AGC_PRKACA (cAMP-dependent protein kinase catalytic subunit alpha)

Total number of chains: 80
Active chains: 52
Uniprot: KAPCA_HUMAN
Kinase Domain Residues: 44 - 298
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 70 87.5% AF-P17612-K1A
DFGin ABAminus 10 12.5% 4AE6A

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PRKACA 4WB8A P17612 16 351 351.0 ATP:60401 ATPlike Active DFGin 5.6838 14.4142 BLAminus -121.45, -177.2 62.67, 77.75 -91.98, 24.58 268.87, 53.09 -58.34, -31.51 in-in in 8.9131 Saltbr-in 2.7592 HRD-in -95.2, -52.32 70.44, 11.38 in-in-in SNCiii in-in ActLoopNT-in 2.9124 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.85, 164.58 APE9-dihe-na 131.46, -156.38 APE8-dihe-in -129.55, 139.43 APE8-rot-in 297.11 APE67-dihe-in -60.54, -22.69 -52.03, -49.04 APE12-dist-in 8.0978 APE11-dist-in 11.3919 APE10-dist-in 5.8266 APE9-dist-in 3.4975 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.164 0.184 A 337.0 336.0 0 25 25 0 [[44, 298]] 1.0 4wb8 AGC_PRKACA_HUMAN AGC 4e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4WB5A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 5.5996 14.452 BLAminus -123.05, 176.84 68.94, 80.02 -91.46, 24.86 270.2, 52.92 -60.74, -31.43 in-in in 9.0296 Saltbr-in 2.7148 HRD-in -92.12, -52.84 69.8, 13.37 in-in-in SNCiii in-in ActLoopNT-in 2.9178 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.48, 163.75 APE9-dihe-na 132.31, -149.49 APE8-dihe-in -132.05, 134.14 APE8-rot-in 301.14 APE67-dihe-in -60.1, -21.12 -48.44, -50.23 APE12-dist-in 8.0121 APE11-dist-in 11.4001 APE10-dist-in 5.799 APE9-dist-in 3.5673 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.641 0.165 0.196 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 4wb5 AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4WB7A P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.4448 14.6485 BLAminus -119.06, -174.39 59.4, 77.28 -89.09, 26.42 267.74, 51.48 -60.48, -28.34 in-in in 8.8699 Saltbr-in 2.7695 HRD-in -93.55, -50.9 68.82, 8.95 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.63, 158.06 APE9-dihe-na 139.02, -156.91 APE8-dihe-in -126.94, 137.23 APE8-rot-in 299.54 APE67-dihe-in -64.26, -23.0 -50.4, -48.13 APE12-dist-in 8.1804 APE11-dist-in 11.5397 APE10-dist-in 5.9545 APE9-dist-in 3.7228 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 4wb7 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4WB7B P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.3799 14.7121 BLAminus -115.93, -176.79 62.38, 75.33 -88.91, 25.18 264.71, 51.71 -56.9, -30.26 in-in in 8.9624 Saltbr-in 2.7732 HRD-in -94.01, -50.55 67.24, 10.48 in-in-in SNCiii in-in ActLoopNT-in 2.9391 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.07, 161.39 APE9-dihe-na 132.31, -156.17 APE8-dihe-in -127.2, 138.18 APE8-rot-in 298.14 APE67-dihe-in -59.62, -23.37 -52.63, -48.78 APE12-dist-in 8.1977 APE11-dist-in 11.5627 APE10-dist-in 5.9704 APE9-dist-in 3.6419 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 4wb7 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6BYRA P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.6263 14.6159 BLAminus -128.29, 177.03 62.06, 86.64 -97.54, 28.59 271.87, 66.62 -63.2, -33.23 in-in in 8.8079 Saltbr-in 3.1965 HRD-in -87.43, -52.47 67.28, 5.18 in-in-in SNCiii in-in ActLoopNT-in 3.1931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.51, 153.24 APE9-dihe-na 149.32, -133.8 APE8-dihe-in -139.35, 133.91 APE8-rot-in 312.31 APE67-dihe-in -68.4, -6.95 -52.73, -48.25 APE12-dist-in 8.7341 APE11-dist-in 11.0763 APE10-dist-in 5.6298 APE9-dist-in 3.4915 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 6byr AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6BYRC P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.6794 14.3401 BLAminus -129.89, 172.29 61.76, 74.25 -79.2, 34.93 281.69, 54.14 -61.8, -27.34 in-in in 8.7335 Saltbr-in 2.4981 HRD-in -93.13, -49.8 64.55, 7.44 in-in-in SNCiii in-in ActLoopNT-in 3.0524 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.29, 161.94 APE9-dihe-na 130.51, -156.26 APE8-dihe-in -112.31, 134.09 APE8-rot-in 302.07 APE67-dihe-in -64.15, -16.52 -52.64, -41.39 APE12-dist-in 8.3162 APE11-dist-in 11.1062 APE10-dist-in 5.7667 APE9-dist-in 3.6182 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 C 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 6byr AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 9EDCA P17612 14 351 351.0 ATP:60400 ATPlike Active DFGin 5.6262 13.772 BLAminus -125.61, -173.52 60.53, 69.6 -81.59, 16.86 273.36, 51.23 -62.38, -30.28 in-in in 9.1286 Saltbr-in 2.9998 HRD-in -112.54, -46.7 65.17, 1.82 in-in-in SNCiii in-in ActLoopNT-in 3.1404 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.87, 159.92 APE9-dihe-na 136.42, -156.18 APE8-dihe-in -101.13, 126.83 APE8-rot-in 299.98 APE67-dihe-in -84.76, -8.6 -60.74, -28.35 APE12-dist-in 7.9989 APE11-dist-in 11.1115 APE10-dist-in 5.7968 APE9-dist-in 3.7475 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 EM 4.18 999.0 999.0 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9edc AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4WB6A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 6.0678 14.3977 BLAminus -118.38, -169.49 51.77, 82.47 -95.61, 17.78 271.18, 55.73 -42.8, -37.29 in-in in 8.8304 Saltbr-in 2.5613 HRD-in -94.17, -52.18 74.17, 2.46 in-in-in SNCiii in-in ActLoopNT-in 2.9483 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.55, 166.68 APE9-dihe-na 116.18, 128.45 APE8-dihe-in -46.62, 128.74 APE8-rot-in 303.5 APE67-dihe-in -58.01, -23.74 -49.09, -50.89 APE12-dist-in 8.0462 APE11-dist-in 11.764 APE10-dist-in 6.2427 APE9-dist-in 3.7665 L206R SEP11,SEP140,TPO198 SEP11,SEP140,TPO198 XRAY 2.1 0.19 0.237 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 4wb6 AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4WB6B P17612 9 351 351.0 ATP:60401 ATPlike Active DFGin 5.8721 14.0727 BLAminus -117.82, -168.32 53.27, 78.35 -91.25, 29.34 274.97, 62.46 -60.26, -35.85 in-in in 8.6873 Saltbr-in 2.7501 HRD-in -101.62, -46.5 64.42, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.9461 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.38, 164.15 APE9-dihe-na 120.83, 133.18 APE8-dihe-in -48.66, 125.41 APE8-rot-in 298.86 APE67-dihe-in -54.58, -37.6 -53.55, -42.52 APE12-dist-in 8.078 APE11-dist-in 11.6173 APE10-dist-in 6.2035 APE9-dist-in 3.8221 L206R SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.19 0.237 B 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 4wb6 AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5J5XA P17612 10 351 351.0 6J9:60404 Allosteric Active DFGin 6.1307 14.2674 BLAminus -130.51, 173.14 68.75, 93.05 -105.74, 27.05 279.27, 61.24 -64.37, -20.92 in-in in 8.4945 Saltbr-in 2.7357 HRD-in -82.45, -52.91 66.97, 1.69 in-in-in SNCiii in-in ActLoopNT-in 2.8965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.53, 148.7 APE9-dihe-na 119.01, 165.11 APE8-dihe-in -70.44, 134.99 APE8-rot-in 296.24 APE67-dihe-in -60.26, -38.48 -54.53, -34.6 APE12-dist-in 7.8109 APE11-dist-in 11.1325 APE10-dist-in 5.6005 APE9-dist-in 3.9887 None TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.24 0.309 A 351.0 342.0 0 25 25 0 [[44, 298]] 1.0 5j5x AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA AF-P17612-K1A P17612 36 306 351.0 No_ligand No_ligand Active DFGin 5.9552 14.1005 BLAminus -112.06, -162.49 41.01, 73.74 -80.57, 22.27 279.02, 69.01 -57.23, -32.63 in-in in 8.7297 Saltbr-in 2.6065 HRD-in -81.22, -48.08 66.27, 5.12 in-in-in SNCiii in-in ActLoopNT-in 2.9414 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.31, 161.49 APE9-dihe-na 113.97, -179.99 APE8-dihe-in -91.88, 135.09 APE8-rot-in 302.21 APE67-dihe-in -65.91, -23.79 -48.59, -45.69 APE12-dist-in 8.0558 APE11-dist-in 11.4784 APE10-dist-in 5.7165 APE9-dist-in 3.4962 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 25 25 0 [[44, 298]] 1.0 AF-P17612-K1 AGC_PRKACA_HUMAN AGC 1.8e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA AF-P17612-K3A P17612 36 306 351.0 No_ligand No_ligand Active DFGin 5.9894 14.1821 BLAminus -127.06, -175.23 47.34, 85.15 -88.29, 17.62 289.75, 82.76 -56.25, -31.52 in-in in 8.7982 Saltbr-in 2.6486 HRD-in -85.43, -51.15 69.13, 5.21 in-in-in SNCiii in-in ActLoopNT-in 2.8708 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.07, 161.67 APE9-dihe-na 110.83, -179.43 APE8-dihe-in -90.4, 132.09 APE8-rot-in 300.17 APE67-dihe-in -66.95, -21.36 -48.38, -45.21 APE12-dist-in 8.0717 APE11-dist-in 11.1565 APE10-dist-in 5.4898 APE9-dist-in 3.4162 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 25 25 0 [[44, 298]] 1.0 AF-P17612-K3 AGC_PRKACA_HUMAN AGC 1.8e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6NO7C P17612 12 351 351.0 No_ligand No_ligand Active DFGin 5.3091 14.0414 BLAminus -119.31, 176.37 65.24, 77.94 -84.43, 19.43 273.37, 51.07 -43.97, -41.52 in-in in 8.987 Saltbr-in 2.3597 HRD-in -94.38, -54.81 73.77, 10.87 in-in-in SNCiii in-in ActLoopNT-in 2.9661 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.7, 149.95 APE9-dihe-na 149.29, -142.75 APE8-dihe-in -132.31, 130.88 APE8-rot-in 297.15 APE67-dihe-in -65.36, -25.54 -38.33, -55.04 APE12-dist-in 8.372 APE11-dist-in 10.8625 APE10-dist-in 5.5723 APE9-dist-in 3.1598 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 C 350.0 340.0 0 25 25 0 [[44, 298]] 1.0 6no7 AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3AGMA P17612 13 351 351.0 No_ligand No_ligand Active DFGin 6.4463 13.4021 BLAminus -121.71, 165.51 70.43, 93.14 -102.22, 24.88 291.91, 69.39 -56.91, -34.43 in-in in 8.7602 Saltbr-in 2.8017 HRD-in -90.0, -49.9 65.54, 1.86 in-in-in SNCiii in-in ActLoopNT-in 2.9866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.66, 155.53 APE9-dihe-na 129.13, -155.89 APE8-dihe-in -119.08, 128.77 APE8-rot-in 315.26 APE67-dihe-in -58.72, -28.41 -42.89, -48.17 APE12-dist-in 7.9624 APE11-dist-in 11.3404 APE10-dist-in 5.7893 APE9-dist-in 3.8393 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.277 0.265 A 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 3agm AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5IZFA P17612 14 351 351.0 No_ligand No_ligand Active DFGin 6.4693 14.6805 BLAminus -115.33, 168.85 66.79, 92.72 -104.07, 26.57 271.02, 67.91 -60.32, -26.19 in-in in 8.9198 Saltbr-in 2.86 HRD-in -91.12, -53.12 70.24, 3.28 in-in-in SNCiii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.28, 154.6 APE9-dihe-na 132.55, -178.51 APE8-dihe-in -93.41, 131.47 APE8-rot-in 300.25 APE67-dihe-in -61.6, -25.88 -48.77, -44.1 APE12-dist-in 7.9991 APE11-dist-in 11.6508 APE10-dist-in 5.9844 APE9-dist-in 4.1432 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.232 0.27 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 5izf AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3NX8A P17612 16 351 351.0 No_ligand No_ligand Active DFGin 6.2174 14.3207 BLAminus -121.41, 174.36 68.59, 92.57 -100.19, 21.71 266.05, 56.03 -54.66, -29.9 in-in in 8.8669 Saltbr-in 3.0948 HRD-in -83.14, -56.31 66.43, 12.16 in-in-in SNCiii in-in ActLoopNT-in 3.0216 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.5, 160.02 APE9-dihe-na 128.98, -158.22 APE8-dihe-in -117.99, 132.74 APE8-rot-in 294.49 APE67-dihe-in -53.23, -32.68 -47.46, -50.82 APE12-dist-in 8.0488 APE11-dist-in 11.4278 APE10-dist-in 5.8527 APE9-dist-in 3.6257 None TPO198,SEP339 TPO198,LGY293,SEP339 XRAY 2.0 0.22 0.288 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 3nx8 AGC_PRKACA_HUMAN AGC 2.9e-94 321.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 9DCDA P17612 14 351 351.0 A1A3J:60401 Type1 Active DFGin 5.9288 14.45 BLAminus -126.13, 173.68 64.63, 91.94 -99.88, 28.46 273.99, 56.84 -61.81, -26.4 in-in in 9.1249 Saltbr-in 2.7292 HRD-in -91.13, -53.48 71.25, 11.66 in-in-in SNCiii in-in ActLoopNT-in 2.8197 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.7, 158.74 APE9-dihe-na 136.61, -155.83 APE8-dihe-in -120.28, 133.14 APE8-rot-in 302.66 APE67-dihe-in -56.79, -23.93 -44.41, -54.9 APE12-dist-in 8.0289 APE11-dist-in 11.4422 APE10-dist-in 5.9126 APE9-dist-in 3.6174 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.7 0.174 0.191 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9dcd AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3AGLA P17612 11 351 351.0 A03:60351 Type1 Active DFGin 6.145 14.1866 BLAminus -123.32, 177.62 64.25, 83.52 -96.46, 22.51 272.11, 61.62 -58.64, -28.46 in-in in 8.4913 Saltbr-in 2.8863 HRD-in -82.44, -53.5 74.32, 9.67 in-in-in SNCiii in-in ActLoopNT-in 2.8897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.19, 166.18 APE9-dihe-na 128.76, -154.1 APE8-dihe-in -126.1, 126.27 APE8-rot-in 292.64 APE67-dihe-in -59.45, -23.51 -43.73, -52.47 APE12-dist-in 8.0899 APE11-dist-in 11.2847 APE10-dist-in 5.6424 APE9-dist-in 3.6922 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.2 0.237 A 351.0 341.0 0 25 25 0 [[44, 298]] 1.0 3agl AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3AGLB P17612 15 351 351.0 A03:60351 Type1 Active DFGin 6.244 14.2587 BLAminus -119.17, 172.99 64.04, 88.92 -97.96, 24.36 271.27, 65.91 -60.24, -24.04 in-in in 8.4832 Saltbr-in 2.838 HRD-in -81.23, -56.2 72.88, 10.89 in-in-in SNCiii in-in ActLoopNT-in 2.8655 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.17, 153.35 APE9-dihe-na 137.51, -153.25 APE8-dihe-in -122.43, 130.68 APE8-rot-in 303.24 APE67-dihe-in -59.0, -24.94 -49.14, -44.94 APE12-dist-in 8.0815 APE11-dist-in 11.3224 APE10-dist-in 5.744 APE9-dist-in 3.8805 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.2 0.237 B 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3agl AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3L9LA P17612 12 351 351.0 L9L:60351 Type1 Active DFGin 6.6864 14.5845 BLAminus -131.42, 170.84 67.14, 98.79 -112.52, 31.48 281.78, 68.95 -76.6, -5.02 in-in in 9.118 Saltbr-in 3.0215 HRD-in -66.86, -56.55 70.6, 11.25 in-in-in SNCiii in-in ActLoopNT-in 2.8997 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.79, 159.06 APE9-dihe-na 115.3, -161.08 APE8-dihe-in -112.72, 124.05 APE8-rot-in 306.01 APE67-dihe-in -58.13, -24.33 -29.04, -60.55 APE12-dist-in 8.3496 APE11-dist-in 11.1877 APE10-dist-in 5.5865 APE9-dist-in 3.5153 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.262 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 3l9l AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3L9LB P17612 13 351 351.0 L9L:60351 Type1 Active DFGin 6.5037 14.7481 BLAminus -126.06, 169.3 70.23, 93.91 -105.72, 28.14 277.25, 72.68 -68.61, -5.61 in-in in 9.1221 Saltbr-in 3.0925 HRD-in -71.18, -54.73 64.89, 13.74 in-in-in SNCiii in-in ActLoopNT-in 2.96 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.39, 167.34 APE9-dihe-na 115.39, -170.56 APE8-dihe-in -110.93, 132.83 APE8-rot-in 304.32 APE67-dihe-in -49.56, -29.7 -32.05, -69.65 APE12-dist-in 8.223 APE11-dist-in 11.2936 APE10-dist-in 5.685 APE9-dist-in 3.5296 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.262 B 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 3l9l AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3OOGA P17612 17 351 351.0 YTP:62001 Type1 Active DFGin 5.8967 14.3236 BLAminus -121.7, 177.27 65.88, 89.72 -99.72, 18.72 271.46, 61.56 -55.08, -24.51 in-in in 9.0925 Saltbr-in 2.5643 HRD-in -88.93, -49.19 62.2, 8.05 in-in-in SNCiii in-in ActLoopNT-in 2.8865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.22, 156.24 APE9-dihe-na 130.48, -158.98 APE8-dihe-in -121.53, 132.57 APE8-rot-in 295.61 APE67-dihe-in -56.76, -31.12 -46.34, -49.72 APE12-dist-in 8.1836 APE11-dist-in 11.5607 APE10-dist-in 5.9904 APE9-dist-in 3.7821 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.276 A 351.0 335.0 0 25 25 0 [[44, 298]] 1.0 3oog AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3OVVA P17612 15 351 351.0 1SB:62001 Type1 Active DFGin 5.6952 14.513 BLAminus -122.03, 173.75 63.75, 85.64 -91.93, 24.88 270.34, 49.38 -58.53, -29.2 in-in in 9.1567 Saltbr-in 2.6429 HRD-in -85.42, -51.64 68.38, 18.21 in-in-in SNCiii in-in ActLoopNT-in 2.9726 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.97, 161.66 APE9-dihe-na 131.92, -151.97 APE8-dihe-in -126.88, 132.92 APE8-rot-in 299.89 APE67-dihe-in -61.32, -22.22 -45.4, -52.6 APE12-dist-in 8.1277 APE11-dist-in 11.5503 APE10-dist-in 5.9067 APE9-dist-in 3.5315 None TPO198,SEP339 TPO198,SEP339 XRAY 1.58 0.186 0.232 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3ovv AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3OWPA P17612 16 351 351.0 2SB:62001 Type1 Active DFGin 5.7967 14.5771 BLAminus -129.79, 179.44 68.22, 88.81 -97.88, 23.63 269.47, 50.63 -59.8, -24.73 in-in in 9.0211 Saltbr-in 2.6482 HRD-in -91.6, -55.1 70.56, 10.08 in-in-in SNCiii in-in ActLoopNT-in 2.8362 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.46, 156.32 APE9-dihe-na 133.26, -159.94 APE8-dihe-in -117.71, 131.95 APE8-rot-in 303.89 APE67-dihe-in -56.68, -26.5 -44.05, -53.81 APE12-dist-in 8.0794 APE11-dist-in 11.5299 APE10-dist-in 5.9471 APE9-dist-in 3.8249 None TPO198,SEP339 TPO198,SEP339 XRAY 1.88 0.172 0.211 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 3owp AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3OXTA P17612 15 351 351.0 3SB:62001 Type1 Active DFGin 5.7237 14.3223 BLAminus -130.49, 176.59 67.71, 88.75 -96.86, 20.88 271.58, 55.14 -54.8, -35.77 in-in in 9.1078 Saltbr-in 2.754 HRD-in -88.64, -56.71 72.64, 4.73 in-in-in SNCiii in-in ActLoopNT-in 2.7833 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.01, 154.62 APE9-dihe-na 133.52, -155.05 APE8-dihe-in -117.36, 129.13 APE8-rot-in 302.02 APE67-dihe-in -56.32, -26.92 -42.89, -52.47 APE12-dist-in 8.2687 APE11-dist-in 11.8606 APE10-dist-in 6.2609 APE9-dist-in 4.1093 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.176 0.239 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3oxt AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3P0MA P17612 15 351 351.0 4SB:60351 Type1 Active DFGin 5.9227 14.5783 BLAminus -120.95, -179.03 59.8, 84.94 -96.45, 19.28 269.08, 54.31 -49.85, -35.86 in-in in 9.0006 Saltbr-in 2.6601 HRD-in -87.41, -52.38 71.61, 9.65 in-in-in SNCiii in-in ActLoopNT-in 2.9521 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.78, 160.64 APE9-dihe-na 131.62, -157.52 APE8-dihe-in -119.88, 133.57 APE8-rot-in 304.97 APE67-dihe-in -52.04, -26.97 -43.23, -57.05 APE12-dist-in 8.0193 APE11-dist-in 11.4768 APE10-dist-in 5.8873 APE9-dist-in 3.6581 None TPO198,SEP339 TPO198,SEP339 XRAY 2.03 0.171 0.205 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3p0m AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3POOA P17612 15 351 351.0 S69:62001 Type1 Active DFGin 5.6882 14.66 BLAminus -122.77, 177.28 59.44, 86.58 -95.62, 24.37 267.18, 52.33 -56.67, -28.22 in-in in 9.2255 Saltbr-in 2.6135 HRD-in -88.33, -52.91 73.26, 10.11 in-in-in SNCiii in-in ActLoopNT-in 2.9542 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.96, 158.93 APE9-dihe-na 133.77, -158.97 APE8-dihe-in -121.67, 134.24 APE8-rot-in 298.67 APE67-dihe-in -57.61, -22.88 -45.78, -52.79 APE12-dist-in 8.0956 APE11-dist-in 11.5265 APE10-dist-in 5.9381 APE9-dist-in 3.5559 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.187 0.212 A 351.0 333.0 0 25 25 0 [[44, 298]] 1.0 3poo AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3VQHA P17612 5 351 351.0 IQB:60401 Type1 Active DFGin 5.8868 14.5091 BLAminus -116.4, -175.47 66.0, 75.68 -94.16, 21.7 272.84, 60.82 -59.14, -31.37 in-in in 8.8982 Saltbr-in 2.6912 HRD-in -94.63, -51.76 70.89, 9.84 in-in-in SNCiii in-in ActLoopNT-in 2.8756 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.13, 162.63 APE9-dihe-na 132.63, -148.92 APE8-dihe-in -128.75, 132.36 APE8-rot-in 300.65 APE67-dihe-in -61.72, -25.75 -46.04, -48.59 APE12-dist-in 8.0578 APE11-dist-in 11.5232 APE10-dist-in 5.8417 APE9-dist-in 3.6408 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.95 0.192 0.234 A 351.0 347.0 0 25 25 0 [[44, 298]] 1.0 3vqh AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4UJ1A P17612 15 351 351.0 NVX:61351 Type1 Active DFGin 6.2416 14.5472 BLAminus -123.61, -163.8 61.68, 70.56 -93.64, 20.6 271.48, 60.79 -64.78, -20.97 in-in in 9.0378 Saltbr-in 2.5518 HRD-in -90.63, -51.42 73.4, 9.87 in-in-in SNCiii in-in ActLoopNT-in 2.9745 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.01, 158.56 APE9-dihe-na 139.11, -156.28 APE8-dihe-in -125.77, 137.11 APE8-rot-in 295.71 APE67-dihe-in -57.89, -23.24 -51.45, -49.94 APE12-dist-in 8.1202 APE11-dist-in 11.3926 APE10-dist-in 5.8666 APE9-dist-in 3.6245 None TPO198,SEP339 TPO198,SEP339 XRAY 1.768 0.168 0.201 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4uj1 AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4UJ2A P17612 15 351 351.0 NVV:61351 Type1 Active DFGin 6.3807 14.5704 BLAminus -125.67, -160.4 61.32, 58.86 -86.58, 22.47 272.1, 62.19 -53.53, -31.63 in-in in 9.0784 Saltbr-in 2.6406 HRD-in -86.14, -55.69 77.07, 9.76 in-in-in SNCiii in-in ActLoopNT-in 2.9495 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.59, 157.48 APE9-dihe-na 137.97, -154.25 APE8-dihe-in -126.65, 132.96 APE8-rot-in 298.62 APE67-dihe-in -53.02, -26.32 -44.15, -55.11 APE12-dist-in 8.245 APE11-dist-in 11.6516 APE10-dist-in 6.1174 APE9-dist-in 3.5607 None TPO198,SEP339 TPO198,SEP339 XRAY 2.019 0.165 0.209 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4uj2 AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4UJ9A P17612 11 351 351.0 S3N:61351 Type1 Active DFGin 6.1337 14.6501 BLAminus -117.52, -171.14 58.79, 71.43 -92.02, 19.19 269.08, 56.18 -56.86, -27.59 in-in in 8.9204 Saltbr-in 2.5062 HRD-in -93.86, -53.97 74.6, 12.42 in-in-in SNCiii in-in ActLoopNT-in 2.9172 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.92, 155.16 APE9-dihe-na 141.7, -146.62 APE8-dihe-in -127.44, 135.95 APE8-rot-in 296.91 APE67-dihe-in -56.69, -21.29 -47.92, -48.81 APE12-dist-in 7.952 APE11-dist-in 11.4276 APE10-dist-in 5.8483 APE9-dist-in 3.4787 None TPO198,SEP339 TPO198,SEP339 XRAY 1.87 0.167 0.206 A 351.0 341.0 0 25 25 0 [[44, 298]] 1.0 4uj9 AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4UJAA P17612 14 351 351.0 4L7:61351 Type1 Active DFGin 6.0974 14.6131 BLAminus -125.31, -163.62 62.94, 64.42 -88.89, 21.72 270.4, 58.9 -55.44, -30.93 in-in in 9.0487 Saltbr-in 2.7771 HRD-in -87.37, -51.28 70.71, 6.14 in-in-in SNCiii in-in ActLoopNT-in 2.9072 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.5, 162.38 APE9-dihe-na 130.88, -155.58 APE8-dihe-in -125.03, 133.85 APE8-rot-in 299.16 APE67-dihe-in -59.42, -24.42 -46.24, -50.45 APE12-dist-in 8.1686 APE11-dist-in 11.5131 APE10-dist-in 5.9673 APE9-dist-in 3.5887 None TPO198,SEP339 TPO198,SEP339 XRAY 1.93 0.166 0.206 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4uja AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4UJBA P17612 5 351 351.0 8BQ:61351 Type1 Active DFGin 5.9468 14.6677 BLAminus -125.29, -162.0 58.42, 69.71 -90.44, 19.28 267.91, 58.77 -53.57, -31.33 in-in in 9.135 Saltbr-in 2.7431 HRD-in -89.96, -52.14 72.96, 12.71 in-in-in SNCiii in-in ActLoopNT-in 2.9078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.56, 161.27 APE9-dihe-na 132.43, -159.75 APE8-dihe-in -122.62, 132.75 APE8-rot-in 302.43 APE67-dihe-in -59.14, -27.14 -46.68, -47.07 APE12-dist-in 8.1376 APE11-dist-in 11.4555 APE10-dist-in 5.9421 APE9-dist-in 3.6035 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.949 0.156 0.19 A 351.0 347.0 0 25 25 0 [[44, 298]] 1.0 4ujb AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5BX6A P17612 6 351 351.0 495:60401 Type1 Active DFGin 6.1832 14.3031 BLAminus -119.55, 164.86 70.92, 91.57 -100.18, 26.65 271.79, 52.76 -61.33, -23.25 in-in in 8.9062 Saltbr-in 2.708 HRD-in -93.87, -50.75 70.32, 10.63 in-in-in SNCiii in-in ActLoopNT-in 2.9595 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.15, 164.21 APE9-dihe-na 125.51, -162.2 APE8-dihe-in -117.48, 134.41 APE8-rot-in 303.65 APE67-dihe-in -56.37, -27.52 -46.12, -51.63 APE12-dist-in 8.0749 APE11-dist-in 11.4551 APE10-dist-in 5.918 APE9-dist-in 3.6014 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.89 0.172 0.218 A 351.0 346.0 0 25 25 0 [[44, 298]] 1.0 5bx6 AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5BX7A P17612 6 350 351.0 4W1:60401 Type1 Active DFGin 5.8928 14.2566 BLAminus -120.21, 170.97 66.4, 95.24 -104.96, 26.38 271.55, 55.44 -58.59, -27.02 in-in in 8.8868 Saltbr-in 2.6463 HRD-in -91.82, -48.84 66.55, 10.61 in-in-in SNCiii in-in ActLoopNT-in 2.9359 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.67, 162.65 APE9-dihe-na 129.46, -159.53 APE8-dihe-in -119.63, 133.68 APE8-rot-in 305.25 APE67-dihe-in -56.25, -25.43 -45.01, -52.75 APE12-dist-in 8.1102 APE11-dist-in 11.5179 APE10-dist-in 5.9614 APE9-dist-in 3.5807 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.89 0.178 0.226 A 351.0 345.0 0 25 25 0 [[44, 298]] 1.0 5bx7 AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5UZKA P17612 15 351 351.0 504:60401 Type1 Active DFGin 6.3811 13.9478 BLAminus -125.23, 159.32 70.49, 97.31 -104.94, 23.81 281.36, 67.83 -60.03, -27.16 in-in in 8.8803 Saltbr-in 2.7654 HRD-in -81.16, -49.29 61.5, 17.59 in-in-in SNCiii in-in ActLoopNT-in 2.9206 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.44, 160.74 APE9-dihe-na 127.01, -154.99 APE8-dihe-in -117.26, 132.5 APE8-rot-in 297.37 APE67-dihe-in -55.36, -26.76 -39.46, -56.34 APE12-dist-in 8.0111 APE11-dist-in 11.3938 APE10-dist-in 5.8297 APE9-dist-in 3.5881 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.191 0.253 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 5uzk AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6QJ7A P17612 14 351 351.0 J4B:60401 Type1 Active DFGin 6.3708 14.8786 BLAminus -117.39, 169.65 69.58, 85.56 -98.1, 21.35 272.03, 58.03 -54.77, -30.7 in-in in 9.2139 Saltbr-in 2.7504 HRD-in -87.29, -50.94 66.9, 9.43 in-in-in SNCiii in-in ActLoopNT-in 2.94 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.01, 157.32 APE9-dihe-na 126.55, -163.63 APE8-dihe-in -112.81, 131.54 APE8-rot-in 300.45 APE67-dihe-in -57.75, -27.43 -43.16, -51.25 APE12-dist-in 8.0042 APE11-dist-in 11.5059 APE10-dist-in 5.846 APE9-dist-in 3.703 None TPO198,SEP339 TPO198,SEP339 XRAY 1.69 0.179 0.214 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 6qj7 AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3MVJA P17612 16 351 351.0 XFE:60351 Type1 Active DFGin 6.1884 13.5821 BLAminus -115.88, 169.36 72.34, 84.05 -100.4, 21.07 284.54, 72.78 -48.33, -32.34 in-in in 8.6933 Saltbr-in 2.9429 HRD-in -94.45, -57.98 81.77, 7.12 in-in-in SNCiii in-in ActLoopNT-in 3.0047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.5, 165.11 APE9-dihe-na 130.23, -153.23 APE8-dihe-in -130.91, 127.14 APE8-rot-in 305.92 APE67-dihe-in -54.4, -32.7 -46.27, -53.24 APE12-dist-in 8.1645 APE11-dist-in 11.4405 APE10-dist-in 5.835 APE9-dist-in 3.6782 None TPO198,SEP339 TPO198,SEP339 XRAY 2.49 0.217 0.304 A 371.0 336.0 0 25 25 0 [[44, 298]] 1.0 3mvj AGC_PRKACA_HUMAN AGC 5.4e-95 323.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3MVJE P17612 16 351 351.0 XFE:60351 Type1 Active DFGin 6.0097 13.9041 BLAminus -120.77, 173.49 75.79, 91.53 -105.05, 22.03 286.9, 73.04 -48.68, -45.44 in-in in 8.7857 Saltbr-in 2.5037 HRD-in -85.62, -59.75 66.22, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.9875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.99, 156.89 APE9-dihe-na 143.78, -161.15 APE8-dihe-in -124.44, 132.79 APE8-rot-in 305.29 APE67-dihe-in -69.91, -25.33 -54.9, -34.25 APE12-dist-in 8.1481 APE11-dist-in 11.447 APE10-dist-in 5.8027 APE9-dist-in 3.8015 None TPO198,SEP339 TPO198,SEP339 XRAY 2.49 0.217 0.304 E 371.0 336.0 0 25 25 0 [[44, 298]] 1.0 3mvj AGC_PRKACA_HUMAN AGC 5.4e-95 323.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3L9MA P17612 12 351 351.0 L9M:60351 Type1 Active DFGin 6.7018 13.6799 BLAminus -123.42, 168.26 64.27, 97.86 -112.03, 32.77 297.13, 76.75 -74.15, -5.52 in-in in 9.0347 Saltbr-in 2.7926 HRD-in -71.88, -60.17 71.32, 14.02 in-in-in SNCiii in-in ActLoopNT-in 2.8886 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.62, 165.36 APE9-dihe-na 118.63, -161.51 APE8-dihe-in -116.7, 125.6 APE8-rot-in 304.73 APE67-dihe-in -59.86, -22.26 -32.71, -59.17 APE12-dist-in 8.1871 APE11-dist-in 11.2087 APE10-dist-in 5.6173 APE9-dist-in 3.5714 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.223 0.27 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 3l9m AGC_PRKACA_HUMAN AGC 5.8e-95 323.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3L9MB P17612 14 351 351.0 L9M:60351 Type1 Active DFGin 6.7673 13.7383 BLAminus -124.39, 166.06 67.02, 98.19 -111.82, 31.79 294.5, 74.52 -67.48, -11.73 in-in in 8.8779 Saltbr-in 2.9129 HRD-in -76.18, -53.82 65.92, 13.75 in-in-in SNCiii in-in ActLoopNT-in 2.9242 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.4, 166.8 APE9-dihe-na 115.45, -164.35 APE8-dihe-in -115.85, 130.97 APE8-rot-in 297.34 APE67-dihe-in -54.51, -26.46 -29.85, -67.98 APE12-dist-in 8.2238 APE11-dist-in 11.2629 APE10-dist-in 5.6584 APE9-dist-in 3.5585 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.223 0.27 B 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 3l9m AGC_PRKACA_HUMAN AGC 5.8e-95 323.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3L9NA P17612 15 351 351.0 L9N:60351 Type1 Active DFGin 6.4227 13.4597 BLAminus -123.73, 167.95 65.98, 97.53 -115.01, 25.76 300.78, 81.96 -66.98, -19.82 in-in in 9.0504 Saltbr-in 2.7445 HRD-in -67.38, -52.97 66.43, 17.24 in-in-in SNCiii in-in ActLoopNT-in 2.9582 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.06, 165.76 APE9-dihe-na 122.47, -160.51 APE8-dihe-in -116.6, 130.05 APE8-rot-in 304.11 APE67-dihe-in -53.81, -24.08 -30.84, -70.07 APE12-dist-in 8.1973 APE11-dist-in 11.3941 APE10-dist-in 5.9345 APE9-dist-in 3.5534 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.217 0.257 A 351.0 334.0 0 25 25 0 [[44, 298]] 1.0 3l9n AGC_PRKACA_HUMAN AGC 5.8e-95 323.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8FE2A P17612 4 351 351.0 XTI:60501 Type1 Active DFGin 6.1423 13.9131 BLAminus -123.85, 174.03 69.38, 86.41 -105.22, 28.0 281.98, 71.1 -68.62, -14.04 in-in in 8.8535 Saltbr-in 2.5144 HRD-in -84.66, -51.16 67.93, 20.04 in-in-in SNCiii in-in ActLoopNT-in 2.7913 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.46, 164.95 APE9-dihe-na 122.51, -154.32 APE8-dihe-in -114.26, 125.71 APE8-rot-in 301.9 APE67-dihe-in -53.15, -32.01 -48.08, -46.83 APE12-dist-in 8.3148 APE11-dist-in 11.573 APE10-dist-in 6.0032 APE9-dist-in 3.9389 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.34 0.199 0.251 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fe2 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8FE2B P17612 4 351 351.0 XTI:60501 Type1 Active DFGin 6.2269 13.875 BLAminus -121.06, -174.83 58.15, 84.69 -101.22, 28.39 282.36, 54.58 -64.33, -23.67 in-in in 8.8613 Saltbr-in 2.9356 HRD-in -86.41, -49.46 70.11, 7.42 in-in-in SNCiii in-in ActLoopNT-in 2.9286 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.54, 160.4 APE9-dihe-na 134.47, -156.72 APE8-dihe-in -118.93, 133.24 APE8-rot-in 292.47 APE67-dihe-in -59.44, -24.84 -53.68, -43.95 APE12-dist-in 8.1124 APE11-dist-in 11.5096 APE10-dist-in 5.8745 APE9-dist-in 3.7916 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.34 0.199 0.251 B 405.0 333.0 0 25 25 0 [[44, 298]] 1.0 8fe2 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8FE5A P17612 3 351 351.0 XTT:60501 Type1 Active DFGin 6.5996 14.2711 BLAminus -118.08, 163.41 75.28, 94.71 -111.66, 23.11 283.47, 69.64 -61.06, -23.26 in-in in 8.6685 Saltbr-in 2.7938 HRD-in -90.95, -53.69 70.13, 22.37 in-in-in SNCiii in-in ActLoopNT-in 2.8938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.31, 157.71 APE9-dihe-na 120.85, -158.74 APE8-dihe-in -109.76, 129.18 APE8-rot-in 307.33 APE67-dihe-in -52.63, -34.99 -47.86, -48.55 APE12-dist-in 8.4091 APE11-dist-in 11.5401 APE10-dist-in 5.9179 APE9-dist-in 3.8815 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.51 0.193 0.243 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fe5 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8FE5B P17612 4 351 351.0 XTT:60501 Type1 Active DFGin 6.5852 14.1601 BLAminus -125.03, 171.21 68.33, 95.08 -111.16, 25.84 279.92, 72.93 -61.92, -29.97 in-in in 8.6935 Saltbr-in 2.6551 HRD-in -80.97, -54.69 77.96, 3.27 in-in-in SNCiii in-in ActLoopNT-in 2.9235 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.98, 153.65 APE9-dihe-na 132.84, -165.24 APE8-dihe-in -101.75, 136.64 APE8-rot-in 293.15 APE67-dihe-in -60.99, -28.63 -57.01, -42.49 APE12-dist-in 8.3434 APE11-dist-in 11.6658 APE10-dist-in 6.0763 APE9-dist-in 3.8646 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.51 0.193 0.243 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fe5 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8FECA P17612 3 351 351.0 XU0:60501 Type1 Active DFGin 5.927 14.4607 BLAminus -126.38, -179.91 61.84, 90.42 -102.64, 31.23 279.77, 62.7 -61.22, -32.63 in-in in 9.1545 Saltbr-in 3.1068 HRD-in -85.43, -52.43 73.91, 14.55 in-in-in SNCiii in-in ActLoopNT-in 2.8343 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.02, 165.29 APE9-dihe-na 137.47, -140.99 APE8-dihe-in -132.86, 123.05 APE8-rot-in 312.11 APE67-dihe-in -60.14, -32.0 -40.12, -49.13 APE12-dist-in 8.2325 APE11-dist-in 11.5617 APE10-dist-in 5.9552 APE9-dist-in 3.6059 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.7 0.214 0.287 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fec AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8FECB P17612 3 351 351.0 XU0:60501 Type1 Active DFGin 5.9754 14.6835 BLAminus -127.65, 171.34 68.29, 92.72 -102.21, 27.6 281.7, 67.04 -60.34, -31.82 in-in in 8.8397 Saltbr-in 2.809 HRD-in -91.52, -53.88 75.61, 9.83 in-in-in SNCiii in-in ActLoopNT-in 2.9418 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.24, 178.4 APE9-dihe-na 115.87, -151.85 APE8-dihe-in -128.69, 124.59 APE8-rot-in 281.12 APE67-dihe-in -60.64, -38.43 -38.43, -52.12 APE12-dist-in 8.1803 APE11-dist-in 11.3776 APE10-dist-in 5.7925 APE9-dist-in 3.4601 None TPO198,SEP339 TPO198,SEP339 XRAY 2.7 0.214 0.287 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fec AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 2GU8A P17612 15 351 351.0 796:61001 Type1 Active DFGin 6.6297 14.3669 BLAminus -112.13, 169.56 64.55, 88.46 -98.67, 24.98 279.28, 59.9 -52.79, -25.6 in-in in 8.9692 Saltbr-in 3.0305 HRD-in -83.27, -51.67 71.2, 9.61 in-in-in SNCiii in-in ActLoopNT-in 2.9056 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.43, 156.76 APE9-dihe-na 146.07, -145.55 APE8-dihe-in -129.46, 134.31 APE8-rot-in 294.43 APE67-dihe-in -57.08, -22.75 -50.07, -49.98 APE12-dist-in 8.0405 APE11-dist-in 11.4687 APE10-dist-in 5.9773 APE9-dist-in 3.5072 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.203 0.261 A 337.0 337.0 0 25 25 0 [[44, 298]] 1.0 2gu8 AGC_PRKACA_HUMAN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5N23A P17612 9 351 351.0 35R:60401 Type1 Active DFGin 5.4212 13.8637 BLAminus -109.83, 165.02 72.7, 94.27 -97.78, 24.01 286.85, 71.32 -58.73, -25.18 in-in in 9.4998 Saltbr-in 2.9266 HRD-in -90.99, -49.74 71.93, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.8779 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.89, 153.96 APE9-dihe-na 137.51, -163.29 APE8-dihe-in -116.51, 133.79 APE8-rot-in 303.7 APE67-dihe-in -56.98, -24.74 -46.64, -52.33 APE12-dist-in 8.0559 APE11-dist-in 11.5849 APE10-dist-in 5.9451 APE9-dist-in 3.6536 K48R,L96Q,M121L,V124A,Q182K,T184A SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.088 0.192 0.239 A 352.0 337.0 0 25 25 0 [[44, 298]] 1.0 5n23 AGC_PRKACA_HUMAN AGC 5.3e-93 316.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3AMAA P17612 2 351 351.0 SKE:60351 Type1 Active DFGin 5.0968 14.0258 BLAminus -113.5, 162.11 72.12, 95.43 -101.12, 20.61 280.01, 66.12 -51.23, -34.47 in-in in 9.396 Saltbr-in 2.7343 HRD-in -88.12, -51.56 68.22, 12.75 in-in-in SNCiii in-in ActLoopNT-in 2.9104 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.04, 164.64 APE9-dihe-na 124.94, -160.1 APE8-dihe-in -123.9, 133.09 APE8-rot-in 298.24 APE67-dihe-in -57.85, -22.29 -46.67, -50.91 APE12-dist-in 8.1018 APE11-dist-in 11.5706 APE10-dist-in 5.9018 APE9-dist-in 3.5818 K48R,L96Q,M121L,V124A,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.75 0.198 0.223 A 351.0 345.0 0 25 25 0 [[44, 298]] 1.0 3ama AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6FRXA P17612 13 351 351.0 E3Z:60401 Type1 Active DFGin 5.2761 14.2424 BLAminus -103.8, 165.76 62.73, 100.4 -98.82, 30.34 278.36, 58.69 -63.79, -25.19 in-in in 9.3071 Saltbr-in 2.6351 HRD-in -83.02, -52.27 73.43, 9.25 in-in-in SNCiii in-in ActLoopNT-in 2.866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.05, 168.13 APE9-dihe-na 109.0, -164.56 APE8-dihe-in -112.4, 132.82 APE8-rot-in 302.54 APE67-dihe-in -55.48, -26.17 -48.65, -50.5 APE12-dist-in 8.3241 APE11-dist-in 11.7113 APE10-dist-in 6.1183 APE9-dist-in 3.716 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.88 0.191 0.226 A 351.0 334.0 0 25 25 0 [[44, 298]] 1.0 6frx AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4AE6A P17612 13 351 351.0 No_ligand No_ligand Inactive DFGin 6.5333 15.789 ABAminus -102.0, -12.32 -149.9, 117.63 -105.31, 23.09 271.72, 75.39 -56.8, -39.15 out-in out 10.0651 Saltbr-in 3.037 HRD-in -80.45, -57.48 71.85, 11.08 in-in-out SNCiio in-out ActLoopNT-in 2.8103 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.83, 165.09 APE9-dihe-na 109.71, 150.17 APE8-dihe-in -70.25, 136.52 APE8-rot-out 76.9 APE67-dihe-in -62.21, -26.49 -48.12, -39.36 APE12-dist-in 8.4839 APE11-dist-in 11.6198 APE10-dist-in 6.1388 APE9-dist-in 4.2493 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.219 0.283 A 343.0 321.0 0 25 25 0 [[44, 298]] 1.0 4ae6 AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4AE6B P17612 17 351 351.0 No_ligand No_ligand Inactive DFGin 6.7262 16.2285 ABAminus -110.11, -21.15 -129.5, 123.25 -122.94, 15.22 289.43, 78.48 -49.18, -40.14 out-out out 10.4783 Saltbr-out 4.4043 HRD-in -72.54, -54.34 51.9, 34.46 out-in-out SNCoio in-out ActLoopNT-in 2.6982 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -140.57, 163.72 APE9-dihe-na 111.27, 158.24 APE8-dihe-in -83.25, 146.52 APE8-rot-out 46.71 APE67-dihe-in -47.41, -26.35 -55.51, -46.4 APE12-dist-in 8.738 APE11-dist-in 11.4408 APE10-dist-in 5.9066 APE9-dist-in 4.36 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.219 0.283 B 343.0 323.0 0 25 25 0 [[44, 298]] 1.0 4ae6 AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4AE9A P17612 13 351 351.0 No_ligand No_ligand Inactive DFGin 6.55 16.001 ABAminus -108.08, 1.25 -143.04, 135.02 -120.31, 26.17 277.62, 67.12 -50.31, -36.29 out-out out 10.2017 Saltbr-out 4.9285 HRD-in -78.87, -60.3 78.37, 10.3 out-in-in SNCoii in-in ActLoopNT-in 2.7466 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.01, 163.39 APE9-dihe-na 112.23, 171.54 APE8-dihe-in -84.52, 127.75 APE8-rot-in 289.6 APE67-dihe-in -56.88, -27.79 -43.6, -44.81 APE12-dist-in 8.2704 APE11-dist-in 11.576 APE10-dist-in 6.0269 APE9-dist-in 4.1577 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.201 0.264 A 343.0 324.0 0 25 25 0 [[44, 298]] 1.0 4ae9 AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 4AE9B P17612 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.7487 16.1613 ABAminus -114.92, -7.43 -130.92, 125.97 -130.48, 16.95 295.44, 81.38 -52.61, -39.79 out-out out 10.6681 Saltbr-out 4.4397 HRD-in -74.27, -49.34 44.92, 35.44 out-in-out SNCoio in-out ActLoopNT-in 2.6317 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -139.93, 157.79 APE9-dihe-na 109.15, 156.62 APE8-dihe-in -68.62, 140.66 APE8-rot-out 10.98 APE67-dihe-in -51.62, -27.57 -42.37, -51.96 APE12-dist-in 8.5473 APE11-dist-in 11.4951 APE10-dist-in 5.9265 APE9-dist-in 4.357 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.201 0.264 B 343.0 324.0 0 25 25 0 [[44, 298]] 1.0 4ae9 AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 7Y1GB P17612 15 351 351.0 I5G:60401 Type1 Inactive DFGin 6.5019 15.3725 ABAminus -112.68, -38.34 -99.79, 125.89 -136.28, 17.99 282.52, 84.22 -66.37, -34.78 in-in in 9.4501 Saltbr-in 2.8689 HRD-in -80.77, -61.43 56.8, 33.17 in-in-out SNCiio in-out ActLoopNT-in 2.95 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.12, 157.52 APE9-dihe-na 119.76, 163.27 APE8-dihe-in -78.91, 145.18 APE8-rot-out 49.01 APE67-dihe-in -67.8, -20.12 -41.99, -42.68 APE12-dist-in 8.186 APE11-dist-in 11.3096 APE10-dist-in 5.7517 APE9-dist-in 4.3013 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.188 0.237 B 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 7y1g AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 9DC6A P17612 16 351 351.0 A1A3I:60501 Type1 Inactive DFGin 5.8215 14.3818 ABAminus -129.15, -5.99 -129.24, 116.18 -111.87, 19.13 279.15, 62.12 -54.37, -20.22 in-in in 9.1087 Saltbr-in 3.3088 HRD-in -90.78, -41.18 70.14, 8.35 in-in-in SNCiii in-in ActLoopNT-in 2.8945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.59, -177.06 APE9-dihe-na 91.67, -156.82 APE8-dihe-in -118.5, 121.2 APE8-rot-in 293.95 APE67-dihe-in -55.19, -30.52 -37.8, -52.71 APE12-dist-in 8.2373 APE11-dist-in 11.5075 APE10-dist-in 6.1047 APE9-dist-in 3.6545 None SEP140,TPO198 SEP140,TPO198 XRAY 2.7 0.237 0.311 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 9dc6 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 9DC6B P17612 16 351 351.0 A1A3I:60501 Type1 Inactive DFGin 6.1262 14.2237 ABAminus -118.96, -25.57 -111.81, 119.46 -118.82, 27.48 291.58, 78.19 -62.06, -32.01 in-in in 8.9675 Saltbr-in 2.88 HRD-in -75.88, -55.9 87.72, 2.66 in-in-in SNCiii in-in ActLoopNT-in 2.8974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.71, 171.27 APE9-dihe-na 114.33, -156.38 APE8-dihe-in -127.33, 134.71 APE8-rot-in 292.26 APE67-dihe-in -63.06, -23.33 -44.45, -51.67 APE12-dist-in 8.5329 APE11-dist-in 11.6121 APE10-dist-in 6.0734 APE9-dist-in 3.5437 None SEP140,TPO198 SEP140,TPO198 XRAY 2.7 0.237 0.311 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 9dc6 AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3AMBA P17612 4 351 351.0 VX6:60351 Type1 Inactive DFGin 5.087 14.2922 ABAminus -95.17, -47.0 -99.94, 115.14 -101.01, 17.86 279.8, 67.75 -53.93, -36.65 in-in in 9.4162 Saltbr-in 2.7867 HRD-in -85.39, -50.26 66.81, 7.13 in-in-in SNCiii in-in ActLoopNT-in 2.8909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.26, 159.46 APE9-dihe-na 131.88, -164.87 APE8-dihe-in -118.92, 127.93 APE8-rot-in 300.49 APE67-dihe-in -60.18, -24.15 -37.91, -53.92 APE12-dist-in 8.1946 APE11-dist-in 11.5803 APE10-dist-in 6.013 APE9-dist-in 3.6414 K48R,L96Q,M121L,V124A,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.25 0.214 0.256 A 351.0 343.0 0 25 25 0 [[44, 298]] 1.0 3amb AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8X5LA P17612 17 351 351.0 RKD:401 Type1 Inactive DFGin 4.1037 12.291 ABAminus -92.81, -18.04 -108.82, 165.79 -131.86, 13.05 303.97, 96.56 69.26, -154.62 in-out in 9.9587 Saltbr-out 4.1566 HRD-in -67.69, -44.07 75.82, -80.8 out-out-out SNCooo out-out ActLoopNT-out 7.1481 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iooo APE10-dihe-na -77.04, -32.9 APE9-dihe-na -87.77, -44.9 APE8-dihe-in -124.02, 60.68 APE8-rot-out 58.39 APE67-dihe-in -63.73, -18.25 -72.69, -25.11 APE12-dist-in 12.2601 APE11-dist-out 15.7603 APE10-dist-out 19.6162 APE9-dist-out 13.5896 None SEP339 SEP339 XRAY 2.75 0.204 0.255 A 352.0 331.0 4 25 21 4 [[44, 298]] 1.0 8x5l AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 8X5LB P17612 17 334 351.0 RKD:401 Type1 Inactive DFGin 4.0878 12.4831 ABAminus -93.45, -16.52 -108.91, 166.44 -130.77, 10.4 300.78, 83.16 68.88, -158.2 out-out out 10.6724 Saltbr-out 4.4614 HRD-in -67.44, -44.97 74.27, -77.51 out-out-out SNCooo out-out ActLoopNT-out 7.1674 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iioo APE10-dihe-na -62.33, 89.14 APE9-dihe-na -96.13, -167.24 APE8-dihe-in -45.35, 129.26 APE8-rot-out 58.75 APE67-dihe-in -60.15, -17.0 -69.42, -27.93 APE12-dist-in 9.2928 APE11-dist-in 11.2327 APE10-dist-out 15.0507 APE9-dist-out 8.3319 None SEP339 SEP339 XRAY 2.75 0.204 0.255 B 352.0 306.0 5 25 20 5 [[44, 298]] 1.0 8x5l AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6NO7E P17612 13 351 351.0 ATP:60403 ATPlike Inactive DFGin 6.9335 14.1655 BLAminus -118.71, 175.9 64.55, 75.01 -86.85, 19.7 273.68, 51.02 -43.49, -41.12 in-out in 9.4189 Saltbr-out 5.4559 HRD-in -91.66, -53.62 73.72, 11.47 out-in-in SNCoii in-in ActLoopNT-in 3.1639 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.9, 150.23 APE9-dihe-na 149.21, -142.3 APE8-dihe-in -132.1, 131.95 APE8-rot-in 297.19 APE67-dihe-in -64.62, -25.64 -37.25, -53.79 APE12-dist-in 8.0557 APE11-dist-in 10.9843 APE10-dist-in 5.7482 APE9-dist-in 3.2156 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 E 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 6no7 AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6NO7G P17612 15 351 351.0 ATP:60403 ATPlike Inactive DFGin 6.0359 14.0844 BLAminus -118.68, 176.55 65.34, 76.32 -85.78, 18.75 273.72, 51.07 -44.34, -41.82 in-out in 9.7125 Saltbr-out 5.2149 HRD-in -91.95, -53.38 74.11, 11.57 out-in-in SNCoii in-in ActLoopNT-in 3.3017 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.42, 149.81 APE9-dihe-na 148.91, -142.4 APE8-dihe-in -132.18, 131.68 APE8-rot-in 297.12 APE67-dihe-in -64.98, -25.0 -37.42, -54.32 APE12-dist-in 7.6679 APE11-dist-in 10.658 APE10-dist-in 5.5534 APE9-dist-in 3.4096 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 G 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 6no7 AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 9EDDA P17612 14 351 351.0 ATP:60400 ATPlike Inactive DFGin 7.6417 15.4797 BLAminus -131.38, -176.44 56.47, 73.0 -86.17, 32.62 269.53, 53.11 -62.17, -29.29 in-out in 9.6174 Saltbr-out 3.9466 HRD-in -100.83, -51.39 64.03, -2.2 out-out-out SNCooo out-out ActLoopNT-out 3.7028 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -126.87, 141.16 APE9-dihe-na 150.41, -172.01 APE8-dihe-in -103.27, 147.74 APE8-rot-out 185.24 APE67-dihe-in -92.0, 3.92 -57.96, -27.57 APE12-dist-in 8.1647 APE11-dist-in 11.2754 APE10-dist-in 5.6275 APE9-dist-in 4.2273 None TPO198,SEP339 TPO198,SEP339 EM 6.3 999.0 999.0 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9edd AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 9EDEA P17612 14 351 351.0 ATP:60400 ATPlike Inactive DFGin 6.6922 15.188 BLAminus -131.57, -176.8 59.06, 65.59 -87.14, 28.49 267.05, 50.71 -66.29, -36.64 in-out in 9.9219 Saltbr-out 4.6819 HRD-in -115.21, -49.18 64.38, 4.15 out-out-out SNCooo out-out ActLoopNT-out 3.632 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.67, 141.1 APE9-dihe-na 158.89, -177.66 APE8-dihe-in -75.58, 154.98 APE8-rot-out 190.35 APE67-dihe-in -109.16, -25.21 -65.33, -8.36 APE12-dist-in 8.3471 APE11-dist-in 11.7825 APE10-dist-in 6.8289 APE9-dist-in 4.9175 None TPO198,SEP339 TPO198,SEP339 EM 5.9 999.0 999.0 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9ede AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5IZJA P17612 15 351 351.0 6J9:60414 Allosteric Inactive DFGin 6.0059 14.882 BLAminus -111.62, 172.78 70.98, 87.77 -97.8, 27.11 278.83, 80.41 -58.58, -30.48 in-out in 9.9394 Saltbr-out 4.1818 HRD-in -81.12, -50.89 44.27, 35.23 out-in-out SNCoio in-out ActLoopNT-in 2.9865 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -140.79, 157.34 APE9-dihe-na 106.02, 164.59 APE8-dihe-in -74.04, 136.38 APE8-rot-out 204.5 APE67-dihe-in -57.37, -26.41 -46.69, -44.98 APE12-dist-in 8.2021 APE11-dist-in 11.523 APE10-dist-in 5.7985 APE9-dist-in 4.2246 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.199 0.226 A 351.0 330.0 0 25 25 0 [[44, 298]] 1.0 5izj AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 5IZJB P17612 15 351 351.0 6J9:60413 Allosteric Inactive DFGin 6.2012 15.2736 BLAminus -109.02, 168.97 75.33, 87.97 -97.67, 24.22 269.13, 57.46 -63.02, -24.98 out-out out 10.2894 Saltbr-out 4.5426 HRD-in -78.48, -51.65 67.16, 12.35 out-in-out SNCoio in-out ActLoopNT-in 2.9093 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.15, 157.15 APE9-dihe-na 105.13, 166.26 APE8-dihe-in -75.85, 137.43 APE8-rot-out 200.52 APE67-dihe-in -61.79, -25.86 -47.32, -41.18 APE12-dist-in 8.2568 APE11-dist-in 11.4828 APE10-dist-in 5.8129 APE9-dist-in 4.0688 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.199 0.226 B 351.0 327.0 0 25 25 0 [[44, 298]] 1.0 5izj AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6BYSA P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.6445 12.8448 BLAminus 176.97, -168.6 35.04, 63.97 -77.13, -0.55 257.78, 43.58 -51.31, -30.32 in-out in 8.4132 Saltbr-out 3.6943 HRD-out -132.08, 139.02 -123.89, -19.92 out-in-in SNCoii in-in ActLoopNT-in 3.1045 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -174.55, -174.54 APE9-dihe-na 119.07, -153.65 APE8-dihe-in -123.63, 121.24 APE8-rot-in 279.88 APE67-dihe-in -80.36, -3.37 -55.82, -41.73 APE12-dist-in 8.6369 APE11-dist-in 11.0634 APE10-dist-in 6.1456 APE9-dist-in 3.4911 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6BYSC P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.5999 13.0168 BLAminus 177.41, -169.47 35.75, 66.26 -79.08, -7.92 257.89, 46.49 -37.01, -39.99 in-out in 8.4312 Saltbr-out 3.6308 HRD-out -132.47, 138.88 -123.68, -21.42 out-in-in SNCoii in-in ActLoopNT-in 3.129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.21, -176.06 APE9-dihe-na 122.36, -150.78 APE8-dihe-in -124.74, 121.46 APE8-rot-in 280.04 APE67-dihe-in -74.72, -2.75 -56.12, -45.35 APE12-dist-in 8.6212 APE11-dist-in 11.0301 APE10-dist-in 6.1698 APE9-dist-in 3.5547 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 C 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6BYSE P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.5995 12.7783 BLAminus 177.63, -170.33 35.66, 68.12 -82.89, -7.7 254.73, 43.9 -34.72, -39.61 in-in in 8.3947 Saltbr-in 3.5304 HRD-out -134.25, 137.62 -124.05, -19.61 in-in-in SNCiii in-in ActLoopNT-in 3.1341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -175.91, -174.99 APE9-dihe-na 120.1, -152.87 APE8-dihe-in -123.78, 120.18 APE8-rot-in 279.49 APE67-dihe-in -74.6, -2.18 -55.44, -46.05 APE12-dist-in 8.5261 APE11-dist-in 11.0087 APE10-dist-in 6.1584 APE9-dist-in 3.4923 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 E 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6BYSG P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.5502 12.8795 BLAminus 177.64, -169.59 35.17, 69.18 -84.06, -7.89 253.42, 50.51 -34.53, -40.01 in-out in 8.4064 Saltbr-out 3.6038 HRD-out -131.78, 137.89 -122.99, -20.45 out-in-in SNCoii in-in ActLoopNT-in 3.091 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -174.78, -177.53 APE9-dihe-na 124.08, -149.25 APE8-dihe-in -124.03, 121.23 APE8-rot-in 280.42 APE67-dihe-in -73.41, -1.98 -56.98, -46.28 APE12-dist-in 8.6175 APE11-dist-in 11.0767 APE10-dist-in 6.1508 APE9-dist-in 3.5427 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 G 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6NO7A P17612 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.5833 14.5513 BLAminus -119.16, 176.65 65.47, 76.79 -85.63, 19.52 273.14, 48.34 -44.12, -41.29 in-out in 9.256 Saltbr-out 3.8369 HRD-in -93.59, -54.13 73.95, 11.29 out-in-in SNCoii in-in ActLoopNT-in 3.0846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.66, 149.89 APE9-dihe-na 148.72, -142.64 APE8-dihe-in -132.35, 131.6 APE8-rot-in 297.3 APE67-dihe-in -65.08, -25.39 -37.56, -54.33 APE12-dist-in 7.8572 APE11-dist-in 10.7351 APE10-dist-in 5.368 APE9-dist-in 3.3109 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 6no7 AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 3MVJB P17612 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.6749 15.0725 BLAminus -107.29, 175.17 69.85, 103.13 -126.62, 31.7 289.12, 86.96 -68.94, -36.62 in-out in 9.8619 Saltbr-out 5.1808 HRD-in -72.7, -45.04 65.83, 8.62 out-in-in SNCoii in-in ActLoopNT-in 2.6815 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.22, 164.94 APE9-dihe-na 113.67, -166.87 APE8-dihe-in -95.86, 130.98 APE8-rot-in 290.81 APE67-dihe-in -63.62, -17.9 -44.08, -47.61 APE12-dist-in 8.4504 APE11-dist-in 11.5319 APE10-dist-in 6.2728 APE9-dist-in 4.219 None TPO198,SEP339 TPO198,SEP339 XRAY 2.49 0.217 0.304 B 371.0 322.0 0 25 25 0 [[44, 298]] 1.0 3mvj AGC_PRKACA_HUMAN AGC 5.4e-95 323.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6WJFA P17612 2 351 351.0 No_ligand No_ligand Inactive DFGin 9.9992 13.4832 BLAminus -126.44, 169.73 60.01, 89.86 -112.86, 1.12 296.86, 95.65 -61.53, -29.79 out-out out 10.0908 Saltbr-out 7.2346 HRD-in -67.55, -42.01 64.88, -66.83 out-out-out SNCooo out-out ActLoopNT-out 3.6866 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -171.91, 116.67 APE9-dihe-na 154.02, -66.34 APE8-dihe-in -113.18, 77.77 APE8-rot-out 47.03 APE67-dihe-in -82.77, -55.57 -68.63, -38.53 APE12-dist-in 8.4814 APE11-dist-in 12.0403 APE10-dist-in 7.8146 APE9-dist-in 4.4462 None None None EM 7.5 999.0 999.0 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 6wjf AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6WJFB P17612 42 351 351.0 No_ligand No_ligand Inactive DFGin 10.0534 15.2293 BLAminus -124.34, 176.36 59.38, 90.58 -123.09, 12.38 277.22, 94.34 -61.71, -29.6 out-out out 11.687 Saltbr-out 6.4309 HRD-out -65.49, -35.93 66.74, -107.09 out-out-out SNCooo out-out ActLoopNT-out 3.9609 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiio APE10-dihe-na -163.85, -158.9 APE9-dihe-na 100.21, -130.3 APE8-dihe-in -150.47, 147.99 APE8-rot-out 180.18 APE67-dihe-in -80.92, 5.22 -58.41, -26.93 APE12-dist-in 8.6814 APE11-dist-in 11.7662 APE10-dist-in 6.7949 APE9-dist-out 6.2996 None None None EM 7.5 999.0 999.0 B 405.0 310.0 27 25 25 0 [[44, 298]] 1.0 6wjf AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6WJGA P17612 42 351 351.0 No_ligand No_ligand Inactive DFGin 9.9992 13.4832 BLAminus -126.44, 169.73 60.01, 89.86 -112.86, 1.12 296.86, 95.65 -61.53, -29.79 out-out out 10.0908 Saltbr-out 7.2346 HRD-in -67.55, -42.01 64.88, -66.83 out-out-out SNCooo out-out ActLoopNT-out 3.6866 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -171.91, 116.67 APE9-dihe-na 154.02, -66.34 APE8-dihe-in -113.18, 77.77 APE8-rot-out 47.03 APE67-dihe-in -82.77, -55.57 -68.63, -38.53 APE12-dist-in 8.4814 APE11-dist-in 12.0403 APE10-dist-in 7.8146 APE9-dist-in 4.4462 None None None EM 6.2 999.0 999.0 A 405.0 310.0 27 25 25 0 [[44, 298]] 1.0 6wjg AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6WJGB P17612 42 351 351.0 No_ligand No_ligand Inactive DFGin 10.0534 15.2293 BLAminus -124.34, 176.36 59.38, 90.58 -123.09, 12.38 277.22, 94.34 -61.71, -29.6 out-out out 11.687 Saltbr-out 6.4309 HRD-out -65.49, -35.93 66.74, -107.09 out-out-out SNCooo out-out ActLoopNT-out 3.9609 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiio APE10-dihe-na -163.85, -158.9 APE9-dihe-na 100.21, -130.3 APE8-dihe-in -150.47, 147.99 APE8-rot-out 180.18 APE67-dihe-in -80.92, 5.22 -58.41, -26.93 APE12-dist-in 8.6814 APE11-dist-in 11.7662 APE10-dist-in 6.7949 APE9-dist-out 6.2996 None None None EM 6.2 999.0 999.0 B 405.0 310.0 27 25 25 0 [[44, 298]] 1.0 6wjg AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 7Y1GA P17612 16 351 351.0 I5G:60500 Type1 Inactive DFGin 6.3413 14.8624 BLAminus -118.48, 174.7 76.77, 103.0 -130.63, 13.32 288.1, 82.33 -55.62, -41.63 in-in in 9.1119 Saltbr-in 2.716 HRD-in -77.78, -56.16 48.65, 33.18 in-in-out SNCiio in-out ActLoopNT-in 2.8984 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -128.96, 160.38 APE9-dihe-na 112.98, 149.31 APE8-dihe-in -54.34, 136.89 APE8-rot-out 199.98 APE67-dihe-in -67.35, -18.71 -49.9, -39.67 APE12-dist-in 8.1184 APE11-dist-in 11.271 APE10-dist-in 5.6336 APE9-dist-in 4.254 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.188 0.237 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 7y1g AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA 6C0UA P17612 12 351 351.0 EE4:60400 Type1 Inactive DFGin 6.4885 14.2621 BLAminus -130.77, 175.54 62.84, 100.35 -119.36, 26.56 282.24, 71.26 -65.52, -23.67 in-in in 8.3667 Saltbr-in 3.028 HRD-in -79.47, -53.84 70.3, 8.89 in-in-out SNCiio in-out ActLoopNT-in 3.0007 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.41, 153.98 APE9-dihe-na 116.73, 155.27 APE8-dihe-in -73.99, 144.03 APE8-rot-out 173.49 APE67-dihe-in -64.51, -15.31 -53.81, -42.18 APE12-dist-in 7.614 APE11-dist-in 10.848 APE10-dist-in 5.4829 APE9-dist-in 3.9348 None TPO198,SEP339 TPO198,SEP339 XRAY 2.65 0.211 0.243 A 354.0 340.0 0 25 25 0 [[44, 298]] 1.0 6c0u AGC_PRKACA_HUMAN AGC 4.7e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha

AGC_PRKACA (cAMP-dependent protein kinase catalytic subunit alpha)

Total number of chains: 452
Active chains: 289
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 363 80.3% AF-P17612-K1A
DFGin ABAminus 80 17.7% 5M6YA
None None 5 1.1% 9DW7G
DFGin None 4 0.9% 4C35A

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PRKACA KAPCA_BOVIN 9DW9G P00517 13 351 351.0 ATP:401 ATPlike Active DFGin 6.5695 15.1264 BLAminus -133.9, -169.96 59.46, 64.31 -83.85, 33.99 275.29, 73.58 -66.33, -24.36 in-in in 9.4988 Saltbr-in 3.2167 HRD-in -92.3, -53.34 68.25, 14.14 in-in-in SNCiii in-in ActLoopNT-in 3.0799 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.91, 151.76 APE9-dihe-na 126.66, -174.62 APE8-dihe-in -92.84, 130.69 APE8-rot-in 299.41 APE67-dihe-in -68.55, -23.13 -58.33, -34.44 APE12-dist-in 8.7033 APE11-dist-in 11.5632 APE10-dist-in 6.1702 APE9-dist-in 4.5677 None TPO198 TPO198 EM 2.8 999.0 999.0 G 351.0 328.0 0 25 25 0 [[44, 298]] 1.0 9dw9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q24A P00517 15 351 351.0 ATP:60400 ATPlike Active DFGin 5.9832 14.3195 BLAminus -113.95, 178.0 66.86, 85.15 -103.99, 32.82 274.7, 64.8 -65.44, -25.66 in-in in 8.779 Saltbr-in 2.742 HRD-in -93.22, -55.61 73.46, 14.95 in-in-in SNCiii in-in ActLoopNT-in 3.0897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.66, 162.77 APE9-dihe-na 133.15, -143.39 APE8-dihe-in -135.22, 127.61 APE8-rot-in 301.89 APE67-dihe-in -67.43, -30.61 -42.63, -46.05 APE12-dist-in 8.0357 APE11-dist-in 11.4473 APE10-dist-in 6.0235 APE9-dist-in 3.486 V124A,L174M TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.202 0.25 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1q24 Bos taurus AGC_PRKACA_BOVIN AGC 4.8e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO7A P00517 15 351 351.0 M05:61351,M05:61352 Allosteric,Type1 Active DFGin 6.0589 13.3545 BLAminus -112.73, 170.06 64.79, 125.13 -129.63, 24.75 288.96, 78.29 -59.84, -27.0 in-in in 8.9212 Saltbr-in 2.5901 HRD-in -91.38, -48.53 69.14, 8.91 in-in-in SNCiii in-in ActLoopNT-in 2.9119 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.06, 161.81 APE9-dihe-na 128.93, -157.64 APE8-dihe-in -120.9, 132.32 APE8-rot-in 302.18 APE67-dihe-in -59.27, -25.29 -43.22, -50.55 APE12-dist-in 8.1025 APE11-dist-in 11.3217 APE10-dist-in 5.7515 APE9-dist-in 3.6251 None TPO198,SEP339 TPO198,SEP339 XRAY 1.98 0.191 0.241 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vo7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNGA P00517 11 351 351.0 No_ligand No_ligand Active DFGin 6.1399 14.2236 BLAminus -119.55, 178.04 62.47, 98.55 -111.03, 25.12 275.63, 67.2 -58.48, -24.65 in-in in 9.0055 Saltbr-in 2.6957 HRD-in -96.2, -52.02 73.83, 11.43 in-in-in SNCiii in-in ActLoopNT-in 2.9239 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.01, 159.86 APE9-dihe-na 129.89, -160.93 APE8-dihe-in -123.36, 138.18 APE8-rot-in 302.01 APE67-dihe-in -59.18, -22.88 -47.61, -51.91 APE12-dist-in 8.0125 APE11-dist-in 11.2898 APE10-dist-in 5.8022 APE9-dist-in 3.5598 L50I,V124M,E128D,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.87 0.198 0.258 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gng Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GFCA P00517 15 351 351.0 No_ligand No_ligand Active DFGin 6.1877 14.0711 BLAminus -117.74, 159.24 72.69, 98.85 -105.34, 28.02 271.26, 59.63 -61.26, -23.71 in-in in 8.6743 Saltbr-in 2.5762 HRD-in -90.3, -52.85 73.44, 9.78 in-in-in SNCiii in-in ActLoopNT-in 2.9736 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.8, 159.7 APE9-dihe-na 133.98, -157.58 APE8-dihe-in -121.29, 135.51 APE8-rot-in 301.46 APE67-dihe-in -58.17, -22.85 -42.97, -54.07 APE12-dist-in 8.0335 APE11-dist-in 11.2552 APE10-dist-in 5.7258 APE9-dist-in 3.5267 None TPO198,SEP339 TPO198,SEP339 XRAY 1.87 0.239 0.239 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 2gfc Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q61A P00517 15 351 351.0 No_ligand No_ligand Active DFGin 6.3166 14.0576 BLAminus -113.32, 171.66 65.32, 95.24 -105.6, 28.35 273.54, 62.22 -60.93, -24.2 in-in in 8.7701 Saltbr-in 2.7918 HRD-in -88.4, -55.05 70.66, 3.99 in-in-in SNCiii in-in ActLoopNT-in 2.7864 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.36, 157.96 APE9-dihe-na 134.42, -161.14 APE8-dihe-in -115.93, 129.95 APE8-rot-in 300.39 APE67-dihe-in -58.76, -26.29 -47.87, -46.79 APE12-dist-in 8.1766 APE11-dist-in 11.5728 APE10-dist-in 6.0171 APE9-dist-in 3.7962 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.184 0.232 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1q61 Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SMHA P00517 2 351 351.0 No_ligand No_ligand Active DFGin 6.7989 14.5799 BLAminus -115.56, -165.58 57.6, 64.56 -89.23, 16.63 272.25, 75.82 -57.78, -31.17 in-in in 8.8477 Saltbr-in 2.4417 HRD-in -96.56, -52.48 70.28, 5.31 in-in-in SNCiii in-in ActLoopNT-in 2.7976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.7, 159.43 APE9-dihe-na 133.86, -177.98 APE8-dihe-in -99.8, 130.8 APE8-rot-in 299.09 APE67-dihe-in -59.18, -25.63 -42.57, -53.75 APE12-dist-in 8.2039 APE11-dist-in 11.557 APE10-dist-in 6.0526 APE9-dist-in 3.7586 Q85E,V124A,L174M,F188L TPO198,SEP339 TPO198,SEP339 XRAY 2.044 0.191 0.238 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1smh Bos taurus AGC_PRKACA_BOVIN AGC 3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q62A P00517 14 351 351.0 No_ligand No_ligand Active DFGin 6.1823 14.2767 BLAminus -104.64, 174.54 66.86, 89.86 -104.82, 25.62 276.34, 54.84 -53.41, -25.33 in-in in 8.9311 Saltbr-in 2.6139 HRD-in -96.79, -53.25 66.13, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.8834 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.96, 166.05 APE9-dihe-na 130.72, -161.89 APE8-dihe-in -113.23, 133.18 APE8-rot-in 300.81 APE67-dihe-in -67.6, -24.51 -42.5, -46.58 APE12-dist-in 8.1409 APE11-dist-in 11.4273 APE10-dist-in 6.0155 APE9-dist-in 3.617 V124A,L174M TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.192 0.252 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1q62 Bos taurus AGC_PRKACA_BOVIN AGC 4.8e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C33A P00517 14 351 351.0 No_ligand No_ligand Active DFGin 6.3698 14.4633 BLAminus -122.61, 167.1 69.2, 93.31 -104.18, 28.64 273.24, 55.76 -56.02, -28.41 in-in in 8.8225 Saltbr-in 2.7134 HRD-in -80.43, -53.85 71.22, 13.56 in-in-in SNCiii in-in ActLoopNT-in 2.937 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.13, 162.95 APE9-dihe-na 124.44, -159.48 APE8-dihe-in -120.39, 137.89 APE8-rot-in 301.42 APE67-dihe-in -62.3, -24.0 -46.94, -49.76 APE12-dist-in 8.0022 APE11-dist-in 11.3971 APE10-dist-in 5.7782 APE9-dist-in 3.4384 F55Y,M121L,V124L,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.158 0.187 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4c33 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNFA P00517 11 351 351.0 Y27:60501 Type1 Active DFGin 6.0407 14.1738 BLAminus -116.96, 178.88 58.65, 105.43 -113.78, 28.7 272.88, 66.05 -63.78, -25.92 in-in in 9.2018 Saltbr-in 2.5932 HRD-in -94.14, -47.78 64.37, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.8822 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -171.34, 163.17 APE9-dihe-na 124.68, -165.19 APE8-dihe-in -121.59, 134.6 APE8-rot-in 288.13 APE67-dihe-in -58.1, -28.51 -44.73, -50.81 APE12-dist-in 8.0234 APE11-dist-in 11.2036 APE10-dist-in 5.8077 APE9-dist-in 3.4001 L50I,V124M,E128D,Q182K,T184A TPO198,SEP339 TPO198,SEP339 XRAY 2.28 0.201 0.258 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gnf Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNJA P00517 15 351 351.0 Y27:60501 Type1 Active DFGin 6.1039 13.6767 BLAminus -125.2, 164.0 75.11, 93.42 -104.04, 27.11 286.53, 71.0 -58.19, -29.08 in-in in 9.0921 Saltbr-in 2.8299 HRD-in -86.57, -53.41 73.77, 21.07 in-in-in SNCiii in-in ActLoopNT-in 2.7763 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.71, 163.04 APE9-dihe-na 124.17, -165.73 APE8-dihe-in -116.96, 135.69 APE8-rot-in 293.77 APE67-dihe-in -62.53, -24.27 -43.03, -48.93 APE12-dist-in 8.108 APE11-dist-in 11.3187 APE10-dist-in 5.7869 APE9-dist-in 3.4239 L50I,Q182K,T184A TPO198,SEP339 TPO198,SEP339 XRAY 2.28 0.19 0.262 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 2gnj Bos taurus AGC_PRKACA_BOVIN AGC 7.3e-95 323.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNLA P00517 12 351 351.0 H52:60501 Type1 Active DFGin 6.3581 14.8769 BLAminus -89.02, -175.74 47.17, 112.42 -122.51, 26.46 259.73, 63.8 -65.5, -20.97 in-in in 9.1821 Saltbr-in 2.6049 HRD-in -84.16, -63.35 83.4, 16.15 in-in-in SNCiii in-in ActLoopNT-in 2.8748 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.63, 164.56 APE9-dihe-na 121.8, -158.16 APE8-dihe-in -125.31, 137.52 APE8-rot-in 295.72 APE67-dihe-in -52.7, -17.18 -53.68, -49.84 APE12-dist-in 8.1164 APE11-dist-in 11.5217 APE10-dist-in 6.1495 APE9-dist-in 3.5167 L50I,Q182K,T184A TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.203 0.303 A 350.0 340.0 0 25 25 0 [[44, 298]] 1.0 2gnl Bos taurus AGC_PRKACA_BOVIN AGC 7.3e-95 323.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZTA P00517 16 351 351.0 SS3:61351 Type1 Active DFGin 6.8713 14.0778 BLAminus -126.85, 167.46 69.43, 90.19 -103.99, 29.38 280.49, 66.47 -59.79, -22.48 in-in in 9.1397 Saltbr-in 2.6911 HRD-in -77.75, -50.42 62.52, 13.49 in-in-in SNCiii in-in ActLoopNT-in 2.9856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -114.56, 156.36 APE9-dihe-na 116.01, -154.02 APE8-dihe-in -130.0, 127.43 APE8-rot-in 298.59 APE67-dihe-in -60.13, -24.22 -31.54, -56.49 APE12-dist-in 7.8297 APE11-dist-in 11.3914 APE10-dist-in 5.7844 APE9-dist-in 3.7237 None None None XRAY 2.1 0.273 0.313 A 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzt Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZUE P00517 16 351 351.0 L20:61351 Type1 Active DFGin 6.5165 14.3927 BLAminus -116.34, 172.4 61.54, 100.04 -109.49, 24.05 269.56, 56.18 -51.88, -19.43 in-in in 8.8645 Saltbr-in 2.5717 HRD-in -79.6, -53.73 68.74, 6.41 in-in-in SNCiii in-in ActLoopNT-in 3.0336 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.25, 159.94 APE9-dihe-na 132.5, -155.2 APE8-dihe-in -127.84, 130.66 APE8-rot-in 306.17 APE67-dihe-in -52.51, -26.75 -31.49, -67.12 APE12-dist-in 7.8584 APE11-dist-in 11.1723 APE10-dist-in 5.7612 APE9-dist-in 3.7464 None None None XRAY 2.4 0.318 0.371 E 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzu Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZVA P00517 16 351 351.0 SS5:61351 Type1 Active DFGin 6.7937 14.3133 BLAminus -133.61, 167.29 69.98, 107.83 -122.87, 25.1 278.16, 55.22 -54.77, -25.94 in-in in 9.0833 Saltbr-in 2.6706 HRD-in -77.51, -58.55 72.39, 6.58 in-in-in SNCiii in-in ActLoopNT-in 3.1559 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.23, 161.95 APE9-dihe-na 131.29, -149.51 APE8-dihe-in -126.03, 139.69 APE8-rot-in 311.31 APE67-dihe-in -45.96, -25.35 -39.61, -69.13 APE12-dist-in 7.7834 APE11-dist-in 11.1969 APE10-dist-in 5.8374 APE9-dist-in 3.677 None None None XRAY 2.5 0.251 0.316 A 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzv Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZWE P00517 16 351 351.0 SS4:61351 Type1 Active DFGin 6.5613 14.5744 BLAminus -112.04, -173.28 55.73, 87.87 -110.12, 39.6 275.39, 62.8 -71.34, -18.15 in-in in 8.8979 Saltbr-in 3.1279 HRD-in -78.88, -49.67 62.72, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.7912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.16, 162.59 APE9-dihe-na 103.28, -160.9 APE8-dihe-in -116.22, 129.17 APE8-rot-in 310.0 APE67-dihe-in -56.35, -23.35 -31.72, -57.46 APE12-dist-in 8.0868 APE11-dist-in 11.3531 APE10-dist-in 5.8387 APE9-dist-in 3.776 None None None XRAY 2.2 0.313 0.328 E 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzw Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q8TA P00517 11 351 351.0 Y27:60930 Type1 Active DFGin 6.1851 14.3139 BLAminus -117.96, 176.23 66.27, 91.07 -99.92, 24.26 275.29, 66.15 -60.05, -23.97 in-in in 9.0544 Saltbr-in 2.5891 HRD-in -93.15, -51.44 72.41, 0.56 in-in-in SNCiii in-in ActLoopNT-in 2.9525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.6, 160.94 APE9-dihe-na 131.1, -162.98 APE8-dihe-in -114.15, 135.68 APE8-rot-in 299.16 APE67-dihe-in -56.85, -26.83 -51.6, -49.02 APE12-dist-in 8.1774 APE11-dist-in 11.4755 APE10-dist-in 5.9128 APE9-dist-in 3.6886 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.182 0.229 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1q8t Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q8WA P00517 15 351 351.0 M77:60960 Type1 Active DFGin 6.5158 14.6907 BLAminus -127.81, 164.07 85.37, 88.74 -113.2, 23.58 288.03, 80.25 -50.72, -40.77 in-in in 8.8645 Saltbr-in 2.7877 HRD-in -88.09, -59.12 85.64, -3.61 in-in-in SNCiii in-in ActLoopNT-in 3.125 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.12, 157.94 APE9-dihe-na 118.72, -168.38 APE8-dihe-in -118.75, 133.72 APE8-rot-in 300.62 APE67-dihe-in -62.19, -20.35 -49.36, -50.33 APE12-dist-in 8.427 APE11-dist-in 11.7879 APE10-dist-in 6.3999 APE9-dist-in 4.0603 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.22 0.295 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1q8w Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SVEA P00517 8 351 351.0 I01:60351 Type1 Active DFGin 6.1664 14.2222 BLAminus -113.6, -176.53 62.78, 78.1 -100.84, 17.81 278.73, 68.66 -48.01, -28.95 in-in in 8.6662 Saltbr-in 2.5697 HRD-in -91.7, -56.06 76.75, 8.37 in-in-in SNCiii in-in ActLoopNT-in 3.0657 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.08, 161.63 APE9-dihe-na 125.64, -173.88 APE8-dihe-in -102.65, 133.23 APE8-rot-in 299.26 APE67-dihe-in -60.18, -26.54 -47.49, -48.66 APE12-dist-in 8.1227 APE11-dist-in 11.4552 APE10-dist-in 5.942 APE9-dist-in 3.5408 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.49 0.202 0.257 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 1sve Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SVGA P00517 11 351 351.0 I04:60351 Type1 Active DFGin 6.2852 14.1972 BLAminus -126.54, 177.16 64.26, 73.95 -91.56, 21.32 279.08, 73.3 -61.43, -19.1 in-in in 8.5805 Saltbr-in 2.6809 HRD-in -92.74, -53.98 73.19, 8.88 in-in-in SNCiii in-in ActLoopNT-in 2.9341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.17, 160.9 APE9-dihe-na 123.57, -169.23 APE8-dihe-in -108.56, 130.67 APE8-rot-in 293.73 APE67-dihe-in -66.93, -24.48 -43.76, -46.84 APE12-dist-in 8.0906 APE11-dist-in 11.5393 APE10-dist-in 6.0517 APE9-dist-in 3.6478 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.02 0.183 0.227 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1svg Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1VEBA P00517 11 351 351.0 I05:60351 Type1 Active DFGin 6.2131 14.2357 BLAminus -112.2, -169.65 49.77, 80.02 -102.5, 31.57 278.86, 61.26 -72.56, -20.75 in-in in 8.5766 Saltbr-in 2.8728 HRD-in -83.01, -49.6 62.13, 5.25 in-in-in SNCiii in-in ActLoopNT-in 3.0408 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.53, 158.22 APE9-dihe-na 134.18, -167.65 APE8-dihe-in -109.96, 136.58 APE8-rot-in 290.96 APE67-dihe-in -71.75, -2.37 -42.82, -49.75 APE12-dist-in 8.1776 APE11-dist-in 11.6793 APE10-dist-in 6.0598 APE9-dist-in 3.7367 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.89 0.187 0.251 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1veb Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH4A P00517 15 351 351.0 R69:60351 Type1 Active DFGin 6.2972 13.619 BLAminus -125.63, 176.59 60.0, 74.66 -89.7, 21.14 287.64, 81.0 -57.7, -30.21 in-in in 8.7553 Saltbr-in 2.5701 HRD-in -85.89, -55.59 71.5, 15.27 in-in-in SNCiii in-in ActLoopNT-in 3.0669 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.1, 158.39 APE9-dihe-na 135.4, -175.25 APE8-dihe-in -99.1, 130.32 APE8-rot-in 300.14 APE67-dihe-in -53.15, -30.05 -47.58, -48.79 APE12-dist-in 8.1288 APE11-dist-in 11.5852 APE10-dist-in 6.0366 APE9-dist-in 3.7183 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.45 0.191 0.242 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1xh4 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH5A P00517 15 351 351.0 R68:61001 Type1 Active DFGin 6.3947 13.2316 BLAminus -125.11, 175.33 63.85, 75.87 -93.6, 21.14 294.45, 75.91 -54.91, -25.56 in-in in 8.7353 Saltbr-in 2.7377 HRD-in -92.22, -50.1 68.22, 14.89 in-in-in SNCiii in-in ActLoopNT-in 2.9658 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.82, 159.18 APE9-dihe-na 129.26, -172.93 APE8-dihe-in -106.77, 134.87 APE8-rot-in 299.04 APE67-dihe-in -60.66, -25.82 -46.87, -48.0 APE12-dist-in 7.9509 APE11-dist-in 11.4133 APE10-dist-in 5.881 APE9-dist-in 3.5909 None TPO198,SEP339 TPO198,SEP339 XRAY 2.05 0.185 0.236 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1xh5 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH6A P00517 19 351 351.0 R94:60351 Type1 Active DFGin 6.1276 13.3787 BLAminus -130.28, 176.51 62.64, 74.17 -91.5, 20.79 288.12, 76.57 -51.25, -30.79 in-in in 8.8185 Saltbr-in 2.708 HRD-in -82.23, -52.65 67.28, 14.23 in-in-in SNCiii in-in ActLoopNT-in 3.0713 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.94, 161.1 APE9-dihe-na 129.62, -161.03 APE8-dihe-in -117.21, 135.0 APE8-rot-in 298.01 APE67-dihe-in -59.91, -22.98 -46.35, -48.26 APE12-dist-in 8.104 APE11-dist-in 11.5006 APE10-dist-in 5.9059 APE9-dist-in 3.4893 None TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.192 0.249 A 350.0 333.0 0 25 25 0 [[44, 298]] 1.0 1xh6 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH7A P00517 11 351 351.0 R96:60351 Type1 Active DFGin 6.3831 13.3018 BLAminus -121.57, 176.46 64.46, 76.56 -95.28, 25.2 293.04, 73.78 -55.65, -33.0 in-in in 8.6628 Saltbr-in 2.6788 HRD-in -88.46, -51.77 72.39, 6.4 in-in-in SNCiii in-in ActLoopNT-in 2.9193 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.76, 163.97 APE9-dihe-na 129.5, -170.45 APE8-dihe-in -100.96, 130.84 APE8-rot-in 305.54 APE67-dihe-in -56.25, -25.46 -42.72, -53.32 APE12-dist-in 7.9889 APE11-dist-in 11.7106 APE10-dist-in 6.0439 APE9-dist-in 3.9196 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.47 0.192 0.254 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1xh7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH8A P00517 13 351 351.0 R55:60351 Type1 Active DFGin 7.2199 14.5512 BLAminus -127.78, 170.11 66.78, 76.25 -93.48, 35.64 282.0, 79.13 -69.55, -13.04 in-in in 8.6647 Saltbr-in 2.5851 HRD-in -73.67, -49.45 69.2, 1.69 in-in-in SNCiii in-in ActLoopNT-in 2.9223 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.86, 150.19 APE9-dihe-na 125.99, -169.91 APE8-dihe-in -111.55, 132.51 APE8-rot-in 296.34 APE67-dihe-in -62.89, -22.39 -42.71, -52.56 APE12-dist-in 8.7908 APE11-dist-in 11.805 APE10-dist-in 6.255 APE9-dist-in 3.5116 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.202 0.236 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1xh8 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3KKVA P00517 14 351 351.0 B99:60351 Type1 Active DFGin 6.2802 14.9874 BLAminus -125.37, 172.94 64.41, 88.24 -101.41, 28.77 274.35, 61.51 -57.52, -30.45 in-in in 9.39 Saltbr-in 2.668 HRD-in -87.09, -58.29 72.04, 20.78 in-in-in SNCiii in-in ActLoopNT-in 2.9138 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.6, 161.14 APE9-dihe-na 126.5, -157.51 APE8-dihe-in -121.76, 131.58 APE8-rot-in 301.24 APE67-dihe-in -59.26, -23.73 -39.89, -55.55 APE12-dist-in 7.9861 APE11-dist-in 11.2507 APE10-dist-in 5.7729 APE9-dist-in 3.4844 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.8 0.203 0.225 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3kkv Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4IJ9A P00517 15 351 351.0 PTV:60401 Type1 Active DFGin 6.6148 14.131 BLAminus -111.94, -175.65 58.73, 79.19 -93.36, 11.75 269.03, 67.58 -54.32, -24.02 in-in in 8.8666 Saltbr-in 3.4017 HRD-in -79.91, -51.1 66.03, 1.36 in-in-in SNCiii in-in ActLoopNT-in 2.9049 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.66, 160.33 APE9-dihe-na 124.74, -169.36 APE8-dihe-in -102.85, 129.95 APE8-rot-in 307.44 APE67-dihe-in -60.51, -31.49 -37.15, -49.85 APE12-dist-in 8.2305 APE11-dist-in 11.4808 APE10-dist-in 5.8096 APE9-dist-in 3.3378 None TPO198,SEP339 TPO198,SEP339 XRAY 2.55 0.175 0.247 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4ij9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2C1AA P00517 15 351 351.0 I5S:61351 Type1 Active DFGin 6.2978 14.6265 BLAminus -124.46, -169.61 66.48, 66.45 -85.13, 21.14 273.21, 64.57 -65.03, -22.49 in-in in 9.003 Saltbr-in 2.6116 HRD-in -90.18, -53.0 74.43, 14.23 in-in-in SNCiii in-in ActLoopNT-in 2.9703 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.63, 158.7 APE9-dihe-na 138.5, -149.83 APE8-dihe-in -130.06, 134.27 APE8-rot-in 299.96 APE67-dihe-in -59.41, -28.42 -45.36, -49.19 APE12-dist-in 7.8481 APE11-dist-in 11.246 APE10-dist-in 5.7402 APE9-dist-in 3.5606 None TPO198,SEP339 TPO198,SEP339 XRAY 1.95 0.176 0.23 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2c1a Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2C1BA P00517 15 351 351.0 CQP:61351 Type1 Active DFGin 6.0179 14.5756 BLAminus -127.46, 168.13 73.41, 94.26 -102.97, 22.93 271.29, 59.53 -60.22, -28.98 in-in in 8.8601 Saltbr-in 2.6005 HRD-in -86.97, -55.45 75.34, 13.69 in-in-in SNCiii in-in ActLoopNT-in 2.9333 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.15, 165.93 APE9-dihe-na 130.88, -155.25 APE8-dihe-in -127.93, 130.25 APE8-rot-in 296.49 APE67-dihe-in -57.75, -24.32 -42.11, -51.87 APE12-dist-in 8.026 APE11-dist-in 11.266 APE10-dist-in 5.7202 APE9-dist-in 3.4692 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.162 0.211 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2c1b Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2F7EE P00517 16 351 351.0 2EA:60351 Type1 Active DFGin 6.4255 14.622 BLAminus -129.37, 172.24 65.85, 87.0 -103.27, 28.23 271.13, 52.64 -61.39, -20.95 in-in in 9.0188 Saltbr-in 2.5724 HRD-in -84.54, -55.3 68.58, 20.0 in-in-in SNCiii in-in ActLoopNT-in 3.0357 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.64, 149.46 APE9-dihe-na 134.17, -155.82 APE8-dihe-in -124.14, 133.58 APE8-rot-in 298.87 APE67-dihe-in -58.46, -26.82 -32.03, -63.88 APE12-dist-in 7.8441 APE11-dist-in 11.2456 APE10-dist-in 5.6686 APE9-dist-in 3.7407 None None None XRAY 2.0 0.283 0.323 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2f7e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2F7XE P00517 16 351 351.0 4EA:60351 Type1 Active DFGin 6.4787 14.4427 BLAminus -134.55, -177.23 60.89, 80.89 -96.41, 28.1 269.37, 55.24 -56.5, -28.29 in-in in 8.9136 Saltbr-in 2.4578 HRD-in -81.93, -53.89 61.67, 20.58 in-in-in SNCiii in-in ActLoopNT-in 2.989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.99, 155.02 APE9-dihe-na 135.32, -157.56 APE8-dihe-in -123.89, 130.78 APE8-rot-in 298.61 APE67-dihe-in -49.48, -26.89 -30.62, -70.43 APE12-dist-in 7.9799 APE11-dist-in 11.4061 APE10-dist-in 5.9418 APE9-dist-in 3.9333 None None None XRAY 1.9 0.268 0.297 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2f7x Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2F7ZE P00517 16 351 351.0 6EA:61000 Type1 Active DFGin 6.2259 13.9549 BLAminus -129.55, -167.66 49.24, 93.04 -110.0, 23.76 275.34, 53.4 -53.66, -28.22 in-in in 8.5633 Saltbr-in 3.0644 HRD-in -65.45, -44.81 59.73, 0.41 in-in-in SNCiii in-in ActLoopNT-in 2.9811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -169.37, 169.07 APE9-dihe-na 126.6, -164.29 APE8-dihe-in -104.93, 138.12 APE8-rot-in 285.38 