.507 APE9-dist-in 2.99 None None None XRAY 2.05 0.209 0.244 A 373 351 11 0 0 0 [[158, 706]] 1.0 1q8y Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
CMGC SKY1 SKY1_YEAST 1Q97A Q03656 144 737 742.0 ATP:60485 ATPlike Active DFGin 5.605 12.648 BLAminus -113.61, -176.06 45.65, 81.54 -92.49, 25.33 294.84, 21.0 -61.4, -14.56 in-in in 8.92 Saltbr-in 2.91 HRD-in -73.18, -42.39 69.86, -2.96 in-in-in SNCiii in-in ActLoopNT-in 2.985 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -115.18, 168.88 APE9-dihe-na 68.54, 141.02 APE8-dihe-in -74.6, 131.99 APE8-rot-in 300.34 APE67-dihe-in -58.79, -28.16 -13.13, -73.4 APE12-dist-in 12.586 APE11-dist-in 10.498 APE10-dist-in 7.631 APE9-dist-in 3.163 None None None XRAY 2.3 0.215 0.264 A 373 351 11 0 0 0 [[158, 706]] 1.0 1q97 Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
CMGC SKY1 SKY1_YEAST 1Q99A Q03656 143 737 742.0 ANP:60901 ATPlike Active DFGin 5.863 12.817 BLAminus -114.29, -177.44 55.8, 69.3 -86.87, 21.69 289.5, 16.74 -63.01, -13.14 in-in in 9.01 Saltbr-in 3.393 HRD-in -74.14, -46.77 73.71, -6.86 in-in-in SNCiii in-in ActLoopNT-in 2.983 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.75, 166.8 APE9-dihe-na 68.75, 148.0 APE8-dihe-in -82.45, 139.06 APE8-rot-in 296.77 APE67-dihe-in -63.19, -13.43 -18.75, -76.87 APE12-dist-in 12.636 APE11-dist-in 10.441 APE10-dist-in 7.678 APE9-dist-in 2.996 None None None XRAY 2.11 0.22 0.26 A 373 354 9 0 0 0 [[158, 706]] 1.0 1q99 Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
CMGC SKY1 SKY1_YEAST 1Q99B Q03656 142 737 742.0 ANP:60902 ATPlike Active DFGin 6.007 13.076 BLAminus -119.51, 178.42 55.8, 73.86 -88.54, 22.76 281.2, 12.04 -67.31, -20.83 in-in in 8.991 Saltbr-in 3.413 HRD-in -77.35, -48.77 76.96, -6.7 in-in-in SNCiii in-in ActLoopNT-in 3.054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.48, 168.06 APE9-dihe-na 68.34, 160.67 APE8-dihe-in -99.08, 126.68 APE8-rot-in 289.43 APE67-dihe-in -64.6, -22.58 -5.08, -74.37 APE12-dist-in 12.556 APE11-dist-in 10.321 APE10-dist-in 7.788 APE9-dist-in 3.158 None None None XRAY 2.11 0.22 0.26 B 373 364 0 0 0 0 [[158, 706]] 1.0 1q99 Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
OTHER BUD32 BUD32_YEAST 4WW7A P53323 4 257 261.0 AMP:301 ATPlike Active DFGin 6.607 15.107 BLAminus -125.65, 168.23 67.12, 79.12 -101.96, 21.21 282.36, 92.63 -52.39, -37.98 in-in in 7.952 Saltbr-in 3.029 HRD-in -80.86, -48.82 95.12, -20.58 in-in-na SNCiia in-na ActLoopNT-in 2.886 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -64.64, -46.2 APE9-dihe-na -61.22, -39.41 APE8-dihe-na -68.4, -38.62 APE8-rot-na 171.99 APE67-dihe-na -60.22, -42.81 -57.37, -50.5 APE12-dist-na 15.675 APE11-dist-na 11.246 APE10-dist-na 14.76 APE9-dist-na 11.687 None None None XRAY 1.669 0.194 0.213 A 261 237 21 0 0 0 [[17, 261]] 1.0 4ww7 Saccharomyces cerevisiae OTHER_BUD32_YEAST TP53RK 5e-44 156.6 8 224 217 181 182 183 185 187 52 76 80 158 160 159 161 198 204 199 198 197 196 195 194 193 107 EKC/KEOPS complex subunit BUD32
OTHER BUD32 BUD32_YEAST 4WW9A P53323 4 259 261.0 ADP:302 ATPlike Active DFGin 6.618 15.283 BLAminus -128.14, 172.87 62.95, 73.82 -100.2, 23.36 281.69, 91.54 -52.55, -36.42 in-in in 7.602 Saltbr-in 2.744 HRD-in -80.98, -51.42 97.59, -12.36 in-in-na SNCiia in-na ActLoopNT-in 2.852 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -61.46, -46.34 APE9-dihe-na -60.52, -40.33 APE8-dihe-na -68.91, -38.47 APE8-rot-na 168.71 APE67-dihe-na -62.48, -38.16 -54.4, -51.68 APE12-dist-na 15.732 APE11-dist-na 11.179 APE10-dist-na 14.687 APE9-dist-na 11.734 None None None XRAY 1.951 0.18 0.209 A 261 238 20 0 0 0 [[17, 261]] 1.0 4ww9 Saccharomyces cerevisiae OTHER_BUD32_YEAST TP53RK 5e-44 156.6 8 224 217 181 182 183 185 187 52 76 80 158 160 159 161 198 204 199 198 197 196 195 194 193 107 EKC/KEOPS complex subunit BUD32
TKL NCGRLOCUS634 A0ACD6BAX3_9POAL 8HO6A A0ACD6BAX3 7 305 312.0 ATP:60401 ATPlike Active DFGin 6.377 15.619 BLAminus -139.79, 171.9 63.28, 66.12 -93.24, 62.65 279.35, 60.61 -82.08, -30.35 in-in in 8.644 Saltbr-in 2.728 HRD-in -60.88, -41.53 70.8, -58.95 in-in-in SNCiii in-in ActLoopNT-in 2.72 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.65, 146.26 APE9-dihe-na 148.14, -156.83 APE8-dihe-in -124.83, 132.59 APE8-rot-in 314.24 APE67-dihe-inflip 93.19, -27.63 -56.53, 137.58 APE12-dist-in 9.991 APE11-dist-in 11.771 APE10-dist-in 6.261 APE9-dist-in 5.587 None TPO184,SEP187,TPO188 TPO184,SEP187,TPO188 XRAY 2.1 0.206 0.234 A 326 281 18 0 0 2 [[22, 302]] 1.0 8ho6 Saccharum hybrid cultivar TKL_NCGRLOCUS634_9POAL TKL 3.7e-60 209.7 4 266 263 170 171 172 174 176 58 74 78 150 152 151 153 212 200 195 194 193 192 191 190 189 104 ScRIPK kinase protein
CK1 CKI1 CKI1_SCHPO 1CSNA P40233 6 298 446.0 ATP:299 ATPlike Active DFGin 6.422 13.79 BLAminus -124.8, 177.22 63.85, 88.12 -109.85, 36.77 298.25, 97.14 -71.61, -21.33 in-in in 8.04 Saltbr-in 3.086 HRD-in -68.74, -48.02 63.6, 9.84 in-in-in SNCiii in-in ActLoopNT-in 2.815 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -97.61, -90.82 APE9-dihe-na -65.25, -165.09 APE8-dihe-in -55.42, 111.92 APE8-rot-in 313.89 APE67-dihe-in -55.02, -31.3 -55.98, -42.83 APE12-dist-in 12.741 APE11-dist-in 13.007 APE10-dist-in 7.16 APE9-dist-in 4.794 None None None XRAY 2.0 0.207 999.0 A 298 293 0 0 0 0 [[12, 280]] 1.0 1csn Schizosaccharomyces pombe CK1_CKI1_SCHPO CK1 8e-95 323.1 1 261 261 153 154 155 157 159 41 55 59 128 130 129 131 200 188 183 182 181 180 179 178 177 86 Casein kinase I homolog 1
AGC PRKACA KAPCA_PIG 1CDKA P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.843 14.33 BLAminus -113.76, -166.2 47.38, 80.03 -85.76, 16.06 278.85, 56.4 -55.46, -28.11 in-in in 9.034 Saltbr-in 2.899 HRD-in -94.66, -56.81 78.16, -3.52 in-in-in SNCiii in-in ActLoopNT-in 2.985 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.51, 155.2 APE9-dihe-na 137.51, -153.75 APE8-dihe-in -125.49, 136.2 APE8-rot-in 297.83 APE67-dihe-in -73.46, -24.38 -35.73, -51.43 APE12-dist-in 7.997 APE11-dist-in 11.418 APE10-dist-in 5.766 APE9-dist-in 3.642 None TPO198 TPO198 XRAY 2.0 0.197 999.0 A 350 343 0 0 0 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_PIG 1CDKB P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.907 14.511 BLAminus -124.27, -171.72 50.82, 76.29 -83.58, 17.26 280.88, 62.25 -47.74, -29.83 in-in in 8.889 Saltbr-in 2.883 HRD-in -87.48, -57.48 77.49, 1.67 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 159.84 APE9-dihe-na 137.3, -140.74 APE8-dihe-in -136.57, 132.27 APE8-rot-in 304.84 APE67-dihe-in -69.16, -27.96 -34.59, -53.92 APE12-dist-in 8.348 APE11-dist-in 11.514 APE10-dist-in 6.08 APE9-dist-in 3.744 None TPO198 TPO198 XRAY 2.0 0.197 999.0 B 350 343 0 0 0 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CMGC TVAG125560 A2F9N1_TRIV3 9AV7A A2F9N1 15 318 320.0 ANP:401 ATPlike Active DFGin 7.636 16.424 BLAminus -120.42, -177.29 61.53, 69.44 -89.47, 18.08 296.84, 80.84 -66.47, -28.11 in-in in 9.462 Saltbr-in 3.092 HRD-in -77.85, -46.91 69.04, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.954 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.39, -177.21 APE9-dihe-na 62.4, -175.9 APE8-dihe-in -115.65, 153.97 APE8-rot-in 297.25 APE67-dihe-inflip 82.79, -6.3 -53.46, 134.7 APE12-dist-in 12.695 APE11-dist-in 10.496 APE10-dist-in 6.317 APE9-dist-in 3.013 None None None XRAY 2.1 0.202 0.246 A 328 304 0 0 0 0 [[27, 312]] 1.0 9av7 Trichomonas vaginalis CMGC_TVAG125560_TRIV3 CMGC 2.3e-51 180.8 1 301 301 162 163 164 166 168 56 69 73 141 143 142 144 202 189 184 183 182 181 180 179 178 102 non-specific serine/threonine protein kinase
CMGC ACK2 CSK2A_MAIZE 1DS5A P28523 1 328 332.0 AMP:60501 ATPlike Active DFGin 7.256 16.138 BLAminus -131.0, -177.8 59.5, 94.79 -110.09, 23.49 292.94, 70.46 -65.1, -12.46 in-in in 9.41 Saltbr-in 2.992 HRD-in -75.82, -4.13 22.93, 18.86 in-in-in SNCiii in-in ActLoopNT-in 2.927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, -170.21 APE9-dihe-na 48.23, -163.7 APE8-dihe-in -120.52, 135.99 APE8-rot-in 299.66 APE67-dihe-in -32.14, -36.61 -18.26, -83.73 APE12-dist-in 12.442 APE11-dist-in 10.293 APE10-dist-in 6.391 APE9-dist-in 3.166 None None None XRAY 3.16 0.214 0.289 A 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha
CMGC ACK2 CSK2A_MAIZE 1DS5B P28523 1 328 332.0 AMP:60801 ATPlike Active DFGin 7.364 16.317 BLAminus -130.6, -175.34 56.5, 69.06 -85.22, 18.36 296.09, 73.67 -62.25, -12.27 in-in in 9.134 Saltbr-in 2.468 HRD-in -78.74, -8.85 28.88, 23.14 in-in-in SNCiii in-in ActLoopNT-in 2.85 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.31, -172.94 APE9-dihe-na 48.86, -163.66 APE8-dihe-in -122.01, 142.21 APE8-rot-in 298.66 APE67-dihe-in -27.41, -40.26 -18.35, -90.48 APE12-dist-in 12.513 APE11-dist-in 10.354 APE10-dist-in 6.441 APE9-dist-in 3.101 None None None XRAY 3.16 0.214 0.289 B 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha
CMGC ACK2 CSK2A_MAIZE 1DS5C P28523 1 328 332.0 AMP:60601 ATPlike Active DFGin 7.431 16.3 BLAminus -130.04, -171.91 47.17, 91.25 -104.25, 20.64 295.37, 72.57 -63.12, -7.55 in-in in 9.164 Saltbr-in 2.64 HRD-in -79.02, -3.04 26.4, 20.9 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.73, -170.98 APE9-dihe-na 48.52, -163.45 APE8-dihe-in -120.17, 138.04 APE8-rot-in 300.76 APE67-dihe-in -34.03, -36.56 -18.28, -84.34 APE12-dist-in 12.439 APE11-dist-in 10.299 APE10-dist-in 6.441 APE9-dist-in 3.093 None None None XRAY 3.16 0.214 0.289 C 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha
CMGC ACK2 CSK2A_MAIZE 1DS5D P28523 1 328 332.0 AMP:60701 ATPlike Active DFGin 7.269 16.174 BLAminus -138.27, -179.17 62.24, 74.19 -94.05, 17.43 296.9, 73.95 -62.87, -11.79 in-in in 9.511 Saltbr-in 2.483 HRD-in -81.25, -4.13 24.81, 26.82 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.11, -172.61 APE9-dihe-na 51.23, -160.96 APE8-dihe-in -124.78, 137.86 APE8-rot-in 294.35 APE67-dihe-in -36.36, -34.26 -18.24, -83.45 APE12-dist-in 12.473 APE11-dist-in 10.246 APE10-dist-in 6.365 APE9-dist-in 3.133 None None None XRAY 3.16 0.214 0.289 D 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha

All / Activity_Active / ATPlike

Total number of chains: 132
Active chains: 132
Total number of genes: 27
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 132 100.0% 6EM7A

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC CKA1 CSK21_ARATH 6XX7A Q08467 77 406 409.0 ANP:60401 ATPlike Active DFGin 7.522 16.054 BLAminus -117.69, -174.69 54.04, 89.21 -108.75, 22.96 298.46, 82.8 -72.45, -17.87 in-in in 9.197 Saltbr-in 3.111 HRD-in -78.14, -48.74 65.41, 21.05 in-in-in SNCiii in-in ActLoopNT-in 2.834 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.12, 170.49 APE9-dihe-na 62.76, -171.63 APE8-dihe-in -114.91, 151.01 APE8-rot-in 304.83 APE67-dihe-in -66.49, -17.41 -50.66, -50.22 APE12-dist-in 12.585 APE11-dist-in 10.283 APE10-dist-in 6.188 APE9-dist-in 3.134 None None None XRAY 2.4 0.198 0.246 A 342 330 0 0 0 0 [[110, 395]] 1.0 6xx7 Arabidopsis thaliana CMGC_CKA1_ARATH CMGC 2.6e-65 226.5 1 301 301 245 246 247 249 251 139 152 156 224 226 225 227 285 272 267 266 265 264 263 262 261 185 Casein kinase II subunit alpha-1
