FDA approved list of protein kinase inhibitors with known structure

Name PDB identifier
Abrocitinib D7D
Adavosertib 8X7
Afatinib 0WM
Alectinib EMH
Alisertib A5B
Alpelisib 1LT
Altiratinib A9I
Alvocidib CPB
Apitolisib 980
Asciminib AY7
Avutometinib CHU
Axitinib AXI
Azenosertib 05J
Bafetinib 406
Baricitinib 3JW
Belizatinib 0UV
Belumosudil ICQ
Belvarafenib V1Y
Bezuclastinib WEJ
Bimiralisib A3W
Binimetinib QO7
Bosutinib DB8
Brigatinib 6GY
Buparlisib SD5
Cabozantinib XIN
Capivasertib 0XZ
Ceritinib 4MK
Cobimetinib EUI
Copanlisib 6E2
Crenolanib 6T2
Crizotinib VGH
Dabrafenib P06
Dacomitinib 1C9
Danusertib 627
Dasatinib 1N1
Decernotinib VJK
Defactinib 7KD
Defosbarasertib YJA
Delgocitinib FHX
Dinaciclib 1QK
Doramapimod B96
Dovitinib 38O
Ebvaciclib WG1
Empesertib 8QW
Entospletinib CG9
Entrectinib YMX
Erdafitinib SSF
Erlotinib AQ4
Evobrutinib MZJ
Fasudil M77
Fedratinib 2TA
Fenebrutinib 9AJ
Filgotinib 2HB
Foretinib 88Z
Fostamatinib 2RC
Futibatinib TZ0
Gedatolisib VL1
Gefitinib IRE
Genistein GEN
Gilteritinib C6F
Golvatinib GV0
Ibrutinib 1E8
Idelalisib 40L
Imatinib STI
Inavolisib X3N
Infigratinib 07J
Ipatasertib 0RF
Izorlisib MMD
Laduviglusib 65C
Lanraplenib R6D
Lapatinib FMM
Lartesertib UGK
Leniolisib 9NQ
Lenvatinib LEV
Lerociclib EG7
Lestaurtinib 2V9
Lorlatinib 5P8
Lucitanib 3ZC
Masitinib G65
Merestinib L1X
Midostaurin 2K2
Milciclib P48
Miransertib 6S1
Mirdametinib 4BM
Mivavotinib 7KG
Momelotinib C87
Motesanib 706
Naporafenib K81
Naquotinib 8RC
Neflamapimod 52P
Nemiralisib VVX
Nemtabrutinib HRA
Neratinib HKI
Nilotinib NIL
Nintedanib XIN
Omipalisib ZIG
Onvansertib 937
Orantinib SU6
Osimertinib YY3
Pacritinib 6T3
Padnarsertib 96Q
Palbociclib LQQ
Pamapimod FLW
Pelitinib 93J
Pemigatinib 8ZF
Peposertib 1IX
Pexidartinib P31
Pictilisib GD9
Pimasertib QOA
Pirtobrutinib Y7W
Ponatinib 0LI
Pralsetinib Q4J
Quizartinib P30
Ravoxertinib 6QB
Rebastinib 919
Refametinib VRA
Repotrectinib 7GI
Ribociclib 6ZZ
Rigosertib 6FS
Rilzabrutinib R1L
Roblitinib FGF
Rociletinib 8JC
Roniciclib R0N
Ruboxistaurin LY4
Ruxolitinib RXT
Samuraciclib I74
Sapanisertib FE5
Saracatinib H8H
Savolitinib V0L
Seliciclib RRC
Selonsertib NJV
Selumetinib 3EW
Semaxanib X2M
Silmitasertib 3NG
Simurosertib O1V
Sorafenib BAX
Sotrastaurin LW4
Sunitinib B49
Talmapimod 469
Tanzisertib KBI
Taselisib 799
Temuterkib KE8
Tepotinib 3E8
Tirbanibulin DN0
Tivantinib TIV
Tivozanib AV9
Tizaterkib LHZ
Toceranib BWC
Tofacitinib MI1
Tomivosertib N45
Tovorafenib QOP
Tozasertib VX6
Trametinib QOM
Triciribine ZJB
Ulixertinib EVK
Vandetanib ZD6
Vemurafenib 32'
Vimseltinib Z6V
Volasertib IBI
Zanubrutinib BA0
Zimlovisertib 8CD
Zoligratinib LWJ
A complete list of FDA approved inhibitors can be obtained here.