| Name | PDB identifier |
|---|---|
| Abrocitinib | D7D |
| Adavosertib | 8X7 |
| Afatinib | 0WM |
| Alectinib | EMH |
| Alisertib | A5B |
| Alpelisib | 1LT |
| Altiratinib | A9I |
| Alvocidib | CPB |
| Apitolisib | 980 |
| Asciminib | AY7 |
| Avutometinib | CHU |
| Axitinib | AXI |
| Azenosertib | 05J |
| Bafetinib | 406 |
| Baricitinib | 3JW |
| Belizatinib | 0UV |
| Belumosudil | ICQ |
| Belvarafenib | V1Y |
| Bezuclastinib | WEJ |
| Bimiralisib | A3W |
| Binimetinib | QO7 |
| Bosutinib | DB8 |
| Brigatinib | 6GY |
| Buparlisib | SD5 |
| Cabozantinib | XIN |
| Capivasertib | 0XZ |
| Ceritinib | 4MK |
| Cobimetinib | EUI |
| Copanlisib | 6E2 |
| Crenolanib | 6T2 |
| Crizotinib | VGH |
| Dabrafenib | P06 |
| Dacomitinib | 1C9 |
| Danusertib | 627 |
| Dasatinib | 1N1 |
| Decernotinib | VJK |
| Defactinib | 7KD |
| Defosbarasertib | YJA |
| Delgocitinib | FHX |
| Dinaciclib | 1QK |
| Doramapimod | B96 |
| Dovitinib | 38O |
| Ebvaciclib | WG1 |
| Empesertib | 8QW |
| Entospletinib | CG9 |
| Entrectinib | YMX |
| Erdafitinib | SSF |
| Erlotinib | AQ4 |
| Evobrutinib | MZJ |
| Fasudil | M77 |
| Fedratinib | 2TA |
| Fenebrutinib | 9AJ |
| Filgotinib | 2HB |
| Foretinib | 88Z |
| Fostamatinib | 2RC |
| Futibatinib | TZ0 |
| Gedatolisib | VL1 |
| Gefitinib | IRE |
| Genistein | GEN |
| Gilteritinib | C6F |
| Golvatinib | GV0 |
| Ibrutinib | 1E8 |
| Idelalisib | 40L |
| Imatinib | STI |
| Inavolisib | X3N |
| Infigratinib | 07J |
| Ipatasertib | 0RF |
| Izorlisib | MMD |
| Laduviglusib | 65C |
| Lanraplenib | R6D |
| Lapatinib | FMM |
| Lartesertib | UGK |
| Leniolisib | 9NQ |
| Lenvatinib | LEV |
| Lerociclib | EG7 |
| Lestaurtinib | 2V9 |
| Lorlatinib | 5P8 |
| Lucitanib | 3ZC |
| Masitinib | G65 |
| Merestinib | L1X |
| Midostaurin | 2K2 |
| Milciclib | P48 |
| Miransertib | 6S1 |
| Mirdametinib | 4BM |
| Mivavotinib | 7KG |
| Momelotinib | C87 |
| Motesanib | 706 |
| Naporafenib | K81 |
| Naquotinib | 8RC |
| Neflamapimod | 52P |
| Nemiralisib | VVX |
| Nemtabrutinib | HRA |
| Neratinib | HKI |
| Nilotinib | NIL |
| Nintedanib | XIN |
| Omipalisib | ZIG |
| Onvansertib | 937 |
| Orantinib | SU6 |
| Osimertinib | YY3 |
| Pacritinib | 6T3 |
| Padnarsertib | 96Q |
| Palbociclib | LQQ |
| Pamapimod | FLW |
| Pelitinib | 93J |
| Pemigatinib | 8ZF |
| Peposertib | 1IX |
| Pexidartinib | P31 |
| Pictilisib | GD9 |
| Pimasertib | QOA |
| Pirtobrutinib | Y7W |
| Ponatinib | 0LI |
| Pralsetinib | Q4J |
| Quizartinib | P30 |
| Ravoxertinib | 6QB |
| Rebastinib | 919 |
| Refametinib | VRA |
| Repotrectinib | 7GI |
| Ribociclib | 6ZZ |
| Rigosertib | 6FS |
| Rilzabrutinib | R1L |
| Roblitinib | FGF |
| Rociletinib | 8JC |
| Roniciclib | R0N |
| Ruboxistaurin | LY4 |
| Ruxolitinib | RXT |
| Samuraciclib | I74 |
| Sapanisertib | FE5 |
| Saracatinib | H8H |
| Savolitinib | V0L |
| Seliciclib | RRC |
| Selonsertib | NJV |
| Selumetinib | 3EW |
| Semaxanib | X2M |
| Silmitasertib | 3NG |
| Simurosertib | O1V |
| Sorafenib | BAX |
| Sotrastaurin | LW4 |
| Sunitinib | B49 |
| Talmapimod | 469 |
| Tanzisertib | KBI |
| Taselisib | 799 |
| Temuterkib | KE8 |
| Tepotinib | 3E8 |
| Tirbanibulin | DN0 |
| Tivantinib | TIV |
| Tivozanib | AV9 |
| Tizaterkib | LHZ |
| Toceranib | BWC |
| Tofacitinib | MI1 |
| Tomivosertib | N45 |
| Tovorafenib | QOP |
| Tozasertib | VX6 |
| Trametinib | QOM |
| Triciribine | ZJB |
| Ulixertinib | EVK |
| Vandetanib | ZD6 |
| Vemurafenib | 32' |
| Vimseltinib | Z6V |
| Volasertib | IBI |
| Zanubrutinib | BA0 |
| Zimlovisertib | 8CD |
| Zoligratinib | LWJ |