TKL BRI1 BRI1_ARATH 5LPBA O22476 867 1160 1196.0 ADP:1201 ATPlike Active DFGin 5.075 15.058 BLAminus -134.68, 179.03 63.17, 81.59 -99.15, 20.06 285.86, 73.26 -60.78, -23.17 in-in in 8.649 Saltbr-in 3.148 HRD-in -69.16, -46.8 71.42, -2.74 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -107.78, 147.47 APE9-dihe-na 145.38, -170.04 APE8-dihe-in -133.78, 133.64 APE8-rot-in 306.07 APE67-dihe-inflip 102.35, -15.45 -46.22, 126.04 APE12-dist-in 9.248 APE11-dist-in 11.275 APE10-dist-in 5.497 APE9-dist-in 3.743 T872A TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 1.98 0.184 0.203 A 296 284 10 0 0 0 [[882, 1157]] 1.0 5lpb Arabidopsis thaliana TKL_BRI1_ARATH TKL 2e-63 220.4 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 5LPVA O22476 867 1160 1196.0 ANP:1200 ATPlike Active DFGin 5.144 14.999 BLAminus -125.7, -177.27 57.44, 79.7 -100.2, 28.83 289.11, 69.34 -64.8, -27.23 in-in in 8.616 Saltbr-in 2.692 HRD-in -72.39, -48.96 69.78, 4.25 in-in-in SNCiii in-in ActLoopNT-in 2.973 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.4, 152.93 APE9-dihe-na 138.14, -175.87 APE8-dihe-in -122.84, 131.25 APE8-rot-in 310.37 APE67-dihe-inflip 103.25, -12.92 -53.02, 126.73 APE12-dist-in 9.499 APE11-dist-in 11.435 APE10-dist-in 5.667 APE9-dist-in 3.671 T872A TPO1039,SEP1042,SEP1044 TPO1039,SEP1042,SEP1044 XRAY 2.7 0.193 0.233 A 296 285 9 0 0 0 [[882, 1157]] 1.0 5lpv Arabidopsis thaliana TKL_BRI1_ARATH TKL 2e-63 220.4 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 5LPYA O22476 867 1160 1196.0 ATP:1200 ATPlike Active DFGin 5.175 15.203 BLAminus -134.16, 179.9 60.37, 82.56 -100.0, 17.51 285.92, 71.71 -57.07, -20.27 in-in in 8.892 Saltbr-in 3.152 HRD-in -70.7, -49.88 77.86, -1.82 in-in-in SNCiii in-in ActLoopNT-in 2.908 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.47, 151.76 APE9-dihe-na 140.48, 176.99 APE8-dihe-in -121.99, 138.13 APE8-rot-in 307.91 APE67-dihe-inflip 92.03, -10.16 -52.79, 133.04 APE12-dist-in 9.609 APE11-dist-in 11.524 APE10-dist-in 5.721 APE9-dist-in 3.885 T872A TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 2.3 0.203 0.248 A 296 286 8 0 0 0 [[882, 1157]] 1.0 5lpy Arabidopsis thaliana TKL_BRI1_ARATH TKL 2e-63 220.4 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 5LPZA O22476 866 1160 1196.0 ADP:1200 ATPlike Active DFGin 5.281 15.229 BLAminus -133.61, -178.19 59.45, 71.09 -88.15, 19.11 288.53, 76.38 -60.79, -23.86 in-in in 8.633 Saltbr-in 2.829 HRD-in -68.17, -37.55 64.9, -2.92 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -69.74, 170.98 APE9-dihe-na 106.33, 162.6 APE8-dihe-in -102.72, 137.46 APE8-rot-in 305.68 APE67-dihe-inflip 102.78, -18.56 -57.05, 134.59 APE12-dist-in 9.342 APE11-dist-in 11.755 APE10-dist-in 5.72 APE9-dist-in 3.579 T872A TPO1039,SEP1042,SEP1044 TPO1039,SEP1042,SEP1044 XRAY 2.48 0.226 0.253 A 332 286 9 0 0 0 [[882, 1157]] 1.0 5lpz Arabidopsis thaliana TKL_BRI1_ARATH TKL 3e-63 219.9 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4OH4A O22476 863 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.109 14.621 BLAminus -140.27, -170.9 60.42, 81.58 -96.75, 17.94 285.65, 72.49 -62.14, -24.45 in-in in 8.43 Saltbr-in 2.981 HRD-in -67.48, -45.07 71.79, 0.23 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.28, 137.25 APE9-dihe-na 143.97, 175.71 APE8-dihe-in -113.05, 131.41 APE8-rot-in 300.18 APE67-dihe-inflip 103.6, -22.59 -52.56, 134.8 APE12-dist-in 10.688 APE11-dist-in 12.06 APE10-dist-in 6.328 APE9-dist-in 4.124 None TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 2.25 0.203 0.236 A 333 292 6 0 0 0 [[882, 1157]] 1.0 4oh4 Arabidopsis thaliana TKL_BRI1_ARATH TKL 3e-63 219.8 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4OH4B O22476 867 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.028 14.866 BLAminus -128.92, -179.57 66.05, 81.1 -97.08, 13.19 285.07, 69.22 -52.61, -27.46 in-in in 8.604 Saltbr-in 2.585 HRD-in -68.96, -46.37 73.67, -10.15 in-in-in SNCiii in-in ActLoopNT-in 2.87 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.43, 142.85 APE9-dihe-na 162.33, 170.81 APE8-dihe-in -132.62, 128.73 APE8-rot-in 297.7 APE67-dihe-inflip 104.71, -30.59 -48.41, 132.44 APE12-dist-in 9.471 APE11-dist-in 10.311 APE10-dist-in 5.146 APE9-dist-in 4.053 None TPO1039,SEP1042,SEP1044,SEP1060 TPO1039,SEP1042,SEP1044,SEP1060 XRAY 2.25 0.203 0.236 B 333 283 11 0 0 0 [[882, 1157]] 1.0 4oh4 Arabidopsis thaliana TKL_BRI1_ARATH TKL 3e-63 219.8 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4Q5JA O22476 863 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.066 14.74 BLAminus -137.9, 174.67 63.19, 85.3 -100.14, 20.42 284.87, 74.71 -62.5, -33.31 in-in in 8.354 Saltbr-in 3.257 HRD-in -68.22, -43.45 65.77, 3.93 in-in-in SNCiii in-in ActLoopNT-in 2.662 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -108.48, 139.01 APE9-dihe-na 175.24, 173.84 APE8-dihe-in -115.42, 129.74 APE8-rot-in 289.59 APE67-dihe-inflip 96.87, -1.52 -53.59, 124.31 APE12-dist-in 10.51 APE11-dist-in 12.065 APE10-dist-in 6.236 APE9-dist-in 4.467 None TPO1039,SEP1042,SEP1044,SEP1060 MSE925,MSE928,MSE959,MSE1010,MSE1030,MSE1034,MSE1037,TPO1039,SEP1042,SEP1044,SEP1060,MSE1117,MSE1148,MSE1152,MSE1154 XRAY 2.772 0.203 0.259 A 341 287 11 0 0 0 [[882, 1157]] 1.0 4q5j Arabidopsis thaliana TKL_BRI1_ARATH TKL 3.2e-63 219.7 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
TKL BRI1 BRI1_ARATH 4Q5JB O22476 867 1160 1196.0 ANP:61201 ATPlike Active DFGin 5.259 14.8 BLAminus -126.47, -178.56 58.45, 93.89 -112.89, 22.9 283.23, 71.66 -57.4, -19.56 in-in in 8.732 Saltbr-in 3.184 HRD-in -81.55, -35.96 67.72, -5.15 in-in-in SNCiii in-in ActLoopNT-in 2.775 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.14, 134.16 APE9-dihe-na 157.62, 164.27 APE8-dihe-in -126.08, 123.8 APE8-rot-in 304.99 APE67-dihe-inflip 120.44, -28.11 -46.98, 122.06 APE12-dist-in 9.403 APE11-dist-in 10.636 APE10-dist-in 5.512 APE9-dist-in 4.081 None TPO1039,SEP1042,SEP1044,SEP1060 MSE925,MSE928,MSE959,MSE1010,MSE1030,MSE1034,MSE1037,TPO1039,SEP1042,SEP1044,SEP1060,MSE1117,MSE1148,MSE1152,MSE1154 XRAY 2.772 0.203 0.259 B 341 283 11 0 0 0 [[882, 1157]] 1.0 4q5j Arabidopsis thaliana TKL_BRI1_ARATH TKL 3.2e-63 219.7 4 266 263 1026 1027 1028 1030 1032 911 927 931 1006 1008 1007 1009 1068 1056 1051 1050 1049 1048 1047 1046 1045 957 Protein BRASSINOSTEROID INSENSITIVE 1
AGC GRK1 GRK1_BOVIN 3T8OA P28327 30 532 561.0 ATP:562 ATPlike Active DFGin 6.784 13.652 BLAminus -147.61, 176.5 66.51, 86.5 -106.39, 20.07 278.45, 121.96 -78.51, -8.51 in-in in 9.131 Saltbr-in 2.946 HRD-in -72.08, -59.57 74.93, 15.13 in-in-in SNCiii in-in ActLoopNT-in 3.034 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.6, 145.4 APE9-dihe-na 140.82, -165.62 APE8-dihe-in -114.33, 123.31 APE8-rot-in 302.45 APE67-dihe-inflip 90.49, -9.25 -48.36, 136.06 APE12-dist-in 10.419 APE11-dist-in 11.645 APE10-dist-in 5.795 APE9-dist-in 4.276 L166K None None XRAY 2.5 0.209 0.245 A 543 493 0 0 0 0 [[187, 452]] 1.0 3t8o Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4WA P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 6.587 13.314 BLAminus -157.51, 175.0 67.79, 80.23 -106.97, 21.1 277.77, 138.55 -72.95, -18.52 in-in in 8.671 Saltbr-in 2.659 HRD-in -67.86, -51.97 60.46, 12.85 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.73, 153.77 APE9-dihe-na 125.45, -175.95 APE8-dihe-in -101.44, 127.92 APE8-rot-in 301.93 APE67-dihe-inflip 97.46, -21.92 -46.81, 133.28 APE12-dist-in 10.007 APE11-dist-in 11.248 APE10-dist-in 5.534 APE9-dist-in 3.508 None TPO8 TPO8 XRAY 2.7 0.192 999.0 A 543 494 0 0 0 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4WB P28327 5 533 561.0 ATP:562 ATPlike Active DFGin 5.963 13.111 BLAminus -155.04, 178.49 64.64, 79.84 -103.28, 19.03 277.57, 109.21 -72.3, -19.68 in-in in 8.548 Saltbr-in 2.84 HRD-in -67.79, -54.67 64.69, 11.83 in-in-in SNCiii in-in ActLoopNT-in 2.958 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.45, 154.48 APE9-dihe-na 126.08, -175.35 APE8-dihe-in -101.18, 126.91 APE8-rot-in 300.91 APE67-dihe-inflip 94.23, -17.08 -47.18, 130.86 APE12-dist-in 10.103 APE11-dist-in 11.254 APE10-dist-in 5.545 APE9-dist-in 3.534 None TPO8 TPO8 XRAY 2.7 0.192 999.0 B 543 519 0 0 0 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4XA P28327 30 533 561.0 ATP:562 ATPlike Active DFGin 6.392 13.294 BLAminus -153.36, -178.73 56.38, 83.66 -101.23, 19.01 282.86, 141.85 -58.01, -33.04 in-in in 8.623 Saltbr-in 2.825 HRD-in -65.41, -52.58 62.44, 13.36 in-in-in SNCiii in-in ActLoopNT-in 2.96 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.48, 144.22 APE9-dihe-na 128.55, -174.69 APE8-dihe-in -103.7, 129.98 APE8-rot-in 314.1 APE67-dihe-inflip 101.04, -22.84 -50.28, 132.61 APE12-dist-in 10.283 APE11-dist-in 11.237 APE10-dist-in 5.726 APE9-dist-in 3.827 None None None XRAY 2.9 0.193 999.0 A 543 496 0 0 0 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4XB P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 5.903 13.063 BLAminus -149.62, 174.69 57.3, 76.73 -95.24, 8.98 282.05, 96.12 -51.11, -35.54 in-in in 8.642 Saltbr-in 2.675 HRD-in -62.32, -48.48 63.55, 4.44 in-in-in SNCiii in-in ActLoopNT-in 3.043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.42, 143.72 APE9-dihe-na 129.46, -175.16 APE8-dihe-in -98.28, 125.3 APE8-rot-in 312.69 APE67-dihe-inflip 98.15, -18.1 -45.11, 129.51 APE12-dist-in 10.201 APE11-dist-in 11.247 APE10-dist-in 5.61 APE9-dist-in 3.639 None None None XRAY 2.9 0.193 999.0 B 543 475 0 0 0 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C4ZA P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.913 13.235 BLAminus -149.46, 171.26 70.91, 78.39 -108.02, 16.47 270.55, 111.24 -69.43, -16.01 in-in in 8.736 Saltbr-in 2.716 HRD-in -71.08, -53.07 69.31, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.878 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.53, 147.45 APE9-dihe-na 134.96, -165.72 APE8-dihe-in -111.39, 128.56 APE8-rot-in 296.58 APE67-dihe-inflip 96.79, -17.75 -54.96, 131.39 APE12-dist-in 10.43 APE11-dist-in 11.113 APE10-dist-in 5.49 APE9-dist-in 3.542 None None None XRAY 1.84 0.193 999.0 A 543 493 0 0 0 0 [[187, 452]] 1.0 3c4z Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C50A P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.075 13.034 BLAminus -142.59, 172.43 68.85, 78.38 -104.12, 14.36 280.99, 104.76 -67.57, -15.07 in-in in 8.602 Saltbr-in 2.925 HRD-in -76.21, -52.36 64.46, 15.62 in-in-in SNCiii in-in ActLoopNT-in 2.795 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.66, 144.27 APE9-dihe-na 130.37, -165.26 APE8-dihe-in -104.68, 131.22 APE8-rot-in 300.48 APE67-dihe-inflip 92.29, -6.18 -56.88, 135.03 APE12-dist-in 10.685 APE11-dist-in 11.469 APE10-dist-in 5.876 APE9-dist-in 3.473 None None None XRAY 2.6 0.19 999.0 A 543 499 0 0 0 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C50B P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.078 13.068 BLAminus -140.52, 175.4 66.53, 77.05 -104.14, 18.55 279.39, 103.87 -67.23, -21.39 in-in in 8.532 Saltbr-in 2.721 HRD-in -71.74, -52.34 63.89, 11.32 in-in-in SNCiii in-in ActLoopNT-in 2.89 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.47, 143.37 APE9-dihe-na 137.53, -168.17 APE8-dihe-in -105.39, 125.32 APE8-rot-in 297.12 APE67-dihe-inflip 95.82, -17.57 -51.32, 135.4 APE12-dist-in 10.129 APE11-dist-in 11.115 APE10-dist-in 5.538 APE9-dist-in 3.418 None None None XRAY 2.6 0.19 999.0 B 543 496 0 0 0 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C51A P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.735 13.235 BLAminus -156.28, 178.74 57.85, 73.51 -84.14, -2.01 283.03, 106.57 -47.35, -22.99 in-in in 8.798 Saltbr-in 2.687 HRD-in -64.41, -45.82 69.5, -19.46 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.64, 142.5 APE9-dihe-na 155.52, -169.52 APE8-dihe-in -101.5, 135.25 APE8-rot-in 300.99 APE67-dihe-inflip 84.91, 4.53 -59.96, 128.0 APE12-dist-in 10.573 APE11-dist-in 11.541 APE10-dist-in 6.152 APE9-dist-in 3.937 None None None XRAY 3.55 0.281 999.0 A 543 487 0 0 0 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3C51B P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.785 13.187 BLAminus -156.29, 175.57 58.57, 74.43 -85.29, -1.69 285.99, 107.07 -47.38, -22.91 in-in in 8.696 Saltbr-in 2.792 HRD-in -66.67, -42.5 63.68, -15.39 in-in-in SNCiii in-in ActLoopNT-in 2.969 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.05, 141.93 APE9-dihe-na 155.26, -171.96 APE8-dihe-in -101.33, 138.35 APE8-rot-in 299.85 APE67-dihe-inflip 84.6, 5.24 -64.39, 128.67 APE12-dist-in 10.537 APE11-dist-in 11.598 APE10-dist-in 6.156 APE9-dist-in 3.94 None None None XRAY 3.55 0.281 999.0 B 543 461 20 0 0 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9A P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.852 13.484 BLAminus -151.04, 174.48 70.22, 99.25 -129.57, 18.73 275.22, 99.19 -61.63, -18.96 in-in in 8.961 Saltbr-in 3.127 HRD-in -61.98, -58.15 73.37, -3.42 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.32, 133.82 APE9-dihe-na 142.48, -169.15 APE8-dihe-in -104.33, 125.71 APE8-rot-in 302.67 APE67-dihe-inflip 104.42, -3.83 -50.74, 122.55 APE12-dist-in 10.356 APE11-dist-in 11.014 APE10-dist-in 5.5 APE9-dist-in 3.664 T8C,N480C None None XRAY 2.7 0.194 0.229 A 543 486 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9B P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.899 13.504 BLAminus -154.17, 173.67 70.5, 100.81 -132.54, 18.75 276.87, 97.69 -56.57, -24.02 in-in in 8.931 Saltbr-in 3.099 HRD-in -65.24, -58.34 73.4, -2.88 in-in-in SNCiii in-in ActLoopNT-in 2.934 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -166.53, 132.45 APE9-dihe-na 145.72, -169.79 APE8-dihe-in -103.09, 126.5 APE8-rot-in 303.38 APE67-dihe-inflip 99.94, -4.73 -52.12, 123.93 APE12-dist-in 10.368 APE11-dist-in 11.038 APE10-dist-in 5.525 APE9-dist-in 3.677 T8C,N480C None None XRAY 2.7 0.194 0.229 B 543 481 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9C P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.868 13.481 BLAminus -151.87, 172.48 72.03, 98.62 -128.19, 19.72 276.34, 98.38 -59.47, -19.79 in-in in 8.951 Saltbr-in 3.107 HRD-in -62.09, -58.44 72.04, -1.68 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.26, 134.05 APE9-dihe-na 142.83, -170.11 APE8-dihe-in -104.04, 126.58 APE8-rot-in 301.36 APE67-dihe-inflip 105.14, -2.81 -49.9, 120.73 APE12-dist-in 10.384 APE11-dist-in 11.018 APE10-dist-in 5.508 APE9-dist-in 3.673 T8C,N480C None None XRAY 2.7 0.194 0.229 C 543 482 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC GRK1 GRK1_BOVIN 3QC9D P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.923 13.517 BLAminus -151.29, 174.11 71.25, 99.27 -130.54, 20.81 276.77, 98.72 -58.99, -24.3 in-in in 8.931 Saltbr-in 3.091 HRD-in -63.44, -57.63 71.87, -0.43 in-in-in SNCiii in-in ActLoopNT-in 2.927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.95, 134.69 APE9-dihe-na 141.2, -168.54 APE8-dihe-in -103.28, 126.55 APE8-rot-in 303.76 APE67-dihe-inflip 102.49, -2.5 -51.29, 121.62 APE12-dist-in 10.397 APE11-dist-in 11.044 APE10-dist-in 5.513 APE9-dist-in 3.693 T8C,N480C None None XRAY 2.7 0.194 0.229 D 543 486 0 0 0 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4 260 257 331 332 333 335 337 216 235 239 311 313 312 314 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