APE67-dihe-in -37.82, -20.53 -38.18, -81.91 APE12-dist-in 7.8361 APE11-dist-in 11.3017 APE10-dist-in 6.2126 APE9-dist-in 3.7238 None None None XRAY 3.0 0.246 0.342 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2f7z Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2JDSA P00517 15 351 351.0 L20:61351 Type1 Active DFGin 6.2975 14.4588 BLAminus -119.85, 164.76 69.86, 95.65 -106.41, 24.64 270.02, 58.03 -63.42, -24.71 in-in in 8.8415 Saltbr-in 2.9556 HRD-in -93.07, -49.96 71.48, 12.63 in-in-in SNCiii in-in ActLoopNT-in 2.9911 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.76, 158.61 APE9-dihe-na 135.6, -151.18 APE8-dihe-in -131.14, 134.0 APE8-rot-in 299.22 APE67-dihe-in -56.34, -24.22 -43.06, -54.13 APE12-dist-in 7.9284 APE11-dist-in 11.2908 APE10-dist-in 5.7662 APE9-dist-in 3.5059 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.211 0.272 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2jds Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2OH0E P00517 16 351 351.0 2PY:60351 Type1 Active DFGin 6.5126 14.6531 BLAminus -127.37, 173.11 66.58, 90.68 -104.37, 27.73 269.87, 52.25 -56.81, -28.64 in-in in 8.9289 Saltbr-in 2.5821 HRD-in -77.86, -55.61 71.73, 4.87 in-in-in SNCiii in-in ActLoopNT-in 2.9184 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.82, 160.53 APE9-dihe-na 132.23, -161.93 APE8-dihe-in -120.81, 133.78 APE8-rot-in 295.17 APE67-dihe-in -53.8, -16.59 -31.38, -69.24 APE12-dist-in 7.8772 APE11-dist-in 11.1968 APE10-dist-in 5.8391 APE9-dist-in 3.6735 None None None XRAY 2.2 0.273 0.32 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2oh0 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2OJFE P00517 16 351 351.0 4PY:61000 Type1 Active DFGin 6.632 13.5749 BLAminus -129.09, 175.09 60.55, 94.36 -110.26, 30.25 290.83, 66.47 -61.76, -22.5 in-in in 8.9951 Saltbr-in 2.6975 HRD-in -83.69, -49.78 65.87, 9.9 in-in-in SNCiii in-in ActLoopNT-in 2.9369 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.63, 160.13 APE9-dihe-na 129.42, -154.83 APE8-dihe-in -123.4, 138.68 APE8-rot-in 295.74 APE67-dihe-in -57.43, -25.96 -38.07, -61.94 APE12-dist-in 7.9119 APE11-dist-in 11.2719 APE10-dist-in 5.8536 APE9-dist-in 3.6707 None None None XRAY 2.1 0.265 0.29 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2ojf Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3AG9B P00517 16 351 351.0 A02:60351 Type1 Active DFGin 6.7069 14.8178 BLAminus -118.08, 165.29 66.01, 91.25 -100.52, 22.8 270.89, 66.31 -51.41, -38.23 in-in in 9.1095 Saltbr-in 2.7494 HRD-in -86.2, -49.67 71.39, 4.04 in-in-in SNCiii in-in ActLoopNT-in 2.8575 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.38, 133.7 APE9-dihe-na 131.92, -165.0 APE8-dihe-in -83.45, 116.32 APE8-rot-in 314.25 APE67-dihe-in -59.66, -23.97 -46.78, -44.32 APE12-dist-in 8.1703 APE11-dist-in 11.9191 APE10-dist-in 6.8174 APE9-dist-in 5.6216 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.23 0.246 B 351.0 319.0 0 25 25 0 [[44, 298]] 1.0 3ag9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO1A P00517 10 351 351.0 SIJ:61351 Type1 Active DFGin 6.3414 14.0562 BLAminus -119.34, -177.25 63.83, 74.63 -95.99, 18.51 283.99, 75.88 -54.4, -29.22 in-in in 9.1037 Saltbr-in 2.6632 HRD-in -85.49, -49.19 68.51, 9.51 in-in-in SNCiii in-in ActLoopNT-in 2.9485 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.19, 161.74 APE9-dihe-na 124.38, -162.01 APE8-dihe-in -111.99, 135.74 APE8-rot-in 300.86 APE67-dihe-in -57.72, -23.86 -43.38, -54.21 APE12-dist-in 7.9994 APE11-dist-in 11.3701 APE10-dist-in 5.7652 APE9-dist-in 3.4439 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.162 0.19 A 351.0 342.0 0 25 25 0 [[44, 298]] 1.0 3zo1 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO4A P00517 15 351 351.0 QWI:61352 Type1 Active DFGin 5.971 14.4316 BLAminus -122.52, 179.4 62.97, 87.47 -105.16, 25.03 272.68, 69.84 -56.89, -28.47 in-in in 8.8067 Saltbr-in 2.6787 HRD-in -83.14, -51.38 69.84, 7.49 in-in-in SNCiii in-in ActLoopNT-in 2.9237 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.86, 163.63 APE9-dihe-na 121.61, -161.92 APE8-dihe-in -113.3, 134.36 APE8-rot-in 304.88 APE67-dihe-in -60.74, -25.7 -43.03, -50.51 APE12-dist-in 8.1783 APE11-dist-in 11.5104 APE10-dist-in 5.91 APE9-dist-in 3.4662 None TPO198,SEP339 TPO198,SEP339 XRAY 1.65 0.17 0.195 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3zo4 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4IE9A P00517 15 351 351.0 PZX:60401 Type1 Active DFGin 6.4403 14.5717 BLAminus -120.62, 176.92 66.27, 86.77 -100.95, 18.69 270.67, 65.37 -56.43, -28.52 in-in in 8.9159 Saltbr-in 2.77 HRD-in -89.08, -49.96 64.8, 10.82 in-in-in SNCiii in-in ActLoopNT-in 2.9618 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.58, 154.28 APE9-dihe-na 136.57, -156.42 APE8-dihe-in -117.79, 131.56 APE8-rot-in 300.22 APE67-dihe-in -56.73, -26.63 -41.25, -54.98 APE12-dist-in 8.1769 APE11-dist-in 11.3836 APE10-dist-in 5.8183 APE9-dist-in 3.6635 None TPO198,SEP339 TPO198,SEP339 XRAY 1.92 0.18 0.232 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4ie9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 5VHBA P00517 19 351 351.0 9CY:60401 Type1 Active DFGin 5.8914 14.4101 BLAminus -119.66, -177.23 60.94, 80.11 -93.35, 23.41 272.21, 58.28 -59.14, -26.18 in-in in 9.0291 Saltbr-in 2.7119 HRD-in -91.92, -50.82 66.2, 13.96 in-in-in SNCiii in-in ActLoopNT-in 2.9438 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.84, 154.36 APE9-dihe-na 131.28, -165.28 APE8-dihe-in -112.93, 137.33 APE8-rot-in 299.96 APE67-dihe-in -60.22, -22.29 -46.36, -53.5 APE12-dist-in 7.9601 APE11-dist-in 11.4577 APE10-dist-in 5.827 APE9-dist-in 3.8655 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.61 0.178 0.204 A 351.0 328.0 0 25 25 0 [[44, 298]] 1.0 5vhb Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 6E99A P00517 19 351 351.0 J0G:60601 Type1 Active DFGin 6.0023 14.6887 BLAminus -119.91, 176.13 61.41, 87.48 -95.36, 20.23 270.62, 61.24 -51.17, -35.89 in-in in 9.2093 Saltbr-in 2.7738 HRD-in -83.71, -54.36 68.2, 17.2 in-in-in SNCiii in-in ActLoopNT-in 3.0278 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.66, 157.43 APE9-dihe-na 126.17, -162.46 APE8-dihe-in -111.15, 131.88 APE8-rot-in 301.0 APE67-dihe-in -61.67, -24.67 -45.52, -49.68 APE12-dist-in 8.1145 APE11-dist-in 11.6023 APE10-dist-in 5.8812 APE9-dist-in 3.7622 None TPO198,SEP339 TPO198,SEP339 XRAY 1.88 0.208 0.23 A 351.0 333.0 0 25 25 0 [[44, 298]] 1.0 6e99 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 6E9LA P00517 18 351 351.0 J0P:60401 Type1 Active DFGin 6.4992 14.4033 BLAminus -98.87, -153.44 32.95, 78.78 -89.6, 15.58 275.81, 59.68 -55.89, -23.51 in-in in 8.8735 Saltbr-in 2.7663 HRD-in -69.86, -50.02 57.75, 17.6 in-in-in SNCiii in-in ActLoopNT-in 3.0358 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.26, 159.36 APE9-dihe-na 132.47, -166.61 APE8-dihe-in -110.57, 132.03 APE8-rot-in 295.04 APE67-dihe-in -57.99, -24.14 -37.74, -55.31 APE12-dist-in 7.9954 APE11-dist-in 11.7663 APE10-dist-in 6.1939 APE9-dist-in 4.0725 None TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.198 0.271 A 351.0 334.0 0 25 25 0 [[44, 298]] 1.0 6e9l Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 8SF8A P00517 13 351 351.0 ZWG:60401 Type1 Active DFGin 6.2798 14.2539 BLAminus -129.1, 170.06 68.03, 97.5 -109.47, 25.84 272.72, 61.91 -63.1, -22.98 in-in in 8.7505 Saltbr-in 2.7564 HRD-in -95.34, -49.3 69.01, 11.41 in-in-in SNCiii in-in ActLoopNT-in 2.8647 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.49, 160.11 APE9-dihe-na 135.6, -161.4 APE8-dihe-in -120.07, 137.81 APE8-rot-in 299.35 APE67-dihe-in -59.91, -22.91 -50.11, -49.66 APE12-dist-in 8.0794 APE11-dist-in 11.2474 APE10-dist-in 5.82 APE9-dist-in 3.5329 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.199 0.22 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 8sf8 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3DNDA P00517 16 351 351.0 LL2:60351 Type1 Active DFGin 6.5437 14.6347 BLAminus -116.16, 171.46 66.82, 93.02 -101.85, 16.18 271.74, 55.59 -52.63, -24.52 in-in in 9.1859 Saltbr-in 2.9585 HRD-in -95.42, -56.13 76.88, 13.37 in-in-in SNCiii in-in ActLoopNT-in 2.8599 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.6, 159.85 APE9-dihe-na 129.5, -152.83 APE8-dihe-in -125.57, 136.21 APE8-rot-in 298.43 APE67-dihe-in -52.95, -28.96 -44.81, -53.93 APE12-dist-in 8.0597 APE11-dist-in 11.3778 APE10-dist-in 5.8234 APE9-dist-in 3.4374 None TPO198,SEP339 TPO198,SEP339 XRAY 2.26 0.19 0.253 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 3dnd Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3DNEA P00517 14 351 351.0 LL1:60351 Type1 Active DFGin 6.437 14.4585 BLAminus -121.1, -178.57 64.95, 70.37 -87.98, 19.34 273.67, 65.23 -66.31, -20.97 in-in in 8.8191 Saltbr-in 2.7351 HRD-in -96.15, -42.67 61.27, 10.37 in-in-in SNCiii in-in ActLoopNT-in 2.8642 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.64, 165.13 APE9-dihe-na 129.71, -157.6 APE8-dihe-in -124.5, 137.89 APE8-rot-in 294.27 APE67-dihe-in -60.97, -25.49 -45.94, -52.87 APE12-dist-in 8.0593 APE11-dist-in 11.1643 APE10-dist-in 5.7175 APE9-dist-in 3.5291 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.179 0.23 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3dne Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4YXRA P00517 16 351 351.0 0RW:60401 Type1 Active DFGin 6.0086 14.2951 BLAminus -119.04, 170.91 66.3, 93.05 -106.53, 24.67 276.07, 60.12 -58.07, -27.2 in-in in 9.0005 Saltbr-in 2.7007 HRD-in -82.28, -52.44 64.39, 8.26 in-in-in SNCiii in-in ActLoopNT-in 2.8702 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.51, 157.24 APE9-dihe-na 130.59, -154.35 APE8-dihe-in -122.35, 133.27 APE8-rot-in 301.51 APE67-dihe-in -58.69, -25.56 -33.6, -61.81 APE12-dist-in 8.0106 APE11-dist-in 11.3632 APE10-dist-in 5.8486 APE9-dist-in 3.6367 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 999.0 0.252 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4yxr Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4YXSA P00517 15 351 351.0 EMU:60401 Type1 Active DFGin 6.2857 13.5939 BLAminus -119.26, 168.5 67.4, 97.14 -108.4, 23.82 281.89, 73.4 -58.43, -25.53 in-in in 8.6608 Saltbr-in 2.6403 HRD-in -81.58, -52.24 65.52, 13.45 in-in-in SNCiii in-in ActLoopNT-in 2.9722 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.78, 159.45 APE9-dihe-na 131.68, -155.75 APE8-dihe-in -118.67, 131.09 APE8-rot-in 300.67 APE67-dihe-in -60.75, -29.57 -37.55, -53.5 APE12-dist-in 7.9379 APE11-dist-in 11.2743 APE10-dist-in 5.702 APE9-dist-in 3.6169 None TPO198,SEP339 TPO198,SEP339 XRAY 2.11 0.179 0.232 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4yxs Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1YDRE P00517 16 351 351.0 IQP:60351 Type1 Active DFGin 6.3291 14.2499 BLAminus -123.41, -178.28 58.45, 85.19 -101.97, 32.19 283.4, 54.35 -61.44, -27.25 in-in in 9.0495 Saltbr-in 2.7847 HRD-in -72.07, -64.76 83.06, 0.73 in-in-in SNCiii in-in ActLoopNT-in 2.8217 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.65, 168.03 APE9-dihe-na 116.01, -166.19 APE8-dihe-in -108.88, 132.42 APE8-rot-in 303.05 APE67-dihe-in -60.22, -26.51 -39.35, -52.68 APE12-dist-in 7.8706 APE11-dist-in 11.2981 APE10-dist-in 5.8958 APE9-dist-in 3.7525 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.188 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1ydr Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1YDSE P00517 16 351 351.0 IQS:60351 Type1 Active DFGin 6.3904 14.2877 BLAminus -112.84, -174.99 60.37, 74.83 -97.86, 29.16 279.73, 63.74 -63.98, -20.15 in-in in 8.9368 Saltbr-in 2.7755 HRD-in -75.45, -57.26 74.03, 4.96 in-in-in SNCiii in-in ActLoopNT-in 2.8322 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.17, 169.02 APE9-dihe-na 97.73, -165.42 APE8-dihe-in -112.69, 125.84 APE8-rot-in 302.88 APE67-dihe-in -57.81, -27.95 -31.43, -56.99 APE12-dist-in 7.9405 APE11-dist-in 11.1848 APE10-dist-in 5.7383 APE9-dist-in 3.6085 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.199 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1yds Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1YDTE P00517 16 351 351.0 IQB:60351 Type1 Active DFGin 6.5625 14.5739 BLAminus -112.01, -173.33 55.77, 87.81 -110.08, 39.59 275.46, 62.76 -71.4, -18.08 in-in in 8.8978 Saltbr-in 3.1275 HRD-in -78.94, -49.64 62.76, 12.37 in-in-in SNCiii in-in ActLoopNT-in 2.7915 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.17, 162.58 APE9-dihe-na 103.22, -160.88 APE8-dihe-in -116.29, 129.25 APE8-rot-in 310.0 APE67-dihe-in -56.34, -23.41 -31.82, -57.38 APE12-dist-in 8.0876 APE11-dist-in 11.3528 APE10-dist-in 5.8378 APE9-dist-in 3.7764 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.194 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1ydt Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SZMA P00517 16 351 351.0 BI4:60351 Type1 Active DFGin 6.3181 15.3683 BLAminus -125.27, 171.81 65.17, 99.61 -108.03, 19.56 272.67, 80.44 -58.01, -35.62 in-in in 9.4925 Saltbr-in 2.5743 HRD-in -86.5, -61.07 68.65, 7.7 in-in-in SNCiii in-in ActLoopNT-in 3.0034 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 163.31 APE9-dihe-na 107.11, 170.89 APE8-dihe-in -74.89, 129.09 APE8-rot-in 328.61 APE67-dihe-in -51.73, -30.1 -54.41, -49.2 APE12-dist-in 8.0399 APE11-dist-in 11.3302 APE10-dist-in 5.7626 APE9-dist-in 3.8064 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 A 350.0 320.0 0 25 25 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4Z84A P00517 15 351 351.0 NVX:60401 Type1 Active DFGin 6.1539 14.585 BLAminus -122.35, -175.47 64.09, 72.13 -88.27, 20.06 271.08, 58.42 -49.77, -31.82 in-in in 9.0164 Saltbr-in 2.7991 HRD-in -96.48, -53.57 76.53, 13.57 in-in-in SNCiii in-in ActLoopNT-in 2.9176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.06, 154.73 APE9-dihe-na 134.03, -158.23 APE8-dihe-in -120.28, 132.43 APE8-rot-in 300.75 APE67-dihe-in -53.91, -23.24 -46.29, -52.23 APE12-dist-in 8.1505 APE11-dist-in 11.5238 APE10-dist-in 5.9254 APE9-dist-in 3.5106 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.554 0.209 0.234 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4z84 Bos taurus AGC_PRKACA_BOVIN AGC 1.7e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XHAA P00517 2 351 351.0 R68:61001 Type1 Active DFGin 6.2641 14.1375 BLAminus -120.5, -174.91 64.53, 71.29 -89.72, 23.88 279.31, 73.73 -56.55, -38.89 in-in in 8.7371 Saltbr-in 2.545 HRD-in -89.15, -49.54 68.47, 12.55 in-in-in SNCiii in-in ActLoopNT-in 2.9376 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.3, 164.66 APE9-dihe-na 127.73, 179.02 APE8-dihe-in -85.45, 132.2 APE8-rot-in 302.59 APE67-dihe-in -55.5, -36.01 -41.3, -53.29 APE12-dist-in 8.4646 APE11-dist-in 11.7786 APE10-dist-in 6.157 APE9-dist-in 3.7469 Q85E,V124A,L174M,F188L TPO198,SEP339 TPO198,SEP339 XRAY 2.46 0.223 0.272 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1xha Bos taurus AGC_PRKACA_BOVIN AGC 3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2JDTA P00517 16 351 351.0 I5S:61351 Type1 Active DFGin 6.2483 14.4539 BLAminus -118.34, -171.87 56.8, 75.79 -95.64, 21.06 274.55, 57.92 -54.25, -28.4 in-in in 8.8407 Saltbr-in 2.7265 HRD-in -87.26, -55.39 77.73, 12.38 in-in-in SNCiii in-in ActLoopNT-in 2.9989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.35, 160.37 APE9-dihe-na 136.22, -156.91 APE8-dihe-in -125.95, 134.07 APE8-rot-in 299.88 APE67-dihe-in -54.81, -22.83 -45.72, -53.17 APE12-dist-in 7.9604 APE11-dist-in 11.3761 APE10-dist-in 5.7901 APE9-dist-in 3.5461 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.15 0.203 0.259 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2jdt Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2JDVA P00517 16 351 351.0 L20:61351 Type1 Active DFGin 6.8915 13.8202 BLAminus -131.77, 167.29 66.94, 91.79 -105.86, 27.67 278.62, 60.56 -53.86, -24.56 in-in in 8.8406 Saltbr-in 2.8778 HRD-in -94.92, -55.32 76.45, 14.41 in-in-in SNCiii in-in ActLoopNT-in 2.9231 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.28, 166.03 APE9-dihe-na 121.76, -153.88 APE8-dihe-in -130.57, 133.66 APE8-rot-in 294.95 APE67-dihe-in -54.68, -28.08 -47.57, -51.85 APE12-dist-in 8.0027 APE11-dist-in 11.3848 APE10-dist-in 5.7807 APE9-dist-in 3.4188 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.08 0.21 0.276 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2jdv Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UVXA P00517 15 351 351.0 GVH:61351 Type1 Active DFGin 6.4797 13.8517 BLAminus -113.02, 171.98 67.75, 90.65 -101.98, 28.22 272.02, 52.69 -58.83, -28.67 in-in in 8.4347 Saltbr-in 2.8578 HRD-in -88.35, -54.63 73.53, 9.81 in-in-in SNCiii in-in ActLoopNT-in 2.9512 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.14, 156.72 APE9-dihe-na 129.39, -155.0 APE8-dihe-in -123.88, 135.4 APE8-rot-in 299.16 APE67-dihe-in -58.73, -23.74 -45.63, -51.62 APE12-dist-in 7.8612 APE11-dist-in 11.2242 APE10-dist-in 5.6959 APE9-dist-in 3.5342 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.175 0.237 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uvx Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UVYA P00517 16 351 351.0 GVI:61351 Type1 Active DFGin 6.6883 13.7301 BLAminus -138.26, 177.38 63.89, 90.39 -103.82, 30.2 278.88, 60.78 -58.29, -25.32 in-in in 8.5322 Saltbr-in 2.8677 HRD-in -91.19, -52.46 73.0, 13.57 in-in-in SNCiii in-in ActLoopNT-in 2.955 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.29, 164.08 APE9-dihe-na 125.27, -164.76 APE8-dihe-in -118.0, 134.0 APE8-rot-in 303.1 APE67-dihe-in -57.9, -24.5 -45.7, -51.96 APE12-dist-in 7.8997 APE11-dist-in 11.319 APE10-dist-in 5.7311 APE9-dist-in 3.5369 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.218 0.253 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uvy Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UVZA P00517 15 351 351.0 GVJ:61351 Type1 Active DFGin 6.4579 13.9569 BLAminus -114.74, -176.7 66.06, 78.43 -99.26, 24.12 270.22, 58.52 -59.61, -24.08 in-in in 8.5257 Saltbr-in 2.6293 HRD-in -92.0, -54.55 74.61, 15.4 in-in-in SNCiii in-in ActLoopNT-in 2.8816 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.48, 161.55 APE9-dihe-na 129.65, -159.59 APE8-dihe-in -126.36, 133.57 APE8-rot-in 300.99 APE67-dihe-in -58.07, -24.11 -45.65, -50.65 APE12-dist-in 7.8629 APE11-dist-in 11.1547 APE10-dist-in 5.6461 APE9-dist-in 3.4616 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.94 0.205 0.245 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uvz Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW0A P00517 15 351 351.0 GVK:61351 Type1 Active DFGin 6.6807 13.8545 BLAminus -123.12, 170.63 63.31, 92.05 -104.17, 27.62 276.86, 57.75 -54.59, -30.88 in-in in 8.6064 Saltbr-in 2.7061 HRD-in -91.98, -52.4 71.75, 13.11 in-in-in SNCiii in-in ActLoopNT-in 2.9563 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.42, 159.97 APE9-dihe-na 125.35, -161.9 APE8-dihe-in -119.06, 132.94 APE8-rot-in 303.5 APE67-dihe-in -59.26, -23.73 -42.54, -53.1 APE12-dist-in 7.95 APE11-dist-in 11.363 APE10-dist-in 5.817 APE9-dist-in 3.5714 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.204 0.248 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw0 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW3A P00517 15 351 351.0 GVG:61351 Type1 Active DFGin 6.5124 13.5734 BLAminus -134.7, 177.07 65.72, 91.81 -107.38, 30.0 281.86, 61.73 -63.9, -19.07 in-in in 8.5145 Saltbr-in 2.9351 HRD-in -92.24, -48.61 69.34, 10.98 in-in-in SNCiii in-in ActLoopNT-in 2.9305 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.62, 157.61 APE9-dihe-na 126.53, -159.5 APE8-dihe-in -119.31, 132.1 APE8-rot-in 301.91 APE67-dihe-in -60.53, -27.24 -45.08, -48.44 APE12-dist-in 7.8948 APE11-dist-in 11.2961 APE10-dist-in 5.7653 APE9-dist-in 3.5543 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.19 0.191 0.252 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw3 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW4A P00517 15 351 351.0 L15:61351 Type1 Active DFGin 6.4921 14.0113 BLAminus -125.98, 178.92 62.3, 87.41 -98.07, 19.83 275.17, 58.86 -56.03, -29.21 in-in in 8.6955 Saltbr-in 2.6847 HRD-in -99.89, -51.11 66.26, 15.03 in-in-in SNCiii in-in ActLoopNT-in 2.9933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.17, 154.32 APE9-dihe-na 136.7, -157.38 APE8-dihe-in -123.04, 134.76 APE8-rot-in 305.65 APE67-dihe-in -59.99, -23.88 -42.91, -53.6 APE12-dist-in 7.8692 APE11-dist-in 11.2922 APE10-dist-in 5.8184 APE9-dist-in 3.8346 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.274 A 351.0 336.0 1 25 25 0 [[44, 298]] 1.0 2uw4 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW5A P00517 16 351 351.0 GVN:61351 Type1 Active DFGin 6.4006 13.8772 BLAminus -133.91, 172.04 65.21, 93.24 -108.15, 25.65 277.97, 62.72 -53.54, -37.02 in-in in 8.7284 Saltbr-in 2.8062 HRD-in -86.0, -54.55 71.01, 10.44 in-in-in SNCiii in-in ActLoopNT-in 2.9816 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.67, 159.27 APE9-dihe-na 130.34, -162.49 APE8-dihe-in -114.97, 133.7 APE8-rot-in 296.24 APE67-dihe-in -62.66, -23.25 -45.46, -47.84 APE12-dist-in 7.9004 APE11-dist-in 11.248 APE10-dist-in 5.7124 APE9-dist-in 3.5694 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.14 0.207 0.259 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uw5 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW6A P00517 15 351 351.0 GVO:61351 Type1 Active DFGin 6.5366 14.032 BLAminus -123.92, -171.55 58.59, 76.44 -99.17, 23.1 278.06, 64.52 -53.95, -28.73 in-in in 8.8994 Saltbr-in 2.6953 HRD-in -89.32, -52.49 72.51, 13.36 in-in-in SNCiii in-in ActLoopNT-in 2.8911 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.65, 165.8 APE9-dihe-na 120.56, -163.15 APE8-dihe-in -118.84, 134.95 APE8-rot-in 297.85 APE67-dihe-in -59.8, -23.71 -47.39, -48.58 APE12-dist-in 7.9462 APE11-dist-in 11.3542 APE10-dist-in 5.7826 APE9-dist-in 3.5043 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.23 0.192 0.244 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw6 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW7A P00517 15 351 351.0 GVP:61351 Type1 Active DFGin 6.6166 13.7352 BLAminus -136.69, 175.22 59.69, 95.21 -111.12, 31.03 278.38, 57.43 -58.09, -25.49 in-in in 8.5612 Saltbr-in 2.7092 HRD-in -86.23, -51.08 72.7, 10.78 in-in-in SNCiii in-in ActLoopNT-in 3.0203 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.27, 162.23 APE9-dihe-na 121.1, -162.52 APE8-dihe-in -116.53, 136.36 APE8-rot-in 303.46 APE67-dihe-in -55.18, -28.45 -48.94, -51.5 APE12-dist-in 7.93 APE11-dist-in 11.4491 APE10-dist-in 5.8017 APE9-dist-in 3.5143 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.239 0.318 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw7 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW8A P00517 15 351 351.0 GVQ:61351 Type1 Active DFGin 6.3045 14.2798 BLAminus -127.77, 173.64 63.87, 90.76 -102.26, 24.27 274.86, 58.11 -57.85, -25.36 in-in in 8.7881 Saltbr-in 2.6187 HRD-in -87.86, -52.11 70.45, 11.81 in-in-in SNCiii in-in ActLoopNT-in 2.9485 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.21, 162.91 APE9-dihe-na 127.4, -162.92 APE8-dihe-in -121.14, 133.97 APE8-rot-in 304.45 APE67-dihe-in -56.86, -24.67 -46.34, -50.57 APE12-dist-in 7.9507 APE11-dist-in 11.2821 APE10-dist-in 5.7747 APE9-dist-in 3.5317 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.188 0.233 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw8 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VNWA P00517 15 351 351.0 M01:61351 Type1 Active DFGin 6.5203 14.2539 BLAminus -99.0, -162.5 57.81, 69.82 -93.2, 19.41 267.8, 58.81 -57.89, -28.06 in-in in 8.608 Saltbr-in 2.7916 HRD-in -93.79, -52.83 75.12, 12.44 in-in-in SNCiii in-in ActLoopNT-in 2.9661 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.21, 164.77 APE9-dihe-na 124.54, -157.72 APE8-dihe-in -125.0, 133.49 APE8-rot-in 299.26 APE67-dihe-in -56.84, -26.04 -43.44, -52.9 APE12-dist-in 7.8989 APE11-dist-in 11.3061 APE10-dist-in 5.7483 APE9-dist-in 3.4375 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.09 0.179 0.247 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vnw Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VNYA P00517 15 351 351.0 M02:61351 Type1 Active DFGin 6.5021 13.8926 BLAminus -119.89, 177.02 61.41, 90.56 -103.09, 29.14 278.68, 50.15 -55.55, -28.57 in-in in 8.4839 Saltbr-in 2.8581 HRD-in -86.58, -53.8 72.94, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.9193 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.32, 164.15 APE9-dihe-na 124.54, -158.42 APE8-dihe-in -121.16, 130.65 APE8-rot-in 300.17 APE67-dihe-in -57.01, -22.39 -43.28, -52.93 APE12-dist-in 7.9208 APE11-dist-in 11.3298 APE10-dist-in 5.8145 APE9-dist-in 3.478 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.96 0.226 0.292 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vny Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO3A P00517 15 351 351.0 M04:61352 Type1 Active DFGin 6.4299 14.4177 BLAminus -103.33, -162.63 58.24, 61.11 -86.11, 18.5 266.87, 55.84 -51.81, -33.51 in-in in 8.7704 Saltbr-in 2.6553 HRD-in -94.44, -55.26 74.28, 15.13 in-in-in SNCiii in-in ActLoopNT-in 2.9179 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.75, 157.39 APE9-dihe-na 131.99, -148.74 APE8-dihe-in -128.37, 129.57 APE8-rot-in 302.29 APE67-dihe-in -55.2, -26.12 -39.48, -55.25 APE12-dist-in 7.9685 APE11-dist-in 11.4444 APE10-dist-in 5.8578 APE9-dist-in 3.6169 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.98 0.189 0.246 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vo3 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO6A P00517 14 351 351.0 M05:61352 Type1 Active DFGin 6.4346 14.1872 BLAminus -116.69, -177.73 56.84, 84.85 -93.23, 27.76 272.38, 55.86 -61.33, -23.85 in-in in 8.6236 Saltbr-in 2.7502 HRD-in -94.44, -52.03 70.59, 14.63 in-in-in SNCiii in-in ActLoopNT-in 2.9129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.43, 161.66 APE9-dihe-na 131.96, -159.34 APE8-dihe-in -122.22, 131.28 APE8-rot-in 303.11 APE67-dihe-in -58.4, -24.83 -41.37, -51.96 APE12-dist-in 7.9982 APE11-dist-in 11.3208 APE10-dist-in 5.7969 APE9-dist-in 3.5782 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.97 0.175 0.229 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 2vo6 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C36A P00517 14 351 351.0 ZO9:61351 Type1 Active DFGin 6.1806 14.4761 BLAminus -118.69, 178.88 60.12, 90.41 -102.76, 21.93 269.17, 67.05 -52.26, -31.89 in-in in 8.958 Saltbr-in 2.7522 HRD-in -81.95, -52.55 68.64, 5.14 in-in-in SNCiii in-in ActLoopNT-in 2.9473 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.13, 158.34 APE9-dihe-na 127.36, -163.94 APE8-dihe-in -108.9, 133.1 APE8-rot-in 299.72 APE67-dihe-in -56.07, -28.95 -40.56, -54.07 APE12-dist-in 8.1424 APE11-dist-in 11.4572 APE10-dist-in 5.8378 APE9-dist-in 3.5366 F55Y,M121L,V124L,L174M,Q182K SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.98 0.158 0.19 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4c36 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C38A P00517 15 351 351.0 VUP:61351 Type1 Active DFGin 6.2217 14.4048 BLAminus -126.62, 165.92 74.69, 93.13 -106.33, 26.68 268.54, 56.88 -59.81, -19.94 in-in in 8.7724 Saltbr-in 2.7124 HRD-in -83.07, -52.03 71.32, 8.89 in-in-in SNCiii in-in ActLoopNT-in 2.9254 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.52, 161.58 APE9-dihe-na 127.55, -160.47 APE8-dihe-in -120.22, 132.35 APE8-rot-in 299.09 APE67-dihe-in -60.14, -23.8 -44.31, -50.86 APE12-dist-in 8.074 APE11-dist-in 11.4506 APE10-dist-in 5.8341 APE9-dist-in 3.5064 F55Y,M121L,V124L,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.58 0.154 0.178 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4c38 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q8UA P00517 8 351 351.0 H52:60961,H52:60962 Type1,Allosteric Active DFGin 6.1919 14.5396 BLAminus -121.34, -175.23 53.4, 94.64 -107.06, 23.52 275.18, 66.66 -55.71, -29.87 in-in in 9.3646 Saltbr-in 2.6498 HRD-in -94.99, -53.62 73.43, 4.82 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.92, 158.63 APE9-dihe-na 129.17, -156.38 APE8-dihe-in -121.51, 130.86 APE8-rot-in 299.83 APE67-dihe-in -61.21, -26.61 -47.69, -47.6 APE12-dist-in 8.2067 APE11-dist-in 11.5494 APE10-dist-in 5.967 APE9-dist-in 3.6469 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.9 0.173 0.206 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 1q8u Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3BWJA P00517 11 351 351.0 ARX:60351,ARX:60352 Type1,Allosteric Active DFGin 6.696 14.4073 BLAminus -110.43, 169.36 68.32, 91.4 -103.19, 23.79 279.15, 62.0 -69.5, -7.66 in-in in 8.6647 Saltbr-in 2.7201 HRD-in -86.31, -55.51 71.76, 12.05 in-in-in SNCiii in-in ActLoopNT-in 2.8621 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.81, 155.85 APE9-dihe-na 142.65, -162.5 APE8-dihe-in -110.95, 130.57 APE8-rot-in 293.64 APE67-dihe-in -63.27, -21.79 -42.33, -48.7 APE12-dist-in 8.115 APE11-dist-in 11.3778 APE10-dist-in 5.9209 APE9-dist-in 3.7349 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.201 0.249 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 3bwj Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4Z83E P00517 15 351 351.0 4L7:60401,4L7:60402 Type1,Allosteric Active DFGin 5.9886 14.5734 BLAminus -130.13, -162.52 52.5, 73.8 -91.1, 22.2 271.01, 60.02 -56.14, -30.3 in-in in 8.9604 Saltbr-in 2.6159 HRD-in -86.75, -50.89 68.08, 10.37 in-in-in SNCiii in-in ActLoopNT-in 2.878 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.2, 158.26 APE9-dihe-na 130.71, -157.52 APE8-dihe-in -119.41, 132.79 APE8-rot-in 303.19 APE67-dihe-in -56.65, -23.66 -45.82, -50.99 APE12-dist-in 8.1208 APE11-dist-in 11.4963 APE10-dist-in 5.9491 APE9-dist-in 3.7101 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.8 0.182 0.217 E 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4z83 Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO0A P00517 9 351 351.0 M03:61354,M03:61355 Type1,Allosteric Active DFGin 6.4684 14.4354 BLAminus -105.06, -163.48 59.05, 63.73 -87.9, 21.77 268.86, 60.16 -61.88, -26.99 in-in in 8.8145 Saltbr-in 2.4561 HRD-in -97.05, -57.43 76.4, 9.67 in-in-in SNCiii in-in ActLoopNT-in 2.8932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.64, 159.11 APE9-dihe-na 131.22, -153.01 APE8-dihe-in -127.42, 133.63 APE8-rot-in 298.09 APE67-dihe-in -55.96, -25.96 -42.79, -54.49 APE12-dist-in 7.9676 APE11-dist-in 11.3833 APE10-dist-in 5.8985 APE9-dist-in 3.6486 V105T,V124A,L174M,Q182K SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.94 0.165 0.216 A 351.0 343.0 0 25 25 0 [[44, 298]] 1.0 2vo0 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CA P00517 8 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.2009 14.4431 BLAminus -125.76, -178.37 54.76, 79.93 -90.51, 28.04 276.07, 57.76 -61.29, -35.5 in-in in 8.8075 Saltbr-in 2.8579 HRD-in -85.03, -54.57 65.22, 22.07 in-in-in SNCiii in-in ActLoopNT-in 2.8219 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.95, 159.1 APE9-dihe-na 118.65, -172.42 APE8-dihe-in -101.75, 128.13 APE8-rot-in 295.06 APE67-dihe-in -58.34, -26.98 -41.06, -49.71 APE12-dist-in 8.0918 APE11-dist-in 11.5524 APE10-dist-in 6.1282 APE9-dist-in 3.9113 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CB P00517 5 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.5319 14.6298 BLAminus -126.7, -178.91 56.82, 78.03 -91.32, 30.19 275.18, 53.57 -61.25, -34.87 in-in in 8.7621 Saltbr-in 3.0566 HRD-in -84.6, -55.03 67.66, 19.16 in-in-in SNCiii in-in ActLoopNT-in 2.8012 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.35, 159.24 APE9-dihe-na 119.5, -170.09 APE8-dihe-in -105.39, 130.22 APE8-rot-in 303.07 APE67-dihe-in -57.44, -28.07 -44.47, -49.51 APE12-dist-in 8.0466 APE11-dist-in 11.5239 APE10-dist-in 6.0242 APE9-dist-in 3.8597 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 B 350.0 347.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CC P00517 8 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.2974 14.7558 BLAminus -125.92, -177.85 55.25, 79.64 -90.5, 29.38 270.76, 52.31 -60.78, -37.14 in-in in 8.8167 Saltbr-in 2.6352 HRD-in -82.84, -55.25 65.25, 20.45 in-in-in SNCiii in-in ActLoopNT-in 2.8166 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.33, 159.63 APE9-dihe-na 118.14, -173.27 APE8-dihe-in -100.83, 130.06 APE8-rot-in 300.03 APE67-dihe-in -60.34, -24.98 -43.86, -49.06 APE12-dist-in 8.0524 APE11-dist-in 11.5266 APE10-dist-in 6.0815 APE9-dist-in 3.9132 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 C 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CD P00517 5 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.4689 14.6139 BLAminus -125.62, -178.32 56.8, 78.69 -92.33, 30.68 274.67, 61.46 -62.35, -34.64 in-in in 8.7979 Saltbr-in 2.6568 HRD-in -84.05, -54.95 66.91, 19.26 in-in-in SNCiii in-in ActLoopNT-in 2.8137 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.6, 160.31 APE9-dihe-na 118.55, -170.22 APE8-dihe-in -103.2, 129.22 APE8-rot-in 310.88 APE67-dihe-in -59.74, -24.78 -43.75, -49.55 APE12-dist-in 8.092 APE11-dist-in 11.4883 APE10-dist-in 6.0672 APE9-dist-in 3.881 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 D 350.0 347.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CE P00517 14 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.4857 14.6047 BLAminus -126.72, -179.02 57.21, 78.54 -91.86, 29.91 275.24, 58.74 -61.76, -34.81 in-in in 8.7747 Saltbr-in 2.8495 HRD-in -84.14, -54.47 66.34, 19.61 in-in-in SNCiii in-in ActLoopNT-in 2.8132 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.41, 160.32 APE9-dihe-na 118.41, -171.62 APE8-dihe-in -103.31, 130.93 APE8-rot-in 316.9 APE67-dihe-in -58.71, -26.13 -46.25, -48.17 APE12-dist-in 8.0859 APE11-dist-in 11.519 APE10-dist-in 6.0608 APE9-dist-in 3.871 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 E 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CF P00517 8 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.204 14.5963 BLAminus -125.48, -179.37 56.48, 79.11 -90.97, 29.84 273.44, 55.64 -61.95, -35.57 in-in in 8.801 Saltbr-in 2.9055 HRD-in -84.03, -54.54 65.26, 20.82 in-in-in SNCiii in-in ActLoopNT-in 2.8163 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.83, 160.18 APE9-dihe-na 118.26, -172.77 APE8-dihe-in -101.93, 130.0 APE8-rot-in 316.95 APE67-dihe-in -59.02, -26.57 -43.48, -49.35 APE12-dist-in 8.0793 APE11-dist-in 11.4951 APE10-dist-in 6.0617 APE9-dist-in 3.8792 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 F 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EA P00517 8 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.3073 14.6275 BLAminus -127.58, 177.12 59.26, 81.09 -89.3, 24.2 272.49, 51.41 -54.01, -38.82 in-in in 8.6228 Saltbr-in 2.6167 HRD-in -86.71, -49.98 69.16, 6.49 in-in-in SNCiii in-in ActLoopNT-in 2.8632 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.99, 154.32 APE9-dihe-na 133.62, -170.54 APE8-dihe-in -106.52, 129.54 APE8-rot-in 301.27 APE67-dihe-in -53.09, -32.91 -42.99, -51.98 APE12-dist-in 8.2069 APE11-dist-in 11.4816 APE10-dist-in 5.9204 APE9-dist-in 3.7722 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EB P00517 13 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.2938 14.7178 BLAminus -125.84, -172.92 50.21, 81.31 -89.14, 23.18 270.21, 58.55 -50.98, -43.5 in-in in 8.6642 Saltbr-in 2.6654 HRD-in -82.38, -53.17 68.54, 5.22 in-in-in SNCiii in-in ActLoopNT-in 2.8797 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.38, 161.75 APE9-dihe-na 128.75, -165.32 APE8-dihe-in -112.15, 133.4 APE8-rot-in 300.5 APE67-dihe-in -58.46, -24.04 -42.84, -57.3 APE12-dist-in 8.0985 APE11-dist-in 11.3489 APE10-dist-in 5.8215 APE9-dist-in 3.724 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 B 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EE P00517 8 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.5022 14.7143 BLAminus -125.94, 177.63 60.28, 78.38 -89.05, 26.68 272.68, 53.04 -58.15, -33.43 in-in in 8.5959 Saltbr-in 2.7412 HRD-in -83.69, -53.19 69.3, 12.83 in-in-in SNCiii in-in ActLoopNT-in 2.9203 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.44, 161.83 APE9-dihe-na 125.18, -160.92 APE8-dihe-in -119.48, 128.06 APE8-rot-in 308.71 APE67-dihe-in -61.97, -23.41 -42.69, -51.33 APE12-dist-in 8.1077 APE11-dist-in 11.5081 APE10-dist-in 5.9999 APE9-dist-in 3.6674 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 E 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EI P00517 4 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.2839 14.6216 BLAminus -121.51, -176.84 52.35, 81.35 -90.04, 28.89 273.59, 58.29 -59.59, -35.26 in-in in 8.5151 Saltbr-in 2.667 HRD-in -96.55, -53.06 68.92, 16.49 in-in-in SNCiii in-in ActLoopNT-in 2.8724 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.85, 164.56 APE9-dihe-na 117.18, -165.89 APE8-dihe-in -113.08, 128.95 APE8-rot-in 295.01 APE67-dihe-in -62.64, -25.23 -41.3, -50.45 APE12-dist-in 8.1826 APE11-dist-in 11.4443 APE10-dist-in 5.9011 APE9-dist-in 3.5317 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 I 350.0 348.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EL P00517 14 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.3558 14.4455 BLAminus -126.34, 179.53 56.51, 87.88 -97.22, 26.99 274.78, 53.86 -54.08, -36.01 in-in in 8.4902 Saltbr-in 2.9058 HRD-in -84.79, -53.72 69.04, 14.43 in-in-in SNCiii in-in ActLoopNT-in 2.9175 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.8, 165.17 APE9-dihe-na 117.16, -168.03 APE8-dihe-in -109.85, 132.76 APE8-rot-in 309.54 APE67-dihe-in -58.05, -25.67 -43.08, -54.13 APE12-dist-in 8.0742 APE11-dist-in 11.4769 APE10-dist-in 5.8902 APE9-dist-in 3.5416 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 L 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EP P00517 8 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.3511 14.4567 BLAminus -129.89, 174.6 59.69, 84.32 -91.75, 22.85 273.06, 63.33 -54.83, -37.28 in-in in 8.5071 Saltbr-in 3.0872 HRD-in -91.09, -52.59 71.75, 13.86 in-in-in SNCiii in-in ActLoopNT-in 2.8806 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.01, 169.23 APE9-dihe-na 113.75, -166.64 APE8-dihe-in -114.16, 128.38 APE8-rot-in 299.83 APE67-dihe-in -58.07, -28.95 -41.88, -52.2 APE12-dist-in 8.1136 APE11-dist-in 11.4255 APE10-dist-in 5.9681 APE9-dist-in 3.5443 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 P 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH9A P00517 14 351 351.0 R69:60351 Type1.5_Front Active DFGin 6.209 14.3533 BLAminus -129.75, -179.11 60.33, 73.87 -88.04, 22.6 274.32, 67.63 -61.73, -24.72 in-in in 8.5813 Saltbr-in 2.6088 HRD-in -83.79, -50.21 70.28, 10.19 in-in-in SNCiii in-in ActLoopNT-in 2.9141 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.47, 163.02 APE9-dihe-na 127.04, -169.55 APE8-dihe-in -104.83, 132.1 APE8-rot-in 300.02 APE67-dihe-in -61.76, -25.27 -43.65, -49.85 APE12-dist-in 8.2976 APE11-dist-in 11.8047 APE10-dist-in 6.2189 APE9-dist-in 3.6955 Q85E,V124A,L174M,Q182K,F188L TPO198,SEP339 TPO198,SEP339 XRAY 1.64 0.166 0.199 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1xh9 Bos taurus AGC_PRKACA_BOVIN AGC 1e-94 322.6 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SVHA P00517 15 351 351.0 I08:60351 Type1.5_Front Active DFGin 6.2901 14.3586 BLAminus -115.3, -171.03 56.71, 72.97 -89.54, 18.36 276.49, 75.83 -65.64, -21.28 in-in in 8.5191 Saltbr-in 2.4169 HRD-in -84.39, -53.98 69.64, 16.78 in-in-in SNCiii in-in ActLoopNT-in 3.0122 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.15, 156.51 APE9-dihe-na 127.45, -173.0 APE8-dihe-in -94.86, 131.95 APE8-rot-in 296.28 APE67-dihe-in -64.98, -17.24 -40.94, -52.95 APE12-dist-in 8.6846 APE11-dist-in 11.7208 APE10-dist-in 6.2204 APE9-dist-in 3.7125 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.214 0.259 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1svh Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNIA P00517 11 351 351.0 M77:60601 Type1 Inactive DFGin 6.1218 13.3386 ABAminus -125.47, 13.51 -148.05, 120.42 -113.28, 22.31 295.85, 71.04 -57.43, -24.9 in-in in 9.2508 Saltbr-in 2.8621 HRD-in -97.25, -49.49 72.22, 6.42 in-in-in SNCiii in-in ActLoopNT-in 2.9904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.86, 164.06 APE9-dihe-na 122.41, -161.87 APE8-dihe-in -119.99, 136.29 APE8-rot-in 295.68 APE67-dihe-in -63.27, -25.72 -47.9, -45.46 APE12-dist-in 8.1408 APE11-dist-in 11.2646 APE10-dist-in 5.7788 APE9-dist-in 3.3758 L50I,V124M,E128D,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.27 0.192 0.268 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gni Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1STCE P00517 16 351 351.0 STU:60351 Type1 Inactive DFGin 6.1254 14.6764 ABAminus -152.28, -21.25 -98.94, 113.28 -112.23, 27.12 284.07, 102.64 -65.61, -29.61 in-in in 9.1737 Saltbr-in 2.6077 HRD-out -84.15, -57.61 42.07, 55.99 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.84, 156.46 APE9-dihe-na 129.45, -158.0 APE8-dihe-in -121.73, 124.56 APE8-rot-in 292.46 APE67-dihe-in -75.12, -21.46 -28.7, -46.78 APE12-dist-in 8.3869 APE11-dist-in 11.1625 APE10-dist-in 5.8257 APE9-dist-in 4.4432 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.3 0.208 0.33 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1stc Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO2A P00517 8 351 351.0 15I:61351 Type1 Inactive DFGin 6.1445 13.7565 ABAminus -111.64, -15.7 -114.7, 103.29 -107.0, 15.63 291.73, 77.0 -53.95, -31.44 in-in in 8.9831 Saltbr-in 2.7087 HRD-in -83.31, -56.68 67.99, 8.34 in-in-in SNCiii in-in ActLoopNT-in 2.9313 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 157.34 APE9-dihe-na 124.98, -162.06 APE8-dihe-in -114.19, 137.15 APE8-rot-in 302.62 APE67-dihe-in -58.09, -28.32 -43.68, -52.1 APE12-dist-in 8.012 APE11-dist-in 11.4691 APE10-dist-in 5.8391 APE9-dist-in 3.6098 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.98 0.158 0.191 A 351.0 344.0 0 25 25 0 [[44, 298]] 1.0 3zo2 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO3A P00517 12 351 351.0 QNI:61351 Type1 Inactive DFGin 5.8139 14.5584 ABAminus -113.45, -3.91 -119.58, 103.74 -104.44, 16.56 281.0, 73.71 -59.51, -27.51 in-in in 9.1187 Saltbr-in 2.7878 HRD-in -88.87, -55.75 64.02, 12.24 in-in-in SNCiii in-in ActLoopNT-in 2.8636 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.07, 157.3 APE9-dihe-na 125.82, -155.48 APE8-dihe-in -117.69, 139.23 APE8-rot-in 297.95 APE67-dihe-in -57.23, -32.24 -46.12, -52.37 APE12-dist-in 7.9721 APE11-dist-in 11.3311 APE10-dist-in 5.7624 APE9-dist-in 3.6518 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.1 0.176 0.21 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 3zo3 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 5VI9A P00517 15 351 351.0 9D4:60401 Type1 Inactive DFGin 6.4135 14.639 ABAminus -108.08, -28.68 -104.39, 134.13 -134.73, 37.16 293.35, 85.38 -60.78, -29.79 in-out in 9.3856 Saltbr-out 3.754 HRD-in -77.99, -57.09 68.94, 10.33 out-in-in SNCoii in-in ActLoopNT-in 2.8473 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.52, 160.7 APE9-dihe-na 121.66, -160.6 APE8-dihe-in -114.63, 135.81 APE8-rot-in 302.32 APE67-dihe-in -61.89, -29.97 -46.88, -46.56 APE12-dist-in 8.0832 APE11-dist-in 11.498 APE10-dist-in 5.8264 APE9-dist-in 3.6359 None TPO198 TPO198 XRAY 1.95 0.209 0.256 A 351.0 307.0 4 25 25 0 [[44, 298]] 1.0 5vi9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 5VIBA P00517 19 351 351.0 9D1:60401 Type1 Inactive DFGin 6.6212 14.8324 ABAminus -107.11, -34.58 -98.31, 117.88 -117.47, 22.93 281.07, 85.16 -57.39, -18.74 in-in in 9.1872 Saltbr-in 3.5607 HRD-in -77.43, -53.28 63.56, 13.71 in-in-in SNCiii in-in ActLoopNT-in 2.8615 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.02, 160.82 APE9-dihe-na 122.63, -164.02 APE8-dihe-in -113.1, 131.73 APE8-rot-in 301.25 APE67-dihe-in -62.36, -27.21 -42.7, -49.96 APE12-dist-in 7.9483 APE11-dist-in 11.4159 APE10-dist-in 5.7564 APE9-dist-in 3.504 None TPO198 TPO198 XRAY 2.37 0.215 0.276 A 351.0 309.0 0 25 25 0 [[44, 298]] 1.0 5vib Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SZMB P00517 15 351 351.0 BI4:60351 Type1 Inactive DFGin 6.9164 16.0168 ABAminus -124.67, -37.03 -119.38, 110.7 -112.86, 23.01 290.52, 94.06 -59.96, -45.74 out-out out 10.6181 Saltbr-out 4.666 HRD-in -70.48, -44.14 31.9, 37.49 out-in-in SNCoii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.49, 166.21 APE9-dihe-na 109.44, 164.47 APE8-dihe-in -71.29, 133.53 APE8-rot-in 294.81 APE67-dihe-in -63.33, -24.2 -45.0, -46.86 APE12-dist-in 8.346 APE11-dist-in 11.522 APE10-dist-in 5.9849 APE9-dist-in 4.4453 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 B 350.0 323.0 0 25 25 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4AXAA P00517 15 351 351.0 RKD:61351 Type1 Inactive DFGin 6.203 13.8956 ABAminus -121.83, -29.08 -102.06, 117.48 -118.59, 24.36 279.49, 73.66 -60.99, -27.08 in-in in 8.7606 Saltbr-in 3.0068 HRD-in -91.45, -56.33 70.15, 3.62 in-in-in SNCiii in-in ActLoopNT-in 2.8879 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.21, 158.94 APE9-dihe-na 126.47, -155.87 APE8-dihe-in -119.74, 130.42 APE8-rot-in 299.77 APE67-dihe-in -59.64, -26.03 -40.97, -51.19 APE12-dist-in 7.9966 APE11-dist-in 11.4177 APE10-dist-in 5.8548 APE9-dist-in 3.7051 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.216 0.256 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4axa Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C34A P00517 11 351 351.0 STU:61351 Type1 Inactive DFGin 6.5166 14.8494 ABAminus -119.31, -40.44 -98.64, 112.68 -107.28, 23.29 283.36, 88.13 -59.12, -19.89 in-in in 8.8642 Saltbr-in 2.9854 HRD-in -78.06, -54.1 69.84, 7.38 in-in-in SNCiii in-in ActLoopNT-in 2.9107 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.66, 162.66 APE9-dihe-na 118.12, -166.39 APE8-dihe-in -111.07, 134.19 APE8-rot-in 303.77 APE67-dihe-in -56.72, -26.94 -46.04, -52.13 APE12-dist-in 8.3983 APE11-dist-in 11.4581 APE10-dist-in 5.7648 APE9-dist-in 3.4077 F55Y,M121L,V124L,L174M,Q182K SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.78 0.18 0.214 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 4c34 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C37A P00517 14 351 351.0 Z21:61351 Type1 Inactive DFGin 6.2618 14.2841 ABAminus -113.24, -47.75 -78.1, 110.9 -112.08, 25.76 272.69, 64.65 -57.89, -26.17 in-in in 8.7279 Saltbr-in 2.7412 HRD-in -81.42, -53.5 70.95, 1.92 in-in-in SNCiii in-in ActLoopNT-in 2.9412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.71, 160.19 APE9-dihe-na 127.27, -162.5 APE8-dihe-in -118.08, 133.43 APE8-rot-in 300.5 APE67-dihe-in -57.54, -26.87 -42.89, -53.17 APE12-dist-in 8.1544 APE11-dist-in 11.5086 APE10-dist-in 5.8833 APE9-dist-in 3.537 F55Y,M121L,V124L,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.157 0.179 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4c37 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNHA P00517 11 351 351.0 H52:60501,H52:60502 Type1,Allosteric Inactive DFGin 5.7262 14.706 ABAminus -128.79, 15.58 -151.1, 122.77 -119.76, 23.12 270.41, 63.78 -48.67, -39.31 in-in in 9.333 Saltbr-in 2.8243 HRD-in -85.53, -55.44 74.29, 10.02 in-in-in SNCiii in-in ActLoopNT-in 2.9565 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.69, 165.93 APE9-dihe-na 124.87, -164.72 APE8-dihe-in -119.96, 131.77 APE8-rot-in 295.2 APE67-dihe-in -55.53, -26.21 -49.22, -48.81 APE12-dist-in 8.1711 APE11-dist-in 11.3893 APE10-dist-in 5.8788 APE9-dist-in 3.4654 L50I,V124M,E128D,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.05 0.198 0.256 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gnh Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3AG9A P00517 15 351 351.0 No_ligand No_ligand Inactive DFGin 7.051 16.1774 BLAminus -121.67, 168.31 69.6, 87.4 -105.16, 26.26 286.68, 81.88 -58.4, -43.3 out-out out 10.486 Saltbr-out 4.7632 HRD-in -75.01, -50.0 50.19, 29.04 out-in-in SNCoii in-in ActLoopNT-in 2.8564 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.66, 167.28 APE9-dihe-na 97.3, 169.91 APE8-dihe-in -87.06, 128.77 APE8-rot-in 296.19 APE67-dihe-in -53.54, -29.25 -42.73, -48.49 APE12-dist-in 8.336 APE11-dist-in 11.2386 APE10-dist-in 5.7464 APE9-dist-in 4.3081 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.23 0.246 A 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3ag9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9FQRXT P00517 26 351 351.0 No_ligand No_ligand Inactive DFGin 7.5042 15.4719 BLAminus -120.43, -175.35 59.39, 66.35 -90.0, 32.7 274.65, 67.61 -64.07, -27.17 in-out in 8.66 Saltbr-out 4.4575 HRD-in -81.78, -57.62 51.32, 20.96 out-in-in SNCoii in-in ActLoopNT-in 3.2154 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.53, 169.85 APE9-dihe-na 132.17, 174.57 APE8-dihe-in -89.75, 132.06 APE8-rot-in 314.38 APE67-dihe-in -73.91, -30.73 -62.64, -19.12 APE12-dist-in 8.4981 APE11-dist-in 10.7604 APE10-dist-in 6.0224 APE9-dist-in 4.8414 None None None EM 5.0 999.0 999.0 Xt 351.0 294.0 0 25 25 0 [[44, 298]] 1.0 9fqr Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C35A P00517 11 351 351.0 NU3:61351 Type1.5_Back Inactive DFGin 5.96 15.1175 None -103.23, -88.31 -54.39, 108.88 -97.56, 11.02 265.67, 64.27 -54.79, -37.29 in-in in 9.1847 Saltbr-in 2.7744 HRD-in -78.97, -53.39 72.53, 0.25 in-in-in SNCiii in-in ActLoopNT-in 2.8688 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.98, 158.62 APE9-dihe-na 121.3, -169.27 APE8-dihe-in -106.38, 130.41 APE8-rot-in 302.02 APE67-dihe-in -58.09, -26.56 -41.09, -54.15 APE12-dist-in 8.7429 APE11-dist-in 11.6126 APE10-dist-in 5.9626 APE9-dist-in 3.4271 F55Y,M121L,V124L,L174M,Q182K SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.19 0.186 0.24 A 351.0 341.0 0 25 25 0 [[44, 298]] 1.0 4c35 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW7G P00517 13 351 351.0 ANP:403 ATPlike Inactive None 999.0 999.0 None -155.4, -162.2 59.11, 63.62 -70.57, 12.19 999.0, 999.0 -65.51, -34.83 out-none out 10.9713 Saltbr-none 999.0 HRD-in -65.14, -55.26 50.7, 27.28 none-in-out SNCnio in-out ActLoopNT-in 2.5754 ActLoopCT-out nonTYR APEdihe_aaini APEdist_iiio APE10-dihe-na -166.96, 170.69 APE9-dihe-na 108.98, -156.8 APE8-dihe-in -102.79, 139.06 APE8-rot-none 999.0 APE67-dihe-in -58.63, -28.81 -67.98, -6.96 APE12-dist-in 9.2283 APE11-dist-in 10.2672 APE10-dist-in 6.4383 APE9-dist-out 6.202 None None None EM 6.0 999.0 999.0 G 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 9dw7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW4K P00517 13 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -155.5, -168.49 59.79, 60.87 -83.31, 16.99 999.0, 999.0 -58.46, -53.69 in-none in 9.8843 Saltbr-none 999.0 HRD-in -75.2, -40.09 55.77, 26.65 none-in-none SNCnin in-none ActLoopNT-in 2.6727 ActLoopCT-none nonTYR APEdihe_aaini APEdist_iiii APE10-dihe-na -174.21, -178.74 APE9-dihe-na 106.6, -165.51 APE8-dihe-in -76.59, 132.39 APE8-rot-none 999.0 APE67-dihe-in -65.14, -23.53 -62.01, -33.48 APE12-dist-in 9.2205 APE11-dist-in 11.7506 APE10-dist-in 7.9925 APE9-dist-in 5.2599 None None None EM 9.0 999.0 999.0 K 351.0 331.0 0 25 25 0 [[44, 298]] 1.0 9dw4 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW7K P00517 13 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -155.25, -168.9 60.19, 60.97 -83.26, 17.04 999.0, 999.0 -58.67, -53.39 in-none in 9.875 Saltbr-none 999.0 HRD-in -75.5, -40.23 55.96, 26.19 none-in-none SNCnin in-none ActLoopNT-in 2.684 ActLoopCT-none nonTYR APEdihe_aaini APEdist_iiii APE10-dihe-na -174.15, -178.86 APE9-dihe-na 106.51, -165.36 APE8-dihe-in -77.09, 132.58 APE8-rot-none 999.0 APE67-dihe-in -65.64, -23.21 -62.33, -33.03 APE12-dist-in 9.2221 APE11-dist-in 11.7466 APE10-dist-in 7.9705 APE9-dist-in 5.2537 None None None EM 6.0 999.0 999.0 K 351.0 331.0 0 25 25 0 [[44, 298]] 1.0 9dw7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW5G P00517 13 351 351.0 ANP:403 ATPlike None DFGin 7.3339 15.8767 BLAminus -126.22, -169.89 60.75, 61.77 -87.02, 21.16 273.51, 93.96 -63.0, -33.74 out-none out 10.2523 Saltbr-none 999.0 HRD-in -80.85, -56.62 73.43, -6.68 none-in-in SNCnii in-in ActLoopNT-in 2.7819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.11, -173.97 APE9-dihe-na 106.0, -157.25 APE8-dihe-in -108.29, 136.12 APE8-rot-in 326.0 APE67-dihe-in -63.46, -43.06 -59.57, -33.75 APE12-dist-in 9.1133 APE11-dist-in 11.9553 APE10-dist-in 6.8101 APE9-dist-in 4.5632 None TPO198 TPO198 EM 3.8 999.0 999.0 G 351.0 330.0 0 25 25 0 [[44, 298]] 1.0 9dw5 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW8G P00517 15 329 351.0 ANP:403 ATPlike None DFGin 6.0696 14.2353 BLAminus -131.43, -174.72 59.27, 66.66 -86.28, 33.46 293.19, 93.28 -61.23, -49.05 in-none in 9.9111 Saltbr-none 999.0 HRD-in -98.32, -49.71 57.42, 11.15 none-in-in SNCnii in-in ActLoopNT-in 2.9612 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.06, 160.73 APE9-dihe-na 123.3, -175.7 APE8-dihe-in -89.52, 132.72 APE8-rot-in 298.44 APE67-dihe-in -69.93, -27.98 -56.75, -38.6 APE12-dist-in 8.7001 APE11-dist-in 11.5933 APE10-dist-in 6.4109 APE9-dist-in 4.8026 None TPO198 TPO198 EM 3.5 999.0 999.0 G 351.0 309.0 0 25 25 0 [[44, 298]] 1.0 9dw8 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EM7A P25321 11 351 351.0 ADP:60403 ATPlike Active DFGin 5.924 14.3384 BLAminus -118.71, 173.1 68.53, 85.06 -96.18, 23.36 270.78, 55.34 -59.75, -28.55 in-in in 8.7405 Saltbr-in 2.7108 HRD-in -88.33, -53.93 74.88, 10.19 in-in-in SNCiii in-in ActLoopNT-in 2.9674 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.73, 159.92 APE9-dihe-na 127.98, -160.75 APE8-dihe-in -119.5, 137.47 APE8-rot-in 298.57 APE67-dihe-in -59.39, -22.73 -49.47, -50.59 APE12-dist-in 8.0499 APE11-dist-in 11.4294 APE10-dist-in 5.809 APE9-dist-in 3.6743 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.238 0.139 0.157 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6em7 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EMAA P25321 12 351 351.0 ATP:60401 ATPlike Active DFGin 6.8466 14.0282 BLAminus -121.3, 163.01 76.03, 95.19 -107.48, 29.41 285.05, 72.84 -63.27, -23.25 in-in in 8.5805 Saltbr-in 2.9123 HRD-in -88.06, -51.23 73.05, 9.34 in-in-in SNCiii in-in ActLoopNT-in 2.8434 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.85, 162.03 APE9-dihe-na 127.51, -167.2 APE8-dihe-in -113.51, 133.85 APE8-rot-in 299.54 APE67-dihe-in -58.99, -24.47 -49.7, -50.19 APE12-dist-in 8.208 APE11-dist-in 11.4336 APE10-dist-in 5.7768 APE9-dist-in 3.5854 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.88 0.184 0.213 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6ema Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ESAA P25321 11 351 351.0 AMP:60401 ATPlike Active DFGin 6.1394 14.3654 BLAminus -120.63, 169.73 70.22, 89.96 -100.72, 24.5 270.85, 56.09 -58.05, -28.66 in-in in 8.6912 Saltbr-in 2.8734 HRD-in -93.01, -53.86 73.79, 10.3 in-in-in SNCiii in-in ActLoopNT-in 2.9643 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.44, 160.95 APE9-dihe-na 124.73, -163.46 APE8-dihe-in -117.05, 136.25 APE8-rot-in 299.26 APE67-dihe-in -59.89, -22.61 -49.24, -49.61 APE12-dist-in 8.0912 APE11-dist-in 11.4994 APE10-dist-in 5.8224 APE9-dist-in 3.6604 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.307 0.132 0.147 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6esa Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y8CA P25321 13 351 351.0 ATP:60402 ATPlike Active DFGin 5.7272 14.3024 BLAminus -123.99, 172.57 69.5, 82.73 -92.15, 25.74 279.44, 63.0 -58.78, -31.82 in-in in 9.1661 Saltbr-in 2.6378 HRD-in -96.49, -52.39 69.1, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.8845 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.28, 160.42 APE9-dihe-na 122.78, -169.96 APE8-dihe-in -106.17, 134.07 APE8-rot-in 304.81 APE67-dihe-in -60.24, -22.7 -48.33, -48.43 APE12-dist-in 8.0442 APE11-dist-in 11.5168 APE10-dist-in 5.9394 APE9-dist-in 3.8952 None TPO198,SEP339 TPO198,SEP339 XRAY 1.76 0.162 0.19 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 6y8c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1NA P25321 1 351 351.0 8G8:60402 Allosteric Active DFGin 6.4141 14.3021 BLAminus -123.89, -172.22 60.93, 80.4 -92.44, 26.18 275.59, 66.61 -60.07, -25.93 in-in in 8.7465 Saltbr-in 3.033 HRD-in -89.37, -52.82 73.6, 7.6 in-in-in SNCiii in-in ActLoopNT-in 2.9227 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.19, 156.64 APE9-dihe-na 134.09, -162.2 APE8-dihe-in -112.34, 129.13 APE8-rot-in 298.42 APE67-dihe-in -61.33, -22.28 -43.88, -53.69 APE12-dist-in 8.451 APE11-dist-in 11.6981 APE10-dist-in 6.1521 APE9-dist-in 3.7784 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.405 0.154 0.179 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 5n1n Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3IA P25321 12 351 351.0 BJQ:60404 Allosteric Active DFGin 6.2036 14.3735 BLAminus -121.15, 165.89 72.6, 94.77 -102.91, 24.31 271.68, 55.3 -58.81, -29.64 in-in in 8.5664 Saltbr-in 2.9174 HRD-in -84.69, -52.32 69.36, 13.72 in-in-in SNCiii in-in ActLoopNT-in 2.9163 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.06, 170.9 APE9-dihe-na 117.62, -155.4 APE8-dihe-in -132.77, 134.35 APE8-rot-in 303.36 APE67-dihe-in -62.11, -19.9 -47.3, -51.17 APE12-dist-in 8.1248 APE11-dist-in 11.1999 APE10-dist-in 5.6654 APE9-dist-in 3.6237 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.14 0.134 0.151 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3i Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3KA P25321 12 351 351.0 GGB:60401 Allosteric Active DFGin 6.1849 14.34 BLAminus -124.6, 161.61 76.98, 90.66 -99.67, 25.29 272.38, 65.33 -61.96, -25.98 in-in in 8.6368 Saltbr-in 3.0012 HRD-in -87.33, -51.9 70.65, 14.42 in-in-in SNCiii in-in ActLoopNT-in 2.9472 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.91, 162.87 APE9-dihe-na 131.35, -156.18 APE8-dihe-in -123.66, 133.94 APE8-rot-in 296.91 APE67-dihe-in -59.29, -22.9 -47.8, -51.08 APE12-dist-in 8.1169 APE11-dist-in 11.1579 APE10-dist-in 5.6584 APE9-dist-in 3.7179 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.33 0.146 0.172 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3k Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Z08A P25321 14 351 351.0 NPO:60401 Allosteric Active DFGin 6.0045 14.3152 BLAminus -122.86, -172.56 56.32, 85.8 -96.13, 22.67 273.1, 62.96 -62.03, -25.78 in-in in 8.7081 Saltbr-in 2.5485 HRD-in -86.99, -51.51 69.72, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.9103 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.61, 168.88 APE9-dihe-na 120.32, -158.83 APE8-dihe-in -126.12, 135.53 APE8-rot-in 304.13 APE67-dihe-in -63.09, -19.11 -50.64, -46.8 APE12-dist-in 8.1729 APE11-dist-in 11.2225 APE10-dist-in 5.7126 APE9-dist-in 3.5871 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.49 0.163 0.185 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6z08 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE2A P25321 13 351 351.0 A1JE1:60504 Allosteric Active DFGin 6.9065 14.6005 BLAminus -130.51, -172.34 64.95, 64.92 -87.74, 25.39 275.14, 64.69 -64.84, -26.39 in-in in 8.9545 Saltbr-in 2.7115 HRD-in -89.39, -50.72 72.95, 14.8 in-in-in SNCiii in-in ActLoopNT-in 2.9921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.73, 162.53 APE9-dihe-na 125.67, -157.85 APE8-dihe-in -124.12, 131.82 APE8-rot-in 303.61 APE67-dihe-in -61.71, -21.87 -46.36, -49.79 APE12-dist-in 8.2745 APE11-dist-in 11.3295 APE10-dist-in 5.8612 APE9-dist-in 3.7356 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.68 0.209 0.233 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9re2 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REMA P25321 12 351 351.0 A1JEL:60401 Allosteric Active DFGin 6.4257 14.5409 BLAminus -124.03, 163.4 76.56, 89.18 -99.82, 25.59 271.66, 58.78 -64.22, -23.78 in-in in 8.6205 Saltbr-in 2.8774 HRD-in -87.63, -52.43 69.95, 13.38 in-in-in SNCiii in-in ActLoopNT-in 2.9373 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.48, 163.83 APE9-dihe-na 114.89, 177.74 APE8-dihe-in -94.85, 132.62 APE8-rot-in 300.61 APE67-dihe-in -61.62, -20.97 -47.15, -48.45 APE12-dist-in 8.263 APE11-dist-in 11.3978 APE10-dist-in 5.9326 APE9-dist-in 4.0207 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.43 0.158 0.173 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rem Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RESA P25321 12 351 351.0 A1JEG:60401 Allosteric Active DFGin 6.1727 14.8814 BLAminus -125.7, 167.74 69.23, 93.16 -97.77, 26.89 271.48, 59.73 -63.11, -29.76 in-in in 9.0438 Saltbr-in 2.7187 HRD-in -87.69, -51.87 66.23, 13.93 in-in-in SNCiii in-in ActLoopNT-in 2.9651 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.16, 154.7 APE9-dihe-na 118.02, 158.85 APE8-dihe-in -77.09, 138.71 APE8-rot-in 297.19 APE67-dihe-in -59.68, -23.56 -52.24, -44.23 APE12-dist-in 8.1974 APE11-dist-in 11.3307 APE10-dist-in 5.7869 APE9-dist-in 4.2474 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.196 0.211 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9res Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RETA P25321 13 351 351.0 A1JEF:60404 Allosteric Active DFGin 6.5025 14.9192 BLAminus -121.64, 161.02 79.66, 89.44 -97.28, 25.84 271.42, 57.67 -59.32, -29.98 in-in in 9.0584 Saltbr-in 2.6884 HRD-in -91.57, -50.28 65.7, 14.34 in-in-in SNCiii in-in ActLoopNT-in 2.9609 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.82, 155.57 APE9-dihe-na 119.38, 155.92 APE8-dihe-in -73.83, 138.5 APE8-rot-in 315.72 APE67-dihe-in -57.32, -25.4 -54.39, -42.36 APE12-dist-in 8.1859 APE11-dist-in 11.4021 APE10-dist-in 5.9522 APE9-dist-in 4.2407 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.75 0.193 0.227 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ret Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N37A P25321 1 351 351.0 8JT:60402,8JT:60403 Allosteric,Allosteric Active DFGin 6.6488 14.4854 BLAminus -123.92, -170.55 59.87, 72.4 -89.59, 22.41 275.2, 67.84 -61.07, -22.15 in-in in 8.6486 Saltbr-in 2.8873 HRD-in -90.3, -49.46 71.47, 2.69 in-in-in SNCiii in-in ActLoopNT-in 2.9099 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.56, 154.71 APE9-dihe-na 136.23, -163.83 APE8-dihe-in -107.21, 128.79 APE8-rot-in 298.22 APE67-dihe-in -60.14, -24.18 -42.74, -52.97 APE12-dist-in 8.5415 APE11-dist-in 11.9362 APE10-dist-in 6.3043 APE9-dist-in 3.975 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.589 0.145 0.167 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n37 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3TA P25321 12 351 351.0 8K2:60401,8K2:60402 Allosteric,Allosteric Active DFGin 6.2089 14.3858 BLAminus -125.21, 167.5 70.97, 90.28 -98.07, 24.21 271.06, 55.85 -60.14, -28.27 in-in in 8.5718 Saltbr-in 2.8524 HRD-in -84.98, -51.06 69.41, 14.03 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.94, 169.7 APE9-dihe-na 118.95, -153.57 APE8-dihe-in -135.51, 135.28 APE8-rot-in 302.46 APE67-dihe-in -63.12, -21.21 -48.68, -48.91 APE12-dist-in 8.1233 APE11-dist-in 11.2089 APE10-dist-in 5.6949 APE9-dist-in 3.706 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.209 0.14 0.157 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3t Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDZA P25321 12 351 351.0 A1JE9:60402,A1JE9:60403 Allosteric,Allosteric Active DFGin 6.37 14.6865 BLAminus -121.86, 166.99 72.88, 89.4 -99.69, 27.1 269.36, 64.25 -60.46, -30.34 in-in in 8.7723 Saltbr-in 2.9001 HRD-in -86.07, -51.02 68.52, 15.31 in-in-in SNCiii in-in ActLoopNT-in 3.0047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.16, 164.09 APE9-dihe-na 123.15, -172.2 APE8-dihe-in -104.62, 134.08 APE8-rot-in 309.64 APE67-dihe-in -61.1, -21.33 -52.23, -44.2 APE12-dist-in 8.2799 APE11-dist-in 11.4033 APE10-dist-in 5.8984 APE9-dist-in 3.9616 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.64 0.18 0.212 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rdz Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REEA P25321 13 351 351.0 A1JEW:60401,A1JEW:60403 Allosteric,Allosteric Active DFGin 6.286 14.26 BLAminus -124.23, 162.89 77.1, 88.42 -96.8, 24.55 273.02, 56.54 -61.31, -24.65 in-in in 8.4623 Saltbr-in 2.9112 HRD-in -83.83, -50.86 69.06, 13.49 in-in-in SNCiii in-in ActLoopNT-in 2.9147 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.82, 159.16 APE9-dihe-na 111.69, 168.82 APE8-dihe-in -86.75, 136.79 APE8-rot-in 296.84 APE67-dihe-in -63.43, -20.25 -47.42, -48.01 APE12-dist-in 8.1052 APE11-dist-in 11.1621 APE10-dist-in 5.684 APE9-dist-in 3.9569 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.34 0.157 0.167 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ree Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RELA P25321 12 351 351.0 D8V:60402,D8V:60403 Allosteric,Allosteric Active DFGin 6.4822 14.5671 BLAminus -123.01, 164.35 74.25, 89.59 -99.6, 28.07 272.56, 59.06 -67.42, -22.86 in-in in 8.6372 Saltbr-in 2.9197 HRD-in -86.71, -52.81 70.71, 15.02 in-in-in SNCiii in-in ActLoopNT-in 2.9775 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.1, 164.56 APE9-dihe-na 121.48, -172.32 APE8-dihe-in -106.43, 133.24 APE8-rot-in 301.52 APE67-dihe-in -61.15, -21.91 -46.09, -49.9 APE12-dist-in 8.3488 APE11-dist-in 11.4781 APE10-dist-in 6.0184 APE9-dist-in 3.9426 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.158 0.177 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rel Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REPA P25321 12 351 351.0 A1JFA:60402,A1JFA:60403,A1JFA:60404 Allosteric,Allosteric,Type1 Active DFGin 6.3781 14.529 BLAminus -120.08, 167.91 74.1, 88.72 -97.52, 23.51 270.46, 58.88 -60.74, -26.54 in-in in 8.6885 Saltbr-in 2.9313 HRD-in -87.33, -51.34 69.9, 12.31 in-in-in SNCiii in-in ActLoopNT-in 2.9651 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.19, 163.24 APE9-dihe-na 117.23, 172.54 APE8-dihe-in -96.3, 137.81 APE8-rot-in 314.32 APE67-dihe-in -63.77, -21.88 -47.87, -48.37 APE12-dist-in 8.1899 APE11-dist-in 11.3609 APE10-dist-in 5.8512 APE9-dist-in 4.0301 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.44 0.157 0.181 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rep Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REOA P25321 13 351 351.0 A1JEJ:60401,A1JEJ:60402,A1JEJ:60403,A1JEJ:60404,A1JEJ:60405 Allosteric,Allosteric,Type1,Type1,Allosteric Active DFGin 6.3145 14.3168 BLAminus -116.84, 173.33 67.79, 85.36 -98.4, 23.6 274.95, 63.33 -57.17, -27.66 in-in in 8.6623 Saltbr-in 2.7528 HRD-in -87.13, -54.16 72.26, 11.26 in-in-in SNCiii in-in ActLoopNT-in 2.8988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.54, 160.85 APE9-dihe-na 115.26, -179.78 APE8-dihe-in -98.51, 134.9 APE8-rot-in 302.45 APE67-dihe-in -59.75, -23.89 -49.35, -45.76 APE12-dist-in 8.1175 APE11-dist-in 11.2447 APE10-dist-in 5.7372 APE9-dist-in 3.9737 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.45 0.152 0.175 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9reo Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7AXVA P25321 1 351 351.0 S95:60401,S95:60402 Allosteric,Type1 Active DFGin 6.5443 14.3191 BLAminus -124.64, 165.56 73.97, 89.92 -106.44, 27.23 290.62, 82.1 -63.98, -25.18 in-in in 9.5168 Saltbr-in 3.1989 HRD-in -92.54, -54.57 72.35, 9.82 in-in-in SNCiii in-in ActLoopNT-in 2.8895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.49, 161.0 APE9-dihe-na 125.29, -162.18 APE8-dihe-in -119.59, 130.9 APE8-rot-in 299.34 APE67-dihe-in -56.02, -27.32 -46.45, -51.94 APE12-dist-in 8.0271 APE11-dist-in 11.475 APE10-dist-in 5.9545 APE9-dist-in 3.8706 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.79 0.2 0.231 A 353.0 344.0 3 25 25 0 [[44, 298]] 1.0 7axv Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE3A P25321 12 351 351.0 A1JE0:60805,A1JE0:60807 Allosteric,Type1 Active DFGin 6.4607 14.6641 BLAminus -120.32, 164.28 77.93, 91.61 -101.65, 25.38 271.39, 59.52 -61.95, -25.41 in-in in 8.7616 Saltbr-in 2.8901 HRD-in -88.06, -50.21 67.37, 14.1 in-in-in SNCiii in-in ActLoopNT-in 3.0126 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.15, 155.76 APE9-dihe-na 126.49, 178.95 APE8-dihe-in -96.29, 137.07 APE8-rot-in 306.5 APE67-dihe-in -59.04, -22.36 -49.62, -47.63 APE12-dist-in 8.2317 APE11-dist-in 11.4892 APE10-dist-in 5.9401 APE9-dist-in 4.1876 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.57 0.185 0.213 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3OA P25321 14 351 351.0 5AO:60403,5AO:60404,5AO:60405 Allosteric,Type1,Allosteric Active DFGin 6.2389 14.3632 BLAminus -124.74, 162.74 72.04, 91.7 -99.25, 24.26 270.68, 57.41 -61.29, -25.0 in-in in 8.56 Saltbr-in 2.8625 HRD-in -84.17, -53.21 70.22, 13.77 in-in-in SNCiii in-in ActLoopNT-in 2.9147 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.1, 167.24 APE9-dihe-na 125.28, -162.2 APE8-dihe-in -119.97, 133.57 APE8-rot-in 304.74 APE67-dihe-in -63.04, -20.65 -49.48, -46.76 APE12-dist-in 8.1083 APE11-dist-in 11.3568 APE10-dist-in 5.8435 APE9-dist-in 3.7337 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.32 0.135 0.158 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 5n3o Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 4WIHA P25321 1 351 351.0 No_ligand No_ligand Active DFGin 6.1605 14.2123 BLAminus -123.3, 174.61 65.19, 98.78 -108.79, 24.75 270.23, 57.89 -53.46, -27.17 in-in in 8.5468 Saltbr-in 2.4651 HRD-in -89.62, -51.49 71.45, 14.2 in-in-in SNCiii in-in ActLoopNT-in 2.9097 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.02, 163.3 APE9-dihe-na 130.98, -159.02 APE8-dihe-in -120.59, 129.78 APE8-rot-in 297.97 APE67-dihe-in -60.37, -23.23 -43.98, -53.0 APE12-dist-in 8.282 APE11-dist-in 11.5665 APE10-dist-in 6.0683 APE9-dist-in 3.608 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.139 0.178 0.191 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 4wih Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0UA P25321 1 351 351.0 No_ligand No_ligand Active DFGin 6.6174 14.7612 BLAminus -120.76, 157.18 78.21, 97.74 -104.6, 26.7 278.38, 71.52 -59.1, -27.35 in-in in 8.7241 Saltbr-in 3.0199 HRD-in -84.58, -52.68 70.27, 15.16 in-in-in SNCiii in-in ActLoopNT-in 2.9195 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.97, 158.74 APE9-dihe-na 125.58, -159.96 APE8-dihe-in -115.4, 133.22 APE8-rot-in 298.31 APE67-dihe-in -57.6, -25.41 -46.26, -52.75 APE12-dist-in 8.2464 APE11-dist-in 11.5188 APE10-dist-in 5.8578 APE9-dist-in 3.5802 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.667 0.154 0.189 A 353.0 347.0 4 25 25 0 [[44, 298]] 1.0 5m0u Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3MA P25321 12 351 351.0 No_ligand No_ligand Active DFGin 6.1801 14.3543 BLAminus -123.75, 157.21 80.77, 89.43 -98.44, 24.43 270.49, 59.51 -61.84, -26.83 in-in in 8.534 Saltbr-in 2.9772 HRD-in -86.44, -51.88 69.6, 14.02 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.37, 162.31 APE9-dihe-na 130.48, -156.87 APE8-dihe-in -124.49, 134.84 APE8-rot-in 297.05 APE67-dihe-in -63.46, -20.29 -50.29, -48.15 APE12-dist-in 8.1166 APE11-dist-in 11.173 APE10-dist-in 5.6762 APE9-dist-in 3.7229 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.229 0.14 0.164 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3m Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EH0A P25321 13 351 351.0 No_ligand No_ligand Active DFGin 6.1366 14.4089 BLAminus -122.27, 162.09 77.35, 95.81 -104.93, 26.7 272.05, 59.25 -60.27, -24.52 in-in in 8.6935 Saltbr-in 3.0251 HRD-in -85.16, -52.91 72.1, 11.56 in-in-in SNCiii in-in ActLoopNT-in 2.9063 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.28, 161.12 APE9-dihe-na 111.18, 173.11 APE8-dihe-in -92.76, 136.72 APE8-rot-in 292.07 APE67-dihe-in -59.99, -23.63 -47.46, -47.75 APE12-dist-in 8.1156 APE11-dist-in 11.2721 APE10-dist-in 5.7898 APE9-dist-in 3.9986 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.49 0.15 0.186 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 6eh0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Z44A P25321 14 351 351.0 No_ligand No_ligand Active DFGin 6.2102 14.4374 BLAminus -128.58, 169.86 73.52, 88.4 -98.57, 23.88 272.06, 58.82 -60.44, -27.11 in-in in 8.6237 Saltbr-in 2.8632 HRD-in -87.15, -51.73 71.04, 12.68 in-in-in SNCiii in-in ActLoopNT-in 2.8909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.29, 164.35 APE9-dihe-na 123.85, -163.53 APE8-dihe-in -119.09, 134.17 APE8-rot-in 300.66 APE67-dihe-in -64.2, -18.89 -49.41, -47.47 APE12-dist-in 8.1442 APE11-dist-in 11.2003 APE10-dist-in 5.6806 APE9-dist-in 3.7234 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.146 0.174 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6z44 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6F14A P25321 9 351 351.0 ISQ:60401 Type1 Active DFGin 6.0674 14.2043 BLAminus -122.05, 170.08 68.01, 92.59 -99.92, 26.02 274.99, 58.24 -62.07, -22.2 in-in in 8.9109 Saltbr-in 2.7518 HRD-in -91.1, -51.98 71.1, 14.05 in-in-in SNCiii in-in ActLoopNT-in 2.9748 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.36, 162.19 APE9-dihe-na 130.64, -162.57 APE8-dihe-in -117.18, 137.06 APE8-rot-in 303.3 APE67-dihe-in -57.84, -25.17 -52.4, -48.63 APE12-dist-in 8.0928 APE11-dist-in 11.4976 APE10-dist-in 5.9364 APE9-dist-in 3.6185 None TPO198,SEP339 TPO198,SEP339 XRAY 1.867 0.176 0.209 A 351.0 339.0 4 25 25 0 [[44, 298]] 1.0 6f14 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCQA P25321 1 351 351.0 6TV:60401 Type1 Active DFGin 6.8807 14.7391 BLAminus -123.17, 161.48 80.79, 88.7 -100.7, 25.58 283.7, 73.56 -69.47, -15.21 in-in in 8.6294 Saltbr-in 2.7912 HRD-in -83.86, -57.44 75.35, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.8709 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.46, 161.6 APE9-dihe-na 121.64, -167.7 APE8-dihe-in -108.93, 132.05 APE8-rot-in 299.43 APE67-dihe-in -61.12, -21.5 -46.6, -52.1 APE12-dist-in 8.2733 APE11-dist-in 11.3689 APE10-dist-in 5.7633 APE9-dist-in 3.5302 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.423 0.143 0.171 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcq Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0BA P25321 1 351 351.0 IQU:60401 Type1 Active DFGin 6.8813 14.7187 BLAminus -123.22, 164.24 73.76, 92.16 -102.04, 24.7 282.81, 75.1 -69.51, -12.32 in-in in 8.6655 Saltbr-in 2.839 HRD-in -84.13, -55.97 72.34, 13.7 in-in-in SNCiii in-in ActLoopNT-in 2.9176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.89, 160.72 APE9-dihe-na 119.74, -166.42 APE8-dihe-in -108.36, 130.85 APE8-rot-in 297.35 APE67-dihe-in -58.39, -24.4 -45.39, -52.68 APE12-dist-in 8.3169 APE11-dist-in 11.472 APE10-dist-in 5.863 APE9-dist-in 3.5368 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.506 0.133 0.159 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m0b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0CA P25321 14 351 351.0 7CB:60401 Type1 Active DFGin 5.9263 14.302 BLAminus -122.77, 175.08 63.79, 89.7 -99.98, 24.75 269.77, 55.83 -60.58, -26.96 in-in in 8.883 Saltbr-in 2.7611 HRD-in -96.62, -51.29 71.36, 13.59 in-in-in SNCiii in-in ActLoopNT-in 2.8962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.73, 162.77 APE9-dihe-na 130.88, -158.33 APE8-dihe-in -121.3, 136.16 APE8-rot-in 298.59 APE67-dihe-in -56.27, -24.31 -50.24, -49.98 APE12-dist-in 8.0159 APE11-dist-in 11.4298 APE10-dist-in 5.8568 APE9-dist-in 3.4765 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.734 0.174 0.2 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 5m0c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1EA P25321 1 351 351.0 9NT:60402 Type1 Active DFGin 6.2704 14.3856 BLAminus -116.94, 171.55 65.1, 106.63 -111.97, 27.73 271.53, 67.85 -63.72, -19.43 in-in in 8.7187 Saltbr-in 3.0209 HRD-in -91.36, -50.95 71.95, 7.79 in-in-in SNCiii in-in ActLoopNT-in 2.9009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.29, 159.66 APE9-dihe-na 132.29, -165.21 APE8-dihe-in -107.94, 127.91 APE8-rot-in 298.37 APE67-dihe-in -61.69, -23.48 -42.18, -52.19 APE12-dist-in 8.4675 APE11-dist-in 11.8233 APE10-dist-in 6.2637 APE9-dist-in 3.8458 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.529 0.149 0.174 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 5n1e Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1LA P25321 1 351 351.0 47V:60401 Type1 Active DFGin 6.396 14.532 BLAminus -123.64, 176.95 64.79, 82.82 -93.93, 24.8 274.07, 62.39 -62.6, -22.74 in-in in 8.8226 Saltbr-in 2.8025 HRD-in -94.52, -51.37 72.06, 10.31 in-in-in SNCiii in-in ActLoopNT-in 2.9192 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.16, 159.72 APE9-dihe-na 135.69, -163.33 APE8-dihe-in -113.56, 130.78 APE8-rot-in 299.09 APE67-dihe-in -60.45, -22.24 -43.7, -53.93 APE12-dist-in 8.2602 APE11-dist-in 11.6708 APE10-dist-in 6.1348 APE9-dist-in 3.8023 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.489 0.144 0.175 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n1l Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1MA P25321 1 351 351.0 BJK:60403 Type1 Active DFGin 6.4585 14.0437 BLAminus -123.41, 174.5 65.19, 101.23 -111.22, 25.09 279.28, 68.63 -59.82, -25.41 in-in in 8.6556 Saltbr-in 3.1051 HRD-in -94.95, -53.6 73.25, 11.15 in-in-in SNCiii in-in ActLoopNT-in 2.9046 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.71, 160.83 APE9-dihe-na 133.31, -164.27 APE8-dihe-in -112.16, 130.84 APE8-rot-in 297.89 APE67-dihe-in -59.92, -22.11 -42.38, -54.95 APE12-dist-in 8.3624 APE11-dist-in 11.6972 APE10-dist-in 6.1444 APE9-dist-in 3.7347 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.436 0.153 0.17 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n1m Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1OA P25321 8 351 351.0 8GB:60402 Type1 Active DFGin 6.3495 14.2152 BLAminus -117.96, -179.86 55.4, 87.26 -94.87, 24.62 276.45, 65.75 -58.72, -27.08 in-in in 8.7307 Saltbr-in 2.9049 HRD-in -90.93, -54.44 74.01, 7.31 in-in-in SNCiii in-in ActLoopNT-in 2.8232 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.08, 159.92 APE9-dihe-na 129.4, -159.5 APE8-dihe-in -111.79, 132.44 APE8-rot-in 298.64 APE67-dihe-in -59.59, -24.34 -46.73, -53.55 APE12-dist-in 8.262 APE11-dist-in 11.7101 APE10-dist-in 6.159 APE9-dist-in 3.7466 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.8 0.172 0.191 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1o Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N33A P25321 1 351 351.0 8JW:60401 Type1 Active DFGin 6.5966 14.3444 BLAminus -124.76, 172.62 66.0, 85.95 -97.34, 23.47 278.51, 67.69 -61.06, -25.74 in-in in 8.6169 Saltbr-in 2.8295 HRD-in -95.51, -52.3 69.58, 12.9 in-in-in SNCiii in-in ActLoopNT-in 2.9142 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.48, 158.46 APE9-dihe-na 134.35, -163.32 APE8-dihe-in -113.73, 130.26 APE8-rot-in 298.83 APE67-dihe-in -60.31, -22.81 -43.61, -54.33 APE12-dist-in 8.2362 APE11-dist-in 11.6201 APE10-dist-in 6.0809 APE9-dist-in 3.77 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.434 0.151 0.174 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n33 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N36A P25321 1 351 351.0 F05:60402 Type1 Active DFGin 6.5556 14.4334 BLAminus -119.92, -178.94 65.61, 75.08 -89.84, 25.76 275.95, 67.66 -63.27, -22.33 in-in in 8.7237 Saltbr-in 2.8129 HRD-in -93.71, -55.54 73.48, 11.23 in-in-in SNCiii in-in ActLoopNT-in 2.9179 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 158.13 APE9-dihe-na 133.34, -160.6 APE8-dihe-in -112.55, 130.07 APE8-rot-in 300.31 APE67-dihe-in -59.23, -24.07 -46.06, -53.12 APE12-dist-in 8.5382 APE11-dist-in 11.8304 APE10-dist-in 6.244 APE9-dist-in 3.8446 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.15 0.186 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n36 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N39A P25321 1 351 351.0 8LZ:60401 Type1 Active DFGin 6.447 14.1735 BLAminus -115.61, 178.64 62.65, 78.33 -93.23, 24.2 279.01, 65.77 -60.59, -24.07 in-in in 8.6058 Saltbr-in 2.9559 HRD-in -92.08, -52.71 73.17, 11.28 in-in-in SNCiii in-in ActLoopNT-in 2.9039 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.98, 161.14 APE9-dihe-na 131.91, -164.98 APE8-dihe-in -111.15, 130.71 APE8-rot-in 297.72 APE67-dihe-in -61.9, -21.74 -44.77, -52.6 APE12-dist-in 8.3392 APE11-dist-in 11.723 APE10-dist-in 6.1957 APE9-dist-in 3.7478 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.45 0.146 0.169 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n39 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3AA P25321 1 351 351.0 46P:60404 Type1 Active DFGin 6.2347 14.3651 BLAminus -119.17, -176.19 62.26, 81.42 -92.16, 24.71 273.8, 62.92 -62.87, -20.2 in-in in 8.749 Saltbr-in 2.7586 HRD-in -88.58, -51.45 73.7, 4.67 in-in-in SNCiii in-in ActLoopNT-in 2.9097 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.23, 158.77 APE9-dihe-na 132.44, -163.77 APE8-dihe-in -109.48, 129.54 APE8-rot-in 298.98 APE67-dihe-in -60.34, -22.78 -43.75, -54.33 APE12-dist-in 8.4518 APE11-dist-in 11.8624 APE10-dist-in 6.299 APE9-dist-in 3.8633 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.404 0.162 0.184 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5n3a Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3BA P25321 5 351 351.0 BJN:60402 Type1 Active DFGin 6.5927 14.4491 BLAminus -127.99, -176.28 55.77, 87.43 -96.19, 25.66 273.47, 67.97 -63.99, -23.38 in-in in 8.7554 Saltbr-in 2.8962 HRD-in -88.77, -50.71 72.06, 10.59 in-in-in SNCiii in-in ActLoopNT-in 2.9448 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.08, 159.78 APE9-dihe-na 131.61, -163.96 APE8-dihe-in -108.68, 131.24 APE8-rot-in 297.72 APE67-dihe-in -59.88, -25.39 -45.07, -52.54 APE12-dist-in 8.4797 APE11-dist-in 11.8507 APE10-dist-in 6.2466 APE9-dist-in 3.8182 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.64 0.169 0.19 A 353.0 346.0 0 25 25 0 [[44, 298]] 1.0 5n3b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3CA P25321 1 351 351.0 8M2:60401 Type1 Active DFGin 6.4695 14.5593 BLAminus -119.65, -170.8 58.89, 76.61 -92.51, 23.35 273.34, 68.51 -61.87, -22.49 in-in in 8.8718 Saltbr-in 2.5903 HRD-in -86.05, -52.6 72.82, 4.64 in-in-in SNCiii in-in ActLoopNT-in 2.9083 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.17, 154.54 APE9-dihe-na 137.81, -166.64 APE8-dihe-in -107.38, 129.58 APE8-rot-in 301.23 APE67-dihe-in -60.59, -21.91 -48.15, -49.13 APE12-dist-in 8.4988 APE11-dist-in 11.881 APE10-dist-in 6.313 APE9-dist-in 3.9442 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.772 0.179 0.196 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 5n3c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3EA P25321 1 351 351.0 46L:60401 Type1 Active DFGin 6.3638 14.5063 BLAminus -127.71, 175.81 62.83, 90.97 -100.32, 25.03 271.8, 65.14 -62.05, -22.27 in-in in 8.7408 Saltbr-in 2.7088 HRD-in -91.8, -51.14 70.51, 10.68 in-in-in SNCiii in-in ActLoopNT-in 2.9031 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.84, 159.06 APE9-dihe-na 132.58, -164.21 APE8-dihe-in -109.56, 127.56 APE8-rot-in 297.32 APE67-dihe-in -58.87, -22.91 -42.91, -53.84 APE12-dist-in 8.3507 APE11-dist-in 11.7235 APE10-dist-in 6.2032 APE9-dist-in 3.8527 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.529 0.157 0.185 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 5n3e Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3HA P25321 12 351 351.0 NCA:60401 Type1 Active DFGin 6.1319 14.3906 BLAminus -122.6, -180.0 63.23, 82.13 -91.36, 22.79 272.99, 56.19 -60.14, -26.14 in-in in 8.7514 Saltbr-in 2.6589 HRD-in -87.2, -51.58 72.04, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.9341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.37, 162.08 APE9-dihe-na 126.78, -160.11 APE8-dihe-in -123.99, 135.79 APE8-rot-in 303.45 APE67-dihe-in -61.89, -20.7 -47.97, -49.67 APE12-dist-in 8.1151 APE11-dist-in 11.2119 APE10-dist-in 5.6695 APE9-dist-in 3.6645 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.36 0.146 0.174 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3h Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3LA P25321 12 351 351.0 E5E:60403 Type1 Active DFGin 6.2595 14.3638 BLAminus -110.0, -170.99 60.26, 70.6 -90.47, 19.96 272.32, 58.23 -61.45, -24.06 in-in in 8.5405 Saltbr-in 2.6938 HRD-in -90.35, -53.09 72.54, 14.7 in-in-in SNCiii in-in ActLoopNT-in 2.9233 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.08, 164.02 APE9-dihe-na 125.78, -157.28 APE8-dihe-in -125.93, 133.76 APE8-rot-in 301.3 APE67-dihe-in -63.07, -21.0 -46.88, -49.04 APE12-dist-in 8.0924 APE11-dist-in 11.2426 APE10-dist-in 5.7077 APE9-dist-in 3.6875 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.38 0.131 0.16 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3l Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3PA P25321 13 351 351.0 5H1:60403 Type1 Active DFGin 6.2436 14.5023 BLAminus -127.2, 167.3 74.22, 87.87 -97.57, 26.23 270.81, 60.43 -61.56, -25.66 in-in in 8.7311 Saltbr-in 2.7657 HRD-in -85.65, -51.7 69.95, 15.28 in-in-in SNCiii in-in ActLoopNT-in 2.9111 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.51, 162.3 APE9-dihe-na 120.29, -172.77 APE8-dihe-in -106.79, 135.49 APE8-rot-in 306.73 APE67-dihe-in -58.76, -22.92 -47.58, -49.08 APE12-dist-in 8.0501 APE11-dist-in 11.1792 APE10-dist-in 5.6741 APE9-dist-in 3.8219 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.159 0.181 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5n3p Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N7PA P25321 1 351 351.0 E9Q:60401 Type1 Active DFGin 6.2715 14.2377 BLAminus -126.92, 176.32 67.6, 84.98 -97.07, 24.3 276.23, 67.65 -61.77, -20.94 in-in in 8.7682 Saltbr-in 2.9318 HRD-in -90.6, -51.66 69.11, 10.85 in-in-in SNCiii in-in ActLoopNT-in 2.891 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.85, 157.28 APE9-dihe-na 137.17, -163.84 APE8-dihe-in -109.53, 129.55 APE8-rot-in 298.93 APE67-dihe-in -61.19, -22.41 -45.09, -51.76 APE12-dist-in 8.4123 APE11-dist-in 11.794 APE10-dist-in 6.2631 APE9-dist-in 3.8866 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.501 0.161 0.186 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5n7p Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N7UA P25321 1 351 351.0 8PQ:60402 Type1 Active DFGin 6.205 14.2991 BLAminus -120.54, 174.37 71.79, 80.65 -93.18, 24.34 271.72, 64.53 -61.67, -22.3 in-in in 8.6689 Saltbr-in 2.7302 HRD-in -88.01, -52.02 72.42, 9.42 in-in-in SNCiii in-in ActLoopNT-in 2.9076 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.34, 159.87 APE9-dihe-na 134.15, -161.5 APE8-dihe-in -113.47, 128.55 APE8-rot-in 298.53 APE67-dihe-in -62.45, -22.0 -41.16, -54.39 APE12-dist-in 8.4156 APE11-dist-in 11.6964 APE10-dist-in 6.1531 APE9-dist-in 3.7318 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.371 0.162 0.177 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5n7u Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EM2A P25321 12 351 351.0 M77:60401 Type1 Active DFGin 6.0983 14.5142 BLAminus -119.73, 168.43 71.45, 87.62 -96.71, 20.34 273.03, 58.25 -60.57, -24.08 in-in in 8.84 Saltbr-in 2.6697 HRD-in -89.33, -54.43 71.02, 10.57 in-in-in SNCiii in-in ActLoopNT-in 2.9443 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.33, 158.5 APE9-dihe-na 116.31, 173.93 APE8-dihe-in -92.1, 134.84 APE8-rot-in 313.8 APE67-dihe-in -63.32, -22.08 -46.46, -47.85 APE12-dist-in 8.0646 APE11-dist-in 11.2814 APE10-dist-in 5.8035 APE9-dist-in 4.0387 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.3 0.133 0.152 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6em2 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPSA P25321 14 351 351.0 LR5:60403 Type1 Active DFGin 6.2417 14.3836 BLAminus -118.18, 155.69 80.72, 97.49 -102.89, 27.66 269.68, 53.66 -61.81, -26.65 in-in in 8.4713 Saltbr-in 2.769 HRD-in -87.72, -49.97 68.25, 13.7 in-in-in SNCiii in-in ActLoopNT-in 2.9052 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.63, 162.08 APE9-dihe-na 121.79, -175.33 APE8-dihe-in -105.81, 135.65 APE8-rot-in 306.18 APE67-dihe-in -63.55, -22.05 -51.22, -42.77 APE12-dist-in 8.112 APE11-dist-in 11.235 APE10-dist-in 5.7263 APE9-dist-in 3.9626 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.65 0.188 0.223 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6sps Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPYA P25321 14 351 351.0 LR8:60401 Type1 Active DFGin 6.2185 14.4051 BLAminus -123.39, 156.64 76.95, 93.24 -100.34, 25.16 268.44, 60.17 -60.59, -28.29 in-in in 8.5574 Saltbr-in 2.8857 HRD-in -87.4, -50.43 70.53, 14.04 in-in-in SNCiii in-in ActLoopNT-in 2.9355 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.4, 165.8 APE9-dihe-na 119.26, -168.59 APE8-dihe-in -114.24, 137.53 APE8-rot-in 310.43 APE67-dihe-in -58.09, -22.25 -52.05, -47.82 APE12-dist-in 8.0826 APE11-dist-in 11.1688 APE10-dist-in 5.6662 APE9-dist-in 3.7027 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.6 0.162 0.182 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6spy Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SQ1A P25321 14 351 351.0 LRT:60403 Type1 Active DFGin 6.2159 14.2505 BLAminus -121.79, 172.1 69.1, 85.08 -99.08, 24.56 277.81, 66.67 -63.84, -22.93 in-in in 8.6518 Saltbr-in 2.6996 HRD-in -89.13, -55.11 71.03, 9.14 in-in-in SNCiii in-in ActLoopNT-in 2.9507 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.84, 157.22 APE9-dihe-na 133.4, -154.71 APE8-dihe-in -125.36, 134.74 APE8-rot-in 298.73 APE67-dihe-in -64.25, -21.15 -48.42, -47.94 APE12-dist-in 7.9507 APE11-dist-in 11.2453 APE10-dist-in 5.8092 APE9-dist-in 3.9436 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.49 0.144 0.177 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6sq1 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y05A P25321 8 351 351.0 ADE:60401 Type1 Active DFGin 6.2038 13.15 BLAminus -122.62, 176.1 60.39, 98.08 -109.84, 29.54 293.58, 72.67 -62.59, -23.96 in-in in 8.9695 Saltbr-in 2.6495 HRD-in -91.46, -52.85 71.13, 13.97 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.05, 162.66 APE9-dihe-na 130.15, -156.07 APE8-dihe-in -123.62, 136.19 APE8-rot-in 301.3 APE67-dihe-in -59.67, -24.1 -52.64, -47.85 APE12-dist-in 8.102 APE11-dist-in 11.5295 APE10-dist-in 5.9277 APE9-dist-in 3.5458 None TPO198,SEP339 TPO198,SEP339 XRAY 1.7 0.178 0.205 A 353.0 344.0 0 25 25 0 [[44, 298]] 1.0 6y05 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y89A P25321 11 351 351.0 OGB:60401 Type1 Active DFGin 5.8698 14.4362 BLAminus -122.55, 174.87 63.65, 84.21 -93.51, 25.44 274.84, 60.12 -60.56, -27.02 in-in in 9.0446 Saltbr-in 2.6615 HRD-in -89.79, -53.04 71.39, 13.28 in-in-in SNCiii in-in ActLoopNT-in 2.8959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.08, 161.18 APE9-dihe-na 130.37, -156.13 APE8-dihe-in -122.12, 132.52 APE8-rot-in 297.86 APE67-dihe-in -57.82, -25.35 -46.57, -49.91 APE12-dist-in 8.0645 APE11-dist-in 11.5446 APE10-dist-in 5.9255 APE9-dist-in 3.5915 None TPO198,SEP339 TPO198,SEP339 XRAY 1.56 0.17 0.192 A 353.0 339.0 2 25 25 0 [[44, 298]] 1.0 6y89 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNAA P25321 1 351 351.0 M77:60402 Type1 Active DFGin 6.2016 14.3343 BLAminus -119.96, 179.81 63.19, 78.66 -92.28, 22.25 273.96, 61.01 -60.67, -22.0 in-in in 8.696 Saltbr-in 2.6397 HRD-in -90.85, -54.18 73.93, 11.37 in-in-in SNCiii in-in ActLoopNT-in 2.9234 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.28, 159.25 APE9-dihe-na 133.12, -164.07 APE8-dihe-in -114.68, 130.03 APE8-rot-in 297.53 APE67-dihe-in -61.88, -21.65 -45.58, -51.04 APE12-dist-in 8.2756 APE11-dist-in 11.6374 APE10-dist-in 6.1355 APE9-dist-in 3.7647 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.47 0.165 0.189 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6yna Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNBA P25321 1 351 351.0 IQU:60401 Type1 Active DFGin 6.3631 14.3492 BLAminus -116.44, -174.16 61.98, 75.89 -98.12, 21.41 275.26, 66.86 -65.3, -20.05 in-in in 8.6085 Saltbr-in 2.4589 HRD-in -95.93, -55.57 72.9, 13.24 in-in-in SNCiii in-in ActLoopNT-in 2.8713 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.81, 160.16 APE9-dihe-na 137.96, -159.84 APE8-dihe-in -118.76, 130.24 APE8-rot-in 299.49 APE67-dihe-in -60.0, -21.74 -44.91, -52.44 APE12-dist-in 8.0367 APE11-dist-in 11.4934 APE10-dist-in 6.0621 APE9-dist-in 3.7628 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.72 0.158 0.201 A 353.0 347.0 1 25 25 0 [[44, 298]] 1.0 6ynb Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNCA P25321 1 351 351.0 7CT:60401 Type1 Active DFGin 6.0405 14.5355 BLAminus -120.79, 169.65 71.14, 83.37 -95.82, 21.95 274.39, 61.02 -58.31, -26.55 in-in in 8.8468 Saltbr-in 2.5305 HRD-in -88.43, -56.03 72.64, 13.22 in-in-in SNCiii in-in ActLoopNT-in 2.9309 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.35, 158.03 APE9-dihe-na 138.45, -155.36 APE8-dihe-in -121.88, 130.9 APE8-rot-in 297.76 APE67-dihe-in -61.6, -20.8 -45.0, -53.23 APE12-dist-in 8.1381 APE11-dist-in 11.5595 APE10-dist-in 6.0828 APE9-dist-in 3.6746 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.4 0.15 0.173 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 6ync Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNRA P25321 11 351 351.0 O72:60403 Type1 Active DFGin 5.8353 14.1484 BLAminus -121.49, -178.1 59.21, 91.48 -99.82, 25.19 274.78, 55.92 -59.5, -24.95 in-in in 9.0384 Saltbr-in 2.6099 HRD-in -85.88, -50.99 69.33, 11.34 in-in-in SNCiii in-in ActLoopNT-in 2.8951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.62, 159.23 APE9-dihe-na 131.94, -160.26 APE8-dihe-in -120.46, 134.53 APE8-rot-in 302.96 APE67-dihe-in -61.79, -24.17 -46.56, -49.51 APE12-dist-in 8.1163 APE11-dist-in 11.3885 APE10-dist-in 5.8269 APE9-dist-in 3.616 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.9 0.189 0.221 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6ynr Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNTA P25321 6 351 351.0 LRT:60405 Type1 Active DFGin 6.0242 14.3498 BLAminus -127.88, -176.71 61.66, 78.46 -90.86, 25.34 272.68, 60.44 -59.78, -24.31 in-in in 9.06 Saltbr-in 2.6983 HRD-in -92.67, -53.37 74.33, 11.71 in-in-in SNCiii in-in ActLoopNT-in 2.9262 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.24, 160.78 APE9-dihe-na 130.38, -159.85 APE8-dihe-in -120.86, 135.61 APE8-rot-in 299.16 APE67-dihe-in -60.2, -23.36 -47.55, -51.43 APE12-dist-in 8.1139 APE11-dist-in 11.3697 APE10-dist-in 5.8425 APE9-dist-in 3.5589 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.52 0.171 0.191 A 353.0 346.0 0 25 25 0 [[44, 298]] 1.0 6ynt Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YOUA P25321 14 351 351.0 P4Q:60401 Type1 Active DFGin 6.1964 14.3182 BLAminus -120.09, 165.39 72.67, 93.33 -100.94, 27.48 272.8, 57.34 -61.54, -27.01 in-in in 8.6014 Saltbr-in 2.6137 HRD-in -87.37, -52.03 71.03, 15.52 in-in-in SNCiii in-in ActLoopNT-in 2.9619 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.59, 163.46 APE9-dihe-na 118.27, -170.34 APE8-dihe-in -109.65, 135.96 APE8-rot-in 311.42 APE67-dihe-in -62.17, -24.35 -52.31, -42.25 APE12-dist-in 8.0511 APE11-dist-in 11.1756 APE10-dist-in 5.7123 APE9-dist-in 3.7508 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.73 0.181 0.216 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6you Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YPPA P25321 13 351 351.0 ISQ:60401 Type1 Active DFGin 6.575 13.8991 BLAminus -125.47, 168.17 69.21, 91.25 -102.12, 26.99 282.19, 66.61 -59.38, -28.47 in-in in 8.4767 Saltbr-in 2.8285 HRD-in -95.67, -54.73 76.34, 8.75 in-in-in SNCiii in-in ActLoopNT-in 2.9182 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.07, 157.89 APE9-dihe-na 135.57, -161.87 APE8-dihe-in -121.03, 135.18 APE8-rot-in 300.65 APE67-dihe-in -60.09, -21.93 -50.41, -52.89 APE12-dist-in 8.005 APE11-dist-in 11.2134 APE10-dist-in 5.7336 APE9-dist-in 3.8634 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.75 0.179 0.203 A 353.0 337.0 2 25 25 0 [[44, 298]] 1.0 6ypp Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YPSA P25321 14 351 351.0 P72:60402 Type1 Active DFGin 6.1571 14.3301 BLAminus -118.18, 171.85 69.73, 80.92 -91.01, 22.0 274.81, 61.35 -59.17, -25.98 in-in in 8.6264 Saltbr-in 2.7911 HRD-in -86.09, -50.96 68.81, 12.1 in-in-in SNCiii in-in ActLoopNT-in 2.9233 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.88, 163.19 APE9-dihe-na 126.1, -161.8 APE8-dihe-in -121.09, 134.4 APE8-rot-in 301.85 APE67-dihe-in -62.56, -20.95 -48.37, -48.27 APE12-dist-in 8.0941 APE11-dist-in 11.1937 APE10-dist-in 5.6911 APE9-dist-in 3.7621 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.35 0.145 0.157 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6yps Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YQIA P25321 1 351 351.0 6TV:60401 Type1 Active DFGin 6.6225 13.8594 BLAminus -120.83, 174.85 73.2, 74.9 -95.37, 21.17 285.79, 72.27 -63.44, -25.21 in-in in 8.555 Saltbr-in 2.8726 HRD-in -91.67, -56.05 72.65, 12.52 in-in-in SNCiii in-in ActLoopNT-in 2.9283 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.98, 159.1 APE9-dihe-na 134.75, -160.96 APE8-dihe-in -117.42, 130.5 APE8-rot-in 297.87 APE67-dihe-in -60.26, -23.17 -43.79, -54.04 APE12-dist-in 8.0852 APE11-dist-in 11.5282 APE10-dist-in 6.0526 APE9-dist-in 3.7076 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.42 0.155 0.18 A 353.0 345.0 3 25 25 0 [[44, 298]] 1.0 6yqi Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YQJA P25321 1 351 351.0 6TX:60401 Type1 Active DFGin 6.536 14.0021 BLAminus -124.1, 170.97 64.75, 82.67 -94.0, 24.22 278.04, 68.57 -64.35, -18.91 in-in in 8.3434 Saltbr-in 2.8114 HRD-in -94.88, -53.22 71.62, 13.76 in-in-in SNCiii in-in ActLoopNT-in 2.9414 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.32, 160.29 APE9-dihe-na 132.83, -156.0 APE8-dihe-in -122.12, 131.13 APE8-rot-in 297.37 APE67-dihe-in -59.98, -22.93 -46.61, -53.18 APE12-dist-in 8.1341 APE11-dist-in 11.5405 APE10-dist-in 6.0266 APE9-dist-in 3.5883 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.16 0.201 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 6yqj Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YQKA P25321 1 351 351.0 7KB:60401 Type1 Active DFGin 6.3842 14.635 BLAminus -116.26, -173.03 63.61, 71.29 -93.36, 20.28 275.04, 72.25 -62.95, -24.83 in-in in 9.2842 Saltbr-in 2.5172 HRD-in -89.64, -52.45 71.24, 12.44 in-in-in SNCiii in-in ActLoopNT-in 2.9122 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.58, 159.9 APE9-dihe-na 130.2, -161.78 APE8-dihe-in -114.54, 132.23 APE8-rot-in 297.68 APE67-dihe-in -62.46, -19.69 -47.44, -50.59 APE12-dist-in 8.2392 APE11-dist-in 11.6243 APE10-dist-in 6.1043 APE9-dist-in 3.8152 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.67 0.167 0.202 A 353.0 344.0 5 25 25 0 [[44, 298]] 1.0 6yqk Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7AXTA P25321 1 351 351.0 S9B:60401 Type1 Active DFGin 6.7184 14.8628 BLAminus -127.34, 164.32 75.46, 88.44 -100.63, 25.42 283.48, 72.18 -68.02, -22.42 in-in in 9.1968 Saltbr-in 3.149 HRD-in -87.43, -53.85 74.57, 8.03 in-in-in SNCiii in-in ActLoopNT-in 2.8964 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.36, 157.27 APE9-dihe-na 128.21, -163.37 APE8-dihe-in -115.52, 132.73 APE8-rot-in 300.39 APE67-dihe-in -59.29, -20.86 -48.29, -50.7 APE12-dist-in 8.1621 APE11-dist-in 11.401 APE10-dist-in 5.8203 APE9-dist-in 3.6485 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.86 0.189 0.226 A 353.0 342.0 5 25 25 0 [[44, 298]] 1.0 7axt Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7BARA P25321 14 351 351.0 T82:60401 Type1 Active DFGin 6.3379 14.4805 BLAminus -129.87, -171.42 62.69, 72.07 -89.88, 23.39 274.09, 65.5 -62.66, -24.64 in-in in 8.7197 Saltbr-in 2.8384 HRD-in -88.26, -52.14 74.09, 12.92 in-in-in SNCiii in-in ActLoopNT-in 2.9197 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.3, 163.6 APE9-dihe-na 129.58, -156.99 APE8-dihe-in -128.55, 134.3 APE8-rot-in 298.64 APE67-dihe-in -61.2, -20.19 -50.31, -49.26 APE12-dist-in 8.0904 APE11-dist-in 11.2272 APE10-dist-in 5.7202 APE9-dist-in 3.6557 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.37 0.153 0.179 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 7bar Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIHA P25321 1 351 351.0 7QW:60401 Type1 Active DFGin 6.6112 14.7767 BLAminus -121.61, 158.3 80.03, 88.23 -96.87, 22.43 285.52, 80.97 -63.48, -26.52 in-in in 9.1964 Saltbr-in 3.0815 HRD-in -85.1, -53.84 72.68, 6.07 in-in-in SNCiii in-in ActLoopNT-in 2.9353 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.04, 157.29 APE9-dihe-na 126.06, -165.16 APE8-dihe-in -115.66, 135.76 APE8-rot-in 299.21 APE67-dihe-in -61.29, -23.28 -48.22, -51.33 APE12-dist-in 8.4106 APE11-dist-in 11.5423 APE10-dist-in 5.9635 APE9-dist-in 3.7416 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.374 0.14 0.157 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pih Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDXA P25321 12 351 351.0 A1JE5:60406 Type1 Active DFGin 6.3947 14.5159 BLAminus -120.9, 176.38 62.83, 88.27 -100.01, 26.71 273.66, 64.38 -63.82, -25.52 in-in in 8.7161 Saltbr-in 2.9652 HRD-in -95.33, -53.05 70.61, 15.96 in-in-in SNCiii in-in ActLoopNT-in 3.0157 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.31, 161.4 APE9-dihe-na 124.9, -173.36 APE8-dihe-in -106.08, 132.1 APE8-rot-in 308.01 APE67-dihe-in -62.99, -20.07 -49.55, -46.7 APE12-dist-in 8.2468 APE11-dist-in 11.4052 APE10-dist-in 5.9001 APE9-dist-in 4.0415 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.193 0.208 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rdx Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE6A P25321 13 351 351.0 A1JEX:60605 Type1 Active DFGin 6.4398 14.6332 BLAminus -123.71, 169.54 74.02, 90.92 -99.73, 23.54 270.67, 62.64 -62.18, -25.3 in-in in 8.7272 Saltbr-in 2.9096 HRD-in -86.3, -51.47 69.33, 11.7 in-in-in SNCiii in-in ActLoopNT-in 2.9767 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.91, 159.32 APE9-dihe-na 117.99, 172.79 APE8-dihe-in -90.66, 139.04 APE8-rot-in 307.68 APE67-dihe-in -64.33, -21.04 -49.6, -45.84 APE12-dist-in 8.1212 APE11-dist-in 11.3054 APE10-dist-in 5.7928 APE9-dist-in 3.9602 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.45 0.177 0.194 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9re6 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RENA P25321 13 351 351.0 A1JEK:60401 Type1 Active DFGin 6.2639 14.538 BLAminus -125.36, 166.83 70.47, 89.12 -96.27, 20.46 272.82, 57.42 -59.85, -25.61 in-in in 8.7615 Saltbr-in 2.7947 HRD-in -89.58, -52.32 70.81, 11.76 in-in-in SNCiii in-in ActLoopNT-in 2.8858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.72, 157.64 APE9-dihe-na 115.87, 172.3 APE8-dihe-in -88.32, 133.56 APE8-rot-in 293.26 APE67-dihe-in -60.41, -22.75 -46.56, -47.75 APE12-dist-in 7.9097 APE11-dist-in 11.1788 APE10-dist-in 5.6755 APE9-dist-in 4.059 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.16 0.181 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ren Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REQA P25321 13 351 351.0 A1JEI:60402 Type1 Active DFGin 6.494 14.6379 BLAminus -119.67, 172.96 64.34, 87.39 -94.55, 24.82 273.79, 57.22 -60.93, -26.75 in-in in 8.8075 Saltbr-in 2.8045 HRD-in -85.13, -51.31 68.74, 14.76 in-in-in SNCiii in-in ActLoopNT-in 2.9545 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.42, 156.59 APE9-dihe-na 122.72, 176.53 APE8-dihe-in -91.46, 139.22 APE8-rot-in 321.17 APE67-dihe-in -64.4, -18.2 -52.5, -47.28 APE12-dist-in 8.1908 APE11-dist-in 11.3155 APE10-dist-in 5.8314 APE9-dist-in 4.0262 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.19 0.225 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9req Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RERA P25321 13 351 351.0 A1JEH:60401 Type1 Active DFGin 6.3318 14.5099 BLAminus -119.15, -175.34 54.86, 83.32 -93.03, 23.56 273.62, 62.86 -62.47, -23.85 in-in in 8.7329 Saltbr-in 2.8226 HRD-in -86.33, -53.68 72.65, 12.74 in-in-in SNCiii in-in ActLoopNT-in 2.9096 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.6, 159.26 APE9-dihe-na 118.95, -179.09 APE8-dihe-in -98.87, 134.79 APE8-rot-in 304.07 APE67-dihe-in -61.62, -21.03 -49.43, -46.1 APE12-dist-in 8.1931 APE11-dist-in 11.2928 APE10-dist-in 5.7953 APE9-dist-in 4.0229 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.45 0.179 0.198 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rer Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0LA P25321 12 351 351.0 7CT:60401,7CT:60402 Type1,Allosteric Active DFGin 5.8124 14.412 BLAminus -125.24, 171.39 72.54, 82.78 -94.45, 21.51 274.7, 58.82 -58.96, -27.86 in-in in 8.9632 Saltbr-in 2.5902 HRD-in -93.78, -54.2 73.09, 11.9 in-in-in SNCiii in-in ActLoopNT-in 2.9318 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.09, 160.85 APE9-dihe-na 134.16, -158.05 APE8-dihe-in -124.56, 135.24 APE8-rot-in 298.63 APE67-dihe-in -59.22, -23.14 -48.63, -50.91 APE12-dist-in 7.9743 APE11-dist-in 11.3295 APE10-dist-in 5.7609 APE9-dist-in 3.6509 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.465 0.153 0.173 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5m0l Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5MHIA P25321 1 351 351.0 7N9:60402,7N9:60403 Type1,Allosteric Active DFGin 6.5271 14.3646 BLAminus -123.97, 171.25 68.38, 93.75 -105.37, 25.41 275.2, 68.89 -61.8, -24.18 in-in in 8.6749 Saltbr-in 2.887 HRD-in -89.75, -51.15 72.09, 10.68 in-in-in SNCiii in-in ActLoopNT-in 2.9159 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.87, 159.66 APE9-dihe-na 135.33, -164.35 APE8-dihe-in -111.34, 128.89 APE8-rot-in 298.07 APE67-dihe-in -61.98, -22.3 -42.2, -53.64 APE12-dist-in 8.4497 APE11-dist-in 11.738 APE10-dist-in 6.2031 APE9-dist-in 3.7917 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.489 0.148 0.165 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5mhi Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1KA P25321 7 351 351.0 489:60401,489:60402 Type1,Allosteric Active DFGin 6.6813 14.3396 BLAminus -129.58, -178.71 64.55, 76.01 -90.26, 23.75 273.79, 68.55 -63.06, -22.76 in-in in 8.7102 Saltbr-in 2.9128 HRD-in -99.27, -50.72 71.29, 6.63 in-in-in SNCiii in-in ActLoopNT-in 2.8362 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.63, 158.5 APE9-dihe-na 132.87, -161.38 APE8-dihe-in -113.27, 127.15 APE8-rot-in 294.21 APE67-dihe-in -60.63, -22.02 -48.01, -50.0 APE12-dist-in 8.5014 APE11-dist-in 11.9334 APE10-dist-in 6.3293 APE9-dist-in 3.9344 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.8 0.176 0.207 A 353.0 342.0 1 25 25 0 [[44, 298]] 1.0 5n1k Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N32A P25321 1 351 351.0 8K5:60401,8K5:60402 Type1,Allosteric Active DFGin 6.4155 14.3999 BLAminus -123.43, 169.73 68.32, 89.82 -99.03, 25.86 273.98, 63.38 -60.64, -27.18 in-in in 8.5541 Saltbr-in 2.9422 HRD-in -95.08, -52.85 72.97, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.8629 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.95, 157.19 APE9-dihe-na 134.82, -164.27 APE8-dihe-in -110.28, 129.88 APE8-rot-in 300.11 APE67-dihe-in -58.64, -21.5 -44.53, -54.28 APE12-dist-in 8.2963 APE11-dist-in 11.7091 APE10-dist-in 6.1918 APE9-dist-in 3.7562 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.833 0.189 0.214 A 353.0 347.0 1 25 25 0 [[44, 298]] 1.0 5n32 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3FA P25321 8 334 351.0 463:60403,463:60404 Type1,Allosteric Active DFGin 6.6384 14.3677 BLAminus -117.37, -176.84 55.46, 81.93 -92.56, 25.55 274.27, 67.55 -63.44, -27.73 in-in in 8.5998 Saltbr-in 2.7496 HRD-in -89.81, -49.01 69.4, 15.01 in-in-in SNCiii in-in ActLoopNT-in 2.8811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.19, 158.49 APE9-dihe-na 131.1, -163.4 APE8-dihe-in -115.17, 131.52 APE8-rot-in 292.11 APE67-dihe-in -62.12, -20.35 -46.17, -51.48 APE12-dist-in 8.2862 APE11-dist-in 11.6832 APE10-dist-in 6.133 APE9-dist-in 3.7286 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.68 0.173 0.193 A 353.0 321.0 3 25 25 0 [[44, 298]] 1.0 5n3f Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3QA P25321 13 351 351.0 3AB:60402,3AB:60403 Type1,Allosteric Active DFGin 6.2826 14.5563 BLAminus -125.56, 161.33 75.46, 92.4 -98.05, 24.41 270.83, 54.38 -60.67, -25.07 in-in in 8.6862 Saltbr-in 3.0245 HRD-in -85.81, -51.8 71.36, 11.13 in-in-in SNCiii in-in ActLoopNT-in 2.932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.6, 158.28 APE9-dihe-na 114.3, 168.0 APE8-dihe-in -88.22, 137.3 APE8-rot-in 301.76 APE67-dihe-in -63.54, -20.32 -47.52, -48.52 APE12-dist-in 8.0466 APE11-dist-in 11.2177 APE10-dist-in 5.6936 APE9-dist-in 3.9813 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.31 0.136 0.155 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5n3q Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SNXA P25321 12 351 351.0 UNU:60401,UNU:60402 Type1,Allosteric Active DFGin 6.0512 12.8501 BLAminus -124.13, 164.79 75.87, 90.3 -99.95, 24.45 300.66, 73.6 -57.58, -27.27 in-in in 8.5952 Saltbr-in 3.0744 HRD-in -86.88, -52.37 71.04, 13.69 in-in-in SNCiii in-in ActLoopNT-in 2.9054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.16, 166.36 APE9-dihe-na 120.96, -160.48 APE8-dihe-in -123.13, 133.39 APE8-rot-in 301.0 APE67-dihe-in -63.1, -19.02 -49.07, -48.25 APE12-dist-in 8.1536 APE11-dist-in 11.1905 APE10-dist-in 5.6481 APE9-dist-in 3.568 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.4 0.142 0.173 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6snx Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YOTA P25321 1 351 351.0 P4W:60401,P4W:60402 Type1,Allosteric Active DFGin 6.3385 14.3597 BLAminus -117.22, 168.15 76.5, 96.51 -113.0, 26.95 288.67, 82.96 -66.18, -20.33 in-in in 9.1602 Saltbr-in 2.6238 HRD-in -88.7, -57.55 74.81, 2.26 in-in-in SNCiii in-in ActLoopNT-in 2.8328 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.9, 156.81 APE9-dihe-na 126.53, -165.91 APE8-dihe-in -115.98, 133.13 APE8-rot-in 299.88 APE67-dihe-in -58.64, -24.04 -48.78, -50.95 APE12-dist-in 8.0985 APE11-dist-in 11.3364 APE10-dist-in 5.8219 APE9-dist-in 3.7365 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.96 0.192 0.213 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6yot Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ZN0A P25321 14 351 351.0 NTN:60404,NTN:60405 Type1,Allosteric Active DFGin 6.3062 14.2933 BLAminus -125.36, 174.33 64.27, 86.94 -95.54, 24.99 272.68, 57.62 -59.97, -26.54 in-in in 8.5423 Saltbr-in 2.7539 HRD-in -87.06, -51.0 70.17, 14.59 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.46, 163.69 APE9-dihe-na 125.37, -162.56 APE8-dihe-in -119.36, 135.19 APE8-rot-in 306.4 APE67-dihe-in -62.76, -20.13 -50.46, -46.23 APE12-dist-in 8.1022 APE11-dist-in 11.185 APE10-dist-in 5.6571 APE9-dist-in 3.7386 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.59 0.156 0.186 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6zn0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE0A P25321 12 351 351.0 A1JE3:60415,A1JE3:60416 Type1,Allosteric Active DFGin 6.4858 14.8008 BLAminus -127.81, 175.95 67.21, 79.76 -92.52, 24.98 274.18, 65.26 -62.68, -27.01 in-in in 8.9734 Saltbr-in 2.7196 HRD-in -89.08, -49.37 68.42, 15.8 in-in-in SNCiii in-in ActLoopNT-in 2.9816 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.81, 165.38 APE9-dihe-na 123.68, -167.92 APE8-dihe-in -111.45, 134.55 APE8-rot-in 307.3 APE67-dihe-in -62.16, -20.99 -49.64, -48.1 APE12-dist-in 8.2307 APE11-dist-in 11.3722 APE10-dist-in 5.8261 APE9-dist-in 3.8272 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.58 0.17 0.199 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE1A P25321 12 351 351.0 A1JE2:60402,A1JE2:60403 Type1,Allosteric Active DFGin 6.357 14.4975 BLAminus -123.64, 170.43 71.38, 82.58 -93.83, 23.94 276.73, 61.78 -63.16, -19.76 in-in in 8.9487 Saltbr-in 2.6912 HRD-in -91.56, -54.72 69.86, 16.16 in-in-in SNCiii in-in ActLoopNT-in 2.9345 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.9, 155.93 APE9-dihe-na 118.62, 174.39 APE8-dihe-in -90.43, 137.72 APE8-rot-in 306.04 APE67-dihe-in -61.66, -22.83 -48.01, -48.11 APE12-dist-in 8.0786 APE11-dist-in 11.2497 APE10-dist-in 5.7715 APE9-dist-in 4.114 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.41 0.158 0.189 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re1 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE8A P25321 13 351 351.0 A1JEQ:60401,A1JEQ:60402 Type1,Allosteric Active DFGin 6.4702 14.2842 BLAminus -121.7, 170.26 70.13, 85.83 -96.63, 25.0 277.83, 62.9 -63.72, -22.81 in-in in 8.5972 Saltbr-in 2.853 HRD-in -94.16, -51.38 66.63, 15.52 in-in-in SNCiii in-in ActLoopNT-in 2.9219 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.45, 162.24 APE9-dihe-na 127.76, -169.19 APE8-dihe-in -105.79, 133.4 APE8-rot-in 307.65 APE67-dihe-in -61.36, -22.52 -49.82, -47.46 APE12-dist-in 8.0545 APE11-dist-in 11.2462 APE10-dist-in 5.7207 APE9-dist-in 3.8389 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.18 0.204 A 353.0 337.0 2 25 25 0 [[44, 298]] 1.0 9re8 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE9A P25321 12 351 351.0 A1JER:60406,A1JER:60407 Type1,Allosteric Active DFGin 6.2139 14.4257 BLAminus -115.45, 174.18 67.64, 91.06 -99.47, 24.72 274.09, 59.88 -62.57, -25.54 in-in in 8.5815 Saltbr-in 2.8645 HRD-in -87.53, -50.86 69.59, 9.72 in-in-in SNCiii in-in ActLoopNT-in 2.9177 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.54, 160.39 APE9-dihe-na 112.91, 168.83 APE8-dihe-in -85.08, 139.5 APE8-rot-in 305.47 APE67-dihe-in -61.28, -24.3 -48.68, -48.83 APE12-dist-in 8.0803 APE11-dist-in 11.1938 APE10-dist-in 5.7056 APE9-dist-in 3.9875 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.41 0.159 0.182 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re9 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE4A P25321 11 351 351.0 A1JEZ:60402,A1JEZ:60403,A1JEZ:60404 Type1,Allosteric,Allosteric Active DFGin 6.4193 14.4719 BLAminus -125.46, 163.88 74.29, 91.54 -99.92, 24.22 273.39, 58.15 -62.6, -24.27 in-in in 8.6037 Saltbr-in 3.0263 HRD-in -87.71, -51.55 69.07, 12.85 in-in-in SNCiii in-in ActLoopNT-in 2.9413 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.46, 156.9 APE9-dihe-na 126.03, -178.78 APE8-dihe-in -98.18, 132.58 APE8-rot-in 299.03 APE67-dihe-in -60.55, -22.76 -49.18, -46.22 APE12-dist-in 8.1382 APE11-dist-in 11.3542 APE10-dist-in 5.8006 APE9-dist-in 4.0873 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.47 0.192 0.208 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 9re4 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE7A P25321 13 351 351.0 D6V:60401,D6V:60402,D6V:60403,D6V:60404 Type1,Allosteric,Allosteric,Allosteric Active DFGin 6.3969 14.3822 BLAminus -125.46, 169.66 70.64, 87.21 -98.97, 25.83 271.46, 63.62 -64.67, -22.85 in-in in 8.6706 Saltbr-in 3.0142 HRD-in -86.12, -51.15 69.09, 13.78 in-in-in SNCiii in-in ActLoopNT-in 2.9179 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.38, 162.49 APE9-dihe-na 118.13, -170.93 APE8-dihe-in -105.88, 133.45 APE8-rot-in 300.33 APE67-dihe-in -56.23, -24.21 -49.65, -50.28 APE12-dist-in 8.2052 APE11-dist-in 11.3507 APE10-dist-in 5.7797 APE9-dist-in 3.8302 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.46 0.156 0.183 A 353.0 337.0 2 25 25 0 [[44, 298]] 1.0 9re7 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REIA P25321 13 351 351.0 A1JEN:60401,A1JEN:60402 Type1,Type1 Active DFGin 6.4427 14.5573 BLAminus -121.53, 160.04 78.3, 90.11 -98.4, 25.75 272.41, 61.56 -62.91, -24.68 in-in in 8.7225 Saltbr-in 2.9878 HRD-in -84.67, -52.43 70.44, 13.57 in-in-in SNCiii in-in ActLoopNT-in 2.9938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.29, 162.32 APE9-dihe-na 123.69, -172.32 APE8-dihe-in -110.41, 137.96 APE8-rot-in 307.06 APE67-dihe-in -63.61, -18.16 -49.51, -49.01 APE12-dist-in 8.2745 APE11-dist-in 11.2994 APE10-dist-in 5.8053 APE9-dist-in 3.9129 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.167 0.199 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rei Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OUAA P25321 1 351 351.0 No_ligand No_ligand Inactive DFGin 6.7177 14.6348 ABAminus -115.87, -28.94 -123.11, 121.25 -116.35, 27.71 279.87, 77.2 -63.52, -23.18 in-in in 8.6437 Saltbr-in 2.9268 HRD-in -81.78, -54.82 73.94, 13.55 in-in-in SNCiii in-in ActLoopNT-in 2.8996 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.08, 165.1 APE9-dihe-na 113.51, -165.37 APE8-dihe-in -110.07, 129.07 APE8-rot-in 298.26 APE67-dihe-in -59.52, -23.19 -44.71, -53.87 APE12-dist-in 8.3252 APE11-dist-in 11.5022 APE10-dist-in 5.7636 APE9-dist-in 3.3871 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.67 0.17 0.194 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5oua Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OUSA P25321 1 351 351.0 No_ligand No_ligand Inactive DFGin 6.5073 15.429 ABAminus -111.6, -55.85 -94.1, 116.86 -107.2, 23.58 279.6, 77.36 -70.84, -13.23 in-none in 9.4454 Saltbr-none 999.0 HRD-in -84.43, -53.59 72.65, 7.3 none-in-in SNCnii in-in ActLoopNT-in 3.002 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.86, 162.52 APE9-dihe-na 121.37, -167.35 APE8-dihe-in -115.92, 134.51 APE8-rot-in 300.98 APE67-dihe-in -58.34, -27.31 -46.95, -49.63 APE12-dist-in 8.2545 APE11-dist-in 11.5502 APE10-dist-in 5.9508 APE9-dist-in 3.6723 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.21 0.196 0.233 A 353.0 348.0 1 25 25 0 [[44, 298]] 1.0 5ous Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5NW8A P25321 12 351 351.0 M77:60402 Type1 Inactive DFGin 6.3364 14.3863 ABAminus -118.68, -32.42 -99.03, 121.53 -122.45, 23.74 290.12, 82.65 -65.48, -23.88 in-in in 8.8836 Saltbr-in 2.7053 HRD-in -87.46, -57.12 74.8, 8.43 in-in-in SNCiii in-in ActLoopNT-in 2.9091 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.41, 158.53 APE9-dihe-na 124.11, -167.34 APE8-dihe-in -113.09, 136.58 APE8-rot-in 301.73 APE67-dihe-in -53.51, -29.49 -47.53, -53.31 APE12-dist-in 8.2041 APE11-dist-in 11.5565 APE10-dist-in 5.9221 APE9-dist-in 3.7724 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.086 0.178 0.212 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 5nw8 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCPA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.5125 14.567 ABAminus -121.65, -30.45 -98.92, 119.1 -122.07, 18.29 284.17, 84.65 -65.16, -27.53 in-in in 8.8992 Saltbr-in 2.7586 HRD-in -92.61, -56.98 71.24, 5.31 in-in-in SNCiii in-in ActLoopNT-in 2.9161 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.37, 152.55 APE9-dihe-na 132.49, -162.49 APE8-dihe-in -118.01, 135.22 APE8-rot-in 296.96 APE67-dihe-in -61.44, -24.53 -48.46, -49.38 APE12-dist-in 8.1866 APE11-dist-in 11.4765 APE10-dist-in 5.9223 APE9-dist-in 3.9486 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.433 0.134 0.166 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcp Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCRA P25321 1 351 351.0 6TX:60401 Type1 Inactive DFGin 6.374 14.6833 ABAminus -120.45, -30.9 -97.04, 125.99 -132.15, 14.59 283.38, 89.54 -63.35, -31.44 in-in in 8.8488 Saltbr-in 2.672 HRD-in -87.18, -55.06 71.63, -3.59 in-in-in SNCiii in-in ActLoopNT-in 2.9015 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.81, 151.9 APE9-dihe-na 132.74, -162.98 APE8-dihe-in -119.91, 132.41 APE8-rot-in 297.04 APE67-dihe-in -57.71, -25.78 -46.99, -51.33 APE12-dist-in 8.2349 APE11-dist-in 11.5396 APE10-dist-in 6.0024 APE9-dist-in 4.0176 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.565 0.157 0.197 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcr Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCTA P25321 1 351 351.0 6TY:60401 Type1 Inactive DFGin 6.5666 14.9722 ABAminus -119.53, -36.47 -94.64, 123.81 -127.4, 15.84 283.42, 88.07 -61.61, -36.92 in-in in 8.9974 Saltbr-in 2.8958 HRD-in -87.59, -53.98 70.09, 3.04 in-in-in SNCiii in-in ActLoopNT-in 2.9272 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.1, 153.93 APE9-dihe-na 129.99, -163.89 APE8-dihe-in -118.91, 134.19 APE8-rot-in 299.57 APE67-dihe-in -59.43, -24.77 -48.83, -49.96 APE12-dist-in 8.3428 APE11-dist-in 11.612 APE10-dist-in 6.0758 APE9-dist-in 3.98 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.615 0.144 0.174 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lct Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCUA P25321 1 351 351.0 IQP:60401 Type1 Inactive DFGin 6.3439 14.5118 ABAminus -118.46, -33.64 -98.48, 122.71 -128.59, 17.69 287.43, 87.65 -64.81, -32.5 in-in in 8.9216 Saltbr-in 2.7757 HRD-in -89.6, -56.25 69.6, 5.54 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.54, 154.63 APE9-dihe-na 129.64, -164.53 APE8-dihe-in -116.54, 134.11 APE8-rot-in 299.55 APE67-dihe-in -60.52, -23.05 -47.34, -51.22 APE12-dist-in 8.1905 APE11-dist-in 11.5415 APE10-dist-in 5.9813 APE9-dist-in 3.9715 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.579 0.154 0.192 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcu Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M6VA P25321 1 351 351.0 H52:60401 Type1 Inactive DFGin 6.6215 14.87 ABAminus -128.93, -36.38 -82.47, 115.78 -126.79, 13.38 284.62, 84.57 -59.9, -36.82 in-in in 9.1455 Saltbr-in 3.0668 HRD-in -85.39, -54.24 70.45, 5.3 in-in-in SNCiii in-in ActLoopNT-in 2.88 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.08, 154.85 APE9-dihe-na 129.1, -162.88 APE8-dihe-in -117.77, 135.16 APE8-rot-in 297.05 APE67-dihe-in -61.78, -23.12 -47.87, -51.09 APE12-dist-in 8.2559 APE11-dist-in 11.5175 APE10-dist-in 5.9805 APE9-dist-in 3.8478 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.418 0.145 0.174 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m6v Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M6YA P25321 1 351 351.0 7KB:60401 Type1 Inactive DFGin 6.3247 14.3886 ABAminus -120.54, -28.06 -100.7, 125.25 -133.25, 5.41 291.12, 89.13 -59.31, -35.83 in-in in 8.9571 Saltbr-in 2.8685 HRD-in -85.55, -56.37 69.79, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.8795 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.17, 152.58 APE9-dihe-na 128.14, -163.48 APE8-dihe-in -117.76, 135.16 APE8-rot-in 298.33 APE67-dihe-in -60.49, -24.28 -48.85, -50.14 APE12-dist-in 8.3076 APE11-dist-in 11.7151 APE10-dist-in 6.2076 APE9-dist-in 4.0604 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.367 0.145 0.166 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m6y Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M71A P25321 1 351 351.0 7K7:60401 Type1 Inactive DFGin 6.5486 14.873 ABAminus -119.85, -32.84 -98.53, 122.12 -124.32, 17.46 284.12, 85.87 -64.55, -31.73 in-in in 9.0558 Saltbr-in 2.7642 HRD-in -87.14, -56.81 71.22, 6.23 in-in-in SNCiii in-in ActLoopNT-in 2.9024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.13, 152.91 APE9-dihe-na 131.38, -162.26 APE8-dihe-in -116.74, 134.6 APE8-rot-in 297.69 APE67-dihe-in -60.19, -23.45 -48.52, -50.53 APE12-dist-in 8.2262 APE11-dist-in 11.5825 APE10-dist-in 5.9903 APE9-dist-in 3.8944 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.488 0.149 0.176 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m71 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M75A P25321 1 351 351.0 9K6:60402 Type1 Inactive DFGin 6.5416 14.7033 ABAminus -122.93, -37.42 -95.22, 118.15 -122.41, 18.78 283.61, 82.19 -61.66, -33.64 in-in in 9.017 Saltbr-in 2.9023 HRD-in -86.66, -56.28 74.63, 2.67 in-in-in SNCiii in-in ActLoopNT-in 2.8945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.02, 157.01 APE9-dihe-na 127.35, -165.16 APE8-dihe-in -116.36, 133.7 APE8-rot-in 297.39 APE67-dihe-in -60.71, -23.5 -48.32, -49.81 APE12-dist-in 8.2248 APE11-dist-in 11.4473 APE10-dist-in 5.9243 APE9-dist-in 3.7682 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.538 0.146 0.174 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m75 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1DA P25321 1 351 351.0 8FZ:60403 Type1 Inactive DFGin 6.4268 14.5221 ABAminus -119.36, -25.35 -95.05, 134.07 -134.0, 35.23 286.49, 84.89 -74.09, -16.92 in-in in 8.9671 Saltbr-in 2.7736 HRD-in -86.75, -53.91 69.79, 6.83 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.28, 160.08 APE9-dihe-na 123.62, -165.42 APE8-dihe-in -115.29, 135.17 APE8-rot-in 295.44 APE67-dihe-in -60.76, -24.93 -47.42, -49.84 APE12-dist-in 8.3805 APE11-dist-in 11.5224 APE10-dist-in 5.9453 APE9-dist-in 3.6307 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.609 0.157 0.186 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n1d Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3DA P25321 1 351 351.0 8NE:60401 Type1 Inactive DFGin 6.3769 14.5132 ABAminus -125.06, 6.06 -141.01, 114.08 -108.34, 25.78 270.84, 67.95 -65.47, -20.45 in-in in 8.8019 Saltbr-in 2.8929 HRD-in -88.66, -53.48 71.74, 8.74 in-in-in SNCiii in-in ActLoopNT-in 2.8859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.56, 155.77 APE9-dihe-na 134.96, -165.87 APE8-dihe-in -106.38, 130.24 APE8-rot-in 300.79 APE67-dihe-in -61.42, -22.58 -44.45, -52.67 APE12-dist-in 8.4623 APE11-dist-in 11.8721 APE10-dist-in 6.2946 APE9-dist-in 3.8887 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.77 0.169 0.193 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 5n3d Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5O0EA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.5233 14.4554 ABAminus -120.87, -28.54 -98.9, 119.84 -125.0, 19.69 283.23, 84.18 -67.0, -26.17 in-in in 8.8606 Saltbr-in 2.7863 HRD-in -91.49, -57.65 74.16, -1.91 in-in-in SNCiii in-in ActLoopNT-in 2.9264 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.49, 154.58 APE9-dihe-na 133.99, -164.02 APE8-dihe-in -122.83, 136.35 APE8-rot-in 298.08 APE67-dihe-in -61.85, -22.28 -48.99, -49.98 APE12-dist-in 8.1871 APE11-dist-in 11.4128 APE10-dist-in 5.8742 APE9-dist-in 4.0603 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.5 0.133 0.17 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5o0e Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5O5MA P25321 10 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.2398 14.1421 ABAminus -103.5, -42.75 -109.64, 134.16 -133.73, 10.26 296.02, 86.96 -61.7, -36.78 in-in in 8.8473 Saltbr-in 2.793 HRD-in -81.57, -55.82 71.03, 6.22 in-in-in SNCiii in-in ActLoopNT-in 2.8906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.12, 155.87 APE9-dihe-na 127.02, -162.8 APE8-dihe-in -117.37, 136.63 APE8-rot-in 301.79 APE67-dihe-in -60.33, -24.0 -47.69, -51.35 APE12-dist-in 8.4177 APE11-dist-in 11.9058 APE10-dist-in 6.3877 APE9-dist-in 3.8023 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.583 0.15 0.182 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5o5m Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OK3A P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.6154 14.4154 ABAminus -120.44, -31.18 -98.89, 117.63 -123.6, 23.39 284.71, 82.73 -69.59, -23.81 in-in in 8.9341 Saltbr-in 2.7392 HRD-in -95.2, -57.86 72.09, 2.44 in-in-in SNCiii in-in ActLoopNT-in 2.9251 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.84, 153.6 APE9-dihe-na 133.87, -163.65 APE8-dihe-in -122.15, 135.18 APE8-rot-in 299.79 APE67-dihe-in -60.82, -23.36 -49.17, -49.56 APE12-dist-in 8.2185 APE11-dist-in 11.4659 APE10-dist-in 5.8784 APE9-dist-in 4.0553 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.588 0.141 0.172 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5ok3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OL3A P25321 11 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.2933 14.1388 ABAminus -103.07, -42.44 -110.53, 139.16 -139.44, 13.42 297.3, 87.11 -59.46, -35.81 in-in in 8.8063 Saltbr-in 2.7003 HRD-in -84.73, -54.59 70.4, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.9398 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.98, 154.3 APE9-dihe-na 129.69, -160.74 APE8-dihe-in -119.81, 133.8 APE8-rot-in 301.31 APE67-dihe-in -59.48, -24.61 -48.47, -50.75 APE12-dist-in 8.5226 APE11-dist-in 12.0085 APE10-dist-in 6.4955 APE9-dist-in 3.7939 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.156 0.199 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 5ol3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OT3A P25321 13 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.3842 14.2359 ABAminus -113.79, -34.42 -102.76, 127.41 -133.44, 15.99 294.3, 89.2 -57.06, -43.48 in-in in 8.8594 Saltbr-in 2.8226 HRD-in -85.16, -56.21 73.39, 3.05 in-in-in SNCiii in-in ActLoopNT-in 2.9097 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.31, 153.48 APE9-dihe-na 129.3, -161.89 APE8-dihe-in -114.87, 136.52 APE8-rot-in 300.43 APE67-dihe-in -56.81, -27.64 -51.93, -48.81 APE12-dist-in 8.2915 APE11-dist-in 11.842 APE10-dist-in 6.3049 APE9-dist-in 4.0341 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.04 0.186 0.228 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5ot3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OTGA P25321 1 351 351.0 AO8:60401 Type1 Inactive DFGin 6.6641 14.8724 ABAminus -116.07, -34.14 -101.63, 135.19 -132.51, 30.55 284.27, 81.94 -65.58, -28.86 in-in in 9.2076 Saltbr-in 2.8838 HRD-in -87.0, -54.6 75.88, 1.07 in-in-in SNCiii in-in ActLoopNT-in 2.9513 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.1, 159.53 APE9-dihe-na 126.93, -164.36 APE8-dihe-in -118.42, 136.98 APE8-rot-in 301.94 APE67-dihe-in -61.55, -22.37 -50.07, -49.22 APE12-dist-in 8.3277 APE11-dist-in 11.5661 APE10-dist-in 5.9649 APE9-dist-in 3.7403 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.73 0.187 0.206 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5otg Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OUCA P25321 1 351 351.0 AO8:60401 Type1 Inactive DFGin 6.5448 14.6897 ABAminus -118.72, -31.35 -98.66, 124.06 -126.19, 22.18 285.25, 84.4 -64.9, -29.38 in-none in 9.0152 Saltbr-none 999.0 HRD-in -89.21, -57.44 74.92, -2.84 none-in-in SNCnii in-in ActLoopNT-in 2.9042 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 152.91 APE9-dihe-na 134.96, -159.63 APE8-dihe-in -125.22, 135.43 APE8-rot-in 300.15 APE67-dihe-in -61.76, -25.06 -48.4, -50.36 APE12-dist-in 8.2727 APE11-dist-in 11.4814 APE10-dist-in 5.9359 APE9-dist-in 4.0149 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.46 0.151 0.175 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5ouc Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EGWA P25321 14 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.0679 14.0517 ABAminus -99.1, -40.07 -111.56, 135.78 -136.64, 9.64 299.83, 90.65 -57.2, -34.91 in-in in 8.8053 Saltbr-in 2.8447 HRD-in -79.79, -53.68 65.28, 14.91 in-in-in SNCiii in-in ActLoopNT-in 2.8654 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.34, 128.68 APE9-dihe-na 131.12, -162.98 APE8-dihe-in -115.37, 129.12 APE8-rot-in 299.83 APE67-dihe-in -57.87, -22.06 -45.69, -53.12 APE12-dist-in 8.5497 APE11-dist-in 12.0347 APE10-dist-in 6.3542 APE9-dist-in 3.7696 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.74 0.173 0.203 A 353.0 336.0 1 25 25 0 [[44, 298]] 1.0 6egw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EH3A P25321 1 351 351.0 B4Z:60401 Type1 Inactive DFGin 6.5603 14.4887 ABAminus -116.24, -28.55 -105.91, 131.63 -131.61, 27.16 287.22, 81.75 -60.81, -31.22 in-out in 9.0058 Saltbr-out 3.7684 HRD-in -84.94, -53.5 72.91, 0.92 out-in-in SNCoii in-in ActLoopNT-in 2.8965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.18, 161.6 APE9-dihe-na 127.52, -167.93 APE8-dihe-in -115.28, 135.37 APE8-rot-in 300.84 APE67-dihe-in -65.2, -22.11 -46.47, -48.64 APE12-dist-in 8.279 APE11-dist-in 11.5005 APE10-dist-in 5.9114 APE9-dist-in 3.8034 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.95 0.175 0.219 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6eh3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERTA P25321 14 351 351.0 BVZ:60401 Type1 Inactive DFGin 6.1937 14.1209 ABAminus -115.39, -20.57 -108.62, 132.15 -135.58, 27.66 297.14, 82.68 -71.36, -3.39 in-in in 8.9653 Saltbr-in 2.8205 HRD-in -85.32, -55.78 74.89, 1.92 in-in-in SNCiii in-in ActLoopNT-in 2.9314 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.5, 160.76 APE9-dihe-na 124.06, -167.42 APE8-dihe-in -111.64, 135.9 APE8-rot-in 303.33 APE67-dihe-in -58.26, -26.08 -52.61, -48.73 APE12-dist-in 8.2618 APE11-dist-in 11.6271 APE10-dist-in 6.0812 APE9-dist-in 3.7549 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.8 0.186 0.218 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6ert Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERWA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.4014 14.4703 ABAminus -121.15, -34.81 -95.55, 109.86 -114.31, 21.73 291.27, 86.69 -64.06, -18.67 in-in in 8.9017 Saltbr-in 2.8745 HRD-in -86.55, -59.04 70.6, 12.67 in-in-in SNCiii in-in ActLoopNT-in 2.8957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.31, 155.57 APE9-dihe-na 122.97, -167.43 APE8-dihe-in -109.73, 134.74 APE8-rot-in 295.31 APE67-dihe-in -57.25, -24.48 -52.2, -50.35 APE12-dist-in 8.161 APE11-dist-in 11.4552 APE10-dist-in 5.8644 APE9-dist-in 3.8464 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.89 0.195 0.229 A 353.0 348.0 3 25 25 0 [[44, 298]] 1.0 6erw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2AA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.6275 14.6347 ABAminus -122.01, -33.61 -93.89, 119.82 -124.65, 22.24 282.35, 82.22 -67.92, -23.48 in-in in 9.1929 Saltbr-in 2.5611 HRD-in -101.03, -58.68 69.95, -0.61 in-in-in SNCiii in-in ActLoopNT-in 2.9412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.26, 150.72 APE9-dihe-na 137.51, -163.36 APE8-dihe-in -120.26, 133.94 APE8-rot-in 301.03 APE67-dihe-in -62.45, -25.53 -48.16, -48.1 APE12-dist-in 8.1207 APE11-dist-in 11.4401 APE10-dist-in 5.8938 APE9-dist-in 4.1543 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.75 0.175 0.207 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6i2a Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2CA P25321 12 351 351.0 M77:60401 Type1 Inactive DFGin 6.5002 14.6062 ABAminus -115.95, -34.45 -102.09, 116.9 -120.62, 23.53 285.01, 87.65 -68.52, -23.98 in-in in 8.8456 Saltbr-in 2.9203 HRD-in -86.43, -55.89 76.54, -1.15 in-in-in SNCiii in-in ActLoopNT-in 2.9438 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.94, 153.26 APE9-dihe-na 129.65, -163.32 APE8-dihe-in -118.65, 136.78 APE8-rot-in 299.53 APE67-dihe-in -56.88, -28.13 -49.75, -50.61 APE12-dist-in 8.3036 APE11-dist-in 11.5191 APE10-dist-in 5.8971 APE9-dist-in 3.7163 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.82 0.187 0.221 A 353.0 338.0 2 25 25 0 [[44, 298]] 1.0 6i2c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2DA P25321 9 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.4857 14.6911 ABAminus -99.68, -45.99 -105.21, 136.79 -132.46, 16.35 286.72, 86.8 -63.64, -34.15 in-in in 8.6624 Saltbr-in 2.922 HRD-in -90.54, -57.71 68.94, 6.05 in-in-in SNCiii in-in ActLoopNT-in 2.9826 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.06, 154.58 APE9-dihe-na 132.32, -163.48 APE8-dihe-in -118.09, 133.54 APE8-rot-in 299.26 APE67-dihe-in -59.06, -24.95 -49.23, -49.12 APE12-dist-in 8.037 APE11-dist-in 11.595 APE10-dist-in 5.9733 APE9-dist-in 3.9587 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.91 0.19 0.222 A 353.0 343.0 0 25 25 0 [[44, 298]] 1.0 6i2d Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2HA P25321 1 351 351.0 AO8:60401 Type1 Inactive DFGin 6.5671 14.8085 ABAminus -115.56, -38.67 -109.61, 104.13 -103.25, 25.9 285.61, 77.71 -66.17, -17.47 in-in in 8.9865 Saltbr-in 2.9304 HRD-in -83.42, -55.73 70.56, 10.93 in-in-in SNCiii in-in ActLoopNT-in 2.8462 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.42, 160.46 APE9-dihe-na 121.97, -162.48 APE8-dihe-in -116.28, 135.78 APE8-rot-in 298.33 APE67-dihe-in -60.57, -22.98 -48.67, -52.6 APE12-dist-in 8.1576 APE11-dist-in 11.371 APE10-dist-in 5.6959 APE9-dist-in 3.5478 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.68 0.182 0.202 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6i2h Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y0BA P25321 1 351 351.0 1LQ:60401 Type1 Inactive DFGin 6.3607 14.3289 ABAminus -119.37, -25.73 -99.15, 124.17 -126.15, 31.35 288.49, 83.65 -71.09, -16.36 in-in in 9.046 Saltbr-in 2.5951 HRD-in -88.77, -52.67 71.85, 3.28 in-in-in SNCiii in-in ActLoopNT-in 2.8228 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.54, 158.64 APE9-dihe-na 129.02, -163.22 APE8-dihe-in -120.14, 133.41 APE8-rot-in 298.13 APE67-dihe-in -64.32, -22.04 -50.27, -45.04 APE12-dist-in 8.2202 APE11-dist-in 11.4198 APE10-dist-in 5.8956 APE9-dist-in 3.6527 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.71 0.181 0.212 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 6y0b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y2UA P25321 1 351 351.0 LRT:60401 Type1 Inactive DFGin 6.3897 14.1273 ABAminus -116.87, -29.74 -101.42, 118.51 -125.0, 17.87 293.73, 84.27 -60.5, -32.85 in-in in 8.8178 Saltbr-in 2.7471 HRD-in -82.23, -56.84 69.37, 8.99 in-in-in SNCiii in-in ActLoopNT-in 2.9228 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.67, 161.61 APE9-dihe-na 116.23, -161.47 APE8-dihe-in -111.19, 132.56 APE8-rot-in 301.77 APE67-dihe-in -58.37, -26.58 -47.25, -49.31 APE12-dist-in 8.1796 APE11-dist-in 11.6373 APE10-dist-in 5.9769 APE9-dist-in 3.8833 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.93 0.187 0.222 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6y2u Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7AXWA P25321 1 351 351.0 1SQ:60401 Type1 Inactive DFGin 6.4035 14.2527 ABAminus -120.14, -30.0 -96.57, 126.41 -127.77, 33.09 287.87, 84.79 -75.22, -10.69 in-in in 8.9432 Saltbr-in 2.6309 HRD-in -88.15, -50.93 71.59, -1.54 in-in-in SNCiii in-in ActLoopNT-in 2.8412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.41, 158.2 APE9-dihe-na 127.83, -163.7 APE8-dihe-in -120.34, 130.94 APE8-rot-in 298.02 APE67-dihe-in -65.73, -21.71 -43.41, -48.57 APE12-dist-in 8.2015 APE11-dist-in 11.4083 APE10-dist-in 5.9311 APE9-dist-in 3.6613 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.69 0.183 0.219 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 7axw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7BAQA P25321 12 351 351.0 T82:60401 Type1 Inactive DFGin 6.6314 14.6407 ABAminus -123.23, -37.41 -116.05, 126.94 -128.82, 27.15 284.58, 82.2 -65.24, -36.99 in-in in 8.8751 Saltbr-in 2.8259 HRD-in -84.32, -54.85 70.47, 4.72 in-in-in SNCiii in-in ActLoopNT-in 2.9304 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.86, 160.75 APE9-dihe-na 122.68, -162.38 APE8-dihe-in -118.09, 132.31 APE8-rot-in 301.89 APE67-dihe-in -58.89, -25.14 -49.52, -49.11 APE12-dist-in 8.2341 APE11-dist-in 11.5243 APE10-dist-in 6.0507 APE9-dist-in 3.7373 None TPO198,SEP339 TPO198,SEP339 XRAY 1.54 0.178 0.22 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 7baq Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIDA P25321 1 351 351.0 7QI:60401 Type1 Inactive DFGin 6.4367 14.9083 ABAminus -118.24, -40.4 -94.33, 114.05 -113.71, 22.91 282.95, 85.12 -67.72, -22.35 in-in in 9.1457 Saltbr-in 3.1967 HRD-in -88.95, -55.75 73.32, 6.65 in-in-in SNCiii in-in ActLoopNT-in 2.9311 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.62, 155.91 APE9-dihe-na 130.66, -167.59 APE8-dihe-in -113.9, 136.41 APE8-rot-in 298.55 APE67-dihe-in -61.41, -23.98 -47.99, -49.83 APE12-dist-in 8.2605 APE11-dist-in 11.4592 APE10-dist-in 5.8679 APE9-dist-in 3.8737 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.496 0.134 0.161 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pid Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIEA P25321 1 351 351.0 7QF:60401 Type1 Inactive DFGin 6.4369 14.7079 ABAminus -120.2, -32.0 -97.5, 116.46 -117.79, 21.67 284.38, 87.37 -67.96, -24.99 in-in in 9.0175 Saltbr-in 2.947 HRD-in -90.08, -55.75 70.92, 8.29 in-in-in SNCiii in-in ActLoopNT-in 2.9298 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.9, 155.75 APE9-dihe-na 129.48, -166.45 APE8-dihe-in -116.19, 135.64 APE8-rot-in 298.32 APE67-dihe-in -59.08, -26.0 -47.12, -51.73 APE12-dist-in 8.298 APE11-dist-in 11.4827 APE10-dist-in 5.9206 APE9-dist-in 3.8942 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.427 0.137 0.158 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 7pie Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIFA P25321 1 351 351.0 7QL:60401 Type1 Inactive DFGin 6.3465 14.218 ABAminus -118.69, -29.14 -100.96, 122.87 -127.55, 15.73 291.19, 87.86 -63.07, -33.16 in-in in 8.9572 Saltbr-in 2.7865 HRD-in -92.08, -57.05 70.77, -0.71 in-in-in SNCiii in-in ActLoopNT-in 2.9092 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.9, 150.21 APE9-dihe-na 133.66, -162.89 APE8-dihe-in -122.64, 134.78 APE8-rot-in 297.75 APE67-dihe-in -60.89, -24.83 -47.76, -50.71 APE12-dist-in 8.3006 APE11-dist-in 11.5735 APE10-dist-in 6.0009 APE9-dist-in 4.1345 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.395 0.135 0.155 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pif Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIGA P25321 1 351 351.0 7QR:60401 Type1 Inactive DFGin 6.4813 14.8758 ABAminus -122.28, -26.17 -100.91, 119.71 -123.06, 20.32 285.86, 92.34 -68.86, -24.06 in-in in 8.9216 Saltbr-in 2.7465 HRD-in -91.36, -59.49 70.09, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.9153 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.9, 150.63 APE9-dihe-na 129.65, -165.04 APE8-dihe-in -112.18, 133.86 APE8-rot-in 299.17 APE67-dihe-in -59.53, -25.5 -47.67, -52.22 APE12-dist-in 8.1547 APE11-dist-in 11.4414 APE10-dist-in 5.8432 APE9-dist-in 4.0681 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.553 0.129 0.154 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pig Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PNSA P25321 10 351 351.0 7W8:60402 Type1 Inactive DFGin 6.5137 14.8169 ABAminus -119.8, -32.67 -110.21, 109.27 -108.01, 28.37 286.1, 78.14 -68.46, -20.09 in-in in 8.9796 Saltbr-in 3.0843 HRD-in -83.54, -55.5 71.62, 9.07 in-in-in SNCiii in-in ActLoopNT-in 2.9078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.45, 157.3 APE9-dihe-na 125.01, -165.6 APE8-dihe-in -110.51, 134.07 APE8-rot-in 302.08 APE67-dihe-in -61.89, -24.52 -46.65, -50.8 APE12-dist-in 8.3238 APE11-dist-in 11.6189 APE10-dist-in 6.0319 APE9-dist-in 3.821 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.855 0.176 0.202 A 353.0 342.0 0 25 25 0 [[44, 298]] 1.0 7pns Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2BA P25321 5 351 351.0 9LQ:60401,9LQ:60402 Type1,Allosteric Inactive DFGin 6.3083 14.5013 ABAminus -99.36, -48.22 -103.96, 139.83 -136.93, 15.62 290.92, 85.14 -58.8, -40.25 in-in in 8.6839 Saltbr-in 2.8063 HRD-in -93.94, -54.86 69.46, 4.74 in-in-in SNCiii in-in ActLoopNT-in 2.9981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.47, 156.84 APE9-dihe-na 128.63, -164.41 APE8-dihe-in -116.79, 133.75 APE8-rot-in 301.48 APE67-dihe-in -59.49, -25.74 -49.19, -49.96 APE12-dist-in 8.1365 APE11-dist-in 11.6214 APE10-dist-in 6.0086 APE9-dist-in 3.9532 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.97 0.212 0.248 A 353.0 345.0 0 25 25 0 [[44, 298]] 1.0 6i2b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REKA P25321 12 351 351.0 D8P:60401,D8P:60402,D8P:60403,D8P:60404 Type1,Allosteric,Allosteric,Allosteric Inactive DFGin 6.3425 14.4394 ABAminus -107.25, -41.44 -100.58, 143.12 -128.51, 27.13 273.04, 65.71 -61.45, -23.67 in-in in 8.578 Saltbr-in 2.7782 HRD-in -87.09, -53.39 71.15, 12.36 in-in-in SNCiii in-in ActLoopNT-in 2.9003 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.7, 168.09 APE9-dihe-na 116.77, -166.86 APE8-dihe-in -118.41, 135.56 APE8-rot-in 302.89 APE67-dihe-in -59.2, -22.22 -49.04, -50.02 APE12-dist-in 8.1717 APE11-dist-in 11.1178 APE10-dist-in 5.6342 APE9-dist-in 3.7371 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.159 0.19 A 353.0 339.0 1 25 25 0 [[44, 298]] 1.0 9rek Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EM6A P25321 12 351 351.0 ADP:60401 ATPlike Inactive DFGin 6.8591 14.8208 BLAminus -128.32, 163.45 74.87, 92.52 -104.27, 28.45 286.23, 74.8 -62.75, -23.58 in-out in 9.7038 Saltbr-out 4.3621 HRD-in -85.36, -55.87 71.35, 12.71 out-in-in SNCoii in-in ActLoopNT-in 2.9302 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 157.75 APE9-dihe-na 127.42, -164.4 APE8-dihe-in -115.9, 133.37 APE8-rot-in 304.12 APE67-dihe-in -57.32, -23.54 -48.16, -51.44 APE12-dist-in 8.0456 APE11-dist-in 11.3093 APE10-dist-in 5.7368 APE9-dist-in 3.819 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.64 0.175 0.191 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6em6 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3NA P25321 12 351 351.0 152:60403 Allosteric Inactive DFGin 6.2448 14.3764 BLAminus -123.59, 163.17 75.18, 93.32 -100.77, 23.69 272.14, 54.48 -60.82, -27.27 in-in in 8.5509 Saltbr-in 2.932 HRD-in -86.04, -51.94 69.91, 12.31 in-in-out SNCiio in-out ActLoopNT-in 2.9316 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.97, 158.43 APE9-dihe-na 112.44, 164.79 APE8-dihe-in -81.93, 141.6 APE8-rot-out 194.34 APE67-dihe-in -62.51, -21.05 -48.48, -48.45 APE12-dist-in 8.1235 APE11-dist-in 11.1935 APE10-dist-in 5.687 APE9-dist-in 3.9939 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.224 0.136 0.153 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3n Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1GA P25321 12 351 351.0 8G5:60403 Allosteric Inactive DFGin 6.3509 14.2952 BLAminus -120.55, 160.72 78.08, 93.75 -100.89, 22.9 268.69, 55.04 -61.15, -25.02 in-in in 8.4501 Saltbr-in 2.8286 HRD-in -85.02, -51.99 68.33, 11.76 in-in-out SNCiio in-out ActLoopNT-in 2.9141 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.3, 157.42 APE9-dihe-na 113.47, 162.71 APE8-dihe-in -82.12, 143.17 APE8-rot-out 195.96 APE67-dihe-in -64.28, -21.72 -48.98, -46.63 APE12-dist-in 8.0256 APE11-dist-in 11.1323 APE10-dist-in 5.6526 APE9-dist-in 4.0142 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.14 0.129 0.141 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1g Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3RA P25321 13 351 351.0 CDT:60401 Allosteric Inactive DFGin 6.2835 14.3648 BLAminus -123.4, 166.85 72.82, 88.41 -96.79, 24.64 271.02, 57.62 -62.08, -26.42 in-in in 8.473 Saltbr-in 2.8507 HRD-in -84.5, -51.65 69.06, 12.07 in-in-out SNCiio in-out ActLoopNT-in 2.9132 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -163.54, 160.53 APE9-dihe-na 112.85, 168.5 APE8-dihe-in -90.49, 143.51 APE8-rot-out 194.17 APE67-dihe-in -64.82, -18.23 -48.56, -47.77 APE12-dist-in 8.01 APE11-dist-in 11.109 APE10-dist-in 5.6694 APE9-dist-in 3.7548 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.36 0.161 0.193 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5n3r Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REHA P25321 13 351 351.0 A1JEO:60410 Allosteric Inactive DFGin 6.3163 14.4571 BLAminus -120.51, 166.33 73.93, 87.07 -97.3, 23.53 273.58, 55.63 -62.98, -24.59 in-in in 8.6439 Saltbr-in 2.934 HRD-in -90.78, -53.04 70.2, 12.8 in-in-out SNCiio in-out ActLoopNT-in 2.9492 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.03, 159.17 APE9-dihe-na 115.21, 161.46 APE8-dihe-in -80.42, 146.14 APE8-rot-out 193.65 APE67-dihe-in -62.8, -23.48 -51.35, -45.43 APE12-dist-in 8.0609 APE11-dist-in 11.138 APE10-dist-in 5.6907 APE9-dist-in 3.9727 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.33 0.14 0.165 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9reh Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3GA P25321 12 351 351.0 8KB:60401,8KB:60402 Allosteric,Allosteric Inactive DFGin 6.2401 14.4188 BLAminus -122.61, 161.7 77.55, 93.02 -100.37, 23.32 270.97, 56.3 -63.09, -23.8 in-in in 8.5755 Saltbr-in 2.9043 HRD-in -86.82, -52.03 69.25, 11.52 in-in-out SNCiio in-out ActLoopNT-in 2.9346 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.35, 154.45 APE9-dihe-na 118.07, 158.61 APE8-dihe-in -78.39, 140.92 APE8-rot-out 196.18 APE67-dihe-in -62.0, -22.59 -47.89, -47.51 APE12-dist-in 8.0381 APE11-dist-in 11.2059 APE10-dist-in 5.7252 APE9-dist-in 4.1113 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.16 0.138 0.157 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3g Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REDA P25321 13 351 351.0 A1JEV:60401,A1JEV:60402 Allosteric,Allosteric Inactive DFGin 6.3136 14.3886 BLAminus -123.16, 164.73 74.85, 89.64 -97.97, 23.84 269.64, 57.8 -61.74, -25.67 in-in in 8.6392 Saltbr-in 2.8089 HRD-in -83.21, -53.37 69.6, 13.68 in-in-out SNCiio in-out ActLoopNT-in 2.9232 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.24, 157.71 APE9-dihe-na 113.1, 163.31 APE8-dihe-in -87.29, 142.42 APE8-rot-out 178.62 APE67-dihe-in -62.59, -21.07 -47.65, -46.78 APE12-dist-in 8.0505 APE11-dist-in 11.1849 APE10-dist-in 5.6941 APE9-dist-in 4.0315 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.31 0.156 0.179 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9red Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDWA P25321 13 351 351.0 A1JE6:60406,A1JE6:60407 Allosteric,Type1 Inactive DFGin 6.3634 14.4936 BLAminus -122.88, 162.57 78.68, 90.66 -100.96, 23.62 273.2, 61.49 -59.58, -26.11 in-in in 8.7111 Saltbr-in 2.8649 HRD-in -93.71, -51.31 69.07, 9.69 in-in-out SNCiio in-out ActLoopNT-in 2.9807 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.99, 155.73 APE9-dihe-na 118.94, 161.67 APE8-dihe-in -80.46, 143.29 APE8-rot-out 194.72 APE67-dihe-in -65.57, -17.76 -53.02, -44.37 APE12-dist-in 8.1355 APE11-dist-in 11.2237 APE10-dist-in 5.7423 APE9-dist-in 4.0797 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.44 0.154 0.164 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rdw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REJA P25321 12 351 351.0 A1JEM:60605,A1JEM:60606,A1JEM:60607 Allosteric,Type1,Allosteric Inactive DFGin 6.2324 14.4868 BLAminus -126.74, 170.31 72.72, 85.79 -95.11, 23.81 271.99, 61.49 -63.12, -25.09 in-in in 8.7773 Saltbr-in 2.7748 HRD-in -87.13, -50.88 67.77, 11.89 in-in-out SNCiio in-out ActLoopNT-in 2.908 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.08, 154.15 APE9-dihe-na 120.77, 160.5 APE8-dihe-in -80.28, 146.64 APE8-rot-out 196.83 APE67-dihe-in -64.07, -19.5 -50.27, -48.33 APE12-dist-in 8.0227 APE11-dist-in 11.1756 APE10-dist-in 5.6937 APE9-dist-in 4.0217 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.4 0.144 0.17 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rej Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SNNA P25321 13 351 351.0 BEZ:60401 Type1 Inactive DFGin 6.3179 14.5684 BLAminus -123.99, 166.66 75.94, 90.28 -99.21, 23.86 273.03, 56.25 -57.99, -30.08 in-in in 8.7995 Saltbr-in 2.708 HRD-in -85.26, -52.12 68.9, 15.2 in-in-out SNCiio in-out ActLoopNT-in 2.9021 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.87, 159.17 APE9-dihe-na 120.69, 167.55 APE8-dihe-in -88.31, 143.26 APE8-rot-out 194.47 APE67-dihe-in -64.07, -19.46 -52.28, -44.33 APE12-dist-in 8.0169 APE11-dist-in 11.2277 APE10-dist-in 5.7795 APE9-dist-in 4.1265 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.817 0.173 0.209 A 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 6snn Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1FA P25321 12 351 351.0 8ET:60403 Type1 Inactive DFGin 6.2781 14.42 BLAminus -125.76, 161.54 76.66, 90.69 -99.25, 24.03 270.12, 55.91 -61.05, -26.16 in-in in 8.6124 Saltbr-in 2.8119 HRD-in -86.34, -52.94 70.41, 12.62 in-in-out SNCiio in-out ActLoopNT-in 2.9272 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.69, 154.25 APE9-dihe-na 121.48, 156.96 APE8-dihe-in -75.85, 143.28 APE8-rot-out 195.81 APE67-dihe-in -63.37, -20.85 -47.21, -48.33 APE12-dist-in 8.0515 APE11-dist-in 11.1739 APE10-dist-in 5.7008 APE9-dist-in 4.0665 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.12 0.138 0.156 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1f Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1HA P25321 12 351 351.0 8G2:60403 Type1 Inactive DFGin 6.2538 14.418 BLAminus -124.07, 161.77 78.11, 91.86 -99.37, 24.42 270.96, 54.95 -60.37, -25.83 in-in in 8.5499 Saltbr-in 2.7935 HRD-in -86.51, -52.46 68.86, 12.98 in-in-out SNCiio in-out ActLoopNT-in 2.9142 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -157.77, 157.58 APE9-dihe-na 112.74, 163.68 APE8-dihe-in -79.44, 140.67 APE8-rot-out 196.71 APE67-dihe-in -63.37, -21.38 -49.53, -46.05 APE12-dist-in 8.0424 APE11-dist-in 11.1779 APE10-dist-in 5.7151 APE9-dist-in 4.0574 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.18 0.137 0.158 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1h Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3JA P25321 12 351 351.0 4NB:60402 Type1 Inactive DFGin 6.2627 14.559 BLAminus -127.12, 170.53 67.64, 82.17 -90.51, 22.12 271.33, 56.9 -61.6, -22.99 in-in in 8.8468 Saltbr-in 2.8105 HRD-in -84.57, -52.62 70.75, 13.79 in-in-out SNCiio in-out ActLoopNT-in 2.9356 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.46, 163.55 APE9-dihe-na 126.07, -167.14 APE8-dihe-in -114.74, 139.99 APE8-rot-out 192.96 APE67-dihe-in -63.96, -20.14 -47.5, -50.51 APE12-dist-in 8.1285 APE11-dist-in 11.1829 APE10-dist-in 5.6989 APE9-dist-in 3.7037 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.12 0.133 0.148 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3j Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3SA P25321 12 351 351.0 HBD:60401 Type1 Inactive DFGin 6.1499 14.4372 BLAminus -125.26, 171.68 71.74, 87.26 -96.68, 22.46 273.22, 56.06 -59.01, -26.75 in-in in 8.6435 Saltbr-in 2.8511 HRD-in -85.53, -52.56 69.97, 13.2 in-in-out SNCiio in-out ActLoopNT-in 2.9152 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.09, 170.83 APE9-dihe-na 117.86, -171.76 APE8-dihe-in -103.86, 138.88 APE8-rot-out 195.12 APE67-dihe-in -65.16, -19.12 -46.21, -48.93 APE12-dist-in 8.1219 APE11-dist-in 11.2071 APE10-dist-in 5.6952 APE9-dist-in 3.6672 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.14 0.129 0.148 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3s Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SOXA P25321 14 351 351.0 LQ2:60401 Type1 Inactive DFGin 6.2914 14.4415 BLAminus -122.0, 165.62 75.03, 89.05 -96.95, 24.43 271.3, 57.97 -61.84, -25.55 in-in in 8.6537 Saltbr-in 2.7949 HRD-in -85.89, -52.44 69.04, 12.72 in-in-out SNCiio in-out ActLoopNT-in 2.9118 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.24, 162.39 APE9-dihe-na 125.76, -160.57 APE8-dihe-in -123.53, 144.98 APE8-rot-out 197.35 APE67-dihe-in -66.0, -18.08 -49.52, -47.22 APE12-dist-in 8.0394 APE11-dist-in 11.1533 APE10-dist-in 5.5947 APE9-dist-in 3.7106 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.147 0.168 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6sox Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPMA P25321 14 351 351.0 3AE:60401 Type1 Inactive DFGin 6.2886 14.4262 BLAminus -121.91, 163.84 77.47, 92.46 -99.73, 24.27 270.82, 55.73 -61.57, -25.41 in-in in 8.5847 Saltbr-in 2.8251 HRD-in -85.39, -51.06 67.89, 13.49 in-in-out SNCiio in-out ActLoopNT-in 2.9167 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -161.47, 161.1 APE9-dihe-na 118.54, 176.4 APE8-dihe-in -99.11, 144.76 APE8-rot-out 192.34 APE67-dihe-in -65.21, -19.46 -48.83, -47.71 APE12-dist-in 8.0367 APE11-dist-in 11.1218 APE10-dist-in 5.6321 APE9-dist-in 3.8448 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.37 0.147 0.17 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6spm Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPUA P25321 14 351 351.0 GAB:60405 Type1 Inactive DFGin 6.3931 14.5224 BLAminus -124.88, 173.78 70.46, 84.77 -97.04, 23.36 270.78, 58.59 -61.61, -26.89 in-in in 8.6469 Saltbr-in 2.7353 HRD-in -87.8, -49.67 67.09, 13.22 in-in-out SNCiio in-out ActLoopNT-in 2.9411 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.63, 160.29 APE9-dihe-na 125.51, -175.3 APE8-dihe-in -107.62, 144.0 APE8-rot-out 190.74 APE67-dihe-in -65.31, -18.62 -49.85, -47.63 APE12-dist-in 8.0401 APE11-dist-in 11.2233 APE10-dist-in 5.7335 APE9-dist-in 3.8932 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.39 0.165 0.184 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6spu Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDYA P25321 13 351 351.0 A1JE4:60407 Type1 Inactive DFGin 6.5032 14.7795 BLAminus -119.69, 163.99 72.62, 91.41 -97.65, 26.8 272.41, 58.85 -66.3, -24.47 in-in in 8.7751 Saltbr-in 3.0572 HRD-in -86.22, -51.39 68.61, 15.07 in-in-out SNCiio in-out ActLoopNT-in 2.9911 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.15, 158.18 APE9-dihe-na 117.75, 172.26 APE8-dihe-in -89.12, 142.62 APE8-rot-out 194.5 APE67-dihe-in -65.89, -17.43 -50.54, -45.34 APE12-dist-in 8.1575 APE11-dist-in 11.3384 APE10-dist-in 5.8329 APE9-dist-in 4.0454 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.184 0.206 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rdy Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REBA P25321 13 351 351.0 A1JET:60401 Type1 Inactive DFGin 6.3729 14.4269 BLAminus -124.82, 162.22 74.38, 86.67 -95.22, 22.64 270.27, 61.04 -62.16, -23.18 in-in in 8.5836 Saltbr-in 2.7104 HRD-in -85.57, -50.84 67.51, 14.65 in-in-out SNCiio in-out ActLoopNT-in 2.9047 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.96, 159.88 APE9-dihe-na 110.85, 164.82 APE8-dihe-in -83.44, 140.37 APE8-rot-out 191.04 APE67-dihe-in -61.86, -20.69 -47.36, -48.95 APE12-dist-in 8.0333 APE11-dist-in 11.1411 APE10-dist-in 5.6672 APE9-dist-in 3.9355 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.39 0.146 0.174 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9reb Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RECA P25321 13 351 351.0 A1JEU:60402 Type1 Inactive DFGin 6.2807 14.4311 BLAminus -123.32, 165.4 76.33, 88.66 -97.16, 21.64 273.57, 56.99 -61.34, -25.37 in-in in 8.6041 Saltbr-in 2.883 HRD-in -87.05, -51.85 67.25, 12.73 in-in-out SNCiio in-out ActLoopNT-in 2.9375 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -157.22, 157.7 APE9-dihe-na 114.58, 158.78 APE8-dihe-in -77.9, 144.78 APE8-rot-out 194.34 APE67-dihe-in -63.76, -21.52 -52.55, -45.26 APE12-dist-in 8.0412 APE11-dist-in 11.196 APE10-dist-in 5.6992 APE9-dist-in 4.0387 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.2 0.152 0.165 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rec Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REFA P25321 13 351 351.0 D8J:60402 Type1 Inactive DFGin 6.2503 14.6131 BLAminus -124.89, 170.59 72.31, 85.37 -94.16, 22.8 273.07, 58.11 -60.12, -25.38 in-in in 8.8919 Saltbr-in 2.7356 HRD-in -89.11, -54.6 71.98, 11.51 in-in-out SNCiio in-out ActLoopNT-in 2.9454 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -155.33, 157.11 APE9-dihe-na 116.63, 160.22 APE8-dihe-in -78.97, 144.44 APE8-rot-out 195.25 APE67-dihe-in -62.66, -21.01 -52.14, -46.04 APE12-dist-in 8.1341 APE11-dist-in 11.1957 APE10-dist-in 5.704 APE9-dist-in 4.0979 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.144 0.177 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ref Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDVA P25321 13 351 351.0 A1JE7:60410,A1JE7:60411 Type1,Allosteric Inactive DFGin 6.2698 14.4325 BLAminus -128.08, 174.02 71.24, 86.46 -98.05, 22.19 274.06, 57.95 -62.58, -23.25 in-in in 8.6164 Saltbr-in 2.8851 HRD-in -88.5, -54.19 70.44, 9.88 in-in-out SNCiio in-out ActLoopNT-in 2.9638 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.52, 152.92 APE9-dihe-na 122.19, 162.12 APE8-dihe-in -80.5, 144.54 APE8-rot-out 193.25 APE67-dihe-in -65.71, -20.97 -51.75, -43.97 APE12-dist-in 8.0721 APE11-dist-in 11.1894 APE10-dist-in 5.7474 APE9-dist-in 4.0335 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.32 0.147 0.175 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rdv Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE5A P25321 13 351 351.0 A1JEY:60401,A1JEY:60402 Type1,Allosteric Inactive DFGin 6.3662 14.4036 BLAminus -125.27, 165.97 74.06, 89.04 -98.29, 23.47 275.71, 58.54 -58.28, -26.28 in-in in 8.6738 Saltbr-in 2.9443 HRD-in -85.09, -53.15 71.59, 14.35 in-in-out SNCiio in-out ActLoopNT-in 2.9386 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.17, 154.61 APE9-dihe-na 122.02, 168.03 APE8-dihe-in -83.24, 142.74 APE8-rot-out 202.42 APE67-dihe-in -65.84, -18.28 -53.64, -43.72 APE12-dist-in 8.1506 APE11-dist-in 11.2611 APE10-dist-in 5.782 APE9-dist-in 4.0696 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.198 0.235 