AGC PRKACA KAPCA_BOVIN 9DW9G P00517 13 351 351.0 ATP:401 ATPlike Active DFGin 6.569 15.126 BLAminus -133.9, -169.96 59.46, 64.31 -83.85, 33.99 275.29, 73.58 -66.33, -24.36 in-in in 9.499 Saltbr-in 3.217 HRD-in -92.3, -53.34 68.25, 14.14 in-in-in SNCiii in-in ActLoopNT-in 3.08 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.91, 151.76 APE9-dihe-na 126.66, -174.62 APE8-dihe-in -92.84, 130.69 APE8-rot-in 299.41 APE67-dihe-in -68.55, -23.13 -58.33, -34.44 APE12-dist-in 8.703 APE11-dist-in 11.563 APE10-dist-in 6.17 APE9-dist-in 4.568 None TPO198 TPO198 EM 2.8 999.0 999.0 G 351 328 0 0 0 0 [[44, 298]] 1.0 9dw9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_BOVIN 1Q24A P00517 15 351 351.0 ATP:60400 ATPlike Active DFGin 5.983 14.319 BLAminus -113.95, 178.0 66.86, 85.15 -103.99, 32.82 274.7, 64.8 -65.44, -25.66 in-in in 8.779 Saltbr-in 2.742 HRD-in -93.22, -55.61 73.46, 14.95 in-in-in SNCiii in-in ActLoopNT-in 3.09 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.66, 162.77 APE9-dihe-na 133.15, -143.39 APE8-dihe-in -135.22, 127.61 APE8-rot-in 301.89 APE67-dihe-in -67.43, -30.61 -42.63, -46.05 APE12-dist-in 8.036 APE11-dist-in 11.447 APE10-dist-in 6.024 APE9-dist-in 3.486 V124A,L174M TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.202 0.25 A 350 337 0 0 0 0 [[44, 298]] 1.0 1q24 Bos taurus AGC_PRKACA_BOVIN AGC 4.8e-94 320.4 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CMGC CKA1 A0A1D8PUA2_CANAL 6O6QA A0A1D8PUA2 4 333 335.0 AMP:401 ATPlike Active DFGin 7.386 16.256 BLAminus -114.24, -174.82 59.27, 62.07 -85.23, 23.85 304.56, 80.46 -69.03, -20.65 in-in in 9.001 Saltbr-in 2.88 HRD-in -68.75, -45.06 62.13, 23.87 in-in-in SNCiii in-in ActLoopNT-in 3.222 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.59, 173.17 APE9-dihe-na 57.84, -166.47 APE8-dihe-in -122.64, 160.2 APE8-rot-in 318.49 APE67-dihe-in -66.36, -14.81 -53.74, -47.77 APE12-dist-in 12.507 APE11-dist-in 10.219 APE10-dist-in 6.094 APE9-dist-in 3.225 None None None XRAY 2.7 0.236 0.287 A 335 326 4 0 0 0 [[43, 327]] 1.0 6o6q Candida albicans CMGC_CKA1_CANAL CMGC 1.1e-62 217.9 1 301 301 178 179 180 182 184 72 85 89 157 159 158 160 218 205 200 199 198 197 196 195 194 118 Casein kinase II subunit alpha
CMGC CKA1 A0A1D8PUA2_CANAL 6O6QB A0A1D8PUA2 5 333 335.0 AMP:401 ATPlike Active DFGin 7.292 15.98 BLAminus -125.13, -179.74 57.94, 64.68 -85.91, 27.32 303.1, 76.17 -70.46, -30.29 in-in in 9.011 Saltbr-in 2.813 HRD-in -81.71, -46.62 63.63, 27.36 in-in-in SNCiii in-in ActLoopNT-in 2.902 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.56, 167.57 APE9-dihe-na 58.76, -171.72 APE8-dihe-in -113.79, 160.74 APE8-rot-in 318.5 APE67-dihe-in -64.2, -12.3 -53.09, -54.06 APE12-dist-in 12.689 APE11-dist-in 10.132 APE10-dist-in 6.255 APE9-dist-in 3.214 None None None XRAY 2.7 0.236 0.287 B 335 325 4 0 0 0 [[43, 327]] 1.0 6o6q Candida albicans CMGC_CKA1_CANAL CMGC 1.1e-62 217.9 1 301 301 178 179 180 182 184 72 85 89 157 159 158 160 218 205 200 199 198 197 196 195 194 118 Casein kinase II subunit alpha
AGC PRKACA KAPCA_CRIGR 6EM7A P25321 11 351 351.0 ADP:60403 ATPlike Active DFGin 5.924 14.338 BLAminus -118.71, 173.1 68.53, 85.06 -96.18, 23.36 270.78, 55.34 -59.75, -28.55 in-in in 8.741 Saltbr-in 2.711 HRD-in -88.33, -53.93 74.88, 10.19 in-in-in SNCiii in-in ActLoopNT-in 2.967 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.73, 159.92 APE9-dihe-na 127.98, -160.75 APE8-dihe-in -119.5, 137.47 APE8-rot-in 298.57 APE67-dihe-in -59.39, -22.73 -49.47, -50.59 APE12-dist-in 8.05 APE11-dist-in 11.429 APE10-dist-in 5.809 APE9-dist-in 3.674 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.238 0.139 0.157 A 353 341 0 0 0 0 [[44, 298]] 1.0 6em7 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_CRIGR 6EMAA P25321 12 351 351.0 ATP:60401 ATPlike Active DFGin 6.847 14.028 BLAminus -121.3, 163.01 76.03, 95.19 -107.48, 29.41 285.05, 72.84 -63.27, -23.25 in-in in 8.581 Saltbr-in 2.912 HRD-in -88.06, -51.23 73.05, 9.34 in-in-in SNCiii in-in ActLoopNT-in 2.843 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.85, 162.03 APE9-dihe-na 127.51, -167.2 APE8-dihe-in -113.51, 133.85 APE8-rot-in 299.54 APE67-dihe-in -58.99, -24.47 -49.7, -50.19 APE12-dist-in 8.208 APE11-dist-in 11.434 APE10-dist-in 5.777 APE9-dist-in 3.585 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.88 0.184 0.213 A 353 340 0 0 0 0 [[44, 298]] 1.0 6ema Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_CRIGR 6ESAA P25321 11 351 351.0 AMP:60401 ATPlike Active DFGin 6.139 14.365 BLAminus -120.63, 169.73 70.22, 89.96 -100.72, 24.5 270.85, 56.09 -58.05, -28.66 in-in in 8.691 Saltbr-in 2.873 HRD-in -93.01, -53.86 73.79, 10.3 in-in-in SNCiii in-in ActLoopNT-in 2.964 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.44, 160.95 APE9-dihe-na 124.73, -163.46 APE8-dihe-in -117.05, 136.25 APE8-rot-in 299.26 APE67-dihe-in -59.89, -22.61 -49.24, -49.61 APE12-dist-in 8.091 APE11-dist-in 11.499 APE10-dist-in 5.822 APE9-dist-in 3.66 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.307 0.132 0.147 A 353 341 0 0 0 0 [[44, 298]] 1.0 6esa Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_CRIGR 6Y8CA P25321 13 351 351.0 ATP:60402 ATPlike Active DFGin 5.727 14.302 BLAminus -123.99, 172.57 69.5, 82.73 -92.15, 25.74 279.44, 63.0 -58.78, -31.82 in-in in 9.166 Saltbr-in 2.638 HRD-in -96.49, -52.39 69.1, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.28, 160.42 APE9-dihe-na 122.78, -169.96 APE8-dihe-in -106.17, 134.07 APE8-rot-in 304.81 APE67-dihe-in -60.24, -22.7 -48.33, -48.43 APE12-dist-in 8.044 APE11-dist-in 11.517 APE10-dist-in 5.939 APE9-dist-in 3.895 None TPO198,SEP339 TPO198,SEP339 XRAY 1.76 0.162 0.19 A 353 339 0 0 0 0 [[44, 298]] 1.0 6y8c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CMGC CK2 Q5KF69_CRYD1 6ISEA Q5KF69 5 331 336.0 ANP:403 ATPlike Active DFGin 7.339 16.208 BLAminus -129.3, -170.99 44.36, 71.77 -91.05, 22.67 299.01, 82.29 -66.02, -23.99 in-in in 9.482 Saltbr-in 3.336 HRD-in -65.48, -54.09 76.82, 9.27 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.0, -19.23 APE9-dihe-na -99.69, -172.72 APE8-dihe-in -80.09, 147.5 APE8-rot-in 301.93 APE67-dihe-in -61.24, -16.59 -47.75, -58.81 APE12-dist-in 12.687 APE11-dist-in 10.631 APE10-dist-in 6.144 APE9-dist-in 3.609 None None None XRAY 2.8 0.198 0.23 A 338 327 0 0 0 0 [[38, 323]] 1.0 6ise Cryptococcus deneoformans CMGC_CK2_CRYD1 CMGC 6e-64 222.0 1 301 301 173 174 175 177 179 67 80 84 152 154 153 155 213 200 195 194 193 192 191 190 189 113 Casein kinase II subunit alpha
CMGC CK2 Q5KF69_CRYD1 6ISEB Q5KF69 5 331 336.0 ANP:403 ATPlike Active DFGin 7.308 16.238 BLAminus -133.11, -171.48 44.36, 73.35 -91.98, 23.51 299.28, 79.86 -68.68, -21.78 in-in in 9.591 Saltbr-in 3.496 HRD-in -67.7, -51.8 75.87, 7.92 in-in-in SNCiii in-in ActLoopNT-in 2.976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.38, 168.0 APE9-dihe-na 74.76, -173.48 APE8-dihe-in -110.86, 148.66 APE8-rot-in 271.82 APE67-dihe-in -65.62, -23.31 -54.68, -45.78 APE12-dist-in 12.576 APE11-dist-in 10.311 APE10-dist-in 6.266 APE9-dist-in 3.367 None None None XRAY 2.8 0.198 0.23 B 338 327 0 0 0 0 [[38, 323]] 1.0 6ise Cryptococcus deneoformans CMGC_CK2_CRYD1 CMGC 6e-64 222.0 1 301 301 173 174 175 177 179 67 80 84 152 154 153 155 213 200 195 194 193 192 191 190 189 113 Casein kinase II subunit alpha
CMGC CKA1 J9VNH4_CRYN9 6KO6B J9VNH4 5 334 338.0 ANP:401 ATPlike Active DFGin 7.298 16.236 BLAminus -115.02, -165.9 52.87, 72.55 -94.97, 21.12 299.2, 77.23 -71.99, -18.35 in-in in 9.324 Saltbr-in 3.151 HRD-in -64.53, -49.64 63.27, 19.41 in-in-in SNCiii in-in ActLoopNT-in 3.055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.45, 156.98 APE9-dihe-na 76.83, -179.82 APE8-dihe-in -92.38, 159.35 APE8-rot-in 277.62 APE67-dihe-in -71.62, -13.46 -53.06, -52.26 APE12-dist-in 12.792 APE11-dist-in 10.474 APE10-dist-in 6.177 APE9-dist-in 3.249 None None None XRAY 2.4 0.238 0.268 B 338 330 0 0 0 0 [[38, 323]] 1.0 6ko6 Cryptococcus neoformans CMGC_CKA1_CRYN9 CMGC 6e-64 222.0 1 301 301 173 174 175 177 179 67 80 84 152 154 153 155 213 200 195 194 193 192 191 190 189 113 Casein kinase II subunit alpha
OTHER PK1 A0A097P1P8_GVCP 6VVGA A0A097P1P8 3 279 279.0 AMP:301 ATPlike Active DFGin 9.47 12.504 BLAminus -139.45, 174.39 59.11, 72.82 -82.01, 20.88 324.49, 136.4 -73.16, -16.8 na-na na 15.471 Saltbr-na 12.976 HRD-in -69.17, -49.37 73.82, 3.86 na-in-in SNCaii in-in ActLoopNT-in 2.866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.58, 157.03 APE9-dihe-na 90.57, -158.23 APE8-dihe-in -103.25, 120.97 APE8-rot-in 311.05 APE67-dihe-in -75.71, -2.76 -55.41, -39.8 APE12-dist-in 10.799 APE11-dist-in 12.039 APE10-dist-in 6.083 APE9-dist-in 4.885 None None None XRAY 2.01 0.195 0.225 A 279 267 10 0 0 0 [[17, 277]] 1.0 6vvg Cydia pomonella granulosis virus OTHER_PK1_GVCP CAMK 1.9e-45 161.2 8 256 249 159 160 161 163 165 49 62 66 138 140 139 141 195 183 178 177 176 175 174 173 172 92 PK-1
OTHER PK1 A0A097P1P8_GVCP 6VVGB A0A097P1P8 3 278 279.0 AMP:301 ATPlike Active DFGin 9.485 12.665 BLAminus -138.4, 172.21 59.64, 73.0 -83.58, 22.42 324.54, 137.78 -67.63, -19.86 na-na na 15.282 Saltbr-na 13.214 HRD-in -58.02, -51.7 78.84, -1.77 na-in-in SNCaii in-in ActLoopNT-in 2.858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.97, 161.51 APE9-dihe-na 88.81, -151.71 APE8-dihe-in -109.06, 113.8 APE8-rot-in 308.85 APE67-dihe-in -72.96, -2.91 -51.95, -43.87 APE12-dist-in 10.828 APE11-dist-in 12.169 APE10-dist-in 6.178 APE9-dist-in 4.697 None None None XRAY 2.01 0.195 0.225 B 279 264 12 0 0 0 [[17, 277]] 1.0 6vvg Cydia pomonella granulosis virus OTHER_PK1_GVCP CAMK 1.9e-45 161.2 8 256 249 159 160 161 163 165 49 62 66 138 140 139 141 195 183 178 177 176 175 174 173 172 92 PK-1
CAMK CAMKII KCC2A_DROME 5FG8A Q00168 7 275 530.0 ADP:301 ATPlike Active DFGin 5.883 14.23 BLAminus -120.35, -179.38 64.2, 77.37 -92.62, 22.59 287.14, 78.3 -59.18, -27.49 in-in in 8.996 Saltbr-in 2.798 HRD-in -79.26, -45.5 78.31, -3.25 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.29, 153.59 APE9-dihe-na 138.39, -158.82 APE8-dihe-in -123.15, 126.57 APE8-rot-in 291.32 APE67-dihe-in -61.12, -15.42 -38.96, -61.46 APE12-dist-in 10.208 APE11-dist-in 11.816 APE10-dist-in 6.289 APE9-dist-in 3.479 None None None XRAY 1.955 0.192 0.221 A 285 269 0 0 0 0 [[14, 272]] 1.0 5fg8 Drosophila melanogaster CAMK_CAMKII_DROME CAMK 6.3e-98 333.1 1 256 256 156 157 158 160 162 43 61 65 133 135 134 136 196 184 179 178 177 176 175 174 173 91 Calcium/calmodulin-dependent protein kinase type II alpha chain
CAMK CAMKII KCC2A_DROME 5H9BA Q00168 7 275 530.0 AN2:301 ATPlike Active DFGin 5.687 14.14 BLAminus -121.83, -177.58 63.45, 84.2 -103.14, 25.35 292.56, 80.33 -62.44, -18.79 in-in in 9.014 Saltbr-in 2.65 HRD-in -79.17, -42.13 69.98, 5.32 in-in-in SNCiii in-in ActLoopNT-in 3.047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.23, 154.68 APE9-dihe-na 138.91, -156.64 APE8-dihe-in -125.98, 126.82 APE8-rot-in 298.36 APE67-dihe-in -64.57, -17.97 -35.44, -64.1 APE12-dist-in 10.217 APE11-dist-in 11.689 APE10-dist-in 6.016 APE9-dist-in 3.419 None None None XRAY 2.25 0.204 0.222 A 285 269 0 0 0 0 [[14, 272]] 1.0 5h9b Drosophila melanogaster CAMK_CAMKII_DROME CAMK 6.3e-98 333.1 1 256 256 156 157 158 160 162 43 61 65 133 135 134 136 196 184 179 178 177 176 175 174 173 91 Calcium/calmodulin-dependent protein kinase type II alpha chain
CAMK CAMKII KCC2A_DROME 5HU3A Q00168 7 272 530.0 ADP:301 ATPlike Active DFGin 5.625 14.217 BLAminus -125.3, -175.54 57.54, 73.58 -90.7, 26.83 289.37, 84.29 -62.44, -29.23 in-in in 8.952 Saltbr-in 2.671 HRD-in -75.88, -45.31 74.57, -1.26 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.12, 157.18 APE9-dihe-na 139.99, -158.88 APE8-dihe-in -121.63, 130.83 APE8-rot-in 294.31 APE67-dihe-in -66.75, -12.95 -42.37, -59.45 APE12-dist-in 10.059 APE11-dist-in 11.766 APE10-dist-in 6.277 APE9-dist-in 3.564 D136N None None XRAY 1.885 0.194 0.228 A 285 266 0 0 0 0 [[14, 272]] 1.0 5hu3 Drosophila melanogaster CAMK_CAMKII_DROME CAMK 5.7e-97 329.9 1 256 256 156 157 158 160 162 43 61 65 133 135 134 136 196 184 179 178 177 176 175 174 173 91 Calcium/calmodulin-dependent protein kinase type II alpha chain
CAMK CDPK Q3HNM4_EIMTE 4YSJA Q3HNM4 26 499 505.0 ADP:60506 ATPlike Active DFGin 6.651 14.005 BLAminus -140.39, -165.72 52.75, 66.63 -84.34, 22.0 285.15, 82.54 -78.31, -16.63 in-in in 8.319 Saltbr-in 3.482 HRD-in -81.29, -53.0 84.02, -6.2 in-in-in SNCiii in-in ActLoopNT-in 2.898 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.58, 142.92 APE9-dihe-na 138.88, -163.22 APE8-dihe-in -136.98, 140.82 APE8-rot-in 303.29 APE67-dihe-in -62.88, -33.46 -45.59, -53.66 APE12-dist-in 9.144 APE11-dist-in 11.564 APE10-dist-in 5.99 APE9-dist-in 3.493 None None None XRAY 2.7 0.249 0.292 A 491 459 10 0 0 0 [[46, 303]] 1.0 4ysj Eimeria tenella CAMK_CDPK_EIMTE CAMK 6.1e-90 307.2 1 256 256 189 190 191 193 195 75 94 98 166 168 167 169 227 216 211 210 209 208 207 206 205 124 non-specific serine/threonine protein kinase