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9re5 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REAA P25321 12 351 351.0 A1JES:60401,A1JES:60402 Type1,Allosteric Inactive DFGin 6.3101 14.3405 BLAminus -123.83, 166.44 72.66, 91.13 -99.23, 26.22 272.18, 57.96 -61.34, -25.61 in-in in 8.5784 Saltbr-in 2.748 HRD-in -86.86, -51.56 67.66, 14.6 in-in-out SNCiio in-out ActLoopNT-in 2.8985 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.49, 157.18 APE9-dihe-na 118.43, 162.88 APE8-dihe-in -80.84, 140.04 APE8-rot-out 193.72 APE67-dihe-in -64.73, -18.44 -50.69, -44.13 APE12-dist-in 8.0587 APE11-dist-in 11.2174 APE10-dist-in 5.7003 APE9-dist-in 4.039 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.52 0.182 0.207 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rea Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REGA P25321 12 351 351.0 A1JEP:60401,A1JEP:60402 Type1,Allosteric Inactive DFGin 6.4159 14.4433 BLAminus -118.38, 168.52 70.87, 88.51 -97.8, 23.03 272.83, 58.59 -60.46, -22.33 in-in in 8.5806 Saltbr-in 2.8704 HRD-in -87.51, -51.33 69.54, 7.76 in-in-out SNCiio in-out ActLoopNT-in 2.9211 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.94, 158.0 APE9-dihe-na 116.11, 163.67 APE8-dihe-in -82.8, 140.78 APE8-rot-out 193.33 APE67-dihe-in -64.93, -19.49 -46.8, -47.18 APE12-dist-in 8.0379 APE11-dist-in 11.2534 APE10-dist-in 5.7331 APE9-dist-in 3.9797 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.35 0.151 0.164 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9reg Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDUA P25321 13 351 351.0 A1JE8:60401,A1JE8:60402,A1JE8:60403 Type1,Allosteric,Allosteric Inactive DFGin 6.3019 14.4794 BLAminus -123.63, 166.88 73.88, 91.53 -100.44, 21.89 271.16, 60.35 -61.62, -25.71 in-in in 8.7016 Saltbr-in 2.8839 HRD-in -88.41, -52.06 67.0, 12.9 in-in-out SNCiio in-out ActLoopNT-in 2.9686 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.03, 154.41 APE9-dihe-na 120.3, 161.03 APE8-dihe-in -78.42, 143.41 APE8-rot-out 195.24 APE67-dihe-in -64.91, -19.59 -51.04, -45.3 APE12-dist-in 8.0736 APE11-dist-in 11.2223 APE10-dist-in 5.7369 APE9-dist-in 4.1351 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.158 0.17 A 353.0 338.0 1 25 25 0 [[44, 298]] 1.0 9rdu Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EH2A P25321 1 351 351.0 AMP:60401 ATPlike None DFGin 6.7638 14.9194 BLAminus -126.18, 164.33 76.56, 92.11 -105.87, 26.81 282.23, 79.7 -66.18, -22.24 in-none in 9.2259 Saltbr-none 999.0 HRD-in -87.75, -53.65 70.54, 10.24 none-in-in SNCnii in-in ActLoopNT-in 2.9384 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.34, 158.08 APE9-dihe-na 131.59, -168.87 APE8-dihe-in -114.41, 135.93 APE8-rot-in 298.36 APE67-dihe-in -58.8, -22.41 -48.5, -50.6 APE12-dist-in 8.2043 APE11-dist-in 11.4263 APE10-dist-in 5.8454 APE9-dist-in 3.7187 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.76 0.177 0.21 A 353.0 343.0 3 25 25 0 [[44, 298]] 1.0 6eh2 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5NTJA P25321 1 351 351.0 No_ligand No_ligand None DFGin 6.7578 15.5887 BLAminus -126.6, 164.17 70.8, 88.44 -97.34, 22.68 279.05, 78.65 -62.01, -27.43 in-none in 9.318 Saltbr-none 999.0 HRD-in -87.71, -52.99 72.74, 12.02 none-in-in SNCnii in-in ActLoopNT-in 2.9259 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.35, 157.73 APE9-dihe-na 127.06, -161.94 APE8-dihe-in -121.61, 135.07 APE8-rot-in 297.67 APE67-dihe-in -60.56, -23.81 -48.81, -50.06 APE12-dist-in 8.1845 APE11-dist-in 11.5082 APE10-dist-in 5.834 APE9-dist-in 3.6606 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.56 0.142 0.177 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 5ntj Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERUA P25321 1 351 351.0 No_ligand No_ligand None DFGin 6.7077 15.3522 BLAminus -122.01, 161.76 78.09, 83.83 -91.35, 27.07 283.0, 77.27 -61.22, -29.16 in-none in 9.3238 Saltbr-none 999.0 HRD-in -85.44, -56.28 74.88, 7.63 none-in-in SNCnii in-in ActLoopNT-in 2.8885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.17, 161.42 APE9-dihe-na 121.37, -170.91 APE8-dihe-in -112.44, 135.97 APE8-rot-in 301.67 APE67-dihe-in -61.32, -23.67 -50.09, -48.07 APE12-dist-in 8.2425 APE11-dist-in 11.5143 APE10-dist-in 5.8561 APE9-dist-in 3.6262 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.15 0.207 0.245 A 353.0 348.0 1 25 25 0 [[44, 298]] 1.0 6eru Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERVA P25321 1 351 351.0 No_ligand No_ligand None DFGin 6.7146 15.3924 BLAminus -125.08, 156.65 78.53, 86.88 -92.73, 25.79 280.28, 78.54 -65.37, -20.87 in-none in 9.2341 Saltbr-none 999.0 HRD-in -86.89, -53.48 76.44, 7.72 none-in-in SNCnii in-in ActLoopNT-in 2.9464 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.6, 158.99 APE9-dihe-na 121.28, -168.45 APE8-dihe-in -116.16, 134.01 APE8-rot-in 298.45 APE67-dihe-in -57.32, -26.83 -47.6, -49.92 APE12-dist-in 8.2352 APE11-dist-in 11.4876 APE10-dist-in 5.9397 APE9-dist-in 3.6445 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.06 0.181 0.217 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6erv Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y2OA P25321 1 351 351.0 O72:60406 Type1 None DFGin 6.4228 14.1352 BLAminus -118.81, 164.94 68.54, 89.57 -98.17, 23.6 280.79, 62.09 -51.58, -34.71 in-none in 8.664 Saltbr-none 999.0 HRD-in -99.33, -52.87 71.55, 6.25 none-in-in SNCnii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.56, 161.43 APE9-dihe-na 131.48, -155.68 APE8-dihe-in -122.0, 132.63 APE8-rot-in 297.96 APE67-dihe-in -62.6, -21.6 -48.71, -46.53 APE12-dist-in 8.1468 APE11-dist-in 11.4733 APE10-dist-in 5.9727 APE9-dist-in 3.6487 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.01 0.223 0.254 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6y2o Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7BB0A P25321 1 351 351.0 T7W:60401 Type1 None DFGin 6.693 15.1674 BLAminus -117.12, 156.8 84.07, 107.01 -120.86, 24.94 282.89, 80.35 -68.76, -26.06 in-none in 9.3444 Saltbr-none 999.0 HRD-in -88.11, -52.74 73.76, 5.71 none-in-in SNCnii in-in ActLoopNT-in 3.0151 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.84, 156.52 APE9-dihe-na 126.29, -168.37 APE8-dihe-in -114.04, 132.32 APE8-rot-in 303.32 APE67-dihe-in -60.17, -25.3 -47.27, -49.42 APE12-dist-in 8.2705 APE11-dist-in 11.5229 APE10-dist-in 5.9799 APE9-dist-in 3.7589 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.75 0.203 0.235 A 353.0 347.0 0 25 25 0 [[44, 298]] 1.0 7bb0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4WB8A P17612 16 351 351.0 ATP:60401 ATPlike Active DFGin 5.6838 14.4142 BLAminus -121.45, -177.2 62.67, 77.75 -91.98, 24.58 268.87, 53.09 -58.34, -31.51 in-in in 8.9131 Saltbr-in 2.7592 HRD-in -95.2, -52.32 70.44, 11.38 in-in-in SNCiii in-in ActLoopNT-in 2.9124 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.85, 164.58 APE9-dihe-na 131.46, -156.38 APE8-dihe-in -129.55, 139.43 APE8-rot-in 297.11 APE67-dihe-in -60.54, -22.69 -52.03, -49.04 APE12-dist-in 8.0978 APE11-dist-in 11.3919 APE10-dist-in 5.8266 APE9-dist-in 3.4975 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.164 0.184 A 337.0 336.0 0 25 25 0 [[44, 298]] 1.0 4wb8 Homo sapiens AGC_PRKACA_HUMAN AGC 4e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4WB5A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 5.5996 14.452 BLAminus -123.05, 176.84 68.94, 80.02 -91.46, 24.86 270.2, 52.92 -60.74, -31.43 in-in in 9.0296 Saltbr-in 2.7148 HRD-in -92.12, -52.84 69.8, 13.37 in-in-in SNCiii in-in ActLoopNT-in 2.9178 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.48, 163.75 APE9-dihe-na 132.31, -149.49 APE8-dihe-in -132.05, 134.14 APE8-rot-in 301.14 APE67-dihe-in -60.1, -21.12 -48.44, -50.23 APE12-dist-in 8.0121 APE11-dist-in 11.4001 APE10-dist-in 5.799 APE9-dist-in 3.5673 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.641 0.165 0.196 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 4wb5 Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4WB7A P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.4448 14.6485 BLAminus -119.06, -174.39 59.4, 77.28 -89.09, 26.42 267.74, 51.48 -60.48, -28.34 in-in in 8.8699 Saltbr-in 2.7695 HRD-in -93.55, -50.9 68.82, 8.95 in-in-in SNCiii in-in ActLoopNT-in 2.942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.63, 158.06 APE9-dihe-na 139.02, -156.91 APE8-dihe-in -126.94, 137.23 APE8-rot-in 299.54 APE67-dihe-in -64.26, -23.0 -50.4, -48.13 APE12-dist-in 8.1804 APE11-dist-in 11.5397 APE10-dist-in 5.9545 APE9-dist-in 3.7228 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 4wb7 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4WB7B P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.3799 14.7121 BLAminus -115.93, -176.79 62.38, 75.33 -88.91, 25.18 264.71, 51.71 -56.9, -30.26 in-in in 8.9624 Saltbr-in 2.7732 HRD-in -94.01, -50.55 67.24, 10.48 in-in-in SNCiii in-in ActLoopNT-in 2.9391 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.07, 161.39 APE9-dihe-na 132.31, -156.17 APE8-dihe-in -127.2, 138.18 APE8-rot-in 298.14 APE67-dihe-in -59.62, -23.37 -52.63, -48.78 APE12-dist-in 8.1977 APE11-dist-in 11.5627 APE10-dist-in 5.9704 APE9-dist-in 3.6419 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.152 0.188 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 4wb7 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6BYRA P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.6263 14.6159 BLAminus -128.29, 177.03 62.06, 86.64 -97.54, 28.59 271.87, 66.62 -63.2, -33.23 in-in in 8.8079 Saltbr-in 3.1965 HRD-in -87.43, -52.47 67.28, 5.18 in-in-in SNCiii in-in ActLoopNT-in 3.1931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.51, 153.24 APE9-dihe-na 149.32, -133.8 APE8-dihe-in -139.35, 133.91 APE8-rot-in 312.31 APE67-dihe-in -68.4, -6.95 -52.73, -48.25 APE12-dist-in 8.7341 APE11-dist-in 11.0763 APE10-dist-in 5.6298 APE9-dist-in 3.4915 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 6byr Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6BYRC P17612 2 351 351.0 ATP:60501 ATPlike Active DFGin 5.6794 14.3401 BLAminus -129.89, 172.29 61.76, 74.25 -79.2, 34.93 281.69, 54.14 -61.8, -27.34 in-in in 8.7335 Saltbr-in 2.4981 HRD-in -93.13, -49.8 64.55, 7.44 in-in-in SNCiii in-in ActLoopNT-in 3.0524 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.29, 161.94 APE9-dihe-na 130.51, -156.26 APE8-dihe-in -112.31, 134.09 APE8-rot-in 302.07 APE67-dihe-in -64.15, -16.52 -52.64, -41.39 APE12-dist-in 8.3162 APE11-dist-in 11.1062 APE10-dist-in 5.7667 APE9-dist-in 3.6182 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.661 0.203 0.249 C 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 6byr Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 9EDCA P17612 14 351 351.0 ATP:60400 ATPlike Active DFGin 5.6262 13.772 BLAminus -125.61, -173.52 60.53, 69.6 -81.59, 16.86 273.36, 51.23 -62.38, -30.28 in-in in 9.1286 Saltbr-in 2.9998 HRD-in -112.54, -46.7 65.17, 1.82 in-in-in SNCiii in-in ActLoopNT-in 3.1404 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.87, 159.92 APE9-dihe-na 136.42, -156.18 APE8-dihe-in -101.13, 126.83 APE8-rot-in 299.98 APE67-dihe-in -84.76, -8.6 -60.74, -28.35 APE12-dist-in 7.9989 APE11-dist-in 11.1115 APE10-dist-in 5.7968 APE9-dist-in 3.7475 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 EM 4.18 999.0 999.0 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9edc Homo sapiens AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4WB6A P17612 14 351 351.0 ATP:60401 ATPlike Active DFGin 6.0678 14.3977 BLAminus -118.38, -169.49 51.77, 82.47 -95.61, 17.78 271.18, 55.73 -42.8, -37.29 in-in in 8.8304 Saltbr-in 2.5613 HRD-in -94.17, -52.18 74.17, 2.46 in-in-in SNCiii in-in ActLoopNT-in 2.9483 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.55, 166.68 APE9-dihe-na 116.18, 128.45 APE8-dihe-in -46.62, 128.74 APE8-rot-in 303.5 APE67-dihe-in -58.01, -23.74 -49.09, -50.89 APE12-dist-in 8.0462 APE11-dist-in 11.764 APE10-dist-in 6.2427 APE9-dist-in 3.7665 L206R SEP11,SEP140,TPO198 SEP11,SEP140,TPO198 XRAY 2.1 0.19 0.237 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 4wb6 Homo sapiens AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4WB6B P17612 9 351 351.0 ATP:60401 ATPlike Active DFGin 5.8721 14.0727 BLAminus -117.82, -168.32 53.27, 78.35 -91.25, 29.34 274.97, 62.46 -60.26, -35.85 in-in in 8.6873 Saltbr-in 2.7501 HRD-in -101.62, -46.5 64.42, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.9461 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.38, 164.15 APE9-dihe-na 120.83, 133.18 APE8-dihe-in -48.66, 125.41 APE8-rot-in 298.86 APE67-dihe-in -54.58, -37.6 -53.55, -42.52 APE12-dist-in 8.078 APE11-dist-in 11.6173 APE10-dist-in 6.2035 APE9-dist-in 3.8221 L206R SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.19 0.237 B 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 4wb6 Homo sapiens AGC_PRKACA_HUMAN AGC 8.6e-94 319.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5J5XA P17612 10 351 351.0 6J9:60404 Allosteric Active DFGin 6.1307 14.2674 BLAminus -130.51, 173.14 68.75, 93.05 -105.74, 27.05 279.27, 61.24 -64.37, -20.92 in-in in 8.4945 Saltbr-in 2.7357 HRD-in -82.45, -52.91 66.97, 1.69 in-in-in SNCiii in-in ActLoopNT-in 2.8965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.53, 148.7 APE9-dihe-na 119.01, 165.11 APE8-dihe-in -70.44, 134.99 APE8-rot-in 296.24 APE67-dihe-in -60.26, -38.48 -54.53, -34.6 APE12-dist-in 7.8109 APE11-dist-in 11.1325 APE10-dist-in 5.6005 APE9-dist-in 3.9887 None TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.24 0.309 A 351.0 342.0 0 25 25 0 [[44, 298]] 1.0 5j5x Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN AF-P17612-K1A P17612 36 306 351.0 No_ligand No_ligand Active DFGin 5.9552 14.1005 BLAminus -112.06, -162.49 41.01, 73.74 -80.57, 22.27 279.02, 69.01 -57.23, -32.63 in-in in 8.7297 Saltbr-in 2.6065 HRD-in -81.22, -48.08 66.27, 5.12 in-in-in SNCiii in-in ActLoopNT-in 2.9414 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.31, 161.49 APE9-dihe-na 113.97, -179.99 APE8-dihe-in -91.88, 135.09 APE8-rot-in 302.21 APE67-dihe-in -65.91, -23.79 -48.59, -45.69 APE12-dist-in 8.0558 APE11-dist-in 11.4784 APE10-dist-in 5.7165 APE9-dist-in 3.4962 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 25 25 0 [[44, 298]] 1.0 AF-P17612-K1 Homo sapiens AGC_PRKACA_HUMAN AGC 1.8e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN AF-P17612-K3A P17612 36 306 351.0 No_ligand No_ligand Active DFGin 5.9894 14.1821 BLAminus -127.06, -175.23 47.34, 85.15 -88.29, 17.62 289.75, 82.76 -56.25, -31.52 in-in in 8.7982 Saltbr-in 2.6486 HRD-in -85.43, -51.15 69.13, 5.21 in-in-in SNCiii in-in ActLoopNT-in 2.8708 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.07, 161.67 APE9-dihe-na 110.83, -179.43 APE8-dihe-in -90.4, 132.09 APE8-rot-in 300.17 APE67-dihe-in -66.95, -21.36 -48.38, -45.21 APE12-dist-in 8.0717 APE11-dist-in 11.1565 APE10-dist-in 5.4898 APE9-dist-in 3.4162 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 25 25 0 [[44, 298]] 1.0 AF-P17612-K3 Homo sapiens AGC_PRKACA_HUMAN AGC 1.8e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6NO7C P17612 12 351 351.0 No_ligand No_ligand Active DFGin 5.3091 14.0414 BLAminus -119.31, 176.37 65.24, 77.94 -84.43, 19.43 273.37, 51.07 -43.97, -41.52 in-in in 8.987 Saltbr-in 2.3597 HRD-in -94.38, -54.81 73.77, 10.87 in-in-in SNCiii in-in ActLoopNT-in 2.9661 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.7, 149.95 APE9-dihe-na 149.29, -142.75 APE8-dihe-in -132.31, 130.88 APE8-rot-in 297.15 APE67-dihe-in -65.36, -25.54 -38.33, -55.04 APE12-dist-in 8.372 APE11-dist-in 10.8625 APE10-dist-in 5.5723 APE9-dist-in 3.1598 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 C 350.0 340.0 0 25 25 0 [[44, 298]] 1.0 6no7 Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3AGMA P17612 13 351 351.0 No_ligand No_ligand Active DFGin 6.4463 13.4021 BLAminus -121.71, 165.51 70.43, 93.14 -102.22, 24.88 291.91, 69.39 -56.91, -34.43 in-in in 8.7602 Saltbr-in 2.8017 HRD-in -90.0, -49.9 65.54, 1.86 in-in-in SNCiii in-in ActLoopNT-in 2.9866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.66, 155.53 APE9-dihe-na 129.13, -155.89 APE8-dihe-in -119.08, 128.77 APE8-rot-in 315.26 APE67-dihe-in -58.72, -28.41 -42.89, -48.17 APE12-dist-in 7.9624 APE11-dist-in 11.3404 APE10-dist-in 5.7893 APE9-dist-in 3.8393 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.277 0.265 A 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 3agm Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5IZFA P17612 14 351 351.0 No_ligand No_ligand Active DFGin 6.4693 14.6805 BLAminus -115.33, 168.85 66.79, 92.72 -104.07, 26.57 271.02, 67.91 -60.32, -26.19 in-in in 8.9198 Saltbr-in 2.86 HRD-in -91.12, -53.12 70.24, 3.28 in-in-in SNCiii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.28, 154.6 APE9-dihe-na 132.55, -178.51 APE8-dihe-in -93.41, 131.47 APE8-rot-in 300.25 APE67-dihe-in -61.6, -25.88 -48.77, -44.1 APE12-dist-in 7.9991 APE11-dist-in 11.6508 APE10-dist-in 5.9844 APE9-dist-in 4.1432 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.232 0.27 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 5izf Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3NX8A P17612 16 351 351.0 No_ligand No_ligand Active DFGin 6.2174 14.3207 BLAminus -121.41, 174.36 68.59, 92.57 -100.19, 21.71 266.05, 56.03 -54.66, -29.9 in-in in 8.8669 Saltbr-in 3.0948 HRD-in -83.14, -56.31 66.43, 12.16 in-in-in SNCiii in-in ActLoopNT-in 3.0216 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.5, 160.02 APE9-dihe-na 128.98, -158.22 APE8-dihe-in -117.99, 132.74 APE8-rot-in 294.49 APE67-dihe-in -53.23, -32.68 -47.46, -50.82 APE12-dist-in 8.0488 APE11-dist-in 11.4278 APE10-dist-in 5.8527 APE9-dist-in 3.6257 None TPO198,SEP339 TPO198,LGY293,SEP339 XRAY 2.0 0.22 0.288 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 3nx8 Homo sapiens AGC_PRKACA_HUMAN AGC 2.9e-94 321.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 9DCDA P17612 14 351 351.0 A1A3J:60401 Type1 Active DFGin 5.9288 14.45 BLAminus -126.13, 173.68 64.63, 91.94 -99.88, 28.46 273.99, 56.84 -61.81, -26.4 in-in in 9.1249 Saltbr-in 2.7292 HRD-in -91.13, -53.48 71.25, 11.66 in-in-in SNCiii in-in ActLoopNT-in 2.8197 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.7, 158.74 APE9-dihe-na 136.61, -155.83 APE8-dihe-in -120.28, 133.14 APE8-rot-in 302.66 APE67-dihe-in -56.79, -23.93 -44.41, -54.9 APE12-dist-in 8.0289 APE11-dist-in 11.4422 APE10-dist-in 5.9126 APE9-dist-in 3.6174 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.7 0.174 0.191 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9dcd Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3AGLA P17612 11 351 351.0 A03:60351 Type1 Active DFGin 6.145 14.1866 BLAminus -123.32, 177.62 64.25, 83.52 -96.46, 22.51 272.11, 61.62 -58.64, -28.46 in-in in 8.4913 Saltbr-in 2.8863 HRD-in -82.44, -53.5 74.32, 9.67 in-in-in SNCiii in-in ActLoopNT-in 2.8897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.19, 166.18 APE9-dihe-na 128.76, -154.1 APE8-dihe-in -126.1, 126.27 APE8-rot-in 292.64 APE67-dihe-in -59.45, -23.51 -43.73, -52.47 APE12-dist-in 8.0899 APE11-dist-in 11.2847 APE10-dist-in 5.6424 APE9-dist-in 3.6922 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.2 0.237 A 351.0 341.0 0 25 25 0 [[44, 298]] 1.0 3agl Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3AGLB P17612 15 351 351.0 A03:60351 Type1 Active DFGin 6.244 14.2587 BLAminus -119.17, 172.99 64.04, 88.92 -97.96, 24.36 271.27, 65.91 -60.24, -24.04 in-in in 8.4832 Saltbr-in 2.838 HRD-in -81.23, -56.2 72.88, 10.89 in-in-in SNCiii in-in ActLoopNT-in 2.8655 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.17, 153.35 APE9-dihe-na 137.51, -153.25 APE8-dihe-in -122.43, 130.68 APE8-rot-in 303.24 APE67-dihe-in -59.0, -24.94 -49.14, -44.94 APE12-dist-in 8.0815 APE11-dist-in 11.3224 APE10-dist-in 5.744 APE9-dist-in 3.8805 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.2 0.237 B 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3agl Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3L9LA P17612 12 351 351.0 L9L:60351 Type1 Active DFGin 6.6864 14.5845 BLAminus -131.42, 170.84 67.14, 98.79 -112.52, 31.48 281.78, 68.95 -76.6, -5.02 in-in in 9.118 Saltbr-in 3.0215 HRD-in -66.86, -56.55 70.6, 11.25 in-in-in SNCiii in-in ActLoopNT-in 2.8997 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.79, 159.06 APE9-dihe-na 115.3, -161.08 APE8-dihe-in -112.72, 124.05 APE8-rot-in 306.01 APE67-dihe-in -58.13, -24.33 -29.04, -60.55 APE12-dist-in 8.3496 APE11-dist-in 11.1877 APE10-dist-in 5.5865 APE9-dist-in 3.5153 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.262 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 3l9l Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3L9LB P17612 13 351 351.0 L9L:60351 Type1 Active DFGin 6.5037 14.7481 BLAminus -126.06, 169.3 70.23, 93.91 -105.72, 28.14 277.25, 72.68 -68.61, -5.61 in-in in 9.1221 Saltbr-in 3.0925 HRD-in -71.18, -54.73 64.89, 13.74 in-in-in SNCiii in-in ActLoopNT-in 2.96 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.39, 167.34 APE9-dihe-na 115.39, -170.56 APE8-dihe-in -110.93, 132.83 APE8-rot-in 304.32 APE67-dihe-in -49.56, -29.7 -32.05, -69.65 APE12-dist-in 8.223 APE11-dist-in 11.2936 APE10-dist-in 5.685 APE9-dist-in 3.5296 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.262 B 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 3l9l Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3OOGA P17612 17 351 351.0 YTP:62001 Type1 Active DFGin 5.8967 14.3236 BLAminus -121.7, 177.27 65.88, 89.72 -99.72, 18.72 271.46, 61.56 -55.08, -24.51 in-in in 9.0925 Saltbr-in 2.5643 HRD-in -88.93, -49.19 62.2, 8.05 in-in-in SNCiii in-in ActLoopNT-in 2.8865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.22, 156.24 APE9-dihe-na 130.48, -158.98 APE8-dihe-in -121.53, 132.57 APE8-rot-in 295.61 APE67-dihe-in -56.76, -31.12 -46.34, -49.72 APE12-dist-in 8.1836 APE11-dist-in 11.5607 APE10-dist-in 5.9904 APE9-dist-in 3.7821 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.276 A 351.0 335.0 0 25 25 0 [[44, 298]] 1.0 3oog Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3OVVA P17612 15 351 351.0 1SB:62001 Type1 Active DFGin 5.6952 14.513 BLAminus -122.03, 173.75 63.75, 85.64 -91.93, 24.88 270.34, 49.38 -58.53, -29.2 in-in in 9.1567 Saltbr-in 2.6429 HRD-in -85.42, -51.64 68.38, 18.21 in-in-in SNCiii in-in ActLoopNT-in 2.9726 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.97, 161.66 APE9-dihe-na 131.92, -151.97 APE8-dihe-in -126.88, 132.92 APE8-rot-in 299.89 APE67-dihe-in -61.32, -22.22 -45.4, -52.6 APE12-dist-in 8.1277 APE11-dist-in 11.5503 APE10-dist-in 5.9067 APE9-dist-in 3.5315 None TPO198,SEP339 TPO198,SEP339 XRAY 1.58 0.186 0.232 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3ovv Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3OWPA P17612 16 351 351.0 2SB:62001 Type1 Active DFGin 5.7967 14.5771 BLAminus -129.79, 179.44 68.22, 88.81 -97.88, 23.63 269.47, 50.63 -59.8, -24.73 in-in in 9.0211 Saltbr-in 2.6482 HRD-in -91.6, -55.1 70.56, 10.08 in-in-in SNCiii in-in ActLoopNT-in 2.8362 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.46, 156.32 APE9-dihe-na 133.26, -159.94 APE8-dihe-in -117.71, 131.95 APE8-rot-in 303.89 APE67-dihe-in -56.68, -26.5 -44.05, -53.81 APE12-dist-in 8.0794 APE11-dist-in 11.5299 APE10-dist-in 5.9471 APE9-dist-in 3.8249 None TPO198,SEP339 TPO198,SEP339 XRAY 1.88 0.172 0.211 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 3owp Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3OXTA P17612 15 351 351.0 3SB:62001 Type1 Active DFGin 5.7237 14.3223 BLAminus -130.49, 176.59 67.71, 88.75 -96.86, 20.88 271.58, 55.14 -54.8, -35.77 in-in in 9.1078 Saltbr-in 2.754 HRD-in -88.64, -56.71 72.64, 4.73 in-in-in SNCiii in-in ActLoopNT-in 2.7833 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.01, 154.62 APE9-dihe-na 133.52, -155.05 APE8-dihe-in -117.36, 129.13 APE8-rot-in 302.02 APE67-dihe-in -56.32, -26.92 -42.89, -52.47 APE12-dist-in 8.2687 APE11-dist-in 11.8606 APE10-dist-in 6.2609 APE9-dist-in 4.1093 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.176 0.239 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3oxt Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3P0MA P17612 15 351 351.0 4SB:60351 Type1 Active DFGin 5.9227 14.5783 BLAminus -120.95, -179.03 59.8, 84.94 -96.45, 19.28 269.08, 54.31 -49.85, -35.86 in-in in 9.0006 Saltbr-in 2.6601 HRD-in -87.41, -52.38 71.61, 9.65 in-in-in SNCiii in-in ActLoopNT-in 2.9521 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.78, 160.64 APE9-dihe-na 131.62, -157.52 APE8-dihe-in -119.88, 133.57 APE8-rot-in 304.97 APE67-dihe-in -52.04, -26.97 -43.23, -57.05 APE12-dist-in 8.0193 APE11-dist-in 11.4768 APE10-dist-in 5.8873 APE9-dist-in 3.6581 None TPO198,SEP339 TPO198,SEP339 XRAY 2.03 0.171 0.205 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3p0m Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3POOA P17612 15 351 351.0 S69:62001 Type1 Active DFGin 5.6882 14.66 BLAminus -122.77, 177.28 59.44, 86.58 -95.62, 24.37 267.18, 52.33 -56.67, -28.22 in-in in 9.2255 Saltbr-in 2.6135 HRD-in -88.33, -52.91 73.26, 10.11 in-in-in SNCiii in-in ActLoopNT-in 2.9542 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.96, 158.93 APE9-dihe-na 133.77, -158.97 APE8-dihe-in -121.67, 134.24 APE8-rot-in 298.67 APE67-dihe-in -57.61, -22.88 -45.78, -52.79 APE12-dist-in 8.0956 APE11-dist-in 11.5265 APE10-dist-in 5.9381 APE9-dist-in 3.5559 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.187 0.212 A 351.0 333.0 0 25 25 0 [[44, 298]] 1.0 3poo Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3VQHA P17612 5 351 351.0 IQB:60401 Type1 Active DFGin 5.8868 14.5091 BLAminus -116.4, -175.47 66.0, 75.68 -94.16, 21.7 272.84, 60.82 -59.14, -31.37 in-in in 8.8982 Saltbr-in 2.6912 HRD-in -94.63, -51.76 70.89, 9.84 in-in-in SNCiii in-in ActLoopNT-in 2.8756 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.13, 162.63 APE9-dihe-na 132.63, -148.92 APE8-dihe-in -128.75, 132.36 APE8-rot-in 300.65 APE67-dihe-in -61.72, -25.75 -46.04, -48.59 APE12-dist-in 8.0578 APE11-dist-in 11.5232 APE10-dist-in 5.8417 APE9-dist-in 3.6408 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.95 0.192 0.234 A 351.0 347.0 0 25 25 0 [[44, 298]] 1.0 3vqh Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4UJ1A P17612 15 351 351.0 NVX:61351 Type1 Active DFGin 6.2416 14.5472 BLAminus -123.61, -163.8 61.68, 70.56 -93.64, 20.6 271.48, 60.79 -64.78, -20.97 in-in in 9.0378 Saltbr-in 2.5518 HRD-in -90.63, -51.42 73.4, 9.87 in-in-in SNCiii in-in ActLoopNT-in 2.9745 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.01, 158.56 APE9-dihe-na 139.11, -156.28 APE8-dihe-in -125.77, 137.11 APE8-rot-in 295.71 APE67-dihe-in -57.89, -23.24 -51.45, -49.94 APE12-dist-in 8.1202 APE11-dist-in 11.3926 APE10-dist-in 5.8666 APE9-dist-in 3.6245 None TPO198,SEP339 TPO198,SEP339 XRAY 1.768 0.168 0.201 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4uj1 Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4UJ2A P17612 15 351 351.0 NVV:61351 Type1 Active DFGin 6.3807 14.5704 BLAminus -125.67, -160.4 61.32, 58.86 -86.58, 22.47 272.1, 62.19 -53.53, -31.63 in-in in 9.0784 Saltbr-in 2.6406 HRD-in -86.14, -55.69 77.07, 9.76 in-in-in SNCiii in-in ActLoopNT-in 2.9495 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.59, 157.48 APE9-dihe-na 137.97, -154.25 APE8-dihe-in -126.65, 132.96 APE8-rot-in 298.62 APE67-dihe-in -53.02, -26.32 -44.15, -55.11 APE12-dist-in 8.245 APE11-dist-in 11.6516 APE10-dist-in 6.1174 APE9-dist-in 3.5607 None TPO198,SEP339 TPO198,SEP339 XRAY 2.019 0.165 0.209 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4uj2 Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4UJ9A P17612 11 351 351.0 S3N:61351 Type1 Active DFGin 6.1337 14.6501 BLAminus -117.52, -171.14 58.79, 71.43 -92.02, 19.19 269.08, 56.18 -56.86, -27.59 in-in in 8.9204 Saltbr-in 2.5062 HRD-in -93.86, -53.97 74.6, 12.42 in-in-in SNCiii in-in ActLoopNT-in 2.9172 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.92, 155.16 APE9-dihe-na 141.7, -146.62 APE8-dihe-in -127.44, 135.95 APE8-rot-in 296.91 APE67-dihe-in -56.69, -21.29 -47.92, -48.81 APE12-dist-in 7.952 APE11-dist-in 11.4276 APE10-dist-in 5.8483 APE9-dist-in 3.4787 None TPO198,SEP339 TPO198,SEP339 XRAY 1.87 0.167 0.206 A 351.0 341.0 0 25 25 0 [[44, 298]] 1.0 4uj9 Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4UJAA P17612 14 351 351.0 4L7:61351 Type1 Active DFGin 6.0974 14.6131 BLAminus -125.31, -163.62 62.94, 64.42 -88.89, 21.72 270.4, 58.9 -55.44, -30.93 in-in in 9.0487 Saltbr-in 2.7771 HRD-in -87.37, -51.28 70.71, 6.14 in-in-in SNCiii in-in ActLoopNT-in 2.9072 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.5, 162.38 APE9-dihe-na 130.88, -155.58 APE8-dihe-in -125.03, 133.85 APE8-rot-in 299.16 APE67-dihe-in -59.42, -24.42 -46.24, -50.45 APE12-dist-in 8.1686 APE11-dist-in 11.5131 APE10-dist-in 5.9673 APE9-dist-in 3.5887 None TPO198,SEP339 TPO198,SEP339 XRAY 1.93 0.166 0.206 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4uja Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4UJBA P17612 5 351 351.0 8BQ:61351 Type1 Active DFGin 5.9468 14.6677 BLAminus -125.29, -162.0 58.42, 69.71 -90.44, 19.28 267.91, 58.77 -53.57, -31.33 in-in in 9.135 Saltbr-in 2.7431 HRD-in -89.96, -52.14 72.96, 12.71 in-in-in SNCiii in-in ActLoopNT-in 2.9078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.56, 161.27 APE9-dihe-na 132.43, -159.75 APE8-dihe-in -122.62, 132.75 APE8-rot-in 302.43 APE67-dihe-in -59.14, -27.14 -46.68, -47.07 APE12-dist-in 8.1376 APE11-dist-in 11.4555 APE10-dist-in 5.9421 APE9-dist-in 3.6035 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.949 0.156 0.19 A 351.0 347.0 0 25 25 0 [[44, 298]] 1.0 4ujb Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5BX6A P17612 6 351 351.0 495:60401 Type1 Active DFGin 6.1832 14.3031 BLAminus -119.55, 164.86 70.92, 91.57 -100.18, 26.65 271.79, 52.76 -61.33, -23.25 in-in in 8.9062 Saltbr-in 2.708 HRD-in -93.87, -50.75 70.32, 10.63 in-in-in SNCiii in-in ActLoopNT-in 2.9595 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.15, 164.21 APE9-dihe-na 125.51, -162.2 APE8-dihe-in -117.48, 134.41 APE8-rot-in 303.65 APE67-dihe-in -56.37, -27.52 -46.12, -51.63 APE12-dist-in 8.0749 APE11-dist-in 11.4551 APE10-dist-in 5.918 APE9-dist-in 3.6014 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.89 0.172 0.218 A 351.0 346.0 0 25 25 0 [[44, 298]] 1.0 5bx6 Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5BX7A P17612 6 350 351.0 4W1:60401 Type1 Active DFGin 5.8928 14.2566 BLAminus -120.21, 170.97 66.4, 95.24 -104.96, 26.38 271.55, 55.44 -58.59, -27.02 in-in in 8.8868 Saltbr-in 2.6463 HRD-in -91.82, -48.84 66.55, 10.61 in-in-in SNCiii in-in ActLoopNT-in 2.9359 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.67, 162.65 APE9-dihe-na 129.46, -159.53 APE8-dihe-in -119.63, 133.68 APE8-rot-in 305.25 APE67-dihe-in -56.25, -25.43 -45.01, -52.75 APE12-dist-in 8.1102 APE11-dist-in 11.5179 APE10-dist-in 5.9614 APE9-dist-in 3.5807 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.89 0.178 0.226 A 351.0 345.0 0 25 25 0 [[44, 298]] 1.0 5bx7 Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5UZKA P17612 15 351 351.0 504:60401 Type1 Active DFGin 6.3811 13.9478 BLAminus -125.23, 159.32 70.49, 97.31 -104.94, 23.81 281.36, 67.83 -60.03, -27.16 in-in in 8.8803 Saltbr-in 2.7654 HRD-in -81.16, -49.29 61.5, 17.59 in-in-in SNCiii in-in ActLoopNT-in 2.9206 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.44, 160.74 APE9-dihe-na 127.01, -154.99 APE8-dihe-in -117.26, 132.5 APE8-rot-in 297.37 APE67-dihe-in -55.36, -26.76 -39.46, -56.34 APE12-dist-in 8.0111 APE11-dist-in 11.3938 APE10-dist-in 5.8297 APE9-dist-in 3.5881 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.191 0.253 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 5uzk Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6QJ7A P17612 14 351 351.0 J4B:60401 Type1 Active DFGin 6.3708 14.8786 BLAminus -117.39, 169.65 69.58, 85.56 -98.1, 21.35 272.03, 58.03 -54.77, -30.7 in-in in 9.2139 Saltbr-in 2.7504 HRD-in -87.29, -50.94 66.9, 9.43 in-in-in SNCiii in-in ActLoopNT-in 2.94 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.01, 157.32 APE9-dihe-na 126.55, -163.63 APE8-dihe-in -112.81, 131.54 APE8-rot-in 300.45 APE67-dihe-in -57.75, -27.43 -43.16, -51.25 APE12-dist-in 8.0042 APE11-dist-in 11.5059 APE10-dist-in 5.846 APE9-dist-in 3.703 None TPO198,SEP339 TPO198,SEP339 XRAY 1.69 0.179 0.214 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 6qj7 Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3MVJA P17612 16 351 351.0 XFE:60351 Type1 Active DFGin 6.1884 13.5821 BLAminus -115.88, 169.36 72.34, 84.05 -100.4, 21.07 284.54, 72.78 -48.33, -32.34 in-in in 8.6933 Saltbr-in 2.9429 HRD-in -94.45, -57.98 81.77, 7.12 in-in-in SNCiii in-in ActLoopNT-in 3.0047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.5, 165.11 APE9-dihe-na 130.23, -153.23 APE8-dihe-in -130.91, 127.14 APE8-rot-in 305.92 APE67-dihe-in -54.4, -32.7 -46.27, -53.24 APE12-dist-in 8.1645 APE11-dist-in 11.4405 APE10-dist-in 5.835 APE9-dist-in 3.6782 None TPO198,SEP339 TPO198,SEP339 XRAY 2.49 0.217 0.304 A 371.0 336.0 0 25 25 0 [[44, 298]] 1.0 3mvj Homo sapiens AGC_PRKACA_HUMAN AGC 5.4e-95 323.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3MVJE P17612 16 351 351.0 XFE:60351 Type1 Active DFGin 6.0097 13.9041 BLAminus -120.77, 173.49 75.79, 91.53 -105.05, 22.03 286.9, 73.04 -48.68, -45.44 in-in in 8.7857 Saltbr-in 2.5037 HRD-in -85.62, -59.75 66.22, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.9875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.99, 156.89 APE9-dihe-na 143.78, -161.15 APE8-dihe-in -124.44, 132.79 APE8-rot-in 305.29 APE67-dihe-in -69.91, -25.33 -54.9, -34.25 APE12-dist-in 8.1481 APE11-dist-in 11.447 APE10-dist-in 5.8027 APE9-dist-in 3.8015 None TPO198,SEP339 TPO198,SEP339 XRAY 2.49 0.217 0.304 E 371.0 336.0 0 25 25 0 [[44, 298]] 1.0 3mvj Homo sapiens AGC_PRKACA_HUMAN AGC 5.4e-95 323.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3L9MA P17612 12 351 351.0 L9M:60351 Type1 Active DFGin 6.7018 13.6799 BLAminus -123.42, 168.26 64.27, 97.86 -112.03, 32.77 297.13, 76.75 -74.15, -5.52 in-in in 9.0347 Saltbr-in 2.7926 HRD-in -71.88, -60.17 71.32, 14.02 in-in-in SNCiii in-in ActLoopNT-in 2.8886 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.62, 165.36 APE9-dihe-na 118.63, -161.51 APE8-dihe-in -116.7, 125.6 APE8-rot-in 304.73 APE67-dihe-in -59.86, -22.26 -32.71, -59.17 APE12-dist-in 8.1871 APE11-dist-in 11.2087 APE10-dist-in 5.6173 APE9-dist-in 3.5714 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.223 0.27 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 3l9m Homo sapiens AGC_PRKACA_HUMAN AGC 5.8e-95 323.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3L9MB P17612 14 351 351.0 L9M:60351 Type1 Active DFGin 6.7673 13.7383 BLAminus -124.39, 166.06 67.02, 98.19 -111.82, 31.79 294.5, 74.52 -67.48, -11.73 in-in in 8.8779 Saltbr-in 2.9129 HRD-in -76.18, -53.82 65.92, 13.75 in-in-in SNCiii in-in ActLoopNT-in 2.9242 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.4, 166.8 APE9-dihe-na 115.45, -164.35 APE8-dihe-in -115.85, 130.97 APE8-rot-in 297.34 APE67-dihe-in -54.51, -26.46 -29.85, -67.98 APE12-dist-in 8.2238 APE11-dist-in 11.2629 APE10-dist-in 5.6584 APE9-dist-in 3.5585 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.223 0.27 B 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 3l9m Homo sapiens AGC_PRKACA_HUMAN AGC 5.8e-95 323.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3L9NA P17612 15 351 351.0 L9N:60351 Type1 Active DFGin 6.4227 13.4597 BLAminus -123.73, 167.95 65.98, 97.53 -115.01, 25.76 300.78, 81.96 -66.98, -19.82 in-in in 9.0504 Saltbr-in 2.7445 HRD-in -67.38, -52.97 66.43, 17.24 in-in-in SNCiii in-in ActLoopNT-in 2.9582 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.06, 165.76 APE9-dihe-na 122.47, -160.51 APE8-dihe-in -116.6, 130.05 APE8-rot-in 304.11 APE67-dihe-in -53.81, -24.08 -30.84, -70.07 APE12-dist-in 8.1973 APE11-dist-in 11.3941 APE10-dist-in 5.9345 APE9-dist-in 3.5534 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.217 0.257 A 351.0 334.0 0 25 25 0 [[44, 298]] 1.0 3l9n Homo sapiens AGC_PRKACA_HUMAN AGC 5.8e-95 323.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8FE2A P17612 4 351 351.0 XTI:60501 Type1 Active DFGin 6.1423 13.9131 BLAminus -123.85, 174.03 69.38, 86.41 -105.22, 28.0 281.98, 71.1 -68.62, -14.04 in-in in 8.8535 Saltbr-in 2.5144 HRD-in -84.66, -51.16 67.93, 20.04 in-in-in SNCiii in-in ActLoopNT-in 2.7913 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.46, 164.95 APE9-dihe-na 122.51, -154.32 APE8-dihe-in -114.26, 125.71 APE8-rot-in 301.9 APE67-dihe-in -53.15, -32.01 -48.08, -46.83 APE12-dist-in 8.3148 APE11-dist-in 11.573 APE10-dist-in 6.0032 APE9-dist-in 3.9389 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.34 0.199 0.251 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fe2 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8FE2B P17612 4 351 351.0 XTI:60501 Type1 Active DFGin 6.2269 13.875 BLAminus -121.06, -174.83 58.15, 84.69 -101.22, 28.39 282.36, 54.58 -64.33, -23.67 in-in in 8.8613 Saltbr-in 2.9356 HRD-in -86.41, -49.46 70.11, 7.42 in-in-in SNCiii in-in ActLoopNT-in 2.9286 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.54, 160.4 APE9-dihe-na 134.47, -156.72 APE8-dihe-in -118.93, 133.24 APE8-rot-in 292.47 APE67-dihe-in -59.44, -24.84 -53.68, -43.95 APE12-dist-in 8.1124 APE11-dist-in 11.5096 APE10-dist-in 5.8745 APE9-dist-in 3.7916 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.34 0.199 0.251 B 405.0 333.0 0 25 25 0 [[44, 298]] 1.0 8fe2 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8FE5A P17612 3 351 351.0 XTT:60501 Type1 Active DFGin 6.5996 14.2711 BLAminus -118.08, 163.41 75.28, 94.71 -111.66, 23.11 283.47, 69.64 -61.06, -23.26 in-in in 8.6685 Saltbr-in 2.7938 HRD-in -90.95, -53.69 70.13, 22.37 in-in-in SNCiii in-in ActLoopNT-in 2.8938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.31, 157.71 APE9-dihe-na 120.85, -158.74 APE8-dihe-in -109.76, 129.18 APE8-rot-in 307.33 APE67-dihe-in -52.63, -34.99 -47.86, -48.55 APE12-dist-in 8.4091 APE11-dist-in 11.5401 APE10-dist-in 5.9179 APE9-dist-in 3.8815 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.51 0.193 0.243 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fe5 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8FE5B P17612 4 351 351.0 XTT:60501 Type1 Active DFGin 6.5852 14.1601 BLAminus -125.03, 171.21 68.33, 95.08 -111.16, 25.84 279.92, 72.93 -61.92, -29.97 in-in in 8.6935 Saltbr-in 2.6551 HRD-in -80.97, -54.69 77.96, 3.27 in-in-in SNCiii in-in ActLoopNT-in 2.9235 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.98, 153.65 APE9-dihe-na 132.84, -165.24 APE8-dihe-in -101.75, 136.64 APE8-rot-in 293.15 APE67-dihe-in -60.99, -28.63 -57.01, -42.49 APE12-dist-in 8.3434 APE11-dist-in 11.6658 APE10-dist-in 6.0763 APE9-dist-in 3.8646 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.51 0.193 0.243 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fe5 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8FECA P17612 3 351 351.0 XU0:60501 Type1 Active DFGin 5.927 14.4607 BLAminus -126.38, -179.91 61.84, 90.42 -102.64, 31.23 279.77, 62.7 -61.22, -32.63 in-in in 9.1545 Saltbr-in 3.1068 HRD-in -85.43, -52.43 73.91, 14.55 in-in-in SNCiii in-in ActLoopNT-in 2.8343 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.02, 165.29 APE9-dihe-na 137.47, -140.99 APE8-dihe-in -132.86, 123.05 APE8-rot-in 312.11 APE67-dihe-in -60.14, -32.0 -40.12, -49.13 APE12-dist-in 8.2325 APE11-dist-in 11.5617 APE10-dist-in 5.9552 APE9-dist-in 3.6059 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.7 0.214 0.287 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fec Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8FECB P17612 3 351 351.0 XU0:60501 Type1 Active DFGin 5.9754 14.6835 BLAminus -127.65, 171.34 68.29, 92.72 -102.21, 27.6 281.7, 67.04 -60.34, -31.82 in-in in 8.8397 Saltbr-in 2.809 HRD-in -91.52, -53.88 75.61, 9.83 in-in-in SNCiii in-in ActLoopNT-in 2.9418 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.24, 178.4 APE9-dihe-na 115.87, -151.85 APE8-dihe-in -128.69, 124.59 APE8-rot-in 281.12 APE67-dihe-in -60.64, -38.43 -38.43, -52.12 APE12-dist-in 8.1803 APE11-dist-in 11.3776 APE10-dist-in 5.7925 APE9-dist-in 3.4601 None TPO198,SEP339 TPO198,SEP339 XRAY 2.7 0.214 0.287 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 8fec Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 2GU8A P17612 15 351 351.0 796:61001 Type1 Active DFGin 6.6297 14.3669 BLAminus -112.13, 169.56 64.55, 88.46 -98.67, 24.98 279.28, 59.9 -52.79, -25.6 in-in in 8.9692 Saltbr-in 3.0305 HRD-in -83.27, -51.67 71.2, 9.61 in-in-in SNCiii in-in ActLoopNT-in 2.9056 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.43, 156.76 APE9-dihe-na 146.07, -145.55 APE8-dihe-in -129.46, 134.31 APE8-rot-in 294.43 APE67-dihe-in -57.08, -22.75 -50.07, -49.98 APE12-dist-in 8.0405 APE11-dist-in 11.4687 APE10-dist-in 5.9773 APE9-dist-in 3.5072 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.203 0.261 A 337.0 337.0 0 25 25 0 [[44, 298]] 1.0 2gu8 Homo sapiens AGC_PRKACA_HUMAN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5N23A P17612 9 351 351.0 35R:60401 Type1 Active DFGin 5.4212 13.8637 BLAminus -109.83, 165.02 72.7, 94.27 -97.78, 24.01 286.85, 71.32 -58.73, -25.18 in-in in 9.4998 Saltbr-in 2.9266 HRD-in -90.99, -49.74 71.93, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.8779 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.89, 153.96 APE9-dihe-na 137.51, -163.29 APE8-dihe-in -116.51, 133.79 APE8-rot-in 303.7 APE67-dihe-in -56.98, -24.74 -46.64, -52.33 APE12-dist-in 8.0559 APE11-dist-in 11.5849 APE10-dist-in 5.9451 APE9-dist-in 3.6536 K48R,L96Q,M121L,V124A,Q182K,T184A SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.088 0.192 0.239 A 352.0 337.0 0 25 25 0 [[44, 298]] 1.0 5n23 Homo sapiens AGC_PRKACA_HUMAN AGC 5.3e-93 316.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3AMAA P17612 2 351 351.0 SKE:60351 Type1 Active DFGin 5.0968 14.0258 BLAminus -113.5, 162.11 72.12, 95.43 -101.12, 20.61 280.01, 66.12 -51.23, -34.47 in-in in 9.396 Saltbr-in 2.7343 HRD-in -88.12, -51.56 68.22, 12.75 in-in-in SNCiii in-in ActLoopNT-in 2.9104 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.04, 164.64 APE9-dihe-na 124.94, -160.1 APE8-dihe-in -123.9, 133.09 APE8-rot-in 298.24 APE67-dihe-in -57.85, -22.29 -46.67, -50.91 APE12-dist-in 8.1018 APE11-dist-in 11.5706 APE10-dist-in 5.9018 APE9-dist-in 3.5818 K48R,L96Q,M121L,V124A,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.75 0.198 0.223 A 351.0 345.0 0 25 25 0 [[44, 298]] 1.0 3ama Homo sapiens AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6FRXA P17612 13 351 351.0 E3Z:60401 Type1 Active DFGin 5.2761 14.2424 BLAminus -103.8, 165.76 62.73, 100.4 -98.82, 30.34 278.36, 58.69 -63.79, -25.19 in-in in 9.3071 Saltbr-in 2.6351 HRD-in -83.02, -52.27 73.43, 9.25 in-in-in SNCiii in-in ActLoopNT-in 2.866 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.05, 168.13 APE9-dihe-na 109.0, -164.56 APE8-dihe-in -112.4, 132.82 APE8-rot-in 302.54 APE67-dihe-in -55.48, -26.17 -48.65, -50.5 APE12-dist-in 8.3241 APE11-dist-in 11.7113 APE10-dist-in 6.1183 APE9-dist-in 3.716 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.88 0.191 0.226 A 351.0 334.0 0 25 25 0 [[44, 298]] 1.0 6frx Homo sapiens AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4AE6A P17612 13 351 351.0 No_ligand No_ligand Inactive DFGin 6.5333 15.789 ABAminus -102.0, -12.32 -149.9, 117.63 -105.31, 23.09 271.72, 75.39 -56.8, -39.15 out-in out 10.0651 Saltbr-in 3.037 HRD-in -80.45, -57.48 71.85, 11.08 in-in-out SNCiio in-out ActLoopNT-in 2.8103 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.83, 165.09 APE9-dihe-na 109.71, 150.17 APE8-dihe-in -70.25, 136.52 APE8-rot-out 76.9 APE67-dihe-in -62.21, -26.49 -48.12, -39.36 APE12-dist-in 8.4839 APE11-dist-in 11.6198 APE10-dist-in 6.1388 APE9-dist-in 4.2493 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.219 0.283 A 343.0 321.0 0 25 25 0 [[44, 298]] 1.0 4ae6 Homo sapiens AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4AE6B P17612 17 351 351.0 No_ligand No_ligand Inactive DFGin 6.7262 16.2285 ABAminus -110.11, -21.15 -129.5, 123.25 -122.94, 15.22 289.43, 78.48 -49.18, -40.14 out-out out 10.4783 Saltbr-out 4.4043 HRD-in -72.54, -54.34 51.9, 34.46 out-in-out SNCoio in-out ActLoopNT-in 2.6982 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -140.57, 163.72 APE9-dihe-na 111.27, 158.24 APE8-dihe-in -83.25, 146.52 APE8-rot-out 46.71 APE67-dihe-in -47.41, -26.35 -55.51, -46.4 APE12-dist-in 8.738 APE11-dist-in 11.4408 APE10-dist-in 5.9066 APE9-dist-in 4.36 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.219 0.283 B 343.0 323.0 0 25 25 0 [[44, 298]] 1.0 4ae6 Homo sapiens AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4AE9A P17612 13 351 351.0 No_ligand No_ligand Inactive DFGin 6.55 16.001 ABAminus -108.08, 1.25 -143.04, 135.02 -120.31, 26.17 277.62, 67.12 -50.31, -36.29 out-out out 10.2017 Saltbr-out 4.9285 HRD-in -78.87, -60.3 78.37, 10.3 out-in-in SNCoii in-in ActLoopNT-in 2.7466 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.01, 163.39 APE9-dihe-na 112.23, 171.54 APE8-dihe-in -84.52, 127.75 APE8-rot-in 289.6 APE67-dihe-in -56.88, -27.79 -43.6, -44.81 APE12-dist-in 8.2704 APE11-dist-in 11.576 APE10-dist-in 6.0269 APE9-dist-in 4.1577 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.201 0.264 A 343.0 324.0 0 25 25 0 [[44, 298]] 1.0 4ae9 Homo sapiens AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 4AE9B P17612 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.7487 16.1613 ABAminus -114.92, -7.43 -130.92, 125.97 -130.48, 16.95 295.44, 81.38 -52.61, -39.79 out-out out 10.6681 Saltbr-out 4.4397 HRD-in -74.27, -49.34 44.92, 35.44 out-in-out SNCoio in-out ActLoopNT-in 2.6317 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -139.93, 157.79 APE9-dihe-na 109.15, 156.62 APE8-dihe-in -68.62, 140.66 APE8-rot-out 10.98 APE67-dihe-in -51.62, -27.57 -42.37, -51.96 APE12-dist-in 8.5473 APE11-dist-in 11.4951 APE10-dist-in 5.9265 APE9-dist-in 4.357 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.201 0.264 B 343.0 324.0 0 25 25 0 [[44, 298]] 1.0 4ae9 Homo sapiens AGC_PRKACA_HUMAN AGC 4.2e-95 323.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 7Y1GB P17612 15 351 351.0 I5G:60401 Type1 Inactive DFGin 6.5019 15.3725 ABAminus -112.68, -38.34 -99.79, 125.89 -136.28, 17.99 282.52, 84.22 -66.37, -34.78 in-in in 9.4501 Saltbr-in 2.8689 HRD-in -80.77, -61.43 56.8, 33.17 in-in-out SNCiio in-out ActLoopNT-in 2.95 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.12, 157.52 APE9-dihe-na 119.76, 163.27 APE8-dihe-in -78.91, 145.18 APE8-rot-out 49.01 APE67-dihe-in -67.8, -20.12 -41.99, -42.68 APE12-dist-in 8.186 APE11-dist-in 11.3096 APE10-dist-in 5.7517 APE9-dist-in 4.3013 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.188 0.237 B 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 7y1g Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 9DC6A P17612 16 351 351.0 A1A3I:60501 Type1 Inactive DFGin 5.8215 14.3818 ABAminus -129.15, -5.99 -129.24, 116.18 -111.87, 19.13 279.15, 62.12 -54.37, -20.22 in-in in 9.1087 Saltbr-in 3.3088 HRD-in -90.78, -41.18 70.14, 8.35 in-in-in SNCiii in-in ActLoopNT-in 2.8945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.59, -177.06 APE9-dihe-na 91.67, -156.82 APE8-dihe-in -118.5, 121.2 APE8-rot-in 293.95 APE67-dihe-in -55.19, -30.52 -37.8, -52.71 APE12-dist-in 8.2373 APE11-dist-in 11.5075 APE10-dist-in 6.1047 APE9-dist-in 3.6545 None SEP140,TPO198 SEP140,TPO198 XRAY 2.7 0.237 0.311 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 9dc6 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 9DC6B P17612 16 351 351.0 A1A3I:60501 Type1 Inactive DFGin 6.1262 14.2237 ABAminus -118.96, -25.57 -111.81, 119.46 -118.82, 27.48 291.58, 78.19 -62.06, -32.01 in-in in 8.9675 Saltbr-in 2.88 HRD-in -75.88, -55.9 87.72, 2.66 in-in-in SNCiii in-in ActLoopNT-in 2.8974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.71, 171.27 APE9-dihe-na 114.33, -156.38 APE8-dihe-in -127.33, 134.71 APE8-rot-in 292.26 APE67-dihe-in -63.06, -23.33 -44.45, -51.67 APE12-dist-in 8.5329 APE11-dist-in 11.6121 APE10-dist-in 6.0734 APE9-dist-in 3.5437 None SEP140,TPO198 SEP140,TPO198 XRAY 2.7 0.237 0.311 B 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 9dc6 Homo sapiens AGC_PRKACA_HUMAN AGC 7e-95 323.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3AMBA P17612 4 351 351.0 VX6:60351 Type1 Inactive DFGin 5.087 14.2922 ABAminus -95.17, -47.0 -99.94, 115.14 -101.01, 17.86 279.8, 67.75 -53.93, -36.65 in-in in 9.4162 Saltbr-in 2.7867 HRD-in -85.39, -50.26 66.81, 7.13 in-in-in SNCiii in-in ActLoopNT-in 2.8909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.26, 159.46 APE9-dihe-na 131.88, -164.87 APE8-dihe-in -118.92, 127.93 APE8-rot-in 300.49 APE67-dihe-in -60.18, -24.15 -37.91, -53.92 APE12-dist-in 8.1946 APE11-dist-in 11.5803 APE10-dist-in 6.013 APE9-dist-in 3.6414 K48R,L96Q,M121L,V124A,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.25 0.214 0.256 A 351.0 343.0 0 25 25 0 [[44, 298]] 1.0 3amb Homo sapiens AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8X5LA P17612 17 351 351.0 RKD:401 Type1 Inactive DFGin 4.1037 12.291 ABAminus -92.81, -18.04 -108.82, 165.79 -131.86, 13.05 303.97, 96.56 69.26, -154.62 in-out in 9.9587 Saltbr-out 4.1566 HRD-in -67.69, -44.07 75.82, -80.8 out-out-out SNCooo out-out ActLoopNT-out 7.1481 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iooo APE10-dihe-na -77.04, -32.9 APE9-dihe-na -87.77, -44.9 APE8-dihe-in -124.02, 60.68 APE8-rot-out 58.39 APE67-dihe-in -63.73, -18.25 -72.69, -25.11 APE12-dist-in 12.2601 APE11-dist-out 15.7603 APE10-dist-out 19.6162 APE9-dist-out 13.5896 None SEP339 SEP339 XRAY 2.75 0.204 0.255 A 352.0 331.0 4 25 21 4 [[44, 298]] 1.0 8x5l Homo sapiens AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 8X5LB P17612 17 334 351.0 RKD:401 Type1 Inactive DFGin 4.0878 12.4831 ABAminus -93.45, -16.52 -108.91, 166.44 -130.77, 10.4 300.78, 83.16 68.88, -158.2 out-out out 10.6724 Saltbr-out 4.4614 HRD-in -67.44, -44.97 74.27, -77.51 out-out-out SNCooo out-out ActLoopNT-out 7.1674 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iioo APE10-dihe-na -62.33, 89.14 APE9-dihe-na -96.13, -167.24 APE8-dihe-in -45.35, 129.26 APE8-rot-out 58.75 APE67-dihe-in -60.15, -17.0 -69.42, -27.93 APE12-dist-in 9.2928 APE11-dist-in 11.2327 APE10-dist-out 15.0507 APE9-dist-out 8.3319 None SEP339 SEP339 XRAY 2.75 0.204 0.255 B 352.0 306.0 5 25 20 5 [[44, 298]] 1.0 8x5l Homo sapiens AGC_PRKACA_HUMAN AGC 7.9e-93 316.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6NO7E P17612 13 351 351.0 ATP:60403 ATPlike Inactive DFGin 6.9335 14.1655 BLAminus -118.71, 175.9 64.55, 75.01 -86.85, 19.7 273.68, 51.02 -43.49, -41.12 in-out in 9.4189 Saltbr-out 5.4559 HRD-in -91.66, -53.62 73.72, 11.47 out-in-in SNCoii in-in ActLoopNT-in 3.1639 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.9, 150.23 APE9-dihe-na 149.21, -142.3 APE8-dihe-in -132.1, 131.95 APE8-rot-in 297.19 APE67-dihe-in -64.62, -25.64 -37.25, -53.79 APE12-dist-in 8.0557 APE11-dist-in 10.9843 APE10-dist-in 5.7482 APE9-dist-in 3.2156 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 E 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 6no7 Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6NO7G P17612 15 351 351.0 ATP:60403 ATPlike Inactive DFGin 6.0359 14.0844 BLAminus -118.68, 176.55 65.34, 76.32 -85.78, 18.75 273.72, 51.07 -44.34, -41.82 in-out in 9.7125 Saltbr-out 5.2149 HRD-in -91.95, -53.38 74.11, 11.57 out-in-in SNCoii in-in ActLoopNT-in 3.3017 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.42, 149.81 APE9-dihe-na 148.91, -142.4 APE8-dihe-in -132.18, 131.68 APE8-rot-in 297.12 APE67-dihe-in -64.98, -25.0 -37.42, -54.32 APE12-dist-in 7.6679 APE11-dist-in 10.658 APE10-dist-in 5.5534 APE9-dist-in 3.4096 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 G 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 6no7 Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 9EDDA P17612 14 351 351.0 ATP:60400 ATPlike Inactive DFGin 7.6417 15.4797 BLAminus -131.38, -176.44 56.47, 73.0 -86.17, 32.62 269.53, 53.11 -62.17, -29.29 in-out in 9.6174 Saltbr-out 3.9466 HRD-in -100.83, -51.39 64.03, -2.2 out-out-out SNCooo out-out ActLoopNT-out 3.7028 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -126.87, 141.16 APE9-dihe-na 150.41, -172.01 APE8-dihe-in -103.27, 147.74 APE8-rot-out 185.24 APE67-dihe-in -92.0, 3.92 -57.96, -27.57 APE12-dist-in 8.1647 APE11-dist-in 11.2754 APE10-dist-in 5.6275 APE9-dist-in 4.2273 None TPO198,SEP339 TPO198,SEP339 EM 6.3 999.0 999.0 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9edd Homo sapiens AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 9EDEA P17612 14 351 351.0 ATP:60400 ATPlike Inactive DFGin 6.6922 15.188 BLAminus -131.57, -176.8 59.06, 65.59 -87.14, 28.49 267.05, 50.71 -66.29, -36.64 in-out in 9.9219 Saltbr-out 4.6819 HRD-in -115.21, -49.18 64.38, 4.15 out-out-out SNCooo out-out ActLoopNT-out 3.632 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.67, 141.1 APE9-dihe-na 158.89, -177.66 APE8-dihe-in -75.58, 154.98 APE8-rot-out 190.35 APE67-dihe-in -109.16, -25.21 -65.33, -8.36 APE12-dist-in 8.3471 APE11-dist-in 11.7825 APE10-dist-in 6.8289 APE9-dist-in 4.9175 None TPO198,SEP339 TPO198,SEP339 EM 5.9 999.0 999.0 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 9ede Homo sapiens AGC_PRKACA_HUMAN AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5IZJA P17612 15 351 351.0 6J9:60414 Allosteric Inactive DFGin 6.0059 14.882 BLAminus -111.62, 172.78 70.98, 87.77 -97.8, 27.11 278.83, 80.41 -58.58, -30.48 in-out in 9.9394 Saltbr-out 4.1818 HRD-in -81.12, -50.89 44.27, 35.23 out-in-out SNCoio in-out ActLoopNT-in 2.9865 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -140.79, 157.34 APE9-dihe-na 106.02, 164.59 APE8-dihe-in -74.04, 136.38 APE8-rot-out 204.5 APE67-dihe-in -57.37, -26.41 -46.69, -44.98 APE12-dist-in 8.2021 APE11-dist-in 11.523 APE10-dist-in 5.7985 APE9-dist-in 4.2246 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.199 0.226 A 351.0 330.0 0 25 25 0 [[44, 298]] 1.0 5izj Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 5IZJB P17612 15 351 351.0 6J9:60413 Allosteric Inactive DFGin 6.2012 15.2736 BLAminus -109.02, 168.97 75.33, 87.97 -97.67, 24.22 269.13, 57.46 -63.02, -24.98 out-out out 10.2894 Saltbr-out 4.5426 HRD-in -78.48, -51.65 67.16, 12.35 out-in-out SNCoio in-out ActLoopNT-in 2.9093 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.15, 157.15 APE9-dihe-na 105.13, 166.26 APE8-dihe-in -75.85, 137.43 APE8-rot-out 200.52 APE67-dihe-in -61.79, -25.86 -47.32, -41.18 APE12-dist-in 8.2568 APE11-dist-in 11.4828 APE10-dist-in 5.8129 APE9-dist-in 4.0688 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.199 0.226 B 351.0 327.0 0 25 25 0 [[44, 298]] 1.0 5izj Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6BYSA P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.6445 12.8448 BLAminus 176.97, -168.6 35.04, 63.97 -77.13, -0.55 257.78, 43.58 -51.31, -30.32 in-out in 8.4132 Saltbr-out 3.6943 HRD-out -132.08, 139.02 -123.89, -19.92 out-in-in SNCoii in-in ActLoopNT-in 3.1045 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -174.55, -174.54 APE9-dihe-na 119.07, -153.65 APE8-dihe-in -123.63, 121.24 APE8-rot-in 279.88 APE67-dihe-in -80.36, -3.37 -55.82, -41.73 APE12-dist-in 8.6369 APE11-dist-in 11.0634 APE10-dist-in 6.1456 APE9-dist-in 3.4911 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6BYSC P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.5999 13.0168 BLAminus 177.41, -169.47 35.75, 66.26 -79.08, -7.92 257.89, 46.49 -37.01, -39.99 in-out in 8.4312 Saltbr-out 3.6308 HRD-out -132.47, 138.88 -123.68, -21.42 out-in-in SNCoii in-in ActLoopNT-in 3.129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.21, -176.06 APE9-dihe-na 122.36, -150.78 APE8-dihe-in -124.74, 121.46 APE8-rot-in 280.04 APE67-dihe-in -74.72, -2.75 -56.12, -45.35 APE12-dist-in 8.6212 APE11-dist-in 11.0301 APE10-dist-in 6.1698 APE9-dist-in 3.5547 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 C 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6BYSE P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.5995 12.7783 BLAminus 177.63, -170.33 35.66, 68.12 -82.89, -7.7 254.73, 43.9 -34.72, -39.61 in-in in 8.3947 Saltbr-in 3.5304 HRD-out -134.25, 137.62 -124.05, -19.61 in-in-in SNCiii in-in ActLoopNT-in 3.1341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -175.91, -174.99 APE9-dihe-na 120.1, -152.87 APE8-dihe-in -123.78, 120.18 APE8-rot-in 279.49 APE67-dihe-in -74.6, -2.18 -55.44, -46.05 APE12-dist-in 8.5261 APE11-dist-in 11.0087 APE10-dist-in 6.1584 APE9-dist-in 3.4923 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 E 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6BYSG P17612 14 351 351.0 No_ligand No_ligand Inactive DFGin 5.5502 12.8795 BLAminus 177.64, -169.59 35.17, 69.18 -84.06, -7.89 253.42, 50.51 -34.53, -40.01 in-out in 8.4064 Saltbr-out 3.6038 HRD-out -131.78, 137.89 -122.99, -20.45 out-in-in SNCoii in-in ActLoopNT-in 3.091 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -174.78, -177.53 APE9-dihe-na 124.08, -149.25 APE8-dihe-in -124.03, 121.23 APE8-rot-in 280.42 APE67-dihe-in -73.41, -1.98 -56.98, -46.28 APE12-dist-in 8.6175 APE11-dist-in 11.0767 APE10-dist-in 6.1508 APE9-dist-in 3.5427 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 4.75 0.216 0.255 G 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 6bys Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6NO7A P17612 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.5833 14.5513 BLAminus -119.16, 176.65 65.47, 76.79 -85.63, 19.52 273.14, 48.34 -44.12, -41.29 in-out in 9.256 Saltbr-out 3.8369 HRD-in -93.59, -54.13 73.95, 11.29 out-in-in SNCoii in-in ActLoopNT-in 3.0846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.66, 149.89 APE9-dihe-na 148.72, -142.64 APE8-dihe-in -132.35, 131.6 APE8-rot-in 297.3 APE67-dihe-in -65.08, -25.39 -37.56, -54.33 APE12-dist-in 7.8572 APE11-dist-in 10.7351 APE10-dist-in 5.368 APE9-dist-in 3.3109 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.55 0.259 0.269 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 6no7 Homo sapiens AGC_PRKACA_HUMAN AGC 4.5e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 3MVJB P17612 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.6749 15.0725 BLAminus -107.29, 175.17 69.85, 103.13 -126.62, 31.7 289.12, 86.96 -68.94, -36.62 in-out in 9.8619 Saltbr-out 5.1808 HRD-in -72.7, -45.04 65.83, 8.62 out-in-in SNCoii in-in ActLoopNT-in 2.6815 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.22, 164.94 APE9-dihe-na 113.67, -166.87 APE8-dihe-in -95.86, 130.98 APE8-rot-in 290.81 APE67-dihe-in -63.62, -17.9 -44.08, -47.61 APE12-dist-in 8.4504 APE11-dist-in 11.5319 APE10-dist-in 6.2728 APE9-dist-in 4.219 None TPO198,SEP339 TPO198,SEP339 XRAY 2.49 0.217 0.304 B 371.0 322.0 0 25 25 0 [[44, 298]] 1.0 3mvj Homo sapiens AGC_PRKACA_HUMAN AGC 5.4e-95 323.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6WJFA P17612 2 351 351.0 No_ligand No_ligand Inactive DFGin 9.9992 13.4832 BLAminus -126.44, 169.73 60.01, 89.86 -112.86, 1.12 296.86, 95.65 -61.53, -29.79 out-out out 10.0908 Saltbr-out 7.2346 HRD-in -67.55, -42.01 64.88, -66.83 out-out-out SNCooo out-out ActLoopNT-out 3.6866 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -171.91, 116.67 APE9-dihe-na 154.02, -66.34 APE8-dihe-in -113.18, 77.77 APE8-rot-out 47.03 APE67-dihe-in -82.77, -55.57 -68.63, -38.53 APE12-dist-in 8.4814 APE11-dist-in 12.0403 APE10-dist-in 7.8146 APE9-dist-in 4.4462 None None None EM 7.5 999.0 999.0 A 405.0 336.0 0 25 25 0 [[44, 298]] 1.0 6wjf Homo sapiens AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6WJFB P17612 42 351 351.0 No_ligand No_ligand Inactive DFGin 10.0534 15.2293 BLAminus -124.34, 176.36 59.38, 90.58 -123.09, 12.38 277.22, 94.34 -61.71, -29.6 out-out out 11.687 Saltbr-out 6.4309 HRD-out -65.49, -35.93 66.74, -107.09 out-out-out SNCooo out-out ActLoopNT-out 3.9609 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiio APE10-dihe-na -163.85, -158.9 APE9-dihe-na 100.21, -130.3 APE8-dihe-in -150.47, 147.99 APE8-rot-out 180.18 APE67-dihe-in -80.92, 5.22 -58.41, -26.93 APE12-dist-in 8.6814 APE11-dist-in 11.7662 APE10-dist-in 6.7949 APE9-dist-out 6.2996 None None None EM 7.5 999.0 999.0 B 405.0 310.0 27 25 25 0 [[44, 298]] 1.0 6wjf Homo sapiens AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6WJGA P17612 42 351 351.0 No_ligand No_ligand Inactive DFGin 9.9992 13.4832 BLAminus -126.44, 169.73 60.01, 89.86 -112.86, 1.12 296.86, 95.65 -61.53, -29.79 out-out out 10.0908 Saltbr-out 7.2346 HRD-in -67.55, -42.01 64.88, -66.83 out-out-out SNCooo out-out ActLoopNT-out 3.6866 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -171.91, 116.67 APE9-dihe-na 154.02, -66.34 APE8-dihe-in -113.18, 77.77 APE8-rot-out 47.03 APE67-dihe-in -82.77, -55.57 -68.63, -38.53 APE12-dist-in 8.4814 APE11-dist-in 12.0403 APE10-dist-in 7.8146 APE9-dist-in 4.4462 None None None EM 6.2 999.0 999.0 A 405.0 310.0 27 25 25 0 [[44, 298]] 1.0 6wjg Homo sapiens AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6WJGB P17612 42 351 351.0 No_ligand No_ligand Inactive DFGin 10.0534 15.2293 BLAminus -124.34, 176.36 59.38, 90.58 -123.09, 12.38 277.22, 94.34 -61.71, -29.6 out-out out 11.687 Saltbr-out 6.4309 HRD-out -65.49, -35.93 66.74, -107.09 out-out-out SNCooo out-out ActLoopNT-out 3.9609 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiio APE10-dihe-na -163.85, -158.9 APE9-dihe-na 100.21, -130.3 APE8-dihe-in -150.47, 147.99 APE8-rot-out 180.18 APE67-dihe-in -80.92, 5.22 -58.41, -26.93 APE12-dist-in 8.6814 APE11-dist-in 11.7662 APE10-dist-in 6.7949 APE9-dist-out 6.2996 None None None EM 6.2 999.0 999.0 B 405.0 310.0 27 25 25 0 [[44, 298]] 1.0 6wjg Homo sapiens AGC_PRKACA_HUMAN AGC 3.3e-94 320.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 7Y1GA P17612 16 351 351.0 I5G:60500 Type1 Inactive DFGin 6.3413 14.8624 BLAminus -118.48, 174.7 76.77, 103.0 -130.63, 13.32 288.1, 82.33 -55.62, -41.63 in-in in 9.1119 Saltbr-in 2.716 HRD-in -77.78, -56.16 48.65, 33.18 in-in-out SNCiio in-out ActLoopNT-in 2.8984 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -128.96, 160.38 APE9-dihe-na 112.98, 149.31 APE8-dihe-in -54.34, 136.89 APE8-rot-out 199.98 APE67-dihe-in -67.35, -18.71 -49.9, -39.67 APE12-dist-in 8.1184 APE11-dist-in 11.271 APE10-dist-in 5.6336 APE9-dist-in 4.254 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.188 0.237 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 7y1g Homo sapiens AGC_PRKACA_HUMAN AGC 4.6e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_HUMAN 6C0UA P17612 12 351 351.0 EE4:60400 Type1 Inactive DFGin 6.4885 14.2621 BLAminus -130.77, 175.54 62.84, 100.35 -119.36, 26.56 282.24, 71.26 -65.52, -23.67 in-in in 8.3667 Saltbr-in 3.028 HRD-in -79.47, -53.84 70.3, 8.89 in-in-out SNCiio in-out ActLoopNT-in 3.0007 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.41, 153.98 APE9-dihe-na 116.73, 155.27 APE8-dihe-in -73.99, 144.03 APE8-rot-out 173.49 APE67-dihe-in -64.51, -15.31 -53.81, -42.18 APE12-dist-in 7.614 APE11-dist-in 10.848 APE10-dist-in 5.4829 APE9-dist-in 3.9348 None TPO198,SEP339 TPO198,SEP339 XRAY 2.65 0.211 0.243 A 354.0 340.0 0 25 25 0 [[44, 298]] 1.0 6c0u Homo sapiens AGC_PRKACA_HUMAN AGC 4.7e-95 323.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4O21A P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 6.0367 14.4393 BLAminus -125.27, 173.53 70.53, 83.75 -96.26, 25.58 272.04, 54.28 -57.91, -27.19 in-in in 8.9531 Saltbr-in 2.7155 HRD-in -83.95, -57.84 75.15, 8.54 in-in-in SNCiii in-in ActLoopNT-in 2.9043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.15, 164.3 APE9-dihe-na 125.14, -151.92 APE8-dihe-in -125.51, 129.66 APE8-rot-in 308.07 APE67-dihe-in -63.53, -19.17 -43.91, -48.76 APE12-dist-in 8.0396 APE11-dist-in 11.4602 APE10-dist-in 5.9112 APE9-dist-in 3.4511 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.17 0.215 A 342.0 336.0 0 25 25 0 [[44, 298]] 1.0 4o21 Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7E11A P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 6.205 14.4514 BLAminus -127.38, -169.19 58.28, 74.22 -96.53, 30.74 276.22, 81.09 -66.46, -21.72 in-in in 9.0533 Saltbr-in 2.5511 HRD-in -91.79, -53.23 62.57, 24.02 in-in-in SNCiii in-in ActLoopNT-in 3.1289 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.39, 155.98 APE9-dihe-na 134.96, -158.62 APE8-dihe-in -113.95, 132.34 APE8-rot-in 301.67 APE67-dihe-in -76.79, -1.28 -53.37, -39.68 APE12-dist-in 8.3091 APE11-dist-in 11.1349 APE10-dist-in 5.7098 APE9-dist-in 3.659 None TPO198,SEP339 TPO198,SEP339 XRAY 3.43 0.262 0.317 A 338.0 337.0 0 25 25 0 [[44, 298]] 1.0 7e11 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3PVBA P05132 7 351 351.0 ANP:60400 ATPlike Active DFGin 5.2614 14.1066 BLAminus -138.85, 171.16 63.11, 82.89 -89.43, -59.95 273.17, 54.43 27.14, -66.26 in-in in 8.6853 Saltbr-in 3.4757 HRD-in -84.36, -35.8 62.24, -18.82 in-in-in SNCiii in-in ActLoopNT-in 3.2175 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -177.84, 157.88 APE9-dihe-na 132.55, -154.74 APE8-dihe-in -122.19, 108.01 APE8-rot-in 318.81 APE67-dihe-in -60.75, -2.24 -13.41, -60.33 APE12-dist-in 7.7331 APE11-dist-in 10.5794 APE10-dist-in 5.5109 APE9-dist-in 4.0421 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 3.3 0.242 0.29 A 345.0 345.0 0 25 25 0 [[44, 298]] 1.0 3pvb Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1BKXA P05132 13 351 351.0 AMP:60351 ATPlike Active DFGin 6.1602 13.9145 BLAminus -117.09, 179.26 61.99, 75.16 -83.18, 21.65 286.96, 82.43 -60.51, -17.53 in-in in 8.7242 Saltbr-in 2.6583 HRD-in -99.39, -38.31 69.2, -9.22 in-in-in SNCiii in-in ActLoopNT-in 3.4681 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.44, 150.62 APE9-dihe-na 113.99, 166.84 APE8-dihe-in -65.88, 134.1 APE8-rot-in 334.22 APE67-dihe-in -70.66, -34.65 -48.92, -27.08 APE12-dist-in 8.2835 APE11-dist-in 11.3505 APE10-dist-in 5.7038 APE9-dist-in 4.2848 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.6 0.219 0.34 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1bkx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1L3RE P05132 2 351 351.0 ADP:60381 ATPlike Active DFGin 5.7538 14.4402 BLAminus -119.14, -174.46 57.18, 81.19 -93.77, 20.31 270.88, 52.04 -50.0, -37.57 in-in in 9.0231 Saltbr-in 2.7924 HRD-in -82.45, -54.36 70.16, 7.26 in-in-in SNCiii in-in ActLoopNT-in 2.9201 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.84, 161.06 APE9-dihe-na 132.7, -149.01 APE8-dihe-in -131.06, 132.91 APE8-rot-in 298.56 APE67-dihe-in -55.27, -27.25 -33.24, -62.94 APE12-dist-in 8.1978 APE11-dist-in 11.2333 APE10-dist-in 5.8253 APE9-dist-in 3.3679 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.0 0.205 0.232 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1l3r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2QCSA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.648 14.2907 BLAminus -119.78, 176.88 65.56, 77.31 -85.05, 19.39 273.35, 51.28 -44.32, -42.51 in-in in 8.7843 Saltbr-in 2.6377 HRD-in -93.14, -54.78 73.52, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.7354 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.52, 149.74 APE9-dihe-na 148.64, -142.53 APE8-dihe-in -132.36, 132.12 APE8-rot-in 297.18 APE67-dihe-in -64.67, -25.45 -36.74, -53.73 APE12-dist-in 8.133 APE11-dist-in 11.3207 APE10-dist-in 5.8515 APE9-dist-in 3.5726 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.194 0.225 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 2qcs Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3FJQE P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.6709 14.4589 BLAminus -119.42, 178.78 63.28, 80.04 -91.81, 23.31 270.73, 57.82 -56.09, -30.86 in-in in 9.1494 Saltbr-in 2.8344 HRD-in -91.33, -52.39 67.42, 13.87 in-in-in SNCiii in-in ActLoopNT-in 2.9056 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.19, 160.44 APE9-dihe-na 133.42, -155.21 APE8-dihe-in -125.75, 136.86 APE8-rot-in 304.0 APE67-dihe-in -61.0, -22.29 -48.87, -49.39 APE12-dist-in 8.0863 APE11-dist-in 11.4084 APE10-dist-in 5.8377 APE9-dist-in 3.5179 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.179 0.205 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 3fjq Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3IDBA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.3459 14.4126 BLAminus -121.17, -175.1 59.7, 79.28 -94.34, 24.01 267.69, 48.22 -48.56, -33.02 in-in in 8.8455 Saltbr-in 2.694 HRD-in -80.07, -50.75 69.18, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.9896 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.99, 160.5 APE9-dihe-na 138.4, -150.07 APE8-dihe-in -124.64, 132.33 APE8-rot-in 296.41 APE67-dihe-in -59.26, -21.93 -30.94, -63.4 APE12-dist-in 8.1019 APE11-dist-in 11.5726 APE10-dist-in 6.0684 APE9-dist-in 3.4448 None TPO198,SEP339 TPO198,SEP339 XRAY 1.62 0.206 0.23 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 3idb Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3IDCA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.079 14.4716 BLAminus -127.31, 174.57 68.22, 96.34 -111.15, 30.11 265.57, 49.45 -62.75, -22.0 in-in in 8.6423 Saltbr-in 3.0306 HRD-in -69.04, -44.03 64.09, 13.38 in-in-in SNCiii in-in ActLoopNT-in 2.8561 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.35, 157.69 APE9-dihe-na 142.7, -132.16 APE8-dihe-in -139.58, 115.88 APE8-rot-in 293.03 APE67-dihe-in -54.66, -5.54 -16.73, -78.3 APE12-dist-in 7.8437 APE11-dist-in 11.3725 APE10-dist-in 6.1644 APE9-dist-in 3.6752 None TPO198,SEP339 TPO198,SEP339 XRAY 2.7 0.241 0.319 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 3idc Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DG0E P05132 11 351 351.0 ANP:60402 ATPlike Active DFGin 5.5834 14.3418 BLAminus -118.87, 179.66 65.44, 79.89 -93.34, 25.25 272.35, 58.42 -52.71, -36.39 in-in in 8.955 Saltbr-in 2.6989 HRD-in -84.35, -52.45 74.02, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.8946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.07, 161.1 APE9-dihe-na 130.81, -146.6 APE8-dihe-in -130.07, 130.32 APE8-rot-in 303.85 APE67-dihe-in -61.09, -22.5 -44.14, -49.24 APE12-dist-in 8.0079 APE11-dist-in 11.4975 APE10-dist-in 5.8998 APE9-dist-in 3.3886 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.196 0.228 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 4dg0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH1A P05132 16 351 351.0 ATP:60402 ATPlike Active DFGin 6.2341 14.3802 BLAminus -130.7, 167.11 69.97, 89.08 -103.01, 26.92 273.93, 57.95 -52.62, -33.38 in-in in 8.9305 Saltbr-in 3.0104 HRD-in -75.69, -51.31 65.95, 10.85 in-in-in SNCiii in-in ActLoopNT-in 2.8868 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.97, 163.54 APE9-dihe-na 128.87, -151.55 APE8-dihe-in -123.52, 135.53 APE8-rot-in 304.09 APE67-dihe-in -55.69, -26.94 -40.23, -59.36 APE12-dist-in 8.1686 APE11-dist-in 11.5574 APE10-dist-in 5.9503 APE9-dist-in 3.5446 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.199 0.234 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH3A P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.9838 14.3792 BLAminus -125.47, 176.75 61.82, 79.89 -92.16, 24.39 276.69, 54.39 -43.39, -47.09 in-in in 9.021 Saltbr-in 2.7225 HRD-in -82.56, -48.22 66.04, -2.33 in-in-in SNCiii in-in ActLoopNT-in 2.9311 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 165.55 APE9-dihe-na 126.96, -149.27 APE8-dihe-in -125.58, 130.88 APE8-rot-in 307.35 APE67-dihe-in -57.88, -25.54 -37.95, -56.15 APE12-dist-in 8.2249 APE11-dist-in 11.5925 APE10-dist-in 6.1036 APE9-dist-in 3.74 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.203 0.233 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH5A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 6.1214 14.3392 BLAminus -125.12, -179.76 61.4, 85.13 -97.61, 27.77 279.05, 62.21 -46.99, -44.52 in-in in 9.0432 Saltbr-in 2.5524 HRD-in -77.92, -53.51 67.68, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.9684 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.88, 153.17 APE9-dihe-na 132.88, -161.89 APE8-dihe-in -112.07, 131.8 APE8-rot-in 304.21 APE67-dihe-in -57.01, -23.17 -41.47, -55.69 APE12-dist-in 8.2186 APE11-dist-in 11.6017 APE10-dist-in 6.0711 APE9-dist-in 3.87 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.187 0.222 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH7A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.5738 14.3492 BLAminus -124.43, -175.45 59.33, 78.79 -93.54, 24.71 270.97, 54.79 -50.12, -38.03 in-in in 9.0247 Saltbr-in 2.7242 HRD-in -76.49, -50.79 66.5, 11.01 in-in-in SNCiii in-in ActLoopNT-in 2.9607 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.18, 162.39 APE9-dihe-na 131.3, -151.54 APE8-dihe-in -126.44, 134.15 APE8-rot-in 300.19 APE67-dihe-in -56.38, -25.77 -37.48, -60.34 APE12-dist-in 8.0928 APE11-dist-in 11.4546 APE10-dist-in 5.87 APE9-dist-in 3.4166 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.8 0.179 0.194 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH8A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.9006 14.014 BLAminus -123.95, -176.77 59.01, 85.18 -98.8, 24.84 279.52, 63.26 -51.76, -30.5 in-in in 8.8003 Saltbr-in 2.7128 HRD-in -77.99, -56.65 70.43, 3.78 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.95, 158.57 APE9-dihe-na 135.16, -154.79 APE8-dihe-in -124.8, 132.89 APE8-rot-in 296.53 APE67-dihe-in -58.95, -25.2 -38.46, -56.52 APE12-dist-in 8.1451 APE11-dist-in 11.4751 APE10-dist-in 5.904 APE9-dist-in 3.5115 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.155 0.188 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh8 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4HPTE P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.7482 14.4242 BLAminus -115.4, 178.03 67.73, 81.09 -92.11, 21.69 273.09, 55.37 -58.71, -29.4 in-in in 9.0532 Saltbr-in 2.6604 HRD-in -90.64, -54.09 71.81, 9.39 in-in-in SNCiii in-in ActLoopNT-in 2.8739 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.27, 162.98 APE9-dihe-na 129.56, -147.32 APE8-dihe-in -127.39, 129.92 APE8-rot-in 299.02 APE67-dihe-in -63.31, -27.9 -40.61, -49.36 APE12-dist-in 8.0686 APE11-dist-in 11.3854 APE10-dist-in 5.8255 APE9-dist-in 3.5734 None TPO198,SEP339 TPO198,SEP339 XRAY 2.15 0.189 0.228 E 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4hpt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4HPUE P05132 13 351 351.0 ANP:60402 ATPlike Active DFGin 5.5508 14.4067 BLAminus -117.63, -178.61 63.83, 78.8 -92.22, 24.46 271.46, 55.23 -53.69, -32.94 in-in in 9.0306 Saltbr-in 2.6916 HRD-in -87.73, -52.35 74.85, 8.01 in-in-in SNCiii in-in ActLoopNT-in 2.9145 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.41, 162.17 APE9-dihe-na 134.1, -149.11 APE8-dihe-in -128.69, 136.04 APE8-rot-in 297.56 APE67-dihe-in -58.67, -24.48 -48.3, -49.81 APE12-dist-in 8.0634 APE11-dist-in 11.5067 APE10-dist-in 5.8865 APE9-dist-in 3.4033 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.173 0.194 E 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 4hpu Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 5JR7A P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.7387 13.6907 BLAminus -145.14, 176.28 64.37, 76.68 -85.75, 18.89 294.14, 59.99 -43.66, -41.86 in-in in 8.6743 Saltbr-in 2.7095 HRD-in -93.38, -54.67 74.91, 7.39 in-in-in SNCiii in-in ActLoopNT-in 2.945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.46, 148.2 APE9-dihe-na 147.95, -159.28 APE8-dihe-in -109.66, 131.32 APE8-rot-in 258.88 APE67-dihe-in -65.5, -25.8 -38.64, -53.47 APE12-dist-in 8.0144 APE11-dist-in 10.772 APE10-dist-in 5.5284 APE9-dist-in 3.8782 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 5JR7C P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.8995 13.1635 BLAminus -138.79, 176.44 54.89, 86.07 -89.1, 7.67 290.95, 62.79 -41.83, -37.01 in-in in 8.1848 Saltbr-in 3.1954 HRD-in -79.11, -50.37 72.48, -21.93 in-in-in SNCiii in-in ActLoopNT-in 2.8194 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.28, 123.46 APE9-dihe-na 160.31, -160.86 APE8-dihe-in -110.49, 124.04 APE8-rot-in 311.35 APE67-dihe-in -70.47, -24.34 -45.9, -42.95 APE12-dist-in 8.1626 APE11-dist-in 10.628 APE10-dist-in 5.0018 APE9-dist-in 4.2619 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 C 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7UJXE P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 5.731 14.3568 BLAminus -121.93, 179.51 64.92, 83.56 -91.91, 29.5 277.22, 63.03 -64.62, -28.12 in-in in 9.1028 Saltbr-in 2.8121 HRD-in -86.19, -57.72 74.11, 16.74 in-in-in SNCiii in-in ActLoopNT-in 2.9312 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.48, 155.47 APE9-dihe-na 127.23, -161.98 APE8-dihe-in -111.77, 133.52 APE8-rot-in 302.04 APE67-dihe-in -65.07, -18.97 -50.87, -44.77 APE12-dist-in 8.1906 APE11-dist-in 11.5001 APE10-dist-in 5.9613 APE9-dist-in 4.0077 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.133 0.176 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 7ujx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7V0GE P05132 17 351 351.0 ADP:60401 ATPlike Active DFGin 5.7389 14.3189 BLAminus -119.5, 177.58 67.43, 82.74 -91.45, 25.21 276.8, 64.92 -62.46, -26.34 in-in in 9.0699 Saltbr-in 2.8017 HRD-in -88.93, -50.41 71.3, 15.33 in-in-in SNCiii in-in ActLoopNT-in 2.9568 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.52, 156.77 APE9-dihe-na 130.04, -162.37 APE8-dihe-in -114.97, 131.2 APE8-rot-in 299.52 APE67-dihe-in -60.0, -22.75 -47.18, -49.61 APE12-dist-in 8.1738 APE11-dist-in 11.5422 APE10-dist-in 6.0368 APE9-dist-in 3.9649 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.118 0.163 E 350.0 335.0 0 25 25 0 [[44, 298]] 1.0 7v0g Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFXE P05132 2 351 351.0 ANP:60402 ATPlike Active DFGin 5.5242 14.2861 BLAminus -116.71, -179.39 66.13, 78.01 -91.08, 23.34 272.63, 51.46 -56.59, -32.27 in-in in 8.8728 Saltbr-in 2.7287 HRD-in -88.99, -54.58 73.79, 11.03 in-in-in SNCiii in-in ActLoopNT-in 2.9336 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.69, 159.64 APE9-dihe-na 138.16, -148.52 APE8-dihe-in -130.4, 136.32 APE8-rot-in 296.63 APE67-dihe-in -59.91, -24.0 -47.38, -49.37 APE12-dist-in 8.0462 APE11-dist-in 11.4097 APE10-dist-in 5.8188 APE9-dist-in 3.3923 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.35 0.157 0.179 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4dfx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4X6RA P05132 2 351 351.0 ATP:60402 ATPlike Active DFGin 6.1334 14.2323 BLAminus -118.92, 178.27 64.18, 79.91 -89.21, 11.01 274.1, 55.74 -49.19, -34.95 in-in in 8.8037 Saltbr-in 2.7288 HRD-in -85.13, -60.38 77.67, -7.87 in-in-in SNCiii in-in ActLoopNT-in 2.7182 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.34, 156.01 APE9-dihe-na 147.33, -149.7 APE8-dihe-in -130.56, 138.51 APE8-rot-in 291.09 APE67-dihe-in -61.2, -24.8 -52.44, -47.95 APE12-dist-in 8.281 APE11-dist-in 11.2462 APE10-dist-in 5.8359 APE9-dist-in 3.6632 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.186 0.234 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4x6r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3X2UA P05132 13 351 351.0 ATP:60501 ATPlike Active DFGin 6.1271 14.5072 BLAminus -122.24, 178.58 59.36, 87.7 -101.54, 25.28 272.61, 50.83 -59.45, -24.26 in-in in 9.2723 Saltbr-in 2.7882 HRD-in -89.58, -50.62 64.84, 17.58 in-in-in SNCiii in-in ActLoopNT-in 2.9297 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.25, 158.3 APE9-dihe-na 134.88, -147.54 APE8-dihe-in -130.4, 131.58 APE8-rot-in 300.12 APE67-dihe-in -61.26, -14.4 -40.08, -55.22 APE12-dist-in 7.9122 APE11-dist-in 11.1375 APE10-dist-in 5.6863 APE9-dist-in 3.4266 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.202 0.239 A 357.0 339.0 0 25 25 0 [[44, 298]] 1.0 3x2u Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3X2VA P05132 18 351 351.0 ATP:60403 ATPlike Active DFGin 5.5167 14.1516 BLAminus -116.69, -175.94 62.92, 80.3 -91.77, 26.26 271.42, 55.44 -51.78, -39.79 in-in in 8.7552 Saltbr-in 2.6541 HRD-in -92.08, -50.84 67.69, 17.07 in-in-in SNCiii in-in ActLoopNT-in 2.8813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.85, 164.45 APE9-dihe-na 134.14, -152.5 APE8-dihe-in -130.83, 133.42 APE8-rot-in 299.77 APE67-dihe-in -58.82, -21.18 -48.96, -48.11 APE12-dist-in 7.9982 APE11-dist-in 11.3458 APE10-dist-in 5.7964 APE9-dist-in 3.4149 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.77 0.185 0.23 A 357.0 334.0 0 25 25 0 [[44, 298]] 1.0 3x2v Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3X2WA P05132 13 351 351.0 ATP:60403 ATPlike Active DFGin 5.6602 14.3902 BLAminus -121.01, -177.68 63.51, 77.56 -90.4, 24.79 270.4, 59.29 -61.83, -28.06 in-in in 8.8217 Saltbr-in 2.6324 HRD-in -81.34, -52.24 70.22, 11.48 in-in-in SNCiii in-in ActLoopNT-in 2.9059 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.19, 162.39 APE9-dihe-na 132.4, -151.44 APE8-dihe-in -129.91, 133.08 APE8-rot-in 300.2 APE67-dihe-in -60.45, -20.83 -45.18, -51.38 APE12-dist-in 8.001 APE11-dist-in 11.4403 APE10-dist-in 5.911 APE9-dist-in 3.4498 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.165 0.198 A 357.0 339.0 0 25 25 0 [[44, 298]] 1.0 3x2w Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IACA P05132 16 351 351.0 ACP:60403 ATPlike Active DFGin 5.7549 14.3121 BLAminus -125.73, -177.16 59.8, 78.08 -94.31, 23.06 273.35, 54.81 -46.36, -37.92 in-in in 8.8851 Saltbr-in 2.7214 HRD-in -73.57, -53.97 72.67, 5.23 in-in-in SNCiii in-in ActLoopNT-in 2.9421 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.57, 156.93 APE9-dihe-na 137.19, -153.99 APE8-dihe-in -123.03, 128.21 APE8-rot-in 300.87 APE67-dihe-in -59.06, -23.99 -31.47, -61.7 APE12-dist-in 8.1573 APE11-dist-in 11.5147 APE10-dist-in 5.9848 APE9-dist-in 3.5015 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.15 0.181 0.212 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iac Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IADA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.6579 14.362 BLAminus -130.04, -179.13 63.0, 77.66 -87.34, 22.78 276.11, 53.54 -55.12, -31.28 in-in in 9.0855 Saltbr-in 2.8296 HRD-in -93.22, -52.19 70.15, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.9352 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.54, 160.6 APE9-dihe-na 133.65, -143.98 APE8-dihe-in -130.05, 134.5 APE8-rot-in 298.49 APE67-dihe-in -67.08, -22.74 -48.94, -44.54 APE12-dist-in 8.0511 APE11-dist-in 11.5496 APE10-dist-in 6.0873 APE9-dist-in 3.5214 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.189 0.243 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4iad Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAFA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.9427 14.1301 BLAminus -121.29, 178.82 64.06, 84.8 -98.0, 27.2 281.56, 65.38 -51.93, -33.25 in-in in 8.8711 Saltbr-in 2.6687 HRD-in -76.48, -53.65 65.3, 9.94 in-in-in SNCiii in-in ActLoopNT-in 2.9738 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.4, 160.11 APE9-dihe-na 128.66, -151.44 APE8-dihe-in -123.86, 135.06 APE8-rot-in 298.27 APE67-dihe-in -57.84, -25.84 -42.55, -55.44 APE12-dist-in 8.1629 APE11-dist-in 11.523 APE10-dist-in 5.9727 APE9-dist-in 3.5632 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.16 0.192 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iaf Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAIA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.4651 14.5028 BLAminus -125.1, 176.4 64.24, 81.88 -90.74, 22.64 269.91, 49.4 -55.45, -35.99 in-in in 9.1007 Saltbr-in 2.7138 HRD-in -91.06, -49.32 68.79, 15.16 in-in-in SNCiii in-in ActLoopNT-in 2.9385 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.75, 156.86 APE9-dihe-na 141.29, -148.36 APE8-dihe-in -128.24, 130.8 APE8-rot-in 300.02 APE67-dihe-in -62.27, -23.0 -47.39, -47.75 APE12-dist-in 7.9453 APE11-dist-in 11.4584 APE10-dist-in 5.8673 APE9-dist-in 3.6084 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.171 0.209 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iai Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAKA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.7052 14.5691 BLAminus -126.92, 179.61 63.08, 81.74 -90.27, 23.65 270.26, 53.44 -59.05, -31.45 in-in in 8.9848 Saltbr-in 2.7471 HRD-in -94.54, -49.89 67.85, 16.15 in-in-in SNCiii in-in ActLoopNT-in 2.9098 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.92, 164.74 APE9-dihe-na 131.87, -148.57 APE8-dihe-in -130.85, 127.67 APE8-rot-in 297.68 APE67-dihe-in -61.28, -21.91 -43.91, -50.7 APE12-dist-in 7.9618 APE11-dist-in 11.4433 APE10-dist-in 5.9794 APE9-dist-in 3.5447 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.6 0.185 0.222 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4iak Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAYA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.806 14.2571 BLAminus -131.74, 174.05 67.76, 85.89 -95.28, 20.31 273.12, 61.73 -48.17, -36.05 in-in in 9.0392 Saltbr-in 2.9406 HRD-in -89.87, -50.65 68.98, 10.01 in-in-in SNCiii in-in ActLoopNT-in 3.055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.39, 159.46 APE9-dihe-na 132.54, -148.24 APE8-dihe-in -127.91, 130.95 APE8-rot-in 300.76 APE67-dihe-in -63.09, -19.35 -45.58, -49.88 APE12-dist-in 8.0893 APE11-dist-in 11.4657 APE10-dist-in 5.991 APE9-dist-in 3.8226 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.182 0.227 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iay Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAZA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 6.1438 14.6353 BLAminus -132.33, 171.23 62.84, 84.78 -94.94, 21.85 278.49, 61.31 -54.74, -28.93 in-in in 9.2192 Saltbr-in 2.747 HRD-in -95.03, -54.93 73.76, 14.73 in-in-in SNCiii in-in ActLoopNT-in 3.017 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.57, 164.74 APE9-dihe-na 127.12, -150.82 APE8-dihe-in -127.02, 138.46 APE8-rot-in 303.51 APE67-dihe-in -63.11, -25.72 -51.71, -47.83 APE12-dist-in 7.9634 APE11-dist-in 11.5144 APE10-dist-in 5.9788 APE9-dist-in 3.5741 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.85 0.201 0.248 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4iaz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IB0A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.7134 14.4391 BLAminus -123.68, 176.86 65.62, 82.22 -94.42, 18.76 272.15, 51.12 -47.84, -35.86 in-in in 9.0645 Saltbr-in 3.0231 HRD-in -84.67, -55.05 71.31, 12.11 in-in-in SNCiii in-in ActLoopNT-in 2.8861 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.67, 157.49 APE9-dihe-na 139.08, -144.95 APE8-dihe-in -131.16, 131.55 APE8-rot-in 306.17 APE67-dihe-in -61.31, -24.54 -46.0, -48.78 APE12-dist-in 8.0592 APE11-dist-in 11.5164 APE10-dist-in 5.9694 APE9-dist-in 3.6924 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.87 0.219 0.287 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4ib0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IB1A P05132 14 351 351.0 ADP:60403 ATPlike Active DFGin 5.6556 14.4434 BLAminus -126.58, 171.72 66.62, 80.69 -90.79, 23.58 274.18, 53.88 -53.03, -31.34 in-in in 9.1208 Saltbr-in 2.6907 HRD-in -82.93, -51.49 69.93, 14.85 in-in-in SNCiii in-in ActLoopNT-in 2.9803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.64, 163.58 APE9-dihe-na 133.1, -151.37 APE8-dihe-in -125.38, 138.08 APE8-rot-in 304.1 APE67-dihe-in -60.15, -23.69 -50.01, -49.7 APE12-dist-in 7.9604 APE11-dist-in 11.404 APE10-dist-in 5.9611 APE9-dist-in 3.6354 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.196 0.223 A 356.0 338.0 0 25 25 0 [[44, 298]] 1.0 4ib1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IB3A P05132 13 351 351.0 ADP:60401 ATPlike Active DFGin 5.973 14.2146 BLAminus -125.69, 173.12 66.37, 84.97 -98.59, 21.41 276.57, 60.51 -51.27, -29.52 in-in in 8.9902 Saltbr-in 2.7598 HRD-in -77.27, -49.79 61.58, 13.48 in-in-in SNCiii in-in ActLoopNT-in 2.8695 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.06, 160.46 APE9-dihe-na 127.6, -161.57 APE8-dihe-in -110.98, 129.89 APE8-rot-in 305.68 APE67-dihe-in -58.89, -23.07 -39.61, -54.94 APE12-dist-in 8.0781 APE11-dist-in 11.5224 APE10-dist-in 5.9229 APE9-dist-in 3.5677 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.182 0.228 A 356.0 339.0 0 25 25 0 [[44, 298]] 1.0 4ib3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4XW4A P05132 15 351 351.0 ANP:60403 ATPlike Active DFGin 5.673 14.5624 BLAminus -117.82, -177.44 65.15, 79.34 -92.69, 26.58 269.45, 57.64 -61.99, -28.36 in-in in 8.9306 Saltbr-in 2.8579 HRD-in -86.05, -50.94 67.2, 15.72 in-in-in SNCiii in-in ActLoopNT-in 3.0139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.62, 159.69 APE9-dihe-na 135.12, -140.29 APE8-dihe-in -136.84, 125.12 APE8-rot-in 301.75 APE67-dihe-in -61.52, -26.6 -45.5, -44.66 APE12-dist-in 7.961 APE11-dist-in 11.4188 APE10-dist-in 5.9353 APE9-dist-in 3.6644 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.82 0.183 0.24 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4xw4 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4XW5A P05132 15 351 351.0 ATP:60403 ATPlike Active DFGin 5.971 14.2215 BLAminus -131.24, 177.82 59.66, 87.19 -93.08, 25.08 282.37, 63.43 -53.77, -29.24 in-in in 9.2129 Saltbr-in 2.673 HRD-in -90.87, -48.94 63.52, 13.92 in-in-in SNCiii in-in ActLoopNT-in 2.8122 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.24, 155.03 APE9-dihe-na 137.47, -160.98 APE8-dihe-in -110.31, 133.6 APE8-rot-in 304.05 APE67-dihe-in -58.14, -25.36 -48.87, -50.12 APE12-dist-in 8.0264 APE11-dist-in 11.6005 APE10-dist-in 6.1002 APE9-dist-in 3.9217 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.185 0.252 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4xw5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4XW6A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.9823 14.431 BLAminus -130.68, 178.48 65.03, 84.15 -99.24, 23.41 276.01, 56.03 -60.45, -23.49 in-in in 9.1497 Saltbr-in 2.7348 HRD-in -94.59, -52.61 68.2, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.7909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.91, 154.59 APE9-dihe-na 136.7, -154.91 APE8-dihe-in -121.39, 127.95 APE8-rot-in 293.9 APE67-dihe-in -62.75, -24.38 -45.59, -46.76 APE12-dist-in 8.0512 APE11-dist-in 11.6319 APE10-dist-in 6.051 APE9-dist-in 3.787 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.186 0.265 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4xw6 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6E21A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.5937 14.0551 BLAminus -122.61, 176.37 63.02, 83.41 -94.2, 28.27 284.3, 46.09 -48.88, -41.13 in-in in 9.0287 Saltbr-in 2.6073 HRD-in -74.35, -56.8 67.48, 11.51 in-in-in SNCiii in-in ActLoopNT-in 2.9072 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.7, 159.01 APE9-dihe-na 131.41, -152.84 APE8-dihe-in -125.29, 130.56 APE8-rot-in 303.23 APE67-dihe-in -58.42, -25.04 -35.36, -60.06 APE12-dist-in 8.0433 APE11-dist-in 11.5842 APE10-dist-in 6.0224 APE9-dist-in 3.5802 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.187 0.217 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 6e21 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7E0ZA P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 5.5662 13.8842 BLAminus -118.85, -174.47 59.93, 79.47 -94.43, 25.89 275.59, 63.85 -59.78, -31.6 in-in in 8.6241 Saltbr-in 2.9777 HRD-in -96.8, -56.38 78.26, 13.74 in-in-in SNCiii in-in ActLoopNT-in 2.9292 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.91, 162.74 APE9-dihe-na 131.67, -149.57 APE8-dihe-in -131.04, 130.65 APE8-rot-in 294.41 APE67-dihe-in -63.42, -12.5 -45.48, -52.1 APE12-dist-in 7.8999 APE11-dist-in 11.1823 APE10-dist-in 5.721 APE9-dist-in 3.4 None TPO198,SEP339 TPO198,SEP339 XRAY 2.162 0.184 0.228 A 358.0 337.0 0 25 25 0 [[44, 298]] 1.0 7e0z Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DG3E P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.4812 14.3421 BLAminus -115.99, -176.62 61.62, 77.98 -90.25, 24.84 270.29, 54.4 -55.44, -35.73 in-in in 8.842 Saltbr-in 2.6947 HRD-in -87.1, -53.93 73.82, 10.76 in-in-in SNCiii in-in ActLoopNT-in 2.8817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.46, 161.61 APE9-dihe-na 135.41, -150.07 APE8-dihe-in -129.52, 135.22 APE8-rot-in 300.3 APE67-dihe-in -58.11, -23.91 -46.28, -51.67 APE12-dist-in 8.1435 APE11-dist-in 11.4816 APE10-dist-in 5.8864 APE9-dist-in 3.4048 R337A SEP140,TPO198 SEP140,TPO198 XRAY 1.8 0.185 0.217 E 371.0 337.0 0 25 25 0 [[44, 298]] 1.0 4dg3 Mus musculus AGC_PRKACA_MOUSE AGC 1.8e-94 321.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3FHIA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.4633 14.263 BLAminus -118.0, -179.45 64.04, 75.7 -86.07, 24.14 267.17, 53.33 -59.82, -32.06 in-in in 8.8874 Saltbr-in 2.7901 HRD-in -94.84, -53.37 68.02, 7.49 in-in-in SNCiii in-in ActLoopNT-in 2.8652 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.67, 136.88 APE9-dihe-na 156.84, -158.52 APE8-dihe-in -126.08, 132.83 APE8-rot-in 296.09 APE67-dihe-in -67.08, -19.88 -42.62, -50.01 APE12-dist-in 8.2333 APE11-dist-in 11.1199 APE10-dist-in 5.402 APE9-dist-in 3.5636 C200A TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.199 0.226 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3fhi Mus musculus AGC_PRKACA_MOUSE AGC 1e-93 319.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3QAME P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.5585 14.1896 BLAminus -125.2, -173.2 57.82, 79.24 -94.32, 24.42 273.28, 56.46 -52.36, -33.22 in-in in 8.9798 Saltbr-in 2.8042 HRD-in -80.54, -55.75 67.52, 12.49 in-in-in SNCiii in-in ActLoopNT-in 2.8883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.45, 157.56 APE9-dihe-na 134.84, -152.56 APE8-dihe-in -129.9, 127.65 APE8-rot-in 298.13 APE67-dihe-in -57.31, -20.14 -26.19, -66.74 APE12-dist-in 8.0939 APE11-dist-in 11.2769 APE10-dist-in 5.8065 APE9-dist-in 3.475 E209A TPO198,SEP339 TPO198,SEP339 XRAY 1.92 0.195 0.228 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 3qam Mus musculus AGC_PRKACA_MOUSE AGC 2.2e-93 318.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3QALE P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.6399 14.4013 BLAminus -123.21, -177.09 59.31, 80.89 -94.71, 25.93 269.1, 56.43 -54.28, -32.32 in-in in 9.0502 Saltbr-in 2.6578 HRD-in -84.64, -51.07 65.64, 14.74 in-in-in SNCiii in-in ActLoopNT-in 2.9615 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.61, 159.73 APE9-dihe-na 131.58, -155.18 APE8-dihe-in -126.66, 132.34 APE8-rot-in 301.51 APE67-dihe-in -57.77, -23.32 -31.31, -63.36 APE12-dist-in 8.0621 APE11-dist-in 11.3091 APE10-dist-in 5.7435 APE9-dist-in 3.5307 R281A TPO198,SEP339 TPO198,SEP339 XRAY 1.7 0.176 0.194 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 3qal Mus musculus AGC_PRKACA_MOUSE AGC 4.5e-93 317.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1RDQE P05132 2 351 351.0 ADP:60599,ATP:60600 ATPlike,ATPlike Active DFGin 5.7065 14.5148 BLAminus -117.27, 178.71 64.74, 81.19 -90.07, 21.82 270.96, 52.48 -58.25, -31.62 in-in in 9.0905 Saltbr-in 2.719 HRD-in -91.16, -53.36 73.19, 12.39 in-in-in SNCiii in-in ActLoopNT-in 2.9357 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.91, 159.57 APE9-dihe-na 132.64, -151.85 APE8-dihe-in -127.7, 133.09 APE8-rot-in 298.45 APE67-dihe-in -59.33, -27.24 -47.42, -47.34 APE12-dist-in 8.1158 APE11-dist-in 11.4138 APE10-dist-in 5.8307 APE9-dist-in 3.5208 Y205A TPO198,SEP339 TPO198,SEP339 XRAY 1.26 0.132 0.162 E 350.0 342.0 0 25 25 0 [[44, 298]] 1.0 1rdq Mus musculus AGC_PRKACA_MOUSE AGC 1.1e-92 315.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4O22A P05132 16 351 351.0 No_ligand No_ligand Active DFGin 6.4485 14.5482 BLAminus -124.93, -179.58 65.24, 83.52 -97.55, 25.76 273.08, 60.4 -61.15, -26.72 in-in in 8.8242 Saltbr-in 2.6383 HRD-in -89.28, -52.27 69.65, 12.56 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.45, 162.83 APE9-dihe-na 131.87, -150.17 APE8-dihe-in -128.05, 135.42 APE8-rot-in 301.96 APE67-dihe-in -61.83, -23.3 -46.45, -50.3 APE12-dist-in 7.9967 APE11-dist-in 11.4143 APE10-dist-in 5.8621 APE9-dist-in 3.5438 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.187 0.219 A 342.0 336.0 0 25 25 0 [[44, 298]] 1.0 4o22 Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1JLUE P05132 13 351 351.0 No_ligand No_ligand Active DFGin 6.2861 14.0335 BLAminus -116.82, 172.06 62.47, 85.22 -99.38, 25.33 280.76, 66.77 -59.89, -25.29 in-in in 8.8849 Saltbr-in 2.9045 HRD-in -82.77, -54.36 73.92, -0.29 in-in-in SNCiii in-in ActLoopNT-in 3.0022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.81, 157.32 APE9-dihe-na 139.21, -153.09 APE8-dihe-in -125.03, 121.3 APE8-rot-in 316.06 APE67-dihe-in -62.91, -9.39 -23.05, -64.85 APE12-dist-in 8.0643 APE11-dist-in 11.3222 APE10-dist-in 6.0555 APE9-dist-in 3.703 None TPO198,SEP339 TPO198,SEP339 XRAY 2.25 0.181 999.0 E 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1jlu Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DG2E P05132 2 351 351.0 No_ligand No_ligand Active DFGin 6.4783 14.3469 BLAminus -123.83, 172.03 63.45, 88.02 -99.08, 27.68 275.25, 59.55 -56.12, -32.76 in-in in 8.8184 Saltbr-in 2.7992 HRD-in -84.63, -52.84 71.55, 8.96 in-in-in SNCiii in-in ActLoopNT-in 2.9185 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.79, 159.19 APE9-dihe-na 134.75, -147.2 APE8-dihe-in -130.86, 129.22 APE8-rot-in 304.99 APE67-dihe-in -62.19, -22.69 -40.4, -52.05 APE12-dist-in 8.0585 APE11-dist-in 11.3519 APE10-dist-in 5.7561 APE9-dist-in 3.4964 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.193 0.211 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4dg2 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFZE P05132 2 351 351.0 No_ligand No_ligand Active DFGin 6.3314 14.3533 BLAminus -124.21, 173.53 63.45, 88.27 -99.9, 27.01 273.13, 59.34 -56.57, -31.28 in-in in 8.7729 Saltbr-in 2.6928 HRD-in -87.8, -52.9 69.53, 11.47 in-in-in SNCiii in-in ActLoopNT-in 2.9057 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.19, 159.25 APE9-dihe-na 132.22, -141.79 APE8-dihe-in -134.47, 128.83 APE8-rot-in 307.05 APE67-dihe-in -59.16, -25.89 -40.01, -52.76 APE12-dist-in 8.0313 APE11-dist-in 11.343 APE10-dist-in 5.7654 APE9-dist-in 3.4388 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.207 0.234 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4dfz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1APME P05132 11 351 351.0 No_ligand No_ligand Active DFGin 6.2608 14.0704 BLAminus -125.0, 178.22 62.58, 88.79 -105.13, 25.26 274.83, 66.5 -57.51, -25.56 in-in in 8.9302 Saltbr-in 2.582 HRD-in -81.09, -58.27 71.67, -2.38 in-in-in SNCiii in-in ActLoopNT-in 3.0534 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.78, 156.67 APE9-dihe-na 136.06, -155.51 APE8-dihe-in -123.48, 123.72 APE8-rot-in 302.63 APE67-dihe-in -54.93, -28.48 -32.82, -58.43 APE12-dist-in 8.2172 APE11-dist-in 11.4562 APE10-dist-in 5.9547 APE9-dist-in 3.7877 S140A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.186 999.0 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1apm Mus musculus AGC_PRKACA_MOUSE AGC 2.2e-94 321.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1BX6A P05132 13 351 351.0 BA1:60351 Type1 Active DFGin 6.0974 14.2707 BLAminus -131.41, 157.86 79.35, 91.47 -96.7, 9.79 287.76, 86.24 -44.29, -77.97 in-in in 8.3994 Saltbr-in 2.6074 HRD-in -60.43, -49.37 65.58, 0.7 in-in-in SNCiii in-in ActLoopNT-in 3.1024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -96.41, 136.41 APE9-dihe-na 139.93, 174.47 APE8-dihe-in -112.82, 117.81 APE8-rot-in 289.91 APE67-dihe-in -32.61, -31.36 -25.94, -76.91 APE12-dist-in 8.7332 APE11-dist-in 11.1899 APE10-dist-in 5.2412 APE9-dist-in 4.7598 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.21 0.34 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1bx6 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1FMOE P05132 14 351 351.0 ADN:60351 Type1 Active DFGin 6.6779 14.2824 BLAminus -114.95, 166.87 67.95, 101.15 -111.54, 7.58 268.05, 65.13 -43.18, -17.52 in-in in 8.5604 Saltbr-in 2.9824 HRD-in -73.08, -60.95 74.44, -3.64 in-in-in SNCiii in-in ActLoopNT-in 2.8596 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.53, 167.98 APE9-dihe-na 127.76, -157.13 APE8-dihe-in -115.17, 123.5 APE8-rot-in 303.04 APE67-dihe-in -62.85, -32.38 -37.72, -49.63 APE12-dist-in 7.9343 APE11-dist-in 11.2764 APE10-dist-in 5.9475 APE9-dist-in 3.7123 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.182 999.0 E 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1fmo Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1REJA P05132 17 351 351.0 B1L:60351 Type1 Active DFGin 6.6885 14.7589 BLAminus -129.16, -166.14 53.21, 69.99 -91.05, 27.11 275.8, 67.71 -67.13, -23.58 in-in in 9.1448 Saltbr-in 2.806 HRD-in -84.89, -51.08 67.36, 19.76 in-in-in SNCiii in-in ActLoopNT-in 2.7199 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.7, 155.59 APE9-dihe-na 102.81, -168.4 APE8-dihe-in -114.34, 132.29 APE8-rot-in 300.68 APE67-dihe-in -62.15, -27.72 -40.87, -53.2 APE12-dist-in 8.0818 APE11-dist-in 11.1003 APE10-dist-in 5.4023 APE9-dist-in 3.4935 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.208 0.291 A 350.0 335.0 0 25 25 0 [[44, 298]] 1.0 1rej Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3OW3A P05132 16 351 351.0 SMY:60401 Type1 Active DFGin 6.1403 14.543 BLAminus -123.88, 175.12 69.78, 83.56 -97.88, 23.25 272.21, 60.42 -52.11, -32.64 in-in in 9.1321 Saltbr-in 2.5499 HRD-in -87.74, -52.86 72.88, 7.11 in-in-in SNCiii in-in ActLoopNT-in 2.9121 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.65, 165.29 APE9-dihe-na 128.58, -156.74 APE8-dihe-in -122.61, 136.92 APE8-rot-in 295.99 APE67-dihe-in -53.86, -28.98 -54.05, -45.53 APE12-dist-in 8.1185 APE11-dist-in 11.5674 APE10-dist-in 5.8554 APE9-dist-in 3.5108 None TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.166 0.21 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 3ow3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2ERZE P05132 16 351 351.0 HFS:60351 Type1 Active DFGin 5.8621 14.2868 BLAminus -120.01, 167.35 70.07, 90.43 -101.1, 32.12 275.39, 49.09 -53.89, -29.79 in-in in 9.0354 Saltbr-in 2.6896 HRD-in -71.67, -48.74 64.28, 7.57 in-in-in SNCiii in-in ActLoopNT-in 2.9432 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.95, 164.31 APE9-dihe-na 126.82, -161.82 APE8-dihe-in -117.41, 128.23 APE8-rot-in 308.76 APE67-dihe-in -49.78, -31.46 -30.24, -67.82 APE12-dist-in 8.1923 APE11-dist-in 11.4229 APE10-dist-in 5.9098 APE9-dist-in 3.5597 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.227 0.287 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2erz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1REKA P05132 14 351 351.0 B8L:60351,PTL:60352 Type1,Allosteric Active DFGin 6.5124 14.951 BLAminus -126.84, -171.52 53.94, 74.01 -96.88, 22.16 273.96, 65.3 -56.46, -42.1 in-in in 8.8618 Saltbr-in 2.7916 HRD-in -90.9, -46.82 65.04, 3.0 in-in-in SNCiii in-in ActLoopNT-in 2.9322 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.61, 143.64 APE9-dihe-na 123.06, -169.72 APE8-dihe-in -113.81, 132.41 APE8-rot-in 289.91 APE67-dihe-in -65.44, -22.63 -41.39, -49.51 APE12-dist-in 8.0968 APE11-dist-in 10.719 APE10-dist-in 5.1557 APE9-dist-in 3.3485 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.218 0.295 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1rek Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM6C P05132 19 351 351.0 ANP:60402 ATPlike Inactive DFGin 6.7799 16.0821 ABAminus -110.74, -8.1 -141.78, 125.75 -126.67, 17.79 291.81, 81.75 -52.6, -43.19 out-out out 10.4027 Saltbr-out 4.4909 HRD-in -64.73, -48.52 44.91, 28.18 out-in-out SNCoio in-out ActLoopNT-in 2.8769 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -155.16, 154.51 APE9-dihe-na 131.73, -155.42 APE8-dihe-in -119.09, 141.73 APE8-rot-out 198.33 APE67-dihe-in -57.79, -26.12 -45.84, -50.95 APE12-dist-in 8.5303 APE11-dist-in 11.8147 APE10-dist-in 6.3058 APE9-dist-in 4.5025 None TPO198,SEP339 TPO198,SEP339 XRAY 2.39 0.225 0.261 C 339.0 322.0 0 25 25 0 [[44, 298]] 1.0 6mm6 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM6E P05132 19 351 351.0 ANP:60401 ATPlike Inactive DFGin 6.7325 15.9653 ABAminus -112.26, -9.59 -137.74, 126.1 -127.73, 18.87 290.52, 82.39 -53.04, -44.19 out-out out 10.2709 Saltbr-out 5.278 HRD-in -66.74, -47.88 44.41, 27.02 out-in-out SNCoio in-out ActLoopNT-in 2.8731 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -157.27, 155.34 APE9-dihe-na 128.78, -154.8 APE8-dihe-in -120.26, 141.99 APE8-rot-out 197.33 APE67-dihe-in -57.79, -26.44 -45.46, -51.33 APE12-dist-in 8.4779 APE11-dist-in 11.8514 APE10-dist-in 6.3306 APE9-dist-in 4.4228 None TPO198,SEP339 TPO198,SEP339 XRAY 2.39 0.225 0.261 E 339.0 320.0 0 25 25 0 [[44, 298]] 1.0 6mm6 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM7A P05132 17 351 351.0 ANP:60406 ATPlike Inactive DFGin 6.7159 15.4284 ABAminus -112.23, -9.6 -137.01, 123.03 -130.15, 19.3 297.15, 81.39 -54.86, -42.58 out-out out 10.2821 Saltbr-out 4.6231 HRD-in -76.47, -53.66 52.13, 28.38 out-in-out SNCoio in-out ActLoopNT-in 2.8634 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -163.99, 161.65 APE9-dihe-na 126.52, -159.69 APE8-dihe-in -119.22, 141.71 APE8-rot-out 195.45 APE67-dihe-in -67.85, -20.3 -44.24, -48.26 APE12-dist-in 8.2035 APE11-dist-in 11.1251 APE10-dist-in 5.7383 APE9-dist-in 3.9708 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.213 0.238 A 339.0 327.0 0 25 25 0 [[44, 298]] 1.0 6mm7 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM7D P05132 16 351 351.0 ANP:60405 ATPlike Inactive DFGin 6.6517 15.4584 ABAminus -113.01, -9.74 -137.13, 123.49 -128.55, 17.46 296.74, 82.18 -52.99, -42.79 out-out out 10.3794 Saltbr-out 5.8168 HRD-in -73.81, -53.25 53.83, 26.23 out-in-out SNCoio in-out ActLoopNT-in 2.8742 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -166.02, 161.72 APE9-dihe-na 122.21, -160.7 APE8-dihe-in -119.01, 142.81 APE8-rot-out 192.42 APE67-dihe-in -67.72, -20.93 -42.31, -48.3 APE12-dist-in 8.2101 APE11-dist-in 11.2017 APE10-dist-in 5.7858 APE9-dist-in 3.9614 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.213 0.238 D 339.0 324.0 0 25 25 0 [[44, 298]] 1.0 6mm7 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM8C P05132 16 351 351.0 ANP:60403 ATPlike Inactive DFGin 6.6132 15.2001 ABAminus -113.8, -10.95 -132.36, 129.54 -134.0, 24.39 301.03, 83.83 -57.02, -38.35 out-out out 10.3401 Saltbr-out 7.3235 HRD-in -73.54, -53.96 54.41, 29.61 out-in-out SNCoio in-out ActLoopNT-in 2.7764 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.79, 167.54 APE9-dihe-na 115.95, -161.99 APE8-dihe-in -118.41, 142.14 APE8-rot-out 195.18 APE67-dihe-in -66.48, -19.98 -46.61, -45.65 APE12-dist-in 8.1252 APE11-dist-in 11.2017 APE10-dist-in 5.8341 APE9-dist-in 3.9965 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.183 0.221 C 339.0 325.0 0 25 25 0 [[44, 298]] 1.0 6mm8 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKND P05132 16 351 351.0 ANP:60400 ATPlike Inactive DFGin 6.6105 14.9582 ABAminus -121.75, -47.3 -93.55, 119.31 -121.12, 22.25 288.77, 83.91 -60.17, -43.74 in-out in 9.6363 Saltbr-out 4.003 HRD-in -71.48, -47.99 39.7, 38.93 out-in-in SNCoii in-in ActLoopNT-in 2.9756 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.1, 161.55 APE9-dihe-na 104.53, 169.82 APE8-dihe-in -72.88, 137.25 APE8-rot-in 280.42 APE67-dihe-in -60.56, -25.71 -55.68, -37.9 APE12-dist-in 8.0946 APE11-dist-in 11.2355 APE10-dist-in 5.8091 APE9-dist-in 4.6921 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 D 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKOE P05132 16 351 351.0 ANP:60403 ATPlike Inactive DFGin 6.0364 14.5957 ABAminus -122.57, -57.22 -79.99, 109.96 -108.47, 33.73 286.2, 84.93 -64.54, -41.62 in-in in 9.7403 Saltbr-in 3.5644 HRD-in -78.91, -48.33 66.16, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.8677 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.15, 159.43 APE9-dihe-na 137.57, -133.12 APE8-dihe-in -144.28, 132.68 APE8-rot-in 289.09 APE67-dihe-in -62.87, -18.89 -48.53, -47.79 APE12-dist-in 8.0799 APE11-dist-in 11.3212 APE10-dist-in 5.8296 APE9-dist-in 3.774 None TPO198,SEP339 TPO198,SEP339 XRAY 2.89 0.213 0.259 E 339.0 336.0 0 25 25 0 [[44, 298]] 1.0 8uko Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKPE P05132 17 351 351.0 ANP:60402 ATPlike Inactive DFGin 6.1336 14.4301 ABAminus -106.11, -56.02 -81.74, 124.54 -123.06, 18.4 279.21, 82.41 -57.4, -55.55 in-out in 9.2794 Saltbr-out 4.1807 HRD-in -89.57, -52.98 66.95, 19.28 out-in-in SNCoii in-in ActLoopNT-in 2.9525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.29, 147.38 APE9-dihe-na 136.74, -150.06 APE8-dihe-in -126.21, 134.43 APE8-rot-in 318.02 APE67-dihe-in -77.56, -4.79 -54.58, -35.83 APE12-dist-in 7.9285 APE11-dist-in 10.8204 APE10-dist-in 5.1851 APE9-dist-in 3.8514 None SEP140,TPO198 SEP140,TPO198 XRAY 2.85 0.242 0.281 E 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukp Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTTB P05132 11 351 351.0 ADP:60401 ATPlike Inactive DFGin 6.5417 14.8798 ABAminus -93.85, -35.44 -119.41, 118.31 -113.9, 43.83 296.85, 78.9 -65.87, -49.34 in-none in 9.8688 Saltbr-none 999.0 HRD-in -94.05, -37.34 60.44, 1.66 none-in-in SNCnii in-in ActLoopNT-in 2.7867 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -166.4, 146.42 APE9-dihe-na 126.7, -158.4 APE8-dihe-in -116.99, 137.33 APE8-rot-in 273.8 APE67-dihe-in -64.02, -34.69 -52.94, -43.07 APE12-dist-in 7.7129 APE11-dist-in 10.7197 APE10-dist-in 5.2983 APE9-dist-in 4.164 K8C TPO198,SEP339 TPO198,SEP339 XRAY 3.5 0.23 0.284 B 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 4ntt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKNC P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.9773 15.8143 ABAminus -121.28, -46.06 -94.44, 119.11 -121.88, 20.98 289.09, 82.99 -60.59, -43.51 out-out out 10.2655 Saltbr-out 3.7763 HRD-in -69.49, -46.7 40.24, 37.27 out-in-in SNCoii in-in ActLoopNT-in 2.8604 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.14, 161.55 APE9-dihe-na 102.26, 166.3 APE8-dihe-in -75.0, 136.39 APE8-rot-in 285.29 APE67-dihe-in -59.55, -25.47 -55.27, -37.71 APE12-dist-in 8.2631 APE11-dist-in 11.3425 APE10-dist-in 5.8906 APE9-dist-in 4.4404 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 C 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKNF P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.8893 15.4858 ABAminus -119.02, -48.36 -94.42, 119.64 -122.07, 21.3 289.06, 84.07 -60.37, -43.79 in-none in 9.9681 Saltbr-none 999.0 HRD-in -70.24, -47.3 40.22, 39.45 none-in-out SNCnio in-out ActLoopNT-in 3.1956 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -150.61, 160.97 APE9-dihe-na 102.69, 167.59 APE8-dihe-in -73.59, 140.15 APE8-rot-out 204.21 APE67-dihe-in -61.18, -25.59 -54.92, -37.71 APE12-dist-in 8.0636 APE11-dist-in 11.1851 APE10-dist-in 5.795 APE9-dist-in 4.6032 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 F 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKNH P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.9904 15.9406 ABAminus -119.65, -47.17 -95.12, 119.59 -123.41, 20.33 289.47, 82.92 -60.29, -43.54 out-out out 10.3777 Saltbr-out 4.1022 HRD-in -70.28, -46.9 40.49, 37.83 out-in-in SNCoii in-in ActLoopNT-in 2.9436 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.73, 160.95 APE9-dihe-na 102.27, 168.23 APE8-dihe-in -75.08, 137.2 APE8-rot-in 283.98 APE67-dihe-in -59.99, -25.87 -55.81, -37.99 APE12-dist-in 8.247 APE11-dist-in 11.3303 APE10-dist-in 5.9313 APE9-dist-in 4.5321 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 H 339.0 325.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3TNPC P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.4124 14.047 ABAminus -115.86, -60.86 -88.32, 106.92 -98.77, 21.04 269.52, 52.68 -48.7, -36.28 in-in in 8.6 Saltbr-in 2.8944 HRD-in -94.29, -50.01 72.25, 4.59 in-in-in SNCiii in-in ActLoopNT-in 2.9018 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.71, 164.13 APE9-dihe-na 136.51, -140.88 APE8-dihe-in -134.73, 130.62 APE8-rot-in 292.72 APE67-dihe-in -54.62, -27.98 -43.74, -54.69 APE12-dist-in 8.0801 APE11-dist-in 11.4918 APE10-dist-in 5.9315 APE9-dist-in 3.4025 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.3 0.226 0.235 C 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 3tnp Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3TNPF P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.4122 14.0463 ABAminus -115.9, -60.86 -88.39, 106.92 -98.78, 21.05 269.48, 52.72 -48.68, -36.31 in-in in 8.5999 Saltbr-in 2.8941 HRD-in -94.19, -50.06 72.23, 4.62 in-in-in SNCiii in-in ActLoopNT-in 2.9156 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.7, 164.08 APE9-dihe-na 136.57, -140.81 APE8-dihe-in -134.76, 130.54 APE8-rot-in 292.72 APE67-dihe-in -54.65, -27.95 -43.69, -54.69 APE12-dist-in 8.0809 APE11-dist-in 11.4916 APE10-dist-in 5.9317 APE9-dist-in 3.4021 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.3 0.226 0.235 F 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 3tnp Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4WBBB P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 5.8987 14.309 ABAminus -133.99, -40.66 -108.42, 103.56 -98.82, 16.34 272.05, 61.48 -51.24, -35.82 in-in in 8.5861 Saltbr-in 2.7679 HRD-in -93.67, -38.46 55.43, 10.07 in-in-in SNCiii in-in ActLoopNT-in 2.8579 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.35, 160.13 APE9-dihe-na 145.06, -138.63 APE8-dihe-in -131.95, 132.94 APE8-rot-in 298.17 APE67-dihe-in -60.16, -16.13 -44.42, -52.54 APE12-dist-in 8.043 APE11-dist-in 11.467 APE10-dist-in 6.061 APE9-dist-in 3.5781 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.8 0.232 0.279 B 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4wbb Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4X6QC P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.5826 13.9706 ABAminus -121.1, -42.58 -93.87, 102.7 -97.14, 17.55 267.16, 62.54 -52.57, -22.85 in-in in 8.4246 Saltbr-in 2.6995 HRD-in -93.89, -54.89 78.5, 7.23 in-in-in SNCiii in-in ActLoopNT-in 3.0582 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.45, 165.62 APE9-dihe-na 127.31, -150.86 APE8-dihe-in -123.77, 131.23 APE8-rot-in 300.08 APE67-dihe-in -68.69, -15.9 -43.09, -45.27 APE12-dist-in 8.1005 APE11-dist-in 11.4859 APE10-dist-in 6.067 APE9-dist-in 3.4046 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.52 0.201 0.261 C 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4x6q Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTSA P05132 9 351 351.0 No_ligand No_ligand Inactive DFGin 6.538 15.9677 ABAminus -126.95, 0.97 -130.38, 129.83 -128.18, 8.25 284.09, 78.17 -52.18, -25.55 out-out out 10.2859 Saltbr-out 5.443 HRD-in -88.58, -45.11 67.09, 10.84 out-in-in SNCoii in-in ActLoopNT-in 2.9409 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.79, 153.47 APE9-dihe-na 119.65, -179.72 APE8-dihe-in -98.33, 124.38 APE8-rot-in 308.71 APE67-dihe-in -60.54, -27.51 -31.45, -47.3 APE12-dist-in 8.167 APE11-dist-in 11.4446 APE10-dist-in 6.0844 APE9-dist-in 4.2286 K8C TPO198,SEP339 TPO198,SEP339 XRAY 2.9 0.247 0.292 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 4nts Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTSB P05132 9 351 351.0 No_ligand No_ligand Inactive DFGin 6.0263 15.2864 ABAminus -111.39, -34.44 -108.24, 143.4 -134.27, 5.96 285.1, 84.22 -48.51, -37.04 in-none in 9.8214 Saltbr-none 999.0 HRD-in -84.15, -38.94 58.73, 4.32 none-in-in SNCnii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.51, 126.13 APE9-dihe-na 95.83, -178.74 APE8-dihe-in -68.15, 137.5 APE8-rot-in 299.78 APE67-dihe-in -69.28, -28.37 -49.3, -45.44 APE12-dist-in 8.2193 APE11-dist-in 10.3859 APE10-dist-in 5.3483 APE9-dist-in 4.0024 K8C TPO198,SEP339 TPO198,SEP339 XRAY 2.9 0.247 0.292 B 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 4nts Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 5X3FB P05132 5 317 351.0 No_ligand No_ligand Inactive DFGin 6.5356 15.8812 ABAminus -125.34, -3.25 -129.13, 129.62 -128.07, 7.73 283.82, 79.52 -54.86, -24.43 out-out out 10.2687 Saltbr-out 5.1184 HRD-in -88.25, -45.2 67.71, 9.27 out-in-in SNCoii in-in ActLoopNT-in 2.9322 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.56, 145.49 APE9-dihe-na 135.48, 176.97 APE8-dihe-in -97.8, 124.17 APE8-rot-in 309.27 APE67-dihe-in -59.29, -29.32 -31.89, -46.62 APE12-dist-in 8.1446 APE11-dist-in 10.7363 APE10-dist-in 5.6264 APE9-dist-in 4.2648 None TPO198 TPO198 XRAY 3.38 0.192 0.227 B 393.0 310.0 0 25 25 0 [[44, 298]] 1.0 5x3f Mus musculus AGC_PRKACA_MOUSE AGC 2.1e-94 321.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM5E P05132 16 351 351.0 ANP:60402 ATPlike Inactive DFGin 5.9604 14.3509 BLAminus -116.65, 159.11 76.02, 91.05 -92.83, 26.22 286.06, 88.09 -52.81, -36.86 in-in in 8.8493 Saltbr-in 2.8003 HRD-in -83.15, -50.88 72.11, -0.72 in-in-out SNCiio in-out ActLoopNT-in 2.8706 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.6, 159.33 APE9-dihe-na 129.67, -150.44 APE8-dihe-in -128.62, 141.57 APE8-rot-out 194.03 APE67-dihe-in -68.05, -20.18 -46.89, -45.89 APE12-dist-in 8.2074 APE11-dist-in 11.3781 APE10-dist-in 5.7976 APE9-dist-in 3.7765 None TPO198,SEP339 TPO198,SEP339 XRAY 1.95 0.183 0.227 E 339.0 336.0 0 25 25 0 [[44, 298]] 1.0 6mm5 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1ATPE P05132 16 351 351.0 ATP:60355 ATPlike Inactive DFGin 6.2296 14.5876 BLAminus -105.27, -165.6 48.73, 87.06 -105.12, 16.76 267.19, 75.22 -52.19, -32.07 in-out in 9.1613 Saltbr-out 3.6341 HRD-in -88.29, -43.64 51.81, 19.16 out-in-in SNCoii in-in ActLoopNT-in 2.8078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.21, 146.28 APE9-dihe-na 146.09, -156.15 APE8-dihe-in -133.3, 119.84 APE8-rot-in 299.98 APE67-dihe-in -65.71, -15.81 -24.26, -60.76 APE12-dist-in 8.3526 APE11-dist-in 11.4096 APE10-dist-in 5.7064 APE9-dist-in 3.9902 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.177 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1atp Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DINA P05132 10 351 351.0 ATP:60400 ATPlike Inactive DFGin 5.792 13.1437 BLAminus -127.84, -176.29 51.22, 102.02 -109.69, 31.05 287.96, 58.2 -47.08, -31.2 in-in in 8.5177 Saltbr-in 3.4979 HRD-out -64.69, -78.02 71.93, 51.46 in-in-out SNCiio in-out ActLoopNT-in 2.9942 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -152.73, 153.23 APE9-dihe-na 130.84, -154.91 APE8-dihe-in -121.15, 137.05 APE8-rot-out 34.65 APE67-dihe-in -46.77, -45.03 -45.98, -63.1 APE12-dist-in 7.9722 APE11-dist-in 10.5875 APE10-dist-in 4.9968 APE9-dist-in 3.53 None TPO198,SEP339 TPO198,SEP339 XRAY 3.7 0.211 0.293 A 350.0 342.0 0 25 25 0 [[44, 298]] 1.0 4din Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7E12A P05132 19 351 351.0 ANP:60401 ATPlike Inactive DFGin 5.3957 14.6175 BLAminus -131.26, -169.7 58.92, 77.12 -93.02, 37.73 266.27, 47.03 -71.49, -23.13 in-in in 8.8067 Saltbr-in 3.2657 HRD-out -127.04, 103.44 -105.61, 37.91 in-in-in SNCiii in-in ActLoopNT-in 2.903 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.78, 159.74 APE9-dihe-na 134.39, -158.49 APE8-dihe-in -118.85, 128.69 APE8-rot-in 308.98 APE67-dihe-in -63.3, -26.53 -50.37, -37.69 APE12-dist-in 8.03 APE11-dist-in 11.3719 APE10-dist-in 5.9651 APE9-dist-in 3.4216 None TPO198,SEP339 TPO198,SEP339 XRAY 2.796 0.208 0.252 A 358.0 333.0 0 25 25 0 [[44, 298]] 1.0 7e12 Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1JBPE P05132 10 351 351.0 ADP:60381 ATPlike Inactive DFGin 6.1283 14.0345 BLAminus -131.98, 178.81 60.97, 83.81 -101.93, 15.49 276.81, 71.17 -55.35, -24.18 in-in in 8.8688 Saltbr-in 2.7492 HRD-out -93.99, 130.53 -128.02, 39.83 in-in-in SNCiii in-in ActLoopNT-in 2.8856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.07, 156.95 APE9-dihe-na 132.9, -168.64 APE8-dihe-in -109.4, 126.7 APE8-rot-in 297.85 APE67-dihe-in -61.28, -20.5 -33.82, -53.02 APE12-dist-in 8.1215 APE11-dist-in 11.4477 APE10-dist-in 6.0125 APE9-dist-in 3.8617 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.175 999.0 E 350.0 342.0 0 25 25 0 [[44, 298]] 1.0 1jbp Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3O7LB P05132 18 351 351.0 ANP:60354 ATPlike Inactive DFGin 5.7904 14.6658 BLAminus -108.29, -170.95 57.63, 74.91 -94.92, 22.34 267.93, 64.07 -48.2, -34.6 in-in in 9.0975 Saltbr-in 2.9978 HRD-in -84.13, -53.04 68.25, 25.66 in-in-out SNCiio in-out ActLoopNT-in 2.9497 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -140.78, 178.73 APE9-dihe-na 123.03, -156.78 APE8-dihe-in -134.79, 129.02 APE8-rot-out 131.03 APE67-dihe-in -64.87, -13.33 -37.09, -52.44 APE12-dist-in 8.1152 APE11-dist-in 11.126 APE10-dist-in 5.5927 APE9-dist-in 3.4797 None TPO198 TPO198 XRAY 2.8 0.216 0.287 B 350.0 327.0 3 25 25 0 [[44, 298]] 1.0 3o7l Mus musculus AGC_PRKACA_MOUSE AGC 8.9e-94 319.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2CPKE P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.9516 14.3527 BLAminus -119.36, 179.9 54.29, 98.05 -110.06, 38.52 269.38, 72.49 -74.59, -10.83 in-in in 8.8905 Saltbr-in 3.0285 HRD-out -89.69, 114.42 -105.18, 29.22 in-in-in SNCiii in-in ActLoopNT-in 2.9084 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.45, 150.79 APE9-dihe-na 149.42, -157.84 APE8-dihe-in -117.51, 129.53 APE8-rot-in 300.38 APE67-dihe-in -65.47, -26.39 -44.25, -41.5 APE12-dist-in 8.076 APE11-dist-in 11.291 APE10-dist-in 5.9045 APE9-dist-in 3.7514 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.7 0.18 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 2cpk Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3O7LD P05132 14 351 351.0 No_ligand No_ligand Inactive DFGin 6.5881 15.3871 BLAminus -122.76, 164.56 73.91, 96.96 -115.5, 27.13 288.86, 72.99 -56.99, -35.58 in-out in 9.6773 Saltbr-out 3.7173 HRD-in -80.64, -45.25 61.11, 19.5 out-in-out SNCoio in-out ActLoopNT-in 2.9631 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -150.51, -38.18 APE9-dihe-na -70.79, 159.72 APE8-dihe-in -54.96, 142.28 APE8-rot-out 27.57 APE67-dihe-in -76.4, -17.97 -49.97, -34.37 APE12-dist-in 7.986 APE11-dist-in 11.3838 APE10-dist-in 5.9066 APE9-dist-in 3.7447 None TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.216 0.287 D 350.0 335.0 0 25 25 0 [[44, 298]] 1.0 3o7l Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 9O7VA P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.9636 14.2333 BLAminus -144.42, 177.21 64.71, 76.79 -85.39, 18.92 274.62, 10.56 -43.43, -41.22 in-out in 9.3028 Saltbr-out 5.1072 HRD-in -93.65, -55.47 73.54, 8.94 out-in-in SNCoii in-in ActLoopNT-in 2.7506 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na 179.97, 149.56 APE9-dihe-na 148.21, -144.81 APE8-dihe-in -132.69, 133.23 APE8-rot-in 300.23 APE67-dihe-in -65.9, -25.09 -38.29, -53.75 APE12-dist-in 8.3267 APE11-dist-in 10.2791 APE10-dist-in 4.966 APE9-dist-in 3.3364 None TPO198,SEP339 TPO198,SEP339 XRAY 3.7 0.234 0.293 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 9o7v Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1RE8A P05132 13 351 351.0 BD2:60351 Type1 Inactive DFGin 6.3634 14.4971 BLAminus -126.74, -163.36 52.92, 64.83 -86.7, 13.59 272.3, 77.12 -53.9, -38.74 in-in in 8.728 Saltbr-in 2.8622 HRD-out -92.25, 100.7 -92.09, 32.79 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.96, 163.56 APE9-dihe-na 123.01, -156.83 APE8-dihe-in -123.97, 134.13 APE8-rot-in 306.64 APE67-dihe-in -79.49, -1.91 -37.94, -51.41 APE12-dist-in 8.1888 APE11-dist-in 11.3883 APE10-dist-in 5.6985 APE9-dist-in 3.5296 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.197 0.252 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1re8 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTTA P05132 11 351 351.0 ADP:60401 ATPlike Inactive DFGin 6.2546 15.2208 None 58.0, -132.96 -135.23, 163.83 -122.73, 17.77 281.43, 74.72 -41.46, -50.2 in-out in 9.9815 Saltbr-out 4.1938 HRD-in -65.11, -40.77 60.9, 3.38 out-in-in SNCoii in-in ActLoopNT-in 2.8637 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.9, 118.31 APE9-dihe-na 164.12, -173.28 APE8-dihe-in -108.19, 123.7 APE8-rot-in 267.93 APE67-dihe-in -75.4, -22.82 -40.35, -37.34 APE12-dist-in 8.1876 APE11-dist-in 11.1589 APE10-dist-in 5.5421 APE9-dist-in 4.3211 None TPO198,SEP339 TPO198,SEP339 XRAY 3.5 0.23 0.284 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 4ntt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1SYKA P05132 2 351 351.0 No_ligand No_ligand Inactive DFGin 6.5487 15.2891 None -131.76, 92.58 153.52, 114.28 -135.97, 14.86 305.19, 86.4 -55.43, -35.39 out-out out 10.6501 Saltbr-out 4.6701 HRD-out -89.49, 87.61 -76.68, 28.19 out-in-in SNCoii in-in ActLoopNT-in 2.8271 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.89, 158.84 APE9-dihe-na 108.08, 161.46 APE8-dihe-in -68.78, 138.01 APE8-rot-in 292.07 APE67-dihe-in -58.35, -9.3 -44.71, -57.38 APE12-dist-in 8.6724 APE11-dist-in 11.389 APE10-dist-in 5.9774 APE9-dist-in 3.618 E231Q TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.202 0.249 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1syk Mus musculus AGC_PRKACA_MOUSE AGC 5.7e-94 320.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1SYKB P05132 14 351 351.0 No_ligand No_ligand Inactive DFGin 6.599 15.2944 None -131.1, 91.72 152.06, 111.8 -131.83, 14.93 304.13, 82.92 -52.5, -38.6 out-out out 10.6973 Saltbr-out 4.5374 HRD-out -89.8, 89.72 -78.69, 28.99 out-in-in SNCoii in-in ActLoopNT-in 2.7813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.75, 160.3 APE9-dihe-na 107.8, 162.07 APE8-dihe-in -68.75, 135.04 APE8-rot-in 292.48 APE67-dihe-in -58.91, -9.06 -42.82, -56.64 APE12-dist-in 8.6623 APE11-dist-in 11.3639 APE10-dist-in 5.9602 APE9-dist-in 3.6147 E231Q TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.202 0.249 B 350.0 325.0 0 25 25 0 [[44, 298]] 1.0 1syk Mus musculus AGC_PRKACA_MOUSE AGC 5.7e-94 320.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFYA P05132 15 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -85.64, -176.8 33.76, 66.58 -80.32, 120.49 999.0, 999.0 -82.07, 106.21 in-none in 9.9071 Saltbr-none 999.0 HRD-in -75.3, -48.75 74.17, -71.89 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanii APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 145.79 APE8-rot-in 341.44 APE67-dihe-in -58.39, -21.24 -48.4, -47.32 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 R195A SEP339 SEP339 XRAY 2.997 0.253 0.286 A 371.0 311.0 12 25 13 12 [[44, 298]] 1.0 4dfy Mus musculus AGC_PRKACA_MOUSE AGC 3.3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFYE P05132 15 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -87.32, -175.53 34.83, 65.83 -79.11, 119.4 999.0, 999.0 -80.98, 105.33 in-out in 9.7937 Saltbr-out 4.0426 HRD-in -70.47, -49.15 73.48, -78.98 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_nnoo APE10-dihe-na 999.0, -39.98 APE9-dihe-na -90.86, -172.73 APE8-dihe-in -82.11, 146.95 APE8-rot-in 336.67 APE67-dihe-in -63.39, -14.5 -53.89, -42.37 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 12.5337 APE9-dist-out 7.8184 R195A SEP339 SEP339 XRAY 2.997 0.253 0.286 E 371.0 313.0 10 25 15 10 [[44, 298]] 1.0 4dfy Mus musculus AGC_PRKACA_MOUSE AGC 3.3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1J3HA P05132 10 351 351.0 No_ligand No_ligand None DFGin 6.9571 16.5294 BLAminus -128.1, 165.84 66.16, 90.29 -100.57, 29.84 267.59, 74.49 -52.61, -63.31 out-none out 10.2685 Saltbr-none 999.0 HRD-in -65.94, -47.85 41.03, 47.95 none-in-in SNCnii in-in ActLoopNT-in 2.8154 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -175.68, 166.03 APE9-dihe-na 96.38, 161.28 APE8-dihe-in -70.8, 121.46 APE8-rot-in 315.06 APE67-dihe-in -64.05, -14.0 -35.32, -45.01 APE12-dist-in 8.2423 APE11-dist-in 11.0778 APE10-dist-in 6.1501 APE9-dist-in 4.8506 None TPO198,SEP339 TPO198,CME200,SEP339 XRAY 2.9 0.257 0.291 A 350.0 332.0 0 25 25 0 [[44, 298]] 1.0 1j3h Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1J3HB P05132 12 351 351.0 No_ligand No_ligand None DFGin 6.9618 16.3184 BLAminus -127.51, 166.45 66.18, 90.08 -100.98, 29.78 267.08, 73.82 -52.31, -60.95 out-none out 10.1864 Saltbr-none 999.0 HRD-in -67.73, -45.7 38.54, 48.86 none-in-in SNCnii in-in ActLoopNT-in 2.811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.43, 169.92 APE9-dihe-na 94.29, 160.8 APE8-dihe-in -70.42, 119.44 APE8-rot-in 315.91 APE67-dihe-in -66.01, -15.04 -33.81, -42.66 APE12-dist-in 8.2628 APE11-dist-in 11.2131 APE10-dist-in 6.1679 APE9-dist-in 4.844 None TPO198,SEP339 TPO198,CME200,SEP339 XRAY 2.9 0.257 0.291 B 350.0 330.0 0 25 25 0 [[44, 298]] 1.0 1j3h Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2QVSE P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1963 14.9955 BLAminus -125.26, 166.13 66.05, 91.61 -98.74, 33.08 286.99, 64.22 -54.01, -35.46 out-none out 10.2631 Saltbr-none 999.0 HRD-in -74.03, -56.5 67.93, 15.74 none-in-in SNCnii in-in ActLoopNT-in 2.9976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.49, 163.74 APE9-dihe-na 132.78, -148.47 APE8-dihe-in -122.84, 132.55 APE8-rot-in 302.63 APE67-dihe-in -52.83, -31.96 -33.3, -62.56 APE12-dist-in 7.8939 APE11-dist-in 11.5512 APE10-dist-in 6.03 APE9-dist-in 3.5577 None TPO198,SEP339 TPO198,SEP339 XRAY 2.5 0.212 0.251 E 350.0 325.0 0 25 25 0 [[44, 298]] 1.0 2qvs Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4QD P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1967 14.9965 BLAminus -125.26, 166.14 66.1, 91.56 -98.68, 33.07 286.99, 61.83 -54.01, -35.41 out-none out 10.2635 Saltbr-none 999.0 HRD-in -74.09, -56.53 67.97, 15.71 none-in-in SNCnii in-in ActLoopNT-in 2.9982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 163.78 APE9-dihe-na 132.71, -148.52 APE8-dihe-in -122.82, 132.51 APE8-rot-in 302.65 APE67-dihe-in -52.8, -31.95 -33.23, -62.65 APE12-dist-in 7.9212 APE11-dist-in 11.55 APE10-dist-in 6.0293 APE9-dist-in 3.5583 None None None EM 35.0 999.0 999.0 D 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4q Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4QE P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1966 14.995 BLAminus -125.26, 166.1 66.04, 91.65 -98.75, 33.06 286.98, 61.89 -53.93, -35.48 out-none out 10.2634 Saltbr-none 999.0 HRD-in -73.99, -56.54 67.98, 15.68 none-in-in SNCnii in-in ActLoopNT-in 2.9973 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.48, 163.78 APE9-dihe-na 132.74, -148.47 APE8-dihe-in -122.8, 132.56 APE8-rot-in 302.67 APE67-dihe-in -52.81, -31.94 -33.33, -62.57 APE12-dist-in 7.922 APE11-dist-in 11.5519 APE10-dist-in 6.0305 APE9-dist-in 3.5582 None None None EM 35.0 999.0 999.0 E 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4q Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4RD P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1972 14.9967 BLAminus -125.31, 166.2 66.04, 91.6 -98.77, 33.16 286.98, 61.82 -54.08, -35.39 out-none out 10.2636 Saltbr-none 999.0 HRD-in -74.03, -56.49 67.97, 15.67 none-in-in SNCnii in-in ActLoopNT-in 2.998 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.51, 163.71 APE9-dihe-na 132.78, -148.41 APE8-dihe-in -122.89, 132.55 APE8-rot-in 302.65 APE67-dihe-in -52.76, -32.01 -33.29, -62.61 APE12-dist-in 7.9206 APE11-dist-in 11.55 APE10-dist-in 6.0293 APE9-dist-in 3.5577 None None None EM 35.0 999.0 999.0 D 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4RE P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1967 14.9951 BLAminus -125.22, 166.12 66.01, 91.59 -98.73, 33.13 286.98, 61.85 -53.97, -35.5 out-none out 10.2637 Saltbr-none 999.0 HRD-in -74.05, -56.46 67.95, 15.66 none-in-in SNCnii in-in ActLoopNT-in 2.9978 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 163.74 APE9-dihe-na 132.8, -148.42 APE8-dihe-in -122.89, 132.51 APE8-rot-in 302.64 APE67-dihe-in -52.86, -31.95 -33.27, -62.57 APE12-dist-in 7.9226 APE11-dist-in 11.5509 APE10-dist-in 6.0296 APE9-dist-in 3.5575 None None None EM 35.0 999.0 999.0 E 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2QURA P05132 12 351 351.0 No_ligand No_ligand None DFGin 6.5556 14.5504 BLAminus -137.47, -167.05 53.68, 73.35 -97.68, 23.63 275.03, 65.42 -50.82, -37.16 in-none in 9.0785 Saltbr-none 999.0 HRD-in -62.2, -51.82 63.3, 0.36 none-in-in SNCnii in-in ActLoopNT-in 2.9356 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.83, 151.09 APE9-dihe-na 135.53, -158.17 APE8-dihe-in -121.8, 126.63 APE8-rot-in 312.25 APE67-dihe-in -60.67, -15.51 -24.4, -62.49 APE12-dist-in 8.1463 APE11-dist-in 11.1283 APE10-dist-in 5.5314 APE9-dist-in 3.2085 K286P,F328A TPO198,SEP339 TPO198,SEP339 XRAY 2.5 0.212 0.265 A 350.0 340.0 0 25 25 0 [[44, 298]] 1.0 2qur Mus musculus AGC_PRKACA_MOUSE AGC 2.3e-94 321.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_RAT 3TNQB P27791 18 351 351.0 ADP:60400 ATPlike Inactive DFGin 6.0256 14.1092 ABAminus -114.77, -42.68 -116.73, 98.61 -86.63, 16.07 279.08, 57.74 -59.27, -13.09 in-in in 8.7647 Saltbr-in 3.2951 HRD-in -83.62, -53.15 67.05, 14.07 in-in-in SNCiii in-in ActLoopNT-in 3.0146 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.54, 167.18 APE9-dihe-na 139.44, -131.54 APE8-dihe-in -144.99, 127.08 APE8-rot-in 312.05 APE67-dihe-in -55.59, -13.34 -44.48, -54.97 APE12-dist-in 8.0951 APE11-dist-in 11.4567 APE10-dist-in 6.1812 APE9-dist-in 3.5888 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 3.097 0.234 0.275 B 350.0 334.0 0 25 25 0 [[44, 298]] 1.0 3tnq Rattus norvegicus AGC_PRKACA_RAT AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CDKA P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.8431 14.3299 BLAminus -113.76, -166.2 47.38, 80.03 -85.76, 16.06 278.85, 56.4 -55.46, -28.11 in-in in 9.0339 Saltbr-in 2.8992 HRD-in -94.66, -56.81 78.16, -3.52 in-in-in SNCiii in-in ActLoopNT-in 2.9853 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.51, 155.2 APE9-dihe-na 137.51, -153.75 APE8-dihe-in -125.49, 136.2 APE8-rot-in 297.83 APE67-dihe-in -73.46, -24.38 -35.73, -51.43 APE12-dist-in 7.9972 APE11-dist-in 11.4183 APE10-dist-in 5.7664 APE9-dist-in 3.6421 None TPO198 TPO198 XRAY 2.0 0.197 999.0 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CDKB P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.907 14.5106 BLAminus -124.27, -171.72 50.82, 76.29 -83.58, 17.26 280.88, 62.25 -47.74, -29.83 in-in in 8.889 Saltbr-in 2.8833 HRD-in -87.48, -57.48 77.49, 1.67 in-in-in SNCiii in-in ActLoopNT-in 2.9631 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 159.84 APE9-dihe-na 137.3, -140.74 APE8-dihe-in -136.57, 132.27 APE8-rot-in 304.84 APE67-dihe-in -69.16, -27.96 -34.59, -53.92 APE12-dist-in 8.3483 APE11-dist-in 11.5142 APE10-dist-in 6.0801 APE9-dist-in 3.7441 None TPO198 TPO198 XRAY 2.0 0.197 999.0 B 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CTPE P36887 8 351 351.0 No_ligand No_ligand Inactive DFGin 6.725 16.055 BLAminus -116.62, 169.7 58.2, 106.1 -115.39, 26.05 266.95, 79.04 -73.93, 13.07 in-out in 9.9631 Saltbr-out 3.6616 HRD-out -67.85, 127.4 -110.51, 32.03 out-in-in SNCoii in-in ActLoopNT-in 3.0743 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.53, 165.54 APE9-dihe-na 119.1, -162.75 APE8-dihe-in -95.5, 138.49 APE8-rot-in 313.62 APE67-dihe-in -63.93, -15.29 -42.58, -58.58 APE12-dist-in 8.6012 APE11-dist-in 11.5506 APE10-dist-in 6.2522 APE9-dist-in 3.8257 None TPO198 TPO198 XRAY 2.9 0.19 999.0 E 350.0 333.0 0 25 25 0 [[44, 298]] 1.0 1ctp Sus scrofa AGC_PRKACA_PIG AGC 3.3e-95 324.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CMKE P36887 2 351 351.0 No_ligand No_ligand Inactive DFGin 7.428 16.0445 BLAminus -105.57, 177.37 63.01, 79.23 -102.18, 28.14 277.96, 75.47 -76.23, -19.76 in-out in 9.8846 Saltbr-out 4.1251 HRD-in -61.54, -38.92 59.61, -1.33 out-in-in SNCoii in-in ActLoopNT-in 3.0635 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.53, 131.84 APE9-dihe-na 157.2, -155.98 APE8-dihe-in -96.86, 135.92 APE8-rot-in 291.44 APE67-dihe-in -53.19, -28.67 -38.32, -50.64 APE12-dist-in 8.1969 APE11-dist-in 11.2119 APE10-dist-in 5.6454 APE9-dist-in 3.8997 None TPO198,SEP339 TPO198,SEP339 XRAY 2.9 0.233 999.0 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1cmk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha

AGC_PRKACA (cAMP-dependent protein kinase catalytic subunit alpha)

Total number of chains: 372
Active chains: 237
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 293 78.8% 5N1FA
DFGin ABAminus 70 18.8% 5M6YA
None None 5 1.3% 9DW7G
DFGin None 4 1.1% 4C35A

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PRKACA KAPCA_BOVIN 9DW9G P00517 13 351 351.0 ATP:401 ATPlike Active DFGin 6.5695 15.1264 BLAminus -133.9, -169.96 59.46, 64.31 -83.85, 33.99 275.29, 73.58 -66.33, -24.36 in-in in 9.4988 Saltbr-in 3.2167 HRD-in -92.3, -53.34 68.25, 14.14 in-in-in SNCiii in-in ActLoopNT-in 3.0799 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.91, 151.76 APE9-dihe-na 126.66, -174.62 APE8-dihe-in -92.84, 130.69 APE8-rot-in 299.41 APE67-dihe-in -68.55, -23.13 -58.33, -34.44 APE12-dist-in 8.7033 APE11-dist-in 11.5632 APE10-dist-in 6.1702 APE9-dist-in 4.5677 None TPO198 TPO198 EM 2.8 999.0 999.0 G 351.0 328.0 0 25 25 0 [[44, 298]] 1.0 9dw9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q24A P00517 15 351 351.0 ATP:60400 ATPlike Active DFGin 5.9832 14.3195 BLAminus -113.95, 178.0 66.86, 85.15 -103.99, 32.82 274.7, 64.8 -65.44, -25.66 in-in in 8.779 Saltbr-in 2.742 HRD-in -93.22, -55.61 73.46, 14.95 in-in-in SNCiii in-in ActLoopNT-in 3.0897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.66, 162.77 APE9-dihe-na 133.15, -143.39 APE8-dihe-in -135.22, 127.61 APE8-rot-in 301.89 APE67-dihe-in -67.43, -30.61 -42.63, -46.05 APE12-dist-in 8.0357 APE11-dist-in 11.4473 APE10-dist-in 6.0235 APE9-dist-in 3.486 V124A,L174M TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.202 0.25 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1q24 Bos taurus AGC_PRKACA_BOVIN AGC 4.8e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO7A P00517 15 351 351.0 M05:61351,M05:61352 Allosteric,Type1 Active DFGin 6.0589 13.3545 BLAminus -112.73, 170.06 64.79, 125.13 -129.63, 24.75 288.96, 78.29 -59.84, -27.0 in-in in 8.9212 Saltbr-in 2.5901 HRD-in -91.38, -48.53 69.14, 8.91 in-in-in SNCiii in-in ActLoopNT-in 2.9119 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.06, 161.81 APE9-dihe-na 128.93, -157.64 APE8-dihe-in -120.9, 132.32 APE8-rot-in 302.18 APE67-dihe-in -59.27, -25.29 -43.22, -50.55 APE12-dist-in 8.1025 APE11-dist-in 11.3217 APE10-dist-in 5.7515 APE9-dist-in 3.6251 None TPO198,SEP339 TPO198,SEP339 XRAY 1.98 0.191 0.241 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vo7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNGA P00517 11 351 351.0 No_ligand No_ligand Active DFGin 6.1399 14.2236 BLAminus -119.55, 178.04 62.47, 98.55 -111.03, 25.12 275.63, 67.2 -58.48, -24.65 in-in in 9.0055 Saltbr-in 2.6957 HRD-in -96.2, -52.02 73.83, 11.43 in-in-in SNCiii in-in ActLoopNT-in 2.9239 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.01, 159.86 APE9-dihe-na 129.89, -160.93 APE8-dihe-in -123.36, 138.18 APE8-rot-in 302.01 APE67-dihe-in -59.18, -22.88 -47.61, -51.91 APE12-dist-in 8.0125 APE11-dist-in 11.2898 APE10-dist-in 5.8022 APE9-dist-in 3.5598 L50I,V124M,E128D,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.87 0.198 0.258 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gng Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GFCA P00517 15 351 351.0 No_ligand No_ligand Active DFGin 6.1877 14.0711 BLAminus -117.74, 159.24 72.69, 98.85 -105.34, 28.02 271.26, 59.63 -61.26, -23.71 in-in in 8.6743 Saltbr-in 2.5762 HRD-in -90.3, -52.85 73.44, 9.78 in-in-in SNCiii in-in ActLoopNT-in 2.9736 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.8, 159.7 APE9-dihe-na 133.98, -157.58 APE8-dihe-in -121.29, 135.51 APE8-rot-in 301.46 APE67-dihe-in -58.17, -22.85 -42.97, -54.07 APE12-dist-in 8.0335 APE11-dist-in 11.2552 APE10-dist-in 5.7258 APE9-dist-in 3.5267 None TPO198,SEP339 TPO198,SEP339 XRAY 1.87 0.239 0.239 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 2gfc Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q61A P00517 15 351 351.0 No_ligand No_ligand Active DFGin 6.3166 14.0576 BLAminus -113.32, 171.66 65.32, 95.24 -105.6, 28.35 273.54, 62.22 -60.93, -24.2 in-in in 8.7701 Saltbr-in 2.7918 HRD-in -88.4, -55.05 70.66, 3.99 in-in-in SNCiii in-in ActLoopNT-in 2.7864 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.36, 157.96 APE9-dihe-na 134.42, -161.14 APE8-dihe-in -115.93, 129.95 APE8-rot-in 300.39 APE67-dihe-in -58.76, -26.29 -47.87, -46.79 APE12-dist-in 8.1766 APE11-dist-in 11.5728 APE10-dist-in 6.0171 APE9-dist-in 3.7962 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.184 0.232 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1q61 Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SMHA P00517 2 351 351.0 No_ligand No_ligand Active DFGin 6.7989 14.5799 BLAminus -115.56, -165.58 57.6, 64.56 -89.23, 16.63 272.25, 75.82 -57.78, -31.17 in-in in 8.8477 Saltbr-in 2.4417 HRD-in -96.56, -52.48 70.28, 5.31 in-in-in SNCiii in-in ActLoopNT-in 2.7976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.7, 159.43 APE9-dihe-na 133.86, -177.98 APE8-dihe-in -99.8, 130.8 APE8-rot-in 299.09 APE67-dihe-in -59.18, -25.63 -42.57, -53.75 APE12-dist-in 8.2039 APE11-dist-in 11.557 APE10-dist-in 6.0526 APE9-dist-in 3.7586 Q85E,V124A,L174M,F188L TPO198,SEP339 TPO198,SEP339 XRAY 2.044 0.191 0.238 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1smh Bos taurus AGC_PRKACA_BOVIN AGC 3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q62A P00517 14 351 351.0 No_ligand No_ligand Active DFGin 6.1823 14.2767 BLAminus -104.64, 174.54 66.86, 89.86 -104.82, 25.62 276.34, 54.84 -53.41, -25.33 in-in in 8.9311 Saltbr-in 2.6139 HRD-in -96.79, -53.25 66.13, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.8834 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.96, 166.05 APE9-dihe-na 130.72, -161.89 APE8-dihe-in -113.23, 133.18 APE8-rot-in 300.81 APE67-dihe-in -67.6, -24.51 -42.5, -46.58 APE12-dist-in 8.1409 APE11-dist-in 11.4273 APE10-dist-in 6.0155 APE9-dist-in 3.617 V124A,L174M TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.192 0.252 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1q62 Bos taurus AGC_PRKACA_BOVIN AGC 4.8e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C33A P00517 14 351 351.0 No_ligand No_ligand Active DFGin 6.3698 14.4633 BLAminus -122.61, 167.1 69.2, 93.31 -104.18, 28.64 273.24, 55.76 -56.02, -28.41 in-in in 8.8225 Saltbr-in 2.7134 HRD-in -80.43, -53.85 71.22, 13.56 in-in-in SNCiii in-in ActLoopNT-in 2.937 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.13, 162.95 APE9-dihe-na 124.44, -159.48 APE8-dihe-in -120.39, 137.89 APE8-rot-in 301.42 APE67-dihe-in -62.3, -24.0 -46.94, -49.76 APE12-dist-in 8.0022 APE11-dist-in 11.3971 APE10-dist-in 5.7782 APE9-dist-in 3.4384 F55Y,M121L,V124L,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.158 0.187 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4c33 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNFA P00517 11 351 351.0 Y27:60501 Type1 Active DFGin 6.0407 14.1738 BLAminus -116.96, 178.88 58.65, 105.43 -113.78, 28.7 272.88, 66.05 -63.78, -25.92 in-in in 9.2018 Saltbr-in 2.5932 HRD-in -94.14, -47.78 64.37, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.8822 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -171.34, 163.17 APE9-dihe-na 124.68, -165.19 APE8-dihe-in -121.59, 134.6 APE8-rot-in 288.13 APE67-dihe-in -58.1, -28.51 -44.73, -50.81 APE12-dist-in 8.0234 APE11-dist-in 11.2036 APE10-dist-in 5.8077 APE9-dist-in 3.4001 L50I,V124M,E128D,Q182K,T184A TPO198,SEP339 TPO198,SEP339 XRAY 2.28 0.201 0.258 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gnf Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNJA P00517 15 351 351.0 Y27:60501 Type1 Active DFGin 6.1039 13.6767 BLAminus -125.2, 164.0 75.11, 93.42 -104.04, 27.11 286.53, 71.0 -58.19, -29.08 in-in in 9.0921 Saltbr-in 2.8299 HRD-in -86.57, -53.41 73.77, 21.07 in-in-in SNCiii in-in ActLoopNT-in 2.7763 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.71, 163.04 APE9-dihe-na 124.17, -165.73 APE8-dihe-in -116.96, 135.69 APE8-rot-in 293.77 APE67-dihe-in -62.53, -24.27 -43.03, -48.93 APE12-dist-in 8.108 APE11-dist-in 11.3187 APE10-dist-in 5.7869 APE9-dist-in 3.4239 L50I,Q182K,T184A TPO198,SEP339 TPO198,SEP339 XRAY 2.28 0.19 0.262 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 2gnj Bos taurus AGC_PRKACA_BOVIN AGC 7.3e-95 323.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNLA P00517 12 351 351.0 H52:60501 Type1 Active DFGin 6.3581 14.8769 BLAminus -89.02, -175.74 47.17, 112.42 -122.51, 26.46 259.73, 63.8 -65.5, -20.97 in-in in 9.1821 Saltbr-in 2.6049 HRD-in -84.16, -63.35 83.4, 16.15 in-in-in SNCiii in-in ActLoopNT-in 2.8748 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.63, 164.56 APE9-dihe-na 121.8, -158.16 APE8-dihe-in -125.31, 137.52 APE8-rot-in 295.72 APE67-dihe-in -52.7, -17.18 -53.68, -49.84 APE12-dist-in 8.1164 APE11-dist-in 11.5217 APE10-dist-in 6.1495 APE9-dist-in 3.5167 L50I,Q182K,T184A TPO198,SEP339 TPO198,SEP339 XRAY 2.6 0.203 0.303 A 350.0 340.0 0 25 25 0 [[44, 298]] 1.0 2gnl Bos taurus AGC_PRKACA_BOVIN AGC 7.3e-95 323.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZTA P00517 16 351 351.0 SS3:61351 Type1 Active DFGin 6.8713 14.0778 BLAminus -126.85, 167.46 69.43, 90.19 -103.99, 29.38 280.49, 66.47 -59.79, -22.48 in-in in 9.1397 Saltbr-in 2.6911 HRD-in -77.75, -50.42 62.52, 13.49 in-in-in SNCiii in-in ActLoopNT-in 2.9856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -114.56, 156.36 APE9-dihe-na 116.01, -154.02 APE8-dihe-in -130.0, 127.43 APE8-rot-in 298.59 APE67-dihe-in -60.13, -24.22 -31.54, -56.49 APE12-dist-in 7.8297 APE11-dist-in 11.3914 APE10-dist-in 5.7844 APE9-dist-in 3.7237 None None None XRAY 2.1 0.273 0.313 A 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzt Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZUE P00517 16 351 351.0 L20:61351 Type1 Active DFGin 6.5165 14.3927 BLAminus -116.34, 172.4 61.54, 100.04 -109.49, 24.05 269.56, 56.18 -51.88, -19.43 in-in in 8.8645 Saltbr-in 2.5717 HRD-in -79.6, -53.73 68.74, 6.41 in-in-in SNCiii in-in ActLoopNT-in 3.0336 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.25, 159.94 APE9-dihe-na 132.5, -155.2 APE8-dihe-in -127.84, 130.66 APE8-rot-in 306.17 APE67-dihe-in -52.51, -26.75 -31.49, -67.12 APE12-dist-in 7.8584 APE11-dist-in 11.1723 APE10-dist-in 5.7612 APE9-dist-in 3.7464 None None None XRAY 2.4 0.318 0.371 E 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzu Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZVA P00517 16 351 351.0 SS5:61351 Type1 Active DFGin 6.7937 14.3133 BLAminus -133.61, 167.29 69.98, 107.83 -122.87, 25.1 278.16, 55.22 -54.77, -25.94 in-in in 9.0833 Saltbr-in 2.6706 HRD-in -77.51, -58.55 72.39, 6.58 in-in-in SNCiii in-in ActLoopNT-in 3.1559 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.23, 161.95 APE9-dihe-na 131.29, -149.51 APE8-dihe-in -126.03, 139.69 APE8-rot-in 311.31 APE67-dihe-in -45.96, -25.35 -39.61, -69.13 APE12-dist-in 7.7834 APE11-dist-in 11.1969 APE10-dist-in 5.8374 APE9-dist-in 3.677 None None None XRAY 2.5 0.251 0.316 A 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzv Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UZWE P00517 16 351 351.0 SS4:61351 Type1 Active DFGin 6.5613 14.5744 BLAminus -112.04, -173.28 55.73, 87.87 -110.12, 39.6 275.39, 62.8 -71.34, -18.15 in-in in 8.8979 Saltbr-in 3.1279 HRD-in -78.88, -49.67 62.72, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.7912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.16, 162.59 APE9-dihe-na 103.28, -160.9 APE8-dihe-in -116.22, 129.17 APE8-rot-in 310.0 APE67-dihe-in -56.35, -23.35 -31.72, -57.46 APE12-dist-in 8.0868 APE11-dist-in 11.3531 APE10-dist-in 5.8387 APE9-dist-in 3.776 None None None XRAY 2.2 0.313 0.328 E 336.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uzw Bos taurus AGC_PRKACA_BOVIN AGC 1.2e-94 322.