CAMK CDPK Q3HNM4_EIMTE 4YSJB Q3HNM4 26 499 505.0 ADP:60506 ATPlike Active DFGin 6.595 13.993 BLAminus -140.54, -165.92 54.1, 65.38 -84.49, 22.28 285.29, 82.38 -78.18, -16.85 in-in in 8.3 Saltbr-in 3.494 HRD-in -81.3, -52.72 84.55, -6.86 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.46, 142.21 APE9-dihe-na 137.64, -162.65 APE8-dihe-in -138.56, 141.54 APE8-rot-in 303.24 APE67-dihe-in -62.83, -32.98 -44.74, -55.37 APE12-dist-in 8.901 APE11-dist-in 11.534 APE10-dist-in 5.979 APE9-dist-in 3.505 None None None XRAY 2.7 0.249 0.292 B 491 462 10 0 0 0 [[46, 303]] 1.0 4ysj Eimeria tenella CAMK_CDPK_EIMTE CAMK 6.1e-90 307.2 1 256 256 189 190 191 193 195 75 94 98 166 168 167 169 227 216 211 210 209 208 207 206 205 124 non-specific serine/threonine protein kinase
TYR PTK2 FAK1_CHICK 6TY4A Q00944 34 686 1053.0 ANP:702 ATPlike Active DFGin 7.546 15.951 BLAminus -124.05, -151.88 51.86, 82.13 -107.99, 32.9 286.39, 85.0 -72.01, -36.58 in-in in 8.437 Saltbr-in 3.562 HRD-in -70.16, -30.0 74.19, -18.38 in-in-in SNCiii in-in ActLoopNT-in 2.815 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -86.31, 66.54 APE9-dihe-in -63.31, 139.75 APE8-dihe-in -64.41, 127.23 APE8-rot-na 22.65 APE67-dihe-in -56.19, -42.03 -70.19, -41.73 APE12-dist-na 11.489 APE11-dist-na 10.184 APE10-dist-na 13.636 APE9-dist-in 7.205 None None None EM 5.96 999.0 999.0 A 658 621 0 0 0 0 [[422, 678]] 1.0 6ty4 Gallus gallus TYR_PTK2_CHICK TYR 1.5e-91 312.7 1 260 260 563 564 565 567 569 454 471 475 543 545 544 546 604 592 587 586 585 584 583 582 581 500 Focal adhesion kinase 1
TYR PTK2 FAK1_CHICK 6TY4B Q00944 34 686 1053.0 ANP:702 ATPlike Active DFGin 7.546 15.95 BLAminus -124.03, -151.9 51.82, 82.14 -107.99, 32.89 286.33, 85.06 -71.97, -36.56 in-in in 8.436 Saltbr-in 3.562 HRD-in -70.15, -30.0 74.26, -18.38 in-in-in SNCiii in-in ActLoopNT-in 2.815 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -86.3, 66.56 APE9-dihe-in -63.34, 139.79 APE8-dihe-in -64.42, 127.23 APE8-rot-na 22.65 APE67-dihe-in -56.21, -42.01 -70.19, -41.71 APE12-dist-na 11.489 APE11-dist-na 10.183 APE10-dist-na 13.636 APE9-dist-in 7.205 None None None EM 5.96 999.0 999.0 B 658 621 0 0 0 0 [[422, 678]] 1.0 6ty4 Gallus gallus TYR_PTK2_CHICK TYR 1.5e-91 312.7 1 260 260 563 564 565 567 569 454 471 475 543 545 544 546 604 592 587 586 585 584 583 582 581 500 Focal adhesion kinase 1
TYR SRC SRC_CHICK 3DQWA P00523 255 533 533.0 AGS:534 ATPlike Active DFGin 6.357 14.133 BLAminus -133.72, -176.8 56.69, 80.14 -98.42, 17.02 297.52, 87.02 -49.14, -41.19 in-in in 7.931 Saltbr-in 2.687 HRD-in -86.31, -48.96 78.42, -4.92 in-in-in SNCiii in-in ActLoopNT-in 3.014 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -125.37, 137.46 APE9-dihe-in -129.59, 150.85 APE8-dihe-in -68.35, 111.94 APE8-rot-na 22.98 APE67-dihe-in -63.37, -24.29 -54.33, -47.45 APE12-dist-na 14.454 APE11-dist-na 9.918 APE10-dist-na 12.726 APE9-dist-in 6.835 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 A 286 279 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQWB P00523 255 533 533.0 AGS:534 ATPlike Active DFGin 6.515 14.112 BLAminus -130.32, -179.28 59.57, 78.46 -98.37, 14.52 296.04, 88.38 -51.47, -39.24 in-in in 7.861 Saltbr-in 2.594 HRD-in -92.73, -49.37 74.2, -0.04 in-in-in SNCiii in-in ActLoopNT-in 2.955 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -118.73, 138.44 APE9-dihe-in -131.19, 150.2 APE8-dihe-in -68.24, 113.76 APE8-rot-na 20.72 APE67-dihe-in -68.02, -21.16 -58.05, -42.12 APE12-dist-na 14.577 APE11-dist-na 10.068 APE10-dist-na 12.667 APE9-dist-in 6.835 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 B 286 279 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQWC P00523 258 533 533.0 AGS:534 ATPlike Active DFGin 7.23 15.586 BLAminus -138.39, -169.49 49.44, 64.48 -88.87, 22.55 279.28, 86.64 -59.44, -34.1 in-in in 7.666 Saltbr-in 3.046 HRD-in -87.18, -49.68 80.05, -15.46 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -114.69, 105.75 APE9-dihe-in -126.06, 131.23 APE8-dihe-in -49.28, 106.82 APE8-rot-na 333.72 APE67-dihe-in -71.67, -16.03 -52.29, -42.49 APE12-dist-na 14.071 APE11-dist-na 9.851 APE10-dist-na 10.947 APE9-dist-in 6.124 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 C 286 276 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQWD P00523 257 533 533.0 AGS:534 ATPlike Active DFGin 7.183 15.5 BLAminus -135.25, -176.07 62.11, 64.12 -89.05, 15.75 281.43, 79.51 -51.86, -37.09 in-in in 7.529 Saltbr-in 3.018 HRD-in -81.74, -56.17 86.4, -15.46 in-in-in SNCiii in-in ActLoopNT-in 2.971 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -120.41, 149.47 APE9-dihe-in -128.09, 155.96 APE8-dihe-in -55.17, 98.07 APE8-rot-na 334.76 APE67-dihe-in -67.99, -16.44 -49.1, -40.45 APE12-dist-na 15.071 APE11-dist-na 10.305 APE10-dist-na 13.293 APE9-dist-in 6.675 T338I PTR416 PTR416 XRAY 2.017 0.207 0.245 D 286 277 0 0 0 0 [[267, 518]] 1.0 3dqw Gallus gallus TYR_SRC_CHICK TYR 6.7e-94 319.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
TYR SRC SRC_CHICK 3DQXB P00523 259 533 533.0 AMP:2 ATPlike Active DFGin 6.808 14.815 BLAminus -123.08, -167.74 51.93, 60.88 -81.23, 10.84 295.11, 95.49 -43.33, -48.19 in-in in 7.906 Saltbr-in 3.425 HRD-in -73.53, -53.77 83.73, -6.08 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -120.36, 128.73 APE9-dihe-in -122.57, 114.22 APE8-dihe-in -63.43, 112.38 APE8-rot-na 23.41 APE67-dihe-in -72.31, -17.76 -46.16, -42.59 APE12-dist-na 10.885 APE11-dist-na 6.755 APE10-dist-na 9.999 APE9-dist-in 5.75 None None None XRAY 2.3 0.194 0.241 B 286 268 7 0 0 7 [[267, 518]] 1.0 3dqx Gallus gallus TYR_SRC_CHICK TYR 3.4e-94 320.9 1 260 260 403 404 405 407 409 295 310 314 383 385 384 386 444 432 427 426 425 424 423 422 421 339 Proto-oncogene tyrosine-protein kinase Src
OTHER LPL0262 Q5WZW9_LEGPL 5CKWA Q5WZW9 15 404 961.0 ANP:60501 ATPlike Active DFGin 5.948 12.719 BLAminus -133.44, 169.43 70.28, 94.79 -117.83, 12.87 299.33, 117.8 -55.88, -8.97 in-in in 6.71 Saltbr-in 2.716 HRD-na-Q -80.53, -48.66 73.11, 5.26 in-in-in SNCiii in-in ActLoopNT-in 2.927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -69.26, -22.18 APE9-dihe-na -101.55, 179.41 APE8-dihe-in -117.11, 122.15 APE8-rot-in 302.21 APE67-dihe-in -64.67, -9.61 -57.44, -37.84 APE12-dist-in 11.762 APE11-dist-in 9.709 APE10-dist-in 4.647 APE9-dist-in 3.347 None None None XRAY 2.49 0.207 0.258 A 451 378 5 0 0 0 [[75, 309]] 1.0 5ckw Legionella pneumophila OTHER_LPL0262_LEGPL NEK 4.8e-15 62.8 10 222 213 212 213 214 216 218 104 119 123 192 194 193 195 249 237 232 231 230 229 228 227 226 146 non-specific serine/threonine protein kinase
OTHER LPL0262 Q5WZW9_LEGPL 5CKWB Q5WZW9 1 404 961.0 ANP:60501 ATPlike Active DFGin 6.189 12.674 BLAminus -144.06, 165.73 65.65, 85.18 -109.61, 21.73 306.46, 113.14 -57.87, -17.2 in-in in 6.769 Saltbr-in 2.882 HRD-na-Q -82.05, -45.94 73.24, -7.24 in-in-in SNCiii in-in ActLoopNT-in 2.976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -76.56, -19.65 APE9-dihe-na -103.71, -175.8 APE8-dihe-in -130.62, 116.65 APE8-rot-in 293.03 APE67-dihe-in -65.48, -28.87 -48.06, -39.07 APE12-dist-in 11.529 APE11-dist-in 9.586 APE10-dist-in 4.483 APE9-dist-in 3.458 None None None XRAY 2.49 0.207 0.258 B 451 399 5 0 0 0 [[75, 309]] 1.0 5ckw Legionella pneumophila OTHER_LPL0262_LEGPL NEK 4.8e-15 62.8 10 222 213 212 213 214 216 218 104 119 123 192 194 193 195 249 237 232 231 230 229 228 227 226 146 non-specific serine/threonine protein kinase
AGC PRKACA KAPCA_MOUSE 4O21A P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 6.037 14.439 BLAminus -125.27, 173.53 70.53, 83.75 -96.26, 25.58 272.04, 54.28 -57.91, -27.19 in-in in 8.953 Saltbr-in 2.716 HRD-in -83.95, -57.84 75.15, 8.54 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.15, 164.3 APE9-dihe-na 125.14, -151.92 APE8-dihe-in -125.51, 129.66 APE8-rot-in 308.07 APE67-dihe-in -63.53, -19.17 -43.91, -48.76 APE12-dist-in 8.04 APE11-dist-in 11.46 APE10-dist-in 5.911 APE9-dist-in 3.451 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.17 0.215 A 342 336 0 0 0 0 [[44, 298]] 1.0 4o21 Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7E11A P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 6.205 14.451 BLAminus -127.38, -169.19 58.28, 74.22 -96.53, 30.74 276.22, 81.09 -66.46, -21.72 in-in in 9.053 Saltbr-in 2.551 HRD-in -91.79, -53.23 62.57, 24.02 in-in-in SNCiii in-in ActLoopNT-in 3.129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.39, 155.98 APE9-dihe-na 134.96, -158.62 APE8-dihe-in -113.95, 132.34 APE8-rot-in 301.67 APE67-dihe-in -76.79, -1.28 -53.37, -39.68 APE12-dist-in 8.309 APE11-dist-in 11.135 APE10-dist-in 5.71 APE9-dist-in 3.659 None TPO198,SEP339 TPO198,SEP339 XRAY 3.43 0.262 0.317 A 338 337 0 0 0 0 [[44, 298]] 1.0 7e11 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3PVBA P05132 7 351 351.0 ANP:60400 ATPlike Active DFGin 5.261 14.107 BLAminus -138.85, 171.16 63.11, 82.89 -89.43, -59.95 273.17, 54.43 27.14, -66.26 in-in in 8.685 Saltbr-in 3.476 HRD-in -84.36, -35.8 62.24, -18.82 in-in-in SNCiii in-in ActLoopNT-in 3.217 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -177.84, 157.88 APE9-dihe-na 132.55, -154.74 APE8-dihe-in -122.19, 108.01 APE8-rot-in 318.81 APE67-dihe-in -60.75, -2.24 -13.41, -60.33 APE12-dist-in 7.733 APE11-dist-in 10.579 APE10-dist-in 5.511 APE9-dist-in 4.042 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 3.3 0.242 0.29 A 345 345 0 0 0 0 [[44, 298]] 1.0 3pvb Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 1BKXA P05132 13 351 351.0 AMP:60351 ATPlike Active DFGin 6.16 13.915 BLAminus -117.09, 179.26 61.99, 75.16 -83.18, 21.65 286.96, 82.43 -60.51, -17.53 in-in in 8.724 Saltbr-in 2.658 HRD-in -99.39, -38.31 69.2, -9.22 in-in-in SNCiii in-in ActLoopNT-in 3.468 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.44, 150.62 APE9-dihe-na 113.99, 166.84 APE8-dihe-in -65.88, 134.1 APE8-rot-in 334.22 APE67-dihe-in -70.66, -34.65 -48.92, -27.08 APE12-dist-in 8.284 APE11-dist-in 11.351 APE10-dist-in 5.704 APE9-dist-in 4.285 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.6 0.219 0.34 A 350 339 0 0 0 0 [[44, 298]] 1.0 1bkx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 1L3RE P05132 2 351 351.0 ADP:60381 ATPlike Active DFGin 5.754 14.44 BLAminus -119.14, -174.46 57.18, 81.19 -93.77, 20.31 270.88, 52.04 -50.0, -37.57 in-in in 9.023 Saltbr-in 2.792 HRD-in -82.45, -54.36 70.16, 7.26 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.84, 161.06 APE9-dihe-na 132.7, -149.01 APE8-dihe-in -131.06, 132.91 APE8-rot-in 298.56 APE67-dihe-in -55.27, -27.25 -33.24, -62.94 APE12-dist-in 8.198 APE11-dist-in 11.233 APE10-dist-in 5.825 APE9-dist-in 3.368 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.0 0.205 0.232 E 350 341 0 0 0 0 [[44, 298]] 1.0 1l3r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 2QCSA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.648 14.291 BLAminus -119.78, 176.88 65.56, 77.31 -85.05, 19.39 273.35, 51.28 -44.32, -42.51 in-in in 8.784 Saltbr-in 2.638 HRD-in -93.14, -54.78 73.52, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.735 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.52, 149.74 APE9-dihe-na 148.64, -142.53 APE8-dihe-in -132.36, 132.12 APE8-rot-in 297.18 APE67-dihe-in -64.67, -25.45 -36.74, -53.73 APE12-dist-in 8.133 APE11-dist-in 11.321 APE10-dist-in 5.851 APE9-dist-in 3.573 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.194 0.225 A 350 338 0 0 0 0 [[44, 298]] 1.0 2qcs Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3FJQE P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.671 14.459 BLAminus -119.42, 178.78 63.28, 80.04 -91.81, 23.31 270.73, 57.82 -56.09, -30.86 in-in in 9.149 Saltbr-in 2.834 HRD-in -91.33, -52.39 67.42, 13.87 in-in-in SNCiii in-in ActLoopNT-in 2.906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.19, 160.44 APE9-dihe-na 133.42, -155.21 APE8-dihe-in -125.75, 136.86 APE8-rot-in 304.0 APE67-dihe-in -61.0, -22.29 -48.87, -49.39 APE12-dist-in 8.086 APE11-dist-in 11.408 APE10-dist-in 5.838 APE9-dist-in 3.518 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.179 0.205 E 350 336 0 0 0 0 [[44, 298]] 1.0 3fjq Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3IDBA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.346 14.413 BLAminus -121.17, -175.1 59.7, 79.28 -94.34, 24.01 267.69, 48.22 -48.56, -33.02 in-in in 8.845 Saltbr-in 2.694 HRD-in -80.07, -50.75 69.18, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.99 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.99, 160.5 APE9-dihe-na 138.4, -150.07 APE8-dihe-in -124.64, 132.33 APE8-rot-in 296.41 APE67-dihe-in -59.26, -21.93 -30.94, -63.4 APE12-dist-in 8.102 