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q8TA P00517 11 351 351.0 Y27:60930 Type1 Active DFGin 6.1851 14.3139 BLAminus -117.96, 176.23 66.27, 91.07 -99.92, 24.26 275.29, 66.15 -60.05, -23.97 in-in in 9.0544 Saltbr-in 2.5891 HRD-in -93.15, -51.44 72.41, 0.56 in-in-in SNCiii in-in ActLoopNT-in 2.9525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.6, 160.94 APE9-dihe-na 131.1, -162.98 APE8-dihe-in -114.15, 135.68 APE8-rot-in 299.16 APE67-dihe-in -56.85, -26.83 -51.6, -49.02 APE12-dist-in 8.1774 APE11-dist-in 11.4755 APE10-dist-in 5.9128 APE9-dist-in 3.6886 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.182 0.229 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1q8t Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q8WA P00517 15 351 351.0 M77:60960 Type1 Active DFGin 6.5158 14.6907 BLAminus -127.81, 164.07 85.37, 88.74 -113.2, 23.58 288.03, 80.25 -50.72, -40.77 in-in in 8.8645 Saltbr-in 2.7877 HRD-in -88.09, -59.12 85.64, -3.61 in-in-in SNCiii in-in ActLoopNT-in 3.125 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.12, 157.94 APE9-dihe-na 118.72, -168.38 APE8-dihe-in -118.75, 133.72 APE8-rot-in 300.62 APE67-dihe-in -62.19, -20.35 -49.36, -50.33 APE12-dist-in 8.427 APE11-dist-in 11.7879 APE10-dist-in 6.3999 APE9-dist-in 4.0603 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.22 0.295 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1q8w Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SVEA P00517 8 351 351.0 I01:60351 Type1 Active DFGin 6.1664 14.2222 BLAminus -113.6, -176.53 62.78, 78.1 -100.84, 17.81 278.73, 68.66 -48.01, -28.95 in-in in 8.6662 Saltbr-in 2.5697 HRD-in -91.7, -56.06 76.75, 8.37 in-in-in SNCiii in-in ActLoopNT-in 3.0657 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.08, 161.63 APE9-dihe-na 125.64, -173.88 APE8-dihe-in -102.65, 133.23 APE8-rot-in 299.26 APE67-dihe-in -60.18, -26.54 -47.49, -48.66 APE12-dist-in 8.1227 APE11-dist-in 11.4552 APE10-dist-in 5.942 APE9-dist-in 3.5408 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.49 0.202 0.257 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 1sve Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SVGA P00517 11 351 351.0 I04:60351 Type1 Active DFGin 6.2852 14.1972 BLAminus -126.54, 177.16 64.26, 73.95 -91.56, 21.32 279.08, 73.3 -61.43, -19.1 in-in in 8.5805 Saltbr-in 2.6809 HRD-in -92.74, -53.98 73.19, 8.88 in-in-in SNCiii in-in ActLoopNT-in 2.9341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.17, 160.9 APE9-dihe-na 123.57, -169.23 APE8-dihe-in -108.56, 130.67 APE8-rot-in 293.73 APE67-dihe-in -66.93, -24.48 -43.76, -46.84 APE12-dist-in 8.0906 APE11-dist-in 11.5393 APE10-dist-in 6.0517 APE9-dist-in 3.6478 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.02 0.183 0.227 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1svg Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1VEBA P00517 11 351 351.0 I05:60351 Type1 Active DFGin 6.2131 14.2357 BLAminus -112.2, -169.65 49.77, 80.02 -102.5, 31.57 278.86, 61.26 -72.56, -20.75 in-in in 8.5766 Saltbr-in 2.8728 HRD-in -83.01, -49.6 62.13, 5.25 in-in-in SNCiii in-in ActLoopNT-in 3.0408 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.53, 158.22 APE9-dihe-na 134.18, -167.65 APE8-dihe-in -109.96, 136.58 APE8-rot-in 290.96 APE67-dihe-in -71.75, -2.37 -42.82, -49.75 APE12-dist-in 8.1776 APE11-dist-in 11.6793 APE10-dist-in 6.0598 APE9-dist-in 3.7367 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.89 0.187 0.251 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1veb Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH4A P00517 15 351 351.0 R69:60351 Type1 Active DFGin 6.2972 13.619 BLAminus -125.63, 176.59 60.0, 74.66 -89.7, 21.14 287.64, 81.0 -57.7, -30.21 in-in in 8.7553 Saltbr-in 2.5701 HRD-in -85.89, -55.59 71.5, 15.27 in-in-in SNCiii in-in ActLoopNT-in 3.0669 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.1, 158.39 APE9-dihe-na 135.4, -175.25 APE8-dihe-in -99.1, 130.32 APE8-rot-in 300.14 APE67-dihe-in -53.15, -30.05 -47.58, -48.79 APE12-dist-in 8.1288 APE11-dist-in 11.5852 APE10-dist-in 6.0366 APE9-dist-in 3.7183 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.45 0.191 0.242 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1xh4 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH5A P00517 15 351 351.0 R68:61001 Type1 Active DFGin 6.3947 13.2316 BLAminus -125.11, 175.33 63.85, 75.87 -93.6, 21.14 294.45, 75.91 -54.91, -25.56 in-in in 8.7353 Saltbr-in 2.7377 HRD-in -92.22, -50.1 68.22, 14.89 in-in-in SNCiii in-in ActLoopNT-in 2.9658 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.82, 159.18 APE9-dihe-na 129.26, -172.93 APE8-dihe-in -106.77, 134.87 APE8-rot-in 299.04 APE67-dihe-in -60.66, -25.82 -46.87, -48.0 APE12-dist-in 7.9509 APE11-dist-in 11.4133 APE10-dist-in 5.881 APE9-dist-in 3.5909 None TPO198,SEP339 TPO198,SEP339 XRAY 2.05 0.185 0.236 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1xh5 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH6A P00517 19 351 351.0 R94:60351 Type1 Active DFGin 6.1276 13.3787 BLAminus -130.28, 176.51 62.64, 74.17 -91.5, 20.79 288.12, 76.57 -51.25, -30.79 in-in in 8.8185 Saltbr-in 2.708 HRD-in -82.23, -52.65 67.28, 14.23 in-in-in SNCiii in-in ActLoopNT-in 3.0713 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.94, 161.1 APE9-dihe-na 129.62, -161.03 APE8-dihe-in -117.21, 135.0 APE8-rot-in 298.01 APE67-dihe-in -59.91, -22.98 -46.35, -48.26 APE12-dist-in 8.104 APE11-dist-in 11.5006 APE10-dist-in 5.9059 APE9-dist-in 3.4893 None TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.192 0.249 A 350.0 333.0 0 25 25 0 [[44, 298]] 1.0 1xh6 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH7A P00517 11 351 351.0 R96:60351 Type1 Active DFGin 6.3831 13.3018 BLAminus -121.57, 176.46 64.46, 76.56 -95.28, 25.2 293.04, 73.78 -55.65, -33.0 in-in in 8.6628 Saltbr-in 2.6788 HRD-in -88.46, -51.77 72.39, 6.4 in-in-in SNCiii in-in ActLoopNT-in 2.9193 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.76, 163.97 APE9-dihe-na 129.5, -170.45 APE8-dihe-in -100.96, 130.84 APE8-rot-in 305.54 APE67-dihe-in -56.25, -25.46 -42.72, -53.32 APE12-dist-in 7.9889 APE11-dist-in 11.7106 APE10-dist-in 6.0439 APE9-dist-in 3.9196 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.47 0.192 0.254 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1xh7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH8A P00517 13 351 351.0 R55:60351 Type1 Active DFGin 7.2199 14.5512 BLAminus -127.78, 170.11 66.78, 76.25 -93.48, 35.64 282.0, 79.13 -69.55, -13.04 in-in in 8.6647 Saltbr-in 2.5851 HRD-in -73.67, -49.45 69.2, 1.69 in-in-in SNCiii in-in ActLoopNT-in 2.9223 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.86, 150.19 APE9-dihe-na 125.99, -169.91 APE8-dihe-in -111.55, 132.51 APE8-rot-in 296.34 APE67-dihe-in -62.89, -22.39 -42.71, -52.56 APE12-dist-in 8.7908 APE11-dist-in 11.805 APE10-dist-in 6.255 APE9-dist-in 3.5116 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.202 0.236 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1xh8 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3KKVA P00517 14 351 351.0 B99:60351 Type1 Active DFGin 6.2802 14.9874 BLAminus -125.37, 172.94 64.41, 88.24 -101.41, 28.77 274.35, 61.51 -57.52, -30.45 in-in in 9.39 Saltbr-in 2.668 HRD-in -87.09, -58.29 72.04, 20.78 in-in-in SNCiii in-in ActLoopNT-in 2.9138 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.6, 161.14 APE9-dihe-na 126.5, -157.51 APE8-dihe-in -121.76, 131.58 APE8-rot-in 301.24 APE67-dihe-in -59.26, -23.73 -39.89, -55.55 APE12-dist-in 7.9861 APE11-dist-in 11.2507 APE10-dist-in 5.7729 APE9-dist-in 3.4844 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.8 0.203 0.225 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3kkv Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4IJ9A P00517 15 351 351.0 PTV:60401 Type1 Active DFGin 6.6148 14.131 BLAminus -111.94, -175.65 58.73, 79.19 -93.36, 11.75 269.03, 67.58 -54.32, -24.02 in-in in 8.8666 Saltbr-in 3.4017 HRD-in -79.91, -51.1 66.03, 1.36 in-in-in SNCiii in-in ActLoopNT-in 2.9049 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.66, 160.33 APE9-dihe-na 124.74, -169.36 APE8-dihe-in -102.85, 129.95 APE8-rot-in 307.44 APE67-dihe-in -60.51, -31.49 -37.15, -49.85 APE12-dist-in 8.2305 APE11-dist-in 11.4808 APE10-dist-in 5.8096 APE9-dist-in 3.3378 None TPO198,SEP339 TPO198,SEP339 XRAY 2.55 0.175 0.247 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4ij9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2C1AA P00517 15 351 351.0 I5S:61351 Type1 Active DFGin 6.2978 14.6265 BLAminus -124.46, -169.61 66.48, 66.45 -85.13, 21.14 273.21, 64.57 -65.03, -22.49 in-in in 9.003 Saltbr-in 2.6116 HRD-in -90.18, -53.0 74.43, 14.23 in-in-in SNCiii in-in ActLoopNT-in 2.9703 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.63, 158.7 APE9-dihe-na 138.5, -149.83 APE8-dihe-in -130.06, 134.27 APE8-rot-in 299.96 APE67-dihe-in -59.41, -28.42 -45.36, -49.19 APE12-dist-in 7.8481 APE11-dist-in 11.246 APE10-dist-in 5.7402 APE9-dist-in 3.5606 None TPO198,SEP339 TPO198,SEP339 XRAY 1.95 0.176 0.23 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2c1a Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2C1BA P00517 15 351 351.0 CQP:61351 Type1 Active DFGin 6.0179 14.5756 BLAminus -127.46, 168.13 73.41, 94.26 -102.97, 22.93 271.29, 59.53 -60.22, -28.98 in-in in 8.8601 Saltbr-in 2.6005 HRD-in -86.97, -55.45 75.34, 13.69 in-in-in SNCiii in-in ActLoopNT-in 2.9333 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.15, 165.93 APE9-dihe-na 130.88, -155.25 APE8-dihe-in -127.93, 130.25 APE8-rot-in 296.49 APE67-dihe-in -57.75, -24.32 -42.11, -51.87 APE12-dist-in 8.026 APE11-dist-in 11.266 APE10-dist-in 5.7202 APE9-dist-in 3.4692 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.162 0.211 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2c1b Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2F7EE P00517 16 351 351.0 2EA:60351 Type1 Active DFGin 6.4255 14.622 BLAminus -129.37, 172.24 65.85, 87.0 -103.27, 28.23 271.13, 52.64 -61.39, -20.95 in-in in 9.0188 Saltbr-in 2.5724 HRD-in -84.54, -55.3 68.58, 20.0 in-in-in SNCiii in-in ActLoopNT-in 3.0357 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.64, 149.46 APE9-dihe-na 134.17, -155.82 APE8-dihe-in -124.14, 133.58 APE8-rot-in 298.87 APE67-dihe-in -58.46, -26.82 -32.03, -63.88 APE12-dist-in 7.8441 APE11-dist-in 11.2456 APE10-dist-in 5.6686 APE9-dist-in 3.7407 None None None XRAY 2.0 0.283 0.323 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2f7e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2F7XE P00517 16 351 351.0 4EA:60351 Type1 Active DFGin 6.4787 14.4427 BLAminus -134.55, -177.23 60.89, 80.89 -96.41, 28.1 269.37, 55.24 -56.5, -28.29 in-in in 8.9136 Saltbr-in 2.4578 HRD-in -81.93, -53.89 61.67, 20.58 in-in-in SNCiii in-in ActLoopNT-in 2.989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.99, 155.02 APE9-dihe-na 135.32, -157.56 APE8-dihe-in -123.89, 130.78 APE8-rot-in 298.61 APE67-dihe-in -49.48, -26.89 -30.62, -70.43 APE12-dist-in 7.9799 APE11-dist-in 11.4061 APE10-dist-in 5.9418 APE9-dist-in 3.9333 None None None XRAY 1.9 0.268 0.297 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2f7x Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2F7ZE P00517 16 351 351.0 6EA:61000 Type1 Active DFGin 6.2259 13.9549 BLAminus -129.55, -167.66 49.24, 93.04 -110.0, 23.76 275.34, 53.4 -53.66, -28.22 in-in in 8.5633 Saltbr-in 3.0644 HRD-in -65.45, -44.81 59.73, 0.41 in-in-in SNCiii in-in ActLoopNT-in 2.9811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -169.37, 169.07 APE9-dihe-na 126.6, -164.29 APE8-dihe-in -104.93, 138.12 APE8-rot-in 285.38 APE67-dihe-in -37.82, -20.53 -38.18, -81.91 APE12-dist-in 7.8361 APE11-dist-in 11.3017 APE10-dist-in 6.2126 APE9-dist-in 3.7238 None None None XRAY 3.0 0.246 0.342 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2f7z Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2JDSA P00517 15 351 351.0 L20:61351 Type1 Active DFGin 6.2975 14.4588 BLAminus -119.85, 164.76 69.86, 95.65 -106.41, 24.64 270.02, 58.03 -63.42, -24.71 in-in in 8.8415 Saltbr-in 2.9556 HRD-in -93.07, -49.96 71.48, 12.63 in-in-in SNCiii in-in ActLoopNT-in 2.9911 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.76, 158.61 APE9-dihe-na 135.6, -151.18 APE8-dihe-in -131.14, 134.0 APE8-rot-in 299.22 APE67-dihe-in -56.34, -24.22 -43.06, -54.13 APE12-dist-in 7.9284 APE11-dist-in 11.2908 APE10-dist-in 5.7662 APE9-dist-in 3.5059 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.211 0.272 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2jds Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2OH0E P00517 16 351 351.0 2PY:60351 Type1 Active DFGin 6.5126 14.6531 BLAminus -127.37, 173.11 66.58, 90.68 -104.37, 27.73 269.87, 52.25 -56.81, -28.64 in-in in 8.9289 Saltbr-in 2.5821 HRD-in -77.86, -55.61 71.73, 4.87 in-in-in SNCiii in-in ActLoopNT-in 2.9184 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.82, 160.53 APE9-dihe-na 132.23, -161.93 APE8-dihe-in -120.81, 133.78 APE8-rot-in 295.17 APE67-dihe-in -53.8, -16.59 -31.38, -69.24 APE12-dist-in 7.8772 APE11-dist-in 11.1968 APE10-dist-in 5.8391 APE9-dist-in 3.6735 None None None XRAY 2.2 0.273 0.32 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2oh0 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2OJFE P00517 16 351 351.0 4PY:61000 Type1 Active DFGin 6.632 13.5749 BLAminus -129.09, 175.09 60.55, 94.36 -110.26, 30.25 290.83, 66.47 -61.76, -22.5 in-in in 8.9951 Saltbr-in 2.6975 HRD-in -83.69, -49.78 65.87, 9.9 in-in-in SNCiii in-in ActLoopNT-in 2.9369 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.63, 160.13 APE9-dihe-na 129.42, -154.83 APE8-dihe-in -123.4, 138.68 APE8-rot-in 295.74 APE67-dihe-in -57.43, -25.96 -38.07, -61.94 APE12-dist-in 7.9119 APE11-dist-in 11.2719 APE10-dist-in 5.8536 APE9-dist-in 3.6707 None None None XRAY 2.1 0.265 0.29 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2ojf Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3AG9B P00517 16 351 351.0 A02:60351 Type1 Active DFGin 6.7069 14.8178 BLAminus -118.08, 165.29 66.01, 91.25 -100.52, 22.8 270.89, 66.31 -51.41, -38.23 in-in in 9.1095 Saltbr-in 2.7494 HRD-in -86.2, -49.67 71.39, 4.04 in-in-in SNCiii in-in ActLoopNT-in 2.8575 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.38, 133.7 APE9-dihe-na 131.92, -165.0 APE8-dihe-in -83.45, 116.32 APE8-rot-in 314.25 APE67-dihe-in -59.66, -23.97 -46.78, -44.32 APE12-dist-in 8.1703 APE11-dist-in 11.9191 APE10-dist-in 6.8174 APE9-dist-in 5.6216 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.23 0.246 B 351.0 319.0 0 25 25 0 [[44, 298]] 1.0 3ag9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO1A P00517 10 351 351.0 SIJ:61351 Type1 Active DFGin 6.3414 14.0562 BLAminus -119.34, -177.25 63.83, 74.63 -95.99, 18.51 283.99, 75.88 -54.4, -29.22 in-in in 9.1037 Saltbr-in 2.6632 HRD-in -85.49, -49.19 68.51, 9.51 in-in-in SNCiii in-in ActLoopNT-in 2.9485 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.19, 161.74 APE9-dihe-na 124.38, -162.01 APE8-dihe-in -111.99, 135.74 APE8-rot-in 300.86 APE67-dihe-in -57.72, -23.86 -43.38, -54.21 APE12-dist-in 7.9994 APE11-dist-in 11.3701 APE10-dist-in 5.7652 APE9-dist-in 3.4439 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.162 0.19 A 351.0 342.0 0 25 25 0 [[44, 298]] 1.0 3zo1 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO4A P00517 15 351 351.0 QWI:61352 Type1 Active DFGin 5.971 14.4316 BLAminus -122.52, 179.4 62.97, 87.47 -105.16, 25.03 272.68, 69.84 -56.89, -28.47 in-in in 8.8067 Saltbr-in 2.6787 HRD-in -83.14, -51.38 69.84, 7.49 in-in-in SNCiii in-in ActLoopNT-in 2.9237 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.86, 163.63 APE9-dihe-na 121.61, -161.92 APE8-dihe-in -113.3, 134.36 APE8-rot-in 304.88 APE67-dihe-in -60.74, -25.7 -43.03, -50.51 APE12-dist-in 8.1783 APE11-dist-in 11.5104 APE10-dist-in 5.91 APE9-dist-in 3.4662 None TPO198,SEP339 TPO198,SEP339 XRAY 1.65 0.17 0.195 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 3zo4 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4IE9A P00517 15 351 351.0 PZX:60401 Type1 Active DFGin 6.4403 14.5717 BLAminus -120.62, 176.92 66.27, 86.77 -100.95, 18.69 270.67, 65.37 -56.43, -28.52 in-in in 8.9159 Saltbr-in 2.77 HRD-in -89.08, -49.96 64.8, 10.82 in-in-in SNCiii in-in ActLoopNT-in 2.9618 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.58, 154.28 APE9-dihe-na 136.57, -156.42 APE8-dihe-in -117.79, 131.56 APE8-rot-in 300.22 APE67-dihe-in -56.73, -26.63 -41.25, -54.98 APE12-dist-in 8.1769 APE11-dist-in 11.3836 APE10-dist-in 5.8183 APE9-dist-in 3.6635 None TPO198,SEP339 TPO198,SEP339 XRAY 1.92 0.18 0.232 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4ie9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 5VHBA P00517 19 351 351.0 9CY:60401 Type1 Active DFGin 5.8914 14.4101 BLAminus -119.66, -177.23 60.94, 80.11 -93.35, 23.41 272.21, 58.28 -59.14, -26.18 in-in in 9.0291 Saltbr-in 2.7119 HRD-in -91.92, -50.82 66.2, 13.96 in-in-in SNCiii in-in ActLoopNT-in 2.9438 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.84, 154.36 APE9-dihe-na 131.28, -165.28 APE8-dihe-in -112.93, 137.33 APE8-rot-in 299.96 APE67-dihe-in -60.22, -22.29 -46.36, -53.5 APE12-dist-in 7.9601 APE11-dist-in 11.4577 APE10-dist-in 5.827 APE9-dist-in 3.8655 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.61 0.178 0.204 A 351.0 328.0 0 25 25 0 [[44, 298]] 1.0 5vhb Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 6E99A P00517 19 351 351.0 J0G:60601 Type1 Active DFGin 6.0023 14.6887 BLAminus -119.91, 176.13 61.41, 87.48 -95.36, 20.23 270.62, 61.24 -51.17, -35.89 in-in in 9.2093 Saltbr-in 2.7738 HRD-in -83.71, -54.36 68.2, 17.2 in-in-in SNCiii in-in ActLoopNT-in 3.0278 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.66, 157.43 APE9-dihe-na 126.17, -162.46 APE8-dihe-in -111.15, 131.88 APE8-rot-in 301.0 APE67-dihe-in -61.67, -24.67 -45.52, -49.68 APE12-dist-in 8.1145 APE11-dist-in 11.6023 APE10-dist-in 5.8812 APE9-dist-in 3.7622 None TPO198,SEP339 TPO198,SEP339 XRAY 1.88 0.208 0.23 A 351.0 333.0 0 25 25 0 [[44, 298]] 1.0 6e99 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 6E9LA P00517 18 351 351.0 J0P:60401 Type1 Active DFGin 6.4992 14.4033 BLAminus -98.87, -153.44 32.95, 78.78 -89.6, 15.58 275.81, 59.68 -55.89, -23.51 in-in in 8.8735 Saltbr-in 2.7663 HRD-in -69.86, -50.02 57.75, 17.6 in-in-in SNCiii in-in ActLoopNT-in 3.0358 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.26, 159.36 APE9-dihe-na 132.47, -166.61 APE8-dihe-in -110.57, 132.03 APE8-rot-in 295.04 APE67-dihe-in -57.99, -24.14 -37.74, -55.31 APE12-dist-in 7.9954 APE11-dist-in 11.7663 APE10-dist-in 6.1939 APE9-dist-in 4.0725 None TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.198 0.271 A 351.0 334.0 0 25 25 0 [[44, 298]] 1.0 6e9l Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 8SF8A P00517 13 351 351.0 ZWG:60401 Type1 Active DFGin 6.2798 14.2539 BLAminus -129.1, 170.06 68.03, 97.5 -109.47, 25.84 272.72, 61.91 -63.1, -22.98 in-in in 8.7505 Saltbr-in 2.7564 HRD-in -95.34, -49.3 69.01, 11.41 in-in-in SNCiii in-in ActLoopNT-in 2.8647 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.49, 160.11 APE9-dihe-na 135.6, -161.4 APE8-dihe-in -120.07, 137.81 APE8-rot-in 299.35 APE67-dihe-in -59.91, -22.91 -50.11, -49.66 APE12-dist-in 8.0794 APE11-dist-in 11.2474 APE10-dist-in 5.82 APE9-dist-in 3.5329 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.199 0.22 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 8sf8 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3DNDA P00517 16 351 351.0 LL2:60351 Type1 Active DFGin 6.5437 14.6347 BLAminus -116.16, 171.46 66.82, 93.02 -101.85, 16.18 271.74, 55.59 -52.63, -24.52 in-in in 9.1859 Saltbr-in 2.9585 HRD-in -95.42, -56.13 76.88, 13.37 in-in-in SNCiii in-in ActLoopNT-in 2.8599 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.6, 159.85 APE9-dihe-na 129.5, -152.83 APE8-dihe-in -125.57, 136.21 APE8-rot-in 298.43 APE67-dihe-in -52.95, -28.96 -44.81, -53.93 APE12-dist-in 8.0597 APE11-dist-in 11.3778 APE10-dist-in 5.8234 APE9-dist-in 3.4374 None TPO198,SEP339 TPO198,SEP339 XRAY 2.26 0.19 0.253 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 3dnd Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3DNEA P00517 14 351 351.0 LL1:60351 Type1 Active DFGin 6.437 14.4585 BLAminus -121.1, -178.57 64.95, 70.37 -87.98, 19.34 273.67, 65.23 -66.31, -20.97 in-in in 8.8191 Saltbr-in 2.7351 HRD-in -96.15, -42.67 61.27, 10.37 in-in-in SNCiii in-in ActLoopNT-in 2.8642 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.64, 165.13 APE9-dihe-na 129.71, -157.6 APE8-dihe-in -124.5, 137.89 APE8-rot-in 294.27 APE67-dihe-in -60.97, -25.49 -45.94, -52.87 APE12-dist-in 8.0593 APE11-dist-in 11.1643 APE10-dist-in 5.7175 APE9-dist-in 3.5291 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.179 0.23 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3dne Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4YXRA P00517 16 351 351.0 0RW:60401 Type1 Active DFGin 6.0086 14.2951 BLAminus -119.04, 170.91 66.3, 93.05 -106.53, 24.67 276.07, 60.12 -58.07, -27.2 in-in in 9.0005 Saltbr-in 2.7007 HRD-in -82.28, -52.44 64.39, 8.26 in-in-in SNCiii in-in ActLoopNT-in 2.8702 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.51, 157.24 APE9-dihe-na 130.59, -154.35 APE8-dihe-in -122.35, 133.27 APE8-rot-in 301.51 APE67-dihe-in -58.69, -25.56 -33.6, -61.81 APE12-dist-in 8.0106 APE11-dist-in 11.3632 APE10-dist-in 5.8486 APE9-dist-in 3.6367 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 999.0 0.252 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4yxr Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4YXSA P00517 15 351 351.0 EMU:60401 Type1 Active DFGin 6.2857 13.5939 BLAminus -119.26, 168.5 67.4, 97.14 -108.4, 23.82 281.89, 73.4 -58.43, -25.53 in-in in 8.6608 Saltbr-in 2.6403 HRD-in -81.58, -52.24 65.52, 13.45 in-in-in SNCiii in-in ActLoopNT-in 2.9722 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.78, 159.45 APE9-dihe-na 131.68, -155.75 APE8-dihe-in -118.67, 131.09 APE8-rot-in 300.67 APE67-dihe-in -60.75, -29.57 -37.55, -53.5 APE12-dist-in 7.9379 APE11-dist-in 11.2743 APE10-dist-in 5.702 APE9-dist-in 3.6169 None TPO198,SEP339 TPO198,SEP339 XRAY 2.11 0.179 0.232 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4yxs Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1YDRE P00517 16 351 351.0 IQP:60351 Type1 Active DFGin 6.3291 14.2499 BLAminus -123.41, -178.28 58.45, 85.19 -101.97, 32.19 283.4, 54.35 -61.44, -27.25 in-in in 9.0495 Saltbr-in 2.7847 HRD-in -72.07, -64.76 83.06, 0.73 in-in-in SNCiii in-in ActLoopNT-in 2.8217 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.65, 168.03 APE9-dihe-na 116.01, -166.19 APE8-dihe-in -108.88, 132.42 APE8-rot-in 303.05 APE67-dihe-in -60.22, -26.51 -39.35, -52.68 APE12-dist-in 7.8706 APE11-dist-in 11.2981 APE10-dist-in 5.8958 APE9-dist-in 3.7525 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.188 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1ydr Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1YDSE P00517 16 351 351.0 IQS:60351 Type1 Active DFGin 6.3904 14.2877 BLAminus -112.84, -174.99 60.37, 74.83 -97.86, 29.16 279.73, 63.74 -63.98, -20.15 in-in in 8.9368 Saltbr-in 2.7755 HRD-in -75.45, -57.26 74.03, 4.96 in-in-in SNCiii in-in ActLoopNT-in 2.8322 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.17, 169.02 APE9-dihe-na 97.73, -165.42 APE8-dihe-in -112.69, 125.84 APE8-rot-in 302.88 APE67-dihe-in -57.81, -27.95 -31.43, -56.99 APE12-dist-in 7.9405 APE11-dist-in 11.1848 APE10-dist-in 5.7383 APE9-dist-in 3.6085 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.199 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1yds Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1YDTE P00517 16 351 351.0 IQB:60351 Type1 Active DFGin 6.5625 14.5739 BLAminus -112.01, -173.33 55.77, 87.81 -110.08, 39.59 275.46, 62.76 -71.4, -18.08 in-in in 8.8978 Saltbr-in 3.1275 HRD-in -78.94, -49.64 62.76, 12.37 in-in-in SNCiii in-in ActLoopNT-in 2.7915 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.17, 162.58 APE9-dihe-na 103.22, -160.88 APE8-dihe-in -116.29, 129.25 APE8-rot-in 310.0 APE67-dihe-in -56.34, -23.41 -31.82, -57.38 APE12-dist-in 8.0876 APE11-dist-in 11.3528 APE10-dist-in 5.8378 APE9-dist-in 3.7764 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.194 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1ydt Bos taurus AGC_PRKACA_BOVIN AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SZMA P00517 16 351 351.0 BI4:60351 Type1 Active DFGin 6.3181 15.3683 BLAminus -125.27, 171.81 65.17, 99.61 -108.03, 19.56 272.67, 80.44 -58.01, -35.62 in-in in 9.4925 Saltbr-in 2.5743 HRD-in -86.5, -61.07 68.65, 7.7 in-in-in SNCiii in-in ActLoopNT-in 3.0034 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 163.31 APE9-dihe-na 107.11, 170.89 APE8-dihe-in -74.89, 129.09 APE8-rot-in 328.61 APE67-dihe-in -51.73, -30.1 -54.41, -49.2 APE12-dist-in 8.0399 APE11-dist-in 11.3302 APE10-dist-in 5.7626 APE9-dist-in 3.8064 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 A 350.0 320.0 0 25 25 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4Z84A P00517 15 351 351.0 NVX:60401 Type1 Active DFGin 6.1539 14.585 BLAminus -122.35, -175.47 64.09, 72.13 -88.27, 20.06 271.08, 58.42 -49.77, -31.82 in-in in 9.0164 Saltbr-in 2.7991 HRD-in -96.48, -53.57 76.53, 13.57 in-in-in SNCiii in-in ActLoopNT-in 2.9176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.06, 154.73 APE9-dihe-na 134.03, -158.23 APE8-dihe-in -120.28, 132.43 APE8-rot-in 300.75 APE67-dihe-in -53.91, -23.24 -46.29, -52.23 APE12-dist-in 8.1505 APE11-dist-in 11.5238 APE10-dist-in 5.9254 APE9-dist-in 3.5106 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.554 0.209 0.234 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4z84 Bos taurus AGC_PRKACA_BOVIN AGC 1.7e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XHAA P00517 2 351 351.0 R68:61001 Type1 Active DFGin 6.2641 14.1375 BLAminus -120.5, -174.91 64.53, 71.29 -89.72, 23.88 279.31, 73.73 -56.55, -38.89 in-in in 8.7371 Saltbr-in 2.545 HRD-in -89.15, -49.54 68.47, 12.55 in-in-in SNCiii in-in ActLoopNT-in 2.9376 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.3, 164.66 APE9-dihe-na 127.73, 179.02 APE8-dihe-in -85.45, 132.2 APE8-rot-in 302.59 APE67-dihe-in -55.5, -36.01 -41.3, -53.29 APE12-dist-in 8.4646 APE11-dist-in 11.7786 APE10-dist-in 6.157 APE9-dist-in 3.7469 Q85E,V124A,L174M,F188L TPO198,SEP339 TPO198,SEP339 XRAY 2.46 0.223 0.272 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1xha Bos taurus AGC_PRKACA_BOVIN AGC 3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2JDTA P00517 16 351 351.0 I5S:61351 Type1 Active DFGin 6.2483 14.4539 BLAminus -118.34, -171.87 56.8, 75.79 -95.64, 21.06 274.55, 57.92 -54.25, -28.4 in-in in 8.8407 Saltbr-in 2.7265 HRD-in -87.26, -55.39 77.73, 12.38 in-in-in SNCiii in-in ActLoopNT-in 2.9989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.35, 160.37 APE9-dihe-na 136.22, -156.91 APE8-dihe-in -125.95, 134.07 APE8-rot-in 299.88 APE67-dihe-in -54.81, -22.83 -45.72, -53.17 APE12-dist-in 7.9604 APE11-dist-in 11.3761 APE10-dist-in 5.7901 APE9-dist-in 3.5461 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.15 0.203 0.259 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2jdt Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2JDVA P00517 16 351 351.0 L20:61351 Type1 Active DFGin 6.8915 13.8202 BLAminus -131.77, 167.29 66.94, 91.79 -105.86, 27.67 278.62, 60.56 -53.86, -24.56 in-in in 8.8406 Saltbr-in 2.8778 HRD-in -94.92, -55.32 76.45, 14.41 in-in-in SNCiii in-in ActLoopNT-in 2.9231 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.28, 166.03 APE9-dihe-na 121.76, -153.88 APE8-dihe-in -130.57, 133.66 APE8-rot-in 294.95 APE67-dihe-in -54.68, -28.08 -47.57, -51.85 APE12-dist-in 8.0027 APE11-dist-in 11.3848 APE10-dist-in 5.7807 APE9-dist-in 3.4188 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.08 0.21 0.276 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2jdv Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UVXA P00517 15 351 351.0 GVH:61351 Type1 Active DFGin 6.4797 13.8517 BLAminus -113.02, 171.98 67.75, 90.65 -101.98, 28.22 272.02, 52.69 -58.83, -28.67 in-in in 8.4347 Saltbr-in 2.8578 HRD-in -88.35, -54.63 73.53, 9.81 in-in-in SNCiii in-in ActLoopNT-in 2.9512 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.14, 156.72 APE9-dihe-na 129.39, -155.0 APE8-dihe-in -123.88, 135.4 APE8-rot-in 299.16 APE67-dihe-in -58.73, -23.74 -45.63, -51.62 APE12-dist-in 7.8612 APE11-dist-in 11.2242 APE10-dist-in 5.6959 APE9-dist-in 3.5342 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.175 0.237 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uvx Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UVYA P00517 16 351 351.0 GVI:61351 Type1 Active DFGin 6.6883 13.7301 BLAminus -138.26, 177.38 63.89, 90.39 -103.82, 30.2 278.88, 60.78 -58.29, -25.32 in-in in 8.5322 Saltbr-in 2.8677 HRD-in -91.19, -52.46 73.0, 13.57 in-in-in SNCiii in-in ActLoopNT-in 2.955 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.29, 164.08 APE9-dihe-na 125.27, -164.76 APE8-dihe-in -118.0, 134.0 APE8-rot-in 303.1 APE67-dihe-in -57.9, -24.5 -45.7, -51.96 APE12-dist-in 7.8997 APE11-dist-in 11.319 APE10-dist-in 5.7311 APE9-dist-in 3.5369 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.218 0.253 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uvy Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UVZA P00517 15 351 351.0 GVJ:61351 Type1 Active DFGin 6.4579 13.9569 BLAminus -114.74, -176.7 66.06, 78.43 -99.26, 24.12 270.22, 58.52 -59.61, -24.08 in-in in 8.5257 Saltbr-in 2.6293 HRD-in -92.0, -54.55 74.61, 15.4 in-in-in SNCiii in-in ActLoopNT-in 2.8816 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.48, 161.55 APE9-dihe-na 129.65, -159.59 APE8-dihe-in -126.36, 133.57 APE8-rot-in 300.99 APE67-dihe-in -58.07, -24.11 -45.65, -50.65 APE12-dist-in 7.8629 APE11-dist-in 11.1547 APE10-dist-in 5.6461 APE9-dist-in 3.4616 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.94 0.205 0.245 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uvz Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW0A P00517 15 351 351.0 GVK:61351 Type1 Active DFGin 6.6807 13.8545 BLAminus -123.12, 170.63 63.31, 92.05 -104.17, 27.62 276.86, 57.75 -54.59, -30.88 in-in in 8.6064 Saltbr-in 2.7061 HRD-in -91.98, -52.4 71.75, 13.11 in-in-in SNCiii in-in ActLoopNT-in 2.9563 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.42, 159.97 APE9-dihe-na 125.35, -161.9 APE8-dihe-in -119.06, 132.94 APE8-rot-in 303.5 APE67-dihe-in -59.26, -23.73 -42.54, -53.1 APE12-dist-in 7.95 APE11-dist-in 11.363 APE10-dist-in 5.817 APE9-dist-in 3.5714 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.204 0.248 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw0 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW3A P00517 15 351 351.0 GVG:61351 Type1 Active DFGin 6.5124 13.5734 BLAminus -134.7, 177.07 65.72, 91.81 -107.38, 30.0 281.86, 61.73 -63.9, -19.07 in-in in 8.5145 Saltbr-in 2.9351 HRD-in -92.24, -48.61 69.34, 10.98 in-in-in SNCiii in-in ActLoopNT-in 2.9305 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.62, 157.61 APE9-dihe-na 126.53, -159.5 APE8-dihe-in -119.31, 132.1 APE8-rot-in 301.91 APE67-dihe-in -60.53, -27.24 -45.08, -48.44 APE12-dist-in 7.8948 APE11-dist-in 11.2961 APE10-dist-in 5.7653 APE9-dist-in 3.5543 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.19 0.191 0.252 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw3 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW4A P00517 15 351 351.0 L15:61351 Type1 Active DFGin 6.4921 14.0113 BLAminus -125.98, 178.92 62.3, 87.41 -98.07, 19.83 275.17, 58.86 -56.03, -29.21 in-in in 8.6955 Saltbr-in 2.6847 HRD-in -99.89, -51.11 66.26, 15.03 in-in-in SNCiii in-in ActLoopNT-in 2.9933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.17, 154.32 APE9-dihe-na 136.7, -157.38 APE8-dihe-in -123.04, 134.76 APE8-rot-in 305.65 APE67-dihe-in -59.99, -23.88 -42.91, -53.6 APE12-dist-in 7.8692 APE11-dist-in 11.2922 APE10-dist-in 5.8184 APE9-dist-in 3.8346 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.219 0.274 A 351.0 336.0 1 25 25 0 [[44, 298]] 1.0 2uw4 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW5A P00517 16 351 351.0 GVN:61351 Type1 Active DFGin 6.4006 13.8772 BLAminus -133.91, 172.04 65.21, 93.24 -108.15, 25.65 277.97, 62.72 -53.54, -37.02 in-in in 8.7284 Saltbr-in 2.8062 HRD-in -86.0, -54.55 71.01, 10.44 in-in-in SNCiii in-in ActLoopNT-in 2.9816 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.67, 159.27 APE9-dihe-na 130.34, -162.49 APE8-dihe-in -114.97, 133.7 APE8-rot-in 296.24 APE67-dihe-in -62.66, -23.25 -45.46, -47.84 APE12-dist-in 7.9004 APE11-dist-in 11.248 APE10-dist-in 5.7124 APE9-dist-in 3.5694 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.14 0.207 0.259 A 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2uw5 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW6A P00517 15 351 351.0 GVO:61351 Type1 Active DFGin 6.5366 14.032 BLAminus -123.92, -171.55 58.59, 76.44 -99.17, 23.1 278.06, 64.52 -53.95, -28.73 in-in in 8.8994 Saltbr-in 2.6953 HRD-in -89.32, -52.49 72.51, 13.36 in-in-in SNCiii in-in ActLoopNT-in 2.8911 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.65, 165.8 APE9-dihe-na 120.56, -163.15 APE8-dihe-in -118.84, 134.95 APE8-rot-in 297.85 APE67-dihe-in -59.8, -23.71 -47.39, -48.58 APE12-dist-in 7.9462 APE11-dist-in 11.3542 APE10-dist-in 5.7826 APE9-dist-in 3.5043 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.23 0.192 0.244 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw6 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW7A P00517 15 351 351.0 GVP:61351 Type1 Active DFGin 6.6166 13.7352 BLAminus -136.69, 175.22 59.69, 95.21 -111.12, 31.03 278.38, 57.43 -58.09, -25.49 in-in in 8.5612 Saltbr-in 2.7092 HRD-in -86.23, -51.08 72.7, 10.78 in-in-in SNCiii in-in ActLoopNT-in 3.0203 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.27, 162.23 APE9-dihe-na 121.1, -162.52 APE8-dihe-in -116.53, 136.36 APE8-rot-in 303.46 APE67-dihe-in -55.18, -28.45 -48.94, -51.5 APE12-dist-in 7.93 APE11-dist-in 11.4491 APE10-dist-in 5.8017 APE9-dist-in 3.5143 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.239 0.318 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw7 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2UW8A P00517 15 351 351.0 GVQ:61351 Type1 Active DFGin 6.3045 14.2798 BLAminus -127.77, 173.64 63.87, 90.76 -102.26, 24.27 274.86, 58.11 -57.85, -25.36 in-in in 8.7881 Saltbr-in 2.6187 HRD-in -87.86, -52.11 70.45, 11.81 in-in-in SNCiii in-in ActLoopNT-in 2.9485 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.21, 162.91 APE9-dihe-na 127.4, -162.92 APE8-dihe-in -121.14, 133.97 APE8-rot-in 304.45 APE67-dihe-in -56.86, -24.67 -46.34, -50.57 APE12-dist-in 7.9507 APE11-dist-in 11.2821 APE10-dist-in 5.7747 APE9-dist-in 3.5317 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.188 0.233 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2uw8 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VNWA P00517 15 351 351.0 M01:61351 Type1 Active DFGin 6.5203 14.2539 BLAminus -99.0, -162.5 57.81, 69.82 -93.2, 19.41 267.8, 58.81 -57.89, -28.06 in-in in 8.608 Saltbr-in 2.7916 HRD-in -93.79, -52.83 75.12, 12.44 in-in-in SNCiii in-in ActLoopNT-in 2.9661 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.21, 164.77 APE9-dihe-na 124.54, -157.72 APE8-dihe-in -125.0, 133.49 APE8-rot-in 299.26 APE67-dihe-in -56.84, -26.04 -43.44, -52.9 APE12-dist-in 7.8989 APE11-dist-in 11.3061 APE10-dist-in 5.7483 APE9-dist-in 3.4375 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.09 0.179 0.247 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vnw Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VNYA P00517 15 351 351.0 M02:61351 Type1 Active DFGin 6.5021 13.8926 BLAminus -119.89, 177.02 61.41, 90.56 -103.09, 29.14 278.68, 50.15 -55.55, -28.57 in-in in 8.4839 Saltbr-in 2.8581 HRD-in -86.58, -53.8 72.94, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.9193 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.32, 164.15 APE9-dihe-na 124.54, -158.42 APE8-dihe-in -121.16, 130.65 APE8-rot-in 300.17 APE67-dihe-in -57.01, -22.39 -43.28, -52.93 APE12-dist-in 7.9208 APE11-dist-in 11.3298 APE10-dist-in 5.8145 APE9-dist-in 3.478 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.96 0.226 0.292 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vny Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO3A P00517 15 351 351.0 M04:61352 Type1 Active DFGin 6.4299 14.4177 BLAminus -103.33, -162.63 58.24, 61.11 -86.11, 18.5 266.87, 55.84 -51.81, -33.51 in-in in 8.7704 Saltbr-in 2.6553 HRD-in -94.44, -55.26 74.28, 15.13 in-in-in SNCiii in-in ActLoopNT-in 2.9179 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.75, 157.39 APE9-dihe-na 131.99, -148.74 APE8-dihe-in -128.37, 129.57 APE8-rot-in 302.29 APE67-dihe-in -55.2, -26.12 -39.48, -55.25 APE12-dist-in 7.9685 APE11-dist-in 11.4444 APE10-dist-in 5.8578 APE9-dist-in 3.6169 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.98 0.189 0.246 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 2vo3 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO6A P00517 14 351 351.0 M05:61352 Type1 Active DFGin 6.4346 14.1872 BLAminus -116.69, -177.73 56.84, 84.85 -93.23, 27.76 272.38, 55.86 -61.33, -23.85 in-in in 8.6236 Saltbr-in 2.7502 HRD-in -94.44, -52.03 70.59, 14.63 in-in-in SNCiii in-in ActLoopNT-in 2.9129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.43, 161.66 APE9-dihe-na 131.96, -159.34 APE8-dihe-in -122.22, 131.28 APE8-rot-in 303.11 APE67-dihe-in -58.4, -24.83 -41.37, -51.96 APE12-dist-in 7.9982 APE11-dist-in 11.3208 APE10-dist-in 5.7969 APE9-dist-in 3.5782 V105T,V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.97 0.175 0.229 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 2vo6 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C36A P00517 14 351 351.0 ZO9:61351 Type1 Active DFGin 6.1806 14.4761 BLAminus -118.69, 178.88 60.12, 90.41 -102.76, 21.93 269.17, 67.05 -52.26, -31.89 in-in in 8.958 Saltbr-in 2.7522 HRD-in -81.95, -52.55 68.64, 5.14 in-in-in SNCiii in-in ActLoopNT-in 2.9473 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.13, 158.34 APE9-dihe-na 127.36, -163.94 APE8-dihe-in -108.9, 133.1 APE8-rot-in 299.72 APE67-dihe-in -56.07, -28.95 -40.56, -54.07 APE12-dist-in 8.1424 APE11-dist-in 11.4572 APE10-dist-in 5.8378 APE9-dist-in 3.5366 F55Y,M121L,V124L,L174M,Q182K SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.98 0.158 0.19 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4c36 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C38A P00517 15 351 351.0 VUP:61351 Type1 Active DFGin 6.2217 14.4048 BLAminus -126.62, 165.92 74.69, 93.13 -106.33, 26.68 268.54, 56.88 -59.81, -19.94 in-in in 8.7724 Saltbr-in 2.7124 HRD-in -83.07, -52.03 71.32, 8.89 in-in-in SNCiii in-in ActLoopNT-in 2.9254 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.52, 161.58 APE9-dihe-na 127.55, -160.47 APE8-dihe-in -120.22, 132.35 APE8-rot-in 299.09 APE67-dihe-in -60.14, -23.8 -44.31, -50.86 APE12-dist-in 8.074 APE11-dist-in 11.4506 APE10-dist-in 5.8341 APE9-dist-in 3.5064 F55Y,M121L,V124L,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.58 0.154 0.178 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4c38 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1Q8UA P00517 8 351 351.0 H52:60961,H52:60962 Type1,Allosteric Active DFGin 6.1919 14.5396 BLAminus -121.34, -175.23 53.4, 94.64 -107.06, 23.52 275.18, 66.66 -55.71, -29.87 in-in in 9.3646 Saltbr-in 2.6498 HRD-in -94.99, -53.62 73.43, 4.82 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.92, 158.63 APE9-dihe-na 129.17, -156.38 APE8-dihe-in -121.51, 130.86 APE8-rot-in 299.83 APE67-dihe-in -61.21, -26.61 -47.69, -47.6 APE12-dist-in 8.2067 APE11-dist-in 11.5494 APE10-dist-in 5.967 APE9-dist-in 3.6469 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.9 0.173 0.206 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 1q8u Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3BWJA P00517 11 351 351.0 ARX:60351,ARX:60352 Type1,Allosteric Active DFGin 6.696 14.4073 BLAminus -110.43, 169.36 68.32, 91.4 -103.19, 23.79 279.15, 62.0 -69.5, -7.66 in-in in 8.6647 Saltbr-in 2.7201 HRD-in -86.31, -55.51 71.76, 12.05 in-in-in SNCiii in-in ActLoopNT-in 2.8621 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.81, 155.85 APE9-dihe-na 142.65, -162.5 APE8-dihe-in -110.95, 130.57 APE8-rot-in 293.64 APE67-dihe-in -63.27, -21.79 -42.33, -48.7 APE12-dist-in 8.115 APE11-dist-in 11.3778 APE10-dist-in 5.9209 APE9-dist-in 3.7349 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.201 0.249 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 3bwj Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4Z83E P00517 15 351 351.0 4L7:60401,4L7:60402 Type1,Allosteric Active DFGin 5.9886 14.5734 BLAminus -130.13, -162.52 52.5, 73.8 -91.1, 22.2 271.01, 60.02 -56.14, -30.3 in-in in 8.9604 Saltbr-in 2.6159 HRD-in -86.75, -50.89 68.08, 10.37 in-in-in SNCiii in-in ActLoopNT-in 2.878 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.2, 158.26 APE9-dihe-na 130.71, -157.52 APE8-dihe-in -119.41, 132.79 APE8-rot-in 303.19 APE67-dihe-in -56.65, -23.66 -45.82, -50.99 APE12-dist-in 8.1208 APE11-dist-in 11.4963 APE10-dist-in 5.9491 APE9-dist-in 3.7101 V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.8 0.182 0.217 E 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4z83 Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2VO0A P00517 9 351 351.0 M03:61354,M03:61355 Type1,Allosteric Active DFGin 6.4684 14.4354 BLAminus -105.06, -163.48 59.05, 63.73 -87.9, 21.77 268.86, 60.16 -61.88, -26.99 in-in in 8.8145 Saltbr-in 2.4561 HRD-in -97.05, -57.43 76.4, 9.67 in-in-in SNCiii in-in ActLoopNT-in 2.8932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.64, 159.11 APE9-dihe-na 131.22, -153.01 APE8-dihe-in -127.42, 133.63 APE8-rot-in 298.09 APE67-dihe-in -55.96, -25.96 -42.79, -54.49 APE12-dist-in 7.9676 APE11-dist-in 11.3833 APE10-dist-in 5.8985 APE9-dist-in 3.6486 V105T,V124A,L174M,Q182K SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.94 0.165 0.216 A 351.0 343.0 0 25 25 0 [[44, 298]] 1.0 2vo0 Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CA P00517 8 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.2009 14.4431 BLAminus -125.76, -178.37 54.76, 79.93 -90.51, 28.04 276.07, 57.76 -61.29, -35.5 in-in in 8.8075 Saltbr-in 2.8579 HRD-in -85.03, -54.57 65.22, 22.07 in-in-in SNCiii in-in ActLoopNT-in 2.8219 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.95, 159.1 APE9-dihe-na 118.65, -172.42 APE8-dihe-in -101.75, 128.13 APE8-rot-in 295.06 APE67-dihe-in -58.34, -26.98 -41.06, -49.71 APE12-dist-in 8.0918 APE11-dist-in 11.5524 APE10-dist-in 6.1282 APE9-dist-in 3.9113 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CB P00517 5 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.5319 14.6298 BLAminus -126.7, -178.91 56.82, 78.03 -91.32, 30.19 275.18, 53.57 -61.25, -34.87 in-in in 8.7621 Saltbr-in 3.0566 HRD-in -84.6, -55.03 67.66, 19.16 in-in-in SNCiii in-in ActLoopNT-in 2.8012 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.35, 159.24 APE9-dihe-na 119.5, -170.09 APE8-dihe-in -105.39, 130.22 APE8-rot-in 303.07 APE67-dihe-in -57.44, -28.07 -44.47, -49.51 APE12-dist-in 8.0466 APE11-dist-in 11.5239 APE10-dist-in 6.0242 APE9-dist-in 3.8597 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 B 350.0 347.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CC P00517 8 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.2974 14.7558 BLAminus -125.92, -177.85 55.25, 79.64 -90.5, 29.38 270.76, 52.31 -60.78, -37.14 in-in in 8.8167 Saltbr-in 2.6352 HRD-in -82.84, -55.25 65.25, 20.45 in-in-in SNCiii in-in ActLoopNT-in 2.8166 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.33, 159.63 APE9-dihe-na 118.14, -173.27 APE8-dihe-in -100.83, 130.06 APE8-rot-in 300.03 APE67-dihe-in -60.34, -24.98 -43.86, -49.06 APE12-dist-in 8.0524 APE11-dist-in 11.5266 APE10-dist-in 6.0815 APE9-dist-in 3.9132 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 C 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CD P00517 5 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.4689 14.6139 BLAminus -125.62, -178.32 56.8, 78.69 -92.33, 30.68 274.67, 61.46 -62.35, -34.64 in-in in 8.7979 Saltbr-in 2.6568 HRD-in -84.05, -54.95 66.91, 19.26 in-in-in SNCiii in-in ActLoopNT-in 2.8137 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.6, 160.31 APE9-dihe-na 118.55, -170.22 APE8-dihe-in -103.2, 129.22 APE8-rot-in 310.88 APE67-dihe-in -59.74, -24.78 -43.75, -49.55 APE12-dist-in 8.092 APE11-dist-in 11.4883 APE10-dist-in 6.0672 APE9-dist-in 3.881 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 D 350.0 347.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CE P00517 14 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.4857 14.6047 BLAminus -126.72, -179.02 57.21, 78.54 -91.86, 29.91 275.24, 58.74 -61.76, -34.81 in-in in 8.7747 Saltbr-in 2.8495 HRD-in -84.14, -54.47 66.34, 19.61 in-in-in SNCiii in-in ActLoopNT-in 2.8132 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.41, 160.32 APE9-dihe-na 118.41, -171.62 APE8-dihe-in -103.31, 130.93 APE8-rot-in 316.9 APE67-dihe-in -58.71, -26.13 -46.25, -48.17 APE12-dist-in 8.0859 APE11-dist-in 11.519 APE10-dist-in 6.0608 APE9-dist-in 3.871 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 E 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8CF P00517 8 351 351.0 G96:60351 Type1.5_Back Active DFGin 6.204 14.5963 BLAminus -125.48, -179.37 56.48, 79.11 -90.97, 29.84 273.44, 55.64 -61.95, -35.57 in-in in 8.801 Saltbr-in 2.9055 HRD-in -84.03, -54.54 65.26, 20.82 in-in-in SNCiii in-in ActLoopNT-in 2.8163 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.83, 160.18 APE9-dihe-na 118.26, -172.77 APE8-dihe-in -101.93, 130.0 APE8-rot-in 316.95 APE67-dihe-in -59.02, -26.57 -43.48, -49.35 APE12-dist-in 8.0793 APE11-dist-in 11.4951 APE10-dist-in 6.0617 APE9-dist-in 3.8792 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.265 0.29 F 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8c Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EA P00517 8 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.3073 14.6275 BLAminus -127.58, 177.12 59.26, 81.09 -89.3, 24.2 272.49, 51.41 -54.01, -38.82 in-in in 8.6228 Saltbr-in 2.6167 HRD-in -86.71, -49.98 69.16, 6.49 in-in-in SNCiii in-in ActLoopNT-in 2.8632 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.99, 154.32 APE9-dihe-na 133.62, -170.54 APE8-dihe-in -106.52, 129.54 APE8-rot-in 301.27 APE67-dihe-in -53.09, -32.91 -42.99, -51.98 APE12-dist-in 8.2069 APE11-dist-in 11.4816 APE10-dist-in 5.9204 APE9-dist-in 3.7722 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 A 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EB P00517 13 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.2938 14.7178 BLAminus -125.84, -172.92 50.21, 81.31 -89.14, 23.18 270.21, 58.55 -50.98, -43.5 in-in in 8.6642 Saltbr-in 2.6654 HRD-in -82.38, -53.17 68.54, 5.22 in-in-in SNCiii in-in ActLoopNT-in 2.8797 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.38, 161.75 APE9-dihe-na 128.75, -165.32 APE8-dihe-in -112.15, 133.4 APE8-rot-in 300.5 APE67-dihe-in -58.46, -24.04 -42.84, -57.3 APE12-dist-in 8.0985 APE11-dist-in 11.3489 APE10-dist-in 5.8215 APE9-dist-in 3.724 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 B 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EE P00517 8 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.5022 14.7143 BLAminus -125.94, 177.63 60.28, 78.38 -89.05, 26.68 272.68, 53.04 -58.15, -33.43 in-in in 8.5959 Saltbr-in 2.7412 HRD-in -83.69, -53.19 69.3, 12.83 in-in-in SNCiii in-in ActLoopNT-in 2.9203 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.44, 161.83 APE9-dihe-na 125.18, -160.92 APE8-dihe-in -119.48, 128.06 APE8-rot-in 308.71 APE67-dihe-in -61.97, -23.41 -42.69, -51.33 APE12-dist-in 8.1077 APE11-dist-in 11.5081 APE10-dist-in 5.9999 APE9-dist-in 3.6674 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 E 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EI P00517 4 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.2839 14.6216 BLAminus -121.51, -176.84 52.35, 81.35 -90.04, 28.89 273.59, 58.29 -59.59, -35.26 in-in in 8.5151 Saltbr-in 2.667 HRD-in -96.55, -53.06 68.92, 16.49 in-in-in SNCiii in-in ActLoopNT-in 2.8724 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.85, 164.56 APE9-dihe-na 117.18, -165.89 APE8-dihe-in -113.08, 128.95 APE8-rot-in 295.01 APE67-dihe-in -62.64, -25.23 -41.3, -50.45 APE12-dist-in 8.1826 APE11-dist-in 11.4443 APE10-dist-in 5.9011 APE9-dist-in 3.5317 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 I 350.0 348.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EL P00517 14 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.3558 14.4455 BLAminus -126.34, 179.53 56.51, 87.88 -97.22, 26.99 274.78, 53.86 -54.08, -36.01 in-in in 8.4902 Saltbr-in 2.9058 HRD-in -84.79, -53.72 69.04, 14.43 in-in-in SNCiii in-in ActLoopNT-in 2.9175 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.8, 165.17 APE9-dihe-na 117.16, -168.03 APE8-dihe-in -109.85, 132.76 APE8-rot-in 309.54 APE67-dihe-in -58.05, -25.67 -43.08, -54.13 APE12-dist-in 8.0742 APE11-dist-in 11.4769 APE10-dist-in 5.8902 APE9-dist-in 3.5416 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 L 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3E8EP P00517 8 351 351.0 G98:60351 Type1.5_Back Active DFGin 6.3511 14.4567 BLAminus -129.89, 174.6 59.69, 84.32 -91.75, 22.85 273.06, 63.33 -54.83, -37.28 in-in in 8.5071 Saltbr-in 3.0872 HRD-in -91.09, -52.59 71.75, 13.86 in-in-in SNCiii in-in ActLoopNT-in 2.8806 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.01, 169.23 APE9-dihe-na 113.75, -166.64 APE8-dihe-in -114.16, 128.38 APE8-rot-in 299.83 APE67-dihe-in -58.07, -28.95 -41.88, -52.2 APE12-dist-in 8.1136 APE11-dist-in 11.4255 APE10-dist-in 5.9681 APE9-dist-in 3.5443 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.245 0.279 P 350.0 344.0 0 25 25 0 [[44, 298]] 1.0 3e8e Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1XH9A P00517 14 351 351.0 R69:60351 Type1.5_Front Active DFGin 6.209 14.3533 BLAminus -129.75, -179.11 60.33, 73.87 -88.04, 22.6 274.32, 67.63 -61.73, -24.72 in-in in 8.5813 Saltbr-in 2.6088 HRD-in -83.79, -50.21 70.28, 10.19 in-in-in SNCiii in-in ActLoopNT-in 2.9141 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.47, 163.02 APE9-dihe-na 127.04, -169.55 APE8-dihe-in -104.83, 132.1 APE8-rot-in 300.02 APE67-dihe-in -61.76, -25.27 -43.65, -49.85 APE12-dist-in 8.2976 APE11-dist-in 11.8047 APE10-dist-in 6.2189 APE9-dist-in 3.6955 Q85E,V124A,L174M,Q182K,F188L TPO198,SEP339 TPO198,SEP339 XRAY 1.64 0.166 0.199 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1xh9 Bos taurus AGC_PRKACA_BOVIN AGC 1e-94 322.6 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SVHA P00517 15 351 351.0 I08:60351 Type1.5_Front Active DFGin 6.2901 14.3586 BLAminus -115.3, -171.03 56.71, 72.97 -89.54, 18.36 276.49, 75.83 -65.64, -21.28 in-in in 8.5191 Saltbr-in 2.4169 HRD-in -84.39, -53.98 69.64, 16.78 in-in-in SNCiii in-in ActLoopNT-in 3.0122 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.15, 156.51 APE9-dihe-na 127.45, -173.0 APE8-dihe-in -94.86, 131.95 APE8-rot-in 296.28 APE67-dihe-in -64.98, -17.24 -40.94, -52.95 APE12-dist-in 8.6846 APE11-dist-in 11.7208 APE10-dist-in 6.2204 APE9-dist-in 3.7125 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.214 0.259 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 1svh Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNIA P00517 11 351 351.0 M77:60601 Type1 Inactive DFGin 6.1218 13.3386 ABAminus -125.47, 13.51 -148.05, 120.42 -113.28, 22.31 295.85, 71.04 -57.43, -24.9 in-in in 9.2508 Saltbr-in 2.8621 HRD-in -97.25, -49.49 72.22, 6.42 in-in-in SNCiii in-in ActLoopNT-in 2.9904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.86, 164.06 APE9-dihe-na 122.41, -161.87 APE8-dihe-in -119.99, 136.29 APE8-rot-in 295.68 APE67-dihe-in -63.27, -25.72 -47.9, -45.46 APE12-dist-in 8.1408 APE11-dist-in 11.2646 APE10-dist-in 5.7788 APE9-dist-in 3.3758 L50I,V124M,E128D,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.27 0.192 0.268 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gni Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1STCE P00517 16 351 351.0 STU:60351 Type1 Inactive DFGin 6.1254 14.6764 ABAminus -152.28, -21.25 -98.94, 113.28 -112.23, 27.12 284.07, 102.64 -65.61, -29.61 in-in in 9.1737 Saltbr-in 2.6077 HRD-out -84.15, -57.61 42.07, 55.99 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.84, 156.46 APE9-dihe-na 129.45, -158.0 APE8-dihe-in -121.73, 124.56 APE8-rot-in 292.46 APE67-dihe-in -75.12, -21.46 -28.7, -46.78 APE12-dist-in 8.3869 APE11-dist-in 11.1625 APE10-dist-in 5.8257 APE9-dist-in 4.4432 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.3 0.208 0.33 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1stc Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO2A P00517 8 351 351.0 15I:61351 Type1 Inactive DFGin 6.1445 13.7565 ABAminus -111.64, -15.7 -114.7, 103.29 -107.0, 15.63 291.73, 77.0 -53.95, -31.44 in-in in 8.9831 Saltbr-in 2.7087 HRD-in -83.31, -56.68 67.99, 8.34 in-in-in SNCiii in-in ActLoopNT-in 2.9313 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 157.34 APE9-dihe-na 124.98, -162.06 APE8-dihe-in -114.19, 137.15 APE8-rot-in 302.62 APE67-dihe-in -58.09, -28.32 -43.68, -52.1 APE12-dist-in 8.012 APE11-dist-in 11.4691 APE10-dist-in 5.8391 APE9-dist-in 3.6098 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.98 0.158 0.191 A 351.0 344.0 0 25 25 0 [[44, 298]] 1.0 3zo2 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3ZO3A P00517 12 351 351.0 QNI:61351 Type1 Inactive DFGin 5.8139 14.5584 ABAminus -113.45, -3.91 -119.58, 103.74 -104.44, 16.56 281.0, 73.71 -59.51, -27.51 in-in in 9.1187 Saltbr-in 2.7878 HRD-in -88.87, -55.75 64.02, 12.24 in-in-in SNCiii in-in ActLoopNT-in 2.8636 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.07, 157.3 APE9-dihe-na 125.82, -155.48 APE8-dihe-in -117.69, 139.23 APE8-rot-in 297.95 APE67-dihe-in -57.23, -32.24 -46.12, -52.37 APE12-dist-in 7.9721 APE11-dist-in 11.3311 APE10-dist-in 5.7624 APE9-dist-in 3.6518 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.1 0.176 0.21 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 3zo3 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 5VI9A P00517 15 351 351.0 9D4:60401 Type1 Inactive DFGin 6.4135 14.639 ABAminus -108.08, -28.68 -104.39, 134.13 -134.73, 37.16 293.35, 85.38 -60.78, -29.79 in-out in 9.3856 Saltbr-out 3.754 HRD-in -77.99, -57.09 68.94, 10.33 out-in-in SNCoii in-in ActLoopNT-in 2.8473 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.52, 160.7 APE9-dihe-na 121.66, -160.6 APE8-dihe-in -114.63, 135.81 APE8-rot-in 302.32 APE67-dihe-in -61.89, -29.97 -46.88, -46.56 APE12-dist-in 8.0832 APE11-dist-in 11.498 APE10-dist-in 5.8264 APE9-dist-in 3.6359 None TPO198 TPO198 XRAY 1.95 0.209 0.256 A 351.0 307.0 4 25 25 0 [[44, 298]] 1.0 5vi9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 5VIBA P00517 19 351 351.0 9D1:60401 Type1 Inactive DFGin 6.6212 14.8324 ABAminus -107.11, -34.58 -98.31, 117.88 -117.47, 22.93 281.07, 85.16 -57.39, -18.74 in-in in 9.1872 Saltbr-in 3.5607 HRD-in -77.43, -53.28 63.56, 13.71 in-in-in SNCiii in-in ActLoopNT-in 2.8615 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.02, 160.82 APE9-dihe-na 122.63, -164.02 APE8-dihe-in -113.1, 131.73 APE8-rot-in 301.25 APE67-dihe-in -62.36, -27.21 -42.7, -49.96 APE12-dist-in 7.9483 APE11-dist-in 11.4159 APE10-dist-in 5.7564 APE9-dist-in 3.504 None TPO198 TPO198 XRAY 2.37 0.215 0.276 A 351.0 309.0 0 25 25 0 [[44, 298]] 1.0 5vib Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 1SZMB P00517 15 351 351.0 BI4:60351 Type1 Inactive DFGin 6.9164 16.0168 ABAminus -124.67, -37.03 -119.38, 110.7 -112.86, 23.01 290.52, 94.06 -59.96, -45.74 out-out out 10.6181 Saltbr-out 4.666 HRD-in -70.48, -44.14 31.9, 37.49 out-in-in SNCoii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.49, 166.21 APE9-dihe-na 109.44, 164.47 APE8-dihe-in -71.29, 133.53 APE8-rot-in 294.81 APE67-dihe-in -63.33, -24.2 -45.0, -46.86 APE12-dist-in 8.346 APE11-dist-in 11.522 APE10-dist-in 5.9849 APE9-dist-in 4.4453 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 B 350.0 323.0 0 25 25 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4AXAA P00517 15 351 351.0 RKD:61351 Type1 Inactive DFGin 6.203 13.8956 ABAminus -121.83, -29.08 -102.06, 117.48 -118.59, 24.36 279.49, 73.66 -60.99, -27.08 in-in in 8.7606 Saltbr-in 3.0068 HRD-in -91.45, -56.33 70.15, 3.62 in-in-in SNCiii in-in ActLoopNT-in 2.8879 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.21, 158.94 APE9-dihe-na 126.47, -155.87 APE8-dihe-in -119.74, 130.42 APE8-rot-in 299.77 APE67-dihe-in -59.64, -26.03 -40.97, -51.19 APE12-dist-in 7.9966 APE11-dist-in 11.4177 APE10-dist-in 5.8548 APE9-dist-in 3.7051 V105T,V124A,L174M,Q182K TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.216 0.256 A 351.0 337.0 0 25 25 0 [[44, 298]] 1.0 4axa Bos taurus AGC_PRKACA_BOVIN AGC 4.5e-94 320.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C34A P00517 11 351 351.0 STU:61351 Type1 Inactive DFGin 6.5166 14.8494 ABAminus -119.31, -40.44 -98.64, 112.68 -107.28, 23.29 283.36, 88.13 -59.12, -19.89 in-in in 8.8642 Saltbr-in 2.9854 HRD-in -78.06, -54.1 69.84, 7.38 in-in-in SNCiii in-in ActLoopNT-in 2.9107 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.66, 162.66 APE9-dihe-na 118.12, -166.39 APE8-dihe-in -111.07, 134.19 APE8-rot-in 303.77 APE67-dihe-in -56.72, -26.94 -46.04, -52.13 APE12-dist-in 8.3983 APE11-dist-in 11.4581 APE10-dist-in 5.7648 APE9-dist-in 3.4077 F55Y,M121L,V124L,L174M,Q182K SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.78 0.18 0.214 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 4c34 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C37A P00517 14 351 351.0 Z21:61351 Type1 Inactive DFGin 6.2618 14.2841 ABAminus -113.24, -47.75 -78.1, 110.9 -112.08, 25.76 272.69, 64.65 -57.89, -26.17 in-in in 8.7279 Saltbr-in 2.7412 HRD-in -81.42, -53.5 70.95, 1.92 in-in-in SNCiii in-in ActLoopNT-in 2.9412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.71, 160.19 APE9-dihe-na 127.27, -162.5 APE8-dihe-in -118.08, 133.43 APE8-rot-in 300.5 APE67-dihe-in -57.54, -26.87 -42.89, -53.17 APE12-dist-in 8.1544 APE11-dist-in 11.5086 APE10-dist-in 5.8833 APE9-dist-in 3.537 F55Y,M121L,V124L,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.157 0.179 A 351.0 338.0 0 25 25 0 [[44, 298]] 1.0 4c37 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 2GNHA P00517 11 351 351.0 H52:60501,H52:60502 Type1,Allosteric Inactive DFGin 5.7262 14.706 ABAminus -128.79, 15.58 -151.1, 122.77 -119.76, 23.12 270.41, 63.78 -48.67, -39.31 in-in in 9.333 Saltbr-in 2.8243 HRD-in -85.53, -55.44 74.29, 10.02 in-in-in SNCiii in-in ActLoopNT-in 2.9565 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.69, 165.93 APE9-dihe-na 124.87, -164.72 APE8-dihe-in -119.96, 131.77 APE8-rot-in 295.2 APE67-dihe-in -55.53, -26.21 -49.22, -48.81 APE12-dist-in 8.1711 APE11-dist-in 11.3893 APE10-dist-in 5.8788 APE9-dist-in 3.4654 L50I,V124M,E128D,Q182K,T184A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.05 0.198 0.256 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 2gnh Bos taurus AGC_PRKACA_BOVIN AGC 2.1e-95 324.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 3AG9A P00517 15 351 351.0 No_ligand No_ligand Inactive DFGin 7.051 16.1774 BLAminus -121.67, 168.31 69.6, 87.4 -105.16, 26.26 286.68, 81.88 -58.4, -43.3 out-out out 10.486 Saltbr-out 4.7632 HRD-in -75.01, -50.0 50.19, 29.04 out-in-in SNCoii in-in ActLoopNT-in 2.8564 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.66, 167.28 APE9-dihe-na 97.3, 169.91 APE8-dihe-in -87.06, 128.77 APE8-rot-in 296.19 APE67-dihe-in -53.54, -29.25 -42.73, -48.49 APE12-dist-in 8.336 APE11-dist-in 11.2386 APE10-dist-in 5.7464 APE9-dist-in 4.3081 None TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.23 0.246 A 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3ag9 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9FQRXT P00517 26 351 351.0 No_ligand No_ligand Inactive DFGin 7.5042 15.4719 BLAminus -120.43, -175.35 59.39, 66.35 -90.0, 32.7 274.65, 67.61 -64.07, -27.17 in-out in 8.66 Saltbr-out 4.4575 HRD-in -81.78, -57.62 51.32, 20.96 out-in-in SNCoii in-in ActLoopNT-in 3.2154 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.53, 169.85 APE9-dihe-na 132.17, 174.57 APE8-dihe-in -89.75, 132.06 APE8-rot-in 314.38 APE67-dihe-in -73.91, -30.73 -62.64, -19.12 APE12-dist-in 8.4981 APE11-dist-in 10.7604 APE10-dist-in 6.0224 APE9-dist-in 4.8414 None None None EM 5.0 999.0 999.0 Xt 351.0 294.0 0 25 25 0 [[44, 298]] 1.0 9fqr Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 4C35A P00517 11 351 351.0 NU3:61351 Type1.5_Back Inactive DFGin 5.96 15.1175 None -103.23, -88.31 -54.39, 108.88 -97.56, 11.02 265.67, 64.27 -54.79, -37.29 in-in in 9.1847 Saltbr-in 2.7744 HRD-in -78.97, -53.39 72.53, 0.25 in-in-in SNCiii in-in ActLoopNT-in 2.8688 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.98, 158.62 APE9-dihe-na 121.3, -169.27 APE8-dihe-in -106.38, 130.41 APE8-rot-in 302.02 APE67-dihe-in -58.09, -26.56 -41.09, -54.15 APE12-dist-in 8.7429 APE11-dist-in 11.6126 APE10-dist-in 5.9626 APE9-dist-in 3.4271 F55Y,M121L,V124L,L174M,Q182K SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.19 0.186 0.24 A 351.0 341.0 0 25 25 0 [[44, 298]] 1.0 4c35 Bos taurus AGC_PRKACA_BOVIN AGC 7.8e-94 319.7 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW7G P00517 13 351 351.0 ANP:403 ATPlike Inactive None 999.0 999.0 None -155.4, -162.2 59.11, 63.62 -70.57, 12.19 999.0, 999.0 -65.51, -34.83 out-none out 10.9713 Saltbr-none 999.0 HRD-in -65.14, -55.26 50.7, 27.28 none-in-out SNCnio in-out ActLoopNT-in 2.5754 ActLoopCT-out nonTYR APEdihe_aaini APEdist_iiio APE10-dihe-na -166.96, 170.69 APE9-dihe-na 108.98, -156.8 APE8-dihe-in -102.79, 139.06 APE8-rot-none 999.0 APE67-dihe-in -58.63, -28.81 -67.98, -6.96 APE12-dist-in 9.2283 APE11-dist-in 10.2672 APE10-dist-in 6.4383 APE9-dist-out 6.202 None None None EM 6.0 999.0 999.0 G 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 9dw7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW4K P00517 13 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -155.5, -168.49 59.79, 60.87 -83.31, 16.99 999.0, 999.0 -58.46, -53.69 in-none in 9.8843 Saltbr-none 999.0 HRD-in -75.2, -40.09 55.77, 26.65 none-in-none SNCnin in-none ActLoopNT-in 2.6727 ActLoopCT-none nonTYR APEdihe_aaini APEdist_iiii APE10-dihe-na -174.21, -178.74 APE9-dihe-na 106.6, -165.51 APE8-dihe-in -76.59, 132.39 APE8-rot-none 999.0 APE67-dihe-in -65.14, -23.53 -62.01, -33.48 APE12-dist-in 9.2205 APE11-dist-in 11.7506 APE10-dist-in 7.9925 APE9-dist-in 5.2599 None None None EM 9.0 999.0 999.0 K 351.0 331.0 0 25 25 0 [[44, 298]] 1.0 9dw4 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW7K P00517 13 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -155.25, -168.9 60.19, 60.97 -83.26, 17.04 999.0, 999.0 -58.67, -53.39 in-none in 9.875 Saltbr-none 999.0 HRD-in -75.5, -40.23 55.96, 26.19 none-in-none SNCnin in-none ActLoopNT-in 2.684 ActLoopCT-none nonTYR APEdihe_aaini APEdist_iiii APE10-dihe-na -174.15, -178.86 APE9-dihe-na 106.51, -165.36 APE8-dihe-in -77.09, 132.58 APE8-rot-none 999.0 APE67-dihe-in -65.64, -23.21 -62.33, -33.03 APE12-dist-in 9.2221 APE11-dist-in 11.7466 APE10-dist-in 7.9705 APE9-dist-in 5.2537 None None None EM 6.0 999.0 999.0 K 351.0 331.0 0 25 25 0 [[44, 298]] 1.0 9dw7 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW5G P00517 13 351 351.0 ANP:403 ATPlike None DFGin 7.3339 15.8767 BLAminus -126.22, -169.89 60.75, 61.77 -87.02, 21.16 273.51, 93.96 -63.0, -33.74 out-none out 10.2523 Saltbr-none 999.0 HRD-in -80.85, -56.62 73.43, -6.68 none-in-in SNCnii in-in ActLoopNT-in 2.7819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.11, -173.97 APE9-dihe-na 106.0, -157.25 APE8-dihe-in -108.29, 136.12 APE8-rot-in 326.0 APE67-dihe-in -63.46, -43.06 -59.57, -33.75 APE12-dist-in 9.1133 APE11-dist-in 11.9553 APE10-dist-in 6.8101 APE9-dist-in 4.5632 None TPO198 TPO198 EM 3.8 999.0 999.0 G 351.0 330.0 0 25 25 0 [[44, 298]] 1.0 9dw5 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_BOVIN 9DW8G P00517 15 329 351.0 ANP:403 ATPlike None DFGin 6.0696 14.2353 BLAminus -131.43, -174.72 59.27, 66.66 -86.28, 33.46 293.19, 93.28 -61.23, -49.05 in-none in 9.9111 Saltbr-none 999.0 HRD-in -98.32, -49.71 57.42, 11.15 none-in-in SNCnii in-in ActLoopNT-in 2.9612 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.06, 160.73 APE9-dihe-na 123.3, -175.7 APE8-dihe-in -89.52, 132.72 APE8-rot-in 298.44 APE67-dihe-in -69.93, -27.98 -56.75, -38.6 APE12-dist-in 8.7001 APE11-dist-in 11.5933 APE10-dist-in 6.4109 APE9-dist-in 4.8026 None TPO198 TPO198 EM 3.5 999.0 999.0 G 351.0 309.0 0 25 25 0 [[44, 298]] 1.0 9dw8 Bos taurus AGC_PRKACA_BOVIN AGC 1.3e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EM7A P25321 11 351 351.0 ADP:60403 ATPlike Active DFGin 5.924 14.3384 BLAminus -118.71, 173.1 68.53, 85.06 -96.18, 23.36 270.78, 55.34 -59.75, -28.55 in-in in 8.7405 Saltbr-in 2.7108 HRD-in -88.33, -53.93 74.88, 10.19 in-in-in SNCiii in-in ActLoopNT-in 2.9674 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.73, 159.92 APE9-dihe-na 127.98, -160.75 APE8-dihe-in -119.5, 137.47 APE8-rot-in 298.57 APE67-dihe-in -59.39, -22.73 -49.47, -50.59 APE12-dist-in 8.0499 APE11-dist-in 11.4294 APE10-dist-in 5.809 APE9-dist-in 3.6743 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.238 0.139 0.157 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6em7 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EMAA P25321 12 351 351.0 ATP:60401 ATPlike Active DFGin 6.8466 14.0282 BLAminus -121.3, 163.01 76.03, 95.19 -107.48, 29.41 285.05, 72.84 -63.27, -23.25 in-in in 8.5805 Saltbr-in 2.9123 HRD-in -88.06, -51.23 73.05, 9.34 in-in-in SNCiii in-in ActLoopNT-in 2.8434 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.85, 162.03 APE9-dihe-na 127.51, -167.2 APE8-dihe-in -113.51, 133.85 APE8-rot-in 299.54 APE67-dihe-in -58.99, -24.47 -49.7, -50.19 APE12-dist-in 8.208 APE11-dist-in 11.4336 APE10-dist-in 5.7768 APE9-dist-in 3.5854 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.88 0.184 0.213 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6ema Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ESAA P25321 11 351 351.0 AMP:60401 ATPlike Active DFGin 6.1394 14.3654 BLAminus -120.63, 169.73 70.22, 89.96 -100.72, 24.5 270.85, 56.09 -58.05, -28.66 in-in in 8.6912 Saltbr-in 2.8734 HRD-in -93.01, -53.86 73.79, 10.3 in-in-in SNCiii in-in ActLoopNT-in 2.9643 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.44, 160.95 APE9-dihe-na 124.73, -163.46 APE8-dihe-in -117.05, 136.25 APE8-rot-in 299.26 APE67-dihe-in -59.89, -22.61 -49.24, -49.61 APE12-dist-in 8.0912 APE11-dist-in 11.4994 APE10-dist-in 5.8224 APE9-dist-in 3.6604 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.307 0.132 0.147 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6esa Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y8CA P25321 13 351 351.0 ATP:60402 ATPlike Active DFGin 5.7272 14.3024 BLAminus -123.99, 172.57 69.5, 82.73 -92.15, 25.74 279.44, 63.0 -58.78, -31.82 in-in in 9.1661 Saltbr-in 2.6378 HRD-in -96.49, -52.39 69.1, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.8845 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.28, 160.42 APE9-dihe-na 122.78, -169.96 APE8-dihe-in -106.17, 134.07 APE8-rot-in 304.81 APE67-dihe-in -60.24, -22.7 -48.33, -48.43 APE12-dist-in 8.0442 APE11-dist-in 11.5168 APE10-dist-in 5.9394 APE9-dist-in 3.8952 None TPO198,SEP339 TPO198,SEP339 XRAY 1.76 0.162 0.19 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 6y8c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1NA P25321 1 351 351.0 8G8:60402 Allosteric Active DFGin 6.4141 14.3021 BLAminus -123.89, -172.22 60.93, 80.4 -92.44, 26.18 275.59, 66.61 -60.07, -25.93 in-in in 8.7465 Saltbr-in 3.033 HRD-in -89.37, -52.82 73.6, 7.6 in-in-in SNCiii in-in ActLoopNT-in 2.9227 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.19, 156.64 APE9-dihe-na 134.09, -162.2 APE8-dihe-in -112.34, 129.13 APE8-rot-in 298.42 APE67-dihe-in -61.33, -22.28 -43.88, -53.69 APE12-dist-in 8.451 APE11-dist-in 11.6981 APE10-dist-in 6.1521 APE9-dist-in 3.7784 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.405 0.154 0.179 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 5n1n Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3IA P25321 12 351 351.0 BJQ:60404 Allosteric Active DFGin 6.2036 14.3735 BLAminus -121.15, 165.89 72.6, 94.77 -102.91, 24.31 271.68, 55.3 -58.81, -29.64 in-in in 8.5664 Saltbr-in 2.9174 HRD-in -84.69, -52.32 69.36, 13.72 in-in-in SNCiii in-in ActLoopNT-in 2.9163 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.06, 170.9 APE9-dihe-na 117.62, -155.4 APE8-dihe-in -132.77, 134.35 APE8-rot-in 303.36 APE67-dihe-in -62.11, -19.9 -47.3, -51.17 APE12-dist-in 8.1248 APE11-dist-in 11.1999 APE10-dist-in 5.6654 APE9-dist-in 3.6237 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.14 0.134 0.151 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3i Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3KA P25321 12 351 351.0 GGB:60401 Allosteric Active DFGin 6.1849 14.34 BLAminus -124.6, 161.61 76.98, 90.66 -99.67, 25.29 272.38, 65.33 -61.96, -25.98 in-in in 8.6368 Saltbr-in 3.0012 HRD-in -87.33, -51.9 70.65, 14.42 in-in-in SNCiii in-in ActLoopNT-in 2.9472 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.91, 162.87 APE9-dihe-na 131.35, -156.18 APE8-dihe-in -123.66, 133.94 APE8-rot-in 296.91 APE67-dihe-in -59.29, -22.9 -47.8, -51.08 APE12-dist-in 8.1169 APE11-dist-in 11.1579 APE10-dist-in 5.6584 APE9-dist-in 3.7179 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.33 0.146 0.172 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3k Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Z08A P25321 14 351 351.0 NPO:60401 Allosteric Active DFGin 6.0045 14.3152 BLAminus -122.86, -172.56 56.32, 85.8 -96.13, 22.67 273.1, 62.96 -62.03, -25.78 in-in in 8.7081 Saltbr-in 2.5485 HRD-in -86.99, -51.51 69.72, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.9103 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.61, 168.88 APE9-dihe-na 120.32, -158.83 APE8-dihe-in -126.12, 135.53 APE8-rot-in 304.13 APE67-dihe-in -63.09, -19.11 -50.64, -46.8 APE12-dist-in 8.1729 APE11-dist-in 11.2225 APE10-dist-in 5.7126 APE9-dist-in 3.5871 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.49 0.163 0.185 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6z08 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE2A P25321 13 351 351.0 A1JE1:60504 Allosteric Active DFGin 6.9065 14.6005 BLAminus -130.51, -172.34 64.95, 64.92 -87.74, 25.39 275.14, 64.69 -64.84, -26.39 in-in in 8.9545 Saltbr-in 2.7115 HRD-in -89.39, -50.72 72.95, 14.8 in-in-in SNCiii in-in ActLoopNT-in 2.9921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.73, 162.53 APE9-dihe-na 125.67, -157.85 APE8-dihe-in -124.12, 131.82 APE8-rot-in 303.61 APE67-dihe-in -61.71, -21.87 -46.36, -49.79 APE12-dist-in 8.2745 APE11-dist-in 11.3295 APE10-dist-in 5.8612 APE9-dist-in 3.7356 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.68 0.209 0.233 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9re2 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REMA P25321 12 351 351.0 A1JEL:60401 Allosteric Active DFGin 6.4257 14.5409 BLAminus -124.03, 163.4 76.56, 89.18 -99.82, 25.59 271.66, 58.78 -64.22, -23.78 in-in in 8.6205 Saltbr-in 2.8774 HRD-in -87.63, -52.43 69.95, 13.38 in-in-in SNCiii in-in ActLoopNT-in 2.9373 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.48, 163.83 APE9-dihe-na 114.89, 177.74 APE8-dihe-in -94.85, 132.62 APE8-rot-in 300.61 APE67-dihe-in -61.62, -20.97 -47.15, -48.45 APE12-dist-in 8.263 APE11-dist-in 11.3978 APE10-dist-in 5.9326 APE9-dist-in 4.0207 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.43 0.158 0.173 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rem Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RESA P25321 12 351 351.0 A1JEG:60401 Allosteric Active DFGin 6.1727 14.8814 BLAminus -125.7, 167.74 69.23, 93.16 -97.77, 26.89 271.48, 59.73 -63.11, -29.76 in-in in 9.0438 Saltbr-in 2.7187 HRD-in -87.69, -51.87 66.23, 13.93 in-in-in SNCiii in-in ActLoopNT-in 2.9651 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.16, 154.7 APE9-dihe-na 118.02, 158.85 APE8-dihe-in -77.09, 138.71 APE8-rot-in 297.19 APE67-dihe-in -59.68, -23.56 -52.24, -44.23 APE12-dist-in 8.1974 APE11-dist-in 11.3307 APE10-dist-in 5.7869 APE9-dist-in 4.2474 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.196 0.211 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9res Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RETA P25321 13 351 351.0 A1JEF:60404 Allosteric Active DFGin 6.5025 14.9192 BLAminus -121.64, 161.02 79.66, 89.44 -97.28, 25.84 271.42, 57.67 -59.32, -29.98 in-in in 9.0584 Saltbr-in 2.6884 HRD-in -91.57, -50.28 65.7, 14.34 in-in-in SNCiii in-in ActLoopNT-in 2.9609 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.82, 155.57 APE9-dihe-na 119.38, 155.92 APE8-dihe-in -73.83, 138.5 APE8-rot-in 315.72 APE67-dihe-in -57.32, -25.4 -54.39, -42.36 APE12-dist-in 8.1859 APE11-dist-in 11.4021 APE10-dist-in 5.9522 APE9-dist-in 4.2407 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.75 0.193 0.227 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ret Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N37A P25321 1 351 351.0 8JT:60402,8JT:60403 Allosteric,Allosteric Active DFGin 6.6488 14.4854 BLAminus -123.92, -170.55 59.87, 72.4 -89.59, 22.41 275.2, 67.84 -61.07, -22.15 in-in in 8.6486 Saltbr-in 2.8873 HRD-in -90.3, -49.46 71.47, 2.69 in-in-in SNCiii in-in ActLoopNT-in 2.9099 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.56, 154.71 APE9-dihe-na 136.23, -163.83 APE8-dihe-in -107.21, 128.79 APE8-rot-in 298.22 APE67-dihe-in -60.14, -24.18 -42.74, -52.97 APE12-dist-in 8.5415 APE11-dist-in 11.9362 APE10-dist-in 6.3043 APE9-dist-in 3.975 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.589 0.145 0.167 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n37 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3TA P25321 12 351 351.0 8K2:60401,8K2:60402 Allosteric,Allosteric Active DFGin 6.2089 14.3858 BLAminus -125.21, 167.5 70.97, 90.28 -98.07, 24.21 271.06, 55.85 -60.14, -28.27 in-in in 8.5718 Saltbr-in 2.8524 HRD-in -84.98, -51.06 69.41, 14.03 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.94, 169.7 APE9-dihe-na 118.95, -153.57 APE8-dihe-in -135.51, 135.28 APE8-rot-in 302.46 APE67-dihe-in -63.12, -21.21 -48.68, -48.91 APE12-dist-in 8.1233 APE11-dist-in 11.2089 APE10-dist-in 5.6949 APE9-dist-in 3.706 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.209 0.14 0.157 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3t Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDZA P25321 12 351 351.0 A1JE9:60402,A1JE9:60403 Allosteric,Allosteric Active DFGin 6.37 14.6865 BLAminus -121.86, 166.99 72.88, 89.4 -99.69, 27.1 269.36, 64.25 -60.46, -30.34 in-in in 8.7723 Saltbr-in 2.9001 HRD-in -86.07, -51.02 68.52, 15.31 in-in-in SNCiii in-in ActLoopNT-in 3.0047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.16, 164.09 APE9-dihe-na 123.15, -172.2 APE8-dihe-in -104.62, 134.08 APE8-rot-in 309.64 APE67-dihe-in -61.1, -21.33 -52.23, -44.2 APE12-dist-in 8.2799 APE11-dist-in 11.4033 APE10-dist-in 5.8984 APE9-dist-in 3.9616 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.64 0.18 0.212 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rdz Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REEA P25321 13 351 351.0 A1JEW:60401,A1JEW:60403 Allosteric,Allosteric Active DFGin 6.286 14.26 BLAminus -124.23, 162.89 77.1, 88.42 -96.8, 24.55 273.02, 56.54 -61.31, -24.65 in-in in 8.4623 Saltbr-in 2.9112 HRD-in -83.83, -50.86 69.06, 13.49 in-in-in SNCiii in-in ActLoopNT-in 2.9147 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.82, 159.16 APE9-dihe-na 111.69, 168.82 APE8-dihe-in -86.75, 136.79 APE8-rot-in 296.84 APE67-dihe-in -63.43, -20.25 -47.42, -48.01 APE12-dist-in 8.1052 APE11-dist-in 11.1621 APE10-dist-in 5.684 APE9-dist-in 3.9569 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.34 0.157 0.167 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ree Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RELA P25321 12 351 351.0 D8V:60402,D8V:60403 Allosteric,Allosteric Active DFGin 6.4822 14.5671 BLAminus -123.01, 164.35 74.25, 89.59 -99.6, 28.07 272.56, 59.06 -67.42, -22.86 in-in in 8.6372 Saltbr-in 2.9197 HRD-in -86.71, -52.81 70.71, 15.02 in-in-in SNCiii in-in ActLoopNT-in 2.9775 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.1, 164.56 APE9-dihe-na 121.48, -172.32 APE8-dihe-in -106.43, 133.24 APE8-rot-in 301.52 APE67-dihe-in -61.15, -21.91 -46.09, -49.9 APE12-dist-in 8.3488 APE11-dist-in 11.4781 APE10-dist-in 6.0184 APE9-dist-in 3.9426 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.158 0.177 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rel Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REPA P25321 12 351 351.0 A1JFA:60402,A1JFA:60403,A1JFA:60404 Allosteric,Allosteric,Type1 Active DFGin 6.3781 14.529 BLAminus -120.08, 167.91 74.1, 88.72 -97.52, 23.51 270.46, 58.88 -60.74, -26.54 in-in in 8.6885 Saltbr-in 2.9313 HRD-in -87.33, -51.34 69.9, 12.31 in-in-in SNCiii in-in ActLoopNT-in 2.9651 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.19, 163.24 APE9-dihe-na 117.23, 172.54 APE8-dihe-in -96.3, 137.81 APE8-rot-in 314.32 APE67-dihe-in -63.77, -21.88 -47.87, -48.37 APE12-dist-in 8.1899 APE11-dist-in 11.3609 APE10-dist-in 5.8512 APE9-dist-in 4.0301 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.44 0.157 0.181 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rep Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REOA P25321 13 351 351.0 A1JEJ:60401,A1JEJ:60402,A1JEJ:60403,A1JEJ:60404,A1JEJ:60405 Allosteric,Allosteric,Type1,Type1,Allosteric Active DFGin 6.3145 14.3168 BLAminus -116.84, 173.33 67.79, 85.36 -98.4, 23.6 274.95, 63.33 -57.17, -27.66 in-in in 8.6623 Saltbr-in 2.7528 HRD-in -87.13, -54.16 72.26, 11.26 in-in-in SNCiii in-in ActLoopNT-in 2.8988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.54, 160.85 APE9-dihe-na 115.26, -179.78 APE8-dihe-in -98.51, 134.9 APE8-rot-in 302.45 APE67-dihe-in -59.75, -23.89 -49.35, -45.76 APE12-dist-in 8.1175 APE11-dist-in 11.2447 APE10-dist-in 5.7372 APE9-dist-in 3.9737 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.45 0.152 0.175 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9reo Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7AXVA P25321 1 351 351.0 S95:60401,S95:60402 Allosteric,Type1 Active DFGin 6.5443 14.3191 BLAminus -124.64, 165.56 73.97, 89.92 -106.44, 27.23 290.62, 82.1 -63.98, -25.18 in-in in 9.5168 Saltbr-in 3.1989 HRD-in -92.54, -54.57 72.35, 9.82 in-in-in SNCiii in-in ActLoopNT-in 2.8895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.49, 161.0 APE9-dihe-na 125.29, -162.18 APE8-dihe-in -119.59, 130.9 APE8-rot-in 299.34 APE67-dihe-in -56.02, -27.32 -46.45, -51.94 APE12-dist-in 8.0271 APE11-dist-in 11.475 APE10-dist-in 5.9545 APE9-dist-in 3.8706 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.79 0.2 0.231 A 353.0 344.0 3 25 25 0 [[44, 298]] 1.0 7axv Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE3A P25321 12 351 351.0 A1JE0:60805,A1JE0:60807 Allosteric,Type1 Active DFGin 6.4607 14.6641 BLAminus -120.32, 164.28 77.93, 91.61 -101.65, 25.38 271.39, 59.52 -61.95, -25.41 in-in in 8.7616 Saltbr-in 2.8901 HRD-in -88.06, -50.21 67.37, 14.1 in-in-in SNCiii in-in ActLoopNT-in 3.0126 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.15, 155.76 APE9-dihe-na 126.49, 178.95 APE8-dihe-in -96.29, 137.07 APE8-rot-in 306.5 APE67-dihe-in -59.04, -22.36 -49.62, -47.63 APE12-dist-in 8.2317 APE11-dist-in 11.4892 APE10-dist-in 5.9401 APE9-dist-in 4.1876 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.57 0.185 0.213 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3OA P25321 14 351 351.0 5AO:60403,5AO:60404,5AO:60405 Allosteric,Type1,Allosteric Active DFGin 6.2389 14.3632 BLAminus -124.74, 162.74 72.04, 91.7 -99.25, 24.26 270.68, 57.41 -61.29, -25.0 in-in in 8.56 Saltbr-in 2.8625 HRD-in -84.17, -53.21 70.22, 13.77 in-in-in SNCiii in-in ActLoopNT-in 2.9147 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.1, 167.24 APE9-dihe-na 125.28, -162.2 APE8-dihe-in -119.97, 133.57 APE8-rot-in 304.74 APE67-dihe-in -63.04, -20.65 -49.48, -46.76 APE12-dist-in 8.1083 APE11-dist-in 11.3568 APE10-dist-in 5.8435 APE9-dist-in 3.7337 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.32 0.135 0.158 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 5n3o Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 4WIHA P25321 1 351 351.0 No_ligand No_ligand Active DFGin 6.1605 14.2123 BLAminus -123.3, 174.61 65.19, 98.78 -108.79, 24.75 270.23, 57.89 -53.46, -27.17 in-in in 8.5468 Saltbr-in 2.4651 HRD-in -89.62, -51.49 71.45, 14.2 in-in-in SNCiii in-in ActLoopNT-in 2.9097 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.02, 163.3 APE9-dihe-na 130.98, -159.02 APE8-dihe-in -120.59, 129.78 APE8-rot-in 297.97 APE67-dihe-in -60.37, -23.23 -43.98, -53.0 APE12-dist-in 8.282 APE11-dist-in 11.5665 APE10-dist-in 6.0683 APE9-dist-in 3.608 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.139 0.178 0.191 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 4wih Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0UA P25321 1 351 351.0 No_ligand No_ligand Active DFGin 6.6174 14.7612 BLAminus -120.76, 157.18 78.21, 97.74 -104.6, 26.7 278.38, 71.52 -59.1, -27.35 in-in in 8.7241 Saltbr-in 3.0199 HRD-in -84.58, -52.68 70.27, 15.16 in-in-in SNCiii in-in ActLoopNT-in 2.9195 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.97, 158.74 APE9-dihe-na 125.58, -159.96 APE8-dihe-in -115.4, 133.22 APE8-rot-in 298.31 APE67-dihe-in -57.6, -25.41 -46.26, -52.75 APE12-dist-in 8.2464 APE11-dist-in 11.5188 APE10-dist-in 5.8578 APE9-dist-in 3.5802 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.667 0.154 0.189 A 353.0 347.0 4 25 25 0 [[44, 298]] 1.0 5m0u Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3MA P25321 12 351 351.0 No_ligand No_ligand Active DFGin 6.1801 14.3543 BLAminus -123.75, 157.21 80.77, 89.43 -98.44, 24.43 270.49, 59.51 -61.84, -26.83 in-in in 8.534 Saltbr-in 2.9772 HRD-in -86.44, -51.88 69.6, 14.02 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.37, 162.31 APE9-dihe-na 130.48, -156.87 APE8-dihe-in -124.49, 134.84 APE8-rot-in 297.05 APE67-dihe-in -63.46, -20.29 -50.29, -48.15 APE12-dist-in 8.1166 APE11-dist-in 11.173 APE10-dist-in 5.6762 APE9-dist-in 3.7229 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.229 0.14 0.164 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3m Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EH0A P25321 13 351 351.0 No_ligand No_ligand Active DFGin 6.1366 14.4089 BLAminus -122.27, 162.09 77.35, 95.81 -104.93, 26.7 272.05, 59.25 -60.27, -24.52 in-in in 8.6935 Saltbr-in 3.0251 HRD-in -85.16, -52.91 72.1, 11.56 in-in-in SNCiii in-in ActLoopNT-in 2.9063 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.28, 161.12 APE9-dihe-na 111.18, 173.11 APE8-dihe-in -92.76, 136.72 APE8-rot-in 292.07 APE67-dihe-in -59.99, -23.63 -47.46, -47.75 APE12-dist-in 8.1156 APE11-dist-in 11.2721 APE10-dist-in 5.7898 APE9-dist-in 3.9986 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.49 0.15 0.186 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 6eh0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Z44A P25321 14 351 351.0 No_ligand No_ligand Active DFGin 6.2102 14.4374 BLAminus -128.58, 169.86 73.52, 88.4 -98.57, 23.88 272.06, 58.82 -60.44, -27.11 in-in in 8.6237 Saltbr-in 2.8632 HRD-in -87.15, -51.73 71.04, 12.68 in-in-in SNCiii in-in ActLoopNT-in 2.8909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.29, 164.35 APE9-dihe-na 123.85, -163.53 APE8-dihe-in -119.09, 134.17 APE8-rot-in 300.66 APE67-dihe-in -64.2, -18.89 -49.41, -47.47 APE12-dist-in 8.1442 APE11-dist-in 11.2003 APE10-dist-in 5.6806 APE9-dist-in 3.7234 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.146 0.174 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6z44 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6F14A P25321 9 351 351.0 ISQ:60401 Type1 Active DFGin 6.0674 14.2043 BLAminus -122.05, 170.08 68.01, 92.59 -99.92, 26.02 274.99, 58.24 -62.07, -22.2 in-in in 8.9109 Saltbr-in 2.7518 HRD-in -91.1, -51.98 71.1, 14.05 in-in-in SNCiii in-in ActLoopNT-in 2.9748 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.36, 162.19 APE9-dihe-na 130.64, -162.57 APE8-dihe-in -117.18, 137.06 APE8-rot-in 303.3 APE67-dihe-in -57.84, -25.17 -52.4, -48.63 APE12-dist-in 8.0928 APE11-dist-in 11.4976 APE10-dist-in 5.9364 APE9-dist-in 3.6185 None TPO198,SEP339 TPO198,SEP339 XRAY 1.867 0.176 0.209 A 351.0 339.0 4 25 25 0 [[44, 298]] 1.0 6f14 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCQA P25321 1 351 351.0 6TV:60401 Type1 Active DFGin 6.8807 14.7391 BLAminus -123.17, 161.48 80.79, 88.7 -100.7, 25.58 283.7, 73.56 -69.47, -15.21 in-in in 8.6294 Saltbr-in 2.7912 HRD-in -83.86, -57.44 75.35, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.8709 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.46, 161.6 APE9-dihe-na 121.64, -167.7 APE8-dihe-in -108.93, 132.05 APE8-rot-in 299.43 APE67-dihe-in -61.12, -21.5 -46.6, -52.1 APE12-dist-in 8.2733 APE11-dist-in 11.3689 APE10-dist-in 5.7633 APE9-dist-in 3.5302 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.423 0.143 0.171 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcq Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0BA P25321 1 351 351.0 IQU:60401 Type1 Active DFGin 6.8813 14.7187 BLAminus -123.22, 164.24 73.76, 92.16 -102.04, 24.7 282.81, 75.1 -69.51, -12.32 in-in in 8.6655 Saltbr-in 2.839 HRD-in -84.13, -55.97 72.34, 13.7 in-in-in SNCiii in-in ActLoopNT-in 2.9176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.89, 160.72 APE9-dihe-na 119.74, -166.42 APE8-dihe-in -108.36, 130.85 APE8-rot-in 297.35 APE67-dihe-in -58.39, -24.4 -45.39, -52.68 APE12-dist-in 8.3169 APE11-dist-in 11.472 APE10-dist-in 5.863 APE9-dist-in 3.5368 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.506 0.133 0.159 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m0b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0CA P25321 14 351 351.0 7CB:60401 Type1 Active DFGin 5.9263 14.302 BLAminus -122.77, 175.08 63.79, 89.7 -99.98, 24.75 269.77, 55.83 -60.58, -26.96 in-in in 8.883 Saltbr-in 2.7611 HRD-in -96.62, -51.29 71.36, 13.59 in-in-in SNCiii in-in ActLoopNT-in 2.8962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.73, 162.77 APE9-dihe-na 130.88, -158.33 APE8-dihe-in -121.3, 136.16 APE8-rot-in 298.59 APE67-dihe-in -56.27, -24.31 -50.24, -49.98 APE12-dist-in 8.0159 APE11-dist-in 11.4298 APE10-dist-in 5.8568 APE9-dist-in 3.4765 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.734 0.174 0.2 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 5m0c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1EA P25321 1 351 351.0 9NT:60402 Type1 Active DFGin 6.2704 14.3856 BLAminus -116.94, 171.55 65.1, 106.63 -111.97, 27.73 271.53, 67.85 -63.72, -19.43 in-in in 8.7187 Saltbr-in 3.0209 HRD-in -91.36, -50.95 71.95, 7.79 in-in-in SNCiii in-in ActLoopNT-in 2.9009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.29, 159.66 APE9-dihe-na 132.29, -165.21 APE8-dihe-in -107.94, 127.91 APE8-rot-in 298.37 APE67-dihe-in -61.69, -23.48 -42.18, -52.19 APE12-dist-in 8.4675 APE11-dist-in 11.8233 APE10-dist-in 6.2637 APE9-dist-in 3.8458 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.529 0.149 0.174 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 5n1e Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1LA P25321 1 351 351.0 47V:60401 Type1 Active DFGin 6.396 14.532 BLAminus -123.64, 176.95 64.79, 82.82 -93.93, 24.8 274.07, 62.39 -62.6, -22.74 in-in in 8.8226 Saltbr-in 2.8025 HRD-in -94.52, -51.37 72.06, 10.31 in-in-in SNCiii in-in ActLoopNT-in 2.9192 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.16, 159.72 APE9-dihe-na 135.69, -163.33 APE8-dihe-in -113.56, 130.78 APE8-rot-in 299.09 APE67-dihe-in -60.45, -22.24 -43.7, -53.93 APE12-dist-in 8.2602 APE11-dist-in 11.6708 APE10-dist-in 6.1348 APE9-dist-in 3.8023 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.489 0.144 0.175 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n1l Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1MA P25321 1 351 351.0 BJK:60403 Type1 Active DFGin 6.4585 14.0437 BLAminus -123.41, 174.5 65.19, 101.23 -111.22, 25.09 279.28, 68.63 -59.82, -25.41 in-in in 8.6556 Saltbr-in 3.1051 HRD-in -94.95, -53.6 73.25, 11.15 in-in-in SNCiii in-in ActLoopNT-in 2.9046 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.71, 160.83 APE9-dihe-na 133.31, -164.27 APE8-dihe-in -112.16, 130.84 APE8-rot-in 297.89 APE67-dihe-in -59.92, -22.11 -42.38, -54.95 APE12-dist-in 8.3624 APE11-dist-in 11.6972 APE10-dist-in 6.1444 APE9-dist-in 3.7347 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.436 0.153 0.17 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n1m Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1OA P25321 8 351 351.0 8GB:60402 Type1 Active DFGin 6.3495 14.2152 BLAminus -117.96, -179.86 55.4, 87.26 -94.87, 24.62 276.45, 65.75 -58.72, -27.08 in-in in 8.7307 Saltbr-in 2.9049 HRD-in -90.93, -54.44 74.01, 7.31 in-in-in SNCiii in-in ActLoopNT-in 2.8232 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.08, 159.92 APE9-dihe-na 129.4, -159.5 APE8-dihe-in -111.79, 132.44 APE8-rot-in 298.64 APE67-dihe-in -59.59, -24.34 -46.73, -53.55 APE12-dist-in 8.262 APE11-dist-in 11.7101 APE10-dist-in 6.159 APE9-dist-in 3.7466 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.8 0.172 0.191 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1o Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N33A P25321 1 351 351.0 8JW:60401 Type1 Active DFGin 6.5966 14.3444 BLAminus -124.76, 172.62 66.0, 85.95 -97.34, 23.47 278.51, 67.69 -61.06, -25.74 in-in in 8.6169 Saltbr-in 2.8295 HRD-in -95.51, -52.3 69.58, 12.9 in-in-in SNCiii in-in ActLoopNT-in 2.9142 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.48, 158.46 APE9-dihe-na 134.35, -163.32 APE8-dihe-in -113.73, 130.26 APE8-rot-in 298.83 APE67-dihe-in -60.31, -22.81 -43.61, -54.33 APE12-dist-in 8.2362 APE11-dist-in 11.6201 APE10-dist-in 6.0809 APE9-dist-in 3.77 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.434 0.151 0.174 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n33 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N36A P25321 1 351 351.0 F05:60402 Type1 Active DFGin 6.5556 14.4334 BLAminus -119.92, -178.94 65.61, 75.08 -89.84, 25.76 275.95, 67.66 -63.27, -22.33 in-in in 8.7237 Saltbr-in 2.8129 HRD-in -93.71, -55.54 73.48, 11.23 in-in-in SNCiii in-in ActLoopNT-in 2.9179 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 158.13 APE9-dihe-na 133.34, -160.6 APE8-dihe-in -112.55, 130.07 APE8-rot-in 300.31 APE67-dihe-in -59.23, -24.07 -46.06, -53.12 APE12-dist-in 8.5382 APE11-dist-in 11.8304 APE10-dist-in 6.244 APE9-dist-in 3.8446 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.15 0.186 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n36 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N39A P25321 1 351 351.0 8LZ:60401 Type1 Active DFGin 6.447 14.1735 BLAminus -115.61, 178.64 62.65, 78.33 -93.23, 24.2 279.01, 65.77 -60.59, -24.07 in-in in 8.6058 Saltbr-in 2.9559 HRD-in -92.08, -52.71 73.17, 11.28 in-in-in SNCiii in-in ActLoopNT-in 2.9039 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.98, 161.14 APE9-dihe-na 131.91, -164.98 APE8-dihe-in -111.15, 130.71 APE8-rot-in 297.72 APE67-dihe-in -61.9, -21.74 -44.77, -52.6 APE12-dist-in 8.3392 APE11-dist-in 11.723 APE10-dist-in 6.1957 APE9-dist-in 3.7478 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.45 0.146 0.169 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n39 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3AA P25321 1 351 351.0 46P:60404 Type1 Active DFGin 6.2347 14.3651 BLAminus -119.17, -176.19 62.26, 81.42 -92.16, 24.71 273.8, 62.92 -62.87, -20.2 in-in in 8.749 Saltbr-in 2.7586 HRD-in -88.58, -51.45 73.7, 4.67 in-in-in SNCiii in-in ActLoopNT-in 2.9097 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.23, 158.77 APE9-dihe-na 132.44, -163.77 APE8-dihe-in -109.48, 129.54 APE8-rot-in 298.98 APE67-dihe-in -60.34, -22.78 -43.75, -54.33 APE12-dist-in 8.4518 APE11-dist-in 11.8624 APE10-dist-in 6.299 APE9-dist-in 3.8633 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.404 0.162 0.184 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5n3a Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3BA P25321 5 351 351.0 BJN:60402 Type1 Active DFGin 6.5927 14.4491 BLAminus -127.99, -176.28 55.77, 87.43 -96.19, 25.66 273.47, 67.97 -63.99, -23.38 in-in in 8.7554 Saltbr-in 2.8962 HRD-in -88.77, -50.71 72.06, 10.59 in-in-in SNCiii in-in ActLoopNT-in 2.9448 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.08, 159.78 APE9-dihe-na 131.61, -163.96 APE8-dihe-in -108.68, 131.24 APE8-rot-in 297.72 APE67-dihe-in -59.88, -25.39 -45.07, -52.54 APE12-dist-in 8.4797 APE11-dist-in 11.8507 APE10-dist-in 6.2466 APE9-dist-in 3.8182 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.64 0.169 0.19 A 353.0 346.0 0 25 25 0 [[44, 298]] 1.0 5n3b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3CA P25321 1 351 351.0 8M2:60401 Type1 Active DFGin 6.4695 14.5593 BLAminus -119.65, -170.8 58.89, 76.61 -92.51, 23.35 273.34, 68.51 -61.87, -22.49 in-in in 8.8718 Saltbr-in 2.5903 HRD-in -86.05, -52.6 72.82, 4.64 in-in-in SNCiii in-in ActLoopNT-in 2.9083 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.17, 154.54 APE9-dihe-na 137.81, -166.64 APE8-dihe-in -107.38, 129.58 APE8-rot-in 301.23 APE67-dihe-in -60.59, -21.91 -48.15, -49.13 APE12-dist-in 8.4988 APE11-dist-in 11.881 APE10-dist-in 6.313 APE9-dist-in 3.9442 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.772 0.179 0.196 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 5n3c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3EA P25321 1 351 351.0 46L:60401 Type1 Active DFGin 6.3638 14.5063 BLAminus -127.71, 175.81 62.83, 90.97 -100.32, 25.03 271.8, 65.14 -62.05, -22.27 in-in in 8.7408 Saltbr-in 2.7088 HRD-in -91.8, -51.14 70.51, 10.68 in-in-in SNCiii in-in ActLoopNT-in 2.9031 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.84, 159.06 APE9-dihe-na 132.58, -164.21 APE8-dihe-in -109.56, 127.56 APE8-rot-in 297.32 APE67-dihe-in -58.87, -22.91 -42.91, -53.84 APE12-dist-in 8.3507 APE11-dist-in 11.7235 APE10-dist-in 6.2032 APE9-dist-in 3.8527 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.529 0.157 0.185 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 5n3e Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3HA P25321 12 351 351.0 NCA:60401 Type1 Active DFGin 6.1319 14.3906 BLAminus -122.6, -180.0 63.23, 82.13 -91.36, 22.79 272.99, 56.19 -60.14, -26.14 in-in in 8.7514 Saltbr-in 2.6589 HRD-in -87.2, -51.58 72.04, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.9341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.37, 162.08 APE9-dihe-na 126.78, -160.11 APE8-dihe-in -123.99, 135.79 APE8-rot-in 303.45 APE67-dihe-in -61.89, -20.7 -47.97, -49.67 APE12-dist-in 8.1151 APE11-dist-in 11.2119 APE10-dist-in 5.6695 APE9-dist-in 3.6645 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.36 0.146 0.174 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3h Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3LA P25321 12 351 351.0 E5E:60403 Type1 Active DFGin 6.2595 14.3638 BLAminus -110.0, -170.99 60.26, 70.6 -90.47, 19.96 272.32, 58.23 -61.45, -24.06 in-in in 8.5405 Saltbr-in 2.6938 HRD-in -90.35, -53.09 72.54, 14.7 in-in-in SNCiii in-in ActLoopNT-in 2.9233 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.08, 164.02 APE9-dihe-na 125.78, -157.28 APE8-dihe-in -125.93, 133.76 APE8-rot-in 301.3 APE67-dihe-in -63.07, -21.0 -46.88, -49.04 APE12-dist-in 8.0924 APE11-dist-in 11.2426 APE10-dist-in 5.7077 APE9-dist-in 3.6875 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.38 0.131 0.16 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3l Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3PA P25321 13 351 351.0 5H1:60403 Type1 Active DFGin 6.2436 14.5023 BLAminus -127.2, 167.3 74.22, 87.87 -97.57, 26.23 270.81, 60.43 -61.56, -25.66 in-in in 8.7311 Saltbr-in 2.7657 HRD-in -85.65, -51.7 69.95, 15.28 in-in-in SNCiii in-in ActLoopNT-in 2.9111 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.51, 162.3 APE9-dihe-na 120.29, -172.77 APE8-dihe-in -106.79, 135.49 APE8-rot-in 306.73 APE67-dihe-in -58.76, -22.92 -47.58, -49.08 APE12-dist-in 8.0501 APE11-dist-in 11.1792 APE10-dist-in 5.6741 APE9-dist-in 3.8219 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.159 0.181 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5n3p Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N7PA P25321 1 351 351.0 E9Q:60401 Type1 Active DFGin 6.2715 14.2377 BLAminus -126.92, 176.32 67.6, 84.98 -97.07, 24.3 276.23, 67.65 -61.77, -20.94 in-in in 8.7682 Saltbr-in 2.9318 HRD-in -90.6, -51.66 69.11, 10.85 in-in-in SNCiii in-in ActLoopNT-in 2.891 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.85, 157.28 APE9-dihe-na 137.17, -163.84 APE8-dihe-in -109.53, 129.55 APE8-rot-in 298.93 APE67-dihe-in -61.19, -22.41 -45.09, -51.76 APE12-dist-in 8.4123 APE11-dist-in 11.794 APE10-dist-in 6.2631 APE9-dist-in 3.8866 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.501 0.161 0.186 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5n7p Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N7UA P25321 1 351 351.0 8PQ:60402 Type1 Active DFGin 6.205 14.2991 BLAminus -120.54, 174.37 71.79, 80.65 -93.18, 24.34 271.72, 64.53 -61.67, -22.3 in-in in 8.6689 Saltbr-in 2.7302 HRD-in -88.01, -52.02 72.42, 9.42 in-in-in SNCiii in-in ActLoopNT-in 2.9076 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.34, 159.87 APE9-dihe-na 134.15, -161.5 APE8-dihe-in -113.47, 128.55 APE8-rot-in 298.53 APE67-dihe-in -62.45, -22.0 -41.16, -54.39 APE12-dist-in 8.4156 APE11-dist-in 11.6964 APE10-dist-in 6.1531 APE9-dist-in 3.7318 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.371 0.162 0.177 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5n7u Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EM2A P25321 12 351 351.0 M77:60401 Type1 Active DFGin 6.0983 14.5142 BLAminus -119.73, 168.43 71.45, 87.62 -96.71, 20.34 273.03, 58.25 -60.57, -24.08 in-in in 8.84 Saltbr-in 2.6697 HRD-in -89.33, -54.43 71.02, 10.57 in-in-in SNCiii in-in ActLoopNT-in 2.9443 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.33, 158.5 APE9-dihe-na 116.31, 173.93 APE8-dihe-in -92.1, 134.84 APE8-rot-in 313.8 APE67-dihe-in -63.32, -22.08 -46.46, -47.85 APE12-dist-in 8.0646 APE11-dist-in 11.2814 APE10-dist-in 5.8035 APE9-dist-in 4.0387 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.3 0.133 0.152 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6em2 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPSA P25321 14 351 351.0 LR5:60403 Type1 Active DFGin 6.2417 14.3836 BLAminus -118.18, 155.69 80.72, 97.49 -102.89, 27.66 269.68, 53.66 -61.81, -26.65 in-in in 8.4713 Saltbr-in 2.769 HRD-in -87.72, -49.97 68.25, 13.7 in-in-in SNCiii in-in ActLoopNT-in 2.9052 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.63, 162.08 APE9-dihe-na 121.79, -175.33 APE8-dihe-in -105.81, 135.65 APE8-rot-in 306.18 APE67-dihe-in -63.55, -22.05 -51.22, -42.77 APE12-dist-in 8.112 APE11-dist-in 11.235 APE10-dist-in 5.7263 APE9-dist-in 3.9626 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.65 0.188 0.223 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6sps Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPYA P25321 14 351 351.0 LR8:60401 Type1 Active DFGin 6.2185 14.4051 BLAminus -123.39, 156.64 76.95, 93.24 -100.34, 25.16 268.44, 60.17 -60.59, -28.29 in-in in 8.5574 Saltbr-in 2.8857 HRD-in -87.4, -50.43 70.53, 14.04 in-in-in SNCiii in-in ActLoopNT-in 2.9355 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.4, 165.8 APE9-dihe-na 119.26, -168.59 APE8-dihe-in -114.24, 137.53 APE8-rot-in 310.43 APE67-dihe-in -58.09, -22.25 -52.05, -47.82 APE12-dist-in 8.0826 APE11-dist-in 11.1688 APE10-dist-in 5.6662 APE9-dist-in 3.7027 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.6 0.162 0.182 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6spy Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SQ1A P25321 14 351 351.0 LRT:60403 Type1 Active DFGin 6.2159 14.2505 BLAminus -121.79, 172.1 69.1, 85.08 -99.08, 24.56 277.81, 66.67 -63.84, -22.93 in-in in 8.6518 Saltbr-in 2.6996 HRD-in -89.13, -55.11 71.03, 9.14 in-in-in SNCiii in-in ActLoopNT-in 2.9507 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.84, 157.22 APE9-dihe-na 133.4, -154.71 APE8-dihe-in -125.36, 134.74 APE8-rot-in 298.73 APE67-dihe-in -64.25, -21.15 -48.42, -47.94 APE12-dist-in 7.9507 APE11-dist-in 11.2453 APE10-dist-in 5.8092 APE9-dist-in 3.9436 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.49 0.144 0.177 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6sq1 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y05A P25321 8 351 351.0 ADE:60401 Type1 Active DFGin 6.2038 13.15 BLAminus -122.62, 176.1 60.39, 98.08 -109.84, 29.54 293.58, 72.67 -62.59, -23.96 in-in in 8.9695 Saltbr-in 2.6495 HRD-in -91.46, -52.85 71.13, 13.97 in-in-in SNCiii in-in ActLoopNT-in 2.944 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.05, 162.66 APE9-dihe-na 130.15, -156.07 APE8-dihe-in -123.62, 136.19 APE8-rot-in 301.3 APE67-dihe-in -59.67, -24.1 -52.64, -47.85 APE12-dist-in 8.102 APE11-dist-in 11.5295 APE10-dist-in 5.9277 APE9-dist-in 3.5458 None TPO198,SEP339 TPO198,SEP339 XRAY 1.7 0.178 0.205 A 353.0 344.0 0 25 25 0 [[44, 298]] 1.0 6y05 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y89A P25321 11 351 351.0 OGB:60401 Type1 Active DFGin 5.8698 14.4362 BLAminus -122.55, 174.87 63.65, 84.21 -93.51, 25.44 274.84, 60.12 -60.56, -27.02 in-in in 9.0446 Saltbr-in 2.6615 HRD-in -89.79, -53.04 71.39, 13.28 in-in-in SNCiii in-in ActLoopNT-in 2.8959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.08, 161.18 APE9-dihe-na 130.37, -156.13 APE8-dihe-in -122.12, 132.52 APE8-rot-in 297.86 APE67-dihe-in -57.82, -25.35 -46.57, -49.91 APE12-dist-in 8.0645 APE11-dist-in 11.5446 APE10-dist-in 5.9255 APE9-dist-in 3.5915 None TPO198,SEP339 TPO198,SEP339 XRAY 1.56 0.17 0.192 A 353.0 339.0 2 25 25 0 [[44, 298]] 1.0 6y89 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNAA P25321 1 351 351.0 M77:60402 Type1 Active DFGin 6.2016 14.3343 BLAminus -119.96, 179.81 63.19, 78.66 -92.28, 22.25 273.96, 61.01 -60.67, -22.0 in-in in 8.696 Saltbr-in 2.6397 HRD-in -90.85, -54.18 73.93, 11.37 in-in-in SNCiii in-in ActLoopNT-in 2.9234 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.28, 159.25 APE9-dihe-na 133.12, -164.07 APE8-dihe-in -114.68, 130.03 APE8-rot-in 297.53 APE67-dihe-in -61.88, -21.65 -45.58, -51.04 APE12-dist-in 8.2756 APE11-dist-in 11.6374 APE10-dist-in 6.1355 APE9-dist-in 3.7647 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.47 0.165 0.189 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6yna Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNBA P25321 1 351 351.0 IQU:60401 Type1 Active DFGin 6.3631 14.3492 BLAminus -116.44, -174.16 61.98, 75.89 -98.12, 21.41 275.26, 66.86 -65.3, -20.05 in-in in 8.6085 Saltbr-in 2.4589 HRD-in -95.93, -55.57 72.9, 13.24 in-in-in SNCiii in-in ActLoopNT-in 2.8713 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.81, 160.16 APE9-dihe-na 137.96, -159.84 APE8-dihe-in -118.76, 130.24 APE8-rot-in 299.49 APE67-dihe-in -60.0, -21.74 -44.91, -52.44 APE12-dist-in 8.0367 APE11-dist-in 11.4934 APE10-dist-in 6.0621 APE9-dist-in 3.7628 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.72 0.158 0.201 A 353.0 347.0 1 25 25 0 [[44, 298]] 1.0 6ynb Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNCA P25321 1 351 351.0 7CT:60401 Type1 Active DFGin 6.0405 14.5355 BLAminus -120.79, 169.65 71.14, 83.37 -95.82, 21.95 274.39, 61.02 -58.31, -26.55 in-in in 8.8468 Saltbr-in 2.5305 HRD-in -88.43, -56.03 72.64, 13.22 in-in-in SNCiii in-in ActLoopNT-in 2.9309 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.35, 158.03 APE9-dihe-na 138.45, -155.36 APE8-dihe-in -121.88, 130.9 APE8-rot-in 297.76 APE67-dihe-in -61.6, -20.8 -45.0, -53.23 APE12-dist-in 8.1381 APE11-dist-in 11.5595 APE10-dist-in 6.0828 APE9-dist-in 3.6746 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.4 0.15 0.173 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 6ync Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNRA P25321 11 351 351.0 O72:60403 Type1 Active DFGin 5.8353 14.1484 BLAminus -121.49, -178.1 59.21, 91.48 -99.82, 25.19 274.78, 55.92 -59.5, -24.95 in-in in 9.0384 Saltbr-in 2.6099 HRD-in -85.88, -50.99 69.33, 11.34 in-in-in SNCiii in-in ActLoopNT-in 2.8951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.62, 159.23 APE9-dihe-na 131.94, -160.26 APE8-dihe-in -120.46, 134.53 APE8-rot-in 302.96 APE67-dihe-in -61.79, -24.17 -46.56, -49.51 APE12-dist-in 8.1163 APE11-dist-in 11.3885 APE10-dist-in 5.8269 APE9-dist-in 3.616 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.9 0.189 0.221 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6ynr Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YNTA P25321 6 351 351.0 LRT:60405 Type1 Active DFGin 6.0242 14.3498 BLAminus -127.88, -176.71 61.66, 78.46 -90.86, 25.34 272.68, 60.44 -59.78, -24.31 in-in in 9.06 Saltbr-in 2.6983 HRD-in -92.67, -53.37 74.33, 11.71 in-in-in SNCiii in-in ActLoopNT-in 2.9262 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.24, 160.78 APE9-dihe-na 130.38, -159.85 APE8-dihe-in -120.86, 135.61 APE8-rot-in 299.16 APE67-dihe-in -60.2, -23.36 -47.55, -51.43 APE12-dist-in 8.1139 APE11-dist-in 11.3697 APE10-dist-in 5.8425 APE9-dist-in 3.5589 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.52 0.171 0.191 A 353.0 346.0 0 25 25 0 [[44, 298]] 1.0 6ynt Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YOUA P25321 14 351 351.0 P4Q:60401 Type1 Active DFGin 6.1964 14.3182 BLAminus -120.09, 165.39 72.67, 93.33 -100.94, 27.48 272.8, 57.34 -61.54, -27.01 in-in in 8.6014 Saltbr-in 2.6137 HRD-in -87.37, -52.03 71.03, 15.52 in-in-in SNCiii in-in ActLoopNT-in 2.9619 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.59, 163.46 APE9-dihe-na 118.27, -170.34 APE8-dihe-in -109.65, 135.96 APE8-rot-in 311.42 APE67-dihe-in -62.17, -24.35 -52.31, -42.25 APE12-dist-in 8.0511 APE11-dist-in 11.1756 APE10-dist-in 5.7123 APE9-dist-in 3.7508 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.73 0.181 0.216 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6you Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YPPA P25321 13 351 351.0 ISQ:60401 Type1 Active DFGin 6.575 13.8991 BLAminus -125.47, 168.17 69.21, 91.25 -102.12, 26.99 282.19, 66.61 -59.38, -28.47 in-in in 8.4767 Saltbr-in 2.8285 HRD-in -95.67, -54.73 76.34, 8.75 in-in-in SNCiii in-in ActLoopNT-in 2.9182 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.07, 157.89 APE9-dihe-na 135.57, -161.87 APE8-dihe-in -121.03, 135.18 APE8-rot-in 300.65 APE67-dihe-in -60.09, -21.93 -50.41, -52.89 APE12-dist-in 8.005 APE11-dist-in 11.2134 APE10-dist-in 5.7336 APE9-dist-in 3.8634 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.75 0.179 0.203 A 353.0 337.0 2 25 25 0 [[44, 298]] 1.0 6ypp Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YPSA P25321 14 351 351.0 P72:60402 Type1 Active DFGin 6.1571 14.3301 BLAminus -118.18, 171.85 69.73, 80.92 -91.01, 22.0 274.81, 61.35 -59.17, -25.98 in-in in 8.6264 Saltbr-in 2.7911 HRD-in -86.09, -50.96 68.81, 12.1 in-in-in SNCiii in-in ActLoopNT-in 2.9233 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.88, 163.19 APE9-dihe-na 126.1, -161.8 APE8-dihe-in -121.09, 134.4 APE8-rot-in 301.85 APE67-dihe-in -62.56, -20.95 -48.37, -48.27 APE12-dist-in 8.0941 APE11-dist-in 11.1937 APE10-dist-in 5.6911 APE9-dist-in 3.7621 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.35 0.145 0.157 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6yps Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YQIA P25321 1 351 351.0 6TV:60401 Type1 Active DFGin 6.6225 13.8594 BLAminus -120.83, 174.85 73.2, 74.9 -95.37, 21.17 285.79, 72.27 -63.44, -25.21 in-in in 8.555 Saltbr-in 2.8726 HRD-in -91.67, -56.05 72.65, 12.52 in-in-in SNCiii in-in ActLoopNT-in 2.9283 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.98, 159.1 APE9-dihe-na 134.75, -160.96 APE8-dihe-in -117.42, 130.5 APE8-rot-in 297.87 APE67-dihe-in -60.26, -23.17 -43.79, -54.04 APE12-dist-in 8.0852 APE11-dist-in 11.5282 APE10-dist-in 6.0526 APE9-dist-in 3.7076 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.42 0.155 0.18 A 353.0 345.0 3 25 25 0 [[44, 298]] 1.0 6yqi Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YQJA P25321 1 351 351.0 6TX:60401 Type1 Active DFGin 6.536 14.0021 BLAminus -124.1, 170.97 64.75, 82.67 -94.0, 24.22 278.04, 68.57 -64.35, -18.91 in-in in 8.3434 Saltbr-in 2.8114 HRD-in -94.88, -53.22 71.62, 13.76 in-in-in SNCiii in-in ActLoopNT-in 2.9414 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.32, 160.29 APE9-dihe-na 132.83, -156.0 APE8-dihe-in -122.12, 131.13 APE8-rot-in 297.37 APE67-dihe-in -59.98, -22.93 -46.61, -53.18 APE12-dist-in 8.1341 APE11-dist-in 11.5405 APE10-dist-in 6.0266 APE9-dist-in 3.5883 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.16 0.201 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 6yqj Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YQKA P25321 1 351 351.0 7KB:60401 Type1 Active DFGin 6.3842 14.635 BLAminus -116.26, -173.03 63.61, 71.29 -93.36, 20.28 275.04, 72.25 -62.95, -24.83 in-in in 9.2842 Saltbr-in 2.5172 HRD-in -89.64, -52.45 71.24, 12.44 in-in-in SNCiii in-in ActLoopNT-in 2.9122 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.58, 159.9 APE9-dihe-na 130.2, -161.78 APE8-dihe-in -114.54, 132.23 APE8-rot-in 297.68 APE67-dihe-in -62.46, -19.69 -47.44, -50.59 APE12-dist-in 8.2392 APE11-dist-in 11.6243 APE10-dist-in 6.1043 APE9-dist-in 3.8152 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.67 0.167 0.202 A 353.0 344.0 5 25 25 0 [[44, 298]] 1.0 6yqk Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7AXTA P25321 1 351 351.0 S9B:60401 Type1 Active DFGin 6.7184 14.8628 BLAminus -127.34, 164.32 75.46, 88.44 -100.63, 25.42 283.48, 72.18 -68.02, -22.42 in-in in 9.1968 Saltbr-in 3.149 HRD-in -87.43, -53.85 74.57, 8.03 in-in-in SNCiii in-in ActLoopNT-in 2.8964 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.36, 157.27 APE9-dihe-na 128.21, -163.37 APE8-dihe-in -115.52, 132.73 APE8-rot-in 300.39 APE67-dihe-in -59.29, -20.86 -48.29, -50.7 APE12-dist-in 8.1621 APE11-dist-in 11.401 APE10-dist-in 5.8203 APE9-dist-in 3.6485 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.86 0.189 0.226 A 353.0 342.0 5 25 25 0 [[44, 298]] 1.0 7axt Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7BARA P25321 14 351 351.0 T82:60401 Type1 Active DFGin 6.3379 14.4805 BLAminus -129.87, -171.42 62.69, 72.07 -89.88, 23.39 274.09, 65.5 -62.66, -24.64 in-in in 8.7197 Saltbr-in 2.8384 HRD-in -88.26, -52.14 74.09, 12.92 in-in-in SNCiii in-in ActLoopNT-in 2.9197 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.3, 163.6 APE9-dihe-na 129.58, -156.99 APE8-dihe-in -128.55, 134.3 APE8-rot-in 298.64 APE67-dihe-in -61.2, -20.19 -50.31, -49.26 APE12-dist-in 8.0904 APE11-dist-in 11.2272 APE10-dist-in 5.7202 APE9-dist-in 3.6557 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.37 0.153 0.179 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 7bar Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIHA P25321 1 351 351.0 7QW:60401 Type1 Active DFGin 6.6112 14.7767 BLAminus -121.61, 158.3 80.03, 88.23 -96.87, 22.43 285.52, 80.97 -63.48, -26.52 in-in in 9.1964 Saltbr-in 3.0815 HRD-in -85.1, -53.84 72.68, 6.07 in-in-in SNCiii in-in ActLoopNT-in 2.9353 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.04, 157.29 APE9-dihe-na 126.06, -165.16 APE8-dihe-in -115.66, 135.76 APE8-rot-in 299.21 APE67-dihe-in -61.29, -23.28 -48.22, -51.33 APE12-dist-in 8.4106 APE11-dist-in 11.5423 APE10-dist-in 5.9635 APE9-dist-in 3.7416 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.374 0.14 0.157 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pih Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDXA P25321 12 351 351.0 A1JE5:60406 Type1 Active DFGin 6.3947 14.5159 BLAminus -120.9, 176.38 62.83, 88.27 -100.01, 26.71 273.66, 64.38 -63.82, -25.52 in-in in 8.7161 Saltbr-in 2.9652 HRD-in -95.33, -53.05 70.61, 15.96 in-in-in SNCiii in-in ActLoopNT-in 3.0157 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.31, 161.4 APE9-dihe-na 124.9, -173.36 APE8-dihe-in -106.08, 132.1 APE8-rot-in 308.01 APE67-dihe-in -62.99, -20.07 -49.55, -46.7 APE12-dist-in 8.2468 APE11-dist-in 11.4052 APE10-dist-in 5.9001 APE9-dist-in 4.0415 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.193 0.208 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rdx Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE6A P25321 13 351 351.0 A1JEX:60605 Type1 Active DFGin 6.4398 14.6332 BLAminus -123.71, 169.54 74.02, 90.92 -99.73, 23.54 270.67, 62.64 -62.18, -25.3 in-in in 8.7272 Saltbr-in 2.9096 HRD-in -86.3, -51.47 69.33, 11.7 in-in-in SNCiii in-in ActLoopNT-in 2.9767 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.91, 159.32 APE9-dihe-na 117.99, 172.79 APE8-dihe-in -90.66, 139.04 APE8-rot-in 307.68 APE67-dihe-in -64.33, -21.04 -49.6, -45.84 APE12-dist-in 8.1212 APE11-dist-in 11.3054 APE10-dist-in 5.7928 APE9-dist-in 3.9602 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.45 0.177 0.194 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9re6 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RENA P25321 13 351 351.0 A1JEK:60401 Type1 Active DFGin 6.2639 14.538 BLAminus -125.36, 166.83 70.47, 89.12 -96.27, 20.46 272.82, 57.42 -59.85, -25.61 in-in in 8.7615 Saltbr-in 2.7947 HRD-in -89.58, -52.32 70.81, 11.76 in-in-in SNCiii in-in ActLoopNT-in 2.8858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.72, 157.64 APE9-dihe-na 115.87, 172.3 APE8-dihe-in -88.32, 133.56 APE8-rot-in 293.26 APE67-dihe-in -60.41, -22.75 -46.56, -47.75 APE12-dist-in 7.9097 APE11-dist-in 11.1788 APE10-dist-in 5.6755 APE9-dist-in 4.059 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.16 0.181 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ren Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REQA P25321 13 351 351.0 A1JEI:60402 Type1 Active DFGin 6.494 14.6379 BLAminus -119.67, 172.96 64.34, 87.39 -94.55, 24.82 273.79, 57.22 -60.93, -26.75 in-in in 8.8075 Saltbr-in 2.8045 HRD-in -85.13, -51.31 68.74, 14.76 in-in-in SNCiii in-in ActLoopNT-in 2.9545 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.42, 156.59 APE9-dihe-na 122.72, 176.53 APE8-dihe-in -91.46, 139.22 APE8-rot-in 321.17 APE67-dihe-in -64.4, -18.2 -52.5, -47.28 APE12-dist-in 8.1908 APE11-dist-in 11.3155 APE10-dist-in 5.8314 APE9-dist-in 4.0262 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.19 0.225 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9req Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RERA P25321 13 351 351.0 A1JEH:60401 Type1 Active DFGin 6.3318 14.5099 BLAminus -119.15, -175.34 54.86, 83.32 -93.03, 23.56 273.62, 62.86 -62.47, -23.85 in-in in 8.7329 Saltbr-in 2.8226 HRD-in -86.33, -53.68 72.65, 12.74 in-in-in SNCiii in-in ActLoopNT-in 2.9096 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.6, 159.26 APE9-dihe-na 118.95, -179.09 APE8-dihe-in -98.87, 134.79 APE8-rot-in 304.07 APE67-dihe-in -61.62, -21.03 -49.43, -46.1 APE12-dist-in 8.1931 APE11-dist-in 11.2928 APE10-dist-in 5.7953 APE9-dist-in 4.0229 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.45 0.179 0.198 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rer Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M0LA P25321 12 351 351.0 7CT:60401,7CT:60402 Type1,Allosteric Active DFGin 5.8124 14.412 BLAminus -125.24, 171.39 72.54, 82.78 -94.45, 21.51 274.7, 58.82 -58.96, -27.86 in-in in 8.9632 Saltbr-in 2.5902 HRD-in -93.78, -54.2 73.09, 11.9 in-in-in SNCiii in-in ActLoopNT-in 2.9318 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.09, 160.85 APE9-dihe-na 134.16, -158.05 APE8-dihe-in -124.56, 135.24 APE8-rot-in 298.63 APE67-dihe-in -59.22, -23.14 -48.63, -50.91 APE12-dist-in 7.9743 APE11-dist-in 11.3295 APE10-dist-in 5.7609 APE9-dist-in 3.6509 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.465 0.153 0.173 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5m0l Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5MHIA P25321 1 351 351.0 7N9:60402,7N9:60403 Type1,Allosteric Active DFGin 6.5271 14.3646 BLAminus -123.97, 171.25 68.38, 93.75 -105.37, 25.41 275.2, 68.89 -61.8, -24.18 in-in in 8.6749 Saltbr-in 2.887 HRD-in -89.75, -51.15 72.09, 10.68 in-in-in SNCiii in-in ActLoopNT-in 2.9159 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.87, 159.66 APE9-dihe-na 135.33, -164.35 APE8-dihe-in -111.34, 128.89 APE8-rot-in 298.07 APE67-dihe-in -61.98, -22.3 -42.2, -53.64 APE12-dist-in 8.4497 APE11-dist-in 11.738 APE10-dist-in 6.2031 APE9-dist-in 3.7917 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.489 0.148 0.165 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5mhi Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1KA P25321 7 351 351.0 489:60401,489:60402 Type1,Allosteric Active DFGin 6.6813 14.3396 BLAminus -129.58, -178.71 64.55, 76.01 -90.26, 23.75 273.79, 68.55 -63.06, -22.76 in-in in 8.7102 Saltbr-in 2.9128 HRD-in -99.27, -50.72 71.29, 6.63 in-in-in SNCiii in-in ActLoopNT-in 2.8362 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.63, 158.5 APE9-dihe-na 132.87, -161.38 APE8-dihe-in -113.27, 127.15 APE8-rot-in 294.21 APE67-dihe-in -60.63, -22.02 -48.01, -50.0 APE12-dist-in 8.5014 APE11-dist-in 11.9334 APE10-dist-in 6.3293 APE9-dist-in 3.9344 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.8 0.176 0.207 A 353.0 342.0 1 25 25 0 [[44, 298]] 1.0 5n1k Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N32A P25321 1 351 351.0 8K5:60401,8K5:60402 Type1,Allosteric Active DFGin 6.4155 14.3999 BLAminus -123.43, 169.73 68.32, 89.82 -99.03, 25.86 273.98, 63.38 -60.64, -27.18 in-in in 8.5541 Saltbr-in 2.9422 HRD-in -95.08, -52.85 72.97, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.8629 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.95, 157.19 APE9-dihe-na 134.82, -164.27 APE8-dihe-in -110.28, 129.88 APE8-rot-in 300.11 APE67-dihe-in -58.64, -21.5 -44.53, -54.28 APE12-dist-in 8.2963 APE11-dist-in 11.7091 APE10-dist-in 6.1918 APE9-dist-in 3.7562 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.833 0.189 0.214 A 353.0 347.0 1 25 25 0 [[44, 298]] 1.0 5n32 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3FA P25321 8 334 351.0 463:60403,463:60404 Type1,Allosteric Active DFGin 6.6384 14.3677 BLAminus -117.37, -176.84 55.46, 81.93 -92.56, 25.55 274.27, 67.55 -63.44, -27.73 in-in in 8.5998 Saltbr-in 2.7496 HRD-in -89.81, -49.01 69.4, 15.01 in-in-in SNCiii in-in ActLoopNT-in 2.8811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.19, 158.49 APE9-dihe-na 131.1, -163.4 APE8-dihe-in -115.17, 131.52 APE8-rot-in 292.11 APE67-dihe-in -62.12, -20.35 -46.17, -51.48 APE12-dist-in 8.2862 APE11-dist-in 11.6832 APE10-dist-in 6.133 APE9-dist-in 3.7286 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.68 0.173 0.193 A 353.0 321.0 3 25 25 0 [[44, 298]] 1.0 5n3f Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3QA P25321 13 351 351.0 3AB:60402,3AB:60403 Type1,Allosteric Active DFGin 6.2826 14.5563 BLAminus -125.56, 161.33 75.46, 92.4 -98.05, 24.41 270.83, 54.38 -60.67, -25.07 in-in in 8.6862 Saltbr-in 3.0245 HRD-in -85.81, -51.8 71.36, 11.13 in-in-in SNCiii in-in ActLoopNT-in 2.932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.6, 158.28 APE9-dihe-na 114.3, 168.0 APE8-dihe-in -88.22, 137.3 APE8-rot-in 301.76 APE67-dihe-in -63.54, -20.32 -47.52, -48.52 APE12-dist-in 8.0466 APE11-dist-in 11.2177 APE10-dist-in 5.6936 APE9-dist-in 3.9813 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.31 0.136 0.155 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5n3q Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SNXA P25321 12 351 351.0 UNU:60401,UNU:60402 Type1,Allosteric Active DFGin 6.0512 12.8501 BLAminus -124.13, 164.79 75.87, 90.3 -99.95, 24.45 300.66, 73.6 -57.58, -27.27 in-in in 8.5952 Saltbr-in 3.0744 HRD-in -86.88, -52.37 71.04, 13.69 in-in-in SNCiii in-in ActLoopNT-in 2.9054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.16, 166.36 APE9-dihe-na 120.96, -160.48 APE8-dihe-in -123.13, 133.39 APE8-rot-in 301.0 APE67-dihe-in -63.1, -19.02 -49.07, -48.25 APE12-dist-in 8.1536 APE11-dist-in 11.1905 APE10-dist-in 5.6481 APE9-dist-in 3.568 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.4 0.142 0.173 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6snx Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6YOTA P25321 1 351 351.0 P4W:60401,P4W:60402 Type1,Allosteric Active DFGin 6.3385 14.3597 BLAminus -117.22, 168.15 76.5, 96.51 -113.0, 26.95 288.67, 82.96 -66.18, -20.33 in-in in 9.1602 Saltbr-in 2.6238 HRD-in -88.7, -57.55 74.81, 2.26 in-in-in SNCiii in-in ActLoopNT-in 2.8328 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.9, 156.81 APE9-dihe-na 126.53, -165.91 APE8-dihe-in -115.98, 133.13 APE8-rot-in 299.88 APE67-dihe-in -58.64, -24.04 -48.78, -50.95 APE12-dist-in 8.0985 APE11-dist-in 11.3364 APE10-dist-in 5.8219 APE9-dist-in 3.7365 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.96 0.192 0.213 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6yot Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ZN0A P25321 14 351 351.0 NTN:60404,NTN:60405 Type1,Allosteric Active DFGin 6.3062 14.2933 BLAminus -125.36, 174.33 64.27, 86.94 -95.54, 24.99 272.68, 57.62 -59.97, -26.54 in-in in 8.5423 Saltbr-in 2.7539 HRD-in -87.06, -51.0 70.17, 14.59 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.46, 163.69 APE9-dihe-na 125.37, -162.56 APE8-dihe-in -119.36, 135.19 APE8-rot-in 306.4 APE67-dihe-in -62.76, -20.13 -50.46, -46.23 APE12-dist-in 8.1022 APE11-dist-in 11.185 APE10-dist-in 5.6571 APE9-dist-in 3.7386 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.59 0.156 0.186 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6zn0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE0A P25321 12 351 351.0 A1JE3:60415,A1JE3:60416 Type1,Allosteric Active DFGin 6.4858 14.8008 BLAminus -127.81, 175.95 67.21, 79.76 -92.52, 24.98 274.18, 65.26 -62.68, -27.01 in-in in 8.9734 Saltbr-in 2.7196 HRD-in -89.08, -49.37 68.42, 15.8 in-in-in SNCiii in-in ActLoopNT-in 2.9816 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.81, 165.38 APE9-dihe-na 123.68, -167.92 APE8-dihe-in -111.45, 134.55 APE8-rot-in 307.3 APE67-dihe-in -62.16, -20.99 -49.64, -48.1 APE12-dist-in 8.2307 APE11-dist-in 11.3722 APE10-dist-in 5.8261 APE9-dist-in 3.8272 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.58 0.17 0.199 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE1A P25321 12 351 351.0 A1JE2:60402,A1JE2:60403 Type1,Allosteric Active DFGin 6.357 14.4975 BLAminus -123.64, 170.43 71.38, 82.58 -93.83, 23.94 276.73, 61.78 -63.16, -19.76 in-in in 8.9487 Saltbr-in 2.6912 HRD-in -91.56, -54.72 69.86, 16.16 in-in-in SNCiii in-in ActLoopNT-in 2.9345 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.9, 155.93 APE9-dihe-na 118.62, 174.39 APE8-dihe-in -90.43, 137.72 APE8-rot-in 306.04 APE67-dihe-in -61.66, -22.83 -48.01, -48.11 APE12-dist-in 8.0786 APE11-dist-in 11.2497 APE10-dist-in 5.7715 APE9-dist-in 4.114 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.41 0.158 0.189 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re1 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE8A P25321 13 351 351.0 A1JEQ:60401,A1JEQ:60402 Type1,Allosteric Active DFGin 6.4702 14.2842 BLAminus -121.7, 170.26 70.13, 85.83 -96.63, 25.0 277.83, 62.9 -63.72, -22.81 in-in in 8.5972 Saltbr-in 2.853 HRD-in -94.16, -51.38 66.63, 15.52 in-in-in SNCiii in-in ActLoopNT-in 2.9219 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.45, 162.24 APE9-dihe-na 127.76, -169.19 APE8-dihe-in -105.79, 133.4 APE8-rot-in 307.65 APE67-dihe-in -61.36, -22.52 -49.82, -47.46 APE12-dist-in 8.0545 APE11-dist-in 11.2462 APE10-dist-in 5.7207 APE9-dist-in 3.8389 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.18 0.204 A 353.0 337.0 2 25 25 0 [[44, 298]] 1.0 9re8 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE9A P25321 12 351 351.0 A1JER:60406,A1JER:60407 Type1,Allosteric Active DFGin 6.2139 14.4257 BLAminus -115.45, 174.18 67.64, 91.06 -99.47, 24.72 274.09, 59.88 -62.57, -25.54 in-in in 8.5815 Saltbr-in 2.8645 HRD-in -87.53, -50.86 69.59, 9.72 in-in-in SNCiii in-in ActLoopNT-in 2.9177 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.54, 160.39 APE9-dihe-na 112.91, 168.83 APE8-dihe-in -85.08, 139.5 APE8-rot-in 305.47 APE67-dihe-in -61.28, -24.3 -48.68, -48.83 APE12-dist-in 8.0803 APE11-dist-in 11.1938 APE10-dist-in 5.7056 APE9-dist-in 3.9875 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.41 0.159 0.182 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9re9 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE4A P25321 11 351 351.0 A1JEZ:60402,A1JEZ:60403,A1JEZ:60404 Type1,Allosteric,Allosteric Active DFGin 6.4193 14.4719 BLAminus -125.46, 163.88 74.29, 91.54 -99.92, 24.22 273.39, 58.15 -62.6, -24.27 in-in in 8.6037 Saltbr-in 3.0263 HRD-in -87.71, -51.55 69.07, 12.85 in-in-in SNCiii in-in ActLoopNT-in 2.9413 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.46, 156.9 APE9-dihe-na 126.03, -178.78 APE8-dihe-in -98.18, 132.58 APE8-rot-in 299.03 APE67-dihe-in -60.55, -22.76 -49.18, -46.22 APE12-dist-in 8.1382 APE11-dist-in 11.3542 APE10-dist-in 5.8006 APE9-dist-in 4.0873 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.47 0.192 0.208 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 9re4 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE7A P25321 13 351 351.0 D6V:60401,D6V:60402,D6V:60403,D6V:60404 Type1,Allosteric,Allosteric,Allosteric Active DFGin 6.3969 14.3822 BLAminus -125.46, 169.66 70.64, 87.21 -98.97, 25.83 271.46, 63.62 -64.67, -22.85 in-in in 8.6706 Saltbr-in 3.0142 HRD-in -86.12, -51.15 69.09, 13.78 in-in-in SNCiii in-in ActLoopNT-in 2.9179 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.38, 162.49 APE9-dihe-na 118.13, -170.93 APE8-dihe-in -105.88, 133.45 APE8-rot-in 300.33 APE67-dihe-in -56.23, -24.21 -49.65, -50.28 APE12-dist-in 8.2052 APE11-dist-in 11.3507 APE10-dist-in 5.7797 APE9-dist-in 3.8302 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.46 0.156 0.183 A 353.0 337.0 2 25 25 0 [[44, 298]] 1.0 9re7 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REIA P25321 13 351 351.0 A1JEN:60401,A1JEN:60402 Type1,Type1 Active DFGin 6.4427 14.5573 BLAminus -121.53, 160.04 78.3, 90.11 -98.4, 25.75 272.41, 61.56 -62.91, -24.68 in-in in 8.7225 Saltbr-in 2.9878 HRD-in -84.67, -52.43 70.44, 13.57 in-in-in SNCiii in-in ActLoopNT-in 2.9938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.29, 162.32 APE9-dihe-na 123.69, -172.32 APE8-dihe-in -110.41, 137.96 APE8-rot-in 307.06 APE67-dihe-in -63.61, -18.16 -49.51, -49.01 APE12-dist-in 8.2745 APE11-dist-in 11.2994 APE10-dist-in 5.8053 APE9-dist-in 3.9129 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.167 0.199 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rei Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OUAA P25321 1 351 351.0 No_ligand No_ligand Inactive DFGin 6.7177 14.6348 ABAminus -115.87, -28.94 -123.11, 121.25 -116.35, 27.71 279.87, 77.2 -63.52, -23.18 in-in in 8.6437 Saltbr-in 2.9268 HRD-in -81.78, -54.82 73.94, 13.55 in-in-in SNCiii in-in ActLoopNT-in 2.8996 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.08, 165.1 APE9-dihe-na 113.51, -165.37 APE8-dihe-in -110.07, 129.07 APE8-rot-in 298.26 APE67-dihe-in -59.52, -23.19 -44.71, -53.87 APE12-dist-in 8.3252 APE11-dist-in 11.5022 APE10-dist-in 5.7636 APE9-dist-in 3.3871 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.67 0.17 0.194 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5oua Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OUSA P25321 1 351 351.0 No_ligand No_ligand Inactive DFGin 6.5073 15.429 ABAminus -111.6, -55.85 -94.1, 116.86 -107.2, 23.58 279.6, 77.36 -70.84, -13.23 in-none in 9.4454 Saltbr-none 999.0 HRD-in -84.43, -53.59 72.65, 7.3 none-in-in SNCnii in-in ActLoopNT-in 3.002 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.86, 162.52 APE9-dihe-na 121.37, -167.35 APE8-dihe-in -115.92, 134.51 APE8-rot-in 300.98 APE67-dihe-in -58.34, -27.31 -46.95, -49.63 APE12-dist-in 8.2545 APE11-dist-in 11.5502 APE10-dist-in 5.9508 APE9-dist-in 3.6723 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.21 0.196 0.233 A 353.0 348.0 1 25 25 0 [[44, 298]] 1.0 5ous Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5NW8A P25321 12 351 351.0 M77:60402 Type1 Inactive DFGin 6.3364 14.3863 ABAminus -118.68, -32.42 -99.03, 121.53 -122.45, 23.74 290.12, 82.65 -65.48, -23.88 in-in in 8.8836 Saltbr-in 2.7053 HRD-in -87.46, -57.12 74.8, 8.43 in-in-in SNCiii in-in ActLoopNT-in 2.9091 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.41, 158.53 APE9-dihe-na 124.11, -167.34 APE8-dihe-in -113.09, 136.58 APE8-rot-in 301.73 APE67-dihe-in -53.51, -29.49 -47.53, -53.31 APE12-dist-in 8.2041 APE11-dist-in 11.5565 APE10-dist-in 5.9221 APE9-dist-in 3.7724 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.086 0.178 0.212 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 5nw8 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCPA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.5125 14.567 ABAminus -121.65, -30.45 -98.92, 119.1 -122.07, 18.29 284.17, 84.65 -65.16, -27.53 in-in in 8.8992 Saltbr-in 2.7586 HRD-in -92.61, -56.98 71.24, 5.31 in-in-in SNCiii in-in ActLoopNT-in 2.9161 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.37, 152.55 APE9-dihe-na 132.49, -162.49 APE8-dihe-in -118.01, 135.22 APE8-rot-in 296.96 APE67-dihe-in -61.44, -24.53 -48.46, -49.38 APE12-dist-in 8.1866 APE11-dist-in 11.4765 APE10-dist-in 5.9223 APE9-dist-in 3.9486 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.433 0.134 0.166 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcp Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCRA P25321 1 351 351.0 6TX:60401 Type1 Inactive DFGin 6.374 14.6833 ABAminus -120.45, -30.9 -97.04, 125.99 -132.15, 14.59 283.38, 89.54 -63.35, -31.44 in-in in 8.8488 Saltbr-in 2.672 HRD-in -87.18, -55.06 71.63, -3.59 in-in-in SNCiii in-in ActLoopNT-in 2.9015 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.81, 151.9 APE9-dihe-na 132.74, -162.98 APE8-dihe-in -119.91, 132.41 APE8-rot-in 297.04 APE67-dihe-in -57.71, -25.78 -46.99, -51.33 APE12-dist-in 8.2349 APE11-dist-in 11.5396 APE10-dist-in 6.0024 APE9-dist-in 4.0176 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.565 0.157 0.197 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcr Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCTA P25321 1 351 351.0 6TY:60401 Type1 Inactive DFGin 6.5666 14.9722 ABAminus -119.53, -36.47 -94.64, 123.81 -127.4, 15.84 283.42, 88.07 -61.61, -36.92 in-in in 8.9974 Saltbr-in 2.8958 HRD-in -87.59, -53.98 70.09, 3.04 in-in-in SNCiii in-in ActLoopNT-in 2.9272 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.1, 153.93 APE9-dihe-na 129.99, -163.89 APE8-dihe-in -118.91, 134.19 APE8-rot-in 299.57 APE67-dihe-in -59.43, -24.77 -48.83, -49.96 APE12-dist-in 8.3428 APE11-dist-in 11.612 APE10-dist-in 6.0758 APE9-dist-in 3.98 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.615 0.144 0.174 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lct Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5LCUA P25321 1 351 351.0 IQP:60401 Type1 Inactive DFGin 6.3439 14.5118 ABAminus -118.46, -33.64 -98.48, 122.71 -128.59, 17.69 287.43, 87.65 -64.81, -32.5 in-in in 8.9216 Saltbr-in 2.7757 HRD-in -89.6, -56.25 69.6, 5.54 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.54, 154.63 APE9-dihe-na 129.64, -164.53 APE8-dihe-in -116.54, 134.11 APE8-rot-in 299.55 APE67-dihe-in -60.52, -23.05 -47.34, -51.22 APE12-dist-in 8.1905 APE11-dist-in 11.5415 APE10-dist-in 5.9813 APE9-dist-in 3.9715 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.579 0.154 0.192 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5lcu Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M6VA P25321 1 351 351.0 H52:60401 Type1 Inactive DFGin 6.6215 14.87 ABAminus -128.93, -36.38 -82.47, 115.78 -126.79, 13.38 284.62, 84.57 -59.9, -36.82 in-in in 9.1455 Saltbr-in 3.0668 HRD-in -85.39, -54.24 70.45, 5.3 in-in-in SNCiii in-in ActLoopNT-in 2.88 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.08, 154.85 APE9-dihe-na 129.1, -162.88 APE8-dihe-in -117.77, 135.16 APE8-rot-in 297.05 APE67-dihe-in -61.78, -23.12 -47.87, -51.09 APE12-dist-in 8.2559 APE11-dist-in 11.5175 APE10-dist-in 5.9805 APE9-dist-in 3.8478 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.418 0.145 0.174 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m6v Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M6YA P25321 1 351 351.0 7KB:60401 Type1 Inactive DFGin 6.3247 14.3886 ABAminus -120.54, -28.06 -100.7, 125.25 -133.25, 5.41 291.12, 89.13 -59.31, -35.83 in-in in 8.9571 Saltbr-in 2.8685 HRD-in -85.55, -56.37 69.79, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.8795 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.17, 152.58 APE9-dihe-na 128.14, -163.48 APE8-dihe-in -117.76, 135.16 APE8-rot-in 298.33 APE67-dihe-in -60.49, -24.28 -48.85, -50.14 APE12-dist-in 8.3076 APE11-dist-in 11.7151 APE10-dist-in 6.2076 APE9-dist-in 4.0604 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.367 0.145 0.166 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m6y Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M71A P25321 1 351 351.0 7K7:60401 Type1 Inactive DFGin 6.5486 14.873 ABAminus -119.85, -32.84 -98.53, 122.12 -124.32, 17.46 284.12, 85.87 -64.55, -31.73 in-in in 9.0558 Saltbr-in 2.7642 HRD-in -87.14, -56.81 71.22, 6.23 in-in-in SNCiii in-in ActLoopNT-in 2.9024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.13, 152.91 APE9-dihe-na 131.38, -162.26 APE8-dihe-in -116.74, 134.6 APE8-rot-in 297.69 APE67-dihe-in -60.19, -23.45 -48.52, -50.53 APE12-dist-in 8.2262 APE11-dist-in 11.5825 APE10-dist-in 5.9903 APE9-dist-in 3.8944 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.488 0.149 0.176 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m71 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5M75A P25321 1 351 351.0 9K6:60402 Type1 Inactive DFGin 6.5416 14.7033 ABAminus -122.93, -37.42 -95.22, 118.15 -122.41, 18.78 283.61, 82.19 -61.66, -33.64 in-in in 9.017 Saltbr-in 2.9023 HRD-in -86.66, -56.28 74.63, 2.67 in-in-in SNCiii in-in ActLoopNT-in 2.8945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.02, 157.01 APE9-dihe-na 127.35, -165.16 APE8-dihe-in -116.36, 133.7 APE8-rot-in 297.39 APE67-dihe-in -60.71, -23.5 -48.32, -49.81 APE12-dist-in 8.2248 APE11-dist-in 11.4473 APE10-dist-in 5.9243 APE9-dist-in 3.7682 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.538 0.146 0.174 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5m75 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1DA P25321 1 351 351.0 8FZ:60403 Type1 Inactive DFGin 6.4268 14.5221 ABAminus -119.36, -25.35 -95.05, 134.07 -134.0, 35.23 286.49, 84.89 -74.09, -16.92 in-in in 8.9671 Saltbr-in 2.7736 HRD-in -86.75, -53.91 69.79, 6.83 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.28, 160.08 APE9-dihe-na 123.62, -165.42 APE8-dihe-in -115.29, 135.17 APE8-rot-in 295.44 APE67-dihe-in -60.76, -24.93 -47.42, -49.84 APE12-dist-in 8.3805 APE11-dist-in 11.5224 APE10-dist-in 5.9453 APE9-dist-in 3.6307 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.609 0.157 0.186 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 5n1d Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3DA P25321 1 351 351.0 8NE:60401 Type1 Inactive DFGin 6.3769 14.5132 ABAminus -125.06, 6.06 -141.01, 114.08 -108.34, 25.78 270.84, 67.95 -65.47, -20.45 in-in in 8.8019 Saltbr-in 2.8929 HRD-in -88.66, -53.48 71.74, 8.74 in-in-in SNCiii in-in ActLoopNT-in 2.8859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.56, 155.77 APE9-dihe-na 134.96, -165.87 APE8-dihe-in -106.38, 130.24 APE8-rot-in 300.79 APE67-dihe-in -61.42, -22.58 -44.45, -52.67 APE12-dist-in 8.4623 APE11-dist-in 11.8721 APE10-dist-in 6.2946 APE9-dist-in 3.8887 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.77 0.169 0.193 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 5n3d Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5O0EA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.5233 14.4554 ABAminus -120.87, -28.54 -98.9, 119.84 -125.0, 19.69 283.23, 84.18 -67.0, -26.17 in-in in 8.8606 Saltbr-in 2.7863 HRD-in -91.49, -57.65 74.16, -1.91 in-in-in SNCiii in-in ActLoopNT-in 2.9264 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.49, 154.58 APE9-dihe-na 133.99, -164.02 APE8-dihe-in -122.83, 136.35 APE8-rot-in 298.08 APE67-dihe-in -61.85, -22.28 -48.99, -49.98 APE12-dist-in 8.1871 APE11-dist-in 11.4128 APE10-dist-in 5.8742 APE9-dist-in 4.0603 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.5 0.133 0.17 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5o0e Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5O5MA P25321 10 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.2398 14.1421 ABAminus -103.5, -42.75 -109.64, 134.16 -133.73, 10.26 296.02, 86.96 -61.7, -36.78 in-in in 8.8473 Saltbr-in 2.793 HRD-in -81.57, -55.82 71.03, 6.22 in-in-in SNCiii in-in ActLoopNT-in 2.8906 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.12, 155.87 APE9-dihe-na 127.02, -162.8 APE8-dihe-in -117.37, 136.63 APE8-rot-in 301.79 APE67-dihe-in -60.33, -24.0 -47.69, -51.35 APE12-dist-in 8.4177 APE11-dist-in 11.9058 APE10-dist-in 6.3877 APE9-dist-in 3.8023 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.583 0.15 0.182 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5o5m Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OK3A P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.6154 14.4154 ABAminus -120.44, -31.18 -98.89, 117.63 -123.6, 23.39 284.71, 82.73 -69.59, -23.81 in-in in 8.9341 Saltbr-in 2.7392 HRD-in -95.2, -57.86 72.09, 2.44 in-in-in SNCiii in-in ActLoopNT-in 2.9251 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.84, 153.6 APE9-dihe-na 133.87, -163.65 APE8-dihe-in -122.15, 135.18 APE8-rot-in 299.79 APE67-dihe-in -60.82, -23.36 -49.17, -49.56 APE12-dist-in 8.2185 APE11-dist-in 11.4659 APE10-dist-in 5.8784 APE9-dist-in 4.0553 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.588 0.141 0.172 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5ok3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OL3A P25321 11 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.2933 14.1388 ABAminus -103.07, -42.44 -110.53, 139.16 -139.44, 13.42 297.3, 87.11 -59.46, -35.81 in-in in 8.8063 Saltbr-in 2.7003 HRD-in -84.73, -54.59 70.4, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.9398 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.98, 154.3 APE9-dihe-na 129.69, -160.74 APE8-dihe-in -119.81, 133.8 APE8-rot-in 301.31 APE67-dihe-in -59.48, -24.61 -48.47, -50.75 APE12-dist-in 8.5226 APE11-dist-in 12.0085 APE10-dist-in 6.4955 APE9-dist-in 3.7939 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.58 0.156 0.199 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 5ol3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OT3A P25321 13 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.3842 14.2359 ABAminus -113.79, -34.42 -102.76, 127.41 -133.44, 15.99 294.3, 89.2 -57.06, -43.48 in-in in 8.8594 Saltbr-in 2.8226 HRD-in -85.16, -56.21 73.39, 3.05 in-in-in SNCiii in-in ActLoopNT-in 2.9097 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.31, 153.48 APE9-dihe-na 129.3, -161.89 APE8-dihe-in -114.87, 136.52 APE8-rot-in 300.43 APE67-dihe-in -56.81, -27.64 -51.93, -48.81 APE12-dist-in 8.2915 APE11-dist-in 11.842 APE10-dist-in 6.3049 APE9-dist-in 4.0341 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.04 0.186 0.228 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5ot3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OTGA P25321 1 351 351.0 AO8:60401 Type1 Inactive DFGin 6.6641 14.8724 ABAminus -116.07, -34.14 -101.63, 135.19 -132.51, 30.55 284.27, 81.94 -65.58, -28.86 in-in in 9.2076 Saltbr-in 2.8838 HRD-in -87.0, -54.6 75.88, 1.07 in-in-in SNCiii in-in ActLoopNT-in 2.9513 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.1, 159.53 APE9-dihe-na 126.93, -164.36 APE8-dihe-in -118.42, 136.98 APE8-rot-in 301.94 APE67-dihe-in -61.55, -22.37 -50.07, -49.22 APE12-dist-in 8.3277 APE11-dist-in 11.5661 APE10-dist-in 5.9649 APE9-dist-in 3.7403 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.73 0.187 0.206 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5otg Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5OUCA P25321 1 351 351.0 AO8:60401 Type1 Inactive DFGin 6.5448 14.6897 ABAminus -118.72, -31.35 -98.66, 124.06 -126.19, 22.18 285.25, 84.4 -64.9, -29.38 in-none in 9.0152 Saltbr-none 999.0 HRD-in -89.21, -57.44 74.92, -2.84 none-in-in SNCnii in-in ActLoopNT-in 2.9042 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 152.91 APE9-dihe-na 134.96, -159.63 APE8-dihe-in -125.22, 135.43 APE8-rot-in 300.15 APE67-dihe-in -61.76, -25.06 -48.4, -50.36 APE12-dist-in 8.2727 APE11-dist-in 11.4814 APE10-dist-in 5.9359 APE9-dist-in 4.0149 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.46 0.151 0.175 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 5ouc Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EGWA P25321 14 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.0679 14.0517 ABAminus -99.1, -40.07 -111.56, 135.78 -136.64, 9.64 299.83, 90.65 -57.2, -34.91 in-in in 8.8053 Saltbr-in 2.8447 HRD-in -79.79, -53.68 65.28, 14.91 in-in-in SNCiii in-in ActLoopNT-in 2.8654 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.34, 128.68 APE9-dihe-na 131.12, -162.98 APE8-dihe-in -115.37, 129.12 APE8-rot-in 299.83 APE67-dihe-in -57.87, -22.06 -45.69, -53.12 APE12-dist-in 8.5497 APE11-dist-in 12.0347 APE10-dist-in 6.3542 APE9-dist-in 3.7696 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.74 0.173 0.203 A 353.0 336.0 1 25 25 0 [[44, 298]] 1.0 6egw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EH3A P25321 1 351 351.0 B4Z:60401 Type1 Inactive DFGin 6.5603 14.4887 ABAminus -116.24, -28.55 -105.91, 131.63 -131.61, 27.16 287.22, 81.75 -60.81, -31.22 in-out in 9.0058 Saltbr-out 3.7684 HRD-in -84.94, -53.5 72.91, 0.92 out-in-in SNCoii in-in ActLoopNT-in 2.8965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.18, 161.6 APE9-dihe-na 127.52, -167.93 APE8-dihe-in -115.28, 135.37 APE8-rot-in 300.84 APE67-dihe-in -65.2, -22.11 -46.47, -48.64 APE12-dist-in 8.279 APE11-dist-in 11.5005 APE10-dist-in 5.9114 APE9-dist-in 3.8034 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.95 0.175 0.219 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6eh3 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERTA P25321 14 351 351.0 BVZ:60401 Type1 Inactive DFGin 6.1937 14.1209 ABAminus -115.39, -20.57 -108.62, 132.15 -135.58, 27.66 297.14, 82.68 -71.36, -3.39 in-in in 8.9653 Saltbr-in 2.8205 HRD-in -85.32, -55.78 74.89, 1.92 in-in-in SNCiii in-in ActLoopNT-in 2.9314 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.5, 160.76 APE9-dihe-na 124.06, -167.42 APE8-dihe-in -111.64, 135.9 APE8-rot-in 303.33 APE67-dihe-in -58.26, -26.08 -52.61, -48.73 APE12-dist-in 8.2618 APE11-dist-in 11.6271 APE10-dist-in 6.0812 APE9-dist-in 3.7549 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.8 0.186 0.218 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6ert Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERWA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.4014 14.4703 ABAminus -121.15, -34.81 -95.55, 109.86 -114.31, 21.73 291.27, 86.69 -64.06, -18.67 in-in in 8.9017 Saltbr-in 2.8745 HRD-in -86.55, -59.04 70.6, 12.67 in-in-in SNCiii in-in ActLoopNT-in 2.8957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.31, 155.57 APE9-dihe-na 122.97, -167.43 APE8-dihe-in -109.73, 134.74 APE8-rot-in 295.31 APE67-dihe-in -57.25, -24.48 -52.2, -50.35 APE12-dist-in 8.161 APE11-dist-in 11.4552 APE10-dist-in 5.8644 APE9-dist-in 3.8464 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.89 0.195 0.229 A 353.0 348.0 3 25 25 0 [[44, 298]] 1.0 6erw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2AA P25321 1 351 351.0 M77:60401 Type1 Inactive DFGin 6.6275 14.6347 ABAminus -122.01, -33.61 -93.89, 119.82 -124.65, 22.24 282.35, 82.22 -67.92, -23.48 in-in in 9.1929 Saltbr-in 2.5611 HRD-in -101.03, -58.68 69.95, -0.61 in-in-in SNCiii in-in ActLoopNT-in 2.9412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.26, 150.72 APE9-dihe-na 137.51, -163.36 APE8-dihe-in -120.26, 133.94 APE8-rot-in 301.03 APE67-dihe-in -62.45, -25.53 -48.16, -48.1 APE12-dist-in 8.1207 APE11-dist-in 11.4401 APE10-dist-in 5.8938 APE9-dist-in 4.1543 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.75 0.175 0.207 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6i2a Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2CA P25321 12 351 351.0 M77:60401 Type1 Inactive DFGin 6.5002 14.6062 ABAminus -115.95, -34.45 -102.09, 116.9 -120.62, 23.53 285.01, 87.65 -68.52, -23.98 in-in in 8.8456 Saltbr-in 2.9203 HRD-in -86.43, -55.89 76.54, -1.15 in-in-in SNCiii in-in ActLoopNT-in 2.9438 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.94, 153.26 APE9-dihe-na 129.65, -163.32 APE8-dihe-in -118.65, 136.78 APE8-rot-in 299.53 APE67-dihe-in -56.88, -28.13 -49.75, -50.61 APE12-dist-in 8.3036 APE11-dist-in 11.5191 APE10-dist-in 5.8971 APE9-dist-in 3.7163 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.82 0.187 0.221 A 353.0 338.0 2 25 25 0 [[44, 298]] 1.0 6i2c Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2DA P25321 9 351 351.0 9LQ:60401 Type1 Inactive DFGin 6.4857 14.6911 ABAminus -99.68, -45.99 -105.21, 136.79 -132.46, 16.35 286.72, 86.8 -63.64, -34.15 in-in in 8.6624 Saltbr-in 2.922 HRD-in -90.54, -57.71 68.94, 6.05 in-in-in SNCiii in-in ActLoopNT-in 2.9826 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.06, 154.58 APE9-dihe-na 132.32, -163.48 APE8-dihe-in -118.09, 133.54 APE8-rot-in 299.26 APE67-dihe-in -59.06, -24.95 -49.23, -49.12 APE12-dist-in 8.037 APE11-dist-in 11.595 APE10-dist-in 5.9733 APE9-dist-in 3.9587 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.91 0.19 0.222 A 353.0 343.0 0 25 25 0 [[44, 298]] 1.0 6i2d Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2HA P25321 1 351 351.0 AO8:60401 Type1 Inactive DFGin 6.5671 14.8085 ABAminus -115.56, -38.67 -109.61, 104.13 -103.25, 25.9 285.61, 77.71 -66.17, -17.47 in-in in 8.9865 Saltbr-in 2.9304 HRD-in -83.42, -55.73 70.56, 10.93 in-in-in SNCiii in-in ActLoopNT-in 2.8462 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.42, 160.46 APE9-dihe-na 121.97, -162.48 APE8-dihe-in -116.28, 135.78 APE8-rot-in 298.33 APE67-dihe-in -60.57, -22.98 -48.67, -52.6 APE12-dist-in 8.1576 APE11-dist-in 11.371 APE10-dist-in 5.6959 APE9-dist-in 3.5478 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.68 0.182 0.202 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6i2h Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y0BA P25321 1 351 351.0 1LQ:60401 Type1 Inactive DFGin 6.3607 14.3289 ABAminus -119.37, -25.73 -99.15, 124.17 -126.15, 31.35 288.49, 83.65 -71.09, -16.36 in-in in 9.046 Saltbr-in 2.5951 HRD-in -88.77, -52.67 71.85, 3.28 in-in-in SNCiii in-in ActLoopNT-in 2.8228 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.54, 158.64 APE9-dihe-na 129.02, -163.22 APE8-dihe-in -120.14, 133.41 APE8-rot-in 298.13 APE67-dihe-in -64.32, -22.04 -50.27, -45.04 APE12-dist-in 8.2202 APE11-dist-in 11.4198 APE10-dist-in 5.8956 APE9-dist-in 3.6527 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.71 0.181 0.212 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 6y0b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y2UA P25321 1 351 351.0 LRT:60401 Type1 Inactive DFGin 6.3897 14.1273 ABAminus -116.87, -29.74 -101.42, 118.51 -125.0, 17.87 293.73, 84.27 -60.5, -32.85 in-in in 8.8178 Saltbr-in 2.7471 HRD-in -82.23, -56.84 69.37, 8.99 in-in-in SNCiii in-in ActLoopNT-in 2.9228 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.67, 161.61 APE9-dihe-na 116.23, -161.47 APE8-dihe-in -111.19, 132.56 APE8-rot-in 301.77 APE67-dihe-in -58.37, -26.58 -47.25, -49.31 APE12-dist-in 8.1796 APE11-dist-in 11.6373 APE10-dist-in 5.9769 APE9-dist-in 3.8833 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.93 0.187 0.222 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6y2u Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7AXWA P25321 1 351 351.0 1SQ:60401 Type1 Inactive DFGin 6.4035 14.2527 ABAminus -120.14, -30.0 -96.57, 126.41 -127.77, 33.09 287.87, 84.79 -75.22, -10.69 in-in in 8.9432 Saltbr-in 2.6309 HRD-in -88.15, -50.93 71.59, -1.54 in-in-in SNCiii in-in ActLoopNT-in 2.8412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.41, 158.2 APE9-dihe-na 127.83, -163.7 APE8-dihe-in -120.34, 130.94 APE8-rot-in 298.02 APE67-dihe-in -65.73, -21.71 -43.41, -48.57 APE12-dist-in 8.2015 APE11-dist-in 11.4083 APE10-dist-in 5.9311 APE9-dist-in 3.6613 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.69 0.183 0.219 A 353.0 349.0 0 25 25 0 [[44, 298]] 1.0 7axw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7BAQA P25321 12 351 351.0 T82:60401 Type1 Inactive DFGin 6.6314 14.6407 ABAminus -123.23, -37.41 -116.05, 126.94 -128.82, 27.15 284.58, 82.2 -65.24, -36.99 in-in in 8.8751 Saltbr-in 2.8259 HRD-in -84.32, -54.85 70.47, 4.72 in-in-in SNCiii in-in ActLoopNT-in 2.9304 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.86, 160.75 APE9-dihe-na 122.68, -162.38 APE8-dihe-in -118.09, 132.31 APE8-rot-in 301.89 APE67-dihe-in -58.89, -25.14 -49.52, -49.11 APE12-dist-in 8.2341 APE11-dist-in 11.5243 APE10-dist-in 6.0507 APE9-dist-in 3.7373 None TPO198,SEP339 TPO198,SEP339 XRAY 1.54 0.178 0.22 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 7baq Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIDA P25321 1 351 351.0 7QI:60401 Type1 Inactive DFGin 6.4367 14.9083 ABAminus -118.24, -40.4 -94.33, 114.05 -113.71, 22.91 282.95, 85.12 -67.72, -22.35 in-in in 9.1457 Saltbr-in 3.1967 HRD-in -88.95, -55.75 73.32, 6.65 in-in-in SNCiii in-in ActLoopNT-in 2.9311 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.62, 155.91 APE9-dihe-na 130.66, -167.59 APE8-dihe-in -113.9, 136.41 APE8-rot-in 298.55 APE67-dihe-in -61.41, -23.98 -47.99, -49.83 APE12-dist-in 8.2605 APE11-dist-in 11.4592 APE10-dist-in 5.8679 APE9-dist-in 3.8737 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.496 0.134 0.161 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pid Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIEA P25321 1 351 351.0 7QF:60401 Type1 Inactive DFGin 6.4369 14.7079 ABAminus -120.2, -32.0 -97.5, 116.46 -117.79, 21.67 284.38, 87.37 -67.96, -24.99 in-in in 9.0175 Saltbr-in 2.947 HRD-in -90.08, -55.75 70.92, 8.29 in-in-in SNCiii in-in ActLoopNT-in 2.9298 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.9, 155.75 APE9-dihe-na 129.48, -166.45 APE8-dihe-in -116.19, 135.64 APE8-rot-in 298.32 APE67-dihe-in -59.08, -26.0 -47.12, -51.73 APE12-dist-in 8.298 APE11-dist-in 11.4827 APE10-dist-in 5.9206 APE9-dist-in 3.8942 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.427 0.137 0.158 A 353.0 350.0 0 25 25 0 [[44, 298]] 1.0 7pie Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIFA P25321 1 351 351.0 7QL:60401 Type1 Inactive DFGin 6.3465 14.218 ABAminus -118.69, -29.14 -100.96, 122.87 -127.55, 15.73 291.19, 87.86 -63.07, -33.16 in-in in 8.9572 Saltbr-in 2.7865 HRD-in -92.08, -57.05 70.77, -0.71 in-in-in SNCiii in-in ActLoopNT-in 2.9092 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.9, 150.21 APE9-dihe-na 133.66, -162.89 APE8-dihe-in -122.64, 134.78 APE8-rot-in 297.75 APE67-dihe-in -60.89, -24.83 -47.76, -50.71 APE12-dist-in 8.3006 APE11-dist-in 11.5735 APE10-dist-in 6.0009 APE9-dist-in 4.1345 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.395 0.135 0.155 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pif Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PIGA P25321 1 351 351.0 7QR:60401 Type1 Inactive DFGin 6.4813 14.8758 ABAminus -122.28, -26.17 -100.91, 119.71 -123.06, 20.32 285.86, 92.34 -68.86, -24.06 in-in in 8.9216 Saltbr-in 2.7465 HRD-in -91.36, -59.49 70.09, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.9153 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.9, 150.63 APE9-dihe-na 129.65, -165.04 APE8-dihe-in -112.18, 133.86 APE8-rot-in 299.17 APE67-dihe-in -59.53, -25.5 -47.67, -52.22 APE12-dist-in 8.1547 APE11-dist-in 11.4414 APE10-dist-in 5.8432 APE9-dist-in 4.0681 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.553 0.129 0.154 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 7pig Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7PNSA P25321 10 351 351.0 7W8:60402 Type1 Inactive DFGin 6.5137 14.8169 ABAminus -119.8, -32.67 -110.21, 109.27 -108.01, 28.37 286.1, 78.14 -68.46, -20.09 in-in in 8.9796 Saltbr-in 3.0843 HRD-in -83.54, -55.5 71.62, 9.07 in-in-in SNCiii in-in ActLoopNT-in 2.9078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.45, 157.3 APE9-dihe-na 125.01, -165.6 APE8-dihe-in -110.51, 134.07 APE8-rot-in 302.08 APE67-dihe-in -61.89, -24.52 -46.65, -50.8 APE12-dist-in 8.3238 APE11-dist-in 11.6189 APE10-dist-in 6.0319 APE9-dist-in 3.821 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.855 0.176 0.202 A 353.0 342.0 0 25 25 0 [[44, 298]] 1.0 7pns Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6I2BA P25321 5 351 351.0 9LQ:60401,9LQ:60402 Type1,Allosteric Inactive DFGin 6.3083 14.5013 ABAminus -99.36, -48.22 -103.96, 139.83 -136.93, 15.62 290.92, 85.14 -58.8, -40.25 in-in in 8.6839 Saltbr-in 2.8063 HRD-in -93.94, -54.86 69.46, 4.74 in-in-in SNCiii in-in ActLoopNT-in 2.9981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.47, 156.84 APE9-dihe-na 128.63, -164.41 APE8-dihe-in -116.79, 133.75 APE8-rot-in 301.48 APE67-dihe-in -59.49, -25.74 -49.19, -49.96 APE12-dist-in 8.1365 APE11-dist-in 11.6214 APE10-dist-in 6.0086 APE9-dist-in 3.9532 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.97 0.212 0.248 A 353.0 345.0 0 25 25 0 [[44, 298]] 1.0 6i2b Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REKA P25321 12 351 351.0 D8P:60401,D8P:60402,D8P:60403,D8P:60404 Type1,Allosteric,Allosteric,Allosteric Inactive DFGin 6.3425 14.4394 ABAminus -107.25, -41.44 -100.58, 143.12 -128.51, 27.13 273.04, 65.71 -61.45, -23.67 in-in in 8.578 Saltbr-in 2.7782 HRD-in -87.09, -53.39 71.15, 12.36 in-in-in SNCiii in-in ActLoopNT-in 2.9003 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.7, 168.09 APE9-dihe-na 116.77, -166.86 APE8-dihe-in -118.41, 135.56 APE8-rot-in 302.89 APE67-dihe-in -59.2, -22.22 -49.04, -50.02 APE12-dist-in 8.1717 APE11-dist-in 11.1178 APE10-dist-in 5.6342 APE9-dist-in 3.7371 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.159 0.19 A 353.0 339.0 1 25 25 0 [[44, 298]] 1.0 9rek Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EM6A P25321 12 351 351.0 ADP:60401 ATPlike Inactive DFGin 6.8591 14.8208 BLAminus -128.32, 163.45 74.87, 92.52 -104.27, 28.45 286.23, 74.8 -62.75, -23.58 in-out in 9.7038 Saltbr-out 4.3621 HRD-in -85.36, -55.87 71.35, 12.71 out-in-in SNCoii in-in ActLoopNT-in 2.9302 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 157.75 APE9-dihe-na 127.42, -164.4 APE8-dihe-in -115.9, 133.37 APE8-rot-in 304.12 APE67-dihe-in -57.32, -23.54 -48.16, -51.44 APE12-dist-in 8.0456 APE11-dist-in 11.3093 APE10-dist-in 5.7368 APE9-dist-in 3.819 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.64 0.175 0.191 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 6em6 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3NA P25321 12 351 351.0 152:60403 Allosteric Inactive DFGin 6.2448 14.3764 BLAminus -123.59, 163.17 75.18, 93.32 -100.77, 23.69 272.14, 54.48 -60.82, -27.27 in-in in 8.5509 Saltbr-in 2.932 HRD-in -86.04, -51.94 69.91, 12.31 in-in-out SNCiio in-out ActLoopNT-in 2.9316 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.97, 158.43 APE9-dihe-na 112.44, 164.79 APE8-dihe-in -81.93, 141.6 APE8-rot-out 194.34 APE67-dihe-in -62.51, -21.05 -48.48, -48.45 APE12-dist-in 8.1235 APE11-dist-in 11.1935 APE10-dist-in 5.687 APE9-dist-in 3.9939 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.224 0.136 0.153 A 351.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3n Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1GA P25321 12 351 351.0 8G5:60403 Allosteric Inactive DFGin 6.3509 14.2952 BLAminus -120.55, 160.72 78.08, 93.75 -100.89, 22.9 268.69, 55.04 -61.15, -25.02 in-in in 8.4501 Saltbr-in 2.8286 HRD-in -85.02, -51.99 68.33, 11.76 in-in-out SNCiio in-out ActLoopNT-in 2.9141 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.3, 157.42 APE9-dihe-na 113.47, 162.71 APE8-dihe-in -82.12, 143.17 APE8-rot-out 195.96 APE67-dihe-in -64.28, -21.72 -48.98, -46.63 APE12-dist-in 8.0256 APE11-dist-in 11.1323 APE10-dist-in 5.6526 APE9-dist-in 4.0142 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.14 0.129 0.141 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1g Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3RA P25321 13 351 351.0 CDT:60401 Allosteric Inactive DFGin 6.2835 14.3648 BLAminus -123.4, 166.85 72.82, 88.41 -96.79, 24.64 271.02, 57.62 -62.08, -26.42 in-in in 8.473 Saltbr-in 2.8507 HRD-in -84.5, -51.65 69.06, 12.07 in-in-out SNCiio in-out ActLoopNT-in 2.9132 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -163.54, 160.53 APE9-dihe-na 112.85, 168.5 APE8-dihe-in -90.49, 143.51 APE8-rot-out 194.17 APE67-dihe-in -64.82, -18.23 -48.56, -47.77 APE12-dist-in 8.01 APE11-dist-in 11.109 APE10-dist-in 5.6694 APE9-dist-in 3.7548 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.36 0.161 0.193 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 5n3r Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REHA P25321 13 351 351.0 A1JEO:60410 Allosteric Inactive DFGin 6.3163 14.4571 BLAminus -120.51, 166.33 73.93, 87.07 -97.3, 23.53 273.58, 55.63 -62.98, -24.59 in-in in 8.6439 Saltbr-in 2.934 HRD-in -90.78, -53.04 70.2, 12.8 in-in-out SNCiio in-out ActLoopNT-in 2.9492 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.03, 159.17 APE9-dihe-na 115.21, 161.46 APE8-dihe-in -80.42, 146.14 APE8-rot-out 193.65 APE67-dihe-in -62.8, -23.48 -51.35, -45.43 APE12-dist-in 8.0609 APE11-dist-in 11.138 APE10-dist-in 5.6907 APE9-dist-in 3.9727 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.33 0.14 0.165 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9reh Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3GA P25321 12 351 351.0 8KB:60401,8KB:60402 Allosteric,Allosteric Inactive DFGin 6.2401 14.4188 BLAminus -122.61, 161.7 77.55, 93.02 -100.37, 23.32 270.97, 56.3 -63.09, -23.8 in-in in 8.5755 Saltbr-in 2.9043 HRD-in -86.82, -52.03 69.25, 11.52 in-in-out SNCiio in-out ActLoopNT-in 2.9346 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.35, 154.45 APE9-dihe-na 118.07, 158.61 APE8-dihe-in -78.39, 140.92 APE8-rot-out 196.18 APE67-dihe-in -62.0, -22.59 -47.89, -47.51 APE12-dist-in 8.0381 APE11-dist-in 11.2059 APE10-dist-in 5.7252 APE9-dist-in 4.1113 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.16 0.138 0.157 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3g Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REDA P25321 13 351 351.0 A1JEV:60401,A1JEV:60402 Allosteric,Allosteric Inactive DFGin 6.3136 14.3886 BLAminus -123.16, 164.73 74.85, 89.64 -97.97, 23.84 269.64, 57.8 -61.74, -25.67 in-in in 8.6392 Saltbr-in 2.8089 HRD-in -83.21, -53.37 69.6, 13.68 in-in-out SNCiio in-out ActLoopNT-in 2.9232 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.24, 157.71 APE9-dihe-na 113.1, 163.31 APE8-dihe-in -87.29, 142.42 APE8-rot-out 178.62 APE67-dihe-in -62.59, -21.07 -47.65, -46.78 APE12-dist-in 8.0505 APE11-dist-in 11.1849 APE10-dist-in 5.6941 APE9-dist-in 4.0315 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.31 0.156 0.179 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9red Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDWA P25321 13 351 351.0 A1JE6:60406,A1JE6:60407 Allosteric,Type1 Inactive DFGin 6.3634 14.4936 BLAminus -122.88, 162.57 78.68, 90.66 -100.96, 23.62 273.2, 61.49 -59.58, -26.11 in-in in 8.7111 Saltbr-in 2.8649 HRD-in -93.71, -51.31 69.07, 9.69 in-in-out SNCiio in-out ActLoopNT-in 2.9807 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.99, 155.73 APE9-dihe-na 118.94, 161.67 APE8-dihe-in -80.46, 143.29 APE8-rot-out 194.72 APE67-dihe-in -65.57, -17.76 -53.02, -44.37 APE12-dist-in 8.1355 APE11-dist-in 11.2237 APE10-dist-in 5.7423 APE9-dist-in 4.0797 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.44 0.154 0.164 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rdw Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REJA P25321 12 351 351.0 A1JEM:60605,A1JEM:60606,A1JEM:60607 Allosteric,Type1,Allosteric Inactive DFGin 6.2324 14.4868 BLAminus -126.74, 170.31 72.72, 85.79 -95.11, 23.81 271.99, 61.49 -63.12, -25.09 in-in in 8.7773 Saltbr-in 2.7748 HRD-in -87.13, -50.88 67.77, 11.89 in-in-out SNCiio in-out ActLoopNT-in 2.908 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.08, 154.15 APE9-dihe-na 120.77, 160.5 APE8-dihe-in -80.28, 146.64 APE8-rot-out 196.83 APE67-dihe-in -64.07, -19.5 -50.27, -48.33 APE12-dist-in 8.0227 APE11-dist-in 11.1756 APE10-dist-in 5.6937 APE9-dist-in 4.0217 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.4 0.144 0.17 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rej Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SNNA P25321 13 351 351.0 BEZ:60401 Type1 Inactive DFGin 6.3179 14.5684 BLAminus -123.99, 166.66 75.94, 90.28 -99.21, 23.86 273.03, 56.25 -57.99, -30.08 in-in in 8.7995 Saltbr-in 2.708 HRD-in -85.26, -52.12 68.9, 15.2 in-in-out SNCiio in-out ActLoopNT-in 2.9021 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.87, 159.17 APE9-dihe-na 120.69, 167.55 APE8-dihe-in -88.31, 143.26 APE8-rot-out 194.47 APE67-dihe-in -64.07, -19.46 -52.28, -44.33 APE12-dist-in 8.0169 APE11-dist-in 11.2277 APE10-dist-in 5.7795 APE9-dist-in 4.1265 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.817 0.173 0.209 A 351.0 339.0 0 25 25 0 [[44, 298]] 1.0 6snn Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.5e-95 323.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1FA P25321 12 351 351.0 8ET:60403 Type1 Inactive DFGin 6.2781 14.42 BLAminus -125.76, 161.54 76.66, 90.69 -99.25, 24.03 270.12, 55.91 -61.05, -26.16 in-in in 8.6124 Saltbr-in 2.8119 HRD-in -86.34, -52.94 70.41, 12.62 in-in-out SNCiio in-out ActLoopNT-in 2.9272 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.69, 154.25 APE9-dihe-na 121.48, 156.96 APE8-dihe-in -75.85, 143.28 APE8-rot-out 195.81 APE67-dihe-in -63.37, -20.85 -47.21, -48.33 APE12-dist-in 8.0515 APE11-dist-in 11.1739 APE10-dist-in 5.7008 APE9-dist-in 4.0665 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.12 0.138 0.156 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1f Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N1HA P25321 12 351 351.0 8G2:60403 Type1 Inactive DFGin 6.2538 14.418 BLAminus -124.07, 161.77 78.11, 91.86 -99.37, 24.42 270.96, 54.95 -60.37, -25.83 in-in in 8.5499 Saltbr-in 2.7935 HRD-in -86.51, -52.46 68.86, 12.98 in-in-out SNCiio in-out ActLoopNT-in 2.9142 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -157.77, 157.58 APE9-dihe-na 112.74, 163.68 APE8-dihe-in -79.44, 140.67 APE8-rot-out 196.71 APE67-dihe-in -63.37, -21.38 -49.53, -46.05 APE12-dist-in 8.0424 APE11-dist-in 11.1779 APE10-dist-in 5.7151 APE9-dist-in 4.0574 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.18 0.137 0.158 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n1h Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3JA P25321 12 351 351.0 4NB:60402 Type1 Inactive DFGin 6.2627 14.559 BLAminus -127.12, 170.53 67.64, 82.17 -90.51, 22.12 271.33, 56.9 -61.6, -22.99 in-in in 8.8468 Saltbr-in 2.8105 HRD-in -84.57, -52.62 70.75, 13.79 in-in-out SNCiio in-out ActLoopNT-in 2.9356 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.46, 163.55 APE9-dihe-na 126.07, -167.14 APE8-dihe-in -114.74, 139.99 APE8-rot-out 192.96 APE67-dihe-in -63.96, -20.14 -47.5, -50.51 APE12-dist-in 8.1285 APE11-dist-in 11.1829 APE10-dist-in 5.6989 APE9-dist-in 3.7037 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.12 0.133 0.148 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3j Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5N3SA P25321 12 351 351.0 HBD:60401 Type1 Inactive DFGin 6.1499 14.4372 BLAminus -125.26, 171.68 71.74, 87.26 -96.68, 22.46 273.22, 56.06 -59.01, -26.75 in-in in 8.6435 Saltbr-in 2.8511 HRD-in -85.53, -52.56 69.97, 13.2 in-in-out SNCiio in-out ActLoopNT-in 2.9152 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.09, 170.83 APE9-dihe-na 117.86, -171.76 APE8-dihe-in -103.86, 138.88 APE8-rot-out 195.12 APE67-dihe-in -65.16, -19.12 -46.21, -48.93 APE12-dist-in 8.1219 APE11-dist-in 11.2071 APE10-dist-in 5.6952 APE9-dist-in 3.6672 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.14 0.129 0.148 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 5n3s Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SOXA P25321 14 351 351.0 LQ2:60401 Type1 Inactive DFGin 6.2914 14.4415 BLAminus -122.0, 165.62 75.03, 89.05 -96.95, 24.43 271.3, 57.97 -61.84, -25.55 in-in in 8.6537 Saltbr-in 2.7949 HRD-in -85.89, -52.44 69.04, 12.72 in-in-out SNCiio in-out ActLoopNT-in 2.9118 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.24, 162.39 APE9-dihe-na 125.76, -160.57 APE8-dihe-in -123.53, 144.98 APE8-rot-out 197.35 APE67-dihe-in -66.0, -18.08 -49.52, -47.22 APE12-dist-in 8.0394 APE11-dist-in 11.1533 APE10-dist-in 5.5947 APE9-dist-in 3.7106 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.38 0.147 0.168 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6sox Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPMA P25321 14 351 351.0 3AE:60401 Type1 Inactive DFGin 6.2886 14.4262 BLAminus -121.91, 163.84 77.47, 92.46 -99.73, 24.27 270.82, 55.73 -61.57, -25.41 in-in in 8.5847 Saltbr-in 2.8251 HRD-in -85.39, -51.06 67.89, 13.49 in-in-out SNCiio in-out ActLoopNT-in 2.9167 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -161.47, 161.1 APE9-dihe-na 118.54, 176.4 APE8-dihe-in -99.11, 144.76 APE8-rot-out 192.34 APE67-dihe-in -65.21, -19.46 -48.83, -47.71 APE12-dist-in 8.0367 APE11-dist-in 11.1218 APE10-dist-in 5.6321 APE9-dist-in 3.8448 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.37 0.147 0.17 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6spm Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6SPUA P25321 14 351 351.0 GAB:60405 Type1 Inactive DFGin 6.3931 14.5224 BLAminus -124.88, 173.78 70.46, 84.77 -97.04, 23.36 270.78, 58.59 -61.61, -26.89 in-in in 8.6469 Saltbr-in 2.7353 HRD-in -87.8, -49.67 67.09, 13.22 in-in-out SNCiio in-out ActLoopNT-in 2.9411 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.63, 160.29 APE9-dihe-na 125.51, -175.3 APE8-dihe-in -107.62, 144.0 APE8-rot-out 190.74 APE67-dihe-in -65.31, -18.62 -49.85, -47.63 APE12-dist-in 8.0401 APE11-dist-in 11.2233 APE10-dist-in 5.7335 APE9-dist-in 3.8932 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.39 0.165 0.184 A 353.0 338.0 0 25 25 0 [[44, 298]] 1.0 6spu Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDYA P25321 13 351 351.0 A1JE4:60407 Type1 Inactive DFGin 6.5032 14.7795 BLAminus -119.69, 163.99 72.62, 91.41 -97.65, 26.8 272.41, 58.85 -66.3, -24.47 in-in in 8.7751 Saltbr-in 3.0572 HRD-in -86.22, -51.39 68.61, 15.07 in-in-out SNCiio in-out ActLoopNT-in 2.9911 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.15, 158.18 APE9-dihe-na 117.75, 172.26 APE8-dihe-in -89.12, 142.62 APE8-rot-out 194.5 APE67-dihe-in -65.89, -17.43 -50.54, -45.34 APE12-dist-in 8.1575 APE11-dist-in 11.3384 APE10-dist-in 5.8329 APE9-dist-in 4.0454 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.5 0.184 0.206 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rdy Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REBA P25321 13 351 351.0 A1JET:60401 Type1 Inactive DFGin 6.3729 14.4269 BLAminus -124.82, 162.22 74.38, 86.67 -95.22, 22.64 270.27, 61.04 -62.16, -23.18 in-in in 8.5836 Saltbr-in 2.7104 HRD-in -85.57, -50.84 67.51, 14.65 in-in-out SNCiio in-out ActLoopNT-in 2.9047 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.96, 159.88 APE9-dihe-na 110.85, 164.82 APE8-dihe-in -83.44, 140.37 APE8-rot-out 191.04 APE67-dihe-in -61.86, -20.69 -47.36, -48.95 APE12-dist-in 8.0333 APE11-dist-in 11.1411 APE10-dist-in 5.6672 APE9-dist-in 3.9355 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.39 0.146 0.174 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9reb Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RECA P25321 13 351 351.0 A1JEU:60402 Type1 Inactive DFGin 6.2807 14.4311 BLAminus -123.32, 165.4 76.33, 88.66 -97.16, 21.64 273.57, 56.99 -61.34, -25.37 in-in in 8.6041 Saltbr-in 2.883 HRD-in -87.05, -51.85 67.25, 12.73 in-in-out SNCiio in-out ActLoopNT-in 2.9375 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -157.22, 157.7 APE9-dihe-na 114.58, 158.78 APE8-dihe-in -77.9, 144.78 APE8-rot-out 194.34 APE67-dihe-in -63.76, -21.52 -52.55, -45.26 APE12-dist-in 8.0412 APE11-dist-in 11.196 APE10-dist-in 5.6992 APE9-dist-in 4.0387 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.2 0.152 0.165 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rec Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REFA P25321 13 351 351.0 D8J:60402 Type1 Inactive DFGin 6.2503 14.6131 BLAminus -124.89, 170.59 72.31, 85.37 -94.16, 22.8 273.07, 58.11 -60.12, -25.38 in-in in 8.8919 Saltbr-in 2.7356 HRD-in -89.11, -54.6 71.98, 11.51 in-in-out SNCiio in-out ActLoopNT-in 2.9454 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -155.33, 157.11 APE9-dihe-na 116.63, 160.22 APE8-dihe-in -78.97, 144.44 APE8-rot-out 195.25 APE67-dihe-in -62.66, -21.01 -52.14, -46.04 APE12-dist-in 8.1341 APE11-dist-in 11.1957 APE10-dist-in 5.704 APE9-dist-in 4.0979 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.144 0.177 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9ref Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDVA P25321 13 351 351.0 A1JE7:60410,A1JE7:60411 Type1,Allosteric Inactive DFGin 6.2698 14.4325 BLAminus -128.08, 174.02 71.24, 86.46 -98.05, 22.19 274.06, 57.95 -62.58, -23.25 in-in in 8.6164 Saltbr-in 2.8851 HRD-in -88.5, -54.19 70.44, 9.88 in-in-out SNCiio in-out ActLoopNT-in 2.9638 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.52, 152.92 APE9-dihe-na 122.19, 162.12 APE8-dihe-in -80.5, 144.54 APE8-rot-out 193.25 APE67-dihe-in -65.71, -20.97 -51.75, -43.97 APE12-dist-in 8.0721 APE11-dist-in 11.1894 APE10-dist-in 5.7474 APE9-dist-in 4.0335 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.32 0.147 0.175 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9rdv Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RE5A P25321 13 351 351.0 A1JEY:60401,A1JEY:60402 Type1,Allosteric Inactive DFGin 6.3662 14.4036 BLAminus -125.27, 165.97 74.06, 89.04 -98.29, 23.47 275.71, 58.54 -58.28, -26.28 in-in in 8.6738 Saltbr-in 2.9443 HRD-in -85.09, -53.15 71.59, 14.35 in-in-out SNCiio in-out ActLoopNT-in 2.9386 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -160.17, 154.61 APE9-dihe-na 122.02, 168.03 APE8-dihe-in -83.24, 142.74 APE8-rot-out 202.42 APE67-dihe-in -65.84, -18.28 -53.64, -43.72 APE12-dist-in 8.1506 APE11-dist-in 11.2611 APE10-dist-in 5.782 APE9-dist-in 4.0696 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.198 0.235 A 353.0 339.0 0 25 25 0 [[44, 298]] 1.0 9re5 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REAA P25321 12 351 351.0 A1JES:60401,A1JES:60402 Type1,Allosteric Inactive DFGin 6.3101 14.3405 BLAminus -123.83, 166.44 72.66, 91.13 -99.23, 26.22 272.18, 57.96 -61.34, -25.61 in-in in 8.5784 Saltbr-in 2.748 HRD-in -86.86, -51.56 67.66, 14.6 in-in-out SNCiio in-out ActLoopNT-in 2.8985 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.49, 157.18 APE9-dihe-na 118.43, 162.88 APE8-dihe-in -80.84, 140.04 APE8-rot-out 193.72 APE67-dihe-in -64.73, -18.44 -50.69, -44.13 APE12-dist-in 8.0587 APE11-dist-in 11.2174 APE10-dist-in 5.7003 APE9-dist-in 4.039 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.52 0.182 0.207 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9rea Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9REGA P25321 12 351 351.0 A1JEP:60401,A1JEP:60402 Type1,Allosteric Inactive DFGin 6.4159 14.4433 BLAminus -118.38, 168.52 70.87, 88.51 -97.8, 23.03 272.83, 58.59 -60.46, -22.33 in-in in 8.5806 Saltbr-in 2.8704 HRD-in -87.51, -51.33 69.54, 7.76 in-in-out SNCiio in-out ActLoopNT-in 2.9211 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -158.94, 158.0 APE9-dihe-na 116.11, 163.67 APE8-dihe-in -82.8, 140.78 APE8-rot-out 193.33 APE67-dihe-in -64.93, -19.49 -46.8, -47.18 APE12-dist-in 8.0379 APE11-dist-in 11.2534 APE10-dist-in 5.7331 APE9-dist-in 3.9797 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.35 0.151 0.164 A 353.0 340.0 0 25 25 0 [[44, 298]] 1.0 9reg Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 9RDUA P25321 13 351 351.0 A1JE8:60401,A1JE8:60402,A1JE8:60403 Type1,Allosteric,Allosteric Inactive DFGin 6.3019 14.4794 BLAminus -123.63, 166.88 73.88, 91.53 -100.44, 21.89 271.16, 60.35 -61.62, -25.71 in-in in 8.7016 Saltbr-in 2.8839 HRD-in -88.41, -52.06 67.0, 12.9 in-in-out SNCiio in-out ActLoopNT-in 2.9686 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.03, 154.41 APE9-dihe-na 120.3, 161.03 APE8-dihe-in -78.42, 143.41 APE8-rot-out 195.24 APE67-dihe-in -64.91, -19.59 -51.04, -45.3 APE12-dist-in 8.0736 APE11-dist-in 11.2223 APE10-dist-in 5.7369 APE9-dist-in 4.1351 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.42 0.158 0.17 A 353.0 338.0 1 25 25 0 [[44, 298]] 1.0 9rdu Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6EH2A P25321 1 351 351.0 AMP:60401 ATPlike None DFGin 6.7638 14.9194 BLAminus -126.18, 164.33 76.56, 92.11 -105.87, 26.81 282.23, 79.7 -66.18, -22.24 in-none in 9.2259 Saltbr-none 999.0 HRD-in -87.75, -53.65 70.54, 10.24 none-in-in SNCnii in-in ActLoopNT-in 2.9384 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.34, 158.08 APE9-dihe-na 131.59, -168.87 APE8-dihe-in -114.41, 135.93 APE8-rot-in 298.36 APE67-dihe-in -58.8, -22.41 -48.5, -50.6 APE12-dist-in 8.2043 APE11-dist-in 11.4263 APE10-dist-in 5.8454 APE9-dist-in 3.7187 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.76 0.177 0.21 A 353.0 343.0 3 25 25 0 [[44, 298]] 1.0 6eh2 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 5NTJA P25321 1 351 351.0 No_ligand No_ligand None DFGin 6.7578 15.5887 BLAminus -126.6, 164.17 70.8, 88.44 -97.34, 22.68 279.05, 78.65 -62.01, -27.43 in-none in 9.318 Saltbr-none 999.0 HRD-in -87.71, -52.99 72.74, 12.02 none-in-in SNCnii in-in ActLoopNT-in 2.9259 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.35, 157.73 APE9-dihe-na 127.06, -161.94 APE8-dihe-in -121.61, 135.07 APE8-rot-in 297.67 APE67-dihe-in -60.56, -23.81 -48.81, -50.06 APE12-dist-in 8.1845 APE11-dist-in 11.5082 APE10-dist-in 5.834 APE9-dist-in 3.6606 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 1.56 0.142 0.177 A 353.0 348.0 0 25 25 0 [[44, 298]] 1.0 5ntj Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERUA P25321 1 351 351.0 No_ligand No_ligand None DFGin 6.7077 15.3522 BLAminus -122.01, 161.76 78.09, 83.83 -91.35, 27.07 283.0, 77.27 -61.22, -29.16 in-none in 9.3238 Saltbr-none 999.0 HRD-in -85.44, -56.28 74.88, 7.63 none-in-in SNCnii in-in ActLoopNT-in 2.8885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.17, 161.42 APE9-dihe-na 121.37, -170.91 APE8-dihe-in -112.44, 135.97 APE8-rot-in 301.67 APE67-dihe-in -61.32, -23.67 -50.09, -48.07 APE12-dist-in 8.2425 APE11-dist-in 11.5143 APE10-dist-in 5.8561 APE9-dist-in 3.6262 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.15 0.207 0.245 A 353.0 348.0 1 25 25 0 [[44, 298]] 1.0 6eru Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6ERVA P25321 1 351 351.0 No_ligand No_ligand None DFGin 6.7146 15.3924 BLAminus -125.08, 156.65 78.53, 86.88 -92.73, 25.79 280.28, 78.54 -65.37, -20.87 in-none in 9.2341 Saltbr-none 999.0 HRD-in -86.89, -53.48 76.44, 7.72 none-in-in SNCnii in-in ActLoopNT-in 2.9464 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.6, 158.99 APE9-dihe-na 121.28, -168.45 APE8-dihe-in -116.16, 134.01 APE8-rot-in 298.45 APE67-dihe-in -57.32, -26.83 -47.6, -49.92 APE12-dist-in 8.2352 APE11-dist-in 11.4876 APE10-dist-in 5.9397 APE9-dist-in 3.6445 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.06 0.181 0.217 A 353.0 341.0 0 25 25 0 [[44, 298]] 1.0 6erv Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 6Y2OA P25321 1 351 351.0 O72:60406 Type1 None DFGin 6.4228 14.1352 BLAminus -118.81, 164.94 68.54, 89.57 -98.17, 23.6 280.79, 62.09 -51.58, -34.71 in-none in 8.664 Saltbr-none 999.0 HRD-in -99.33, -52.87 71.55, 6.25 none-in-in SNCnii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.56, 161.43 APE9-dihe-na 131.48, -155.68 APE8-dihe-in -122.0, 132.63 APE8-rot-in 297.96 APE67-dihe-in -62.6, -21.6 -48.71, -46.53 APE12-dist-in 8.1468 APE11-dist-in 11.4733 APE10-dist-in 5.9727 APE9-dist-in 3.6487 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.01 0.223 0.254 A 353.0 351.0 0 25 25 0 [[44, 298]] 1.0 6y2o Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_CRIGR 7BB0A P25321 1 351 351.0 T7W:60401 Type1 None DFGin 6.693 15.1674 BLAminus -117.12, 156.8 84.07, 107.01 -120.86, 24.94 282.89, 80.35 -68.76, -26.06 in-none in 9.3444 Saltbr-none 999.0 HRD-in -88.11, -52.74 73.76, 5.71 none-in-in SNCnii in-in ActLoopNT-in 3.0151 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.84, 156.52 APE9-dihe-na 126.29, -168.37 APE8-dihe-in -114.04, 132.32 APE8-rot-in 303.32 APE67-dihe-in -60.17, -25.3 -47.27, -49.42 APE12-dist-in 8.2705 APE11-dist-in 11.5229 APE10-dist-in 5.9799 APE9-dist-in 3.7589 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 1.75 0.203 0.235 A 353.0 347.0 0 25 25 0 [[44, 298]] 1.0 7bb0 Cricetulus griseus AGC_PRKACA_CRIGR AGC 6.6e-95 323.