APE11-dist-in 11.573 APE10-dist-in 6.068 APE9-dist-in 3.445 None TPO198,SEP339 TPO198,SEP339 XRAY 1.62 0.206 0.23 A 350 343 0 0 0 0 [[44, 298]] 1.0 3idb Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3IDCA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.079 14.472 BLAminus -127.31, 174.57 68.22, 96.34 -111.15, 30.11 265.57, 49.45 -62.75, -22.0 in-in in 8.642 Saltbr-in 3.031 HRD-in -69.04, -44.03 64.09, 13.38 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.35, 157.69 APE9-dihe-na 142.7, -132.16 APE8-dihe-in -139.58, 115.88 APE8-rot-in 293.03 APE67-dihe-in -54.66, -5.54 -16.73, -78.3 APE12-dist-in 7.844 APE11-dist-in 11.373 APE10-dist-in 6.164 APE9-dist-in 3.675 None TPO198,SEP339 TPO198,SEP339 XRAY 2.7 0.241 0.319 A 350 343 0 0 0 0 [[44, 298]] 1.0 3idc Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DG0E P05132 11 351 351.0 ANP:60402 ATPlike Active DFGin 5.583 14.342 BLAminus -118.87, 179.66 65.44, 79.89 -93.34, 25.25 272.35, 58.42 -52.71, -36.39 in-in in 8.955 Saltbr-in 2.699 HRD-in -84.35, -52.45 74.02, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.07, 161.1 APE9-dihe-na 130.81, -146.6 APE8-dihe-in -130.07, 130.32 APE8-rot-in 303.85 APE67-dihe-in -61.09, -22.5 -44.14, -49.24 APE12-dist-in 8.008 APE11-dist-in 11.498 APE10-dist-in 5.9 APE9-dist-in 3.389 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.196 0.228 E 350 341 0 0 0 0 [[44, 298]] 1.0 4dg0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH1A P05132 16 351 351.0 ATP:60402 ATPlike Active DFGin 6.234 14.38 BLAminus -130.7, 167.11 69.97, 89.08 -103.01, 26.92 273.93, 57.95 -52.62, -33.38 in-in in 8.931 Saltbr-in 3.01 HRD-in -75.69, -51.31 65.95, 10.85 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.97, 163.54 APE9-dihe-na 128.87, -151.55 APE8-dihe-in -123.52, 135.53 APE8-rot-in 304.09 APE67-dihe-in -55.69, -26.94 -40.23, -59.36 APE12-dist-in 8.169 APE11-dist-in 11.557 APE10-dist-in 5.95 APE9-dist-in 3.545 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.199 0.234 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH3A P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.984 14.379 BLAminus -125.47, 176.75 61.82, 79.89 -92.16, 24.39 276.69, 54.39 -43.39, -47.09 in-in in 9.021 Saltbr-in 2.723 HRD-in -82.56, -48.22 66.04, -2.33 in-in-in SNCiii in-in ActLoopNT-in 2.931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 165.55 APE9-dihe-na 126.96, -149.27 APE8-dihe-in -125.58, 130.88 APE8-rot-in 307.35 APE67-dihe-in -57.88, -25.54 -37.95, -56.15 APE12-dist-in 8.225 APE11-dist-in 11.592 APE10-dist-in 6.104 APE9-dist-in 3.74 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.203 0.233 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH5A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 6.121 14.339 BLAminus -125.12, -179.76 61.4, 85.13 -97.61, 27.77 279.05, 62.21 -46.99, -44.52 in-in in 9.043 Saltbr-in 2.552 HRD-in -77.92, -53.51 67.68, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.88, 153.17 APE9-dihe-na 132.88, -161.89 APE8-dihe-in -112.07, 131.8 APE8-rot-in 304.21 APE67-dihe-in -57.01, -23.17 -41.47, -55.69 APE12-dist-in 8.219 APE11-dist-in 11.602 APE10-dist-in 6.071 APE9-dist-in 3.87 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.187 0.222 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH7A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.574 14.349 BLAminus -124.43, -175.45 59.33, 78.79 -93.54, 24.71 270.97, 54.79 -50.12, -38.03 in-in in 9.025 Saltbr-in 2.724 HRD-in -76.49, -50.79 66.5, 11.01 in-in-in SNCiii in-in ActLoopNT-in 2.961 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.18, 162.39 APE9-dihe-na 131.3, -151.54 APE8-dihe-in -126.44, 134.15 APE8-rot-in 300.19 APE67-dihe-in -56.38, -25.77 -37.48, -60.34 APE12-dist-in 8.093 APE11-dist-in 11.455 APE10-dist-in 5.87 APE9-dist-in 3.417 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.8 0.179 0.194 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DH8A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.901 14.014 BLAminus -123.95, -176.77 59.01, 85.18 -98.8, 24.84 279.52, 63.26 -51.76, -30.5 in-in in 8.8 Saltbr-in 2.713 HRD-in -77.99, -56.65 70.43, 3.78 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.95, 158.57 APE9-dihe-na 135.16, -154.79 APE8-dihe-in -124.8, 132.89 APE8-rot-in 296.53 APE67-dihe-in -58.95, -25.2 -38.46, -56.52 APE12-dist-in 8.145 APE11-dist-in 11.475 APE10-dist-in 5.904 APE9-dist-in 3.511 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.155 0.188 A 350 336 0 0 0 0 [[44, 298]] 1.0 4dh8 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4HPTE P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.748 14.424 BLAminus -115.4, 178.03 67.73, 81.09 -92.11, 21.69 273.09, 55.37 -58.71, -29.4 in-in in 9.053 Saltbr-in 2.66 HRD-in -90.64, -54.09 71.81, 9.39 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.27, 162.98 APE9-dihe-na 129.56, -147.32 APE8-dihe-in -127.39, 129.92 APE8-rot-in 299.02 APE67-dihe-in -63.31, -27.9 -40.61, -49.36 APE12-dist-in 8.069 APE11-dist-in 11.385 APE10-dist-in 5.825 APE9-dist-in 3.573 None TPO198,SEP339 TPO198,SEP339 XRAY 2.15 0.189 0.228 E 350 337 0 0 0 0 [[44, 298]] 1.0 4hpt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4HPUE P05132 13 351 351.0 ANP:60402 ATPlike Active DFGin 5.551 14.407 BLAminus -117.63, -178.61 63.83, 78.8 -92.22, 24.46 271.46, 55.23 -53.69, -32.94 in-in in 9.031 Saltbr-in 2.692 HRD-in -87.73, -52.35 74.85, 8.01 in-in-in SNCiii in-in ActLoopNT-in 2.914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.41, 162.17 APE9-dihe-na 134.1, -149.11 APE8-dihe-in -128.69, 136.04 APE8-rot-in 297.56 APE67-dihe-in -58.67, -24.48 -48.3, -49.81 APE12-dist-in 8.063 APE11-dist-in 11.507 APE10-dist-in 5.886 APE9-dist-in 3.403 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.173 0.194 E 350 339 0 0 0 0 [[44, 298]] 1.0 4hpu Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 5JR7A P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.739 13.691 BLAminus -145.14, 176.28 64.37, 76.68 -85.75, 18.89 294.14, 59.99 -43.66, -41.86 in-in in 8.674 Saltbr-in 2.709 HRD-in -93.38, -54.67 74.91, 7.39 in-in-in SNCiii in-in ActLoopNT-in 2.945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.46, 148.2 APE9-dihe-na 147.95, -159.28 APE8-dihe-in -109.66, 131.32 APE8-rot-in 258.88 APE67-dihe-in -65.5, -25.8 -38.64, -53.47 APE12-dist-in 8.014 APE11-dist-in 10.772 APE10-dist-in 5.528 APE9-dist-in 3.878 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 A 350 338 0 0 0 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 5JR7C P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.899 13.164 BLAminus -138.79, 176.44 54.89, 86.07 -89.1, 7.67 290.95, 62.79 -41.83, -37.01 in-in in 8.185 Saltbr-in 3.195 HRD-in -79.11, -50.37 72.48, -21.93 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.28, 123.46 APE9-dihe-na 160.31, -160.86 APE8-dihe-in -110.49, 124.04 APE8-rot-in 311.35 APE67-dihe-in -70.47, -24.34 -45.9, -42.95 APE12-dist-in 8.163 APE11-dist-in 10.628 APE10-dist-in 5.002 APE9-dist-in 4.262 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 C 350 338 0 0 0 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7UJXE P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 5.731 14.357 BLAminus -121.93, 179.51 64.92, 83.56 -91.91, 29.5 277.22, 63.03 -64.62, -28.12 in-in in 9.103 Saltbr-in 2.812 HRD-in -86.19, -57.72 74.11, 16.74 in-in-in SNCiii in-in ActLoopNT-in 2.931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.48, 155.47 APE9-dihe-na 127.23, -161.98 APE8-dihe-in -111.77, 133.52 APE8-rot-in 302.04 APE67-dihe-in -65.07, -18.97 -50.87, -44.77 APE12-dist-in 8.191 APE11-dist-in 11.5 APE10-dist-in 5.961 APE9-dist-in 4.008 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.133 0.176 E 350 336 0 0 0 0 [[44, 298]] 1.0 7ujx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7V0GE P05132 17 351 351.0 ADP:60401 ATPlike Active DFGin 5.739 14.319 BLAminus -119.5, 177.58 67.43, 82.74 -91.45, 25.21 276.8, 64.92 -62.46, -26.34 in-in in 9.07 Saltbr-in 2.802 HRD-in -88.93, -50.41 71.3, 15.33 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.52, 156.77 APE9-dihe-na 130.04, -162.37 APE8-dihe-in -114.97, 131.2 APE8-rot-in 299.52 APE67-dihe-in -60.0, -22.75 -47.18, -49.61 APE12-dist-in 8.174 APE11-dist-in 11.542 APE10-dist-in 6.037 APE9-dist-in 3.965 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.118 0.163 E 350 335 0 0 0 0 [[44, 298]] 1.0 7v0g Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DFXE P05132 2 351 351.0 ANP:60402 ATPlike Active DFGin 5.524 14.286 BLAminus -116.71, -179.39 66.13, 78.01 -91.08, 23.34 272.63, 51.46 -56.59, -32.27 in-in in 8.873 Saltbr-in 2.729 HRD-in -88.99, -54.58 73.79, 11.03 in-in-in SNCiii in-in ActLoopNT-in 2.934 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.69, 159.64 APE9-dihe-na 138.16, -148.52 APE8-dihe-in -130.4, 136.32 APE8-rot-in 296.63 APE67-dihe-in -59.91, -24.0 -47.38, -49.37 APE12-dist-in 8.046 APE11-dist-in 11.41 APE10-dist-in 5.819 APE9-dist-in 3.392 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.35 0.157 0.179 E 350 350 0 0 0 0 [[44, 298]] 1.0 4dfx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4X6RA P05132 2 351 351.0 ATP:60402 ATPlike Active DFGin 6.133 14.232 BLAminus -118.92, 178.27 64.18, 79.91 -89.21, 11.01 274.1, 55.74 -49.19, -34.95 in-in in 8.804 Saltbr-in 2.729 HRD-in -85.13, -60.38 77.67, -7.87 in-in-in SNCiii in-in ActLoopNT-in 2.718 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.34, 156.01 APE9-dihe-na 147.33, -149.7 APE8-dihe-in -130.56, 138.51 APE8-rot-in 291.09 APE67-dihe-in -61.2, -24.8 -52.44, -47.95 APE12-dist-in 8.281 APE11-dist-in 11.246 APE10-dist-in 5.836 APE9-dist-in 3.663 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.186 0.234 A 350 350 0 0 0 0 [[44, 298]] 1.0 4x6r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3X2UA P05132 13 351 351.0 ATP:60501 ATPlike Active DFGin 6.127 14.507 BLAminus -122.24, 178.58 59.36, 87.7 -101.54, 25.28 272.61, 50.83 -59.45, -24.26 in-in in 9.272 Saltbr-in 2.788 HRD-in -89.58, -50.62 64.84, 17.58 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.25, 158.3 APE9-dihe-na 134.88, -147.54 APE8-dihe-in -130.4, 131.58 APE8-rot-in 300.12 APE67-dihe-in -61.26, -14.4 -40.08, -55.22 APE12-dist-in 7.912 APE11-dist-in 11.137 APE10-dist-in 5.686 APE9-dist-in 3.427 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.202 0.239 A 357 339 0 0 0 0 [[44, 298]] 1.0 3x2u Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3X2VA P05132 18 351 351.0 ATP:60403 ATPlike Active DFGin 5.517 14.152 BLAminus -116.69, -175.94 62.92, 80.3 -91.77, 26.26 271.42, 55.44 -51.78, -39.79 in-in in 8.755 Saltbr-in 2.654 HRD-in -92.08, -50.84 67.69, 17.07 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.85, 164.45 APE9-dihe-na 134.14, -152.5 APE8-dihe-in -130.83, 133.42 APE8-rot-in 299.77 APE67-dihe-in -58.82, -21.18 -48.96, -48.11 APE12-dist-in 7.998 APE11-dist-in 11.346 APE10-dist-in 5.796 APE9-dist-in 3.415 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.77 0.185 0.23 A 357 334 0 0 0 0 [[44, 298]] 1.0 3x2v Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3X2WA P05132 13 351 351.0 ATP:60403 ATPlike Active DFGin 5.66 14.39 BLAminus -121.01, -177.68 63.51, 77.56 -90.4, 24.79 270.4, 59.29 -61.83, -28.06 in-in in 8.822 Saltbr-in 2.632 HRD-in -81.34, -52.24 70.22, 11.48 in-in-in SNCiii in-in ActLoopNT-in 2.906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.19, 162.39 APE9-dihe-na 132.4, -151.44 APE8-dihe-in -129.91, 133.08 APE8-rot-in 300.2 APE67-dihe-in -60.45, -20.83 -45.18, -51.38 APE12-dist-in 8.001 APE11-dist-in 11.44 APE10-dist-in 5.911 APE9-dist-in 3.45 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.165 0.198 A 357 339 0 0 0 0 [[44, 298]] 1.0 3x2w Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IACA P05132 16 351 351.0 ACP:60403 ATPlike Active DFGin 5.755 14.312 BLAminus -125.73, -177.16 59.8, 78.08 -94.31, 23.06 273.35, 54.81 -46.36, -37.92 in-in in 8.885 Saltbr-in 2.721 HRD-in -73.57, -53.97 72.67, 5.23 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.57, 156.93 APE9-dihe-na 137.19, -153.99 APE8-dihe-in -123.03, 128.21 APE8-rot-in 300.87 APE67-dihe-in -59.06, -23.99 -31.47, -61.7 APE12-dist-in 8.157 APE11-dist-in 11.515 APE10-dist-in 5.985 APE9-dist-in 3.502 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.15 0.181 0.212 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iac Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IADA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.658 14.362 BLAminus -130.04, -179.13 63.0, 77.66 -87.34, 22.78 276.11, 53.54 -55.12, -31.28 in-in in 9.085 Saltbr-in 2.83 HRD-in -93.22, -52.19 70.15, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.935 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.54, 160.6 APE9-dihe-na 133.65, -143.98 APE8-dihe-in -130.05, 134.5 APE8-rot-in 298.49 APE67-dihe-in -67.08, -22.74 -48.94, -44.54 APE12-dist-in 8.051 APE11-dist-in 11.55 APE10-dist-in 6.087 APE9-dist-in 3.521 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.189 0.243 A 356 337 0 0 0 0 [[44, 298]] 1.0 4iad Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAFA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.943 14.13 BLAminus -121.29, 178.82 64.06, 84.8 -98.0, 27.2 281.56, 65.38 -51.93, -33.25 in-in in 8.871 Saltbr-in 2.669 HRD-in -76.48, -53.65 65.3, 9.94 in-in-in SNCiii in-in ActLoopNT-in 2.974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.4, 160.11 APE9-dihe-na 128.66, -151.44 APE8-dihe-in -123.86, 135.06 APE8-rot-in 298.27 APE67-dihe-in -57.84, -25.84 -42.55, -55.44 APE12-dist-in 8.163 APE11-dist-in 11.523 APE10-dist-in 5.973 APE9-dist-in 3.563 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.16 0.192 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iaf Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAIA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.465 14.503 BLAminus -125.1, 176.4 64.24, 81.88 -90.74, 22.64 269.91, 49.4 -55.45, -35.99 in-in in 9.101 Saltbr-in 2.714 HRD-in -91.06, -49.32 68.79, 15.16 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.75, 156.86 APE9-dihe-na 141.29, -148.36 APE8-dihe-in -128.24, 130.8 APE8-rot-in 300.02 APE67-dihe-in -62.27, -23.0 -47.39, -47.75 APE12-dist-in 7.945 APE11-dist-in 11.458 APE10-dist-in 5.867 APE9-dist-in 3.608 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.171 0.209 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iai Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAKA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.705 14.569 BLAminus -126.92, 179.61 63.08, 81.74 -90.27, 23.65 270.26, 53.44 -59.05, -31.45 in-in in 8.985 Saltbr-in 2.747 HRD-in -94.54, -49.89 67.85, 16.15 in-in-in SNCiii in-in ActLoopNT-in 2.91 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.92, 164.74 APE9-dihe-na 131.87, -148.57 APE8-dihe-in -130.85, 127.67 APE8-rot-in 297.68 APE67-dihe-in -61.28, -21.91 -43.91, -50.7 APE12-dist-in 7.962 APE11-dist-in 11.443 APE10-dist-in 5.979 APE9-dist-in 3.545 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.6 0.185 0.222 A 356 337 0 0 0 0 [[44, 298]] 1.0 4iak Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAYA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.806 14.257 BLAminus -131.74, 174.05 67.76, 85.89 -95.28, 20.31 273.12, 61.73 -48.17, -36.05 in-in in 9.039 Saltbr-in 2.941 HRD-in -89.87, -50.65 68.98, 10.01 in-in-in SNCiii in-in ActLoopNT-in 3.055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.39, 159.46 APE9-dihe-na 132.54, -148.24 APE8-dihe-in -127.91, 130.95 APE8-rot-in 300.76 APE67-dihe-in -63.09, -19.35 -45.58, -49.88 APE12-dist-in 8.089 APE11-dist-in 11.466 APE10-dist-in 5.991 APE9-dist-in 3.823 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.182 0.227 A 356 336 0 0 0 0 [[44, 298]] 1.0 4iay Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IAZA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 6.144 14.635 BLAminus -132.33, 171.23 62.84, 84.78 -94.94, 21.85 278.49, 61.31 -54.74, -28.93 in-in in 9.219 Saltbr-in 2.747 HRD-in -95.03, -54.93 73.76, 14.73 in-in-in SNCiii in-in ActLoopNT-in 3.017 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.57, 164.74 APE9-dihe-na 127.12, -150.82 APE8-dihe-in -127.02, 138.46 APE8-rot-in 303.51 APE67-dihe-in -63.11, -25.72 -51.71, -47.83 APE12-dist-in 7.963 APE11-dist-in 11.514 APE10-dist-in 5.979 APE9-dist-in 3.574 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.85 0.201 0.248 A 356 337 0 0 0 0 [[44, 298]] 1.0 4iaz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IB0A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.713 14.439 BLAminus -123.68, 176.86 65.62, 82.22 -94.42, 18.76 272.15, 51.12 -47.84, -35.86 in-in in 9.065 Saltbr-in 3.023 HRD-in -84.67, -55.05 71.31, 12.11 in-in-in SNCiii in-in ActLoopNT-in 2.886 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.67, 157.49 APE9-dihe-na 139.08, -144.95 APE8-dihe-in -131.16, 131.55 APE8-rot-in 306.17 APE67-dihe-in -61.31, -24.54 -46.0, -48.78 APE12-dist-in 8.059 APE11-dist-in 11.516 APE10-dist-in 5.969 APE9-dist-in 3.692 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.87 0.219 0.287 A 356 337 0 0 0 0 [[44, 298]] 1.0 4ib0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IB1A P05132 14 351 351.0 ADP:60403 ATPlike Active DFGin 5.656 14.443 BLAminus -126.58, 171.72 66.62, 80.69 -90.79, 23.58 274.18, 53.88 -53.03, -31.34 in-in in 9.121 Saltbr-in 2.691 HRD-in -82.93, -51.49 69.93, 14.85 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.64, 163.58 APE9-dihe-na 133.1, -151.37 APE8-dihe-in -125.38, 138.08 APE8-rot-in 304.1 APE67-dihe-in -60.15, -23.69 -50.01, -49.7 APE12-dist-in 7.96 APE11-dist-in 11.404 APE10-dist-in 5.961 APE9-dist-in 3.635 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.196 0.223 A 356 338 0 0 0 0 [[44, 298]] 1.0 4ib1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4IB3A P05132 13 351 351.0 ADP:60401 ATPlike Active DFGin 5.973 14.215 BLAminus -125.69, 173.12 66.37, 84.97 -98.59, 21.41 276.57, 60.51 -51.27, -29.52 in-in in 8.99 Saltbr-in 2.76 HRD-in -77.27, -49.79 61.58, 13.48 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.06, 160.46 APE9-dihe-na 127.6, -161.57 APE8-dihe-in -110.98, 129.89 APE8-rot-in 305.68 APE67-dihe-in -58.89, -23.07 -39.61, -54.94 APE12-dist-in 8.078 APE11-dist-in 11.522 APE10-dist-in 5.923 APE9-dist-in 3.568 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.182 0.228 A 356 339 0 0 0 0 [[44, 298]] 1.0 4ib3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4XW4A P05132 15 351 351.0 ANP:60403 ATPlike Active DFGin 5.673 14.562 BLAminus -117.82, -177.44 65.15, 79.34 -92.69, 26.58 269.45, 57.64 -61.99, -28.36 in-in in 8.931 Saltbr-in 2.858 HRD-in -86.05, -50.94 67.2, 15.72 in-in-in SNCiii in-in ActLoopNT-in 3.014 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.62, 159.69 APE9-dihe-na 135.12, -140.29 APE8-dihe-in -136.84, 125.12 APE8-rot-in 301.75 APE67-dihe-in -61.52, -26.6 -45.5, -44.66 APE12-dist-in 7.961 APE11-dist-in 11.419 APE10-dist-in 5.935 APE9-dist-in 3.664 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.82 0.183 0.24 A 356 337 0 0 0 0 [[44, 298]] 1.0 4xw4 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4XW5A P05132 15 351 351.0 ATP:60403 ATPlike Active DFGin 5.971 14.222 BLAminus -131.24, 177.82 59.66, 87.19 -93.08, 25.08 282.37, 63.43 -53.77, -29.24 in-in in 9.213 Saltbr-in 2.673 HRD-in -90.87, -48.94 63.52, 13.92 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.24, 155.03 APE9-dihe-na 137.47, -160.98 APE8-dihe-in -110.31, 133.6 APE8-rot-in 304.05 APE67-dihe-in -58.14, -25.36 -48.87, -50.12 APE12-dist-in 8.026 APE11-dist-in 11.601 APE10-dist-in 6.1 APE9-dist-in 3.922 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.185 0.252 A 356 337 0 0 0 0 [[44, 298]] 1.0 4xw5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4XW6A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.982 14.431 BLAminus -130.68, 178.48 65.03, 84.15 -99.24, 23.41 276.01, 56.03 -60.45, -23.49 in-in in 9.15 Saltbr-in 2.735 HRD-in -94.59, -52.61 68.2, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.791 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.91, 154.59 APE9-dihe-na 136.7, -154.91 APE8-dihe-in -121.39, 127.95 APE8-rot-in 293.9 APE67-dihe-in -62.75, -24.38 -45.59, -46.76 APE12-dist-in 8.051 APE11-dist-in 11.632 APE10-dist-in 6.051 APE9-dist-in 3.787 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.186 0.265 A 356 337 0 0 0 0 [[44, 298]] 1.0 4xw6 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 6E21A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.594 14.055 BLAminus -122.61, 176.37 63.02, 83.41 -94.2, 28.27 284.3, 46.09 -48.88, -41.13 in-in in 9.029 Saltbr-in 2.607 HRD-in -74.35, -56.8 67.48, 11.51 in-in-in SNCiii in-in ActLoopNT-in 2.907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.7, 159.01 APE9-dihe-na 131.41, -152.84 APE8-dihe-in -125.29, 130.56 APE8-rot-in 303.23 APE67-dihe-in -58.42, -25.04 -35.36, -60.06 APE12-dist-in 8.043 APE11-dist-in 11.584 APE10-dist-in 6.022 APE9-dist-in 3.58 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.187 0.217 A 356 336 0 0 0 0 [[44, 298]] 1.0 6e21 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 7E0ZA P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 5.566 13.884 BLAminus -118.85, -174.47 59.93, 79.47 -94.43, 25.89 275.59, 63.85 -59.78, -31.6 in-in in 8.624 Saltbr-in 2.978 HRD-in -96.8, -56.38 78.26, 13.74 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.91, 162.74 APE9-dihe-na 131.67, -149.57 APE8-dihe-in -131.04, 130.65 APE8-rot-in 294.41 APE67-dihe-in -63.42, -12.5 -45.48, -52.1 APE12-dist-in 7.9 APE11-dist-in 11.182 APE10-dist-in 5.721 APE9-dist-in 3.4 None TPO198,SEP339 TPO198,SEP339 XRAY 2.162 0.184 0.228 A 358 337 0 0 0 0 [[44, 298]] 1.0 7e0z Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 4DG3E P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.481 14.342 BLAminus -115.99, -176.62 61.62, 77.98 -90.25, 24.84 270.29, 54.4 -55.44, -35.73 in-in in 8.842 Saltbr-in 2.695 HRD-in -87.1, -53.93 73.82, 10.76 in-in-in SNCiii in-in ActLoopNT-in 2.882 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.46, 161.61 APE9-dihe-na 135.41, -150.07 APE8-dihe-in -129.52, 135.22 APE8-rot-in 300.3 APE67-dihe-in -58.11, -23.91 -46.28, -51.67 APE12-dist-in 8.143 APE11-dist-in 11.482 APE10-dist-in 5.886 APE9-dist-in 3.405 R337A SEP140,TPO198 SEP140,TPO198 XRAY 1.8 0.185 0.217 E 371 337 0 0 0 0 [[44, 298]] 1.0 4dg3 Mus musculus AGC_PRKACA_MOUSE AGC 1.8e-94 321.8 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3FHIA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.463 14.263 BLAminus -118.0, -179.45 64.04, 75.7 -86.07, 24.14 267.17, 53.33 -59.82, -32.06 in-in in 8.887 Saltbr-in 2.79 HRD-in -94.84, -53.37 68.02, 7.49 in-in-in SNCiii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.67, 136.88 APE9-dihe-na 156.84, -158.52 APE8-dihe-in -126.08, 132.83 APE8-rot-in 296.09 APE67-dihe-in -67.08, -19.88 -42.62, -50.01 APE12-dist-in 8.233 APE11-dist-in 11.12 APE10-dist-in 5.402 APE9-dist-in 3.564 C200A TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.199 0.226 A 350 338 0 0 0 0 [[44, 298]] 1.0 3fhi Mus musculus AGC_PRKACA_MOUSE AGC 1e-93 319.3 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3QAME P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.559 14.19 BLAminus -125.2, -173.2 57.82, 79.24 -94.32, 24.42 273.28, 56.46 -52.36, -33.22 in-in in 8.98 Saltbr-in 2.804 HRD-in -80.54, -55.75 67.52, 12.49 in-in-in SNCiii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.45, 157.56 APE9-dihe-na 134.84, -152.56 APE8-dihe-in -129.9, 127.65 APE8-rot-in 298.13 APE67-dihe-in -57.31, -20.14 -26.19, -66.74 APE12-dist-in 8.094 APE11-dist-in 11.277 APE10-dist-in 5.806 APE9-dist-in 3.475 E209A TPO198,SEP339 TPO198,SEP339 XRAY 1.92 0.195 0.228 E 350 350 0 0 0 0 [[44, 298]] 1.0 3qam Mus musculus AGC_PRKACA_MOUSE AGC 2.2e-93 318.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_MOUSE 3QALE P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.64 14.401 BLAminus -123.21, -177.09 59.31, 80.89 -94.71, 25.93 269.1, 56.43 -54.28, -32.32 in-in in 9.05 Saltbr-in 2.658 HRD-in -84.64, -51.07 65.64, 14.74 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.61, 159.73 APE9-dihe-na 131.58, -155.18 APE8-dihe-in -126.66, 132.34 APE8-rot-in 301.51 APE67-dihe-in -57.77, -23.32 -31.31, -63.36 APE12-dist-in 8.062 APE11-dist-in 11.309 APE10-dist-in 5.744 APE9-dist-in 3.531 R281A TPO198,SEP339 TPO198,SEP339 XRAY 1.7 0.176 0.194 E 350 341 0 0 0 0 [[44, 298]] 1.0 3qal Mus musculus AGC_PRKACA_MOUSE AGC 4.5e-93 317.2 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CAMK CAMK2A KCC2A_MOUSE 7B56B P11798 5 307 478.0 ANP:60401 ATPlike Active DFGin 6.729 14.232 BLAminus -127.69, 175.68 61.5, 79.97 -89.44, 23.96 289.95, 77.46 -66.33, -24.14 in-in in 8.963 Saltbr-in 2.797 HRD-in -75.83, -42.64 71.61, -6.11 in-in-in SNCiii in-in ActLoopNT-in 2.891 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.35, 145.48 APE9-dihe-na 136.45, -166.63 APE8-dihe-in -115.36, 130.21 APE8-rot-in 297.52 APE67-dihe-in -66.37, -13.84 -48.36, -50.63 APE12-dist-in 10.406 APE11-dist-in 11.67 APE10-dist-in 5.883 APE9-dist-in 3.799 T305A,T306A None None XRAY 1.45 0.191 0.215 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b56 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK CAMK2A KCC2A_MOUSE 7B57B P11798 5 307 478.0 ADP:603 ATPlike Active DFGin 6.612 14.081 BLAminus -127.42, 175.73 58.47, 86.34 -93.82, 26.41 288.57, 77.62 -63.18, -29.51 in-in in 8.79 Saltbr-in 2.799 HRD-in -66.41, -49.66 65.98, 1.57 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.13, 142.7 APE9-dihe-na 131.67, 177.43 APE8-dihe-in -91.43, 131.98 APE8-rot-in 302.75 APE67-dihe-in -62.31, -16.39 -48.04, -47.99 APE12-dist-in 10.368 APE11-dist-in 11.44 APE10-dist-in 5.743 APE9-dist-in 3.998 T305A,T306A None None XRAY 1.95 0.206 0.247 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b57 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
CAMK DAPK2 DAPK2_MOUSE 2YAAA Q8VDF3 12 311 370.0 ATP:61302 ATPlike Active DFGin 6.531 14.282 BLAminus -119.44, -173.75 61.63, 82.55 -100.44, 26.82 279.23, 73.82 -61.71, -30.38 in-in in 9.437 Saltbr-in 2.945 HRD-in -69.91, -51.35 70.12, 4.4 in-in-in SNCiii in-in ActLoopNT-in 2.83 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.66, 179.02 APE9-dihe-na 88.17, 165.82 APE8-dihe-in -83.03, 124.75 APE8-rot-in 307.34 APE67-dihe-in -54.24, -28.42 -45.93, -43.89 APE12-dist-in 8.679 APE11-dist-in 11.592 APE10-dist-in 6.391 APE9-dist-in 4.926 None None None XRAY 2.3 0.219 0.271 A 361 300 0 0 0 0 [[23, 285]] 1.0 2yaa Mus musculus CAMK_DAPK2_MOUSE CAMK 1.1e-93 319.4 1 256 256 170 171 172 174 176 52 74 78 146 148 147 149 209 197 192 191 190 189 188 187 186 104 Death-associated protein kinase 2
CAMK DAPK2 DAPK2_MOUSE 2YABA Q8VDF3 13 311 370.0 AMP:61302 ATPlike Active DFGin 6.504 14.098 BLAminus -124.73, -175.5 61.61, 83.44 -98.66, 29.53 280.86, 70.25 -68.26, -23.3 in-in in 9.084 Saltbr-in 2.894 HRD-in -75.19, -47.84 69.74, 6.94 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.38, -177.82 APE9-dihe-na 87.95, 171.12 APE8-dihe-in -92.08, 123.94 APE8-rot-in 301.03 APE67-dihe-in -53.06, -29.06 -44.13, -47.2 APE12-dist-in 8.535 APE11-dist-in 11.604 APE10-dist-in 6.372 APE9-dist-in 4.88 None None None XRAY 1.9 0.174 0.215 A 361 299 0 0 0 0 [[23, 285]] 1.0 2yab Mus musculus CAMK_DAPK2_MOUSE CAMK 1.1e-93 319.4 1 256 256 170 171 172 174 176 52 74 78 146 148 147 149 209 197 192 191 190 189 188 187 186 104 Death-associated protein kinase 2
CMGC GSK3B GSK3B_MOUSE 8VMFA Q9WV60 27 383 420.0 ADP:60504 ATPlike Active DFGin 6.612 14.1 BLAminus -148.4, -167.57 58.53, 66.72 -90.57, 24.21 287.49, 78.37 -75.04, -7.89 in-in in 8.66 Saltbr-in 2.678 HRD-in -67.34, -47.3 70.6, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.84 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.01, -20.74 APE9-dihe-na -93.16, -168.14 APE8-dihe-in -112.8, 164.36 APE8-rot-in 304.6 APE67-dihe-inflip 78.98, -8.38 -56.8, 140.56 APE12-dist-in 13.183 APE11-dist-in 10.949 APE10-dist-in 6.514 APE9-dist-in 3.308 None None None XRAY 2.5 0.21 0.251 A 364 354 0 0 0 0 [[56, 340]] 1.0 8vmf Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_MOUSE 8VMGA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 7.0 13.999 BLAminus -139.67, -176.86 60.44, 73.06 -89.27, 27.07 283.1, 81.19 -73.23, -12.63 in-in in 8.478 Saltbr-in 2.688 HRD-in -67.64, -48.38 72.75, 3.36 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.26, 164.63 APE9-dihe-na 72.45, 142.8 APE8-dihe-in -66.41, 146.08 APE8-rot-in 307.07 APE67-dihe-in -64.3, -22.81 -57.43, -46.54 APE12-dist-in 13.278 APE11-dist-in 11.627 APE10-dist-in 6.941 APE9-dist-in 2.984 None None None XRAY 2.45 0.195 0.23 A 364 358 0 0 0 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_MOUSE 8VMEA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 6.469 13.844 BLAminus -131.0, -171.33 63.41, 73.0 -92.56, 22.88 289.27, 83.61 -79.03, -1.02 in-in in 8.753 Saltbr-in 2.78 HRD-in -67.9, -47.67 70.4, 7.52 in-in-in SNCiii in-in ActLoopNT-in 2.731 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.18, 168.01 APE9-dihe-na 68.83, 161.19 APE8-dihe-in -90.7, 152.54 APE8-rot-in 290.93 APE67-dihe-inflip 82.32, -22.26 -51.38, 150.9 APE12-dist-in 13.288 APE11-dist-in 12.071 APE10-dist-in 6.934 APE9-dist-in 3.292 None None None XRAY 2.3 0.183 0.23 A 365 355 0 0 0 0 [[56, 340]] 1.0 8vme Mus musculus CMGC_GSK3B_MOUSE CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC GSK3B GSK3B_MOUSE 4NU1A Q9WV60 6 383 420.0 ADP:405 ATPlike Active DFGin 6.109 13.677 BLAminus -140.27, -172.8 60.29, 88.19 -108.14, 24.39 289.57, 88.21 -68.01, -14.99 in-in in 8.691 Saltbr-in 2.793 HRD-in -66.76, -45.51 62.96, 19.85 in-in-in SNCiii in-in ActLoopNT-in 2.682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.38, 172.68 APE9-dihe-na 66.76, 153.81 APE8-dihe-in -82.08, 156.46 APE8-rot-in 299.93 APE67-dihe-inflip 76.53, -25.22 -54.39, 158.45 APE12-dist-in 13.51 APE11-dist-in 11.621 APE10-dist-in 7.126 APE9-dist-in 3.15 None SEP9 SEP9 XRAY 2.5 0.194 0.245 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nu1 Mus musculus CMGC_GSK3B_MOUSE CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
CMGC MAPK14 MK14_MOUSE 5NZZE P47811 4 353 360.0 AGS:60401 ATPlike Active DFGin 6.514 14.981 BLAminus -122.06, 164.78 72.33, 78.3 -82.97, 27.83 284.83, 92.09 -68.73, -16.77 in-in in 9.475 Saltbr-in 3.566 HRD-in -92.47, -52.47 76.16, -3.26 in-in-in SNCiii in-in ActLoopNT-in 2.855 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.62, 176.88 APE9-dihe-na 58.43, 166.45 APE8-dihe-in -84.96, 144.19 APE8-rot-in 316.3 APE67-dihe-in -61.16, -25.49 -55.46, -53.03 APE12-dist-in 11.933 APE11-dist-in 11.395 APE10-dist-in 7.236 APE9-dist-in 3.126 None TPO180,PTR182 TPO180,PTR182 XRAY 2.6 0.221 0.271 E 360 345 5 0 0 0 [[24, 308]] 1.0 5nzz Mus musculus CMGC_MAPK14_MOUSE CMGC 1.9e-85 292.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_MOUSE 5NZZF P47811 5 353 360.0 AGS:60401 ATPlike Active DFGin 6.581 14.746 BLAminus -104.46, 169.41 67.42, 93.44 -106.87, 21.93 284.61, 82.38 -60.31, -14.32 in-in in 9.318 Saltbr-in 2.692 HRD-in -84.83, -58.57 70.0, 21.45 in-in-in SNCiii in-in ActLoopNT-in 3.066 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.79, 145.31 APE9-dihe-na 83.88, 162.38 APE8-dihe-in -79.27, 130.51 APE8-rot-in 303.15 APE67-dihe-in -54.1, -23.47 -46.06, -59.5 APE12-dist-in 11.925 APE11-dist-in 11.532 APE10-dist-in 7.245 APE9-dist-in 3.334 None TPO180,PTR182 TPO180,PTR182 XRAY 2.6 0.221 0.271 F 360 343 6 0 0 0 [[24, 308]] 1.0 5nzz Mus musculus CMGC_MAPK14_MOUSE CMGC 1.9e-85 292.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
TYR LYN LYN_MOUSE 2ZV8A P25911 239 501 512.0 ANP:60001 ATPlike Active DFGin 6.207 14.166 BLAminus -127.46, 176.54 66.14, 76.26 -98.89, 34.27 306.37, 82.39 -66.23, -26.52 in-in in 8.182 Saltbr-in 2.888 HRD-na-N -93.92, -49.32 76.02, -10.27 in-in-in SNCiii in-in ActLoopNT-in 2.954 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -123.91, 116.52 APE9-dihe-in -60.43, 148.58 APE8-dihe-in -80.52, 92.26 APE8-rot-na 28.17 APE67-dihe-in -68.44, -3.54 -43.41, -52.9 APE12-dist-na 9.634 APE11-dist-na 5.923 APE10-dist-na 9.729 APE9-dist-in 5.004 None None None XRAY 2.7 0.201 0.245 A 279 256 7 0 0 7 [[247, 499]] 1.0 2zv8 Mus musculus TYR_LYN_MOUSE TYR 4.1e-95 323.9 1 260 260 384 385 386 388 390 275 290 294 364 366 365 367 425 413 408 407 406 405 404 403 402 320 Tyrosine-protein kinase Lyn
CAMK PHKG1 PHKG1_RABIT 2PHKA P00518 15 291 387.0 ATP:60381 ATPlike Active DFGin 6.355 14.931 BLAminus -137.29, -164.32 48.12, 82.5 -104.58, 35.29 286.95, 71.57 -66.18, -30.51 in-in in 9.223 Saltbr-in 2.867 HRD-in -75.14, -51.03 75.46, 17.9 in-in-in SNCiii in-in ActLoopNT-in 2.885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.02, 157.52 APE9-dihe-na 142.39, -153.7 APE8-dihe-in -119.73, 129.29 APE8-rot-in 312.14 APE67-dihe-in -75.97, -3.06 -46.22, -51.97 APE12-dist-in 9.188 APE11-dist-in 12.037 APE10-dist-in 6.565 APE9-dist-in 4.187 None None None XRAY 2.6 0.253 0.3 A 277 277 0 0 0 0 [[20, 288]] 1.0 2phk Oryctolagus cuniculus CAMK_PHKG1_RABIT CAMK 3e-86 294.8 1 256 256 167 168 169 171 173 49 74 78 147 149 148 150 212 194 189 188 187 186 185 184 183 105 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
CAMK PHKG1 PHKG1_RABIT 1QL6A P00518 12 292 387.0 ATP:60301 ATPlike Active DFGin 6.367 14.614 BLAminus -136.63, -170.42 53.21, 74.77 -97.04, 26.39 287.52, 75.09 -70.06, -14.72 in-in in 9.205 Saltbr-in 3.1 HRD-in -59.97, -49.78 67.92, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.896 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.76, 155.97 APE9-dihe-na 109.55, 169.96 APE8-dihe-in -76.43, 127.92 APE8-rot-in 308.32 APE67-dihe-in -67.24, -23.63 -51.61, -34.62 APE12-dist-in 9.259 APE11-dist-in 11.445 APE10-dist-in 6.11 APE9-dist-in 4.369 E183S None None XRAY 2.4 0.24 0.33 A 298 281 0 0 0 0 [[20, 288]] 1.0 1ql6 Oryctolagus cuniculus CAMK_PHKG1_RABIT CAMK 5.1e-86 294.1 1 256 256 167 168 169 171 173 49 74 78 147 149 148 150 212 194 189 188 187 186 185 184 183 105 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
CAMK PHKG1 PHKG1_RABIT 1PHKA P00518 16 292 387.0 ATP:60381 ATPlike Active DFGin 6.147 14.336 BLAminus -126.89, -173.45 56.12, 79.25 -99.09, 29.57 290.92, 76.23 -67.63, -19.58 in-in in 8.993 Saltbr-in 2.825 HRD-in -77.33, -46.36 68.03, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.41, 147.14 APE9-dihe-na 116.4, 168.87 APE8-dihe-in -72.55, 120.48 APE8-rot-in 295.05 APE67-dihe-in -62.26, -27.58 -41.92, -42.38 APE12-dist-in 8.836 APE11-dist-in 11.43 APE10-dist-in 6.157 APE9-dist-in 4.492 None None None XRAY 2.2 0.21 0.288 A 298 277 0 0 0 0 [[20, 288]] 1.0 1phk Oryctolagus cuniculus CAMK_PHKG1_RABIT CAMK 4e-86 294.4 1 256 256 167 168 169 171 173 49 74 78 147 149 148 150 212 194 189 188 187 186 185 184 183 105 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
OTHER PINK1 PINK1_PEDHC 8UYHA E0W1I1 115 574 575.0 ANP:601 ATPlike Active DFGin 9.322 14.819 BLAminus -130.08, -169.42 57.7, 62.71 -86.71, 26.39 286.61, 80.23 -66.61, -35.48 in-in in 7.967 Saltbr-in 3.27 HRD-in -73.02, -43.12 61.9, 7.28 in-in-in SNCiii in-in ActLoopNT-in 2.764 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 161.16, -131.74 APE9-dihe-na -112.83, -108.55 APE8-dihe-in -69.42, 145.98 APE8-rot-na 76.98 APE67-dihe-in -73.97, -39.08 -95.26, -9.75 APE12-dist-in 8.048 APE11-dist-in 10.262 APE10-dist-in 5.834 APE9-dist-in 3.572 None TPO305 TPO305 EM 2.84 999.0 999.0 A 463 375 49 0 0 0 [[64, 514]] 1.0 8uyh Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
OTHER PINK1 PINK1_PEDHC 8UYHB E0W1I1 121 574 575.0 ANP:601 ATPlike Active DFGin 9.449 14.871 BLAminus -129.89, -169.12 59.53, 64.83 -87.85, 20.05 283.99, 82.98 -70.23, -23.56 in-in in 7.846 Saltbr-in 2.387 HRD-in -70.23, -41.92 63.21, 0.58 in-in-in SNCiii in-in ActLoopNT-in 2.932 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 144.56, -157.47 APE9-dihe-na -105.64, -99.0 APE8-dihe-in -70.54, 139.11 APE8-rot-na 52.17 APE67-dihe-in -71.03, -46.42 -78.22, -15.68 APE12-dist-in 7.74 APE11-dist-in 10.385 APE10-dist-in 6.127 APE9-dist-in 3.781 None TPO305 TPO305 EM 2.84 999.0 999.0 B 463 370 50 0 0 0 [[64, 514]] 1.0 8uyh Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
OTHER PINK1 PINK1_PEDHC 8UYIA E0W1I1 120 572 575.0 ADP:601 ATPlike Active DFGin 9.472 14.492 BLAminus -126.54, -170.24 58.08, 66.04 -87.71, 25.91 289.34, 85.25 -66.89, -21.8 in-in in 7.734 Saltbr-in 2.489 HRD-in -72.82, -45.28 62.7, 4.34 in-in-in SNCiii in-in ActLoopNT-in 2.793 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 149.48, -127.57 APE9-dihe-na -109.63, -105.35 APE8-dihe-in -70.24, 160.24 APE8-rot-na 51.46 APE67-dihe-in -90.34, -42.74 -107.64, 8.21 APE12-dist-in 8.485 APE11-dist-in 10.413 APE10-dist-in 5.828 APE9-dist-in 3.643 None SEP202,TPO305 SEP202,TPO305 EM 3.13 999.0 999.0 A 463 369 49 0 0 0 [[64, 514]] 1.0 8uyi Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
OTHER PINK1 PINK1_PEDHC 8UYIB E0W1I1 122 574 575.0 ADP:601 ATPlike Active DFGin 9.37 14.767 BLAminus -128.32, -168.79 58.11, 64.54 -83.54, 12.33 278.78, 92.3 -66.63, -13.93 in-in in 8.001 Saltbr-in 2.363 HRD-in -66.42, -44.15 62.85, 2.17 in-in-in SNCiii in-in ActLoopNT-in 2.974 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na 143.29, -143.85 APE9-dihe-na -111.19, -100.88 APE8-dihe-in -71.36, 134.31 APE8-rot-na 50.34 APE67-dihe-in -67.38, -41.28 -74.79, -24.08 APE12-dist-in 8.473 APE11-dist-in 10.806 APE10-dist-in 6.227 APE9-dist-in 3.553 None SEP202,TPO305 SEP202,TPO305 EM 3.13 999.0 999.0 B 463 369 51 0 0 0 [[64, 514]] 1.0 8uyi Pediculus humanus OTHER_PINK1_PEDHC PINK1 1e-86 297.1 4 367 364 356 357 358 360 362 193 214 218 331 333 332 334 408 390 385 384 383 382 381 380 379 291 Serine/threonine-protein kinase Pink1, mitochondrial
CAMK CDPK1 CDPK1_PLABA 3Q5IA A0A509AHB6 38 518 523.0 ANP:61634 ATPlike Active DFGin 6.767 14.466 BLAminus -128.23, -176.48 60.5, 79.46 -95.96, 19.56 285.65, 75.94 -57.69, -30.19 in-in in 9.237 Saltbr-in 3.124 HRD-in -79.9, -50.9 74.57, -2.92 in-in-in SNCiii in-in ActLoopNT-in 2.988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.44, 148.94 APE9-dihe-na 143.23, -165.03 APE8-dihe-in -126.86, 133.51 APE8-rot-in 304.61 APE67-dihe-in -56.9, -32.89 -45.51, -52.84 APE12-dist-in 8.589 APE11-dist-in 11.465 APE10-dist-in 5.667 APE9-dist-in 3.634 None None None XRAY 2.1 0.197 0.25 A 504 461 18 0 0 0 [[57, 324]] 1.0 3q5i Plasmodium berghei CAMK_CDPK1_PLABA CAMK 4e-85 291.5 4 256 253 210 211 212 214 216 86 115 119 187 189 188 190 248 237 232 231 230 229 228 227 226 145 Calcium-dependent protein kinase 1
CMGC PSTK1 Q8IL19_PLAF7 3LLTA Q8IL19 535 875 881.0 ANP:877 ATPlike Active DFGin 7.143 15.216 BLAminus -123.92, -179.42 67.73, 65.46 -96.96, 21.34 280.85, 86.26 -60.95, -43.39 in-in in 9.013 Saltbr-in 2.621 HRD-in -67.76, -41.54 71.0, -10.38 in-in-in SNCiii in-in ActLoopNT-in 2.854 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.91, 173.39 APE9-dihe-na 75.57, 154.71 APE8-dihe-in -70.15, 136.15 APE8-rot-in 300.24 APE67-dihe-in -71.32, -17.13 -39.04, -49.24 APE12-dist-in 13.205 APE11-dist-in 11.39 APE10-dist-in 7.514 APE9-dist-in 2.941 None None None XRAY 2.5 0.225 0.267 A 360 341 0 0 0 0 [[552, 874]] 1.0 3llt Plasmodium falciparum CMGC_PSTK1_PLAF7 CMGC 8.3e-71 244.6 2 301 300 719 720 721 723 725 581 596 600 674 676 675 677 756 744 739 738 737 736 735 734 733 631 Protein serine/threonine kinase-1
STE TAOK2 TAOK2_RAT 1U5RA Q9JLS3 12 320 1235.0 ATP:411 ATPlike Active DFGin 6.99 14.24 BLAminus -128.27, -174.18 56.24, 80.49 -99.99, 21.83 293.09, 83.93 -60.11, -26.41 in-in in 8.687 Saltbr-in 2.887 HRD-in -75.95, -53.43 76.2, -2.14 in-in-in SNCiii in-in ActLoopNT-in 2.767 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.19, 153.0 APE9-dihe-na 135.08, -166.49 APE8-dihe-in -116.65, 119.51 APE8-rot-in 301.53 APE67-dihe-in -56.87, -24.9 -27.41, -63.55 APE12-dist-in 8.446 APE11-dist-in 11.391 APE10-dist-in 5.507 APE9-dist-in 3.279 None SEP181 SEP181 XRAY 2.1 0.211 0.244 A 348 309 0 0 0 0 [[28, 281]] 1.0 1u5r Rattus norvegicus STE_TAOK2_RAT STE 1.4e-89 305.8 2 257 256 168 169 170 172 174 57 76 80 148 150 149 151 207 192 187 186 185 184 183 182 181 106 Serine/threonine-protein kinase TAO2
STE TAOK2 TAOK2_RAT 1U5RB Q9JLS3 12 320 1235.0 ATP:412 ATPlike Active DFGin 6.763 13.896 BLAminus -129.03, -178.62 56.08, 82.23 -96.99, 22.88 295.53, 83.61 -63.46, -23.11 in-in in 8.772 Saltbr-in 2.623 HRD-in -71.62, -50.86 71.95, 2.83 in-in-in SNCiii in-in ActLoopNT-in 2.776 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.4, 155.39 APE9-dihe-na 130.83, -165.29 APE8-dihe-in -116.7, 116.24 APE8-rot-in 302.47 APE67-dihe-in -61.68, -22.51 -24.84, -62.59 APE12-dist-in 8.905 APE11-dist-in 11.02 APE10-dist-in 5.282 APE9-dist-in 3.304 None SEP181 SEP181 XRAY 2.1 0.211 0.244 B 348 309 0 0 0 0 [[28, 281]] 1.0 1u5r Rattus norvegicus STE_TAOK2_RAT STE 1.4e-89 305.8 2 257 256 168 169 170 172 174 57 76 80 148 150 149 151 207 192 187 186 185 184 183 182 181 106 Serine/threonine-protein kinase TAO2
CMGC SKY1 SKY1_YEAST 1Q8YA Q03656 144 737 742.0 ADP:60810 ATPlike Active DFGin 5.554 12.776 BLAminus -120.8, -179.55 50.32, 80.87 -92.72, 24.06 294.38, 19.86 -63.4, -18.16 in-in in 8.712 Saltbr-in 2.74 HRD-in -75.73, -45.78 71.18, -6.61 in-in-in SNCiii in-in ActLoopNT-in 2.965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.41, 175.98 APE9-dihe-na 63.08, 152.12 APE8-dihe-in -90.87, 131.26 APE8-rot-in 290.95 APE67-dihe-in -56.18, -26.85 -9.03, -76.03 APE12-dist-in 12.534 APE11-dist-in 10.496 APE10-dist-in 7.507 APE9-dist-in 2.99 None None None XRAY 2.05 0.209 0.244 A 373 351 11 0 0 0 [[158, 706]] 1.0 1q8y Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
CMGC SKY1 SKY1_YEAST 1Q97A Q03656 144 737 742.0 ATP:60485 ATPlike Active DFGin 5.605 12.648 BLAminus -113.61, -176.06 45.65, 81.54 -92.49, 25.33 294.84, 21.0 -61.4, -14.56 in-in in 8.92 Saltbr-in 2.91 HRD-in -73.18, -42.39 69.86, -2.96 in-in-in SNCiii in-in ActLoopNT-in 2.985 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -115.18, 168.88 APE9-dihe-na 68.54, 141.02 APE8-dihe-in -74.6, 131.99 APE8-rot-in 300.34 APE67-dihe-in -58.79, -28.16 -13.13, -73.4 APE12-dist-in 12.586 APE11-dist-in 10.498 APE10-dist-in 7.631 APE9-dist-in 3.163 None None None XRAY 2.3 0.215 0.264 A 373 351 11 0 0 0 [[158, 706]] 1.0 1q97 Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
CMGC SKY1 SKY1_YEAST 1Q99A Q03656 143 737 742.0 ANP:60901 ATPlike Active DFGin 5.863 12.817 BLAminus -114.29, -177.44 55.8, 69.3 -86.87, 21.69 289.5, 16.74 -63.01, -13.14 in-in in 9.01 Saltbr-in 3.393 HRD-in -74.14, -46.77 73.71, -6.86 in-in-in SNCiii in-in ActLoopNT-in 2.983 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.75, 166.8 APE9-dihe-na 68.75, 148.0 APE8-dihe-in -82.45, 139.06 APE8-rot-in 296.77 APE67-dihe-in -63.19, -13.43 -18.75, -76.87 APE12-dist-in 12.636 APE11-dist-in 10.441 APE10-dist-in 7.678 APE9-dist-in 2.996 None None None XRAY 2.11 0.22 0.26 A 373 354 9 0 0 0 [[158, 706]] 1.0 1q99 Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
CMGC SKY1 SKY1_YEAST 1Q99B Q03656 142 737 742.0 ANP:60902 ATPlike Active DFGin 6.007 13.076 BLAminus -119.51, 178.42 55.8, 73.86 -88.54, 22.76 281.2, 12.04 -67.31, -20.83 in-in in 8.991 Saltbr-in 3.413 HRD-in -77.35, -48.77 76.96, -6.7 in-in-in SNCiii in-in ActLoopNT-in 3.054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.48, 168.06 APE9-dihe-na 68.34, 160.67 APE8-dihe-in -99.08, 126.68 APE8-rot-in 289.43 APE67-dihe-in -64.6, -22.58 -5.08, -74.37 APE12-dist-in 12.556 APE11-dist-in 10.321 APE10-dist-in 7.788 APE9-dist-in 3.158 None None None XRAY 2.11 0.22 0.26 B 373 364 0 0 0 0 [[158, 706]] 1.0 1q99 Saccharomyces cerevisiae CMGC_SKY1_YEAST CMGC 8.8e-100 339.7 1 301 301 549 550 551 553 555 187 202 206 291 293 292 294 586 574 569 568 567 566 565 564 563 247 Serine/threonine-protein kinase SKY1
OTHER BUD32 BUD32_YEAST 4WW7A P53323 4 257 261.0 AMP:301 ATPlike Active DFGin 6.607 15.107 BLAminus -125.65, 168.23 67.12, 79.12 -101.96, 21.21 282.36, 92.63 -52.39, -37.98 in-in in 7.952 Saltbr-in 3.029 HRD-in -80.86, -48.82 95.12, -20.58 in-in-na SNCiia in-na ActLoopNT-in 2.886 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -64.64, -46.2 APE9-dihe-na -61.22, -39.41 APE8-dihe-na -68.4, -38.62 APE8-rot-na 171.99 APE67-dihe-na -60.22, -42.81 -57.37, -50.5 APE12-dist-na 15.675 APE11-dist-na 11.246 APE10-dist-na 14.76 APE9-dist-na 11.687 None None None XRAY 1.669 0.194 0.213 A 261 237 21 0 0 0 [[17, 261]] 1.0 4ww7 Saccharomyces cerevisiae OTHER_BUD32_YEAST TP53RK 5e-44 156.6 8 224 217 181 182 183 185 187 52 76 80 158 160 159 161 198 204 199 198 197 196 195 194 193 107 EKC/KEOPS complex subunit BUD32
OTHER BUD32 BUD32_YEAST 4WW9A P53323 4 259 261.0 ADP:302 ATPlike Active DFGin 6.618 15.283 BLAminus -128.14, 172.87 62.95, 73.82 -100.2, 23.36 281.69, 91.54 -52.55, -36.42 in-in in 7.602 Saltbr-in 2.744 HRD-in -80.98, -51.42 97.59, -12.36 in-in-na SNCiia in-na ActLoopNT-in 2.852 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -61.46, -46.34 APE9-dihe-na -60.52, -40.33 APE8-dihe-na -68.91, -38.47 APE8-rot-na 168.71 APE67-dihe-na -62.48, -38.16 -54.4, -51.68 APE12-dist-na 15.732 APE11-dist-na 11.179 APE10-dist-na 14.687 APE9-dist-na 11.734 None None None XRAY 1.951 0.18 0.209 A 261 238 20 0 0 0 [[17, 261]] 1.0 4ww9 Saccharomyces cerevisiae OTHER_BUD32_YEAST TP53RK 5e-44 156.6 8 224 217 181 182 183 185 187 52 76 80 158 160 159 161 198 204 199 198 197 196 195 194 193 107 EKC/KEOPS complex subunit BUD32
TKL NCGRLOCUS634 A0ACD6BAX3_9POAL 8HO6A A0ACD6BAX3 7 305 312.0 ATP:60401 ATPlike Active DFGin 6.377 15.619 BLAminus -139.79, 171.9 63.28, 66.12 -93.24, 62.65 279.35, 60.61 -82.08, -30.35 in-in in 8.644 Saltbr-in 2.728 HRD-in -60.88, -41.53 70.8, -58.95 in-in-in SNCiii in-in ActLoopNT-in 2.72 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.65, 146.26 APE9-dihe-na 148.14, -156.83 APE8-dihe-in -124.83, 132.59 APE8-rot-in 314.24 APE67-dihe-inflip 93.19, -27.63 -56.53, 137.58 APE12-dist-in 9.991 APE11-dist-in 11.771 APE10-dist-in 6.261 APE9-dist-in 5.587 None TPO184,SEP187,TPO188 TPO184,SEP187,TPO188 XRAY 2.1 0.206 0.234 A 326 281 18 0 0 2 [[22, 302]] 1.0 8ho6 Saccharum hybrid cultivar TKL_NCGRLOCUS634_9POAL TKL 3.7e-60 209.7 4 266 263 170 171 172 174 176 58 74 78 150 152 151 153 212 200 195 194 193 192 191 190 189 104 ScRIPK kinase protein
CK1 CKI1 CKI1_SCHPO 1CSNA P40233 6 298 446.0 ATP:299 ATPlike Active DFGin 6.422 13.79 BLAminus -124.8, 177.22 63.85, 88.12 -109.85, 36.77 298.25, 97.14 -71.61, -21.33 in-in in 8.04 Saltbr-in 3.086 HRD-in -68.74, -48.02 63.6, 9.84 in-in-in SNCiii in-in ActLoopNT-in 2.815 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -97.61, -90.82 APE9-dihe-na -65.25, -165.09 APE8-dihe-in -55.42, 111.92 APE8-rot-in 313.89 APE67-dihe-in -55.02, -31.3 -55.98, -42.83 APE12-dist-in 12.741 APE11-dist-in 13.007 APE10-dist-in 7.16 APE9-dist-in 4.794 None None None XRAY 2.0 0.207 999.0 A 298 293 0 0 0 0 [[12, 280]] 1.0 1csn Schizosaccharomyces pombe CK1_CKI1_SCHPO CK1 8e-95 323.1 1 261 261 153 154 155 157 159 41 55 59 128 130 129 131 200 188 183 182 181 180 179 178 177 86 Casein kinase I homolog 1
AGC PRKACA KAPCA_PIG 1CDKA P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.843 14.33 BLAminus -113.76, -166.2 47.38, 80.03 -85.76, 16.06 278.85, 56.4 -55.46, -28.11 in-in in 9.034 Saltbr-in 2.899 HRD-in -94.66, -56.81 78.16, -3.52 in-in-in SNCiii in-in ActLoopNT-in 2.985 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.51, 155.2 APE9-dihe-na 137.51, -153.75 APE8-dihe-in -125.49, 136.2 APE8-rot-in 297.83 APE67-dihe-in -73.46, -24.38 -35.73, -51.43 APE12-dist-in 7.997 APE11-dist-in 11.418 APE10-dist-in 5.766 APE9-dist-in 3.642 None TPO198 TPO198 XRAY 2.0 0.197 999.0 A 350 343 0 0 0 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_PIG 1CDKB P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.907 14.511 BLAminus -124.27, -171.72 50.82, 76.29 -83.58, 17.26 280.88, 62.25 -47.74, -29.83 in-in in 8.889 Saltbr-in 2.883 HRD-in -87.48, -57.48 77.49, 1.67 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 159.84 APE9-dihe-na 137.3, -140.74 APE8-dihe-in -136.57, 132.27 APE8-rot-in 304.84 APE67-dihe-in -69.16, -27.96 -34.59, -53.92 APE12-dist-in 8.348 APE11-dist-in 11.514 APE10-dist-in 6.08 APE9-dist-in 3.744 None TPO198 TPO198 XRAY 2.0 0.197 999.0 B 350 343 0 0 0 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
CMGC TVAG125560 A2F9N1_TRIV3 9AV7A A2F9N1 15 318 320.0 ANP:401 ATPlike Active DFGin 7.636 16.424 BLAminus -120.42, -177.29 61.53, 69.44 -89.47, 18.08 296.84, 80.84 -66.47, -28.11 in-in in 9.462 Saltbr-in 3.092 HRD-in -77.85, -46.91 69.04, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.954 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.39, -177.21 APE9-dihe-na 62.4, -175.9 APE8-dihe-in -115.65, 153.97 APE8-rot-in 297.25 APE67-dihe-inflip 82.79, -6.3 -53.46, 134.7 APE12-dist-in 12.695 APE11-dist-in 10.496 APE10-dist-in 6.317 APE9-dist-in 3.013 None None None XRAY 2.1 0.202 0.246 A 328 304 0 0 0 0 [[27, 312]] 1.0 9av7 Trichomonas vaginalis CMGC_TVAG125560_TRIV3 CMGC 2.3e-51 180.8 1 301 301 162 163 164 166 168 56 69 73 141 143 142 144 202 189 184 183 182 181 180 179 178 102 non-specific serine/threonine protein kinase
CMGC ACK2 CSK2A_MAIZE 1DS5A P28523 1 328 332.0 AMP:60501 ATPlike Active DFGin 7.256 16.138 BLAminus -131.0, -177.8 59.5, 94.79 -110.09, 23.49 292.94, 70.46 -65.1, -12.46 in-in in 9.41 Saltbr-in 2.992 HRD-in -75.82, -4.13 22.93, 18.86 in-in-in SNCiii in-in ActLoopNT-in 2.927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, -170.21 APE9-dihe-na 48.23, -163.7 APE8-dihe-in -120.52, 135.99 APE8-rot-in 299.66 APE67-dihe-in -32.14, -36.61 -18.26, -83.73 APE12-dist-in 12.442 APE11-dist-in 10.293 APE10-dist-in 6.391 APE9-dist-in 3.166 None None None XRAY 3.16 0.214 0.289 A 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha
CMGC ACK2 CSK2A_MAIZE 1DS5B P28523 1 328 332.0 AMP:60801 ATPlike Active DFGin 7.364 16.317 BLAminus -130.6, -175.34 56.5, 69.06 -85.22, 18.36 296.09, 73.67 -62.25, -12.27 in-in in 9.134 Saltbr-in 2.468 HRD-in -78.74, -8.85 28.88, 23.14 in-in-in SNCiii in-in ActLoopNT-in 2.85 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.31, -172.94 APE9-dihe-na 48.86, -163.66 APE8-dihe-in -122.01, 142.21 APE8-rot-in 298.66 APE67-dihe-in -27.41, -40.26 -18.35, -90.48 APE12-dist-in 12.513 APE11-dist-in 10.354 APE10-dist-in 6.441 APE9-dist-in 3.101 None None None XRAY 3.16 0.214 0.289 B 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha
CMGC ACK2 CSK2A_MAIZE 1DS5C P28523 1 328 332.0 AMP:60601 ATPlike Active DFGin 7.431 16.3 BLAminus -130.04, -171.91 47.17, 91.25 -104.25, 20.64 295.37, 72.57 -63.12, -7.55 in-in in 9.164 Saltbr-in 2.64 HRD-in -79.02, -3.04 26.4, 20.9 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.73, -170.98 APE9-dihe-na 48.52, -163.45 APE8-dihe-in -120.17, 138.04 APE8-rot-in 300.76 APE67-dihe-in -34.03, -36.56 -18.28, -84.34 APE12-dist-in 12.439 APE11-dist-in 10.299 APE10-dist-in 6.441 APE9-dist-in 3.093 None None None XRAY 3.16 0.214 0.289 C 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha
CMGC ACK2 CSK2A_MAIZE 1DS5D P28523 1 328 332.0 AMP:60701 ATPlike Active DFGin 7.269 16.174 BLAminus -138.27, -179.17 62.24, 74.19 -94.05, 17.43 296.9, 73.95 -62.87, -11.79 in-in in 9.511 Saltbr-in 2.483 HRD-in -81.25, -4.13 24.81, 26.82 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.11, -172.61 APE9-dihe-na 51.23, -160.96 APE8-dihe-in -124.78, 137.86 APE8-rot-in 294.35 APE67-dihe-in -36.36, -34.26 -18.24, -83.45 APE12-dist-in 12.473 APE11-dist-in 10.246 APE10-dist-in 6.365 APE9-dist-in 3.133 None None None XRAY 3.16 0.214 0.289 D 332 328 0 0 0 0 [[34, 319]] 1.0 1ds5 Zea mays CMGC_ACK2_MAIZE CMGC 1.8e-65 227.0 1 301 301 169 170 171 173 175 63 76 80 148 150 149 151 209 196 191 190 189 188 187 186 185 109 Casein kinase II subunit alpha