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4O21A P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 6.0367 14.4393 BLAminus -125.27, 173.53 70.53, 83.75 -96.26, 25.58 272.04, 54.28 -57.91, -27.19 in-in in 8.9531 Saltbr-in 2.7155 HRD-in -83.95, -57.84 75.15, 8.54 in-in-in SNCiii in-in ActLoopNT-in 2.9043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.15, 164.3 APE9-dihe-na 125.14, -151.92 APE8-dihe-in -125.51, 129.66 APE8-rot-in 308.07 APE67-dihe-in -63.53, -19.17 -43.91, -48.76 APE12-dist-in 8.0396 APE11-dist-in 11.4602 APE10-dist-in 5.9112 APE9-dist-in 3.4511 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.17 0.215 A 342.0 336.0 0 25 25 0 [[44, 298]] 1.0 4o21 Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7E11A P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 6.205 14.4514 BLAminus -127.38, -169.19 58.28, 74.22 -96.53, 30.74 276.22, 81.09 -66.46, -21.72 in-in in 9.0533 Saltbr-in 2.5511 HRD-in -91.79, -53.23 62.57, 24.02 in-in-in SNCiii in-in ActLoopNT-in 3.1289 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.39, 155.98 APE9-dihe-na 134.96, -158.62 APE8-dihe-in -113.95, 132.34 APE8-rot-in 301.67 APE67-dihe-in -76.79, -1.28 -53.37, -39.68 APE12-dist-in 8.3091 APE11-dist-in 11.1349 APE10-dist-in 5.7098 APE9-dist-in 3.659 None TPO198,SEP339 TPO198,SEP339 XRAY 3.43 0.262 0.317 A 338.0 337.0 0 25 25 0 [[44, 298]] 1.0 7e11 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3PVBA P05132 7 351 351.0 ANP:60400 ATPlike Active DFGin 5.2614 14.1066 BLAminus -138.85, 171.16 63.11, 82.89 -89.43, -59.95 273.17, 54.43 27.14, -66.26 in-in in 8.6853 Saltbr-in 3.4757 HRD-in -84.36, -35.8 62.24, -18.82 in-in-in SNCiii in-in ActLoopNT-in 3.2175 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -177.84, 157.88 APE9-dihe-na 132.55, -154.74 APE8-dihe-in -122.19, 108.01 APE8-rot-in 318.81 APE67-dihe-in -60.75, -2.24 -13.41, -60.33 APE12-dist-in 7.7331 APE11-dist-in 10.5794 APE10-dist-in 5.5109 APE9-dist-in 4.0421 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 3.3 0.242 0.29 A 345.0 345.0 0 25 25 0 [[44, 298]] 1.0 3pvb Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1BKXA P05132 13 351 351.0 AMP:60351 ATPlike Active DFGin 6.1602 13.9145 BLAminus -117.09, 179.26 61.99, 75.16 -83.18, 21.65 286.96, 82.43 -60.51, -17.53 in-in in 8.7242 Saltbr-in 2.6583 HRD-in -99.39, -38.31 69.2, -9.22 in-in-in SNCiii in-in ActLoopNT-in 3.4681 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.44, 150.62 APE9-dihe-na 113.99, 166.84 APE8-dihe-in -65.88, 134.1 APE8-rot-in 334.22 APE67-dihe-in -70.66, -34.65 -48.92, -27.08 APE12-dist-in 8.2835 APE11-dist-in 11.3505 APE10-dist-in 5.7038 APE9-dist-in 4.2848 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.6 0.219 0.34 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1bkx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1L3RE P05132 2 351 351.0 ADP:60381 ATPlike Active DFGin 5.7538 14.4402 BLAminus -119.14, -174.46 57.18, 81.19 -93.77, 20.31 270.88, 52.04 -50.0, -37.57 in-in in 9.0231 Saltbr-in 2.7924 HRD-in -82.45, -54.36 70.16, 7.26 in-in-in SNCiii in-in ActLoopNT-in 2.9201 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.84, 161.06 APE9-dihe-na 132.7, -149.01 APE8-dihe-in -131.06, 132.91 APE8-rot-in 298.56 APE67-dihe-in -55.27, -27.25 -33.24, -62.94 APE12-dist-in 8.1978 APE11-dist-in 11.2333 APE10-dist-in 5.8253 APE9-dist-in 3.3679 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.0 0.205 0.232 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1l3r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2QCSA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.648 14.2907 BLAminus -119.78, 176.88 65.56, 77.31 -85.05, 19.39 273.35, 51.28 -44.32, -42.51 in-in in 8.7843 Saltbr-in 2.6377 HRD-in -93.14, -54.78 73.52, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.7354 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.52, 149.74 APE9-dihe-na 148.64, -142.53 APE8-dihe-in -132.36, 132.12 APE8-rot-in 297.18 APE67-dihe-in -64.67, -25.45 -36.74, -53.73 APE12-dist-in 8.133 APE11-dist-in 11.3207 APE10-dist-in 5.8515 APE9-dist-in 3.5726 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.194 0.225 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 2qcs Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3FJQE P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.6709 14.4589 BLAminus -119.42, 178.78 63.28, 80.04 -91.81, 23.31 270.73, 57.82 -56.09, -30.86 in-in in 9.1494 Saltbr-in 2.8344 HRD-in -91.33, -52.39 67.42, 13.87 in-in-in SNCiii in-in ActLoopNT-in 2.9056 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.19, 160.44 APE9-dihe-na 133.42, -155.21 APE8-dihe-in -125.75, 136.86 APE8-rot-in 304.0 APE67-dihe-in -61.0, -22.29 -48.87, -49.39 APE12-dist-in 8.0863 APE11-dist-in 11.4084 APE10-dist-in 5.8377 APE9-dist-in 3.5179 None TPO198,SEP339 TPO198,SEP339 XRAY 1.6 0.179 0.205 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 3fjq Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3IDBA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.3459 14.4126 BLAminus -121.17, -175.1 59.7, 79.28 -94.34, 24.01 267.69, 48.22 -48.56, -33.02 in-in in 8.8455 Saltbr-in 2.694 HRD-in -80.07, -50.75 69.18, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.9896 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.99, 160.5 APE9-dihe-na 138.4, -150.07 APE8-dihe-in -124.64, 132.33 APE8-rot-in 296.41 APE67-dihe-in -59.26, -21.93 -30.94, -63.4 APE12-dist-in 8.1019 APE11-dist-in 11.5726 APE10-dist-in 6.0684 APE9-dist-in 3.4448 None TPO198,SEP339 TPO198,SEP339 XRAY 1.62 0.206 0.23 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 3idb Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3IDCA P05132 9 351 351.0 ANP:60450 ATPlike Active DFGin 5.079 14.4716 BLAminus -127.31, 174.57 68.22, 96.34 -111.15, 30.11 265.57, 49.45 -62.75, -22.0 in-in in 8.6423 Saltbr-in 3.0306 HRD-in -69.04, -44.03 64.09, 13.38 in-in-in SNCiii in-in ActLoopNT-in 2.8561 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.35, 157.69 APE9-dihe-na 142.7, -132.16 APE8-dihe-in -139.58, 115.88 APE8-rot-in 293.03 APE67-dihe-in -54.66, -5.54 -16.73, -78.3 APE12-dist-in 7.8437 APE11-dist-in 11.3725 APE10-dist-in 6.1644 APE9-dist-in 3.6752 None TPO198,SEP339 TPO198,SEP339 XRAY 2.7 0.241 0.319 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 3idc Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DG0E P05132 11 351 351.0 ANP:60402 ATPlike Active DFGin 5.5834 14.3418 BLAminus -118.87, 179.66 65.44, 79.89 -93.34, 25.25 272.35, 58.42 -52.71, -36.39 in-in in 8.955 Saltbr-in 2.6989 HRD-in -84.35, -52.45 74.02, 7.32 in-in-in SNCiii in-in ActLoopNT-in 2.8946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.07, 161.1 APE9-dihe-na 130.81, -146.6 APE8-dihe-in -130.07, 130.32 APE8-rot-in 303.85 APE67-dihe-in -61.09, -22.5 -44.14, -49.24 APE12-dist-in 8.0079 APE11-dist-in 11.4975 APE10-dist-in 5.8998 APE9-dist-in 3.3886 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.196 0.228 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 4dg0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH1A P05132 16 351 351.0 ATP:60402 ATPlike Active DFGin 6.2341 14.3802 BLAminus -130.7, 167.11 69.97, 89.08 -103.01, 26.92 273.93, 57.95 -52.62, -33.38 in-in in 8.9305 Saltbr-in 3.0104 HRD-in -75.69, -51.31 65.95, 10.85 in-in-in SNCiii in-in ActLoopNT-in 2.8868 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.97, 163.54 APE9-dihe-na 128.87, -151.55 APE8-dihe-in -123.52, 135.53 APE8-rot-in 304.09 APE67-dihe-in -55.69, -26.94 -40.23, -59.36 APE12-dist-in 8.1686 APE11-dist-in 11.5574 APE10-dist-in 5.9503 APE9-dist-in 3.5446 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.199 0.234 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH3A P05132 16 351 351.0 ATP:60403 ATPlike Active DFGin 5.9838 14.3792 BLAminus -125.47, 176.75 61.82, 79.89 -92.16, 24.39 276.69, 54.39 -43.39, -47.09 in-in in 9.021 Saltbr-in 2.7225 HRD-in -82.56, -48.22 66.04, -2.33 in-in-in SNCiii in-in ActLoopNT-in 2.9311 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 165.55 APE9-dihe-na 126.96, -149.27 APE8-dihe-in -125.58, 130.88 APE8-rot-in 307.35 APE67-dihe-in -57.88, -25.54 -37.95, -56.15 APE12-dist-in 8.2249 APE11-dist-in 11.5925 APE10-dist-in 6.1036 APE9-dist-in 3.74 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.203 0.233 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH5A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 6.1214 14.3392 BLAminus -125.12, -179.76 61.4, 85.13 -97.61, 27.77 279.05, 62.21 -46.99, -44.52 in-in in 9.0432 Saltbr-in 2.5524 HRD-in -77.92, -53.51 67.68, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.9684 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.88, 153.17 APE9-dihe-na 132.88, -161.89 APE8-dihe-in -112.07, 131.8 APE8-rot-in 304.21 APE67-dihe-in -57.01, -23.17 -41.47, -55.69 APE12-dist-in 8.2186 APE11-dist-in 11.6017 APE10-dist-in 6.0711 APE9-dist-in 3.87 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.187 0.222 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH7A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.5738 14.3492 BLAminus -124.43, -175.45 59.33, 78.79 -93.54, 24.71 270.97, 54.79 -50.12, -38.03 in-in in 9.0247 Saltbr-in 2.7242 HRD-in -76.49, -50.79 66.5, 11.01 in-in-in SNCiii in-in ActLoopNT-in 2.9607 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.18, 162.39 APE9-dihe-na 131.3, -151.54 APE8-dihe-in -126.44, 134.15 APE8-rot-in 300.19 APE67-dihe-in -56.38, -25.77 -37.48, -60.34 APE12-dist-in 8.0928 APE11-dist-in 11.4546 APE10-dist-in 5.87 APE9-dist-in 3.4166 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.8 0.179 0.194 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DH8A P05132 16 351 351.0 ANP:60403 ATPlike Active DFGin 5.9006 14.014 BLAminus -123.95, -176.77 59.01, 85.18 -98.8, 24.84 279.52, 63.26 -51.76, -30.5 in-in in 8.8003 Saltbr-in 2.7128 HRD-in -77.99, -56.65 70.43, 3.78 in-in-in SNCiii in-in ActLoopNT-in 2.968 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.95, 158.57 APE9-dihe-na 135.16, -154.79 APE8-dihe-in -124.8, 132.89 APE8-rot-in 296.53 APE67-dihe-in -58.95, -25.2 -38.46, -56.52 APE12-dist-in 8.1451 APE11-dist-in 11.4751 APE10-dist-in 5.904 APE9-dist-in 3.5115 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.3 0.155 0.188 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 4dh8 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4HPTE P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.7482 14.4242 BLAminus -115.4, 178.03 67.73, 81.09 -92.11, 21.69 273.09, 55.37 -58.71, -29.4 in-in in 9.0532 Saltbr-in 2.6604 HRD-in -90.64, -54.09 71.81, 9.39 in-in-in SNCiii in-in ActLoopNT-in 2.8739 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.27, 162.98 APE9-dihe-na 129.56, -147.32 APE8-dihe-in -127.39, 129.92 APE8-rot-in 299.02 APE67-dihe-in -63.31, -27.9 -40.61, -49.36 APE12-dist-in 8.0686 APE11-dist-in 11.3854 APE10-dist-in 5.8255 APE9-dist-in 3.5734 None TPO198,SEP339 TPO198,SEP339 XRAY 2.15 0.189 0.228 E 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4hpt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4HPUE P05132 13 351 351.0 ANP:60402 ATPlike Active DFGin 5.5508 14.4067 BLAminus -117.63, -178.61 63.83, 78.8 -92.22, 24.46 271.46, 55.23 -53.69, -32.94 in-in in 9.0306 Saltbr-in 2.6916 HRD-in -87.73, -52.35 74.85, 8.01 in-in-in SNCiii in-in ActLoopNT-in 2.9145 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.41, 162.17 APE9-dihe-na 134.1, -149.11 APE8-dihe-in -128.69, 136.04 APE8-rot-in 297.56 APE67-dihe-in -58.67, -24.48 -48.3, -49.81 APE12-dist-in 8.0634 APE11-dist-in 11.5067 APE10-dist-in 5.8865 APE9-dist-in 3.4033 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.173 0.194 E 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 4hpu Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 5JR7A P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.7387 13.6907 BLAminus -145.14, 176.28 64.37, 76.68 -85.75, 18.89 294.14, 59.99 -43.66, -41.86 in-in in 8.6743 Saltbr-in 2.7095 HRD-in -93.38, -54.67 74.91, 7.39 in-in-in SNCiii in-in ActLoopNT-in 2.945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.46, 148.2 APE9-dihe-na 147.95, -159.28 APE8-dihe-in -109.66, 131.32 APE8-rot-in 258.88 APE67-dihe-in -65.5, -25.8 -38.64, -53.47 APE12-dist-in 8.0144 APE11-dist-in 10.772 APE10-dist-in 5.5284 APE9-dist-in 3.8782 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 5JR7C P05132 14 351 351.0 ADP:60400 ATPlike Active DFGin 5.8995 13.1635 BLAminus -138.79, 176.44 54.89, 86.07 -89.1, 7.67 290.95, 62.79 -41.83, -37.01 in-in in 8.1848 Saltbr-in 3.1954 HRD-in -79.11, -50.37 72.48, -21.93 in-in-in SNCiii in-in ActLoopNT-in 2.8194 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.28, 123.46 APE9-dihe-na 160.31, -160.86 APE8-dihe-in -110.49, 124.04 APE8-rot-in 311.35 APE67-dihe-in -70.47, -24.34 -45.9, -42.95 APE12-dist-in 8.1626 APE11-dist-in 10.628 APE10-dist-in 5.0018 APE9-dist-in 4.2619 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 3.56 0.269 0.322 C 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 5jr7 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7UJXE P05132 16 351 351.0 ADP:60401 ATPlike Active DFGin 5.731 14.3568 BLAminus -121.93, 179.51 64.92, 83.56 -91.91, 29.5 277.22, 63.03 -64.62, -28.12 in-in in 9.1028 Saltbr-in 2.8121 HRD-in -86.19, -57.72 74.11, 16.74 in-in-in SNCiii in-in ActLoopNT-in 2.9312 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.48, 155.47 APE9-dihe-na 127.23, -161.98 APE8-dihe-in -111.77, 133.52 APE8-rot-in 302.04 APE67-dihe-in -65.07, -18.97 -50.87, -44.77 APE12-dist-in 8.1906 APE11-dist-in 11.5001 APE10-dist-in 5.9613 APE9-dist-in 4.0077 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.133 0.176 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 7ujx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7V0GE P05132 17 351 351.0 ADP:60401 ATPlike Active DFGin 5.7389 14.3189 BLAminus -119.5, 177.58 67.43, 82.74 -91.45, 25.21 276.8, 64.92 -62.46, -26.34 in-in in 9.0699 Saltbr-in 2.8017 HRD-in -88.93, -50.41 71.3, 15.33 in-in-in SNCiii in-in ActLoopNT-in 2.9568 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.52, 156.77 APE9-dihe-na 130.04, -162.37 APE8-dihe-in -114.97, 131.2 APE8-rot-in 299.52 APE67-dihe-in -60.0, -22.75 -47.18, -49.61 APE12-dist-in 8.1738 APE11-dist-in 11.5422 APE10-dist-in 6.0368 APE9-dist-in 3.9649 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.118 0.163 E 350.0 335.0 0 25 25 0 [[44, 298]] 1.0 7v0g Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFXE P05132 2 351 351.0 ANP:60402 ATPlike Active DFGin 5.5242 14.2861 BLAminus -116.71, -179.39 66.13, 78.01 -91.08, 23.34 272.63, 51.46 -56.59, -32.27 in-in in 8.8728 Saltbr-in 2.7287 HRD-in -88.99, -54.58 73.79, 11.03 in-in-in SNCiii in-in ActLoopNT-in 2.9336 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.69, 159.64 APE9-dihe-na 138.16, -148.52 APE8-dihe-in -130.4, 136.32 APE8-rot-in 296.63 APE67-dihe-in -59.91, -24.0 -47.38, -49.37 APE12-dist-in 8.0462 APE11-dist-in 11.4097 APE10-dist-in 5.8188 APE9-dist-in 3.3923 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.35 0.157 0.179 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4dfx Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4X6RA P05132 2 351 351.0 ATP:60402 ATPlike Active DFGin 6.1334 14.2323 BLAminus -118.92, 178.27 64.18, 79.91 -89.21, 11.01 274.1, 55.74 -49.19, -34.95 in-in in 8.8037 Saltbr-in 2.7288 HRD-in -85.13, -60.38 77.67, -7.87 in-in-in SNCiii in-in ActLoopNT-in 2.7182 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.34, 156.01 APE9-dihe-na 147.33, -149.7 APE8-dihe-in -130.56, 138.51 APE8-rot-in 291.09 APE67-dihe-in -61.2, -24.8 -52.44, -47.95 APE12-dist-in 8.281 APE11-dist-in 11.2462 APE10-dist-in 5.8359 APE9-dist-in 3.6632 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.186 0.234 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4x6r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3X2UA P05132 13 351 351.0 ATP:60501 ATPlike Active DFGin 6.1271 14.5072 BLAminus -122.24, 178.58 59.36, 87.7 -101.54, 25.28 272.61, 50.83 -59.45, -24.26 in-in in 9.2723 Saltbr-in 2.7882 HRD-in -89.58, -50.62 64.84, 17.58 in-in-in SNCiii in-in ActLoopNT-in 2.9297 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.25, 158.3 APE9-dihe-na 134.88, -147.54 APE8-dihe-in -130.4, 131.58 APE8-rot-in 300.12 APE67-dihe-in -61.26, -14.4 -40.08, -55.22 APE12-dist-in 7.9122 APE11-dist-in 11.1375 APE10-dist-in 5.6863 APE9-dist-in 3.4266 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.4 0.202 0.239 A 357.0 339.0 0 25 25 0 [[44, 298]] 1.0 3x2u Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3X2VA P05132 18 351 351.0 ATP:60403 ATPlike Active DFGin 5.5167 14.1516 BLAminus -116.69, -175.94 62.92, 80.3 -91.77, 26.26 271.42, 55.44 -51.78, -39.79 in-in in 8.7552 Saltbr-in 2.6541 HRD-in -92.08, -50.84 67.69, 17.07 in-in-in SNCiii in-in ActLoopNT-in 2.8813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.85, 164.45 APE9-dihe-na 134.14, -152.5 APE8-dihe-in -130.83, 133.42 APE8-rot-in 299.77 APE67-dihe-in -58.82, -21.18 -48.96, -48.11 APE12-dist-in 7.9982 APE11-dist-in 11.3458 APE10-dist-in 5.7964 APE9-dist-in 3.4149 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.77 0.185 0.23 A 357.0 334.0 0 25 25 0 [[44, 298]] 1.0 3x2v Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3X2WA P05132 13 351 351.0 ATP:60403 ATPlike Active DFGin 5.6602 14.3902 BLAminus -121.01, -177.68 63.51, 77.56 -90.4, 24.79 270.4, 59.29 -61.83, -28.06 in-in in 8.8217 Saltbr-in 2.6324 HRD-in -81.34, -52.24 70.22, 11.48 in-in-in SNCiii in-in ActLoopNT-in 2.9059 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.19, 162.39 APE9-dihe-na 132.4, -151.44 APE8-dihe-in -129.91, 133.08 APE8-rot-in 300.2 APE67-dihe-in -60.45, -20.83 -45.18, -51.38 APE12-dist-in 8.001 APE11-dist-in 11.4403 APE10-dist-in 5.911 APE9-dist-in 3.4498 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.165 0.198 A 357.0 339.0 0 25 25 0 [[44, 298]] 1.0 3x2w Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IACA P05132 16 351 351.0 ACP:60403 ATPlike Active DFGin 5.7549 14.3121 BLAminus -125.73, -177.16 59.8, 78.08 -94.31, 23.06 273.35, 54.81 -46.36, -37.92 in-in in 8.8851 Saltbr-in 2.7214 HRD-in -73.57, -53.97 72.67, 5.23 in-in-in SNCiii in-in ActLoopNT-in 2.9421 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.57, 156.93 APE9-dihe-na 137.19, -153.99 APE8-dihe-in -123.03, 128.21 APE8-rot-in 300.87 APE67-dihe-in -59.06, -23.99 -31.47, -61.7 APE12-dist-in 8.1573 APE11-dist-in 11.5147 APE10-dist-in 5.9848 APE9-dist-in 3.5015 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.15 0.181 0.212 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iac Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IADA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.6579 14.362 BLAminus -130.04, -179.13 63.0, 77.66 -87.34, 22.78 276.11, 53.54 -55.12, -31.28 in-in in 9.0855 Saltbr-in 2.8296 HRD-in -93.22, -52.19 70.15, 14.14 in-in-in SNCiii in-in ActLoopNT-in 2.9352 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.54, 160.6 APE9-dihe-na 133.65, -143.98 APE8-dihe-in -130.05, 134.5 APE8-rot-in 298.49 APE67-dihe-in -67.08, -22.74 -48.94, -44.54 APE12-dist-in 8.0511 APE11-dist-in 11.5496 APE10-dist-in 6.0873 APE9-dist-in 3.5214 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.189 0.243 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4iad Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAFA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.9427 14.1301 BLAminus -121.29, 178.82 64.06, 84.8 -98.0, 27.2 281.56, 65.38 -51.93, -33.25 in-in in 8.8711 Saltbr-in 2.6687 HRD-in -76.48, -53.65 65.3, 9.94 in-in-in SNCiii in-in ActLoopNT-in 2.9738 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.4, 160.11 APE9-dihe-na 128.66, -151.44 APE8-dihe-in -123.86, 135.06 APE8-rot-in 298.27 APE67-dihe-in -57.84, -25.84 -42.55, -55.44 APE12-dist-in 8.1629 APE11-dist-in 11.523 APE10-dist-in 5.9727 APE9-dist-in 3.5632 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.16 0.192 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iaf Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAIA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.4651 14.5028 BLAminus -125.1, 176.4 64.24, 81.88 -90.74, 22.64 269.91, 49.4 -55.45, -35.99 in-in in 9.1007 Saltbr-in 2.7138 HRD-in -91.06, -49.32 68.79, 15.16 in-in-in SNCiii in-in ActLoopNT-in 2.9385 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.75, 156.86 APE9-dihe-na 141.29, -148.36 APE8-dihe-in -128.24, 130.8 APE8-rot-in 300.02 APE67-dihe-in -62.27, -23.0 -47.39, -47.75 APE12-dist-in 7.9453 APE11-dist-in 11.4584 APE10-dist-in 5.8673 APE9-dist-in 3.6084 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.55 0.171 0.209 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iai Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAKA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.7052 14.5691 BLAminus -126.92, 179.61 63.08, 81.74 -90.27, 23.65 270.26, 53.44 -59.05, -31.45 in-in in 8.9848 Saltbr-in 2.7471 HRD-in -94.54, -49.89 67.85, 16.15 in-in-in SNCiii in-in ActLoopNT-in 2.9098 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.92, 164.74 APE9-dihe-na 131.87, -148.57 APE8-dihe-in -130.85, 127.67 APE8-rot-in 297.68 APE67-dihe-in -61.28, -21.91 -43.91, -50.7 APE12-dist-in 7.9618 APE11-dist-in 11.4433 APE10-dist-in 5.9794 APE9-dist-in 3.5447 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.6 0.185 0.222 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4iak Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAYA P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.806 14.2571 BLAminus -131.74, 174.05 67.76, 85.89 -95.28, 20.31 273.12, 61.73 -48.17, -36.05 in-in in 9.0392 Saltbr-in 2.9406 HRD-in -89.87, -50.65 68.98, 10.01 in-in-in SNCiii in-in ActLoopNT-in 3.055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.39, 159.46 APE9-dihe-na 132.54, -148.24 APE8-dihe-in -127.91, 130.95 APE8-rot-in 300.76 APE67-dihe-in -63.09, -19.35 -45.58, -49.88 APE12-dist-in 8.0893 APE11-dist-in 11.4657 APE10-dist-in 5.991 APE9-dist-in 3.8226 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.182 0.227 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 4iay Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IAZA P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 6.1438 14.6353 BLAminus -132.33, 171.23 62.84, 84.78 -94.94, 21.85 278.49, 61.31 -54.74, -28.93 in-in in 9.2192 Saltbr-in 2.747 HRD-in -95.03, -54.93 73.76, 14.73 in-in-in SNCiii in-in ActLoopNT-in 3.017 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.57, 164.74 APE9-dihe-na 127.12, -150.82 APE8-dihe-in -127.02, 138.46 APE8-rot-in 303.51 APE67-dihe-in -63.11, -25.72 -51.71, -47.83 APE12-dist-in 7.9634 APE11-dist-in 11.5144 APE10-dist-in 5.9788 APE9-dist-in 3.5741 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.85 0.201 0.248 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4iaz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IB0A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.7134 14.4391 BLAminus -123.68, 176.86 65.62, 82.22 -94.42, 18.76 272.15, 51.12 -47.84, -35.86 in-in in 9.0645 Saltbr-in 3.0231 HRD-in -84.67, -55.05 71.31, 12.11 in-in-in SNCiii in-in ActLoopNT-in 2.8861 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.67, 157.49 APE9-dihe-na 139.08, -144.95 APE8-dihe-in -131.16, 131.55 APE8-rot-in 306.17 APE67-dihe-in -61.31, -24.54 -46.0, -48.78 APE12-dist-in 8.0592 APE11-dist-in 11.5164 APE10-dist-in 5.9694 APE9-dist-in 3.6924 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.87 0.219 0.287 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4ib0 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IB1A P05132 14 351 351.0 ADP:60403 ATPlike Active DFGin 5.6556 14.4434 BLAminus -126.58, 171.72 66.62, 80.69 -90.79, 23.58 274.18, 53.88 -53.03, -31.34 in-in in 9.1208 Saltbr-in 2.6907 HRD-in -82.93, -51.49 69.93, 14.85 in-in-in SNCiii in-in ActLoopNT-in 2.9803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.64, 163.58 APE9-dihe-na 133.1, -151.37 APE8-dihe-in -125.38, 138.08 APE8-rot-in 304.1 APE67-dihe-in -60.15, -23.69 -50.01, -49.7 APE12-dist-in 7.9604 APE11-dist-in 11.404 APE10-dist-in 5.9611 APE9-dist-in 3.6354 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.63 0.196 0.223 A 356.0 338.0 0 25 25 0 [[44, 298]] 1.0 4ib1 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4IB3A P05132 13 351 351.0 ADP:60401 ATPlike Active DFGin 5.973 14.2146 BLAminus -125.69, 173.12 66.37, 84.97 -98.59, 21.41 276.57, 60.51 -51.27, -29.52 in-in in 8.9902 Saltbr-in 2.7598 HRD-in -77.27, -49.79 61.58, 13.48 in-in-in SNCiii in-in ActLoopNT-in 2.8695 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.06, 160.46 APE9-dihe-na 127.6, -161.57 APE8-dihe-in -110.98, 129.89 APE8-rot-in 305.68 APE67-dihe-in -58.89, -23.07 -39.61, -54.94 APE12-dist-in 8.0781 APE11-dist-in 11.5224 APE10-dist-in 5.9229 APE9-dist-in 3.5677 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.2 0.182 0.228 A 356.0 339.0 0 25 25 0 [[44, 298]] 1.0 4ib3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4XW4A P05132 15 351 351.0 ANP:60403 ATPlike Active DFGin 5.673 14.5624 BLAminus -117.82, -177.44 65.15, 79.34 -92.69, 26.58 269.45, 57.64 -61.99, -28.36 in-in in 8.9306 Saltbr-in 2.8579 HRD-in -86.05, -50.94 67.2, 15.72 in-in-in SNCiii in-in ActLoopNT-in 3.0139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.62, 159.69 APE9-dihe-na 135.12, -140.29 APE8-dihe-in -136.84, 125.12 APE8-rot-in 301.75 APE67-dihe-in -61.52, -26.6 -45.5, -44.66 APE12-dist-in 7.961 APE11-dist-in 11.4188 APE10-dist-in 5.9353 APE9-dist-in 3.6644 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.82 0.183 0.24 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4xw4 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4XW5A P05132 15 351 351.0 ATP:60403 ATPlike Active DFGin 5.971 14.2215 BLAminus -131.24, 177.82 59.66, 87.19 -93.08, 25.08 282.37, 63.43 -53.77, -29.24 in-in in 9.2129 Saltbr-in 2.673 HRD-in -90.87, -48.94 63.52, 13.92 in-in-in SNCiii in-in ActLoopNT-in 2.8122 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.24, 155.03 APE9-dihe-na 137.47, -160.98 APE8-dihe-in -110.31, 133.6 APE8-rot-in 304.05 APE67-dihe-in -58.14, -25.36 -48.87, -50.12 APE12-dist-in 8.0264 APE11-dist-in 11.6005 APE10-dist-in 6.1002 APE9-dist-in 3.9217 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.95 0.185 0.252 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4xw5 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4XW6A P05132 15 351 351.0 ADP:60403 ATPlike Active DFGin 5.9823 14.431 BLAminus -130.68, 178.48 65.03, 84.15 -99.24, 23.41 276.01, 56.03 -60.45, -23.49 in-in in 9.1497 Saltbr-in 2.7348 HRD-in -94.59, -52.61 68.2, 15.9 in-in-in SNCiii in-in ActLoopNT-in 2.7909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.91, 154.59 APE9-dihe-na 136.7, -154.91 APE8-dihe-in -121.39, 127.95 APE8-rot-in 293.9 APE67-dihe-in -62.75, -24.38 -45.59, -46.76 APE12-dist-in 8.0512 APE11-dist-in 11.6319 APE10-dist-in 6.051 APE9-dist-in 3.787 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.9 0.186 0.265 A 356.0 337.0 0 25 25 0 [[44, 298]] 1.0 4xw6 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6E21A P05132 16 351 351.0 ADP:60403 ATPlike Active DFGin 5.5937 14.0551 BLAminus -122.61, 176.37 63.02, 83.41 -94.2, 28.27 284.3, 46.09 -48.88, -41.13 in-in in 9.0287 Saltbr-in 2.6073 HRD-in -74.35, -56.8 67.48, 11.51 in-in-in SNCiii in-in ActLoopNT-in 2.9072 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.7, 159.01 APE9-dihe-na 131.41, -152.84 APE8-dihe-in -125.29, 130.56 APE8-rot-in 303.23 APE67-dihe-in -58.42, -25.04 -35.36, -60.06 APE12-dist-in 8.0433 APE11-dist-in 11.5842 APE10-dist-in 6.0224 APE9-dist-in 3.5802 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.187 0.217 A 356.0 336.0 0 25 25 0 [[44, 298]] 1.0 6e21 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7E0ZA P05132 14 351 351.0 ANP:60401 ATPlike Active DFGin 5.5662 13.8842 BLAminus -118.85, -174.47 59.93, 79.47 -94.43, 25.89 275.59, 63.85 -59.78, -31.6 in-in in 8.6241 Saltbr-in 2.9777 HRD-in -96.8, -56.38 78.26, 13.74 in-in-in SNCiii in-in ActLoopNT-in 2.9292 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.91, 162.74 APE9-dihe-na 131.67, -149.57 APE8-dihe-in -131.04, 130.65 APE8-rot-in 294.41 APE67-dihe-in -63.42, -12.5 -45.48, -52.1 APE12-dist-in 7.8999 APE11-dist-in 11.1823 APE10-dist-in 5.721 APE9-dist-in 3.4 None TPO198,SEP339 TPO198,SEP339 XRAY 2.162 0.184 0.228 A 358.0 337.0 0 25 25 0 [[44, 298]] 1.0 7e0z Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DG3E P05132 15 351 351.0 ANP:60401 ATPlike Active DFGin 5.4812 14.3421 BLAminus -115.99, -176.62 61.62, 77.98 -90.25, 24.84 270.29, 54.4 -55.44, -35.73 in-in in 8.842 Saltbr-in 2.6947 HRD-in -87.1, -53.93 73.82, 10.76 in-in-in SNCiii in-in ActLoopNT-in 2.8817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.46, 161.61 APE9-dihe-na 135.41, -150.07 APE8-dihe-in -129.52, 135.22 APE8-rot-in 300.3 APE67-dihe-in -58.11, -23.91 -46.28, -51.67 APE12-dist-in 8.1435 APE11-dist-in 11.4816 APE10-dist-in 5.8864 APE9-dist-in 3.4048 R337A SEP140,TPO198 SEP140,TPO198 XRAY 1.8 0.185 0.217 E 371.0 337.0 0 25 25 0 [[44, 298]] 1.0 4dg3 Mus musculus AGC_PRKACA_MOUSE AGC 1.8e-94 321.8 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3FHIA P05132 14 351 351.0 ANP:60400 ATPlike Active DFGin 5.4633 14.263 BLAminus -118.0, -179.45 64.04, 75.7 -86.07, 24.14 267.17, 53.33 -59.82, -32.06 in-in in 8.8874 Saltbr-in 2.7901 HRD-in -94.84, -53.37 68.02, 7.49 in-in-in SNCiii in-in ActLoopNT-in 2.8652 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.67, 136.88 APE9-dihe-na 156.84, -158.52 APE8-dihe-in -126.08, 132.83 APE8-rot-in 296.09 APE67-dihe-in -67.08, -19.88 -42.62, -50.01 APE12-dist-in 8.2333 APE11-dist-in 11.1199 APE10-dist-in 5.402 APE9-dist-in 3.5636 C200A TPO198,SEP339 TPO198,SEP339 XRAY 2.0 0.199 0.226 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 3fhi Mus musculus AGC_PRKACA_MOUSE AGC 1e-93 319.3 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3QAME P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.5585 14.1896 BLAminus -125.2, -173.2 57.82, 79.24 -94.32, 24.42 273.28, 56.46 -52.36, -33.22 in-in in 8.9798 Saltbr-in 2.8042 HRD-in -80.54, -55.75 67.52, 12.49 in-in-in SNCiii in-in ActLoopNT-in 2.8883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.45, 157.56 APE9-dihe-na 134.84, -152.56 APE8-dihe-in -129.9, 127.65 APE8-rot-in 298.13 APE67-dihe-in -57.31, -20.14 -26.19, -66.74 APE12-dist-in 8.0939 APE11-dist-in 11.2769 APE10-dist-in 5.8065 APE9-dist-in 3.475 E209A TPO198,SEP339 TPO198,SEP339 XRAY 1.92 0.195 0.228 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 3qam Mus musculus AGC_PRKACA_MOUSE AGC 2.2e-93 318.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3QALE P05132 2 351 351.0 ATP:60351 ATPlike Active DFGin 5.6399 14.4013 BLAminus -123.21, -177.09 59.31, 80.89 -94.71, 25.93 269.1, 56.43 -54.28, -32.32 in-in in 9.0502 Saltbr-in 2.6578 HRD-in -84.64, -51.07 65.64, 14.74 in-in-in SNCiii in-in ActLoopNT-in 2.9615 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.61, 159.73 APE9-dihe-na 131.58, -155.18 APE8-dihe-in -126.66, 132.34 APE8-rot-in 301.51 APE67-dihe-in -57.77, -23.32 -31.31, -63.36 APE12-dist-in 8.0621 APE11-dist-in 11.3091 APE10-dist-in 5.7435 APE9-dist-in 3.5307 R281A TPO198,SEP339 TPO198,SEP339 XRAY 1.7 0.176 0.194 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 3qal Mus musculus AGC_PRKACA_MOUSE AGC 4.5e-93 317.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1RDQE P05132 2 351 351.0 ADP:60599,ATP:60600 ATPlike,ATPlike Active DFGin 5.7065 14.5148 BLAminus -117.27, 178.71 64.74, 81.19 -90.07, 21.82 270.96, 52.48 -58.25, -31.62 in-in in 9.0905 Saltbr-in 2.719 HRD-in -91.16, -53.36 73.19, 12.39 in-in-in SNCiii in-in ActLoopNT-in 2.9357 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.91, 159.57 APE9-dihe-na 132.64, -151.85 APE8-dihe-in -127.7, 133.09 APE8-rot-in 298.45 APE67-dihe-in -59.33, -27.24 -47.42, -47.34 APE12-dist-in 8.1158 APE11-dist-in 11.4138 APE10-dist-in 5.8307 APE9-dist-in 3.5208 Y205A TPO198,SEP339 TPO198,SEP339 XRAY 1.26 0.132 0.162 E 350.0 342.0 0 25 25 0 [[44, 298]] 1.0 1rdq Mus musculus AGC_PRKACA_MOUSE AGC 1.1e-92 315.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4O22A P05132 16 351 351.0 No_ligand No_ligand Active DFGin 6.4485 14.5482 BLAminus -124.93, -179.58 65.24, 83.52 -97.55, 25.76 273.08, 60.4 -61.15, -26.72 in-in in 8.8242 Saltbr-in 2.6383 HRD-in -89.28, -52.27 69.65, 12.56 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.45, 162.83 APE9-dihe-na 131.87, -150.17 APE8-dihe-in -128.05, 135.42 APE8-rot-in 301.96 APE67-dihe-in -61.83, -23.3 -46.45, -50.3 APE12-dist-in 7.9967 APE11-dist-in 11.4143 APE10-dist-in 5.8621 APE9-dist-in 3.5438 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 1.7 0.187 0.219 A 342.0 336.0 0 25 25 0 [[44, 298]] 1.0 4o22 Mus musculus AGC_PRKACA_MOUSE AGC 1.4e-94 322.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1JLUE P05132 13 351 351.0 No_ligand No_ligand Active DFGin 6.2861 14.0335 BLAminus -116.82, 172.06 62.47, 85.22 -99.38, 25.33 280.76, 66.77 -59.89, -25.29 in-in in 8.8849 Saltbr-in 2.9045 HRD-in -82.77, -54.36 73.92, -0.29 in-in-in SNCiii in-in ActLoopNT-in 3.0022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.81, 157.32 APE9-dihe-na 139.21, -153.09 APE8-dihe-in -125.03, 121.3 APE8-rot-in 316.06 APE67-dihe-in -62.91, -9.39 -23.05, -64.85 APE12-dist-in 8.0643 APE11-dist-in 11.3222 APE10-dist-in 6.0555 APE9-dist-in 3.703 None TPO198,SEP339 TPO198,SEP339 XRAY 2.25 0.181 999.0 E 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1jlu Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DG2E P05132 2 351 351.0 No_ligand No_ligand Active DFGin 6.4783 14.3469 BLAminus -123.83, 172.03 63.45, 88.02 -99.08, 27.68 275.25, 59.55 -56.12, -32.76 in-in in 8.8184 Saltbr-in 2.7992 HRD-in -84.63, -52.84 71.55, 8.96 in-in-in SNCiii in-in ActLoopNT-in 2.9185 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.79, 159.19 APE9-dihe-na 134.75, -147.2 APE8-dihe-in -130.86, 129.22 APE8-rot-in 304.99 APE67-dihe-in -62.19, -22.69 -40.4, -52.05 APE12-dist-in 8.0585 APE11-dist-in 11.3519 APE10-dist-in 5.7561 APE9-dist-in 3.4964 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.193 0.211 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4dg2 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFZE P05132 2 351 351.0 No_ligand No_ligand Active DFGin 6.3314 14.3533 BLAminus -124.21, 173.53 63.45, 88.27 -99.9, 27.01 273.13, 59.34 -56.57, -31.28 in-in in 8.7729 Saltbr-in 2.6928 HRD-in -87.8, -52.9 69.53, 11.47 in-in-in SNCiii in-in ActLoopNT-in 2.9057 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.19, 159.25 APE9-dihe-na 132.22, -141.79 APE8-dihe-in -134.47, 128.83 APE8-rot-in 307.05 APE67-dihe-in -59.16, -25.89 -40.01, -52.76 APE12-dist-in 8.0313 APE11-dist-in 11.343 APE10-dist-in 5.7654 APE9-dist-in 3.4388 K8C SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.0 0.207 0.234 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 4dfz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1APME P05132 11 351 351.0 No_ligand No_ligand Active DFGin 6.2608 14.0704 BLAminus -125.0, 178.22 62.58, 88.79 -105.13, 25.26 274.83, 66.5 -57.51, -25.56 in-in in 8.9302 Saltbr-in 2.582 HRD-in -81.09, -58.27 71.67, -2.38 in-in-in SNCiii in-in ActLoopNT-in 3.0534 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.78, 156.67 APE9-dihe-na 136.06, -155.51 APE8-dihe-in -123.48, 123.72 APE8-rot-in 302.63 APE67-dihe-in -54.93, -28.48 -32.82, -58.43 APE12-dist-in 8.2172 APE11-dist-in 11.4562 APE10-dist-in 5.9547 APE9-dist-in 3.7877 S140A SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.0 0.186 999.0 E 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 1apm Mus musculus AGC_PRKACA_MOUSE AGC 2.2e-94 321.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1BX6A P05132 13 351 351.0 BA1:60351 Type1 Active DFGin 6.0974 14.2707 BLAminus -131.41, 157.86 79.35, 91.47 -96.7, 9.79 287.76, 86.24 -44.29, -77.97 in-in in 8.3994 Saltbr-in 2.6074 HRD-in -60.43, -49.37 65.58, 0.7 in-in-in SNCiii in-in ActLoopNT-in 3.1024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -96.41, 136.41 APE9-dihe-na 139.93, 174.47 APE8-dihe-in -112.82, 117.81 APE8-rot-in 289.91 APE67-dihe-in -32.61, -31.36 -25.94, -76.91 APE12-dist-in 8.7332 APE11-dist-in 11.1899 APE10-dist-in 5.2412 APE9-dist-in 4.7598 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.1 0.21 0.34 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1bx6 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1FMOE P05132 14 351 351.0 ADN:60351 Type1 Active DFGin 6.6779 14.2824 BLAminus -114.95, 166.87 67.95, 101.15 -111.54, 7.58 268.05, 65.13 -43.18, -17.52 in-in in 8.5604 Saltbr-in 2.9824 HRD-in -73.08, -60.95 74.44, -3.64 in-in-in SNCiii in-in ActLoopNT-in 2.8596 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.53, 167.98 APE9-dihe-na 127.76, -157.13 APE8-dihe-in -115.17, 123.5 APE8-rot-in 303.04 APE67-dihe-in -62.85, -32.38 -37.72, -49.63 APE12-dist-in 7.9343 APE11-dist-in 11.2764 APE10-dist-in 5.9475 APE9-dist-in 3.7123 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.182 999.0 E 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1fmo Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1REJA P05132 17 351 351.0 B1L:60351 Type1 Active DFGin 6.6885 14.7589 BLAminus -129.16, -166.14 53.21, 69.99 -91.05, 27.11 275.8, 67.71 -67.13, -23.58 in-in in 9.1448 Saltbr-in 2.806 HRD-in -84.89, -51.08 67.36, 19.76 in-in-in SNCiii in-in ActLoopNT-in 2.7199 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.7, 155.59 APE9-dihe-na 102.81, -168.4 APE8-dihe-in -114.34, 132.29 APE8-rot-in 300.68 APE67-dihe-in -62.15, -27.72 -40.87, -53.2 APE12-dist-in 8.0818 APE11-dist-in 11.1003 APE10-dist-in 5.4023 APE9-dist-in 3.4935 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.208 0.291 A 350.0 335.0 0 25 25 0 [[44, 298]] 1.0 1rej Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3OW3A P05132 16 351 351.0 SMY:60401 Type1 Active DFGin 6.1403 14.543 BLAminus -123.88, 175.12 69.78, 83.56 -97.88, 23.25 272.21, 60.42 -52.11, -32.64 in-in in 9.1321 Saltbr-in 2.5499 HRD-in -87.74, -52.86 72.88, 7.11 in-in-in SNCiii in-in ActLoopNT-in 2.9121 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.65, 165.29 APE9-dihe-na 128.58, -156.74 APE8-dihe-in -122.61, 136.92 APE8-rot-in 295.99 APE67-dihe-in -53.86, -28.98 -54.05, -45.53 APE12-dist-in 8.1185 APE11-dist-in 11.5674 APE10-dist-in 5.8554 APE9-dist-in 3.5108 None TPO198,SEP339 TPO198,SEP339 XRAY 1.9 0.166 0.21 A 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 3ow3 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2ERZE P05132 16 351 351.0 HFS:60351 Type1 Active DFGin 5.8621 14.2868 BLAminus -120.01, 167.35 70.07, 90.43 -101.1, 32.12 275.39, 49.09 -53.89, -29.79 in-in in 9.0354 Saltbr-in 2.6896 HRD-in -71.67, -48.74 64.28, 7.57 in-in-in SNCiii in-in ActLoopNT-in 2.9432 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.95, 164.31 APE9-dihe-na 126.82, -161.82 APE8-dihe-in -117.41, 128.23 APE8-rot-in 308.76 APE67-dihe-in -49.78, -31.46 -30.24, -67.82 APE12-dist-in 8.1923 APE11-dist-in 11.4229 APE10-dist-in 5.9098 APE9-dist-in 3.5597 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.227 0.287 E 351.0 336.0 0 25 25 0 [[44, 298]] 1.0 2erz Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1REKA P05132 14 351 351.0 B8L:60351,PTL:60352 Type1,Allosteric Active DFGin 6.5124 14.951 BLAminus -126.84, -171.52 53.94, 74.01 -96.88, 22.16 273.96, 65.3 -56.46, -42.1 in-in in 8.8618 Saltbr-in 2.7916 HRD-in -90.9, -46.82 65.04, 3.0 in-in-in SNCiii in-in ActLoopNT-in 2.9322 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.61, 143.64 APE9-dihe-na 123.06, -169.72 APE8-dihe-in -113.81, 132.41 APE8-rot-in 289.91 APE67-dihe-in -65.44, -22.63 -41.39, -49.51 APE12-dist-in 8.0968 APE11-dist-in 10.719 APE10-dist-in 5.1557 APE9-dist-in 3.3485 None TPO198,SEP339 TPO198,SEP339 XRAY 2.3 0.218 0.295 A 350.0 338.0 0 25 25 0 [[44, 298]] 1.0 1rek Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM6C P05132 19 351 351.0 ANP:60402 ATPlike Inactive DFGin 6.7799 16.0821 ABAminus -110.74, -8.1 -141.78, 125.75 -126.67, 17.79 291.81, 81.75 -52.6, -43.19 out-out out 10.4027 Saltbr-out 4.4909 HRD-in -64.73, -48.52 44.91, 28.18 out-in-out SNCoio in-out ActLoopNT-in 2.8769 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -155.16, 154.51 APE9-dihe-na 131.73, -155.42 APE8-dihe-in -119.09, 141.73 APE8-rot-out 198.33 APE67-dihe-in -57.79, -26.12 -45.84, -50.95 APE12-dist-in 8.5303 APE11-dist-in 11.8147 APE10-dist-in 6.3058 APE9-dist-in 4.5025 None TPO198,SEP339 TPO198,SEP339 XRAY 2.39 0.225 0.261 C 339.0 322.0 0 25 25 0 [[44, 298]] 1.0 6mm6 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM6E P05132 19 351 351.0 ANP:60401 ATPlike Inactive DFGin 6.7325 15.9653 ABAminus -112.26, -9.59 -137.74, 126.1 -127.73, 18.87 290.52, 82.39 -53.04, -44.19 out-out out 10.2709 Saltbr-out 5.278 HRD-in -66.74, -47.88 44.41, 27.02 out-in-out SNCoio in-out ActLoopNT-in 2.8731 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -157.27, 155.34 APE9-dihe-na 128.78, -154.8 APE8-dihe-in -120.26, 141.99 APE8-rot-out 197.33 APE67-dihe-in -57.79, -26.44 -45.46, -51.33 APE12-dist-in 8.4779 APE11-dist-in 11.8514 APE10-dist-in 6.3306 APE9-dist-in 4.4228 None TPO198,SEP339 TPO198,SEP339 XRAY 2.39 0.225 0.261 E 339.0 320.0 0 25 25 0 [[44, 298]] 1.0 6mm6 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM7A P05132 17 351 351.0 ANP:60406 ATPlike Inactive DFGin 6.7159 15.4284 ABAminus -112.23, -9.6 -137.01, 123.03 -130.15, 19.3 297.15, 81.39 -54.86, -42.58 out-out out 10.2821 Saltbr-out 4.6231 HRD-in -76.47, -53.66 52.13, 28.38 out-in-out SNCoio in-out ActLoopNT-in 2.8634 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -163.99, 161.65 APE9-dihe-na 126.52, -159.69 APE8-dihe-in -119.22, 141.71 APE8-rot-out 195.45 APE67-dihe-in -67.85, -20.3 -44.24, -48.26 APE12-dist-in 8.2035 APE11-dist-in 11.1251 APE10-dist-in 5.7383 APE9-dist-in 3.9708 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.213 0.238 A 339.0 327.0 0 25 25 0 [[44, 298]] 1.0 6mm7 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM7D P05132 16 351 351.0 ANP:60405 ATPlike Inactive DFGin 6.6517 15.4584 ABAminus -113.01, -9.74 -137.13, 123.49 -128.55, 17.46 296.74, 82.18 -52.99, -42.79 out-out out 10.3794 Saltbr-out 5.8168 HRD-in -73.81, -53.25 53.83, 26.23 out-in-out SNCoio in-out ActLoopNT-in 2.8742 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -166.02, 161.72 APE9-dihe-na 122.21, -160.7 APE8-dihe-in -119.01, 142.81 APE8-rot-out 192.42 APE67-dihe-in -67.72, -20.93 -42.31, -48.3 APE12-dist-in 8.2101 APE11-dist-in 11.2017 APE10-dist-in 5.7858 APE9-dist-in 3.9614 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.213 0.238 D 339.0 324.0 0 25 25 0 [[44, 298]] 1.0 6mm7 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM8C P05132 16 351 351.0 ANP:60403 ATPlike Inactive DFGin 6.6132 15.2001 ABAminus -113.8, -10.95 -132.36, 129.54 -134.0, 24.39 301.03, 83.83 -57.02, -38.35 out-out out 10.3401 Saltbr-out 7.3235 HRD-in -73.54, -53.96 54.41, 29.61 out-in-out SNCoio in-out ActLoopNT-in 2.7764 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.79, 167.54 APE9-dihe-na 115.95, -161.99 APE8-dihe-in -118.41, 142.14 APE8-rot-out 195.18 APE67-dihe-in -66.48, -19.98 -46.61, -45.65 APE12-dist-in 8.1252 APE11-dist-in 11.2017 APE10-dist-in 5.8341 APE9-dist-in 3.9965 None TPO198,SEP339 TPO198,SEP339 XRAY 1.85 0.183 0.221 C 339.0 325.0 0 25 25 0 [[44, 298]] 1.0 6mm8 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKND P05132 16 351 351.0 ANP:60400 ATPlike Inactive DFGin 6.6105 14.9582 ABAminus -121.75, -47.3 -93.55, 119.31 -121.12, 22.25 288.77, 83.91 -60.17, -43.74 in-out in 9.6363 Saltbr-out 4.003 HRD-in -71.48, -47.99 39.7, 38.93 out-in-in SNCoii in-in ActLoopNT-in 2.9756 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.1, 161.55 APE9-dihe-na 104.53, 169.82 APE8-dihe-in -72.88, 137.25 APE8-rot-in 280.42 APE67-dihe-in -60.56, -25.71 -55.68, -37.9 APE12-dist-in 8.0946 APE11-dist-in 11.2355 APE10-dist-in 5.8091 APE9-dist-in 4.6921 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 D 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKOE P05132 16 351 351.0 ANP:60403 ATPlike Inactive DFGin 6.0364 14.5957 ABAminus -122.57, -57.22 -79.99, 109.96 -108.47, 33.73 286.2, 84.93 -64.54, -41.62 in-in in 9.7403 Saltbr-in 3.5644 HRD-in -78.91, -48.33 66.16, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.8677 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.15, 159.43 APE9-dihe-na 137.57, -133.12 APE8-dihe-in -144.28, 132.68 APE8-rot-in 289.09 APE67-dihe-in -62.87, -18.89 -48.53, -47.79 APE12-dist-in 8.0799 APE11-dist-in 11.3212 APE10-dist-in 5.8296 APE9-dist-in 3.774 None TPO198,SEP339 TPO198,SEP339 XRAY 2.89 0.213 0.259 E 339.0 336.0 0 25 25 0 [[44, 298]] 1.0 8uko Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKPE P05132 17 351 351.0 ANP:60402 ATPlike Inactive DFGin 6.1336 14.4301 ABAminus -106.11, -56.02 -81.74, 124.54 -123.06, 18.4 279.21, 82.41 -57.4, -55.55 in-out in 9.2794 Saltbr-out 4.1807 HRD-in -89.57, -52.98 66.95, 19.28 out-in-in SNCoii in-in ActLoopNT-in 2.9525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.29, 147.38 APE9-dihe-na 136.74, -150.06 APE8-dihe-in -126.21, 134.43 APE8-rot-in 318.02 APE67-dihe-in -77.56, -4.79 -54.58, -35.83 APE12-dist-in 7.9285 APE11-dist-in 10.8204 APE10-dist-in 5.1851 APE9-dist-in 3.8514 None SEP140,TPO198 SEP140,TPO198 XRAY 2.85 0.242 0.281 E 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukp Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTTB P05132 11 351 351.0 ADP:60401 ATPlike Inactive DFGin 6.5417 14.8798 ABAminus -93.85, -35.44 -119.41, 118.31 -113.9, 43.83 296.85, 78.9 -65.87, -49.34 in-none in 9.8688 Saltbr-none 999.0 HRD-in -94.05, -37.34 60.44, 1.66 none-in-in SNCnii in-in ActLoopNT-in 2.7867 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -166.4, 146.42 APE9-dihe-na 126.7, -158.4 APE8-dihe-in -116.99, 137.33 APE8-rot-in 273.8 APE67-dihe-in -64.02, -34.69 -52.94, -43.07 APE12-dist-in 7.7129 APE11-dist-in 10.7197 APE10-dist-in 5.2983 APE9-dist-in 4.164 K8C TPO198,SEP339 TPO198,SEP339 XRAY 3.5 0.23 0.284 B 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 4ntt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKNC P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.9773 15.8143 ABAminus -121.28, -46.06 -94.44, 119.11 -121.88, 20.98 289.09, 82.99 -60.59, -43.51 out-out out 10.2655 Saltbr-out 3.7763 HRD-in -69.49, -46.7 40.24, 37.27 out-in-in SNCoii in-in ActLoopNT-in 2.8604 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.14, 161.55 APE9-dihe-na 102.26, 166.3 APE8-dihe-in -75.0, 136.39 APE8-rot-in 285.29 APE67-dihe-in -59.55, -25.47 -55.27, -37.71 APE12-dist-in 8.2631 APE11-dist-in 11.3425 APE10-dist-in 5.8906 APE9-dist-in 4.4404 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 C 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKNF P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.8893 15.4858 ABAminus -119.02, -48.36 -94.42, 119.64 -122.07, 21.3 289.06, 84.07 -60.37, -43.79 in-none in 9.9681 Saltbr-none 999.0 HRD-in -70.24, -47.3 40.22, 39.45 none-in-out SNCnio in-out ActLoopNT-in 3.1956 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -150.61, 160.97 APE9-dihe-na 102.69, 167.59 APE8-dihe-in -73.59, 140.15 APE8-rot-out 204.21 APE67-dihe-in -61.18, -25.59 -54.92, -37.71 APE12-dist-in 8.0636 APE11-dist-in 11.1851 APE10-dist-in 5.795 APE9-dist-in 4.6032 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 F 339.0 323.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 8UKNH P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.9904 15.9406 ABAminus -119.65, -47.17 -95.12, 119.59 -123.41, 20.33 289.47, 82.92 -60.29, -43.54 out-out out 10.3777 Saltbr-out 4.1022 HRD-in -70.28, -46.9 40.49, 37.83 out-in-in SNCoii in-in ActLoopNT-in 2.9436 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.73, 160.95 APE9-dihe-na 102.27, 168.23 APE8-dihe-in -75.08, 137.2 APE8-rot-in 283.98 APE67-dihe-in -59.99, -25.87 -55.81, -37.99 APE12-dist-in 8.247 APE11-dist-in 11.3303 APE10-dist-in 5.9313 APE9-dist-in 4.5321 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.75 0.197 0.232 H 339.0 325.0 0 25 25 0 [[44, 298]] 1.0 8ukn Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3TNPC P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.4124 14.047 ABAminus -115.86, -60.86 -88.32, 106.92 -98.77, 21.04 269.52, 52.68 -48.7, -36.28 in-in in 8.6 Saltbr-in 2.8944 HRD-in -94.29, -50.01 72.25, 4.59 in-in-in SNCiii in-in ActLoopNT-in 2.9018 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.71, 164.13 APE9-dihe-na 136.51, -140.88 APE8-dihe-in -134.73, 130.62 APE8-rot-in 292.72 APE67-dihe-in -54.62, -27.98 -43.74, -54.69 APE12-dist-in 8.0801 APE11-dist-in 11.4918 APE10-dist-in 5.9315 APE9-dist-in 3.4025 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.3 0.226 0.235 C 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 3tnp Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3TNPF P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.4122 14.0463 ABAminus -115.9, -60.86 -88.39, 106.92 -98.78, 21.05 269.48, 52.72 -48.68, -36.31 in-in in 8.5999 Saltbr-in 2.8941 HRD-in -94.19, -50.06 72.23, 4.62 in-in-in SNCiii in-in ActLoopNT-in 2.9156 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.7, 164.08 APE9-dihe-na 136.57, -140.81 APE8-dihe-in -134.76, 130.54 APE8-rot-in 292.72 APE67-dihe-in -54.65, -27.95 -43.69, -54.69 APE12-dist-in 8.0809 APE11-dist-in 11.4916 APE10-dist-in 5.9317 APE9-dist-in 3.4021 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 2.3 0.226 0.235 F 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 3tnp Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4WBBB P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 5.8987 14.309 ABAminus -133.99, -40.66 -108.42, 103.56 -98.82, 16.34 272.05, 61.48 -51.24, -35.82 in-in in 8.5861 Saltbr-in 2.7679 HRD-in -93.67, -38.46 55.43, 10.07 in-in-in SNCiii in-in ActLoopNT-in 2.8579 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.35, 160.13 APE9-dihe-na 145.06, -138.63 APE8-dihe-in -131.95, 132.94 APE8-rot-in 298.17 APE67-dihe-in -60.16, -16.13 -44.42, -52.54 APE12-dist-in 8.043 APE11-dist-in 11.467 APE10-dist-in 6.061 APE9-dist-in 3.5781 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.8 0.232 0.279 B 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4wbb Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4X6QC P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.5826 13.9706 ABAminus -121.1, -42.58 -93.87, 102.7 -97.14, 17.55 267.16, 62.54 -52.57, -22.85 in-in in 8.4246 Saltbr-in 2.6995 HRD-in -93.89, -54.89 78.5, 7.23 in-in-in SNCiii in-in ActLoopNT-in 3.0582 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.45, 165.62 APE9-dihe-na 127.31, -150.86 APE8-dihe-in -123.77, 131.23 APE8-rot-in 300.08 APE67-dihe-in -68.69, -15.9 -43.09, -45.27 APE12-dist-in 8.1005 APE11-dist-in 11.4859 APE10-dist-in 6.067 APE9-dist-in 3.4046 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.52 0.201 0.261 C 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 4x6q Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTSA P05132 9 351 351.0 No_ligand No_ligand Inactive DFGin 6.538 15.9677 ABAminus -126.95, 0.97 -130.38, 129.83 -128.18, 8.25 284.09, 78.17 -52.18, -25.55 out-out out 10.2859 Saltbr-out 5.443 HRD-in -88.58, -45.11 67.09, 10.84 out-in-in SNCoii in-in ActLoopNT-in 2.9409 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.79, 153.47 APE9-dihe-na 119.65, -179.72 APE8-dihe-in -98.33, 124.38 APE8-rot-in 308.71 APE67-dihe-in -60.54, -27.51 -31.45, -47.3 APE12-dist-in 8.167 APE11-dist-in 11.4446 APE10-dist-in 6.0844 APE9-dist-in 4.2286 K8C TPO198,SEP339 TPO198,SEP339 XRAY 2.9 0.247 0.292 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 4nts Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTSB P05132 9 351 351.0 No_ligand No_ligand Inactive DFGin 6.0263 15.2864 ABAminus -111.39, -34.44 -108.24, 143.4 -134.27, 5.96 285.1, 84.22 -48.51, -37.04 in-none in 9.8214 Saltbr-none 999.0 HRD-in -84.15, -38.94 58.73, 4.32 none-in-in SNCnii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.51, 126.13 APE9-dihe-na 95.83, -178.74 APE8-dihe-in -68.15, 137.5 APE8-rot-in 299.78 APE67-dihe-in -69.28, -28.37 -49.3, -45.44 APE12-dist-in 8.2193 APE11-dist-in 10.3859 APE10-dist-in 5.3483 APE9-dist-in 4.0024 K8C TPO198,SEP339 TPO198,SEP339 XRAY 2.9 0.247 0.292 B 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 4nts Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 5X3FB P05132 5 317 351.0 No_ligand No_ligand Inactive DFGin 6.5356 15.8812 ABAminus -125.34, -3.25 -129.13, 129.62 -128.07, 7.73 283.82, 79.52 -54.86, -24.43 out-out out 10.2687 Saltbr-out 5.1184 HRD-in -88.25, -45.2 67.71, 9.27 out-in-in SNCoii in-in ActLoopNT-in 2.9322 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.56, 145.49 APE9-dihe-na 135.48, 176.97 APE8-dihe-in -97.8, 124.17 APE8-rot-in 309.27 APE67-dihe-in -59.29, -29.32 -31.89, -46.62 APE12-dist-in 8.1446 APE11-dist-in 10.7363 APE10-dist-in 5.6264 APE9-dist-in 4.2648 None TPO198 TPO198 XRAY 3.38 0.192 0.227 B 393.0 310.0 0 25 25 0 [[44, 298]] 1.0 5x3f Mus musculus AGC_PRKACA_MOUSE AGC 2.1e-94 321.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 6MM5E P05132 16 351 351.0 ANP:60402 ATPlike Inactive DFGin 5.9604 14.3509 BLAminus -116.65, 159.11 76.02, 91.05 -92.83, 26.22 286.06, 88.09 -52.81, -36.86 in-in in 8.8493 Saltbr-in 2.8003 HRD-in -83.15, -50.88 72.11, -0.72 in-in-out SNCiio in-out ActLoopNT-in 2.8706 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -156.6, 159.33 APE9-dihe-na 129.67, -150.44 APE8-dihe-in -128.62, 141.57 APE8-rot-out 194.03 APE67-dihe-in -68.05, -20.18 -46.89, -45.89 APE12-dist-in 8.2074 APE11-dist-in 11.3781 APE10-dist-in 5.7976 APE9-dist-in 3.7765 None TPO198,SEP339 TPO198,SEP339 XRAY 1.95 0.183 0.227 E 339.0 336.0 0 25 25 0 [[44, 298]] 1.0 6mm5 Mus musculus AGC_PRKACA_MOUSE AGC 1.3e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1ATPE P05132 16 351 351.0 ATP:60355 ATPlike Inactive DFGin 6.2296 14.5876 BLAminus -105.27, -165.6 48.73, 87.06 -105.12, 16.76 267.19, 75.22 -52.19, -32.07 in-out in 9.1613 Saltbr-out 3.6341 HRD-in -88.29, -43.64 51.81, 19.16 out-in-in SNCoii in-in ActLoopNT-in 2.8078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.21, 146.28 APE9-dihe-na 146.09, -156.15 APE8-dihe-in -133.3, 119.84 APE8-rot-in 299.98 APE67-dihe-in -65.71, -15.81 -24.26, -60.76 APE12-dist-in 8.3526 APE11-dist-in 11.4096 APE10-dist-in 5.7064 APE9-dist-in 3.9902 None TPO198,SEP339 TPO198,SEP339 XRAY 2.2 0.177 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 1atp Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DINA P05132 10 351 351.0 ATP:60400 ATPlike Inactive DFGin 5.792 13.1437 BLAminus -127.84, -176.29 51.22, 102.02 -109.69, 31.05 287.96, 58.2 -47.08, -31.2 in-in in 8.5177 Saltbr-in 3.4979 HRD-out -64.69, -78.02 71.93, 51.46 in-in-out SNCiio in-out ActLoopNT-in 2.9942 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -152.73, 153.23 APE9-dihe-na 130.84, -154.91 APE8-dihe-in -121.15, 137.05 APE8-rot-out 34.65 APE67-dihe-in -46.77, -45.03 -45.98, -63.1 APE12-dist-in 7.9722 APE11-dist-in 10.5875 APE10-dist-in 4.9968 APE9-dist-in 3.53 None TPO198,SEP339 TPO198,SEP339 XRAY 3.7 0.211 0.293 A 350.0 342.0 0 25 25 0 [[44, 298]] 1.0 4din Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 7E12A P05132 19 351 351.0 ANP:60401 ATPlike Inactive DFGin 5.3957 14.6175 BLAminus -131.26, -169.7 58.92, 77.12 -93.02, 37.73 266.27, 47.03 -71.49, -23.13 in-in in 8.8067 Saltbr-in 3.2657 HRD-out -127.04, 103.44 -105.61, 37.91 in-in-in SNCiii in-in ActLoopNT-in 2.903 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.78, 159.74 APE9-dihe-na 134.39, -158.49 APE8-dihe-in -118.85, 128.69 APE8-rot-in 308.98 APE67-dihe-in -63.3, -26.53 -50.37, -37.69 APE12-dist-in 8.03 APE11-dist-in 11.3719 APE10-dist-in 5.9651 APE9-dist-in 3.4216 None TPO198,SEP339 TPO198,SEP339 XRAY 2.796 0.208 0.252 A 358.0 333.0 0 25 25 0 [[44, 298]] 1.0 7e12 Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1JBPE P05132 10 351 351.0 ADP:60381 ATPlike Inactive DFGin 6.1283 14.0345 BLAminus -131.98, 178.81 60.97, 83.81 -101.93, 15.49 276.81, 71.17 -55.35, -24.18 in-in in 8.8688 Saltbr-in 2.7492 HRD-out -93.99, 130.53 -128.02, 39.83 in-in-in SNCiii in-in ActLoopNT-in 2.8856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.07, 156.95 APE9-dihe-na 132.9, -168.64 APE8-dihe-in -109.4, 126.7 APE8-rot-in 297.85 APE67-dihe-in -61.28, -20.5 -33.82, -53.02 APE12-dist-in 8.1215 APE11-dist-in 11.4477 APE10-dist-in 6.0125 APE9-dist-in 3.8617 None SEP11,TPO198,SEP339 SEP11,TPO198,SEP339 XRAY 2.2 0.175 999.0 E 350.0 342.0 0 25 25 0 [[44, 298]] 1.0 1jbp Mus musculus AGC_PRKACA_MOUSE AGC 1.6e-94 321.9 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3O7LB P05132 18 351 351.0 ANP:60354 ATPlike Inactive DFGin 5.7904 14.6658 BLAminus -108.29, -170.95 57.63, 74.91 -94.92, 22.34 267.93, 64.07 -48.2, -34.6 in-in in 9.0975 Saltbr-in 2.9978 HRD-in -84.13, -53.04 68.25, 25.66 in-in-out SNCiio in-out ActLoopNT-in 2.9497 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -140.78, 178.73 APE9-dihe-na 123.03, -156.78 APE8-dihe-in -134.79, 129.02 APE8-rot-out 131.03 APE67-dihe-in -64.87, -13.33 -37.09, -52.44 APE12-dist-in 8.1152 APE11-dist-in 11.126 APE10-dist-in 5.5927 APE9-dist-in 3.4797 None TPO198 TPO198 XRAY 2.8 0.216 0.287 B 350.0 327.0 3 25 25 0 [[44, 298]] 1.0 3o7l Mus musculus AGC_PRKACA_MOUSE AGC 8.9e-94 319.5 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2CPKE P05132 16 351 351.0 No_ligand No_ligand Inactive DFGin 6.9516 14.3527 BLAminus -119.36, 179.9 54.29, 98.05 -110.06, 38.52 269.38, 72.49 -74.59, -10.83 in-in in 8.8905 Saltbr-in 3.0285 HRD-out -89.69, 114.42 -105.18, 29.22 in-in-in SNCiii in-in ActLoopNT-in 2.9084 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.45, 150.79 APE9-dihe-na 149.42, -157.84 APE8-dihe-in -117.51, 129.53 APE8-rot-in 300.38 APE67-dihe-in -65.47, -26.39 -44.25, -41.5 APE12-dist-in 8.076 APE11-dist-in 11.291 APE10-dist-in 5.9045 APE9-dist-in 3.7514 None SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.7 0.18 999.0 E 350.0 336.0 0 25 25 0 [[44, 298]] 1.0 2cpk Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3O7LD P05132 14 351 351.0 No_ligand No_ligand Inactive DFGin 6.5881 15.3871 BLAminus -122.76, 164.56 73.91, 96.96 -115.5, 27.13 288.86, 72.99 -56.99, -35.58 in-out in 9.6773 Saltbr-out 3.7173 HRD-in -80.64, -45.25 61.11, 19.5 out-in-out SNCoio in-out ActLoopNT-in 2.9631 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -150.51, -38.18 APE9-dihe-na -70.79, 159.72 APE8-dihe-in -54.96, 142.28 APE8-rot-out 27.57 APE67-dihe-in -76.4, -17.97 -49.97, -34.37 APE12-dist-in 7.986 APE11-dist-in 11.3838 APE10-dist-in 5.9066 APE9-dist-in 3.7447 None TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.216 0.287 D 350.0 335.0 0 25 25 0 [[44, 298]] 1.0 3o7l Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 9O7VA P05132 15 351 351.0 No_ligand No_ligand Inactive DFGin 6.9636 14.2333 BLAminus -144.42, 177.21 64.71, 76.79 -85.39, 18.92 274.62, 10.56 -43.43, -41.22 in-out in 9.3028 Saltbr-out 5.1072 HRD-in -93.65, -55.47 73.54, 8.94 out-in-in SNCoii in-in ActLoopNT-in 2.7506 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na 179.97, 149.56 APE9-dihe-na 148.21, -144.81 APE8-dihe-in -132.69, 133.23 APE8-rot-in 300.23 APE67-dihe-in -65.9, -25.09 -38.29, -53.75 APE12-dist-in 8.3267 APE11-dist-in 10.2791 APE10-dist-in 4.966 APE9-dist-in 3.3364 None TPO198,SEP339 TPO198,SEP339 XRAY 3.7 0.234 0.293 A 350.0 337.0 0 25 25 0 [[44, 298]] 1.0 9o7v Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1RE8A P05132 13 351 351.0 BD2:60351 Type1 Inactive DFGin 6.3634 14.4971 BLAminus -126.74, -163.36 52.92, 64.83 -86.7, 13.59 272.3, 77.12 -53.9, -38.74 in-in in 8.728 Saltbr-in 2.8622 HRD-out -92.25, 100.7 -92.09, 32.79 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.96, 163.56 APE9-dihe-na 123.01, -156.83 APE8-dihe-in -123.97, 134.13 APE8-rot-in 306.64 APE67-dihe-in -79.49, -1.91 -37.94, -51.41 APE12-dist-in 8.1888 APE11-dist-in 11.3883 APE10-dist-in 5.6985 APE9-dist-in 3.5296 None TPO198,SEP339 TPO198,SEP339 XRAY 2.1 0.197 0.252 A 350.0 339.0 0 25 25 0 [[44, 298]] 1.0 1re8 Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4NTTA P05132 11 351 351.0 ADP:60401 ATPlike Inactive DFGin 6.2546 15.2208 None 58.0, -132.96 -135.23, 163.83 -122.73, 17.77 281.43, 74.72 -41.46, -50.2 in-out in 9.9815 Saltbr-out 4.1938 HRD-in -65.11, -40.77 60.9, 3.38 out-in-in SNCoii in-in ActLoopNT-in 2.8637 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.9, 118.31 APE9-dihe-na 164.12, -173.28 APE8-dihe-in -108.19, 123.7 APE8-rot-in 267.93 APE67-dihe-in -75.4, -22.82 -40.35, -37.34 APE12-dist-in 8.1876 APE11-dist-in 11.1589 APE10-dist-in 5.5421 APE9-dist-in 4.3211 None TPO198,SEP339 TPO198,SEP339 XRAY 3.5 0.23 0.284 A 350.0 341.0 0 25 25 0 [[44, 298]] 1.0 4ntt Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1SYKA P05132 2 351 351.0 No_ligand No_ligand Inactive DFGin 6.5487 15.2891 None -131.76, 92.58 153.52, 114.28 -135.97, 14.86 305.19, 86.4 -55.43, -35.39 out-out out 10.6501 Saltbr-out 4.6701 HRD-out -89.49, 87.61 -76.68, 28.19 out-in-in SNCoii in-in ActLoopNT-in 2.8271 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.89, 158.84 APE9-dihe-na 108.08, 161.46 APE8-dihe-in -68.78, 138.01 APE8-rot-in 292.07 APE67-dihe-in -58.35, -9.3 -44.71, -57.38 APE12-dist-in 8.6724 APE11-dist-in 11.389 APE10-dist-in 5.9774 APE9-dist-in 3.618 E231Q TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.202 0.249 A 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1syk Mus musculus AGC_PRKACA_MOUSE AGC 5.7e-94 320.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1SYKB P05132 14 351 351.0 No_ligand No_ligand Inactive DFGin 6.599 15.2944 None -131.1, 91.72 152.06, 111.8 -131.83, 14.93 304.13, 82.92 -52.5, -38.6 out-out out 10.6973 Saltbr-out 4.5374 HRD-out -89.8, 89.72 -78.69, 28.99 out-in-in SNCoii in-in ActLoopNT-in 2.7813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.75, 160.3 APE9-dihe-na 107.8, 162.07 APE8-dihe-in -68.75, 135.04 APE8-rot-in 292.48 APE67-dihe-in -58.91, -9.06 -42.82, -56.64 APE12-dist-in 8.6623 APE11-dist-in 11.3639 APE10-dist-in 5.9602 APE9-dist-in 3.6147 E231Q TPO198,SEP339 TPO198,SEP339 XRAY 2.8 0.202 0.249 B 350.0 325.0 0 25 25 0 [[44, 298]] 1.0 1syk Mus musculus AGC_PRKACA_MOUSE AGC 5.7e-94 320.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFYA P05132 15 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -85.64, -176.8 33.76, 66.58 -80.32, 120.49 999.0, 999.0 -82.07, 106.21 in-none in 9.9071 Saltbr-none 999.0 HRD-in -75.3, -48.75 74.17, -71.89 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanii APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 145.79 APE8-rot-in 341.44 APE67-dihe-in -58.39, -21.24 -48.4, -47.32 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 R195A SEP339 SEP339 XRAY 2.997 0.253 0.286 A 371.0 311.0 12 25 13 12 [[44, 298]] 1.0 4dfy Mus musculus AGC_PRKACA_MOUSE AGC 3.3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 4DFYE P05132 15 351 351.0 No_ligand No_ligand Inactive None 999.0 999.0 None -87.32, -175.53 34.83, 65.83 -79.11, 119.4 999.0, 999.0 -80.98, 105.33 in-out in 9.7937 Saltbr-out 4.0426 HRD-in -70.47, -49.15 73.48, -78.98 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_nnoo APE10-dihe-na 999.0, -39.98 APE9-dihe-na -90.86, -172.73 APE8-dihe-in -82.11, 146.95 APE8-rot-in 336.67 APE67-dihe-in -63.39, -14.5 -53.89, -42.37 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 12.5337 APE9-dist-out 7.8184 R195A SEP339 SEP339 XRAY 2.997 0.253 0.286 E 371.0 313.0 10 25 15 10 [[44, 298]] 1.0 4dfy Mus musculus AGC_PRKACA_MOUSE AGC 3.3e-94 321.0 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1J3HA P05132 10 351 351.0 No_ligand No_ligand None DFGin 6.9571 16.5294 BLAminus -128.1, 165.84 66.16, 90.29 -100.57, 29.84 267.59, 74.49 -52.61, -63.31 out-none out 10.2685 Saltbr-none 999.0 HRD-in -65.94, -47.85 41.03, 47.95 none-in-in SNCnii in-in ActLoopNT-in 2.8154 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -175.68, 166.03 APE9-dihe-na 96.38, 161.28 APE8-dihe-in -70.8, 121.46 APE8-rot-in 315.06 APE67-dihe-in -64.05, -14.0 -35.32, -45.01 APE12-dist-in 8.2423 APE11-dist-in 11.0778 APE10-dist-in 6.1501 APE9-dist-in 4.8506 None TPO198,SEP339 TPO198,CME200,SEP339 XRAY 2.9 0.257 0.291 A 350.0 332.0 0 25 25 0 [[44, 298]] 1.0 1j3h Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 1J3HB P05132 12 351 351.0 No_ligand No_ligand None DFGin 6.9618 16.3184 BLAminus -127.51, 166.45 66.18, 90.08 -100.98, 29.78 267.08, 73.82 -52.31, -60.95 out-none out 10.1864 Saltbr-none 999.0 HRD-in -67.73, -45.7 38.54, 48.86 none-in-in SNCnii in-in ActLoopNT-in 2.811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.43, 169.92 APE9-dihe-na 94.29, 160.8 APE8-dihe-in -70.42, 119.44 APE8-rot-in 315.91 APE67-dihe-in -66.01, -15.04 -33.81, -42.66 APE12-dist-in 8.2628 APE11-dist-in 11.2131 APE10-dist-in 6.1679 APE9-dist-in 4.844 None TPO198,SEP339 TPO198,CME200,SEP339 XRAY 2.9 0.257 0.291 B 350.0 330.0 0 25 25 0 [[44, 298]] 1.0 1j3h Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2QVSE P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1963 14.9955 BLAminus -125.26, 166.13 66.05, 91.61 -98.74, 33.08 286.99, 64.22 -54.01, -35.46 out-none out 10.2631 Saltbr-none 999.0 HRD-in -74.03, -56.5 67.93, 15.74 none-in-in SNCnii in-in ActLoopNT-in 2.9976 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.49, 163.74 APE9-dihe-na 132.78, -148.47 APE8-dihe-in -122.84, 132.55 APE8-rot-in 302.63 APE67-dihe-in -52.83, -31.96 -33.3, -62.56 APE12-dist-in 7.8939 APE11-dist-in 11.5512 APE10-dist-in 6.03 APE9-dist-in 3.5577 None TPO198,SEP339 TPO198,SEP339 XRAY 2.5 0.212 0.251 E 350.0 325.0 0 25 25 0 [[44, 298]] 1.0 2qvs Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4QD P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1967 14.9965 BLAminus -125.26, 166.14 66.1, 91.56 -98.68, 33.07 286.99, 61.83 -54.01, -35.41 out-none out 10.2635 Saltbr-none 999.0 HRD-in -74.09, -56.53 67.97, 15.71 none-in-in SNCnii in-in ActLoopNT-in 2.9982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 163.78 APE9-dihe-na 132.71, -148.52 APE8-dihe-in -122.82, 132.51 APE8-rot-in 302.65 APE67-dihe-in -52.8, -31.95 -33.23, -62.65 APE12-dist-in 7.9212 APE11-dist-in 11.55 APE10-dist-in 6.0293 APE9-dist-in 3.5583 None None None EM 35.0 999.0 999.0 D 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4q Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4QE P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1966 14.995 BLAminus -125.26, 166.1 66.04, 91.65 -98.75, 33.06 286.98, 61.89 -53.93, -35.48 out-none out 10.2634 Saltbr-none 999.0 HRD-in -73.99, -56.54 67.98, 15.68 none-in-in SNCnii in-in ActLoopNT-in 2.9973 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.48, 163.78 APE9-dihe-na 132.74, -148.47 APE8-dihe-in -122.8, 132.56 APE8-rot-in 302.67 APE67-dihe-in -52.81, -31.94 -33.33, -62.57 APE12-dist-in 7.922 APE11-dist-in 11.5519 APE10-dist-in 6.0305 APE9-dist-in 3.5582 None None None EM 35.0 999.0 999.0 E 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4q Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4RD P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1972 14.9967 BLAminus -125.31, 166.2 66.04, 91.6 -98.77, 33.16 286.98, 61.82 -54.08, -35.39 out-none out 10.2636 Saltbr-none 999.0 HRD-in -74.03, -56.49 67.97, 15.67 none-in-in SNCnii in-in ActLoopNT-in 2.998 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.51, 163.71 APE9-dihe-na 132.78, -148.41 APE8-dihe-in -122.89, 132.55 APE8-rot-in 302.65 APE67-dihe-in -52.76, -32.01 -33.29, -62.61 APE12-dist-in 7.9206 APE11-dist-in 11.55 APE10-dist-in 6.0293 APE9-dist-in 3.5577 None None None EM 35.0 999.0 999.0 D 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 3J4RE P05132 14 351 351.0 No_ligand No_ligand None DFGin 6.1967 14.9951 BLAminus -125.22, 166.12 66.01, 91.59 -98.73, 33.13 286.98, 61.85 -53.97, -35.5 out-none out 10.2637 Saltbr-none 999.0 HRD-in -74.05, -56.46 67.95, 15.66 none-in-in SNCnii in-in ActLoopNT-in 2.9978 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.47, 163.74 APE9-dihe-na 132.8, -148.42 APE8-dihe-in -122.89, 132.51 APE8-rot-in 302.64 APE67-dihe-in -52.86, -31.95 -33.27, -62.57 APE12-dist-in 7.9226 APE11-dist-in 11.5509 APE10-dist-in 6.0296 APE9-dist-in 3.5575 None None None EM 35.0 999.0 999.0 E 351.0 325.0 0 25 25 0 [[44, 298]] 1.0 3j4r Mus musculus AGC_PRKACA_MOUSE AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_MOUSE 2QURA P05132 12 351 351.0 No_ligand No_ligand None DFGin 6.5556 14.5504 BLAminus -137.47, -167.05 53.68, 73.35 -97.68, 23.63 275.03, 65.42 -50.82, -37.16 in-none in 9.0785 Saltbr-none 999.0 HRD-in -62.2, -51.82 63.3, 0.36 none-in-in SNCnii in-in ActLoopNT-in 2.9356 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.83, 151.09 APE9-dihe-na 135.53, -158.17 APE8-dihe-in -121.8, 126.63 APE8-rot-in 312.25 APE67-dihe-in -60.67, -15.51 -24.4, -62.49 APE12-dist-in 8.1463 APE11-dist-in 11.1283 APE10-dist-in 5.5314 APE9-dist-in 3.2085 K286P,F328A TPO198,SEP339 TPO198,SEP339 XRAY 2.5 0.212 0.265 A 350.0 340.0 0 25 25 0 [[44, 298]] 1.0 2qur Mus musculus AGC_PRKACA_MOUSE AGC 2.3e-94 321.4 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_RAT 3TNQB P27791 18 351 351.0 ADP:60400 ATPlike Inactive DFGin 6.0256 14.1092 ABAminus -114.77, -42.68 -116.73, 98.61 -86.63, 16.07 279.08, 57.74 -59.27, -13.09 in-in in 8.7647 Saltbr-in 3.2951 HRD-in -83.62, -53.15 67.05, 14.07 in-in-in SNCiii in-in ActLoopNT-in 3.0146 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.54, 167.18 APE9-dihe-na 139.44, -131.54 APE8-dihe-in -144.99, 127.08 APE8-rot-in 312.05 APE67-dihe-in -55.59, -13.34 -44.48, -54.97 APE12-dist-in 8.0951 APE11-dist-in 11.4567 APE10-dist-in 6.1812 APE9-dist-in 3.5888 None SEP11,SEP140,TPO198,SEP339 SEP11,SEP140,TPO198,SEP339 XRAY 3.097 0.234 0.275 B 350.0 334.0 0 25 25 0 [[44, 298]] 1.0 3tnq Rattus norvegicus AGC_PRKACA_RAT AGC 1.5e-94 322.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CDKA P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.8431 14.3299 BLAminus -113.76, -166.2 47.38, 80.03 -85.76, 16.06 278.85, 56.4 -55.46, -28.11 in-in in 9.0339 Saltbr-in 2.8992 HRD-in -94.66, -56.81 78.16, -3.52 in-in-in SNCiii in-in ActLoopNT-in 2.9853 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.51, 155.2 APE9-dihe-na 137.51, -153.75 APE8-dihe-in -125.49, 136.2 APE8-rot-in 297.83 APE67-dihe-in -73.46, -24.38 -35.73, -51.43 APE12-dist-in 7.9972 APE11-dist-in 11.4183 APE10-dist-in 5.7664 APE9-dist-in 3.6421 None TPO198 TPO198 XRAY 2.0 0.197 999.0 A 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CDKB P36887 9 351 351.0 ANP:60400 ATPlike Active DFGin 5.907 14.5106 BLAminus -124.27, -171.72 50.82, 76.29 -83.58, 17.26 280.88, 62.25 -47.74, -29.83 in-in in 8.889 Saltbr-in 2.8833 HRD-in -87.48, -57.48 77.49, 1.67 in-in-in SNCiii in-in ActLoopNT-in 2.9631 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.91, 159.84 APE9-dihe-na 137.3, -140.74 APE8-dihe-in -136.57, 132.27 APE8-rot-in 304.84 APE67-dihe-in -69.16, -27.96 -34.59, -53.92 APE12-dist-in 8.3483 APE11-dist-in 11.5142 APE10-dist-in 6.0801 APE9-dist-in 3.7441 None TPO198 TPO198 XRAY 2.0 0.197 999.0 B 350.0 343.0 0 25 25 0 [[44, 298]] 1.0 1cdk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CTPE P36887 8 351 351.0 No_ligand No_ligand Inactive DFGin 6.725 16.055 BLAminus -116.62, 169.7 58.2, 106.1 -115.39, 26.05 266.95, 79.04 -73.93, 13.07 in-out in 9.9631 Saltbr-out 3.6616 HRD-out -67.85, 127.4 -110.51, 32.03 out-in-in SNCoii in-in ActLoopNT-in 3.0743 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.53, 165.54 APE9-dihe-na 119.1, -162.75 APE8-dihe-in -95.5, 138.49 APE8-rot-in 313.62 APE67-dihe-in -63.93, -15.29 -42.58, -58.58 APE12-dist-in 8.6012 APE11-dist-in 11.5506 APE10-dist-in 6.2522 APE9-dist-in 3.8257 None TPO198 TPO198 XRAY 2.9 0.19 999.0 E 350.0 333.0 0 25 25 0 [[44, 298]] 1.0 1ctp Sus scrofa AGC_PRKACA_PIG AGC 3.3e-95 324.2 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
PRKACA KAPCA_PIG 1CMKE P36887 2 351 351.0 No_ligand No_ligand Inactive DFGin 7.428 16.0445 BLAminus -105.57, 177.37 63.01, 79.23 -102.18, 28.14 277.96, 75.47 -76.23, -19.76 in-out in 9.8846 Saltbr-out 4.1251 HRD-in -61.54, -38.92 59.61, -1.33 out-in-in SNCoii in-in ActLoopNT-in 3.0635 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.53, 131.84 APE9-dihe-na 157.2, -155.98 APE8-dihe-in -96.86, 135.92 APE8-rot-in 291.44 APE67-dihe-in -53.19, -28.67 -38.32, -50.64 APE12-dist-in 8.1969 APE11-dist-in 11.2119 APE10-dist-in 5.6454 APE9-dist-in 3.8997 None TPO198,SEP339 TPO198,SEP339 XRAY 2.9 0.233 999.0 E 350.0 350.0 0 25 25 0 [[44, 298]] 1.0 1cmk Sus scrofa AGC_PRKACA_PIG AGC 3.5e-95 324.1 1.0 260.0 260.0 184 185 186 188 190 73 92 96 164 166 165 167.0 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha