| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|---|---|---|---|
| DFGin | BLAminus | 78 | 46.4% | 4AW0A |
| DFGin | ABAminus | 20 | 11.9% | 4C57A |
| DFGin | BLAplus | 19 | 11.3% | 9UHIA |
| DFGin | None | 16 | 9.5% | 8B9EA |
| DFGin | BLBplus | 10 | 6.0% | 3ZCLA |
| DFGout | None | 9 | 5.4% | 3VO3A |
| DFGout | BBAminus | 8 | 4.8% | 4MXCA |
| DFGin | BLBminus | 3 | 1.8% | 5XYYA |
| DFGin | BLBtrans | 2 | 1.2% | 2R3IA |
| None | None | 2 | 1.2% | 5IEXA |
| DFGinter | None | 1 | 0.6% | 4EBWA |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | AKT1 | AKT1_HUMAN | 4EKLA | P31749 | 144 | 478 | 480.0 | 0RF:501 | Type1 | Active | DFGin | 6.496 | 13.423 | BLAminus | -130.08, 156.46 | 77.16, 99.77 | -112.66, 14.16 | 298.65, 90.33 | -61.32, -30.96 | in-in | in | 8.958 | Saltbr-in | 2.452 | HRD-in | -78.38, -44.96 | 68.93, -13.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.757 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.83, 160.76 | APE9-dihe-na | 116.71, 166.32 | APE8-dihe-in | -83.66, 133.51 | APE8-rot-in | 293.53 | APE67-dihe-in | -68.09, -18.95 | -43.13, -46.31 | APE12-dist-in | 8.36 | APE11-dist-in | 11.512 | APE10-dist-in | 6.011 | APE9-dist-in | 4.443 | S473D | TPO308 | TPO308 | XRAY | 2.0 | 0.175 | 0.235 | A | 341 | 330 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekl | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AGC | GRK5 | GRK5_HUMAN | 9BRPA | P34947 | 25 | 542 | 590.0 | A1ARF:601 | Type1 | Inactive | DFGin | 6.253 | 12.479 | ABAminus | -116.3, -61.02 | -91.04, 101.81 | -97.25, 10.66 | 289.92, 84.11 | -59.57, -18.7 | in-in | in | 8.91 | Saltbr-in | 3.037 | HRD-in | -85.07, -56.86 | 71.89, 13.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.105 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.18, 177.63 | APE9-dihe-na | 122.23, -155.28 | APE8-dihe-in | -122.73, 136.27 | APE8-rot-in | 286.0 | APE67-dihe-inflip | 100.9, -21.88 | -54.82, 128.22 | APE12-dist-in | 9.574 | APE11-dist-in | 11.932 | APE10-dist-in | 6.253 | APE9-dist-in | 4.143 | D311N | None | None | XRAY | 2.8 | 0.245 | 0.283 | A | 598 | 502 | 0 | 0 | 0 | 0 | [[186, 448]] | 1.0 | 9brp | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1 | 260 | 260 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | GRK5 | GRK5_HUMAN | 9BREA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Active | DFGin | 6.176 | 12.564 | BLAminus | -128.67, 172.15 | 57.35, 77.75 | -93.22, 24.8 | 286.17, 72.14 | -63.15, -21.99 | in-in | in | 8.801 | Saltbr-in | 2.458 | HRD-in | -88.2, -51.09 | 67.29, 13.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.127 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.49, 165.19 | APE9-dihe-na | 125.58, -150.88 | APE8-dihe-in | -124.55, 138.39 | APE8-rot-in | 312.36 | APE67-dihe-inflip | 92.11, -16.19 | -53.44, 132.83 | APE12-dist-in | 9.943 | APE11-dist-in | 12.131 | APE10-dist-in | 6.337 | APE9-dist-in | 4.122 | D311N | None | None | XRAY | 2.8 | 0.215 | 0.26 | A | 598 | 503 | 0 | 0 | 0 | 0 | [[186, 448]] | 1.0 | 9bre | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1 | 260 | 260 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | GRK5 | GRK5_HUMAN | 8UAQA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Inactive | DFGin | 6.02 | 12.841 | None | -112.48, -65.82 | -86.97, 96.33 | -93.06, 17.75 | 286.66, 70.13 | -64.2, -19.76 | in-in | in | 9.334 | Saltbr-in | 3.369 | HRD-in | -90.24, -57.5 | 70.99, -0.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.037 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.56, 170.13 | APE9-dihe-na | 119.68, -157.85 | APE8-dihe-in | -112.7, 143.6 | APE8-rot-in | 314.4 | APE67-dihe-inflip | 89.64, -4.73 | -59.54, 131.81 | APE12-dist-in | 9.916 | APE11-dist-in | 12.102 | APE10-dist-in | 6.306 | APE9-dist-in | 4.174 | D311N | None | None | XRAY | 2.8 | 0.232 | 0.277 | A | 598 | 501 | 0 | 0 | 0 | 0 | [[186, 448]] | 1.0 | 8uaq | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1 | 260 | 260 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | PDPK1 | PDPK1_HUMAN | 4AW0A | O15530 | 75 | 359 | 556.0 | ATP:500,MJF:600 | ATPlike,Allosteric | Active | DFGin | 6.531 | 14.993 | BLAminus | -134.84, 177.25 | 78.73, 76.19 | -106.3, 8.53 | 283.51, 97.11 | -69.63, -19.36 | in-in | in | 8.595 | Saltbr-in | 3.009 | HRD-in | -83.05, -53.03 | 79.45, -12.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.934 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.69, 159.04 | APE9-dihe-na | 139.48, -167.8 | APE8-dihe-in | -131.87, 132.42 | APE8-rot-in | 295.45 | APE67-dihe-in | -61.29, -25.28 | -54.74, -42.17 | APE12-dist-in | 7.509 | APE11-dist-in | 10.601 | APE10-dist-in | 5.026 | APE9-dist-in | 3.58 | Y288G,Q292A | SEP241 | SEP241,CME260 | XRAY | 1.43 | 0.171 | 0.188 | A | 311 | 285 | 0 | 0 | 0 | 0 | [[82, 342]] | 1.0 | 4aw0 | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1 | 260 | 260 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PRKCH | KPCL_HUMAN | 8FP1A | P24723 | 349 | 676 | 683.0 | XXF:9000 | Type1 | Active | DFGin | 6.04 | 12.861 | BLAminus | -134.17, 160.39 | 76.6, 103.68 | -113.44, 14.82 | 306.37, 103.97 | -62.81, -37.48 | in-in | in | 8.529 | Saltbr-in | 2.747 | HRD-in | -71.28, -48.4 | 60.66, 8.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.042 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -168.52, 169.89 | APE9-dihe-na | 121.68, 166.05 | APE8-dihe-in | -83.39, 128.15 | APE8-rot-in | 297.95 | APE67-dihe-in | -61.25, -27.98 | -43.8, -44.17 | APE12-dist-in | 8.666 | APE11-dist-in | 11.701 | APE10-dist-in | 6.365 | APE9-dist-in | 3.566 | S675E | TPO513,TPO656 | TPO513,TPO656 | XRAY | 1.85 | 0.2 | 0.234 | A | 353 | 328 | 0 | 0 | 0 | 0 | [[355, 614]] | 1.0 | 8fp1 | AGC_PRKCH_HUMAN | AGC | 1.6e-97 | 331.6 | 1 | 260 | 260 | 496 | 497 | 498 | 500 | 502 | 384 | 403 | 407 | 476 | 478 | 477 | 479 | 536 | 524 | 519 | 518 | 517 | 516 | 515 | 514 | 513 | 434 | Protein kinase C eta type |
| CAMK | AURKA | AURKA_HUMAN | 8C1DA | O14965 | 127 | 388 | 403.0 | T2F:401,ADP:402,T5L:405 | Allosteric,ATPlike,Allosteric | Inactive | DFGin | 5.59 | 14.77 | BLAminus | -129.39, 179.64 | 57.3, 80.97 | -92.88, 23.53 | 280.13, 79.47 | -56.16, -33.44 | in-in | in | 9.306 | Saltbr-in | 2.936 | HRD-in | -72.1, -50.49 | 67.69, -1.24 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.796 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 144.85 | APE8-dihe-in | -64.26, 154.27 | APE8-rot-out | 88.6 | APE67-dihe-in | -39.49, -36.75 | -82.32, -6.09 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.088 | C290A | None | None | XRAY | 2.115 | 0.212 | 0.238 | A | 265 | 259 | 3 | 0 | 0 | 3 | [[133, 383]] | 1.0 | 8c1d | CAMK_AURKA_HUMAN | CAMK | 7.2e-79 | 270.6 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | AURKA | AURKA_HUMAN | 2W1FA | O14965 | 127 | 389 | 403.0 | L0F:61390 | Type1 | Inactive | DFGin | 5.655 | 15.703 | BLAminus | -96.26, 172.45 | 62.06, 107.69 | -118.91, 38.89 | 289.12, 66.42 | -59.62, -48.4 | out-out | out | 10.139 | Saltbr-out | 5.12 | HRD-in | -78.79, -54.88 | 78.03, -25.41 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.676 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -157.03 | APE8-dihe-in | -58.47, 105.92 | APE8-rot-out | 190.33 | APE67-dihe-in | -42.4, -27.58 | -64.36, -20.47 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.774 | None | None | None | XRAY | 2.85 | 0.246 | 0.348 | A | 275 | 253 | 10 | 0 | 0 | 10 | [[133, 383]] | 1.0 | 2w1f | CAMK_AURKA_HUMAN | CAMK | 6.7e-80 | 274.0 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | AURKA | AURKA_HUMAN | 3O51A | O14965 | 126 | 388 | 403.0 | LJF:1 | Type1.5_Front | Inactive | DFGout | 12.921 | 9.215 | None | -125.94, 46.56 | -78.14, 156.47 | -164.09, 999.0 | 59.42, 112.33 | 999.0, 999.0 | out-none | out | 12.863 | Saltbr-none | 999.0 | HRD-out | -126.02, 153.87 | -92.88, -115.51 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -57.91, -10.7 | 999.0, -51.84 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 3.2 | 0.288 | 0.304 | A | 267 | 246 | 17 | 0 | 0 | 17 | [[133, 383]] | 1.0 | 3o51 | CAMK_AURKA_HUMAN | CAMK | 6e-80 | 274.2 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | CAMK2A | KCC2A_HUMAN | 2VZ6A | Q9UQM7 | 9 | 299 | 478.0 | FEF:60600 | Type1 | Active | DFGin | 7.124 | 13.93 | BLAminus | -130.3, 144.9 | 77.59, 104.3 | -118.45, 37.91 | 281.19, 70.53 | -60.86, -31.43 | in-in | in | 9.032 | Saltbr-in | 2.623 | HRD-in | -71.43, -45.76 | 75.34, -9.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.805 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.76, 148.02 | APE9-dihe-na | 132.07, -168.34 | APE8-dihe-in | -120.79, 126.49 | APE8-rot-in | 299.71 | APE67-dihe-in | -63.07, -18.83 | -35.01, -58.7 | APE12-dist-in | 10.327 | APE11-dist-in | 11.819 | APE10-dist-in | 5.993 | APE9-dist-in | 3.832 | None | None | None | XRAY | 2.3 | 0.165 | 0.203 | A | 313 | 289 | 2 | 0 | 0 | 0 | [[13, 271]] | 1.0 | 2vz6 | CAMK_CAMK2A_HUMAN | CAMK | 1.6e-96 | 328.7 | 1 | 256 | 256 | 155 | 156 | 157 | 159 | 161 | 42 | 60 | 64 | 132 | 134 | 133 | 135 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 90 | Calcium/calmodulin-dependent protein kinase type II subunit alpha |
| CAMK | CAMK2A | KCC2A_HUMAN | 2VZ6B | Q9UQM7 | 9 | 300 | 478.0 | FEF:60600 | Type1 | Active | DFGin | 6.865 | 14.032 | BLAminus | -131.92, 139.26 | 77.54, 110.88 | -122.08, 32.95 | 286.68, 71.96 | -61.55, -26.54 | in-in | in | 9.31 | Saltbr-in | 2.931 | HRD-in | -73.12, -44.65 | 73.93, -20.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.874 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -148.21, 149.78 | APE9-dihe-na | 143.11, -171.05 | APE8-dihe-in | -118.3, 128.44 | APE8-rot-in | 303.95 | APE67-dihe-in | -66.72, -18.78 | -39.97, -52.82 | APE12-dist-in | 10.252 | APE11-dist-in | 11.756 | APE10-dist-in | 5.996 | APE9-dist-in | 3.963 | None | None | None | XRAY | 2.3 | 0.165 | 0.203 | B | 313 | 292 | 0 | 0 | 0 | 0 | [[13, 271]] | 1.0 | 2vz6 | CAMK_CAMK2A_HUMAN | CAMK | 1.6e-96 | 328.7 | 1 | 256 | 256 | 155 | 156 | 157 | 159 | 161 | 42 | 60 | 64 | 132 | 134 | 133 | 135 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 90 | Calcium/calmodulin-dependent protein kinase type II subunit alpha |
| CAMK | CHEK1 | CHK1_HUMAN | 8E80A | O14757 | 8 | 271 | 476.0 | UUF:301 | Type1 | Active | DFGin | 6.948 | 13.561 | BLAminus | -116.38, 163.51 | 69.37, 105.0 | -111.89, 20.17 | 292.16, 81.73 | -65.53, -30.68 | in-in | in | 8.579 | Saltbr-in | 2.859 | HRD-in | -73.57, -45.75 | 72.69, 0.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.949 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -163.33, 170.54 | APE9-dihe-na | 117.83, -149.18 | APE8-dihe-in | -134.92, 121.74 | APE8-rot-in | 303.05 | APE67-dihe-in | -62.91, -20.27 | -44.12, -51.23 | APE12-dist-in | 9.365 | APE11-dist-in | 11.644 | APE10-dist-in | 6.142 | APE9-dist-in | 3.497 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | None | XRAY | 1.49 | 0.209 | 0.242 | A | 297 | 258 | 6 | 0 | 0 | 0 | [[9, 265]] | 1.0 | 8e80 | CAMK_CHEK1_HUMAN | CAMK | 4.8e-69 | 238.4 | 2 | 256 | 255 | 147 | 148 | 149 | 151 | 153 | 38 | 55 | 59 | 127 | 129 | 128 | 130 | 190 | 177 | 172 | 171 | 170 | 169 | 168 | 167 | 166 | 85 | Serine/threonine-protein kinase Chk1 |
| CAMK | CHEK2 | CHK2_HUMAN | 2YCFA | O96017 | 210 | 510 | 543.0 | YCF:600 | Type1 | Inactive | DFGin | 6.651 | 14.425 | BLAminus | -133.14, 179.08 | 68.92, 89.26 | -105.02, 26.49 | 290.18, 77.38 | -65.99, -23.19 | in-out | in | 9.994 | Saltbr-out | 8.56 | HRD-in | -70.72, -52.98 | 75.15, -0.9 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.905 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -72.28, -26.54 | APE9-dihe-na | -96.81, -179.54 | APE8-dihe-in | -85.38, 132.85 | APE8-rot-in | 297.44 | APE67-dihe-in | -44.53, -40.92 | -82.1, 28.65 | APE12-dist-out | 25.231 | APE11-dist-out | 27.289 | APE10-dist-out | 29.363 | APE9-dist-out | 33.105 | None | None | None | XRAY | 1.77 | 0.197 | 0.218 | A | 322 | 286 | 15 | 0 | 0 | 0 | [[220, 486]] | 1.0 | 2ycf | CAMK_CHEK2_HUMAN | CAMK | 2e-85 | 292.2 | 1 | 256 | 256 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | DAPK1 | DAPK1_HUMAN | 6AARA | P53355 | 2 | 277 | 1430.0 | 9TF:300 | Type1 | Inactive | DFGin | 6.743 | 14.342 | BLAminus | -121.31, 178.32 | 64.29, 78.62 | -87.38, 15.28 | 286.92, 75.84 | -59.31, -26.74 | in-in | in | 9.386 | Saltbr-in | 2.811 | HRD-in | -76.03, -46.41 | 70.92, -12.19 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.921 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -137.91, 116.13 | APE9-dihe-na | -97.58, -145.9 | APE8-dihe-in | -81.4, 124.5 | APE8-rot-in | 302.0 | APE67-dihe-in | -55.21, -31.9 | -47.73, -42.04 | APE12-dist-in | 11.019 | APE11-dist-out | 6.26 | APE10-dist-out | 9.242 | APE9-dist-in | 4.805 | None | None | None | XRAY | 1.95 | 0.182 | 0.22 | A | 293 | 269 | 7 | 0 | 0 | 0 | [[13, 275]] | 1.0 | 6aar | CAMK_DAPK1_HUMAN | CAMK | 6.1e-95 | 323.3 | 1 | 256 | 256 | 160 | 161 | 162 | 164 | 166 | 42 | 64 | 68 | 136 | 138 | 137 | 139 | 199 | 187 | 182 | 181 | 180 | 179 | 178 | 177 | 176 | 94 | Death-associated protein kinase 1 |
| CAMK | MAPKAPK2 | MAPK2_HUMAN | 3M42A | P49137 | 47 | 364 | 400.0 | HGF:365 | Type1 | None | DFGin | 4.265 | 13.765 | BLAminus | -127.28, 170.7 | 71.87, 101.44 | -103.87, 20.75 | 277.01, 69.5 | -61.92, -8.22 | in-in | in | 9.26 | Saltbr-in | 3.091 | HRD-in | -73.72, -58.45 | 76.25, 11.76 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.912 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | P237G | None | None | XRAY | 2.68 | 0.186 | 0.232 | A | 299 | 290 | 7 | 0 | 0 | 0 | [[63, 325]] | 1.0 | 3m42 | CAMK_MAPKAPK2_HUMAN | CAMK | 1.9e-36 | 228.6 | 3 | 154 | 236 | 206 | 207 | 208 | 210 | 212 | 93 | 104 | 108 | 183 | 185 | 184 | 186 | 245 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 139 | MAP kinase-activated protein kinase 2 |
| CAMK | MELK | MELK_HUMAN | 5IH9A | Q14680 | 3 | 327 | 651.0 | 6BF:60401 | Type1 | None | DFGin | 6.939 | 15.146 | BLAminus | -123.48, 176.08 | 58.26, 79.91 | -95.72, 21.84 | 280.98, 78.3 | -67.92, -25.97 | in-in | in | 8.72 | Saltbr-in | 2.587 | HRD-in | -71.83, -48.59 | 72.02, -0.04 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.992 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -4.81 | APE8-rot-in | 291.01 | APE67-dihe-in | -55.95, -27.86 | -55.75, -43.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.79 | 0.174 | 0.2 | A | 335 | 307 | 18 | 0 | 0 | 14 | [[11, 263]] | 1.0 | 5ih9 | CAMK_MELK_HUMAN | CAMK | 9.7e-89 | 303.1 | 1 | 256 | 256 | 149 | 150 | 151 | 153 | 155 | 40 | 57 | 61 | 129 | 131 | 130 | 132 | 191 | 178 | 173 | 172 | 171 | 170 | 169 | 168 | 167 | 87 | Maternal embryonic leucine zipper kinase |
| CAMK | PIM1 | PIM1_HUMAN | 5KGIA | P11309 | 33 | 305 | 313.0 | 6SF:414 | Type1 | Active | DFGin | 6.196 | 14.678 | BLAminus | -128.85, 173.72 | 58.37, 80.83 | -91.15, 15.65 | 283.15, 78.86 | -67.29, -15.19 | in-in | in | 8.898 | Saltbr-in | 2.699 | HRD-na-A | -66.85, -48.52 | 69.49, 3.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.854 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.48, 30.3 | APE9-dihe-na | -88.67, -155.26 | APE8-dihe-in | -89.24, 121.14 | APE8-rot-in | 310.96 | APE67-dihe-in | -66.24, -12.88 | -55.29, -44.34 | APE12-dist-in | 9.723 | APE11-dist-in | 8.735 | APE10-dist-in | 5.642 | APE9-dist-in | 3.74 | None | None | None | XRAY | 2.13 | 0.173 | 0.186 | A | 276 | 273 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 5kgi | CAMK_PIM1_HUMAN | CAMK | 2.5e-65 | 226.2 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 6L13A | P11309 | 33 | 305 | 313.0 | E2F:401 | Type1 | Active | DFGin | 6.19 | 14.786 | BLAminus | -130.24, 168.2 | 68.46, 80.68 | -89.17, 16.05 | 288.1, 80.31 | -69.01, -19.61 | in-in | in | 9.105 | Saltbr-in | 2.936 | HRD-na-A | -68.46, -51.8 | 71.9, 8.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.778 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.76, 29.56 | APE9-dihe-na | -92.34, -153.25 | APE8-dihe-in | -98.43, 124.2 | APE8-rot-in | 303.55 | APE67-dihe-in | -68.48, -12.49 | -58.68, -45.06 | APE12-dist-in | 9.5 | APE11-dist-in | 8.511 | APE10-dist-in | 5.099 | APE9-dist-in | 3.659 | None | SEP261 | SEP261 | XRAY | 2.24 | 0.18 | 0.214 | A | 289 | 273 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 6l13 | CAMK_PIM1_HUMAN | CAMK | 3e-65 | 226.0 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 2O65A | P11309 | 33 | 306 | 313.0 | MYF:501 | Type1 | Active | DFGin | 5.773 | 14.223 | BLAminus | -134.9, 170.04 | 60.08, 89.22 | -101.35, 10.62 | 287.34, 92.73 | -63.96, -9.9 | in-in | in | 8.704 | Saltbr-in | 2.471 | HRD-na-A | -65.14, -47.59 | 70.03, -4.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.98 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.66, 34.64 | APE9-dihe-na | -104.35, -148.26 | APE8-dihe-in | -83.11, 121.1 | APE8-rot-in | 316.59 | APE67-dihe-in | -62.15, -16.44 | -57.04, -47.52 | APE12-dist-in | 9.988 | APE11-dist-in | 8.628 | APE10-dist-in | 5.289 | APE9-dist-in | 4.136 | None | None | None | XRAY | 2.85 | 0.21 | 0.262 | A | 293 | 274 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 2o65 | CAMK_PIM1_HUMAN | CAMK | 3.2e-65 | 226.0 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 8R0WA | P11309 | 33 | 305 | 313.0 | XGF:405 | Type1 | Active | DFGin | 5.997 | 14.384 | BLAminus | -131.73, 166.77 | 65.97, 82.46 | -89.79, 16.41 | 289.35, 79.56 | -63.02, -16.4 | in-in | in | 8.812 | Saltbr-in | 2.643 | HRD-na-A | -73.15, -45.35 | 65.43, 10.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.23, 17.26 | APE9-dihe-na | -81.93, -156.28 | APE8-dihe-in | -91.39, 121.88 | APE8-rot-in | 296.84 | APE67-dihe-in | -71.92, -8.94 | -64.52, -38.27 | APE12-dist-in | 9.559 | APE11-dist-in | 8.479 | APE10-dist-in | 5.116 | APE9-dist-in | 3.713 | R250G | SEP261 | SEP261 | XRAY | 1.95 | 0.167 | 0.201 | A | 313 | 273 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 8r0w | CAMK_PIM1_HUMAN | CAMK | 1.5e-64 | 223.7 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 8AFRA | P11309 | 33 | 305 | 313.0 | M0F:401 | Type1 | Active | DFGin | 6.024 | 14.406 | BLAminus | -126.46, 177.16 | 55.61, 83.44 | -89.48, 19.88 | 284.93, 74.96 | -67.33, -13.52 | in-in | in | 8.831 | Saltbr-in | 2.648 | HRD-na-A | -72.52, -48.51 | 66.56, 10.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.815 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.4, 19.87 | APE9-dihe-na | -78.39, -149.93 | APE8-dihe-in | -97.85, 123.61 | APE8-rot-in | 301.25 | APE67-dihe-in | -68.16, -10.25 | -64.9, -40.75 | APE12-dist-in | 9.727 | APE11-dist-in | 8.467 | APE10-dist-in | 5.304 | APE9-dist-in | 3.645 | R250G | SEP261 | SEP261 | XRAY | 2.15 | 0.166 | 0.191 | A | 309 | 264 | 7 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 8afr | CAMK_PIM1_HUMAN | CAMK | 3.1e-62 | 216.2 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CMGC | CDK12 | CDK12_HUMAN | 8BU5B | Q9NYV4 | 713 | 1044 | 1490.0 | RMF:1101 | Type1 | Inactive | DFGin | 6.801 | 14.701 | ABAminus | -126.95, -66.04 | -93.95, 105.24 | -102.41, 30.18 | 293.69, 100.66 | -84.84, -22.58 | in-out | in | 8.305 | Saltbr-out | 3.933 | HRD-out | -78.59, 106.12 | -94.17, 5.74 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.828 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -136.91, -22.25 | APE9-dihe-na | -109.89, 157.52 | APE8-dihe-in | -56.01, 131.78 | APE8-rot-in | 308.02 | APE67-dihe-in | -60.99, -26.61 | -52.03, -40.26 | APE12-dist-out | 14.28 | APE11-dist-in | 11.941 | APE10-dist-in | 7.36 | APE9-dist-in | 3.767 | K965R | TPO893 | TPO893 | XRAY | 3.134 | 0.2 | 0.22 | B | 344 | 332 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bu5 | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BU5H | Q9NYV4 | 713 | 1043 | 1490.0 | RMF:1101 | Type1 | Inactive | DFGin | 7.015 | 14.978 | ABAminus | -128.46, -54.53 | -90.71, 103.12 | -97.22, 31.8 | 290.43, 81.59 | -85.33, -25.69 | in-in | in | 8.479 | Saltbr-in | 3.527 | HRD-in | -73.55, -49.58 | 63.85, -4.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.629 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.5, -28.02 | APE9-dihe-na | -97.36, 153.71 | APE8-dihe-in | -57.72, 135.61 | APE8-rot-in | 311.07 | APE67-dihe-in | -63.38, -27.52 | -50.57, -39.59 | APE12-dist-in | 13.941 | APE11-dist-in | 12.128 | APE10-dist-in | 7.258 | APE9-dist-in | 3.497 | K965R | TPO893 | TPO893 | XRAY | 3.134 | 0.2 | 0.22 | H | 344 | 331 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bu5 | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BUNB | Q9NYV4 | 715 | 1041 | 1490.0 | RNF:61101 | Type1 | Inactive | DFGin | 7.009 | 15.297 | ABAminus | -131.36, -49.43 | -89.83, 91.44 | -92.44, 32.63 | 287.3, 77.5 | -75.27, -18.22 | in-in | in | 7.748 | Saltbr-in | 3.279 | HRD-in | -75.67, -53.71 | 75.4, -0.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.923 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.12, -39.12 | APE9-dihe-na | -104.98, 151.97 | APE8-dihe-in | -58.93, 142.91 | APE8-rot-in | 279.94 | APE67-dihe-in | -65.42, -33.6 | -55.06, -35.14 | APE12-dist-in | 13.388 | APE11-dist-in | 11.695 | APE10-dist-in | 7.099 | APE9-dist-in | 3.657 | K965R | TPO893 | TPO893 | XRAY | 3.08 | 0.187 | 0.211 | B | 344 | 327 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bun | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BUNH | Q9NYV4 | 715 | 1043 | 1490.0 | RNF:61101 | Type1 | Inactive | DFGin | 7.045 | 15.286 | ABAminus | -125.24, -50.09 | -100.69, 94.75 | -92.24, 30.97 | 286.18, 71.82 | -75.42, -18.26 | in-in | in | 7.834 | Saltbr-in | 3.373 | HRD-in | -77.6, -54.36 | 73.0, -1.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.74 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.56, -41.65 | APE9-dihe-na | -95.79, 153.05 | APE8-dihe-in | -58.87, 144.43 | APE8-rot-in | 305.25 | APE67-dihe-in | -65.98, -31.29 | -55.83, -37.71 | APE12-dist-in | 13.775 | APE11-dist-in | 11.972 | APE10-dist-in | 6.957 | APE9-dist-in | 3.478 | K965R | TPO893 | TPO893 | XRAY | 3.08 | 0.187 | 0.211 | H | 344 | 329 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bun | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 9FMRE | Q9NYV4 | 714 | 1042 | 1490.0 | RMF:61101 | Type1 | Inactive | DFGin | 6.793 | 14.64 | ABAminus | -113.83, -79.52 | -84.15, 118.47 | -115.27, 16.16 | 293.54, 100.02 | -64.02, -34.33 | in-out | in | 9.633 | Saltbr-out | 3.612 | HRD-out | -79.17, 82.22 | -59.96, 8.89 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.026 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -148.14, -27.51 | APE9-dihe-na | -104.44, 148.12 | APE8-dihe-in | -51.45, 137.55 | APE8-rot-in | 306.02 | APE67-dihe-in | -70.5, -21.3 | -54.61, -36.19 | APE12-dist-out | 14.298 | APE11-dist-in | 12.211 | APE10-dist-in | 7.469 | APE9-dist-in | 3.767 | None | TPO893 | TPO893 | XRAY | 3.9 | 0.209 | 0.25 | E | 351 | 329 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 9fmr | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 9FMRH | Q9NYV4 | 714 | 1044 | 1490.0 | RMF:61101 | Type1 | Inactive | DFGin | 6.801 | 14.603 | ABAminus | -113.95, -78.4 | -84.85, 124.02 | -118.87, 17.95 | 291.29, 89.7 | -63.88, -35.4 | in-in | in | 8.592 | Saltbr-in | 3.552 | HRD-in | -72.47, -40.65 | 59.82, 5.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.74, -27.71 | APE9-dihe-na | -103.25, 148.34 | APE8-dihe-in | -51.07, 136.63 | APE8-rot-in | 306.14 | APE67-dihe-in | -69.99, -21.15 | -54.39, -34.8 | APE12-dist-in | 13.823 | APE11-dist-in | 12.098 | APE10-dist-in | 7.255 | APE9-dist-in | 3.608 | None | TPO893 | TPO893 | XRAY | 3.9 | 0.209 | 0.25 | H | 351 | 331 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 9fmr | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BUNE | Q9NYV4 | 715 | 1039 | 1490.0 | RNF:61101 | Type1 | Inactive | DFGin | 7.217 | 15.313 | BLAminus | -143.55, -179.06 | 50.55, 77.42 | -92.12, 34.85 | 285.27, 76.47 | -72.26, -18.51 | in-in | in | 7.824 | Saltbr-in | 3.046 | HRD-in | -77.13, -53.65 | 75.0, -0.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.924 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -105.31, -34.23 | APE9-dihe-na | -92.08, 151.91 | APE8-dihe-in | -57.84, 145.99 | APE8-rot-out | 175.35 | APE67-dihe-in | -65.98, -29.37 | -55.72, -38.5 | APE12-dist-in | 13.18 | APE11-dist-in | 12.611 | APE10-dist-in | 7.008 | APE9-dist-in | 3.432 | K965R | TPO893 | TPO893 | XRAY | 3.08 | 0.187 | 0.211 | E | 344 | 325 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bun | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8P81A | Q9NYV4 | 716 | 1035 | 1490.0 | RMF:1101 | Type1 | Active | DFGin | 7.095 | 14.446 | BLAminus | -134.83, -178.64 | 59.2, 72.19 | -89.53, 34.88 | 291.56, 80.44 | -67.97, -22.73 | in-in | in | 8.359 | Saltbr-in | 3.057 | HRD-in | -81.5, -42.97 | 59.01, 18.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.963 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.63, 165.61 | APE9-dihe-na | 67.08, 139.25 | APE8-dihe-in | -61.99, 152.33 | APE8-rot-in | 316.49 | APE67-dihe-in | -68.12, -20.85 | -57.98, -41.98 | APE12-dist-in | 12.679 | APE11-dist-in | 10.561 | APE10-dist-in | 6.52 | APE9-dist-in | 3.212 | None | TPO893 | TPO893 | XRAY | 2.68 | 0.212 | 0.255 | A | 351 | 320 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8p81 | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BU5E | Q9NYV4 | 713 | 1043 | 1490.0 | RMF:1101 | Type1 | Inactive | DFGin | 6.942 | 15.122 | None | -123.64, -63.66 | -81.97, -51.09 | 56.28, 22.54 | 292.49, 98.9 | -91.33, -28.22 | in-out | in | 8.371 | Saltbr-out | 3.622 | HRD-in | -72.77, -54.57 | 74.45, -4.91 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.759 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -134.16, -27.33 | APE9-dihe-na | -98.05, 157.33 | APE8-dihe-in | -51.55, 136.25 | APE8-rot-in | 308.17 | APE67-dihe-in | -63.16, -26.85 | -49.17, -41.17 | APE12-dist-out | 14.125 | APE11-dist-in | 12.168 | APE10-dist-in | 7.286 | APE9-dist-in | 3.726 | K965R | TPO893 | TPO893 | XRAY | 3.134 | 0.2 | 0.22 | E | 344 | 331 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bu5 | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 9FMRB | Q9NYV4 | 714 | 1047 | 1490.0 | RMF:61101 | Type1 | Inactive | DFGin | 7.124 | 15.031 | None | -111.49, -74.26 | -77.99, -72.15 | 68.85, 12.84 | 296.16, 89.8 | -66.22, -36.51 | in-out | in | 8.332 | Saltbr-out | 4.45 | HRD-in | -70.8, -35.56 | 62.81, 1.22 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.072 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.03, -25.75 | APE9-dihe-na | -103.56, 146.88 | APE8-dihe-in | -51.72, 138.27 | APE8-rot-in | 305.58 | APE67-dihe-in | -69.51, -21.36 | -53.61, -35.19 | APE12-dist-in | 13.987 | APE11-dist-in | 12.27 | APE10-dist-in | 7.331 | APE9-dist-in | 3.865 | None | TPO893 | TPO893 | XRAY | 3.9 | 0.209 | 0.25 | B | 351 | 334 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 9fmr | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK16 | CDK16_HUMAN | 3MTLA | Q00536 | 163 | 473 | 496.0 | FEF:60668 | Type1 | Inactive | DFGout | 17.399 | 7.472 | None | -75.13, 154.32 | -88.9, 77.74 | -154.62, 116.54 | 227.56, 88.74 | 78.03, 21.89 | in-in | in | 8.385 | Saltbr-in | 2.641 | HRD-out | -101.69, 108.56 | -74.19, -25.04 | in-out-out | SNCioo | out-out | ActLoopNT-out | 5.164 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 102.89 | APE8-rot-out | 156.53 | APE67-dihe-in | -61.54, -35.29 | -78.56, -14.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | S319D | None | None | XRAY | 2.4 | 0.198 | 0.263 | A | 324 | 293 | 18 | 0 | 0 | 12 | [[165, 446]] | 1.0 | 3mtl | CMGC_CDK16_HUMAN | CMGC | 1.3e-83 | 286.9 | 1 | 301 | 301 | 303 | 304 | 305 | 307 | 309 | 194 | 211 | 215 | 283 | 285 | 284 | 286 | 344 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 241 | Cyclin-dependent kinase 16 |
| CMGC | CDK2 | CDK2_HUMAN | 9ESWA | P24941 | 1 | 294 | 298.0 | IJF:60301,IJF:60302,IJF:60303,IJF:60304 | Allosteric,Type1,Allosteric,Allosteric | Active | DFGin | 6.515 | 15.297 | BLAminus | -143.94, 174.07 | 58.52, 82.55 | -94.4, 25.35 | 278.47, 68.95 | -74.76, -22.16 | in-in | in | 8.637 | Saltbr-in | 3.197 | HRD-in | -81.26, -58.57 | 77.56, 16.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.996 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -61.44, 160.94 | APE9-dihe-na | 81.67, 126.4 | APE8-dihe-in | -51.25, 136.17 | APE8-rot-in | 300.7 | APE67-dihe-in | -59.48, -16.12 | -52.59, -48.63 | APE12-dist-in | 12.997 | APE11-dist-in | 11.897 | APE10-dist-in | 7.023 | APE9-dist-in | 3.204 | None | TPO160 | TPO160 | XRAY | 2.38 | 0.233 | 0.239 | A | 302 | 294 | 0 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 9esw | CMGC_CDK2_HUMAN | CMGC | 6.7e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 9ESWC | P24941 | 1 | 296 | 298.0 | IJF:60301,IJF:60302,IJF:60303,IJF:60304 | Allosteric,Type1,Allosteric,Allosteric | Active | DFGin | 6.576 | 15.209 | BLAminus | -137.9, -176.23 | 48.55, 71.41 | -85.05, 25.18 | 283.44, 66.65 | -62.35, -32.95 | in-in | in | 8.417 | Saltbr-in | 2.763 | HRD-in | -83.58, -58.72 | 75.84, 9.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.887 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.32, 151.2 | APE9-dihe-na | 72.23, 131.64 | APE8-dihe-in | -58.77, 140.82 | APE8-rot-in | 312.4 | APE67-dihe-in | -51.92, -26.23 | -42.04, -57.02 | APE12-dist-in | 12.776 | APE11-dist-in | 10.195 | APE10-dist-in | 6.943 | APE9-dist-in | 3.236 | None | TPO160 | TPO160 | XRAY | 2.38 | 0.233 | 0.239 | C | 302 | 269 | 27 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 9esw | CMGC_CDK2_HUMAN | CMGC | 6.7e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 9OB4A | P24941 | 1 | 298 | 298.0 | A1CAF:301 | Type1 | Active | DFGin | 7.07 | 15.433 | BLAminus | -140.78, 171.16 | 58.81, 81.21 | -94.48, 18.25 | 279.35, 70.51 | -60.63, -24.89 | in-in | in | 8.702 | Saltbr-in | 2.578 | HRD-in | -77.49, -52.8 | 70.85, 9.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.858 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -103.4, 171.78 | APE9-dihe-na | 71.79, 138.58 | APE8-dihe-in | -59.97, 144.28 | APE8-rot-in | 298.9 | APE67-dihe-in | -65.05, -23.77 | -53.99, -47.04 | APE12-dist-in | 13.149 | APE11-dist-in | 12.232 | APE10-dist-in | 7.357 | APE9-dist-in | 3.261 | None | TPO160 | TPO160 | XRAY | 1.95 | 0.211 | 0.251 | A | 301 | 298 | 0 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 9ob4 | CMGC_CDK2_HUMAN | CMGC | 6.6e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 4BCQA | P24941 | 1 | 295 | 298.0 | TJF:61296 | Type1 | Active | DFGin | 6.591 | 15.979 | BLAminus | -145.97, 170.46 | 62.82, 84.99 | -99.38, 29.59 | 282.23, 71.6 | -71.19, -18.61 | in-in | in | 9.404 | Saltbr-in | 3.453 | HRD-in | -85.05, -58.94 | 78.36, 12.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.147 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.8, 176.97 | APE9-dihe-na | 69.33, 133.29 | APE8-dihe-in | -55.38, 139.69 | APE8-rot-in | 304.09 | APE67-dihe-in | -55.84, -22.0 | -49.63, -50.65 | APE12-dist-in | 13.625 | APE11-dist-in | 12.543 | APE10-dist-in | 7.498 | APE9-dist-in | 3.511 | None | TPO160 | TPO160 | XRAY | 2.4 | 0.217 | 0.252 | A | 301 | 290 | 5 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 4bcq | CMGC_CDK2_HUMAN | CMGC | 6.6e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 4BCQC | P24941 | 1 | 294 | 298.0 | TJF:61295 | Type1 | Active | DFGin | 6.54 | 16.003 | BLAminus | -147.36, 170.23 | 59.21, 86.27 | -98.9, 28.16 | 278.44, 72.82 | -71.37, -12.42 | in-in | in | 9.598 | Saltbr-in | 3.261 | HRD-in | -88.13, -59.99 | 74.18, 19.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.909 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.48, 157.26 | APE9-dihe-na | 69.58, 129.95 | APE8-dihe-in | -57.66, 135.49 | APE8-rot-in | 301.27 | APE67-dihe-in | -62.84, -20.05 | -48.44, -46.81 | APE12-dist-in | 13.54 | APE11-dist-in | 10.682 | APE10-dist-in | 7.689 | APE9-dist-in | 3.66 | None | TPO160 | TPO160 | XRAY | 2.4 | 0.217 | 0.252 | C | 301 | 292 | 2 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 4bcq | CMGC_CDK2_HUMAN | CMGC | 6.6e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 7S9XA | P24941 | 3 | 298 | 298.0 | 8KF:301 | Type3 | Inactive | DFGin | 9.152 | 14.904 | BLBminus | -140.51, 174.83 | 55.24, 52.61 | -60.52, 155.06 | 283.44, 65.83 | -96.54, 51.03 | out-out | out | 17.021 | Saltbr-out | 17.405 | HRD-in | -80.98, -57.39 | 84.63, -18.55 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.299 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, 131.76 | APE9-dihe-na | -82.0, 133.39 | APE8-dihe-in | -82.83, 123.04 | APE8-rot-in | 299.71 | APE67-dihe-in | -59.76, -23.84 | -102.49, -0.32 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.12 | APE9-dist-out | 11.022 | None | None | None | XRAY | 1.69 | 0.231 | 0.262 | A | 298 | 269 | 27 | 0 | 0 | 12 | [[4, 286]] | 1.0 | 7s9x | CMGC_CDK2_HUMAN | CMGC | 6.3e-90 | 307.9 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 2W1HA | P24941 | 1 | 298 | 298.0 | L0F:1299 | Type1 | Inactive | DFGin | 10.307 | 17.775 | BLBtrans | -130.06, 151.5 | 79.56, 18.75 | -69.93, 141.61 | 226.73, 121.67 | 69.65, -12.05 | out-out | out | 14.489 | Saltbr-out | 16.038 | HRD-in | -88.39, -56.31 | 79.17, -16.22 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.457 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 121.46 | APE8-dihe-in | -76.22, 142.93 | APE8-rot-out | 186.46 | APE67-dihe-in | -49.35, -36.85 | -110.85, -4.12 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.805 | None | None | None | XRAY | 2.15 | 0.263 | 0.308 | A | 298 | 283 | 15 | 0 | 0 | 11 | [[4, 286]] | 1.0 | 2w1h | CMGC_CDK2_HUMAN | CMGC | 6.3e-90 | 307.9 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 2R3IA | P24941 | 1 | 298 | 298.0 | SCF:60501 | Type1 | Inactive | DFGin | 10.929 | 18.24 | BLBtrans | -100.61, 149.54 | 71.45, 21.63 | -58.2, 134.86 | 231.09, 103.4 | 83.18, -10.48 | out-out | out | 15.057 | Saltbr-out | 16.345 | HRD-in | -91.01, -59.76 | 82.13, -15.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.707 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -70.45, 127.61 | APE9-dihe-na | -74.97, 122.45 | APE8-dihe-in | -60.32, 144.67 | APE8-rot-out | 191.76 | APE67-dihe-in | -59.78, -26.25 | -99.25, -5.87 | APE12-dist-out | 20.169 | APE11-dist-out | 17.538 | APE10-dist-out | 18.889 | APE9-dist-out | 9.991 | None | None | CSD177 | XRAY | 1.28 | 0.178 | 0.202 | A | 299 | 291 | 7 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 2r3i | CMGC_CDK2_HUMAN | CMGC | 6.4e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 5IEXA | P24941 | 1 | 298 | 298.0 | 6AF:1001 | Type1 | Inactive | None | 11.106 | 18.344 | None | -105.6, 149.53 | 71.37, 22.65 | -61.85, 135.15 | 236.62, 103.3 | 74.49, -10.58 | out-out | out | 15.176 | Saltbr-out | 15.226 | HRD-in | -80.72, -65.3 | 84.99, -26.41 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.802 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 111.81 | APE8-dihe-in | -112.57, 117.73 | APE8-rot-in | 277.98 | APE67-dihe-in | -67.92, -29.52 | -99.02, -2.25 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.275 | None | None | None | XRAY | 2.03 | 0.206 | 0.254 | A | 298 | 285 | 13 | 0 | 0 | 8 | [[4, 286]] | 1.0 | 5iex | CMGC_CDK2_HUMAN | CMGC | 6.3e-90 | 307.9 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK6 | CDK6_HUMAN | 9PE7A | Q00534 | 10 | 301 | 326.0 | A1CIF:900 | Type1 | Inactive | DFGin | 6.872 | 13.127 | BLBplus | -137.4, 169.29 | 57.4, 61.63 | -142.77, 164.35 | 61.09, 86.59 | 91.92, -16.71 | out-out | out | 12.416 | Saltbr-out | 9.93 | HRD-in | -63.73, -52.58 | 73.19, -16.54 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, 162.46 | APE9-dihe-na | -100.9, 174.34 | APE8-dihe-in | -134.69, 96.5 | APE8-rot-in | 306.93 | APE67-dihe-in | -54.43, -27.6 | -93.0, -5.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 22.373 | APE9-dist-out | 12.123 | E21V,K26T,T106R,Q149E | None | None | XRAY | 2.05 | 0.216 | 0.267 | A | 307 | 262 | 30 | 0 | 0 | 12 | [[13, 300]] | 1.0 | 9pe7 | CMGC_CDK6_HUMAN | CMGC | 3.7e-84 | 289.5 | 1 | 301 | 301 | 162 | 163 | 164 | 166 | 168 | 43 | 61 | 65 | 142 | 144 | 143 | 145 | 201 | 189 | 184 | 183 | 182 | 181 | 180 | 179 | 178 | 99 | Cyclin-dependent kinase 6 |
| CMGC | CDK7 | CDK7_HUMAN | 8P71J | P50613 | 10 | 310 | 346.0 | X4F:60401 | Type1 | Active | DFGin | 6.832 | 15.304 | BLAminus | -139.46, 179.9 | 57.59, 64.02 | -82.45, 17.71 | 282.17, 74.47 | -64.72, -19.22 | in-in | in | 8.103 | Saltbr-in | 2.694 | HRD-in | -67.33, -49.46 | 65.63, 5.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.639 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.68, 168.49 | APE9-dihe-na | 67.33, 140.05 | APE8-dihe-in | -60.3, 143.93 | APE8-rot-in | 294.53 | APE67-dihe-in | -61.0, -25.19 | -55.87, -41.76 | APE12-dist-in | 13.411 | APE11-dist-in | 11.192 | APE10-dist-in | 6.803 | APE9-dist-in | 3.276 | None | None | None | EM | 2.0 | 999.0 | 999.0 | J | 349 | 286 | 15 | 0 | 0 | 0 | [[12, 295]] | 1.0 | 8p71 | CMGC_CDK7_HUMAN | CMGC | 1.6e-78 | 271.7 | 1 | 301 | 301 | 154 | 155 | 156 | 158 | 160 | 41 | 62 | 66 | 134 | 136 | 135 | 137 | 195 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Cyclin-dependent kinase 7 |
| CMGC | CDK8 | CDK8_HUMAN | 9H8SA | P49336 | 1 | 362 | 464.0 | A1ITF:60509 | Type1 | Inactive | DFGin | 7.344 | 13.924 | BLAminus | -119.28, 163.44 | 74.84, 82.25 | -92.61, 11.91 | 298.93, 132.0 | -87.41, 10.8 | in-in | in | 8.612 | Saltbr-in | 2.624 | HRD-in | -75.25, -51.5 | 79.06, -6.52 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.659 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 160.05 | APE8-rot-out | 75.96 | APE67-dihe-in | -54.19, -23.95 | -111.96, 19.45 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.157 | 0.197 | 0.248 | A | 414 | 335 | 27 | 0 | 0 | 17 | [[22, 335]] | 1.0 | 9h8s | CMGC_CDK8_HUMAN | CMGC | 6.3e-82 | 281.3 | 5 | 301 | 297 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 8AEMA | P68400 | 3 | 329 | 391.0 | LVF:407,ATP:408 | Allosteric,ATPlike | Active | DFGin | 7.399 | 16.187 | BLAminus | -114.2, -178.47 | 56.21, 75.05 | -90.39, 15.9 | 296.69, 81.8 | -66.43, -20.83 | in-in | in | 9.132 | Saltbr-in | 2.816 | HRD-in | -72.91, -51.16 | 68.69, 11.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.905 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.83, 169.06 | APE9-dihe-na | 58.87, 157.76 | APE8-dihe-in | -77.1, 150.54 | APE8-rot-in | 294.73 | APE67-dihe-in | -68.78, -13.55 | -40.19, -53.95 | APE12-dist-in | 12.744 | APE11-dist-in | 10.417 | APE10-dist-in | 6.256 | APE9-dist-in | 3.215 | R21S,K74A,K75A,K76A | None | None | XRAY | 1.6 | 0.19 | 0.212 | A | 328 | 327 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 8aem | CMGC_CSNK2A1_HUMAN | CMGC | 8.1e-69 | 238.0 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9EPWB | P68400 | 3 | 333 | 391.0 | A1H6F:406 | Type1 | Active | DFGin | 7.386 | 16.279 | BLAminus | -118.5, 178.76 | 54.91, 76.82 | -86.63, 13.68 | 291.49, 81.55 | -67.5, -20.83 | out-in | out | 10.046 | Saltbr-in | 3.292 | HRD-in | -71.7, -52.07 | 70.7, 14.03 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.882 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.62, 167.98 | APE9-dihe-na | 70.49, 159.89 | APE8-dihe-in | -76.41, 141.74 | APE8-rot-in | 289.66 | APE67-dihe-in | -68.82, -20.3 | -42.56, -42.98 | APE12-dist-in | 12.795 | APE11-dist-in | 10.921 | APE10-dist-in | 6.279 | APE9-dist-in | 3.382 | None | None | None | XRAY | 2.3 | 0.261 | 0.308 | B | 338 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9epw | CMGC_CSNK2A1_HUMAN | CMGC | 1.4e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 2ZJWA | P68400 | 1 | 332 | 391.0 | REF:336 | Type1 | Inactive | DFGin | 7.316 | 16.527 | BLAminus | -109.16, -168.7 | 44.38, 76.01 | -90.89, 24.26 | 297.46, 77.89 | -76.15, -7.13 | in-in | in | 9.417 | Saltbr-in | 2.731 | HRD-in | -72.0, -50.11 | 70.44, 13.49 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.907 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -14.58, 161.89 | APE9-dihe-na | 62.59, 163.98 | APE8-dihe-in | -84.5, 146.1 | APE8-rot-out | 153.88 | APE67-dihe-in | -63.0, -17.21 | -40.84, -52.94 | APE12-dist-in | 12.607 | APE11-dist-in | 8.948 | APE10-dist-in | 5.933 | APE9-dist-in | 2.992 | None | None | None | XRAY | 2.4 | 0.222 | 0.274 | A | 340 | 332 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 2zjw | CMGC_CSNK2A1_HUMAN | CMGC | 1.4e-69 | 240.5 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 7I8AA | P68400 | 3 | 329 | 391.0 | A1B0F:401 | Type1 | Active | DFGin | 7.457 | 16.071 | BLAminus | -110.77, 179.22 | 49.98, 83.2 | -97.8, 27.66 | 295.37, 80.49 | -74.55, -21.62 | in-in | in | 8.964 | Saltbr-in | 2.748 | HRD-in | -69.35, -49.91 | 66.48, 13.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.27, 172.69 | APE9-dihe-na | 60.01, 160.49 | APE8-dihe-in | -88.34, 150.2 | APE8-rot-in | 298.89 | APE67-dihe-in | -68.6, -15.9 | -36.65, -52.88 | APE12-dist-in | 12.62 | APE11-dist-in | 10.174 | APE10-dist-in | 6.101 | APE9-dist-in | 3.048 | R21S,K74A,K75A,K76A | None | None | XRAY | 1.84 | 0.196 | 0.234 | A | 328 | 323 | 4 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 7i8a | CMGC_CSNK2A1_HUMAN | CMGC | 8.1e-69 | 238.0 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | DYRK1A | DYR1A_HUMAN | 6A1FA | Q13627 | 134 | 483 | 763.0 | 9OF:807 | Type1 | Active | DFGin | 7.205 | 15.092 | BLAminus | -125.52, 173.04 | 69.56, 79.06 | -100.37, 18.23 | 289.23, 81.85 | -66.74, -28.25 | in-in | in | 8.712 | Saltbr-in | 2.843 | HRD-in | -63.72, -44.37 | 75.39, -2.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.826 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.51, 164.33 | APE9-dihe-na | 78.19, 142.16 | APE8-dihe-in | -71.23, 146.24 | APE8-rot-in | 287.31 | APE67-dihe-in | -64.89, -24.24 | -54.81, -45.1 | APE12-dist-in | 13.001 | APE11-dist-in | 10.937 | APE10-dist-in | 7.397 | APE9-dist-in | 3.189 | None | PTR321 | PTR321 | XRAY | 1.5 | 0.178 | 0.195 | A | 360 | 346 | 4 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 6a1f | CMGC_DYRK1A_HUMAN | CMGC | 8.3e-91 | 310.2 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK2 | DYRK2_HUMAN | 7DH9A | Q92630 | 215 | 538 | 601.0 | H7F:601 | Type1 | Inactive | DFGin | 6.955 | 15.393 | BLAminus | -118.25, -176.44 | 52.33, 72.66 | -86.4, 22.32 | 285.5, 71.17 | -68.46, -16.6 | in-in | in | 9.091 | Saltbr-in | 2.818 | HRD-in | -67.52, -48.86 | 77.78, -1.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.826 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.21, 165.64 | APE9-dihe-na | 77.26, 152.01 | APE8-dihe-in | -71.35, 136.19 | APE8-rot-out | 186.16 | APE67-dihe-in | -56.24, -27.47 | -53.15, -48.91 | APE12-dist-in | 13.085 | APE11-dist-in | 11.935 | APE10-dist-in | 7.588 | APE9-dist-in | 3.308 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.194 | 0.19 | 0.218 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dh9 | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| CMGC | GSK3B | GSK3B_HUMAN | 9PE9A | P49841 | 36 | 382 | 420.0 | A1CIF:900 | Type1 | Inactive | DFGin | 7.072 | 14.229 | BLAminus | -128.7, -179.96 | 59.31, 84.1 | -97.11, 26.91 | 283.64, 74.63 | -73.69, -18.15 | in-in | in | 8.351 | Saltbr-in | 2.725 | HRD-in | -68.62, -45.57 | 65.7, 16.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.925 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -143.94, 165.33 | APE9-dihe-na | 76.34, 152.28 | APE8-dihe-in | -69.82, 130.62 | APE8-rot-out | 176.66 | APE67-dihe-in | -58.68, -26.71 | -39.69, -56.4 | APE12-dist-in | 13.28 | APE11-dist-in | 11.758 | APE10-dist-in | 7.093 | APE9-dist-in | 3.155 | None | PTR216 | PTR216 | XRAY | 2.11 | 0.221 | 0.247 | A | 359 | 332 | 13 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 9pe9 | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 9PE9B | P49841 | 36 | 382 | 420.0 | A1CIF:900 | Type1 | Inactive | DFGin | 7.058 | 14.218 | BLAminus | -128.76, -179.81 | 59.6, 84.42 | -97.78, 27.09 | 283.79, 74.38 | -73.25, -17.71 | in-in | in | 8.353 | Saltbr-in | 2.713 | HRD-in | -68.49, -44.82 | 64.55, 18.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.94 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -144.27, 163.74 | APE9-dihe-na | 77.64, 152.05 | APE8-dihe-in | -69.14, 130.82 | APE8-rot-out | 177.12 | APE67-dihe-in | -58.92, -26.81 | -39.96, -55.88 | APE12-dist-in | 13.36 | APE11-dist-in | 11.824 | APE10-dist-in | 7.161 | APE9-dist-in | 3.172 | None | PTR216 | PTR216 | XRAY | 2.11 | 0.221 | 0.247 | B | 359 | 332 | 13 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 9pe9 | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 4PTEA | P49841 | 36 | 382 | 420.0 | 2WF:501 | Type1 | Active | DFGin | 6.932 | 14.017 | BLAminus | -141.21, 178.04 | 57.99, 89.39 | -100.23, 24.26 | 286.38, 75.9 | -68.08, -19.02 | in-in | in | 8.716 | Saltbr-in | 2.635 | HRD-in | -73.56, -44.45 | 69.11, 4.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.792 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.74, 175.98 | APE9-dihe-na | 75.98, 148.82 | APE8-dihe-in | -103.79, 152.51 | APE8-rot-in | 295.33 | APE67-dihe-inflip | 95.08, -28.26 | -38.95, 126.56 | APE12-dist-in | 12.979 | APE11-dist-in | 10.89 | APE10-dist-in | 5.883 | APE9-dist-in | 3.088 | None | None | None | XRAY | 2.033 | 0.17 | 0.195 | A | 441 | 341 | 6 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 4pte | CMGC_GSK3B_HUMAN | CMGC | 3.7e-70 | 242.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 4PTEB | P49841 | 36 | 385 | 420.0 | 2WF:501 | Type1 | Active | DFGin | 6.918 | 13.937 | BLAminus | -137.07, 179.43 | 58.52, 88.98 | -101.38, 27.88 | 284.28, 76.88 | -69.85, -20.65 | in-in | in | 8.484 | Saltbr-in | 2.685 | HRD-in | -70.9, -46.61 | 73.05, 2.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.887 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -87.76, 178.59 | APE9-dihe-na | 72.73, 147.77 | APE8-dihe-in | -103.48, 150.66 | APE8-rot-in | 296.89 | APE67-dihe-inflip | 94.67, -27.57 | -36.66, 125.81 | APE12-dist-in | 12.935 | APE11-dist-in | 10.88 | APE10-dist-in | 5.877 | APE9-dist-in | 3.154 | None | None | None | XRAY | 2.033 | 0.17 | 0.195 | B | 441 | 347 | 3 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 4pte | CMGC_GSK3B_HUMAN | CMGC | 3.7e-70 | 242.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | MAPK1 | MK01_HUMAN | 5BVDA | P28482 | 9 | 358 | 360.0 | 4VF:60401 | Type1 | None | DFGin | 7.012 | 14.82 | BLAminus | -120.88, -174.96 | 58.49, 83.25 | -99.87, 23.43 | 283.53, 71.8 | -56.85, -34.73 | in-in | in | 9.264 | Saltbr-in | 2.627 | HRD-in | -80.64, -49.81 | 78.16, -6.37 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.72 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 122.19 | APE8-rot-in | 306.38 | APE67-dihe-in | -62.44, -24.22 | -51.26, -49.02 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.9 | 0.172 | 0.207 | A | 361 | 330 | 20 | 0 | 0 | 16 | [[25, 313]] | 1.0 | 5bvd | CMGC_MAPK1_HUMAN | CMGC | 9.2e-86 | 293.7 | 1 | 301 | 301 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 8AO6A | P28482 | 11 | 356 | 360.0 | N9F:406 | Type1 | Inactive | DFGin | 6.771 | 16.337 | BLAminus | -129.81, 177.88 | 71.62, 78.81 | -103.22, 23.44 | 283.23, 73.97 | -64.0, -29.38 | out-in | out | 10.371 | Saltbr-in | 2.597 | HRD-in | -72.45, -50.74 | 72.14, 4.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.785 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -96.92, -36.24 | APE9-dihe-na | -66.98, 156.39 | APE8-dihe-in | -51.35, 125.27 | APE8-rot-in | 311.93 | APE67-dihe-in | -64.42, -17.18 | -56.32, -47.54 | APE12-dist-out | 14.414 | APE11-dist-in | 11.107 | APE10-dist-in | 7.103 | APE9-dist-in | 4.264 | None | None | CME127,CME161 | XRAY | 1.811 | 0.175 | 0.222 | A | 368 | 338 | 0 | 0 | 0 | 0 | [[25, 313]] | 1.0 | 8ao6 | CMGC_MAPK1_HUMAN | CMGC | 9.9e-86 | 293.6 | 1 | 301 | 301 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 8AO9A | P28482 | 11 | 356 | 360.0 | N4F:406 | Type1 | Inactive | DFGin | 6.837 | 16.45 | BLAminus | -129.5, 178.83 | 61.88, 81.37 | -96.97, 21.21 | 286.14, 78.83 | -59.7, -30.7 | out-out | out | 10.301 | Saltbr-out | 3.765 | HRD-in | -72.95, -49.65 | 72.84, 3.98 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.854 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -91.06, -44.4 | APE9-dihe-na | -60.28, 156.59 | APE8-dihe-in | -55.09, 130.24 | APE8-rot-in | 307.62 | APE67-dihe-in | -64.58, -17.09 | -62.44, -44.52 | APE12-dist-out | 14.27 | APE11-dist-in | 10.981 | APE10-dist-in | 6.789 | APE9-dist-in | 4.23 | None | None | CME161 | XRAY | 1.624 | 0.184 | 0.232 | A | 368 | 338 | 2 | 0 | 0 | 0 | [[25, 313]] | 1.0 | 8ao9 | CMGC_MAPK1_HUMAN | CMGC | 9.9e-86 | 293.6 | 1 | 301 | 301 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK10 | MK10_HUMAN | 3CGFA | P53779 | 45 | 400 | 464.0 | JNF:523 | Type1 | Inactive | DFGin | 3.719 | 14.039 | ABAminus | -89.59, -53.32 | -106.99, -179.49 | -117.03, 20.53 | 309.75, 79.33 | 76.52, -162.79 | in-out | in | 9.602 | Saltbr-out | 3.611 | HRD-in | -43.19, -70.09 | 72.17, 4.64 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -63.93, 178.32 | APE9-dihe-na | -126.54, 145.54 | APE8-dihe-in | -86.07, 133.09 | APE8-rot-in | 307.62 | APE67-dihe-in | -51.07, -34.7 | -123.34, -6.64 | APE12-dist-out | 21.335 | APE11-dist-out | 17.893 | APE10-dist-out | 16.615 | APE9-dist-out | 11.474 | None | None | None | XRAY | 3.0 | 0.225 | 0.317 | A | 365 | 346 | 5 | 0 | 0 | 5 | [[64, 359]] | 1.0 | 3cgf | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.1 | 1 | 301 | 301 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 7YL1A | P53779 | 45 | 400 | 464.0 | J6F:501 | Type1 | Inactive | DFGin | 3.995 | 14.06 | ABAminus | -80.16, -27.18 | -141.36, 174.64 | -114.52, 17.98 | 302.24, 85.17 | 76.51, -161.32 | in-in | in | 9.23 | Saltbr-in | 2.755 | HRD-in | -85.09, -59.15 | 76.16, -2.31 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.441 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -89.31, 134.84 | APE9-dihe-na | -84.54, 138.55 | APE8-dihe-in | -77.28, 127.44 | APE8-rot-in | 291.87 | APE67-dihe-in | -54.76, -19.99 | -106.7, -13.11 | APE12-dist-out | 20.721 | APE11-dist-out | 15.877 | APE10-dist-out | 16.196 | APE9-dist-out | 11.273 | None | None | None | XRAY | 2.48 | 0.208 | 0.294 | A | 464 | 352 | 2 | 0 | 0 | 2 | [[64, 359]] | 1.0 | 7yl1 | CMGC_MAPK10_HUMAN | CMGC | 3e-85 | 292.1 | 1 | 301 | 301 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK14 | MK14_HUMAN | 6ZQSA | Q16539 | 4 | 353 | 360.0 | 3FF:400 | Type1 | Inactive | DFGin | 7.131 | 15.007 | BLAminus | -100.05, 172.92 | 58.72, 89.64 | -100.69, 26.63 | 286.71, 76.86 | -66.14, -26.38 | out-out | out | 10.282 | Saltbr-out | 3.92 | HRD-in | -83.97, -53.39 | 74.81, 10.18 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.23, 173.02 | APE9-dihe-na | 73.87, 161.94 | APE8-dihe-in | -91.46, 139.33 | APE8-rot-in | 294.96 | APE67-dihe-in | -66.05, -18.45 | -53.95, -45.87 | APE12-dist-in | 11.599 | APE11-dist-in | 11.174 | APE10-dist-in | 6.771 | APE9-dist-in | 3.046 | None | TPO180,PTR182 | TPO180,PTR182 | XRAY | 1.95 | 0.178 | 0.223 | A | 362 | 350 | 0 | 0 | 0 | 0 | [[24, 308]] | 1.0 | 6zqs | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 5XYYA | Q16539 | 4 | 352 | 360.0 | P0F:401 | Type1.5_Back | Inactive | DFGin | 8.144 | 16.25 | BLBminus | -111.25, 174.05 | 61.59, 81.71 | -109.03, 145.8 | 286.82, 89.51 | 69.26, 21.62 | in-in | in | 8.942 | Saltbr-in | 2.649 | HRD-in | -68.14, -52.86 | 82.9, -10.64 | in-out-out | SNCioo | out-out | ActLoopNT-out | 11.476 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_oooo | APE10-dihe-na | -136.86, 131.59 | APE9-dihe-na | -62.4, -17.36 | APE8-dihe-out | -62.41, -19.09 | APE8-rot-out | 53.75 | APE67-dihe-in | -64.55, -20.22 | -114.48, -18.89 | APE12-dist-out | 21.139 | APE11-dist-out | 22.895 | APE10-dist-out | 17.093 | APE9-dist-out | 11.759 | None | None | None | XRAY | 1.7 | 0.18 | 0.201 | A | 380 | 343 | 6 | 0 | 0 | 0 | [[24, 308]] | 1.0 | 5xyy | CMGC_MAPK14_HUMAN | CMGC | 7e-85 | 290.9 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 2QD9A | Q16539 | 5 | 352 | 360.0 | LGF:361 | Type1 | Inactive | DFGin | 5.134 | 13.797 | BLBplus | -108.86, 148.96 | 74.79, 24.8 | -73.05, 150.79 | 49.54, 82.76 | 82.07, 6.15 | in-in | in | 9.155 | Saltbr-in | 2.557 | HRD-in | -76.06, -55.95 | 78.8, -20.76 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -59.56, -22.52 | 999.0, -59.62 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.7 | 0.252 | 0.282 | A | 366 | 330 | 18 | 0 | 0 | 13 | [[24, 308]] | 1.0 | 2qd9 | CMGC_MAPK14_HUMAN | CMGC | 6.2e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3QUDA | Q16539 | 4 | 354 | 360.0 | N3F:361 | Type1 | Inactive | DFGin | 10.801 | 12.553 | None | -93.66, 153.34 | -68.51, -47.3 | -136.82, 128.38 | 301.98, 103.1 | -95.02, -166.54 | in-in | in | 9.269 | Saltbr-in | 3.555 | HRD-in | -63.42, -58.28 | 80.41, -12.58 | in-out-out | SNCioo | out-out | ActLoopNT-out | 20.801 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, 112.75 | APE9-dihe-na | -76.37, 136.79 | APE8-dihe-out | -65.47, -38.0 | APE8-rot-in | 295.71 | APE67-dihe-in | -57.05, -26.46 | -56.48, -28.08 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 10.762 | APE9-dist-out | 12.652 | None | None | None | XRAY | 2.0 | 0.234 | 0.278 | A | 360 | 345 | 6 | 0 | 0 | 6 | [[24, 308]] | 1.0 | 3qud | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3QUEA | Q16539 | 5 | 353 | 360.0 | 3FF:362 | Type1 | Inactive | DFGin | 10.642 | 12.339 | None | -82.41, 155.86 | -75.27, -54.23 | -130.98, 134.23 | 308.77, 88.25 | -97.08, -170.31 | in-in | in | 8.96 | Saltbr-in | 2.657 | HRD-in | -64.83, -54.13 | 86.66, -27.06 | in-out-out | SNCioo | out-out | ActLoopNT-out | 21.279 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, 66.84 | APE9-dihe-na | -77.78, 135.56 | APE8-dihe-out | -48.89, -54.16 | APE8-rot-in | 280.74 | APE67-dihe-in | -53.38, -25.8 | -51.95, -34.65 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 9.195 | APE9-dist-out | 11.393 | None | None | None | XRAY | 2.7 | 0.23 | 0.311 | A | 360 | 343 | 6 | 0 | 0 | 6 | [[24, 308]] | 1.0 | 3que | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 4R3CA | Q16539 | 4 | 352 | 360.0 | 3GF:402,3GF:403 | Type1,Allosteric | Inactive | DFGin | 4.924 | 13.134 | None | -118.67, 171.2 | 49.4, 42.48 | -86.86, 999.0 | 38.51, 75.43 | 999.0, 999.0 | in-out | in | 9.543 | Saltbr-out | 3.908 | HRD-in | -66.01, -56.32 | 81.1, -14.57 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 103.85 | APE9-dihe-na | -65.1, 130.86 | APE8-dihe-out | -51.86, -39.46 | APE8-rot-in | 289.55 | APE67-dihe-in | -62.53, -25.36 | -48.44, -37.03 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.264 | None | None | CME162 | XRAY | 2.06 | 0.178 | 0.217 | A | 383 | 336 | 13 | 0 | 0 | 13 | [[24, 308]] | 1.0 | 4r3c | CMGC_MAPK14_HUMAN | CMGC | 7.2e-85 | 290.9 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3L8SA | Q16539 | 4 | 353 | 360.0 | BFF:361 | Type1 | Inactive | DFGout | 15.489 | 11.977 | None | -119.54, 162.4 | -99.13, -16.66 | 31.92, 999.0 | 247.73, 144.9 | 999.0, 999.0 | in-in | in | 9.497 | Saltbr-in | 2.817 | HRD-in | -77.51, -50.13 | 90.87, -25.05 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, 107.11 | APE9-dihe-na | -94.83, 118.78 | APE8-dihe-out | -62.16, -3.07 | APE8-rot-out | 173.18 | APE67-dihe-in | -59.13, -22.21 | -95.45, -15.35 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.2 | C119S,C162S,A172C,F327L | None | None | XRAY | 2.35 | 0.242 | 0.307 | A | 360 | 334 | 16 | 0 | 0 | 13 | [[24, 308]] | 1.0 | 3l8s | CMGC_MAPK14_HUMAN | CMGC | 4.4e-84 | 288.3 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3UVRA | Q16539 | 5 | 351 | 360.0 | 06F:361 | Type2 | Inactive | DFGout | 15.561 | 8.524 | None | -148.63, 178.6 | -133.58, 101.18 | -90.01, -1.78 | 195.55, 17.77 | -54.07, 127.45 | in-in | in | 8.211 | Saltbr-in | 2.627 | HRD-in | -62.71, -55.49 | 83.79, -17.62 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -56.89 | APE8-dihe-out | -51.15, -30.26 | APE8-rot-in | 300.71 | APE67-dihe-in | -70.54, -25.21 | -93.95, -15.4 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.621 | None | None | None | XRAY | 2.1 | 0.204 | 0.245 | A | 360 | 331 | 16 | 0 | 0 | 12 | [[24, 308]] | 1.0 | 3uvr | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK8 | MK08_HUMAN | 8PTAA | P45983 | 8 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.923 | 14.477 | ABAminus | -80.58, -61.37 | -103.85, 165.38 | -100.79, 23.99 | 295.77, 91.74 | 73.84, -149.47 | in-in | in | 9.79 | Saltbr-in | 3.126 | HRD-in | -78.59, -61.53 | 62.23, 7.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.47 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iooo | APE10-dihe-na | -130.45, 138.38 | APE9-dihe-na | -101.99, 109.25 | APE8-dihe-in | -118.89, 112.23 | APE8-rot-out | 53.5 | APE67-dihe-in | -51.79, -30.07 | -95.29, -17.54 | APE12-dist-in | 10.569 | APE11-dist-out | 7.033 | APE10-dist-out | 10.183 | APE9-dist-out | 8.598 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | A | 366 | 354 | 2 | 0 | 0 | 2 | [[26, 321]] | 1.0 | 8pta | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| CMGC | MAPK8 | MK08_HUMAN | 8PTAB | P45983 | 7 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.577 | 13.179 | ABAminus | -81.24, -57.35 | -101.3, 158.61 | -105.36, 14.2 | 308.93, 93.28 | 64.59, -148.13 | in-in | in | 9.366 | Saltbr-in | 3.536 | HRD-in | -77.41, -61.25 | 61.49, 9.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -112.33, 168.25 | APE9-dihe-na | -116.9, 36.67 | APE8-dihe-in | -104.63, 91.0 | APE8-rot-out | 52.55 | APE67-dihe-in | -56.88, -29.41 | -95.02, -21.65 | APE12-dist-in | 11.784 | APE11-dist-in | 9.152 | APE10-dist-out | 11.242 | APE9-dist-out | 10.214 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | B | 366 | 352 | 5 | 0 | 0 | 5 | [[26, 321]] | 1.0 | 8pta | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| CMGC | MAPK8 | MK08_HUMAN | 8PTAC | P45983 | 8 | 361 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.826 | 14.088 | ABAminus | -83.97, -56.35 | -97.04, 154.46 | -105.76, 13.83 | 294.99, 32.04 | 63.79, -147.27 | in-out | in | 9.723 | Saltbr-out | 4.528 | HRD-in | -77.01, -60.9 | 63.25, 7.56 | out-out-out | SNCooo | out-out | ActLoopNT-out | 4.611 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -137.59 | APE9-dihe-na | -94.11, 17.64 | APE8-dihe-in | -81.48, 63.35 | APE8-rot-out | 71.39 | APE67-dihe-in | -58.68, -26.77 | -108.19, -24.77 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 12.467 | APE9-dist-out | 10.78 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | C | 366 | 351 | 3 | 0 | 0 | 3 | [[26, 321]] | 1.0 | 8pta | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| CMGC | MAPK9 | MK09_HUMAN | 3E7OA | P45984 | 9 | 361 | 424.0 | 35F:1 | Type1 | Inactive | DFGin | 4.266 | 14.526 | ABAminus | -84.35, -29.35 | -149.55, 177.24 | -106.27, 9.79 | 301.22, 95.14 | 60.95, -143.01 | in-in | in | 9.439 | Saltbr-in | 2.686 | HRD-in | -64.97, -51.12 | 67.58, -6.1 | in-out-out | SNCioo | out-out | ActLoopNT-out | 5.519 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_oooo | APE10-dihe-na | -84.71, -45.82 | APE9-dihe-na | -76.84, -178.43 | APE8-dihe-in | -88.6, 137.99 | APE8-rot-in | 266.04 | APE67-dihe-out | -72.72, -13.34 | -138.1, 64.96 | APE12-dist-out | 20.29 | APE11-dist-out | 15.686 | APE10-dist-out | 19.328 | APE9-dist-out | 14.665 | C177S,C222S,K250A,K251A,K265A,K270A | None | None | XRAY | 2.14 | 0.219 | 0.25 | A | 360 | 342 | 2 | 0 | 0 | 0 | [[26, 321]] | 1.0 | 3e7o | CMGC_MAPK9_HUMAN | CMGC | 2.7e-84 | 288.8 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 9 |
| CMGC | MAPK9 | MK09_HUMAN | 3E7OB | P45984 | 8 | 362 | 424.0 | 35F:2 | Type1 | Inactive | DFGin | 4.276 | 14.318 | ABAminus | -85.32, -37.61 | -133.45, 175.33 | -107.39, 15.94 | 299.45, 88.14 | 90.36, 999.0 | in-in | in | 9.466 | Saltbr-in | 2.801 | HRD-in | -71.07, -57.75 | 72.11, -12.31 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -39.52 | APE8-rot-out | 181.64 | APE67-dihe-in | -65.99, -17.44 | -49.19, -35.22 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | C177S,C222S,K250A,K251A,K265A,K270A | None | None | XRAY | 2.14 | 0.219 | 0.25 | B | 360 | 326 | 19 | 0 | 0 | 16 | [[26, 321]] | 1.0 | 3e7o | CMGC_MAPK9_HUMAN | CMGC | 2.7e-84 | 288.8 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 9 |
| OTHER | CDC7 | CDC7_HUMAN | 6YA8A | O00311 | 38 | 572 | 574.0 | ADP:60601,BEF:60603 | ATPlike,Allosteric | None | DFGin | 6.168 | 14.087 | BLAminus | -118.93, 173.08 | 76.34, 83.66 | -102.33, 21.87 | 291.62, 81.2 | -67.07, -22.7 | in-in | in | 8.709 | Saltbr-in | 2.738 | HRD-in | -65.76, -44.2 | 72.35, -4.4 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.755 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | -83.06, -154.71 | APE8-dihe-in | -48.63, 132.1 | APE8-rot-in | 306.86 | APE67-dihe-in | -66.07, -7.37 | -59.08, -35.16 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.888 | None | None | None | XRAY | 1.79 | 0.167 | 0.197 | A | 359 | 338 | 13 | 0 | 0 | 13 | [[58, 569]] | 1.0 | 6ya8 | OTHER_CDC7_HUMAN | CMGC | 2e-18 | 137.3 | 1 | 161 | 296 | 195 | 196 | 197 | 199 | 201 | 90 | 104 | 108 | 174 | 176 | 175 | 177 | 396 | 383 | 378 | 377 | 376 | 375 | 0 | 0 | 0 | 135 | Cell division cycle 7-related protein kinase |
| OTHER | GAK | GAK_HUMAN | 4C57A | O14976 | 25 | 334 | 1311.0 | FEF:1340 | Type1 | Inactive | DFGin | 5.754 | 14.141 | ABAminus | -112.53, -37.31 | -102.07, 134.52 | -132.21, 22.67 | 297.88, 98.14 | -59.75, -31.11 | in-out | in | 9.993 | Saltbr-out | 4.057 | HRD-in | -62.14, -51.36 | 70.7, -5.09 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.895 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.34, 3.52 | APE9-dihe-na | -124.99, 156.99 | APE8-dihe-in | -84.98, 122.71 | APE8-rot-in | 297.75 | APE67-dihe-in | -71.57, -19.62 | -46.23, -44.89 | APE12-dist-in | 11.779 | APE11-dist-in | 8.573 | APE10-dist-in | 4.33 | APE9-dist-in | 4.07 | None | None | None | XRAY | 2.55 | 0.18 | 0.228 | A | 340 | 310 | 0 | 0 | 0 | 0 | [[40, 313]] | 1.0 | 4c57 | OTHER_GAK_HUMAN | CAMK | 5.3e-44 | 156.7 | 3 | 252 | 250 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | GAK | GAK_HUMAN | 4C57B | O14976 | 27 | 334 | 1311.0 | FEF:1337 | Type1 | Inactive | DFGin | 5.769 | 14.233 | ABAminus | -105.07, -37.59 | -101.51, 133.86 | -130.57, 22.88 | 297.9, 97.48 | -60.27, -26.81 | out-out | out | 10.065 | Saltbr-out | 4.056 | HRD-in | -62.14, -52.49 | 71.3, -9.85 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.891 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.07, 5.67 | APE9-dihe-na | -124.2, 156.66 | APE8-dihe-in | -83.72, 121.96 | APE8-rot-in | 296.0 | APE67-dihe-in | -71.56, -19.42 | -45.7, -45.17 | APE12-dist-in | 11.928 | APE11-dist-in | 8.658 | APE10-dist-in | 4.358 | APE9-dist-in | 4.086 | None | None | None | XRAY | 2.55 | 0.18 | 0.228 | B | 340 | 308 | 0 | 0 | 0 | 0 | [[40, 313]] | 1.0 | 4c57 | OTHER_GAK_HUMAN | CAMK | 5.3e-44 | 156.7 | 3 | 252 | 250 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | GAK | GAK_HUMAN | 4C59A | O14976 | 27 | 333 | 1311.0 | FEF:1334 | Type1 | Inactive | DFGin | 5.815 | 13.68 | ABAminus | -134.62, -10.32 | -105.18, 88.43 | -107.04, 23.92 | 300.54, 105.0 | -81.95, -10.0 | in-in | in | 9.093 | Saltbr-in | 2.855 | HRD-in | -82.36, -54.36 | 82.63, -15.13 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.838 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.8 | 0.205 | 0.262 | A | 340 | 266 | 41 | 0 | 0 | 27 | [[40, 313]] | 1.0 | 4c59 | OTHER_GAK_HUMAN | CAMK | 5.3e-44 | 156.7 | 3 | 252 | 250 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | HASPIN | HASP_HUMAN | 9FLTA | Q8TF76 | 471 | 798 | 798.0 | A1IDF:801 | Type1 | Active | DFGin | 5.178 | 12.218 | BLAminus | -141.02, 178.95 | 59.99, 70.73 | -81.95, 27.03 | 316.78, 141.24 | -69.29, -28.67 | in-in | in | 8.759 | Saltbr-in | 2.463 | HRD-na-N | -66.6, -53.16 | 75.71, 6.9 | in-in-na | SNCiia | in-na | ActLoopNT-in | 2.905 | ActLoopCT-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | APE10-dihe-na | -131.58, 41.34 | APE9-dihe-na | -102.69, 164.5 | APE8-dihe-na | -162.68, -171.46 | APE8-rot-na | 41.52 | APE67-dihe-na | -134.91, 146.64 | 100.36, -24.97 | APE12-dist-na | 9.64 | APE11-dist-na | 13.509 | APE10-dist-na | 17.247 | APE9-dist-na | 13.279 | None | None | None | XRAY | 2.4 | 0.187 | 0.239 | A | 336 | 320 | 8 | 0 | 0 | 0 | [[484, 797]] | 1.0 | 9flt | OTHER_HASPIN_HUMAN | HASP | 1.1e-226 | 756.9 | 1 | 314 | 314 | 686 | 687 | 688 | 690 | 692 | 511 | 535 | 539 | 646 | 648 | 647 | 649 | 741 | 721 | 716 | 715 | 714 | 713 | 712 | 711 | 710 | 604 | Serine/threonine-protein kinase haspin |
| OTHER | TTK | TTK_HUMAN | 4JS8A | P33981 | 515 | 793 | 857.0 | 1PF:801 | Type1 | Inactive | DFGin | 4.246 | 15.018 | ABAminus | -84.57, -49.34 | -133.98, 167.4 | -109.17, 14.51 | 305.07, 151.28 | 67.69, 15.63 | in-out | in | 9.993 | Saltbr-out | 6.699 | HRD-in | -62.96, -52.34 | 70.46, -10.5 | out-out-out | SNCooo | out-out | ActLoopNT-out | 12.036 | ActLoopCT-out | nonTYR | APEdihe_aaini | APEdist_nnoo | APE10-dihe-na | 999.0, 112.01 | APE9-dihe-na | -104.69, -175.56 | APE8-dihe-in | -119.7, 153.55 | APE8-rot-none | 999.0 | APE67-dihe-in | -65.36, -29.34 | -115.57, 0.38 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.198 | APE9-dist-out | 12.111 | None | TPO675,TPO686 | TPO675,TPO686 | XRAY | 1.94 | 0.232 | 0.253 | A | 281 | 261 | 18 | 0 | 0 | 8 | [[525, 791]] | 1.0 | 4js8 | OTHER_TTK_HUMAN | CAMK | 5.6e-54 | 189.1 | 1 | 256 | 256 | 663 | 664 | 665 | 667 | 669 | 553 | 571 | 575 | 644 | 646 | 645 | 647 | 716 | 693 | 688 | 687 | 686 | 685 | 684 | 683 | 682 | 603 | Dual specificity protein kinase TTK |
| OTHER | TTK | TTK_HUMAN | 7CHMA | P33981 | 516 | 794 | 857.0 | FZF:801 | Type1 | Inactive | DFGin | 4.413 | 14.608 | None | -111.88, -71.82 | -63.89, 158.67 | -119.5, 9.1 | 283.45, 179.72 | 82.92, -15.75 | in-in | in | 9.56 | Saltbr-in | 3.396 | HRD-in | -57.59, -51.23 | 60.31, 6.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 12.264 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnoo | APE10-dihe-na | 999.0, -62.47 | APE9-dihe-na | 66.11, 172.68 | APE8-dihe-out | -121.28, -175.85 | APE8-rot-none | 999.0 | APE67-dihe-in | -54.56, -33.62 | -132.81, 0.36 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 19.863 | APE9-dist-out | 12.904 | None | TPO675,TPO686 | TPO675,TPO686 | XRAY | 2.65 | 0.212 | 0.253 | A | 281 | 260 | 19 | 0 | 0 | 8 | [[525, 791]] | 1.0 | 7chm | OTHER_TTK_HUMAN | CAMK | 5.6e-54 | 189.1 | 1 | 256 | 256 | 663 | 664 | 665 | 667 | 669 | 553 | 571 | 575 | 644 | 646 | 645 | 647 | 716 | 693 | 688 | 687 | 686 | 685 | 684 | 683 | 682 | 603 | Dual specificity protein kinase TTK |
| OTHER | ULK1 | ULK1_HUMAN | 4WNOA | O75385 | 8 | 280 | 1050.0 | 3RF:401 | Type1 | Active | DFGin | 6.889 | 14.949 | BLAminus | -117.94, 169.26 | 64.81, 74.6 | -94.14, 20.86 | 282.18, 71.59 | -63.55, -24.11 | in-in | in | 7.662 | Saltbr-in | 2.77 | HRD-in | -82.57, -51.36 | 80.06, -2.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.966 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -155.03, 162.62 | APE9-dihe-na | 120.91, -162.5 | APE8-dihe-in | -119.54, 124.2 | APE8-rot-in | 305.96 | APE67-dihe-in | -67.71, -19.19 | -53.63, -37.75 | APE12-dist-in | 8.214 | APE11-dist-in | 11.212 | APE10-dist-in | 5.675 | APE9-dist-in | 3.309 | E37A,K38A | TPO180 | TPO180 | XRAY | 1.56 | 0.18 | 0.208 | A | 287 | 273 | 0 | 0 | 0 | 0 | [[14, 278]] | 1.0 | 4wno | OTHER_ULK1_HUMAN | ULK | 2.1e-132 | 446.2 | 1 | 256 | 256 | 164 | 165 | 166 | 168 | 170 | 46 | 63 | 67 | 135 | 137 | 136 | 138 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 93 | Serine/threonine-protein kinase ULK1 |
| STE | MAP2K1 | MP2K1_HUMAN | 7UMBC | Q02750 | 41 | 381 | 393.0 | ANP:401,U9F:402 | ATPlike,Type3 | Inactive | DFGin | 6.169 | 13.767 | BLBplus | -162.24, 171.11 | 70.21, 49.7 | -113.95, 160.88 | 44.65, 94.08 | -79.06, 81.13 | out-out | out | 15.559 | Saltbr-out | 15.273 | HRD-in | -66.12, -48.09 | 76.83, -9.86 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.591 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -127.94, 139.36 | APE9-dihe-na | -138.86, -160.81 | APE8-dihe-out | -82.2, -18.64 | APE8-rot-out | 50.9 | APE67-dihe-out | -106.39, 139.13 | -104.8, 110.61 | APE12-dist-out | 16.699 | APE11-dist-out | 19.666 | APE10-dist-out | 21.57 | APE9-dist-out | 14.915 | None | None | None | XRAY | 3.231 | 0.231 | 0.268 | C | 384 | 303 | 38 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 7umb | STE_MAP2K1_HUMAN | STE | 2.3e-97 | 331.4 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K7 | MP2K7_HUMAN | 6YG3A | O14733 | 103 | 400 | 419.0 | 6HF:60510 | Type1 | None | DFGin | 6.195 | 14.549 | BLAminus | -146.55, 178.23 | 54.3, 83.97 | -103.73, 30.03 | 316.89, 91.95 | -57.17, -29.89 | na-na | na | 8.345 | Saltbr-na | 3.36 | HRD-in | -81.36, -52.29 | 76.4, 12.98 | na-in-none | SNCain | in-none | ActLoopNT-in | 2.982 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.05 | 0.191 | 0.235 | A | 307 | 265 | 33 | 0 | 0 | 19 | [[120, 380]] | 1.0 | 6yg3 | STE_MAP2K7_HUMAN | STE | 2.4e-80 | 275.5 | 2 | 257 | 256 | 260 | 261 | 262 | 264 | 266 | 149 | 166 | 170 | 240 | 242 | 241 | 243 | 304 | 287 | 282 | 281 | 280 | 279 | 278 | 277 | 276 | 197 | Dual specificity mitogen-activated protein kinase kinase 7 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4A | Q92918 | 4 | 293 | 833.0 | XXF:60401 | Type1 | Inactive | DFGin | 6.846 | 14.475 | BLAminus | -131.99, 171.23 | 62.34, 86.7 | -92.12, 20.1 | 289.3, 88.42 | -59.7, -48.05 | in-in | in | 9.232 | Saltbr-in | 2.734 | HRD-in | -67.47, -51.18 | 67.4, 4.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.199 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -73.65, -44.57 | APE9-dihe-na | 76.29, -171.23 | APE8-dihe-in | -62.48, 141.12 | APE8-rot-out | 34.25 | APE67-dihe-in | -59.58, -27.68 | -102.29, 0.49 | APE12-dist-out | 20.304 | APE11-dist-out | 21.079 | APE10-dist-out | 21.421 | APE9-dist-out | 27.259 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | A | 331 | 290 | 0 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 8fh4 | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4B | Q92918 | 6 | 302 | 833.0 | XXF:60402 | Type1 | Inactive | DFGin | 6.551 | 14.294 | BLAminus | -141.43, 174.43 | 62.64, 85.33 | -93.2, 13.55 | 285.99, 85.49 | -57.34, -45.75 | in-in | in | 8.939 | Saltbr-in | 2.697 | HRD-in | -67.85, -50.88 | 67.73, 2.48 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.309 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -67.39, -32.57 | APE9-dihe-na | 75.42, -167.37 | APE8-dihe-in | -61.44, 126.8 | APE8-rot-out | 59.49 | APE67-dihe-in | -56.24, -30.95 | -97.05, -0.91 | APE12-dist-out | 19.464 | APE11-dist-out | 20.586 | APE10-dist-out | 21.665 | APE9-dist-out | 28.047 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | B | 331 | 297 | 0 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 8fh4 | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4C | Q92918 | 1 | 292 | 833.0 | XXF:60401 | Type1 | Inactive | DFGin | 6.824 | 14.118 | BLAminus | -136.31, 172.65 | 64.01, 85.1 | -95.02, 19.77 | 288.84, 83.7 | -61.21, -46.39 | in-in | in | 8.967 | Saltbr-in | 2.733 | HRD-in | -69.91, -50.19 | 67.9, 0.86 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.08 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -67.7, -68.85 | APE9-dihe-na | -109.26, -27.15 | APE8-dihe-in | -115.11, 101.44 | APE8-rot-out | 62.11 | APE67-dihe-in | -65.51, -20.35 | -96.81, 16.0 | APE12-dist-out | 19.318 | APE11-dist-out | 20.935 | APE10-dist-out | 23.085 | APE9-dist-out | 28.365 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | C | 331 | 292 | 0 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 8fh4 | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4D | Q92918 | 8 | 292 | 833.0 | XXF:60401 | Type1 | Inactive | DFGin | 6.646 | 14.023 | BLAminus | -135.73, 170.9 | 66.66, 83.46 | -93.58, 25.1 | 289.61, 94.72 | -69.05, -41.66 | in-in | in | 9.022 | Saltbr-in | 2.745 | HRD-in | -74.6, -51.27 | 71.89, -5.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.134 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -170.02 | APE8-dihe-in | -67.05, 131.5 | APE8-rot-out | 192.16 | APE67-dihe-in | -57.98, -30.82 | -102.78, -3.16 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 27.427 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | D | 331 | 276 | 9 | 0 | 0 | 4 | [[17, 274]] | 1.0 | 8fh4 | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 9QT6A | Q92918 | 6 | 292 | 833.0 | A1JAF:301 | Type1 | Inactive | DFGin | 6.463 | 13.765 | None | -60.93, -35.58 | -154.04, -176.9 | -79.86, 1.42 | 63.88, 19.01 | 105.02, -157.57 | out-out | out | 13.28 | Saltbr-out | 10.782 | HRD-in | -74.09, -55.53 | 70.27, 5.38 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.582 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioo | APE10-dihe-na | -59.89, -40.77 | APE9-dihe-na | -92.18, -16.28 | APE8-dihe-in | -142.86, 74.69 | APE8-rot-in | 316.27 | APE67-dihe-in | -56.11, -27.62 | -91.41, -1.8 | APE12-dist-in | 9.809 | APE11-dist-in | 11.134 | APE10-dist-out | 15.153 | APE9-dist-out | 12.698 | T165E,S171E | None | None | XRAY | 1.76 | 0.198 | 0.226 | A | 294 | 285 | 2 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 9qt6 | STE_MAP4K1_HUMAN | STE | 4.1e-92 | 314.1 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8CIJA | Q92918 | 14 | 294 | 833.0 | USF:401 | Type1 | Inactive | DFGout | 11.213 | 7.331 | None | -112.58, 122.54 | -96.1, 115.56 | -121.01, 999.0 | 297.98, 106.95 | 999.0, 999.0 | out-out | out | 13.535 | Saltbr-out | 11.8 | HRD-in | -61.67, -48.53 | 69.18, 2.25 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | -87.98, 122.06 | APE9-dihe-na | 145.78, 142.84 | APE8-dihe-in | -120.8, 116.13 | APE8-rot-in | 320.07 | APE67-dihe-in | -58.16, -27.75 | -31.5, -57.68 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.681 | None | None | None | XRAY | 2.821 | 0.239 | 0.266 | A | 307 | 264 | 17 | 0 | 0 | 12 | [[17, 274]] | 1.0 | 8cij | STE_MAP4K1_HUMAN | STE | 4.8e-92 | 313.9 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K4 | M4K4_HUMAN | 5DI1A | O95819 | 13 | 309 | 1239.0 | 5DF:4000 | Type1 | Inactive | DFGin | 4.26 | 13.366 | BLBplus | -145.12, 159.02 | 72.53, 52.2 | -89.55, 138.32 | 48.51, 95.38 | -80.62, 999.0 | in-out | in | 9.403 | Saltbr-out | 3.985 | HRD-in | -61.2, -47.09 | 79.65, -23.06 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | -102.21, 124.07 | APE9-dihe-na | -81.57, -147.04 | APE8-dihe-in | -74.95, 131.45 | APE8-rot-out | 195.98 | APE67-dihe-in | -46.35, -33.38 | -85.44, -21.52 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.602 | None | None | None | XRAY | 2.9 | 0.2 | 0.249 | A | 310 | 285 | 12 | 0 | 0 | 12 | [[25, 289]] | 1.0 | 5di1 | STE_MAP4K4_HUMAN | STE | 1.3e-102 | 348.4 | 1 | 257 | 257 | 170 | 171 | 172 | 174 | 176 | 54 | 69 | 73 | 150 | 152 | 151 | 153 | 215 | 198 | 193 | 192 | 191 | 190 | 189 | 188 | 187 | 106 | Mitogen-activated protein kinase kinase kinase kinase 4 |
| TKL | ACVR1 | ACVR1_HUMAN | 3MTFA | Q04771 | 203 | 498 | 509.0 | A3F:1 | Type1 | Inactive | DFGin | 7.09 | 13.208 | BLAminus | -126.1, 157.67 | 76.9, 82.69 | -86.05, 21.36 | 306.23, 175.03 | -61.66, -24.97 | in-out | in | 8.331 | Saltbr-out | 4.196 | HRD-in | -82.54, -58.57 | 79.29, -1.49 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.913 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -103.22, 162.67 | APE9-dihe-na | -69.88, 165.81 | APE8-dihe-in | -53.93, 121.99 | APE8-rot-in | 312.82 | APE67-dihe-in | -59.42, -28.32 | -57.34, -37.41 | APE12-dist-in | 10.671 | APE11-dist-out | 6.476 | APE10-dist-out | 9.482 | APE9-dist-in | 4.073 | Q207D | None | None | XRAY | 2.15 | 0.185 | 0.244 | A | 301 | 296 | 0 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 3mtf | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 3MTFB | Q04771 | 202 | 499 | 509.0 | A3F:501 | Type1 | Inactive | DFGin | 7.578 | 13.323 | BLAminus | -114.45, 160.06 | 82.35, 87.49 | -104.83, 25.86 | 291.12, 164.81 | -75.29, -13.54 | in-out | in | 8.5 | Saltbr-out | 4.232 | HRD-in | -82.5, -60.12 | 85.3, -4.39 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.869 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -111.75, 153.3 | APE9-dihe-na | -57.45, 170.81 | APE8-dihe-in | -65.39, 131.64 | APE8-rot-in | 306.28 | APE67-dihe-in | -49.77, -35.33 | -68.1, -43.23 | APE12-dist-in | 10.611 | APE11-dist-out | 6.453 | APE10-dist-out | 9.396 | APE9-dist-in | 4.119 | Q207D | None | None | XRAY | 2.15 | 0.185 | 0.244 | B | 301 | 298 | 0 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 3mtf | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6EIXA | Q04771 | 192 | 503 | 509.0 | A3F:601 | Type1 | Inactive | DFGin | 7.305 | 13.382 | BLAminus | -122.31, 163.89 | 74.01, 85.68 | -98.53, 23.31 | 310.02, 174.96 | -66.89, -23.04 | in-out | in | 9.083 | Saltbr-out | 5.16 | HRD-in | -81.6, -53.66 | 78.97, -2.54 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.023 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -113.45, 165.41 | APE9-dihe-na | -59.94, 163.8 | APE8-dihe-in | -59.76, 126.51 | APE8-rot-in | 307.55 | APE67-dihe-in | -58.05, -30.26 | -58.58, -41.78 | APE12-dist-in | 10.589 | APE11-dist-out | 6.415 | APE10-dist-out | 9.311 | APE9-dist-in | 3.871 | Q207E | None | None | XRAY | 2.3 | 0.191 | 0.249 | A | 340 | 312 | 0 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 6eix | TKL_ACVR1_HUMAN | TKL | 2.9e-85 | 292.0 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 8PODA | Q04771 | 172 | 498 | 509.0 | 7IO:60501,F:60502 | Type1,Allosteric | Inactive | DFGin | 7.181 | 13.248 | BLAminus | -129.23, 172.96 | 64.95, 88.23 | -102.11, 21.22 | 307.17, 178.99 | -69.46, -24.05 | in-out | in | 8.75 | Saltbr-out | 5.24 | HRD-in | -77.46, -49.01 | 73.0, -1.63 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.105 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -104.74, 151.99 | APE9-dihe-na | -69.89, 170.49 | APE8-dihe-in | -67.7, 124.46 | APE8-rot-in | 304.29 | APE67-dihe-in | -63.94, -28.35 | -69.6, -32.91 | APE12-dist-in | 10.74 | APE11-dist-out | 6.542 | APE10-dist-out | 9.732 | APE9-dist-in | 4.647 | None | None | None | XRAY | 2.59 | 0.236 | 0.255 | A | 330 | 320 | 1 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 8pod | TKL_ACVR1_HUMAN | TKL | 2.6e-85 | 292.1 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | BRAF | BRAF_HUMAN | 4YHTA | P15056 | 449 | 719 | 766.0 | 4EF:61002 | Type1 | Inactive | DFGin | 6.44 | 13.919 | BLAminus | -130.91, -175.71 | 59.89, 88.64 | -101.88, 16.92 | 281.61, 73.69 | -54.19, -26.07 | in-in | in | 8.608 | Saltbr-in | 2.731 | HRD-in | -63.73, -42.35 | 62.62, 3.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.881 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -6.83 | APE8-dihe-in | -100.18, 82.06 | APE8-rot-in | 287.27 | APE67-dihe-in | -63.55, -16.06 | -74.16, -21.42 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.11 | I543T,I544N,I551T,L706T,L716T | None | None | XRAY | 3.05 | 0.2 | 0.233 | A | 272 | 256 | 15 | 0 | 0 | 13 | [[457, 716]] | 1.0 | 4yht | TKL_BRAF_HUMAN | TKL | 2.7e-84 | 288.8 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 4YHTB | P15056 | 449 | 720 | 766.0 | 4EF:60802 | Type1 | Inactive | DFGin | 6.405 | 13.921 | BLAminus | -128.69, -172.56 | 54.11, 90.89 | -102.92, 13.66 | 281.86, 71.12 | -49.43, -28.96 | in-in | in | 8.583 | Saltbr-in | 2.701 | HRD-in | -63.82, -42.99 | 62.91, 4.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.864 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -6.59 | APE8-dihe-in | -97.87, 80.96 | APE8-rot-in | 285.28 | APE67-dihe-in | -62.85, -18.47 | -75.71, -20.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.034 | I543T,I544N,I551T,L706T,L716T | None | None | XRAY | 3.05 | 0.2 | 0.233 | B | 272 | 258 | 14 | 0 | 0 | 12 | [[457, 716]] | 1.0 | 4yht | TKL_BRAF_HUMAN | TKL | 2.7e-84 | 288.8 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 3Q96A | P15056 | 449 | 722 | 766.0 | 0NF:1 | Type2 | Inactive | DFGout | 12.887 | 10.676 | BBAminus | -160.13, -172.44 | -118.2, 91.86 | -79.01, 12.35 | 294.04, 84.62 | -59.8, 141.31 | in-in | in | 8.392 | Saltbr-in | 2.855 | HRD-in | -57.31, -47.78 | 82.12, -11.82 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -115.71 | APE8-rot-in | 265.02 | APE67-dihe-in | -61.58, -24.04 | -87.09, -36.86 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 3.1 | 0.233 | 0.288 | A | 282 | 253 | 21 | 0 | 0 | 18 | [[457, 716]] | 1.0 | 3q96 | TKL_BRAF_HUMAN | TKL | 8e-82 | 280.7 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 3Q96B | P15056 | 449 | 720 | 766.0 | 0NF:1 | Type2 | Inactive | DFGout | 12.338 | 11.655 | BBAminus | -159.06, -168.23 | -117.43, 81.54 | -79.68, 17.57 | 296.0, 82.29 | -26.83, 105.54 | in-in | in | 8.586 | Saltbr-in | 3.176 | HRD-in | -76.92, -42.58 | 73.28, -12.97 | in-out-out | SNCioo | out-out | ActLoopNT-out | 18.49 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 159.44 | APE8-dihe-in | -92.55, 126.53 | APE8-rot-in | 290.06 | APE67-dihe-in | -62.77, -20.3 | -102.35, -28.12 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.232 | None | None | None | XRAY | 3.1 | 0.233 | 0.288 | B | 282 | 262 | 10 | 0 | 0 | 10 | [[457, 716]] | 1.0 | 3q96 | TKL_BRAF_HUMAN | TKL | 8e-82 | 280.7 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8A | Q9NWZ3 | 164 | 459 | 460.0 | 4GF:501 | Type1 | Active | DFGin | 6.842 | 14.163 | BLAminus | -130.64, 178.89 | 61.7, 76.88 | -103.53, 25.67 | 310.66, 96.36 | -67.74, -31.55 | in-in | in | 8.778 | Saltbr-in | 3.549 | HRD-in | -57.79, -50.73 | 76.7, -3.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.775 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.21, 150.97 | APE9-dihe-na | 140.01, -173.97 | APE8-dihe-in | -103.61, 115.43 | APE8-rot-in | 309.9 | APE67-dihe-in | -66.28, -16.88 | -42.43, -50.13 | APE12-dist-in | 10.008 | APE11-dist-in | 11.614 | APE10-dist-in | 6.326 | APE9-dist-in | 3.918 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | A | 301 | 287 | 9 | 0 | 0 | 4 | [[183, 456]] | 1.0 | 4yp8 | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8B | Q9NWZ3 | 161 | 459 | 460.0 | 4GF:501 | Type1 | Inactive | DFGin | 6.917 | 14.444 | BLAminus | -129.86, 179.56 | 60.17, 77.95 | -104.22, 26.32 | 310.53, 95.0 | -66.78, -33.18 | in-out | in | 8.685 | Saltbr-out | 3.962 | HRD-in | -57.85, -50.75 | 76.66, -4.15 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.853 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.74, 150.82 | APE9-dihe-na | 140.12, -173.75 | APE8-dihe-in | -103.4, 115.49 | APE8-rot-in | 310.63 | APE67-dihe-in | -65.34, -17.03 | -41.64, -51.23 | APE12-dist-in | 10.045 | APE11-dist-in | 11.581 | APE10-dist-in | 6.319 | APE9-dist-in | 3.905 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | B | 301 | 281 | 18 | 0 | 0 | 6 | [[183, 456]] | 1.0 | 4yp8 | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8C | Q9NWZ3 | 164 | 460 | 460.0 | 4GF:501 | Type1 | Inactive | DFGin | 6.821 | 14.409 | BLAminus | -129.81, 179.51 | 59.35, 79.05 | -103.24, 26.6 | 309.61, 96.69 | -66.38, -34.02 | in-out | in | 8.851 | Saltbr-out | 4.684 | HRD-in | -59.31, -50.52 | 77.45, -5.42 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.789 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.88, 150.51 | APE9-dihe-na | 141.79, -174.18 | APE8-dihe-in | -103.25, 114.63 | APE8-rot-in | 311.45 | APE67-dihe-in | -64.61, -17.76 | -41.38, -51.75 | APE12-dist-in | 10.149 | APE11-dist-in | 11.626 | APE10-dist-in | 6.34 | APE9-dist-in | 3.945 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | C | 301 | 290 | 7 | 0 | 0 | 4 | [[183, 456]] | 1.0 | 4yp8 | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8D | Q9NWZ3 | 164 | 459 | 460.0 | 4GF:501 | Type1 | Inactive | DFGin | 6.854 | 14.319 | BLAminus | -129.62, 178.91 | 61.84, 77.53 | -103.67, 26.43 | 310.15, 95.74 | -66.28, -34.21 | in-out | in | 8.915 | Saltbr-out | 3.802 | HRD-in | -59.75, -49.91 | 75.93, -3.95 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.79 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.59, 153.02 | APE9-dihe-na | 138.42, -174.86 | APE8-dihe-in | -103.4, 114.55 | APE8-rot-in | 310.75 | APE67-dihe-in | -64.11, -17.03 | -41.21, -51.68 | APE12-dist-in | 10.015 | APE11-dist-in | 11.585 | APE10-dist-in | 6.327 | APE9-dist-in | 3.922 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | D | 301 | 288 | 8 | 0 | 0 | 4 | [[183, 456]] | 1.0 | 4yp8 | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYA | Q9NWZ3 | 163 | 458 | 460.0 | EXF:501 | Type1 | Inactive | DFGin | 6.997 | 14.049 | BLAminus | -130.85, 177.02 | 62.25, 85.69 | -105.57, 13.21 | 307.3, 97.03 | -58.17, -30.36 | in-out | in | 8.929 | Saltbr-out | 5.362 | HRD-in | -67.47, -54.1 | 77.02, 0.48 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.819 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.95, 147.66 | APE9-dihe-na | 135.07, -175.38 | APE8-dihe-in | -106.14, 112.07 | APE8-rot-in | 312.29 | APE67-dihe-in | -59.29, -20.88 | -52.35, -43.4 | APE12-dist-in | 10.191 | APE11-dist-in | 11.704 | APE10-dist-in | 6.439 | APE9-dist-in | 4.357 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | A | 305 | 294 | 2 | 0 | 0 | 2 | [[183, 456]] | 1.0 | 6lxy | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYB | Q9NWZ3 | 163 | 459 | 460.0 | EXF:502 | Type1 | None | DFGin | 6.973 | 14.137 | BLAminus | -129.45, 177.84 | 61.74, 86.54 | -106.07, 12.43 | 306.08, 97.48 | -57.61, -29.04 | in-none | in | 9.098 | Saltbr-none | 999.0 | HRD-in | -68.65, -53.21 | 75.68, 1.0 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.807 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.47, 149.33 | APE9-dihe-na | 135.3, -175.41 | APE8-dihe-in | -105.49, 112.4 | APE8-rot-in | 312.11 | APE67-dihe-in | -59.55, -21.17 | -51.5, -42.55 | APE12-dist-in | 10.189 | APE11-dist-in | 11.686 | APE10-dist-in | 6.444 | APE9-dist-in | 4.332 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | B | 305 | 297 | 0 | 0 | 0 | 0 | [[183, 456]] | 1.0 | 6lxy | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYD | Q9NWZ3 | 162 | 459 | 460.0 | EXF:502 | Type1 | Inactive | DFGin | 7.002 | 14.116 | BLAminus | -130.62, 177.55 | 62.4, 85.91 | -106.35, 12.8 | 307.19, 98.16 | -58.64, -30.18 | in-out | in | 8.943 | Saltbr-out | 5.354 | HRD-in | -67.38, -53.42 | 77.14, -1.48 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.786 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.01, 149.8 | APE9-dihe-na | 134.89, -175.28 | APE8-dihe-in | -104.95, 111.45 | APE8-rot-in | 311.34 | APE67-dihe-in | -58.57, -21.72 | -44.58, -48.25 | APE12-dist-in | 10.314 | APE11-dist-in | 11.954 | APE10-dist-in | 6.613 | APE9-dist-in | 4.254 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | D | 305 | 293 | 5 | 0 | 0 | 5 | [[183, 456]] | 1.0 | 6lxy | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYE | Q9NWZ3 | 164 | 458 | 460.0 | EXF:502 | Type1 | Inactive | DFGin | 6.954 | 14.159 | BLAminus | -130.3, 176.57 | 62.62, 85.73 | -105.89, 13.23 | 306.79, 97.59 | -58.45, -29.69 | in-out | in | 8.931 | Saltbr-out | 5.391 | HRD-in | -66.96, -52.89 | 76.03, -0.37 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.795 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.25, 150.73 | APE9-dihe-na | 134.77, -173.9 | APE8-dihe-in | -105.72, 111.9 | APE8-rot-in | 311.85 | APE67-dihe-in | -56.93, -22.86 | -45.56, -48.25 | APE12-dist-in | 10.309 | APE11-dist-in | 11.905 | APE10-dist-in | 6.607 | APE9-dist-in | 4.292 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | E | 305 | 288 | 7 | 0 | 0 | 7 | [[183, 456]] | 1.0 | 6lxy | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | MAP3K12 | M3K12_HUMAN | 5CEQA | Q12852 | 117 | 398 | 859.0 | 50F:4000 | Type1 | Inactive | DFGin | 6.285 | 14.143 | BLBplus | -139.34, 175.24 | 65.23, 33.46 | -103.17, 163.52 | 57.07, 90.2 | 71.88, 999.0 | na-na | na | 13.937 | Saltbr-na | 13.245 | HRD-in | -61.44, -57.14 | 79.98, -14.5 | na-none-out | SNCano | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | -71.43, -48.01 | APE9-dihe-na | -72.5, -0.08 | APE8-dihe-out | -118.56, -4.99 | APE8-rot-out | 184.08 | APE67-dihe-in | -55.04, -30.89 | -63.03, -27.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.132 | None | None | None | XRAY | 1.911 | 0.171 | 0.218 | A | 300 | 269 | 13 | 0 | 0 | 13 | [[118, 372]] | 1.0 | 5ceq | TKL_MAP3K12_HUMAN | MAP3K123 | 1.5e-137 | 462.8 | 1 | 254 | 254 | 253 | 254 | 255 | 257 | 259 | 152 | 161 | 165 | 233 | 235 | 234 | 236 | 292 | 280 | 275 | 274 | 273 | 272 | 271 | 270 | 269 | 191 | Mitogen-activated protein kinase kinase kinase 12 |
| TKL | MAP3K7 | M3K7_HUMAN | 5J9LA | O43318 | 31 | 496 | 606.0 | 6HF:60501 | Type1 | Inactive | DFGout | 12.964 | 7.575 | None | -126.7, 106.14 | -55.49, -39.75 | -39.65, 999.0 | 105.32, 93.88 | 999.0, 999.0 | in-out | in | 9.619 | Saltbr-out | 4.662 | HRD-in | -64.53, -55.8 | 74.12, -2.79 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 124.52 | APE8-dihe-out | -91.5, 21.0 | APE8-rot-in | 299.75 | APE67-dihe-in | -63.93, -32.31 | -64.12, -36.48 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.7 | None | None | None | XRAY | 2.752 | 0.214 | 0.243 | A | 307 | 253 | 20 | 0 | 0 | 14 | [[36, 286]] | 1.0 | 5j9l | TKL_MAP3K7_HUMAN | TKL | 3.7e-74 | 255.5 | 2 | 266 | 265 | 174 | 175 | 176 | 178 | 180 | 63 | 77 | 81 | 153 | 155 | 154 | 156 | 211 | 199 | 194 | 193 | 192 | 191 | 190 | 189 | 188 | 105 | Mitogen-activated protein kinase kinase kinase 7 |
| TKL | RIPK1 | RIPK1_HUMAN | 7FCZA | Q13546 | 10 | 294 | 671.0 | 3IF:301 | Type3 | Inactive | DFGout | 13.865 | 10.379 | BBAminus | -121.61, 171.92 | -133.79, 66.08 | -70.41, -22.3 | 302.99, 177.02 | -85.6, 3.29 | out-out | out | 15.002 | Saltbr-out | 12.85 | HRD-in | -69.8, -48.63 | 73.26, -13.72 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.074 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 77.72 | APE8-dihe-in | -67.19, 127.43 | APE8-rot-in | 294.95 | APE67-dihe-in | -62.33, -29.47 | -101.92, 1.17 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.476 | C34A,C127A,C233A,C240A | None | None | XRAY | 2.21 | 0.236 | 0.257 | A | 297 | 248 | 37 | 0 | 0 | 18 | [[17, 287]] | 1.0 | 7fcz | TKL_RIPK1_HUMAN | TKL | 1.3e-72 | 250.5 | 6 | 265 | 260 | 155 | 156 | 157 | 159 | 161 | 45 | 63 | 67 | 135 | 137 | 136 | 138 | 210 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 93 | Receptor-interacting serine/threonine-protein kinase 1 |
| TKL | RIPK1 | RIPK1_HUMAN | 7FCZB | Q13546 | 7 | 294 | 671.0 | 3IF:301 | Type3 | Inactive | DFGout | 13.913 | 10.028 | BBAminus | -118.21, 174.22 | -136.13, 64.53 | -68.29, -24.74 | 303.09, 178.58 | -83.09, -0.43 | out-out | out | 14.189 | Saltbr-out | 12.575 | HRD-in | -73.47, -53.47 | 80.61, -17.48 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.139 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 101.37 | APE8-dihe-in | -64.4, 143.44 | APE8-rot-out | 179.16 | APE67-dihe-in | -62.08, -29.26 | -100.06, -1.15 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.634 | C34A,C127A,C233A,C240A | None | None | XRAY | 2.21 | 0.236 | 0.257 | B | 297 | 263 | 25 | 0 | 0 | 17 | [[17, 287]] | 1.0 | 7fcz | TKL_RIPK1_HUMAN | TKL | 1.3e-72 | 250.5 | 6 | 265 | 260 | 155 | 156 | 157 | 159 | 161 | 45 | 63 | 67 | 135 | 137 | 136 | 138 | 210 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 93 | Receptor-interacting serine/threonine-protein kinase 1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 2WOUA | P36897 | 200 | 496 | 503.0 | ZZF:61500 | Type1 | Active | DFGin | 6.124 | 13.039 | BLAminus | -133.49, -169.53 | 51.05, 62.4 | -92.04, 13.34 | 298.31, 178.69 | -62.77, -27.98 | in-in | in | 7.586 | Saltbr-in | 2.752 | HRD-in | -65.52, -56.03 | 81.95, -3.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.039 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.77, -22.31 | APE9-dihe-na | -79.77, -172.15 | APE8-dihe-in | -73.94, 125.36 | APE8-rot-in | 306.35 | APE67-dihe-in | -52.11, -29.79 | -56.64, -45.19 | APE12-dist-in | 13.078 | APE11-dist-in | 11.935 | APE10-dist-in | 6.041 | APE9-dist-in | 3.629 | None | None | None | XRAY | 2.3 | 0.229 | 0.302 | A | 306 | 297 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2wou | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAA | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 5.904 | 13.047 | BLAminus | -165.74, 163.41 | 74.29, 54.12 | -79.67, 24.05 | 317.06, 176.62 | -56.68, -51.28 | in-in | in | 8.001 | Saltbr-in | 2.936 | HRD-in | -45.11, -27.8 | 52.25, 11.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.111 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.43, -171.19 | APE9-dihe-na | 80.03, 171.79 | APE8-dihe-in | -67.98, 121.11 | APE8-rot-in | 302.91 | APE67-dihe-in | -99.71, -73.49 | -46.09, -5.99 | APE12-dist-in | 11.624 | APE11-dist-in | 11.967 | APE10-dist-in | 6.015 | APE9-dist-in | 4.061 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | A | 342 | 328 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAB | P36897 | 171 | 501 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.017 | 13.306 | BLAminus | -136.45, -176.24 | 60.04, 54.86 | -81.47, 12.98 | 307.95, 5.19 | -52.57, -45.29 | in-in | in | 8.1 | Saltbr-in | 3.037 | HRD-in | -75.89, -39.75 | 60.74, 14.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.115 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.32, 175.24 | APE9-dihe-na | 101.52, 166.7 | APE8-dihe-in | -70.87, 127.35 | APE8-rot-in | 315.28 | APE67-dihe-in | -36.34, -44.33 | -43.95, -69.54 | APE12-dist-in | 11.94 | APE11-dist-in | 12.0 | APE10-dist-in | 6.373 | APE9-dist-in | 4.084 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAC | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Inactive | DFGin | 6.142 | 13.141 | BLAminus | -126.27, 176.42 | 50.71, 78.49 | -102.58, 30.06 | 320.3, 19.34 | -66.31, -17.95 | in-in | in | 7.99 | Saltbr-in | 2.662 | HRD-in | -67.56, -21.99 | 46.1, 19.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.947 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -120.66, 131.05 | APE9-dihe-na | 148.7, 175.0 | APE8-dihe-in | -102.93, 87.73 | APE8-rot-in | 305.5 | APE67-dihe-out | -28.83, -55.82 | 5.18, -84.04 | APE12-dist-in | 11.481 | APE11-dist-in | 12.149 | APE10-dist-in | 6.247 | APE9-dist-in | 4.208 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAD | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.26 | 13.168 | BLAminus | -151.5, 176.63 | 62.94, 64.2 | -90.99, 26.98 | 302.19, 4.38 | -66.56, -19.34 | in-in | in | 7.809 | Saltbr-in | 2.745 | HRD-in | -63.44, -55.82 | 78.14, 1.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.86, 174.28 | APE9-dihe-na | 87.09, 173.14 | APE8-dihe-in | -66.87, 116.28 | APE8-rot-in | 325.42 | APE67-dihe-in | -60.47, -38.15 | -48.63, -36.35 | APE12-dist-in | 11.714 | APE11-dist-in | 11.894 | APE10-dist-in | 6.37 | APE9-dist-in | 4.229 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAE | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.355 | 13.366 | BLAminus | -131.48, -168.05 | 37.37, 86.28 | -107.7, 26.02 | 296.92, 176.17 | -65.92, -19.56 | in-in | in | 7.781 | Saltbr-in | 3.095 | HRD-in | -66.77, -57.93 | 79.95, 12.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.85 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.13, 169.87 | APE9-dihe-na | 90.72, 172.5 | APE8-dihe-in | -64.72, 129.04 | APE8-rot-in | 310.98 | APE67-dihe-in | -56.46, -40.64 | -59.57, -42.14 | APE12-dist-in | 11.99 | APE11-dist-in | 12.056 | APE10-dist-in | 6.57 | APE9-dist-in | 3.982 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR2 | TGFR2_HUMAN | 7DV6A | P37173 | 240 | 543 | 567.0 | HJF:9000 | Type1 | Active | DFGin | 7.131 | 13.432 | BLAminus | -156.15, -164.95 | 57.9, 60.45 | -93.44, 15.51 | 294.56, 110.64 | -56.6, -36.89 | in-in | in | 7.444 | Saltbr-in | 2.659 | HRD-in | -60.78, -51.79 | 74.77, -4.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.86 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.14, 141.57 | APE9-dihe-na | 113.33, -173.4 | APE8-dihe-in | -82.04, 128.94 | APE8-rot-in | 303.35 | APE67-dihe-in | -55.96, -36.36 | -60.86, -38.17 | APE12-dist-in | 11.508 | APE11-dist-in | 11.89 | APE10-dist-in | 6.046 | APE9-dist-in | 3.912 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.39 | 0.163 | 0.224 | A | 323 | 304 | 0 | 0 | 0 | 0 | [[244, 540]] | 1.0 | 7dv6 | TKL_TGFBR2_HUMAN | TKL | 2.1e-77 | 266.2 | 2 | 266 | 265 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TYR | ALK | ALK_HUMAN | 4CCUA | Q9UM73 | 1093 | 1402 | 1620.0 | AWF:1500 | Type1 | Inactive | DFGin | 6.02 | 14.623 | ABAminus | -118.73, -9.8 | -132.17, 139.04 | -133.56, 37.48 | 295.42, 86.35 | -74.53, -27.89 | in-out | in | 8.277 | Saltbr-out | 4.689 | HRD-in | -77.94, -47.73 | 82.62, -10.67 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.803 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.98, -27.23 | APE9-dihe-in | -56.62, 135.11 | APE8-dihe-in | -75.38, 65.75 | APE8-rot-na | 29.29 | APE67-dihe-in | -70.29, -14.23 | -60.1, -29.45 | APE12-dist-na | 14.525 | APE11-dist-na | 15.17 | APE10-dist-na | 10.028 | APE9-dist-in | 7.796 | None | None | None | XRAY | 2.0 | 0.202 | 0.233 | A | 327 | 293 | 17 | 0 | 0 | 6 | [[1116, 1385]] | 1.0 | 4ccu | TYR_ALK_HUMAN | TYR | 1.4e-90 | 309.1 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | ALK | ALK_HUMAN | 4FNZA | Q9UM73 | 1093 | 1402 | 1620.0 | NZF:1501 | Type1 | Inactive | DFGin | 5.291 | 12.8 | ABAminus | -135.46, 12.02 | -152.76, 153.63 | -83.97, -38.55 | 283.31, 122.35 | 73.66, 999.0 | in-in | in | 8.5 | Saltbr-in | 2.812 | HRD-in | -72.66, -49.3 | 78.9, -9.45 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -97.65, -24.93 | APE9-dihe-in | -50.61, 132.71 | APE8-dihe-in | -79.34, 69.48 | APE8-rot-na | 27.73 | APE67-dihe-in | -74.42, -13.21 | -56.44, -36.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.83 | C1097S | None | None | XRAY | 2.6 | 0.202 | 0.261 | A | 327 | 287 | 23 | 0 | 0 | 15 | [[1116, 1385]] | 1.0 | 4fnz | TYR_ALK_HUMAN | TYR | 1.4e-90 | 309.1 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | ALK | ALK_HUMAN | 4DCEA | Q9UM73 | 1093 | 1402 | 1620.0 | 0JF:1501 | Type1 | Inactive | DFGin | 5.63 | 13.823 | None | -137.27, 16.47 | -161.52, 152.14 | -94.73, 164.26 | 291.72, 122.64 | -76.17, 999.0 | in-in | in | 8.482 | Saltbr-in | 2.883 | HRD-in | -75.4, -48.78 | 85.77, -10.33 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -96.83, -20.84 | APE9-dihe-in | -55.51, 136.7 | APE8-dihe-in | -77.28, 70.08 | APE8-rot-na | 28.6 | APE67-dihe-in | -68.31, -8.92 | -56.77, -41.62 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.974 | C1097S | None | None | XRAY | 2.03 | 0.211 | 0.256 | A | 333 | 288 | 22 | 0 | 0 | 14 | [[1116, 1385]] | 1.0 | 4dce | TYR_ALK_HUMAN | TYR | 1.5e-90 | 309.0 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | ALK | ALK_HUMAN | 4DCEB | Q9UM73 | 1094 | 1402 | 1620.0 | 0JF:1501 | Type1 | Inactive | DFGin | 5.747 | 13.628 | None | -141.04, 18.73 | -165.26, 150.02 | -96.5, 167.37 | 286.77, 120.17 | -70.38, 999.0 | in-in | in | 8.563 | Saltbr-in | 2.99 | HRD-in | -72.56, -48.26 | 83.87, -14.3 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -96.41, -12.56 | APE9-dihe-in | -59.98, 136.0 | APE8-dihe-in | -80.48, 64.18 | APE8-rot-na | 31.8 | APE67-dihe-in | -66.1, -14.3 | -52.07, -41.53 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.713 | C1097S | None | None | XRAY | 2.03 | 0.211 | 0.256 | B | 333 | 284 | 25 | 0 | 0 | 15 | [[1116, 1385]] | 1.0 | 4dce | TYR_ALK_HUMAN | TYR | 1.5e-90 | 309.0 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | BTK | BTK_HUMAN | 5FBNC | Q06187 | 395 | 658 | 659.0 | 5WF:701,5WE:702 | Type1.5_Front,Allosteric | Inactive | DFGin | 6.234 | 13.485 | BLBplus | -138.97, 172.93 | 64.41, 21.2 | -64.91, 134.85 | 43.34, 89.93 | 78.28, -17.1 | out-out | out | 15.007 | Saltbr-out | 15.714 | HRD-in | -67.81, -54.89 | 86.66, -24.42 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.194 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | 143.31, -31.01 | APE9-dihe-in | -63.12, 135.49 | APE8-dihe-in | -76.38, 65.1 | APE8-rot-na | 32.35 | APE67-dihe-in | -72.98, -10.12 | -50.46, -47.16 | APE12-dist-na | 999.0 | APE11-dist-na | 17.831 | APE10-dist-na | 12.608 | APE9-dist-out | 8.181 | None | None | None | XRAY | 1.8 | 0.182 | 0.226 | C | 271 | 256 | 8 | 0 | 0 | 8 | [[402, 653]] | 1.0 | 5fbn | TYR_BTK_HUMAN | TYR | 6e-93 | 316.8 | 1 | 258 | 258 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 5FBND | Q06187 | 394 | 658 | 659.0 | 5WF:702,5WE:703,5WE:704,5WE:705 | Type1.5_Front,Allosteric,Allosteric,Allosteric | Inactive | DFGin | 6.25 | 13.472 | BLBplus | -137.76, 172.64 | 65.66, 19.16 | -62.24, 135.48 | 45.56, 88.91 | 74.32, -16.76 | out-out | out | 15.056 | Saltbr-out | 15.752 | HRD-in | -65.32, -54.88 | 86.04, -26.38 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.195 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 136.18 | APE8-dihe-in | -78.24, 64.6 | APE8-rot-na | 31.95 | APE67-dihe-in | -74.36, -8.3 | -50.81, -46.27 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.898 | None | None | None | XRAY | 1.8 | 0.182 | 0.226 | D | 271 | 255 | 10 | 0 | 0 | 10 | [[402, 653]] | 1.0 | 5fbn | TYR_BTK_HUMAN | TYR | 6e-93 | 316.8 | 1 | 258 | 258 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | DDR1 | DDR1_HUMAN | 5SAUA | Q08345 | 604 | 912 | 913.0 | 1IF:61000 | Type2 | Inactive | DFGout | 12.628 | 9.672 | BBAminus | -137.39, -170.54 | -153.95, 108.1 | -100.48, 5.9 | 289.81, 101.12 | 83.39, -174.73 | in-in | in | 8.355 | Saltbr-in | 2.869 | HRD-in | -71.66, -48.67 | 82.15, -10.52 | in-out-in | SNCioi | out-in | ActLoopNT-out | 18.139 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.56, 139.94 | APE9-dihe-in | -129.66, 123.98 | APE8-dihe-in | -80.56, 70.77 | APE8-rot-na | 35.49 | APE67-dihe-in | -73.85, -9.33 | -63.13, -31.85 | APE12-dist-na | 13.331 | APE11-dist-na | 10.312 | APE10-dist-na | 5.884 | APE9-dist-in | 7.555 | None | None | None | XRAY | 1.8 | 0.201 | 0.231 | A | 321 | 287 | 16 | 0 | 0 | 0 | [[610, 907]] | 1.0 | 5sau | TYR_DDR1_HUMAN | TYR | 1.4e-92 | 315.7 | 1 | 260 | 260 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | EPHA2 | EPHA2_HUMAN | 8BOCA | P29317 | 605 | 888 | 976.0 | QUF:1001 | Type2 | Inactive | DFGout | 13.583 | 10.813 | BBAminus | -139.62, -179.28 | -151.24, 106.28 | -78.98, -6.2 | 302.64, 171.21 | 84.05, 5.79 | in-in | in | 8.869 | Saltbr-in | 3.501 | HRD-in | -70.68, -54.7 | 83.35, -19.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 12.248 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.53, 160.37 | APE9-dihe-in | -116.01, 148.45 | APE8-dihe-in | -79.02, 97.78 | APE8-rot-na | 34.23 | APE67-dihe-in | -77.84, -8.8 | -56.96, -40.4 | APE12-dist-na | 12.844 | APE11-dist-na | 9.325 | APE10-dist-na | 7.892 | APE9-dist-in | 5.837 | None | None | None | XRAY | 1.9 | 0.248 | 0.286 | A | 306 | 271 | 13 | 0 | 0 | 0 | [[613, 873]] | 1.0 | 8boc | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2 | 261 | 260 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHB4 | EPHB4_HUMAN | 2X9FA | P54760 | 608 | 888 | 987.0 | X9F:1889 | Type1 | Inactive | DFGin | 6.208 | 14.33 | BLBminus | -134.1, -172.08 | 65.01, 71.96 | -106.66, 162.22 | 301.36, 107.12 | 163.16, 158.85 | in-in | in | 7.543 | Saltbr-in | 2.703 | HRD-in | -73.92, -48.13 | 77.71, -16.54 | in-out-in | SNCioi | out-in | ActLoopNT-out | 9.79 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -102.56, 149.08 | APE9-dihe-in | -55.67, 129.32 | APE8-dihe-in | -83.14, 89.74 | APE8-rot-na | 29.6 | APE67-dihe-in | -62.34, -22.56 | -52.45, -48.78 | APE12-dist-na | 8.363 | APE11-dist-na | 11.417 | APE10-dist-na | 15.416 | APE9-dist-in | 6.34 | Y774E | None | None | XRAY | 1.75 | 0.159 | 0.194 | A | 302 | 265 | 16 | 0 | 0 | 13 | [[615, 876]] | 1.0 | 2x9f | TYR_EPHB4_HUMAN | TYR | 3.9e-104 | 353.5 | 2 | 261 | 260 | 757 | 758 | 759 | 761 | 763 | 647 | 664 | 668 | 737 | 739 | 738 | 740 | 802 | 790 | 785 | 784 | 783 | 782 | 781 | 780 | 779 | 694 | Ephrin type-B receptor 4 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIA | P11362 | 458 | 764 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.058 | 13.436 | BLAplus | -111.91, 163.26 | 62.65, 26.85 | -80.22, -19.74 | 58.59, 88.0 | -94.12, 4.52 | in-in | in | 8.251 | Saltbr-in | 2.888 | HRD-in | -74.14, -50.3 | 78.02, -11.1 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.511 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -88.77, 149.44 | APE9-dihe-in | -108.01, 98.39 | APE8-dihe-out | -63.46, -15.87 | APE8-rot-na | 3.35 | APE67-dihe-in | -71.69, -10.38 | -55.45, -26.93 | APE12-dist-na | 17.216 | APE11-dist-na | 19.672 | APE10-dist-na | 16.685 | APE9-dist-out | 11.083 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | A | 310 | 307 | 0 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 9uhi | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIB | P11362 | 458 | 763 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.213 | 12.738 | BLAplus | -108.15, 164.77 | 66.41, 24.28 | -84.34, -17.16 | 58.96, 83.83 | -89.87, -8.4 | in-in | in | 7.768 | Saltbr-in | 3.449 | HRD-in | -77.39, -52.67 | 76.89, -15.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -74.45, 132.66 | APE9-dihe-in | -102.74, 93.19 | APE8-dihe-out | -60.68, -21.29 | APE8-rot-na | 332.28 | APE67-dihe-in | -72.11, -2.38 | -56.87, -27.58 | APE12-dist-na | 17.352 | APE11-dist-na | 20.682 | APE10-dist-na | 16.965 | APE9-dist-out | 11.364 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | B | 310 | 286 | 20 | 0 | 0 | 7 | [[478, 756]] | 1.0 | 9uhi | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FA | P11362 | 464 | 765 | 822.0 | C4F:1 | Type1.5_Back | Inactive | DFGin | 5.114 | 13.318 | BLAplus | -110.44, 159.78 | 58.59, 34.58 | -81.02, -11.31 | 51.22, 81.2 | -119.48, 23.64 | in-out | in | 7.866 | Saltbr-out | 4.632 | HRD-in | -67.82, -57.48 | 84.79, -17.47 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.069 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.31, 173.6 | APE9-dihe-in | -111.71, 110.92 | APE8-dihe-out | -49.57, -28.9 | APE8-rot-na | 335.93 | APE67-dihe-in | -76.49, -6.67 | -57.78, -16.15 | APE12-dist-na | 19.292 | APE11-dist-na | 21.121 | APE10-dist-na | 19.395 | APE9-dist-out | 11.757 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | A | 302 | 290 | 12 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 3c4f | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FB | P11362 | 464 | 765 | 822.0 | C4F:2 | Type1.5_Back | Inactive | DFGin | 5.186 | 13.096 | BLAplus | -113.87, 161.2 | 54.21, 44.76 | -88.95, -14.38 | 49.14, 89.01 | -114.94, 24.21 | in-in | in | 7.831 | Saltbr-in | 3.248 | HRD-in | -69.91, -54.09 | 86.4, -33.67 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.934 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.54, 164.12 | APE9-dihe-in | -103.97, 111.75 | APE8-dihe-out | -49.46, -30.24 | APE8-rot-na | 330.07 | APE67-dihe-in | -74.8, -7.14 | -56.82, -17.81 | APE12-dist-na | 19.37 | APE11-dist-na | 21.296 | APE10-dist-na | 19.671 | APE9-dist-out | 11.643 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | B | 302 | 290 | 12 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 3c4f | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5EW8A | P11362 | 464 | 765 | 822.0 | 5SF:803 | Type1.5_Back | Inactive | DFGin | 4.948 | 13.265 | BLAplus | -106.94, 161.6 | 53.73, 34.99 | -75.93, -13.84 | 56.0, 83.89 | -112.21, 7.75 | in-in | in | 7.954 | Saltbr-in | 2.801 | HRD-in | -68.23, -51.53 | 79.48, -14.26 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.067 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.87, 162.8 | APE9-dihe-in | -100.01, 112.78 | APE8-dihe-out | -57.6, -21.18 | APE8-rot-na | 333.77 | APE67-dihe-in | -70.4, -6.07 | -56.33, -25.26 | APE12-dist-na | 19.37 | APE11-dist-na | 20.743 | APE10-dist-na | 19.216 | APE9-dist-out | 11.882 | None | None | None | XRAY | 1.63 | 0.186 | 0.206 | A | 309 | 291 | 11 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 5ew8 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5EW8B | P11362 | 461 | 765 | 822.0 | 5SF:802 | Type1.5_Back | Inactive | DFGin | 5.002 | 13.124 | BLAplus | -109.75, 160.16 | 55.05, 34.73 | -78.35, -12.87 | 54.65, 85.31 | -106.64, 12.94 | in-in | in | 7.88 | Saltbr-in | 2.807 | HRD-in | -67.52, -52.32 | 78.89, -12.97 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.38 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.81, 162.42 | APE9-dihe-in | -99.2, 111.94 | APE8-dihe-out | -57.42, -21.49 | APE8-rot-na | 334.53 | APE67-dihe-in | -69.99, -6.88 | -56.65, -24.13 | APE12-dist-na | 19.902 | APE11-dist-na | 21.169 | APE10-dist-na | 19.654 | APE9-dist-out | 11.767 | None | None | None | XRAY | 1.63 | 0.186 | 0.206 | B | 309 | 290 | 15 | 0 | 0 | 2 | [[478, 756]] | 1.0 | 5ew8 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7WCLA | P11362 | 459 | 764 | 822.0 | 8ZF:60801 | Type1.5_Back | Inactive | DFGin | 5.032 | 13.511 | BLAplus | -110.65, 158.43 | 54.71, 42.71 | -89.1, -11.93 | 53.54, 87.56 | -114.63, 26.86 | in-in | in | 8.234 | Saltbr-in | 2.943 | HRD-in | -65.51, -45.04 | 70.13, -0.28 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.98 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.05, 142.67 | APE9-dihe-in | -99.82, 98.85 | APE8-dihe-out | -66.04, -10.56 | APE8-rot-na | 23.45 | APE67-dihe-in | -75.78, -2.11 | -60.96, -29.19 | APE12-dist-na | 16.725 | APE11-dist-na | 19.067 | APE10-dist-na | 16.226 | APE9-dist-out | 11.223 | C584S | None | None | XRAY | 2.495 | 0.195 | 0.23 | A | 310 | 306 | 0 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 7wcl | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7WCLB | P11362 | 458 | 763 | 822.0 | 8ZF:60801 | Type1.5_Back | Inactive | DFGin | 5.686 | 13.297 | BLAplus | -116.0, 164.36 | 53.53, 38.11 | -89.51, -19.74 | 50.41, 88.95 | -102.65, 11.92 | in-in | in | 8.381 | Saltbr-in | 2.804 | HRD-in | -77.55, -44.61 | 69.5, -1.67 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -124.03, 166.88 | APE9-dihe-in | -112.63, 116.79 | APE8-dihe-out | -58.21, -18.36 | APE8-rot-na | 340.54 | APE67-dihe-in | -81.23, 2.92 | -65.55, -20.31 | APE12-dist-na | 18.6 | APE11-dist-na | 21.605 | APE10-dist-na | 19.498 | APE9-dist-out | 11.402 | C584S | None | None | XRAY | 2.495 | 0.195 | 0.23 | B | 310 | 285 | 21 | 0 | 0 | 8 | [[478, 756]] | 1.0 | 7wcl | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDTA | P22607 | 457 | 756 | 806.0 | MLT:61001,MLT:61002,WGF:61003 | Allosteric,Allosteric,Type1.5_Front | Inactive | DFGin | 5.441 | 13.493 | BLAplus | -114.8, 158.79 | 55.69, 43.2 | -82.19, -34.37 | 42.84, 89.08 | -83.27, -4.41 | in-out | in | 8.383 | Saltbr-out | 5.287 | HRD-in | -68.34, -46.54 | 75.89, -9.4 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.921 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 112.29 | APE8-dihe-out | -63.06, -32.23 | APE8-rot-na | 340.92 | APE67-dihe-in | -68.35, -26.42 | -62.13, -28.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.198 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | A | 297 | 284 | 4 | 0 | 0 | 4 | [[472, 750]] | 1.0 | 8udt | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1 | 260 | 260 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDTB | P22607 | 457 | 754 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.258 | 13.71 | BLAplus | -108.64, 157.87 | 56.15, 40.62 | -79.39, -35.54 | 45.72, 88.06 | -80.67, 0.1 | in-out | in | 8.445 | Saltbr-out | 5.398 | HRD-in | -67.98, -43.8 | 74.91, -8.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.867 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -64.67 | APE9-dihe-out | -68.82, -39.67 | APE8-dihe-out | -56.45, -17.85 | APE8-rot-na | 337.42 | APE67-dihe-in | -61.76, -27.35 | -59.02, -40.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.666 | APE9-dist-out | 10.854 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | B | 297 | 283 | 3 | 0 | 0 | 3 | [[472, 750]] | 1.0 | 8udt | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1 | 260 | 260 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDTC | P22607 | 457 | 756 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.258 | 13.824 | BLAplus | -109.74, 157.08 | 55.91, 40.67 | -78.94, -35.79 | 45.97, 87.77 | -81.04, -4.46 | in-out | in | 8.545 | Saltbr-out | 4.103 | HRD-in | -68.09, -46.3 | 75.11, -4.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.87 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -150.08 | APE9-dihe-out | -67.3, -42.56 | APE8-dihe-out | -46.98, -31.66 | APE8-rot-na | 333.46 | APE67-dihe-in | -60.08, -29.46 | -58.03, -43.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.405 | APE9-dist-out | 11.049 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | C | 297 | 284 | 4 | 0 | 0 | 4 | [[472, 750]] | 1.0 | 8udt | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1 | 260 | 260 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR4 | FGFR4_HUMAN | 7WCXA | P22455 | 453 | 752 | 802.0 | 90F:801 | Type1 | Inactive | DFGin | 5.263 | 13.141 | BLAplus | -114.81, 160.0 | 54.39, 48.08 | -89.68, -16.38 | 44.55, 83.39 | -109.65, 26.27 | in-in | in | 7.792 | Saltbr-in | 2.511 | HRD-in | -76.2, -43.73 | 72.01, -8.39 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.644 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -80.24, 137.24 | APE9-dihe-in | -109.54, 93.42 | APE8-dihe-out | -57.65, -19.77 | APE8-rot-na | 335.57 | APE67-dihe-in | -71.93, -5.42 | -64.19, -25.82 | APE12-dist-na | 19.074 | APE11-dist-na | 20.85 | APE10-dist-na | 16.822 | APE9-dist-out | 11.904 | C477A,R664E | None | None | XRAY | 2.175 | 0.173 | 0.221 | A | 309 | 300 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 7wcx | TYR_FGFR4_HUMAN | TYR | 7e-101 | 342.8 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7WCWA | P22455 | 453 | 752 | 802.0 | 90F:801 | Type1 | Inactive | DFGin | 5.839 | 13.063 | BLAplus | -123.48, 161.59 | 54.95, 50.1 | -96.76, -24.53 | 39.59, 83.16 | -101.63, 31.89 | in-in | in | 7.582 | Saltbr-in | 3.4 | HRD-in | -77.43, -45.16 | 72.65, -7.54 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.633 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -81.49, 135.61 | APE9-dihe-in | -107.87, 94.77 | APE8-dihe-out | -59.45, -18.22 | APE8-rot-na | 336.81 | APE67-dihe-in | -74.15, -1.22 | -67.3, -23.03 | APE12-dist-na | 19.435 | APE11-dist-na | 20.996 | APE10-dist-na | 16.929 | APE9-dist-out | 11.84 | C477A,R664E | None | None | XRAY | 2.317 | 0.179 | 0.221 | A | 309 | 300 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 7wcw | TYR_FGFR4_HUMAN | TYR | 1.9e-100 | 341.4 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 6JPJA | P22455 | 454 | 752 | 802.0 | FGF:800 | Type1 | Inactive | DFGin | 5.301 | 12.658 | BLAplus | -117.71, 161.57 | 53.08, 42.72 | -89.02, -4.4 | 50.47, 87.12 | -117.52, 24.43 | in-in | in | 7.247 | Saltbr-in | 2.318 | HRD-out | -71.89, 98.16 | -78.45, 15.53 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.002 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -85.03, 139.81 | APE9-dihe-in | -112.83, 87.62 | APE8-dihe-out | -50.76, -19.28 | APE8-rot-na | 332.54 | APE67-dihe-in | -80.03, 5.83 | -68.35, -18.64 | APE12-dist-na | 19.294 | APE11-dist-na | 21.068 | APE10-dist-na | 17.129 | APE9-dist-out | 12.054 | C477A,R664E | None | None | XRAY | 2.638 | 0.198 | 0.243 | A | 311 | 299 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 6jpj | TYR_FGFR4_HUMAN | TYR | 1.3e-100 | 341.9 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7VJLA | P22455 | 454 | 753 | 802.0 | 7IF:801 | Type1 | Inactive | DFGin | 5.301 | 12.42 | BLAplus | -114.78, 170.3 | 57.71, 40.42 | -94.32, 21.48 | 55.77, 90.38 | -107.29, 999.0 | in-in | in | 7.485 | Saltbr-in | 2.904 | HRD-out | -79.19, -58.83 | -98.34, 2.36 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 2.26 | APE8-rot-na | 31.94 | APE67-dihe-in | -59.38, -20.97 | -56.11, -39.64 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.9 | 0.212 | 0.273 | A | 301 | 263 | 37 | 0 | 0 | 19 | [[467, 745]] | 1.0 | 7vjl | TYR_FGFR4_HUMAN | TYR | 1.1e-100 | 342.2 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7VJLB | P22455 | 453 | 753 | 802.0 | 7IF:801 | Type1 | Inactive | DFGin | 5.405 | 13.204 | BLAplus | -123.58, 175.88 | 60.77, 35.86 | -95.6, 5.83 | 48.51, 81.65 | -122.94, 999.0 | in-in | in | 7.876 | Saltbr-in | 2.665 | HRD-out | -72.76, -57.66 | -103.85, -18.8 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 6.57 | APE8-rot-na | 30.25 | APE67-dihe-in | -55.58, -34.43 | -70.09, -36.28 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.9 | 0.212 | 0.273 | B | 301 | 266 | 35 | 0 | 0 | 19 | [[467, 745]] | 1.0 | 7vjl | TYR_FGFR4_HUMAN | TYR | 1.1e-100 | 342.2 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 6YI8A | P22455 | 453 | 753 | 802.0 | FGF:801 | Type1 | Inactive | DFGin | 5.052 | 12.585 | BLAplus | -114.37, 162.1 | 61.01, 37.7 | -86.22, -22.44 | 57.75, 86.82 | -88.83, -1.63 | in-in | in | 7.21 | Saltbr-in | 2.807 | HRD-in | -68.35, -54.97 | 79.66, -18.38 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 137.99 | APE9-dihe-in | -91.08, 144.79 | APE8-dihe-in | -80.88, 56.75 | APE8-rot-na | 32.63 | APE67-dihe-in | -69.74, -13.54 | -50.67, -37.69 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 19.129 | APE9-dist-out | 9.562 | None | None | None | XRAY | 2.13 | 0.198 | 0.231 | A | 307 | 277 | 24 | 0 | 0 | 15 | [[467, 745]] | 1.0 | 6yi8 | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.1 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 6YI8B | P22455 | 451 | 752 | 802.0 | FGF:801 | Type1 | Inactive | DFGin | 5.551 | 13.074 | BLAplus | -114.83, 168.14 | 49.73, 54.77 | -99.35, -32.03 | 46.0, 89.99 | -71.98, 999.0 | in-in | in | 7.399 | Saltbr-in | 2.814 | HRD-in | -67.69, -51.4 | 79.31, -36.01 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 133.49 | APE8-dihe-in | -88.73, 63.1 | APE8-rot-na | 25.93 | APE67-dihe-in | -70.74, -12.22 | -53.82, -35.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.081 | None | None | None | XRAY | 2.13 | 0.198 | 0.231 | B | 307 | 270 | 32 | 0 | 0 | 18 | [[467, 745]] | 1.0 | 6yi8 | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.1 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7WCTA | P22455 | 453 | 752 | 802.0 | 90F:801 | Type1 | Inactive | DFGin | 5.499 | 13.008 | BLAplus | -115.75, 158.15 | 54.59, 44.67 | -82.33, -22.35 | 42.51, 87.35 | -106.03, 33.12 | in-in | in | 7.476 | Saltbr-in | 2.881 | HRD-in | -76.31, -44.07 | 70.33, -3.05 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.497 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -84.18, 139.68 | APE9-dihe-in | -111.32, 93.14 | APE8-dihe-out | -55.09, -20.87 | APE8-rot-na | 333.3 | APE67-dihe-in | -74.74, -3.5 | -65.15, -23.14 | APE12-dist-na | 19.463 | APE11-dist-na | 21.045 | APE10-dist-na | 17.074 | APE9-dist-out | 11.772 | R664E | None | None | XRAY | 2.106 | 0.184 | 0.217 | A | 311 | 300 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 7wct | TYR_FGFR4_HUMAN | TYR | 1.9e-100 | 341.4 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 5XFJA | P22455 | 453 | 750 | 802.0 | 6LF:801 | Type1 | Inactive | DFGin | 5.021 | 13.251 | None | -115.6, 133.16 | 70.83, 138.96 | -157.69, 175.22 | 19.16, 82.91 | -161.9, 174.05 | in-out | in | 8.31 | Saltbr-out | 4.274 | HRD-out | -142.96, 112.57 | -85.34, -51.29 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -47.84 | APE8-dihe-in | -93.04, 75.41 | APE8-rot-na | 34.31 | APE67-dihe-in | -59.81, -17.88 | -81.83, -32.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.229 | V550M | None | None | XRAY | 3.25 | 0.284 | 0.336 | A | 311 | 266 | 32 | 0 | 0 | 17 | [[467, 745]] | 1.0 | 5xfj | TYR_FGFR4_HUMAN | TYR | 4.5e-101 | 343.4 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 5XFFA | P22455 | 453 | 750 | 802.0 | 6LF:801 | Type1 | Inactive | DFGin | 7.251 | 13.8 | None | -91.81, 157.14 | 71.12, 141.83 | -151.53, 140.75 | 303.34, 100.5 | -174.03, 158.26 | in-in | in | 7.907 | Saltbr-in | 3.562 | HRD-out | -144.83, 101.6 | -75.14, -41.6 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -18.13 | APE8-dihe-in | -83.47, 67.75 | APE8-rot-na | 31.32 | APE67-dihe-in | -75.73, 1.3 | -73.66, -27.62 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.541 | V550L | None | None | XRAY | 2.7 | 0.27 | 0.32 | A | 311 | 269 | 29 | 0 | 0 | 17 | [[467, 745]] | 1.0 | 5xff | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.0 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 5JKGA | P22455 | 453 | 750 | 802.0 | 6LF:801 | Type1 | Inactive | DFGin | 4.645 | 13.415 | None | -80.35, 138.57 | 42.13, 154.03 | -151.26, -44.79 | 29.5, 89.83 | 59.57, 154.84 | in-in | in | 7.788 | Saltbr-in | 2.748 | HRD-out | -157.35, 80.6 | -45.38, -51.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -51.98 | APE8-dihe-in | -77.75, 74.49 | APE8-rot-na | 28.85 | APE67-dihe-in | -78.7, 0.61 | -72.33, -28.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.405 | None | None | None | XRAY | 2.352 | 0.237 | 0.277 | A | 311 | 266 | 32 | 0 | 0 | 17 | [[467, 745]] | 1.0 | 5jkg | TYR_FGFR4_HUMAN | TYR | 8.4e-101 | 342.6 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FLT3 | FLT3_HUMAN | 6JQRA | P36888 | 571 | 951 | 993.0 | C6F:1001 | Type1 | Inactive | DFGout | 15.394 | 10.885 | None | -119.73, 157.71 | -104.23, 115.68 | 77.2, 999.0 | 255.94, 91.42 | 999.0, 999.0 | in-in | in | 8.326 | Saltbr-in | 2.804 | HRD-out | -98.26, 117.82 | -85.48, 11.47 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.05, 100.76 | APE9-dihe-in | -103.87, 123.04 | APE8-dihe-in | -78.74, 70.62 | APE8-rot-na | 34.5 | APE67-dihe-in | -69.1, -11.06 | -54.04, -46.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.223 | None | None | None | XRAY | 2.2 | 0.181 | 0.213 | A | 330 | 301 | 29 | 0 | 0 | 6 | [[610, 945]] | 1.0 | 6jqr | TYR_FLT3_HUMAN | TYR | 8.5e-103 | 349.1 | 1 | 259 | 259 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| TYR | HCK | HCK_HUMAN | 3VS4A | P08631 | 81 | 526 | 526.0 | VSF:60603 | Type1.5_Back | Inactive | DFGin | 5.296 | 12.617 | BLBplus | -129.05, 156.5 | 78.18, 7.28 | -55.31, 122.08 | 48.34, 94.72 | 91.65, -36.18 | out-out | out | 13.53 | Saltbr-out | 14.391 | HRD-in | -89.51, -57.9 | 84.08, -11.13 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.875 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 47.3 | APE8-dihe-in | -93.7, 67.91 | APE8-rot-na | 28.82 | APE67-dihe-in | -68.45, -16.47 | -64.44, -22.55 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.697 | Q523E,Q524E,Q525I | PTR522 | PTR522 | XRAY | 2.747 | 0.265 | 0.265 | A | 454 | 429 | 11 | 0 | 0 | 11 | [[262, 513]] | 1.0 | 3vs4 | TYR_HCK_HUMAN | TYR | 1.4e-95 | 325.6 | 1 | 260 | 260 | 398 | 399 | 400 | 402 | 404 | 290 | 305 | 309 | 378 | 380 | 379 | 381 | 439 | 427 | 422 | 421 | 420 | 419 | 418 | 417 | 416 | 334 | Tyrosine-protein kinase HCK |
| TYR | HCK | HCK_HUMAN | 3VS4B | P08631 | 81 | 526 | 526.0 | VSF:60603 | Type1.5_Back | Inactive | DFGin | 5.285 | 12.665 | BLBplus | -120.89, 167.83 | 61.49, 15.86 | -62.02, 121.53 | 47.24, 95.4 | 75.03, 10.7 | out-out | out | 13.766 | Saltbr-out | 15.042 | HRD-in | -94.45, -46.27 | 74.87, -7.2 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.135 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 48.23 | APE8-dihe-in | -84.31, 74.96 | APE8-rot-na | 34.0 | APE67-dihe-in | -71.24, -2.76 | -88.69, -13.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.595 | Q523E,Q524E,Q525I | PTR522 | PTR522 | XRAY | 2.747 | 0.265 | 0.265 | B | 454 | 434 | 12 | 0 | 0 | 12 | [[262, 513]] | 1.0 | 3vs4 | TYR_HCK_HUMAN | TYR | 1.4e-95 | 325.6 | 1 | 260 | 260 | 398 | 399 | 400 | 402 | 404 | 290 | 305 | 309 | 378 | 380 | 379 | 381 | 439 | 427 | 422 | 421 | 420 | 419 | 418 | 417 | 416 | 334 | Tyrosine-protein kinase HCK |
| TYR | JAK2-1 | JAK2_HUMAN | 8B9EA | O60674 | 536 | 809 | 1132.0 | Q7F:1003 | Type1 | Pseudo | DFGin | 5.769 | 13.226 | None | -72.27, 175.04 | -67.31, 162.54 | -76.41, -26.42 | 340.6, 33.67 | 78.05, -163.23 | out-na | out | 11.726 | Saltbr-na | 999.0 | HRD-in | -83.9, -60.17 | 88.41, -6.41 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 8.95 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -67.18, -39.02 | APE9-dihe-out | -59.74, -28.13 | APE8-dihe-out | -86.36, 6.28 | APE8-rot-na | 284.57 | APE67-dihe-out | -105.41, 26.85 | -68.63, 134.78 | APE12-dist-na | 9.613 | APE11-dist-na | 11.316 | APE10-dist-na | 15.854 | APE9-dist-out | 12.106 | W777A,F794H | None | None | XRAY | 1.5 | 0.17 | 0.194 | A | 289 | 274 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 8b9e | TYR_JAK2-1_HUMAN | TYR | 6.4e-64 | 221.7 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 8B9HA | O60674 | 536 | 809 | 1132.0 | Q7F:901 | Type1 | Pseudo | DFGin | 6.01 | 13.307 | None | -84.93, -177.89 | -74.12, 157.3 | -67.76, -31.57 | 343.4, 32.07 | 81.26, -168.8 | out-na | out | 12.097 | Saltbr-na | 999.0 | HRD-in | -82.25, -60.3 | 91.76, -5.32 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.143 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -65.85, -39.85 | APE9-dihe-out | -62.27, -26.85 | APE8-dihe-out | -86.04, 1.76 | APE8-rot-na | 292.25 | APE67-dihe-out | -100.68, 23.58 | -62.84, 136.16 | APE12-dist-na | 9.712 | APE11-dist-na | 11.434 | APE10-dist-na | 15.933 | APE9-dist-out | 12.428 | W659A,W777A,F794H | None | None | XRAY | 1.5 | 0.182 | 0.208 | A | 289 | 274 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 8b9h | TYR_JAK2-1_HUMAN | TYR | 1.9e-64 | 223.4 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | KDR | VGFR2_HUMAN | 3VO3A | P35968 | 812 | 1168 | 1356.0 | 0KF:2001 | Type2 | Inactive | DFGout | 16.448 | 8.215 | None | -125.16, 179.81 | -141.05, 99.79 | -70.03, -34.74 | 215.55, 55.41 | 59.77, -120.61 | in-in | in | 7.357 | Saltbr-in | 2.898 | HRD-in | -84.45, -53.71 | 76.95, -3.4 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.477 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.91, 109.54 | APE9-dihe-in | -120.7, 147.5 | APE8-dihe-in | -78.09, 65.8 | APE8-rot-na | 32.33 | APE67-dihe-in | -67.73, -12.3 | -53.4, -39.21 | APE12-dist-na | 17.03 | APE11-dist-na | 14.067 | APE10-dist-na | 11.393 | APE9-dist-in | 7.997 | None | None | None | XRAY | 1.52 | 0.162 | 0.182 | A | 318 | 303 | 4 | 0 | 0 | 0 | [[834, 1162]] | 1.0 | 3vo3 | TYR_KDR_HUMAN | TYR | 4.2e-100 | 340.3 | 1 | 260 | 260 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| TYR | KDR | VGFR2_HUMAN | 1YWNA | P35968 | 820 | 1171 | 1356.0 | LIF:60301 | Type1 | Inactive | None | 999.0 | 999.0 | None | -128.91, 171.96 | -143.62, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 7.21 | Saltbr-in | 2.725 | HRD-in | -77.88, -50.07 | 82.87, -17.6 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -141.39, 161.44 | APE9-dihe-in | -104.18, 100.32 | APE8-dihe-out | -56.09, -24.71 | APE8-rot-na | 336.02 | APE67-dihe-in | -70.59, -14.0 | -51.58, -32.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.239 | E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.71 | 0.206 | 0.23 | A | 316 | 281 | 21 | 0 | 0 | 6 | [[834, 1162]] | 1.0 | 1ywn | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1 | 260 | 260 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| TYR | LCK | LCK_HUMAN | 2ZM1A | P06239 | 231 | 501 | 509.0 | KSF:513 | Type1 | Active | DFGin | 6.499 | 14.193 | BLAminus | -132.48, -160.42 | 31.13, 88.01 | -99.25, 22.14 | 293.45, 97.67 | -69.47, -32.89 | in-in | in | 8.512 | Saltbr-in | 2.933 | HRD-in | -100.89, -51.07 | 73.44, -7.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.929 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.43, 148.33 | APE9-dihe-in | -138.82, 152.04 | APE8-dihe-in | -57.54, 117.05 | APE8-rot-na | 333.13 | APE67-dihe-in | -71.51, -24.6 | -61.57, -39.74 | APE12-dist-na | 15.101 | APE11-dist-na | 10.35 | APE10-dist-na | 13.014 | APE9-dist-in | 6.822 | None | PTR394 | PTR394 | XRAY | 2.1 | 0.172 | 0.232 | A | 285 | 271 | 0 | 0 | 0 | 0 | [[245, 496]] | 1.0 | 2zm1 | TYR_LCK_HUMAN | TYR | 1.5e-94 | 322.1 | 1 | 260 | 260 | 381 | 382 | 383 | 385 | 387 | 273 | 288 | 292 | 361 | 363 | 362 | 364 | 422 | 410 | 405 | 404 | 403 | 402 | 401 | 400 | 399 | 317 | Tyrosine-protein kinase Lck |
| TYR | MERTK | MERTK_HUMAN | 9BHIA | Q12866 | 578 | 864 | 999.0 | A1APF:60901 | Type1.5_Front | Inactive | DFGin | 6.992 | 12.805 | BLAminus | -138.66, -158.87 | 44.96, 74.5 | -90.39, 18.73 | 305.52, 137.7 | -55.48, -30.3 | out-out | out | 13.615 | Saltbr-out | 13.031 | HRD-in | -81.75, -51.8 | 68.35, 6.62 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.82 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.15, 11.33 | APE9-dihe-in | -72.53, 150.77 | APE8-dihe-in | -64.75, 117.67 | APE8-rot-na | 25.92 | APE67-dihe-in | -73.91, -0.64 | -53.67, -34.29 | APE12-dist-na | 7.154 | APE11-dist-na | 12.056 | APE10-dist-na | 11.657 | APE9-dist-in | 6.71 | None | None | None | XRAY | 2.07 | 0.211 | 0.23 | A | 323 | 278 | 9 | 0 | 0 | 2 | [[587, 856]] | 1.0 | 9bhi | TYR_MERTK_HUMAN | TYR | 1.6e-92 | 315.5 | 2 | 261 | 260 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| TYR | MERTK | MERTK_HUMAN | 7AB1A | Q12866 | 571 | 862 | 999.0 | C6F:60901 | Type1 | Inactive | DFGin | 5.872 | 13.527 | None | -150.27, 178.21 | 48.78, 48.66 | -107.87, 999.0 | 41.9, 85.18 | 999.0, 999.0 | out-out | out | 12.844 | Saltbr-out | 9.566 | HRD-in | -84.92, -52.07 | 85.67, -41.55 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 62.29 | APE8-rot-na | 36.31 | APE67-dihe-in | -65.53, -14.5 | -57.08, -42.11 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | K591R,K693R,K702R,K856R | None | None | XRAY | 1.93 | 0.237 | 0.298 | A | 298 | 267 | 25 | 0 | 0 | 20 | [[587, 856]] | 1.0 | 7ab1 | TYR_MERTK_HUMAN | TYR | 2.3e-92 | 314.9 | 2 | 260 | 259 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| TYR | MET | MET_HUMAN | 3ZCLA | P08581 | 1052 | 1345 | 1390.0 | 5TF:1 | Type1 | Inactive | DFGin | 5.341 | 14.033 | BLBplus | -130.37, -159.34 | 48.43, 53.41 | -147.61, 165.56 | 74.15, 92.01 | 59.61, -131.84 | out-out | out | 14.636 | Saltbr-out | 12.785 | HRD-in | -76.45, -51.81 | 82.5, -13.86 | out-out-in | SNCooi | out-in | ActLoopNT-out | 10.735 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.5, 109.91 | APE9-dihe-in | -127.18, 152.9 | APE8-dihe-in | -78.54, 68.73 | APE8-rot-na | 30.54 | APE67-dihe-in | -82.79, -0.65 | -60.11, -28.04 | APE12-dist-na | 22.937 | APE11-dist-na | 18.131 | APE10-dist-na | 17.771 | APE9-dist-in | 7.357 | None | None | None | XRAY | 1.4 | 0.194 | 0.211 | A | 306 | 291 | 3 | 0 | 0 | 0 | [[1078, 1339]] | 1.0 | 3zcl | TYR_MET_HUMAN | TYR | 6.7e-92 | 313.6 | 2 | 260 | 259 | 1221 | 1222 | 1223 | 1225 | 1227 | 1110 | 1127 | 1131 | 1201 | 1203 | 1202 | 1204 | 1265 | 1253 | 1248 | 1247 | 1246 | 1245 | 1244 | 1243 | 1242 | 1158 | Hepatocyte growth factor receptor |
| TYR | MET | MET_HUMAN | 4MXCA | P08581 | 1052 | 1346 | 1390.0 | DWF:1401 | Type2 | Inactive | DFGout | 14.41 | 10.337 | BBAminus | -151.35, -174.18 | -156.99, 122.43 | -67.95, -16.78 | 287.52, 70.23 | 58.23, -116.98 | in-in | in | 8.929 | Saltbr-in | 3.515 | HRD-in | -73.25, -51.06 | 80.68, -17.87 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.287 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -88.68, 108.68 | APE9-dihe-in | -118.71, 133.81 | APE8-dihe-in | -79.71, 72.93 | APE8-rot-na | 28.81 | APE67-dihe-in | -75.71, -5.79 | -60.94, -31.89 | APE12-dist-na | 999.0 | APE11-dist-na | 13.628 | APE10-dist-na | 10.273 | APE9-dist-in | 7.344 | None | None | None | XRAY | 1.632 | 0.18 | 0.207 | A | 319 | 290 | 5 | 0 | 0 | 5 | [[1078, 1339]] | 1.0 | 4mxc | TYR_MET_HUMAN | TYR | 7.7e-92 | 313.7 | 2 | 260 | 259 | 1221 | 1222 | 1223 | 1225 | 1227 | 1110 | 1127 | 1131 | 1201 | 1203 | 1202 | 1204 | 1265 | 1253 | 1248 | 1247 | 1246 | 1245 | 1244 | 1243 | 1242 | 1158 | Hepatocyte growth factor receptor |
| TYR | NTRK1 | NTRK1_HUMAN | 5H3QA | P04629 | 484 | 796 | 796.0 | 7HF:1001 | Type1 | Inactive | DFGout | 12.708 | 6.583 | BBAminus | 172.54, 156.19 | -157.42, 160.24 | -99.39, 17.97 | 295.12, 97.4 | 79.34, 29.52 | in-out | in | 9.447 | Saltbr-out | 5.851 | HRD-in | -81.9, -52.58 | 77.47, -12.71 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.801 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -128.94, 112.39 | APE9-dihe-in | -107.73, 133.13 | APE8-dihe-in | -79.15, 63.42 | APE8-rot-na | 34.45 | APE67-dihe-in | -63.33, -18.08 | -61.61, -34.65 | APE12-dist-na | 13.748 | APE11-dist-na | 15.2 | APE10-dist-na | 10.681 | APE9-dist-in | 7.568 | None | None | None | XRAY | 2.1 | 0.19 | 0.215 | A | 324 | 303 | 10 | 0 | 0 | 0 | [[510, 783]] | 1.0 | 5h3q | TYR_NTRK1_HUMAN | TYR | 2.4e-100 | 341.1 | 2 | 260 | 259 | 667 | 668 | 669 | 671 | 673 | 544 | 560 | 564 | 647 | 649 | 648 | 650 | 709 | 697 | 692 | 691 | 690 | 689 | 688 | 687 | 686 | 590 | High affinity nerve growth factor receptor |
| TYR | NTRK1 | NTRK1_HUMAN | 5KMJA | P04629 | 486 | 795 | 796.0 | 6UF:901 | Type3 | Inactive | DFGout | 12.074 | 7.602 | None | 156.98, 152.76 | -155.56, 161.93 | -106.33, 28.22 | 308.11, 127.92 | 67.17, 26.59 | in-in | in | 9.714 | Saltbr-in | 2.772 | HRD-in | -79.87, -55.53 | 78.72, -12.42 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.107 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -122.86, 120.05 | APE9-dihe-in | -107.69, 130.38 | APE8-dihe-in | -83.48, 63.94 | APE8-rot-na | 32.0 | APE67-dihe-in | -63.64, -21.11 | -52.37, -37.83 | APE12-dist-na | 15.016 | APE11-dist-na | 15.494 | APE10-dist-na | 11.096 | APE9-dist-in | 7.6 | None | None | None | XRAY | 2.04 | 0.196 | 0.226 | A | 329 | 300 | 6 | 0 | 0 | 0 | [[510, 783]] | 1.0 | 5kmj | TYR_NTRK1_HUMAN | TYR | 2.5e-100 | 341.0 | 2 | 260 | 259 | 667 | 668 | 669 | 671 | 673 | 544 | 560 | 564 | 647 | 649 | 648 | 650 | 709 | 697 | 692 | 691 | 690 | 689 | 688 | 687 | 686 | 590 | High affinity nerve growth factor receptor |
| TYR | PTK2 | FAK1_HUMAN | 4EBWA | Q05397 | 411 | 686 | 1052.0 | 0PF:700 | Type1 | Inactive | DFGinter | 10.52 | 8.023 | None | -156.77, 167.19 | -119.55, 38.35 | -154.8, 160.1 | 57.14, 97.67 | -105.09, 155.15 | in-in | in | 7.232 | Saltbr-in | 3.021 | HRD-out | -85.85, 108.83 | -92.42, -13.42 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 105.2 | APE9-dihe-in | -103.42, 143.85 | APE8-dihe-in | -74.96, 72.04 | APE8-rot-na | 29.05 | APE67-dihe-in | -70.29, -24.24 | -52.29, -39.56 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 17.857 | APE9-dist-out | 9.391 | None | None | None | XRAY | 2.65 | 0.186 | 0.273 | A | 304 | 259 | 17 | 0 | 0 | 15 | [[422, 678]] | 1.0 | 4ebw | TYR_PTK2_HUMAN | TYR | 4.7e-93 | 317.2 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | SYK | KSYK_HUMAN | 5LMBA | P43405 | 364 | 634 | 635.0 | 6ZF:701 | Type1 | Active | DFGin | 6.448 | 14.283 | BLAminus | -131.02, -173.87 | 62.28, 69.39 | -93.16, 19.0 | 290.08, 82.25 | -59.68, -28.46 | in-in | in | 7.696 | Saltbr-in | 2.454 | HRD-in | -78.06, -53.9 | 76.38, 4.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.963 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.66, 104.96 | APE9-dihe-in | -108.73, 152.4 | APE8-dihe-in | -79.7, 70.25 | APE8-rot-na | 31.84 | APE67-dihe-in | -69.34, -16.13 | -51.43, -34.69 | APE12-dist-na | 13.073 | APE11-dist-na | 10.546 | APE10-dist-na | 11.448 | APE9-dist-in | 6.959 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | A | 277 | 265 | 6 | 0 | 0 | 0 | [[370, 628]] | 1.0 | 5lmb | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 5LMBB | P43405 | 364 | 630 | 635.0 | 6ZF:701 | Type1 | None | DFGin | 6.542 | 14.207 | BLAminus | -133.05, -174.7 | 62.98, 72.21 | -97.02, 21.38 | 290.54, 88.36 | -62.52, -32.46 | in-in | in | 7.737 | Saltbr-in | 2.556 | HRD-in | -77.26, -52.74 | 74.6, 8.57 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.872 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 129.43 | APE8-dihe-in | -80.7, 73.18 | APE8-rot-na | 30.16 | APE67-dihe-in | -64.42, -18.25 | -49.18, -37.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.948 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | B | 277 | 262 | 5 | 0 | 0 | 5 | [[370, 628]] | 1.0 | 5lmb | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 4YJOA | P43405 | 363 | 632 | 635.0 | 4DF:701 | Type1 | Active | DFGin | 7.151 | 15.404 | BLAminus | -136.57, 178.57 | 59.58, 80.7 | -95.16, 22.65 | 286.36, 75.19 | -55.96, -31.16 | in-in | in | 8.32 | Saltbr-in | 3.044 | HRD-in | -80.48, -52.4 | 72.29, 6.84 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.957 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -56.5, 127.44 | APE9-dihe-in | -144.08, 83.31 | APE8-dihe-in | -75.74, 70.97 | APE8-rot-na | 33.07 | APE67-dihe-in | -63.43, -16.56 | -52.99, -37.5 | APE12-dist-na | 999.0 | APE11-dist-na | 10.63 | APE10-dist-na | 7.9 | APE9-dist-in | 7.507 | None | None | None | XRAY | 1.6 | 0.186 | 0.23 | A | 281 | 267 | 3 | 0 | 0 | 3 | [[370, 628]] | 1.0 | 4yjo | TYR_SYK_HUMAN | TYR | 4.8e-90 | 307.3 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 5TT7A | P43405 | 358 | 635 | 635.0 | 7KF:60901 | Type1 | Active | DFGin | 6.311 | 14.341 | BLAminus | -130.62, -177.29 | 62.11, 72.82 | -94.96, 21.67 | 289.95, 80.8 | -60.6, -26.94 | in-in | in | 7.709 | Saltbr-in | 2.84 | HRD-in | -77.7, -52.28 | 69.96, 13.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.878 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.65, 88.09 | APE9-dihe-in | -107.14, 140.48 | APE8-dihe-in | -78.3, 78.38 | APE8-rot-na | 32.04 | APE67-dihe-in | -64.56, -15.37 | -56.64, -35.35 | APE12-dist-na | 13.888 | APE11-dist-na | 10.557 | APE10-dist-na | 10.342 | APE9-dist-in | 6.849 | None | None | None | XRAY | 1.77 | 0.208 | 0.234 | A | 289 | 270 | 8 | 0 | 0 | 0 | [[370, 628]] | 1.0 | 5tt7 | TYR_SYK_HUMAN | TYR | 5.4e-90 | 307.1 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 4FYOA | P43405 | 363 | 635 | 635.0 | 0VF:60701 | Type1 | None | DFGin | 6.527 | 14.676 | BLAminus | -132.65, -177.95 | 62.23, 72.42 | -93.99, 21.12 | 289.45, 90.18 | -61.07, -25.58 | in-in | in | 7.75 | Saltbr-in | 2.757 | HRD-in | -74.26, -50.97 | 72.76, 4.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.952 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 140.05 | APE9-dihe-in | -108.11, 144.2 | APE8-dihe-in | -76.07, 73.27 | APE8-rot-na | 27.85 | APE67-dihe-in | -65.29, -14.44 | -52.41, -38.79 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.947 | APE9-dist-in | 7.308 | None | None | None | XRAY | 1.4 | 0.22 | 0.24 | A | 291 | 263 | 10 | 0 | 0 | 4 | [[370, 628]] | 1.0 | 4fyo | TYR_SYK_HUMAN | TYR | 5.5e-90 | 307.1 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 4GFGA | P43405 | 363 | 635 | 635.0 | 0XF:60701 | Type1 | Active | DFGin | 6.382 | 14.706 | BLAminus | -133.41, -165.6 | 61.44, 68.78 | -94.44, 29.51 | 290.84, 74.86 | -64.09, -30.1 | in-in | in | 8.551 | Saltbr-in | 3.497 | HRD-in | -86.12, -47.8 | 68.36, 5.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.866 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -53.12, 138.6 | APE9-dihe-in | -110.15, 137.21 | APE8-dihe-in | -65.63, 68.92 | APE8-rot-na | 25.72 | APE67-dihe-in | -68.08, -17.47 | -52.98, -35.53 | APE12-dist-na | 9.582 | APE11-dist-na | 10.629 | APE10-dist-na | 11.706 | APE9-dist-in | 7.231 | None | None | None | XRAY | 2.35 | 0.221 | 0.246 | A | 291 | 273 | 0 | 0 | 0 | 0 | [[370, 628]] | 1.0 | 4gfg | TYR_SYK_HUMAN | TYR | 5.5e-90 | 307.1 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|---|---|---|---|
| DFGin | BLAminus | 86 | 47.5% | 4AW0A |
| DFGin | ABAminus | 22 | 12.2% | 7PIEA |
| DFGin | BLAplus | 19 | 10.5% | 9UHIA |
| DFGin | None | 16 | 8.8% | 8B9EA |
| DFGin | BLBplus | 10 | 5.5% | 3ZCLA |
| DFGout | BBAminus | 10 | 5.5% | 4MXCA |
| DFGout | None | 9 | 5.0% | 3VO3A |
| DFGin | BLBminus | 4 | 2.2% | 5R9OA |
| DFGin | BLBtrans | 2 | 1.1% | 2R3IA |
| None | None | 2 | 1.1% | 5IEXA |
| DFGinter | None | 1 | 0.6% | 4EBWA |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_CRIGR | 7PIEA | P25321 | 1 | 351 | 351.0 | 7QF:60401 | Type1 | Inactive | DFGin | 6.437 | 14.708 | ABAminus | -120.2, -32.0 | -97.5, 116.46 | -117.79, 21.67 | 284.38, 87.37 | -67.96, -24.99 | in-in | in | 9.018 | Saltbr-in | 2.947 | HRD-in | -90.08, -55.75 | 70.92, 8.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.9, 155.75 | APE9-dihe-na | 129.48, -166.45 | APE8-dihe-in | -116.19, 135.64 | APE8-rot-in | 298.32 | APE67-dihe-in | -59.08, -26.0 | -47.12, -51.73 | APE12-dist-in | 8.298 | APE11-dist-in | 11.483 | APE10-dist-in | 5.921 | APE9-dist-in | 3.894 | None | SEP11,SEP140,TPO198,SEP339 | SEP11,SEP140,TPO198,SEP339 | XRAY | 1.427 | 0.137 | 0.158 | A | 353 | 350 | 0 | 0 | 0 | 0 | [[44, 298]] | 1.0 | 7pie | Cricetulus griseus | AGC_PRKACA_CRIGR | AGC | 6.6e-95 | 323.2 | 1 | 260 | 260 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_CRIGR | 9RETA | P25321 | 13 | 351 | 351.0 | A1JEF:60404 | Allosteric | Active | DFGin | 6.503 | 14.919 | BLAminus | -121.64, 161.02 | 79.66, 89.44 | -97.28, 25.84 | 271.42, 57.67 | -59.32, -29.98 | in-in | in | 9.058 | Saltbr-in | 2.688 | HRD-in | -91.57, -50.28 | 65.7, 14.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.961 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.82, 155.57 | APE9-dihe-na | 119.38, 155.92 | APE8-dihe-in | -73.83, 138.5 | APE8-rot-in | 315.72 | APE67-dihe-in | -57.32, -25.4 | -54.39, -42.36 | APE12-dist-in | 8.186 | APE11-dist-in | 11.402 | APE10-dist-in | 5.952 | APE9-dist-in | 4.241 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 1.75 | 0.193 | 0.227 | A | 353 | 339 | 0 | 0 | 0 | 0 | [[44, 298]] | 1.0 | 9ret | Cricetulus griseus | AGC_PRKACA_CRIGR | AGC | 6.6e-95 | 323.2 | 1 | 260 | 260 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| TYR | SRC | SRC_CHICK | 5SYSA | P00523 | 258 | 533 | 533.0 | 72F:600 | Type2 | Inactive | DFGout | 13.354 | 9.801 | BBAminus | -126.48, -173.83 | -168.38, 115.62 | -104.78, -47.96 | 311.28, 146.33 | 163.56, 999.0 | in-in | in | 8.579 | Saltbr-in | 3.03 | HRD-in | -86.37, -44.08 | 72.1, 11.73 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -16.31 | APE8-rot-na | 5.39 | APE67-dihe-in | -61.6, -39.03 | -88.61, -20.33 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | V281C | None | None | XRAY | 2.8 | 0.288 | 0.334 | A | 286 | 258 | 18 | 0 | 0 | 18 | [[267, 518]] | 1.0 | 5sys | Gallus gallus | TYR_SRC_CHICK | TYR | 4.2e-93 | 317.3 | 1 | 260 | 260 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 5SYSB | P00523 | 258 | 533 | 533.0 | 72F:600 | Type2 | Inactive | DFGout | 13.413 | 10.163 | BBAminus | -126.31, -175.1 | -166.31, 115.77 | -103.34, -47.57 | 306.63, 130.98 | 67.96, 999.0 | in-in | in | 8.321 | Saltbr-in | 3.044 | HRD-in | -86.54, -44.23 | 72.2, 11.45 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -18.84 | APE8-rot-na | 6.43 | APE67-dihe-in | -61.0, -39.73 | -89.58, -19.88 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | V281C | None | None | XRAY | 2.8 | 0.288 | 0.334 | B | 286 | 258 | 18 | 0 | 0 | 18 | [[267, 518]] | 1.0 | 5sys | Gallus gallus | TYR_SRC_CHICK | TYR | 4.2e-93 | 317.3 | 1 | 260 | 260 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| AGC | AKT1 | AKT1_HUMAN | 4EKLA | P31749 | 144 | 478 | 480.0 | 0RF:501 | Type1 | Active | DFGin | 6.496 | 13.423 | BLAminus | -130.08, 156.46 | 77.16, 99.77 | -112.66, 14.16 | 298.65, 90.33 | -61.32, -30.96 | in-in | in | 8.958 | Saltbr-in | 2.452 | HRD-in | -78.38, -44.96 | 68.93, -13.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.757 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.83, 160.76 | APE9-dihe-na | 116.71, 166.32 | APE8-dihe-in | -83.66, 133.51 | APE8-rot-in | 293.53 | APE67-dihe-in | -68.09, -18.95 | -43.13, -46.31 | APE12-dist-in | 8.36 | APE11-dist-in | 11.512 | APE10-dist-in | 6.011 | APE9-dist-in | 4.443 | S473D | TPO308 | TPO308 | XRAY | 2.0 | 0.175 | 0.235 | A | 341 | 330 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekl | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AGC | GRK5 | GRK5_HUMAN | 9BRPA | P34947 | 25 | 542 | 590.0 | A1ARF:601 | Type1 | Inactive | DFGin | 6.253 | 12.479 | ABAminus | -116.3, -61.02 | -91.04, 101.81 | -97.25, 10.66 | 289.92, 84.11 | -59.57, -18.7 | in-in | in | 8.91 | Saltbr-in | 3.037 | HRD-in | -85.07, -56.86 | 71.89, 13.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.105 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.18, 177.63 | APE9-dihe-na | 122.23, -155.28 | APE8-dihe-in | -122.73, 136.27 | APE8-rot-in | 286.0 | APE67-dihe-inflip | 100.9, -21.88 | -54.82, 128.22 | APE12-dist-in | 9.574 | APE11-dist-in | 11.932 | APE10-dist-in | 6.253 | APE9-dist-in | 4.143 | D311N | None | None | XRAY | 2.8 | 0.245 | 0.283 | A | 598 | 502 | 0 | 0 | 0 | 0 | [[186, 448]] | 1.0 | 9brp | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1 | 260 | 260 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | GRK5 | GRK5_HUMAN | 9BREA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Active | DFGin | 6.176 | 12.564 | BLAminus | -128.67, 172.15 | 57.35, 77.75 | -93.22, 24.8 | 286.17, 72.14 | -63.15, -21.99 | in-in | in | 8.801 | Saltbr-in | 2.458 | HRD-in | -88.2, -51.09 | 67.29, 13.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.127 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.49, 165.19 | APE9-dihe-na | 125.58, -150.88 | APE8-dihe-in | -124.55, 138.39 | APE8-rot-in | 312.36 | APE67-dihe-inflip | 92.11, -16.19 | -53.44, 132.83 | APE12-dist-in | 9.943 | APE11-dist-in | 12.131 | APE10-dist-in | 6.337 | APE9-dist-in | 4.122 | D311N | None | None | XRAY | 2.8 | 0.215 | 0.26 | A | 598 | 503 | 0 | 0 | 0 | 0 | [[186, 448]] | 1.0 | 9bre | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1 | 260 | 260 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | GRK5 | GRK5_HUMAN | 8UAQA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Inactive | DFGin | 6.02 | 12.841 | None | -112.48, -65.82 | -86.97, 96.33 | -93.06, 17.75 | 286.66, 70.13 | -64.2, -19.76 | in-in | in | 9.334 | Saltbr-in | 3.369 | HRD-in | -90.24, -57.5 | 70.99, -0.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.037 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.56, 170.13 | APE9-dihe-na | 119.68, -157.85 | APE8-dihe-in | -112.7, 143.6 | APE8-rot-in | 314.4 | APE67-dihe-inflip | 89.64, -4.73 | -59.54, 131.81 | APE12-dist-in | 9.916 | APE11-dist-in | 12.102 | APE10-dist-in | 6.306 | APE9-dist-in | 4.174 | D311N | None | None | XRAY | 2.8 | 0.232 | 0.277 | A | 598 | 501 | 0 | 0 | 0 | 0 | [[186, 448]] | 1.0 | 8uaq | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1 | 260 | 260 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | PDPK1 | PDPK1_HUMAN | 4AW0A | O15530 | 75 | 359 | 556.0 | ATP:500,MJF:600 | ATPlike,Allosteric | Active | DFGin | 6.531 | 14.993 | BLAminus | -134.84, 177.25 | 78.73, 76.19 | -106.3, 8.53 | 283.51, 97.11 | -69.63, -19.36 | in-in | in | 8.595 | Saltbr-in | 3.009 | HRD-in | -83.05, -53.03 | 79.45, -12.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.934 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.69, 159.04 | APE9-dihe-na | 139.48, -167.8 | APE8-dihe-in | -131.87, 132.42 | APE8-rot-in | 295.45 | APE67-dihe-in | -61.29, -25.28 | -54.74, -42.17 | APE12-dist-in | 7.509 | APE11-dist-in | 10.601 | APE10-dist-in | 5.026 | APE9-dist-in | 3.58 | Y288G,Q292A | SEP241 | SEP241,CME260 | XRAY | 1.43 | 0.171 | 0.188 | A | 311 | 285 | 0 | 0 | 0 | 0 | [[82, 342]] | 1.0 | 4aw0 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1 | 260 | 260 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PRKCH | KPCL_HUMAN | 8FP1A | P24723 | 349 | 676 | 683.0 | XXF:9000 | Type1 | Active | DFGin | 6.04 | 12.861 | BLAminus | -134.17, 160.39 | 76.6, 103.68 | -113.44, 14.82 | 306.37, 103.97 | -62.81, -37.48 | in-in | in | 8.529 | Saltbr-in | 2.747 | HRD-in | -71.28, -48.4 | 60.66, 8.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.042 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -168.52, 169.89 | APE9-dihe-na | 121.68, 166.05 | APE8-dihe-in | -83.39, 128.15 | APE8-rot-in | 297.95 | APE67-dihe-in | -61.25, -27.98 | -43.8, -44.17 | APE12-dist-in | 8.666 | APE11-dist-in | 11.701 | APE10-dist-in | 6.365 | APE9-dist-in | 3.566 | S675E | TPO513,TPO656 | TPO513,TPO656 | XRAY | 1.85 | 0.2 | 0.234 | A | 353 | 328 | 0 | 0 | 0 | 0 | [[355, 614]] | 1.0 | 8fp1 | Homo sapiens | AGC_PRKCH_HUMAN | AGC | 1.6e-97 | 331.6 | 1 | 260 | 260 | 496 | 497 | 498 | 500 | 502 | 384 | 403 | 407 | 476 | 478 | 477 | 479 | 536 | 524 | 519 | 518 | 517 | 516 | 515 | 514 | 513 | 434 | Protein kinase C eta type |
| CAMK | AURKA | AURKA_HUMAN | 8C1DA | O14965 | 127 | 388 | 403.0 | T2F:401,ADP:402,T5L:405 | Allosteric,ATPlike,Allosteric | Inactive | DFGin | 5.59 | 14.77 | BLAminus | -129.39, 179.64 | 57.3, 80.97 | -92.88, 23.53 | 280.13, 79.47 | -56.16, -33.44 | in-in | in | 9.306 | Saltbr-in | 2.936 | HRD-in | -72.1, -50.49 | 67.69, -1.24 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.796 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 144.85 | APE8-dihe-in | -64.26, 154.27 | APE8-rot-out | 88.6 | APE67-dihe-in | -39.49, -36.75 | -82.32, -6.09 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.088 | C290A | None | None | XRAY | 2.115 | 0.212 | 0.238 | A | 265 | 259 | 3 | 0 | 0 | 3 | [[133, 383]] | 1.0 | 8c1d | Homo sapiens | CAMK_AURKA_HUMAN | CAMK | 7.2e-79 | 270.6 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | AURKA | AURKA_HUMAN | 2W1FA | O14965 | 127 | 389 | 403.0 | L0F:61390 | Type1 | Inactive | DFGin | 5.655 | 15.703 | BLAminus | -96.26, 172.45 | 62.06, 107.69 | -118.91, 38.89 | 289.12, 66.42 | -59.62, -48.4 | out-out | out | 10.139 | Saltbr-out | 5.12 | HRD-in | -78.79, -54.88 | 78.03, -25.41 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.676 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -157.03 | APE8-dihe-in | -58.47, 105.92 | APE8-rot-out | 190.33 | APE67-dihe-in | -42.4, -27.58 | -64.36, -20.47 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.774 | None | None | None | XRAY | 2.85 | 0.246 | 0.348 | A | 275 | 253 | 10 | 0 | 0 | 10 | [[133, 383]] | 1.0 | 2w1f | Homo sapiens | CAMK_AURKA_HUMAN | CAMK | 6.7e-80 | 274.0 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | AURKA | AURKA_HUMAN | 3O51A | O14965 | 126 | 388 | 403.0 | LJF:1 | Type1.5_Front | Inactive | DFGout | 12.921 | 9.215 | None | -125.94, 46.56 | -78.14, 156.47 | -164.09, 999.0 | 59.42, 112.33 | 999.0, 999.0 | out-none | out | 12.863 | Saltbr-none | 999.0 | HRD-out | -126.02, 153.87 | -92.88, -115.51 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -57.91, -10.7 | 999.0, -51.84 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 3.2 | 0.288 | 0.304 | A | 267 | 246 | 17 | 0 | 0 | 17 | [[133, 383]] | 1.0 | 3o51 | Homo sapiens | CAMK_AURKA_HUMAN | CAMK | 6e-80 | 274.2 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | CAMK2A | KCC2A_HUMAN | 2VZ6A | Q9UQM7 | 9 | 299 | 478.0 | FEF:60600 | Type1 | Active | DFGin | 7.124 | 13.93 | BLAminus | -130.3, 144.9 | 77.59, 104.3 | -118.45, 37.91 | 281.19, 70.53 | -60.86, -31.43 | in-in | in | 9.032 | Saltbr-in | 2.623 | HRD-in | -71.43, -45.76 | 75.34, -9.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.805 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.76, 148.02 | APE9-dihe-na | 132.07, -168.34 | APE8-dihe-in | -120.79, 126.49 | APE8-rot-in | 299.71 | APE67-dihe-in | -63.07, -18.83 | -35.01, -58.7 | APE12-dist-in | 10.327 | APE11-dist-in | 11.819 | APE10-dist-in | 5.993 | APE9-dist-in | 3.832 | None | None | None | XRAY | 2.3 | 0.165 | 0.203 | A | 313 | 289 | 2 | 0 | 0 | 0 | [[13, 271]] | 1.0 | 2vz6 | Homo sapiens | CAMK_CAMK2A_HUMAN | CAMK | 1.6e-96 | 328.7 | 1 | 256 | 256 | 155 | 156 | 157 | 159 | 161 | 42 | 60 | 64 | 132 | 134 | 133 | 135 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 90 | Calcium/calmodulin-dependent protein kinase type II subunit alpha |
| CAMK | CAMK2A | KCC2A_HUMAN | 2VZ6B | Q9UQM7 | 9 | 300 | 478.0 | FEF:60600 | Type1 | Active | DFGin | 6.865 | 14.032 | BLAminus | -131.92, 139.26 | 77.54, 110.88 | -122.08, 32.95 | 286.68, 71.96 | -61.55, -26.54 | in-in | in | 9.31 | Saltbr-in | 2.931 | HRD-in | -73.12, -44.65 | 73.93, -20.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.874 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -148.21, 149.78 | APE9-dihe-na | 143.11, -171.05 | APE8-dihe-in | -118.3, 128.44 | APE8-rot-in | 303.95 | APE67-dihe-in | -66.72, -18.78 | -39.97, -52.82 | APE12-dist-in | 10.252 | APE11-dist-in | 11.756 | APE10-dist-in | 5.996 | APE9-dist-in | 3.963 | None | None | None | XRAY | 2.3 | 0.165 | 0.203 | B | 313 | 292 | 0 | 0 | 0 | 0 | [[13, 271]] | 1.0 | 2vz6 | Homo sapiens | CAMK_CAMK2A_HUMAN | CAMK | 1.6e-96 | 328.7 | 1 | 256 | 256 | 155 | 156 | 157 | 159 | 161 | 42 | 60 | 64 | 132 | 134 | 133 | 135 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 90 | Calcium/calmodulin-dependent protein kinase type II subunit alpha |
| CAMK | CHEK1 | CHK1_HUMAN | 8E80A | O14757 | 8 | 271 | 476.0 | UUF:301 | Type1 | Active | DFGin | 6.948 | 13.561 | BLAminus | -116.38, 163.51 | 69.37, 105.0 | -111.89, 20.17 | 292.16, 81.73 | -65.53, -30.68 | in-in | in | 8.579 | Saltbr-in | 2.859 | HRD-in | -73.57, -45.75 | 72.69, 0.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.949 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -163.33, 170.54 | APE9-dihe-na | 117.83, -149.18 | APE8-dihe-in | -134.92, 121.74 | APE8-rot-in | 303.05 | APE67-dihe-in | -62.91, -20.27 | -44.12, -51.23 | APE12-dist-in | 9.365 | APE11-dist-in | 11.644 | APE10-dist-in | 6.142 | APE9-dist-in | 3.497 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | None | XRAY | 1.49 | 0.209 | 0.242 | A | 297 | 258 | 6 | 0 | 0 | 0 | [[9, 265]] | 1.0 | 8e80 | Homo sapiens | CAMK_CHEK1_HUMAN | CAMK | 4.8e-69 | 238.4 | 2 | 256 | 255 | 147 | 148 | 149 | 151 | 153 | 38 | 55 | 59 | 127 | 129 | 128 | 130 | 190 | 177 | 172 | 171 | 170 | 169 | 168 | 167 | 166 | 85 | Serine/threonine-protein kinase Chk1 |
| CAMK | CHEK2 | CHK2_HUMAN | 2YCFA | O96017 | 210 | 510 | 543.0 | YCF:600 | Type1 | Inactive | DFGin | 6.651 | 14.425 | BLAminus | -133.14, 179.08 | 68.92, 89.26 | -105.02, 26.49 | 290.18, 77.38 | -65.99, -23.19 | in-out | in | 9.994 | Saltbr-out | 8.56 | HRD-in | -70.72, -52.98 | 75.15, -0.9 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.905 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -72.28, -26.54 | APE9-dihe-na | -96.81, -179.54 | APE8-dihe-in | -85.38, 132.85 | APE8-rot-in | 297.44 | APE67-dihe-in | -44.53, -40.92 | -82.1, 28.65 | APE12-dist-out | 25.231 | APE11-dist-out | 27.289 | APE10-dist-out | 29.363 | APE9-dist-out | 33.105 | None | None | None | XRAY | 1.77 | 0.197 | 0.218 | A | 322 | 286 | 15 | 0 | 0 | 0 | [[220, 486]] | 1.0 | 2ycf | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 2e-85 | 292.2 | 1 | 256 | 256 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | DAPK1 | DAPK1_HUMAN | 6AARA | P53355 | 2 | 277 | 1430.0 | 9TF:300 | Type1 | Inactive | DFGin | 6.743 | 14.342 | BLAminus | -121.31, 178.32 | 64.29, 78.62 | -87.38, 15.28 | 286.92, 75.84 | -59.31, -26.74 | in-in | in | 9.386 | Saltbr-in | 2.811 | HRD-in | -76.03, -46.41 | 70.92, -12.19 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.921 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -137.91, 116.13 | APE9-dihe-na | -97.58, -145.9 | APE8-dihe-in | -81.4, 124.5 | APE8-rot-in | 302.0 | APE67-dihe-in | -55.21, -31.9 | -47.73, -42.04 | APE12-dist-in | 11.019 | APE11-dist-out | 6.26 | APE10-dist-out | 9.242 | APE9-dist-in | 4.805 | None | None | None | XRAY | 1.95 | 0.182 | 0.22 | A | 293 | 269 | 7 | 0 | 0 | 0 | [[13, 275]] | 1.0 | 6aar | Homo sapiens | CAMK_DAPK1_HUMAN | CAMK | 6.1e-95 | 323.3 | 1 | 256 | 256 | 160 | 161 | 162 | 164 | 166 | 42 | 64 | 68 | 136 | 138 | 137 | 139 | 199 | 187 | 182 | 181 | 180 | 179 | 178 | 177 | 176 | 94 | Death-associated protein kinase 1 |
| CAMK | MAPKAPK2 | MAPK2_HUMAN | 3M42A | P49137 | 47 | 364 | 400.0 | HGF:365 | Type1 | None | DFGin | 4.265 | 13.765 | BLAminus | -127.28, 170.7 | 71.87, 101.44 | -103.87, 20.75 | 277.01, 69.5 | -61.92, -8.22 | in-in | in | 9.26 | Saltbr-in | 3.091 | HRD-in | -73.72, -58.45 | 76.25, 11.76 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.912 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | P237G | None | None | XRAY | 2.68 | 0.186 | 0.232 | A | 299 | 290 | 7 | 0 | 0 | 0 | [[63, 325]] | 1.0 | 3m42 | Homo sapiens | CAMK_MAPKAPK2_HUMAN | CAMK | 1.9e-36 | 228.6 | 3 | 154 | 236 | 206 | 207 | 208 | 210 | 212 | 93 | 104 | 108 | 183 | 185 | 184 | 186 | 245 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 139 | MAP kinase-activated protein kinase 2 |
| CAMK | MELK | MELK_HUMAN | 5IH9A | Q14680 | 3 | 327 | 651.0 | 6BF:60401 | Type1 | None | DFGin | 6.939 | 15.146 | BLAminus | -123.48, 176.08 | 58.26, 79.91 | -95.72, 21.84 | 280.98, 78.3 | -67.92, -25.97 | in-in | in | 8.72 | Saltbr-in | 2.587 | HRD-in | -71.83, -48.59 | 72.02, -0.04 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.992 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -4.81 | APE8-rot-in | 291.01 | APE67-dihe-in | -55.95, -27.86 | -55.75, -43.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.79 | 0.174 | 0.2 | A | 335 | 307 | 18 | 0 | 0 | 14 | [[11, 263]] | 1.0 | 5ih9 | Homo sapiens | CAMK_MELK_HUMAN | CAMK | 9.7e-89 | 303.1 | 1 | 256 | 256 | 149 | 150 | 151 | 153 | 155 | 40 | 57 | 61 | 129 | 131 | 130 | 132 | 191 | 178 | 173 | 172 | 171 | 170 | 169 | 168 | 167 | 87 | Maternal embryonic leucine zipper kinase |
| CAMK | PIM1 | PIM1_HUMAN | 5KGIA | P11309 | 33 | 305 | 313.0 | 6SF:414 | Type1 | Active | DFGin | 6.196 | 14.678 | BLAminus | -128.85, 173.72 | 58.37, 80.83 | -91.15, 15.65 | 283.15, 78.86 | -67.29, -15.19 | in-in | in | 8.898 | Saltbr-in | 2.699 | HRD-na-A | -66.85, -48.52 | 69.49, 3.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.854 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.48, 30.3 | APE9-dihe-na | -88.67, -155.26 | APE8-dihe-in | -89.24, 121.14 | APE8-rot-in | 310.96 | APE67-dihe-in | -66.24, -12.88 | -55.29, -44.34 | APE12-dist-in | 9.723 | APE11-dist-in | 8.735 | APE10-dist-in | 5.642 | APE9-dist-in | 3.74 | None | None | None | XRAY | 2.13 | 0.173 | 0.186 | A | 276 | 273 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 5kgi | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 2.5e-65 | 226.2 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 6L13A | P11309 | 33 | 305 | 313.0 | E2F:401 | Type1 | Active | DFGin | 6.19 | 14.786 | BLAminus | -130.24, 168.2 | 68.46, 80.68 | -89.17, 16.05 | 288.1, 80.31 | -69.01, -19.61 | in-in | in | 9.105 | Saltbr-in | 2.936 | HRD-na-A | -68.46, -51.8 | 71.9, 8.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.778 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.76, 29.56 | APE9-dihe-na | -92.34, -153.25 | APE8-dihe-in | -98.43, 124.2 | APE8-rot-in | 303.55 | APE67-dihe-in | -68.48, -12.49 | -58.68, -45.06 | APE12-dist-in | 9.5 | APE11-dist-in | 8.511 | APE10-dist-in | 5.099 | APE9-dist-in | 3.659 | None | SEP261 | SEP261 | XRAY | 2.24 | 0.18 | 0.214 | A | 289 | 273 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 6l13 | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 3e-65 | 226.0 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 2O65A | P11309 | 33 | 306 | 313.0 | MYF:501 | Type1 | Active | DFGin | 5.773 | 14.223 | BLAminus | -134.9, 170.04 | 60.08, 89.22 | -101.35, 10.62 | 287.34, 92.73 | -63.96, -9.9 | in-in | in | 8.704 | Saltbr-in | 2.471 | HRD-na-A | -65.14, -47.59 | 70.03, -4.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.98 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.66, 34.64 | APE9-dihe-na | -104.35, -148.26 | APE8-dihe-in | -83.11, 121.1 | APE8-rot-in | 316.59 | APE67-dihe-in | -62.15, -16.44 | -57.04, -47.52 | APE12-dist-in | 9.988 | APE11-dist-in | 8.628 | APE10-dist-in | 5.289 | APE9-dist-in | 4.136 | None | None | None | XRAY | 2.85 | 0.21 | 0.262 | A | 293 | 274 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 2o65 | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 3.2e-65 | 226.0 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 8R0WA | P11309 | 33 | 305 | 313.0 | XGF:405 | Type1 | Active | DFGin | 5.997 | 14.384 | BLAminus | -131.73, 166.77 | 65.97, 82.46 | -89.79, 16.41 | 289.35, 79.56 | -63.02, -16.4 | in-in | in | 8.812 | Saltbr-in | 2.643 | HRD-na-A | -73.15, -45.35 | 65.43, 10.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.23, 17.26 | APE9-dihe-na | -81.93, -156.28 | APE8-dihe-in | -91.39, 121.88 | APE8-rot-in | 296.84 | APE67-dihe-in | -71.92, -8.94 | -64.52, -38.27 | APE12-dist-in | 9.559 | APE11-dist-in | 8.479 | APE10-dist-in | 5.116 | APE9-dist-in | 3.713 | R250G | SEP261 | SEP261 | XRAY | 1.95 | 0.167 | 0.201 | A | 313 | 273 | 0 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 8r0w | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 1.5e-64 | 223.7 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CAMK | PIM1 | PIM1_HUMAN | 8AFRA | P11309 | 33 | 305 | 313.0 | M0F:401 | Type1 | Active | DFGin | 6.024 | 14.406 | BLAminus | -126.46, 177.16 | 55.61, 83.44 | -89.48, 19.88 | 284.93, 74.96 | -67.33, -13.52 | in-in | in | 8.831 | Saltbr-in | 2.648 | HRD-na-A | -72.52, -48.51 | 66.56, 10.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.815 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.4, 19.87 | APE9-dihe-na | -78.39, -149.93 | APE8-dihe-in | -97.85, 123.61 | APE8-rot-in | 301.25 | APE67-dihe-in | -68.16, -10.25 | -64.9, -40.75 | APE12-dist-in | 9.727 | APE11-dist-in | 8.467 | APE10-dist-in | 5.304 | APE9-dist-in | 3.645 | R250G | SEP261 | SEP261 | XRAY | 2.15 | 0.166 | 0.191 | A | 309 | 264 | 7 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 8afr | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 3.1e-62 | 216.2 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CMGC | CDK12 | CDK12_HUMAN | 8BU5B | Q9NYV4 | 713 | 1044 | 1490.0 | RMF:1101 | Type1 | Inactive | DFGin | 6.801 | 14.701 | ABAminus | -126.95, -66.04 | -93.95, 105.24 | -102.41, 30.18 | 293.69, 100.66 | -84.84, -22.58 | in-out | in | 8.305 | Saltbr-out | 3.933 | HRD-out | -78.59, 106.12 | -94.17, 5.74 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.828 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -136.91, -22.25 | APE9-dihe-na | -109.89, 157.52 | APE8-dihe-in | -56.01, 131.78 | APE8-rot-in | 308.02 | APE67-dihe-in | -60.99, -26.61 | -52.03, -40.26 | APE12-dist-out | 14.28 | APE11-dist-in | 11.941 | APE10-dist-in | 7.36 | APE9-dist-in | 3.767 | K965R | TPO893 | TPO893 | XRAY | 3.134 | 0.2 | 0.22 | B | 344 | 332 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bu5 | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BU5H | Q9NYV4 | 713 | 1043 | 1490.0 | RMF:1101 | Type1 | Inactive | DFGin | 7.015 | 14.978 | ABAminus | -128.46, -54.53 | -90.71, 103.12 | -97.22, 31.8 | 290.43, 81.59 | -85.33, -25.69 | in-in | in | 8.479 | Saltbr-in | 3.527 | HRD-in | -73.55, -49.58 | 63.85, -4.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.629 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.5, -28.02 | APE9-dihe-na | -97.36, 153.71 | APE8-dihe-in | -57.72, 135.61 | APE8-rot-in | 311.07 | APE67-dihe-in | -63.38, -27.52 | -50.57, -39.59 | APE12-dist-in | 13.941 | APE11-dist-in | 12.128 | APE10-dist-in | 7.258 | APE9-dist-in | 3.497 | K965R | TPO893 | TPO893 | XRAY | 3.134 | 0.2 | 0.22 | H | 344 | 331 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bu5 | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BUNB | Q9NYV4 | 715 | 1041 | 1490.0 | RNF:61101 | Type1 | Inactive | DFGin | 7.009 | 15.297 | ABAminus | -131.36, -49.43 | -89.83, 91.44 | -92.44, 32.63 | 287.3, 77.5 | -75.27, -18.22 | in-in | in | 7.748 | Saltbr-in | 3.279 | HRD-in | -75.67, -53.71 | 75.4, -0.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.923 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.12, -39.12 | APE9-dihe-na | -104.98, 151.97 | APE8-dihe-in | -58.93, 142.91 | APE8-rot-in | 279.94 | APE67-dihe-in | -65.42, -33.6 | -55.06, -35.14 | APE12-dist-in | 13.388 | APE11-dist-in | 11.695 | APE10-dist-in | 7.099 | APE9-dist-in | 3.657 | K965R | TPO893 | TPO893 | XRAY | 3.08 | 0.187 | 0.211 | B | 344 | 327 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bun | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BUNH | Q9NYV4 | 715 | 1043 | 1490.0 | RNF:61101 | Type1 | Inactive | DFGin | 7.045 | 15.286 | ABAminus | -125.24, -50.09 | -100.69, 94.75 | -92.24, 30.97 | 286.18, 71.82 | -75.42, -18.26 | in-in | in | 7.834 | Saltbr-in | 3.373 | HRD-in | -77.6, -54.36 | 73.0, -1.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.74 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.56, -41.65 | APE9-dihe-na | -95.79, 153.05 | APE8-dihe-in | -58.87, 144.43 | APE8-rot-in | 305.25 | APE67-dihe-in | -65.98, -31.29 | -55.83, -37.71 | APE12-dist-in | 13.775 | APE11-dist-in | 11.972 | APE10-dist-in | 6.957 | APE9-dist-in | 3.478 | K965R | TPO893 | TPO893 | XRAY | 3.08 | 0.187 | 0.211 | H | 344 | 329 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bun | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 9FMRE | Q9NYV4 | 714 | 1042 | 1490.0 | RMF:61101 | Type1 | Inactive | DFGin | 6.793 | 14.64 | ABAminus | -113.83, -79.52 | -84.15, 118.47 | -115.27, 16.16 | 293.54, 100.02 | -64.02, -34.33 | in-out | in | 9.633 | Saltbr-out | 3.612 | HRD-out | -79.17, 82.22 | -59.96, 8.89 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.026 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -148.14, -27.51 | APE9-dihe-na | -104.44, 148.12 | APE8-dihe-in | -51.45, 137.55 | APE8-rot-in | 306.02 | APE67-dihe-in | -70.5, -21.3 | -54.61, -36.19 | APE12-dist-out | 14.298 | APE11-dist-in | 12.211 | APE10-dist-in | 7.469 | APE9-dist-in | 3.767 | None | TPO893 | TPO893 | XRAY | 3.9 | 0.209 | 0.25 | E | 351 | 329 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 9fmr | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 9FMRH | Q9NYV4 | 714 | 1044 | 1490.0 | RMF:61101 | Type1 | Inactive | DFGin | 6.801 | 14.603 | ABAminus | -113.95, -78.4 | -84.85, 124.02 | -118.87, 17.95 | 291.29, 89.7 | -63.88, -35.4 | in-in | in | 8.592 | Saltbr-in | 3.552 | HRD-in | -72.47, -40.65 | 59.82, 5.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.74, -27.71 | APE9-dihe-na | -103.25, 148.34 | APE8-dihe-in | -51.07, 136.63 | APE8-rot-in | 306.14 | APE67-dihe-in | -69.99, -21.15 | -54.39, -34.8 | APE12-dist-in | 13.823 | APE11-dist-in | 12.098 | APE10-dist-in | 7.255 | APE9-dist-in | 3.608 | None | TPO893 | TPO893 | XRAY | 3.9 | 0.209 | 0.25 | H | 351 | 331 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 9fmr | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BUNE | Q9NYV4 | 715 | 1039 | 1490.0 | RNF:61101 | Type1 | Inactive | DFGin | 7.217 | 15.313 | BLAminus | -143.55, -179.06 | 50.55, 77.42 | -92.12, 34.85 | 285.27, 76.47 | -72.26, -18.51 | in-in | in | 7.824 | Saltbr-in | 3.046 | HRD-in | -77.13, -53.65 | 75.0, -0.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.924 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -105.31, -34.23 | APE9-dihe-na | -92.08, 151.91 | APE8-dihe-in | -57.84, 145.99 | APE8-rot-out | 175.35 | APE67-dihe-in | -65.98, -29.37 | -55.72, -38.5 | APE12-dist-in | 13.18 | APE11-dist-in | 12.611 | APE10-dist-in | 7.008 | APE9-dist-in | 3.432 | K965R | TPO893 | TPO893 | XRAY | 3.08 | 0.187 | 0.211 | E | 344 | 325 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bun | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8P81A | Q9NYV4 | 716 | 1035 | 1490.0 | RMF:1101 | Type1 | Active | DFGin | 7.095 | 14.446 | BLAminus | -134.83, -178.64 | 59.2, 72.19 | -89.53, 34.88 | 291.56, 80.44 | -67.97, -22.73 | in-in | in | 8.359 | Saltbr-in | 3.057 | HRD-in | -81.5, -42.97 | 59.01, 18.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.963 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.63, 165.61 | APE9-dihe-na | 67.08, 139.25 | APE8-dihe-in | -61.99, 152.33 | APE8-rot-in | 316.49 | APE67-dihe-in | -68.12, -20.85 | -57.98, -41.98 | APE12-dist-in | 12.679 | APE11-dist-in | 10.561 | APE10-dist-in | 6.52 | APE9-dist-in | 3.212 | None | TPO893 | TPO893 | XRAY | 2.68 | 0.212 | 0.255 | A | 351 | 320 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8p81 | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 8BU5E | Q9NYV4 | 713 | 1043 | 1490.0 | RMF:1101 | Type1 | Inactive | DFGin | 6.942 | 15.122 | None | -123.64, -63.66 | -81.97, -51.09 | 56.28, 22.54 | 292.49, 98.9 | -91.33, -28.22 | in-out | in | 8.371 | Saltbr-out | 3.622 | HRD-in | -72.77, -54.57 | 74.45, -4.91 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.759 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -134.16, -27.33 | APE9-dihe-na | -98.05, 157.33 | APE8-dihe-in | -51.55, 136.25 | APE8-rot-in | 308.17 | APE67-dihe-in | -63.16, -26.85 | -49.17, -41.17 | APE12-dist-out | 14.125 | APE11-dist-in | 12.168 | APE10-dist-in | 7.286 | APE9-dist-in | 3.726 | K965R | TPO893 | TPO893 | XRAY | 3.134 | 0.2 | 0.22 | E | 344 | 331 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 8bu5 | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 5.4e-84 | 287.9 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK12 | CDK12_HUMAN | 9FMRB | Q9NYV4 | 714 | 1047 | 1490.0 | RMF:61101 | Type1 | Inactive | DFGin | 7.124 | 15.031 | None | -111.49, -74.26 | -77.99, -72.15 | 68.85, 12.84 | 296.16, 89.8 | -66.22, -36.51 | in-out | in | 8.332 | Saltbr-out | 4.45 | HRD-in | -70.8, -35.56 | 62.81, 1.22 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.072 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.03, -25.75 | APE9-dihe-na | -103.56, 146.88 | APE8-dihe-in | -51.72, 138.27 | APE8-rot-in | 305.58 | APE67-dihe-in | -69.51, -21.36 | -53.61, -35.19 | APE12-dist-in | 13.987 | APE11-dist-in | 12.27 | APE10-dist-in | 7.331 | APE9-dist-in | 3.865 | None | TPO893 | TPO893 | XRAY | 3.9 | 0.209 | 0.25 | B | 351 | 334 | 0 | 0 | 0 | 0 | [[727, 1020]] | 1.0 | 9fmr | Homo sapiens | CMGC_CDK12_HUMAN | CMGC | 2.9e-84 | 288.8 | 1 | 301 | 301 | 876 | 877 | 878 | 880 | 882 | 756 | 774 | 778 | 856 | 858 | 857 | 859 | 918 | 905 | 900 | 899 | 898 | 897 | 896 | 895 | 894 | 814 | Cyclin-dependent kinase 12 |
| CMGC | CDK16 | CDK16_HUMAN | 3MTLA | Q00536 | 163 | 473 | 496.0 | FEF:60668 | Type1 | Inactive | DFGout | 17.399 | 7.472 | None | -75.13, 154.32 | -88.9, 77.74 | -154.62, 116.54 | 227.56, 88.74 | 78.03, 21.89 | in-in | in | 8.385 | Saltbr-in | 2.641 | HRD-out | -101.69, 108.56 | -74.19, -25.04 | in-out-out | SNCioo | out-out | ActLoopNT-out | 5.164 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 102.89 | APE8-rot-out | 156.53 | APE67-dihe-in | -61.54, -35.29 | -78.56, -14.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | S319D | None | None | XRAY | 2.4 | 0.198 | 0.263 | A | 324 | 293 | 18 | 0 | 0 | 12 | [[165, 446]] | 1.0 | 3mtl | Homo sapiens | CMGC_CDK16_HUMAN | CMGC | 1.3e-83 | 286.9 | 1 | 301 | 301 | 303 | 304 | 305 | 307 | 309 | 194 | 211 | 215 | 283 | 285 | 284 | 286 | 344 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 241 | Cyclin-dependent kinase 16 |
| CMGC | CDK2 | CDK2_HUMAN | 9ESWA | P24941 | 1 | 294 | 298.0 | IJF:60301,IJF:60302,IJF:60303,IJF:60304 | Allosteric,Type1,Allosteric,Allosteric | Active | DFGin | 6.515 | 15.297 | BLAminus | -143.94, 174.07 | 58.52, 82.55 | -94.4, 25.35 | 278.47, 68.95 | -74.76, -22.16 | in-in | in | 8.637 | Saltbr-in | 3.197 | HRD-in | -81.26, -58.57 | 77.56, 16.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.996 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -61.44, 160.94 | APE9-dihe-na | 81.67, 126.4 | APE8-dihe-in | -51.25, 136.17 | APE8-rot-in | 300.7 | APE67-dihe-in | -59.48, -16.12 | -52.59, -48.63 | APE12-dist-in | 12.997 | APE11-dist-in | 11.897 | APE10-dist-in | 7.023 | APE9-dist-in | 3.204 | None | TPO160 | TPO160 | XRAY | 2.38 | 0.233 | 0.239 | A | 302 | 294 | 0 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 9esw | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.7e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 9ESWC | P24941 | 1 | 296 | 298.0 | IJF:60301,IJF:60302,IJF:60303,IJF:60304 | Allosteric,Type1,Allosteric,Allosteric | Active | DFGin | 6.576 | 15.209 | BLAminus | -137.9, -176.23 | 48.55, 71.41 | -85.05, 25.18 | 283.44, 66.65 | -62.35, -32.95 | in-in | in | 8.417 | Saltbr-in | 2.763 | HRD-in | -83.58, -58.72 | 75.84, 9.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.887 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.32, 151.2 | APE9-dihe-na | 72.23, 131.64 | APE8-dihe-in | -58.77, 140.82 | APE8-rot-in | 312.4 | APE67-dihe-in | -51.92, -26.23 | -42.04, -57.02 | APE12-dist-in | 12.776 | APE11-dist-in | 10.195 | APE10-dist-in | 6.943 | APE9-dist-in | 3.236 | None | TPO160 | TPO160 | XRAY | 2.38 | 0.233 | 0.239 | C | 302 | 269 | 27 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 9esw | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.7e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 9OB4A | P24941 | 1 | 298 | 298.0 | A1CAF:301 | Type1 | Active | DFGin | 7.07 | 15.433 | BLAminus | -140.78, 171.16 | 58.81, 81.21 | -94.48, 18.25 | 279.35, 70.51 | -60.63, -24.89 | in-in | in | 8.702 | Saltbr-in | 2.578 | HRD-in | -77.49, -52.8 | 70.85, 9.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.858 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -103.4, 171.78 | APE9-dihe-na | 71.79, 138.58 | APE8-dihe-in | -59.97, 144.28 | APE8-rot-in | 298.9 | APE67-dihe-in | -65.05, -23.77 | -53.99, -47.04 | APE12-dist-in | 13.149 | APE11-dist-in | 12.232 | APE10-dist-in | 7.357 | APE9-dist-in | 3.261 | None | TPO160 | TPO160 | XRAY | 1.95 | 0.211 | 0.251 | A | 301 | 298 | 0 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 9ob4 | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.6e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 4BCQA | P24941 | 1 | 295 | 298.0 | TJF:61296 | Type1 | Active | DFGin | 6.591 | 15.979 | BLAminus | -145.97, 170.46 | 62.82, 84.99 | -99.38, 29.59 | 282.23, 71.6 | -71.19, -18.61 | in-in | in | 9.404 | Saltbr-in | 3.453 | HRD-in | -85.05, -58.94 | 78.36, 12.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.147 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.8, 176.97 | APE9-dihe-na | 69.33, 133.29 | APE8-dihe-in | -55.38, 139.69 | APE8-rot-in | 304.09 | APE67-dihe-in | -55.84, -22.0 | -49.63, -50.65 | APE12-dist-in | 13.625 | APE11-dist-in | 12.543 | APE10-dist-in | 7.498 | APE9-dist-in | 3.511 | None | TPO160 | TPO160 | XRAY | 2.4 | 0.217 | 0.252 | A | 301 | 290 | 5 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 4bcq | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.6e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 4BCQC | P24941 | 1 | 294 | 298.0 | TJF:61295 | Type1 | Active | DFGin | 6.54 | 16.003 | BLAminus | -147.36, 170.23 | 59.21, 86.27 | -98.9, 28.16 | 278.44, 72.82 | -71.37, -12.42 | in-in | in | 9.598 | Saltbr-in | 3.261 | HRD-in | -88.13, -59.99 | 74.18, 19.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.909 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.48, 157.26 | APE9-dihe-na | 69.58, 129.95 | APE8-dihe-in | -57.66, 135.49 | APE8-rot-in | 301.27 | APE67-dihe-in | -62.84, -20.05 | -48.44, -46.81 | APE12-dist-in | 13.54 | APE11-dist-in | 10.682 | APE10-dist-in | 7.689 | APE9-dist-in | 3.66 | None | TPO160 | TPO160 | XRAY | 2.4 | 0.217 | 0.252 | C | 301 | 292 | 2 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 4bcq | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.6e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 7S9XA | P24941 | 3 | 298 | 298.0 | 8KF:301 | Type3 | Inactive | DFGin | 9.152 | 14.904 | BLBminus | -140.51, 174.83 | 55.24, 52.61 | -60.52, 155.06 | 283.44, 65.83 | -96.54, 51.03 | out-out | out | 17.021 | Saltbr-out | 17.405 | HRD-in | -80.98, -57.39 | 84.63, -18.55 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.299 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, 131.76 | APE9-dihe-na | -82.0, 133.39 | APE8-dihe-in | -82.83, 123.04 | APE8-rot-in | 299.71 | APE67-dihe-in | -59.76, -23.84 | -102.49, -0.32 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.12 | APE9-dist-out | 11.022 | None | None | None | XRAY | 1.69 | 0.231 | 0.262 | A | 298 | 269 | 27 | 0 | 0 | 12 | [[4, 286]] | 1.0 | 7s9x | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.3e-90 | 307.9 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 2W1HA | P24941 | 1 | 298 | 298.0 | L0F:1299 | Type1 | Inactive | DFGin | 10.307 | 17.775 | BLBtrans | -130.06, 151.5 | 79.56, 18.75 | -69.93, 141.61 | 226.73, 121.67 | 69.65, -12.05 | out-out | out | 14.489 | Saltbr-out | 16.038 | HRD-in | -88.39, -56.31 | 79.17, -16.22 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.457 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 121.46 | APE8-dihe-in | -76.22, 142.93 | APE8-rot-out | 186.46 | APE67-dihe-in | -49.35, -36.85 | -110.85, -4.12 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.805 | None | None | None | XRAY | 2.15 | 0.263 | 0.308 | A | 298 | 283 | 15 | 0 | 0 | 11 | [[4, 286]] | 1.0 | 2w1h | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.3e-90 | 307.9 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 2R3IA | P24941 | 1 | 298 | 298.0 | SCF:60501 | Type1 | Inactive | DFGin | 10.929 | 18.24 | BLBtrans | -100.61, 149.54 | 71.45, 21.63 | -58.2, 134.86 | 231.09, 103.4 | 83.18, -10.48 | out-out | out | 15.057 | Saltbr-out | 16.345 | HRD-in | -91.01, -59.76 | 82.13, -15.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.707 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -70.45, 127.61 | APE9-dihe-na | -74.97, 122.45 | APE8-dihe-in | -60.32, 144.67 | APE8-rot-out | 191.76 | APE67-dihe-in | -59.78, -26.25 | -99.25, -5.87 | APE12-dist-out | 20.169 | APE11-dist-out | 17.538 | APE10-dist-out | 18.889 | APE9-dist-out | 9.991 | None | None | CSD177 | XRAY | 1.28 | 0.178 | 0.202 | A | 299 | 291 | 7 | 0 | 0 | 0 | [[4, 286]] | 1.0 | 2r3i | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.4e-90 | 307.8 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK2 | CDK2_HUMAN | 5IEXA | P24941 | 1 | 298 | 298.0 | 6AF:1001 | Type1 | Inactive | None | 11.106 | 18.344 | None | -105.6, 149.53 | 71.37, 22.65 | -61.85, 135.15 | 236.62, 103.3 | 74.49, -10.58 | out-out | out | 15.176 | Saltbr-out | 15.226 | HRD-in | -80.72, -65.3 | 84.99, -26.41 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.802 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 111.81 | APE8-dihe-in | -112.57, 117.73 | APE8-rot-in | 277.98 | APE67-dihe-in | -67.92, -29.52 | -99.02, -2.25 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.275 | None | None | None | XRAY | 2.03 | 0.206 | 0.254 | A | 298 | 285 | 13 | 0 | 0 | 8 | [[4, 286]] | 1.0 | 5iex | Homo sapiens | CMGC_CDK2_HUMAN | CMGC | 6.3e-90 | 307.9 | 1 | 301 | 301 | 144 | 145 | 146 | 148 | 150 | 33 | 51 | 55 | 124 | 126 | 125 | 127 | 185 | 172 | 167 | 166 | 165 | 164 | 163 | 162 | 161 | 81 | Cyclin-dependent kinase 2 |
| CMGC | CDK6 | CDK6_HUMAN | 9PE7A | Q00534 | 10 | 301 | 326.0 | A1CIF:900 | Type1 | Inactive | DFGin | 6.872 | 13.127 | BLBplus | -137.4, 169.29 | 57.4, 61.63 | -142.77, 164.35 | 61.09, 86.59 | 91.92, -16.71 | out-out | out | 12.416 | Saltbr-out | 9.93 | HRD-in | -63.73, -52.58 | 73.19, -16.54 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, 162.46 | APE9-dihe-na | -100.9, 174.34 | APE8-dihe-in | -134.69, 96.5 | APE8-rot-in | 306.93 | APE67-dihe-in | -54.43, -27.6 | -93.0, -5.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 22.373 | APE9-dist-out | 12.123 | E21V,K26T,T106R,Q149E | None | None | XRAY | 2.05 | 0.216 | 0.267 | A | 307 | 262 | 30 | 0 | 0 | 12 | [[13, 300]] | 1.0 | 9pe7 | Homo sapiens | CMGC_CDK6_HUMAN | CMGC | 3.7e-84 | 289.5 | 1 | 301 | 301 | 162 | 163 | 164 | 166 | 168 | 43 | 61 | 65 | 142 | 144 | 143 | 145 | 201 | 189 | 184 | 183 | 182 | 181 | 180 | 179 | 178 | 99 | Cyclin-dependent kinase 6 |
| CMGC | CDK7 | CDK7_HUMAN | 8P71J | P50613 | 10 | 310 | 346.0 | X4F:60401 | Type1 | Active | DFGin | 6.832 | 15.304 | BLAminus | -139.46, 179.9 | 57.59, 64.02 | -82.45, 17.71 | 282.17, 74.47 | -64.72, -19.22 | in-in | in | 8.103 | Saltbr-in | 2.694 | HRD-in | -67.33, -49.46 | 65.63, 5.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.639 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.68, 168.49 | APE9-dihe-na | 67.33, 140.05 | APE8-dihe-in | -60.3, 143.93 | APE8-rot-in | 294.53 | APE67-dihe-in | -61.0, -25.19 | -55.87, -41.76 | APE12-dist-in | 13.411 | APE11-dist-in | 11.192 | APE10-dist-in | 6.803 | APE9-dist-in | 3.276 | None | None | None | EM | 2.0 | 999.0 | 999.0 | J | 349 | 286 | 15 | 0 | 0 | 0 | [[12, 295]] | 1.0 | 8p71 | Homo sapiens | CMGC_CDK7_HUMAN | CMGC | 1.6e-78 | 271.7 | 1 | 301 | 301 | 154 | 155 | 156 | 158 | 160 | 41 | 62 | 66 | 134 | 136 | 135 | 137 | 195 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Cyclin-dependent kinase 7 |
| CMGC | CDK8 | CDK8_HUMAN | 9H8SA | P49336 | 1 | 362 | 464.0 | A1ITF:60509 | Type1 | Inactive | DFGin | 7.344 | 13.924 | BLAminus | -119.28, 163.44 | 74.84, 82.25 | -92.61, 11.91 | 298.93, 132.0 | -87.41, 10.8 | in-in | in | 8.612 | Saltbr-in | 2.624 | HRD-in | -75.25, -51.5 | 79.06, -6.52 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.659 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 160.05 | APE8-rot-out | 75.96 | APE67-dihe-in | -54.19, -23.95 | -111.96, 19.45 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.157 | 0.197 | 0.248 | A | 414 | 335 | 27 | 0 | 0 | 17 | [[22, 335]] | 1.0 | 9h8s | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 6.3e-82 | 281.3 | 5 | 301 | 297 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 8AEMA | P68400 | 3 | 329 | 391.0 | LVF:407,ATP:408 | Allosteric,ATPlike | Active | DFGin | 7.399 | 16.187 | BLAminus | -114.2, -178.47 | 56.21, 75.05 | -90.39, 15.9 | 296.69, 81.8 | -66.43, -20.83 | in-in | in | 9.132 | Saltbr-in | 2.816 | HRD-in | -72.91, -51.16 | 68.69, 11.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.905 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.83, 169.06 | APE9-dihe-na | 58.87, 157.76 | APE8-dihe-in | -77.1, 150.54 | APE8-rot-in | 294.73 | APE67-dihe-in | -68.78, -13.55 | -40.19, -53.95 | APE12-dist-in | 12.744 | APE11-dist-in | 10.417 | APE10-dist-in | 6.256 | APE9-dist-in | 3.215 | R21S,K74A,K75A,K76A | None | None | XRAY | 1.6 | 0.19 | 0.212 | A | 328 | 327 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 8aem | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 8.1e-69 | 238.0 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9EPWB | P68400 | 3 | 333 | 391.0 | A1H6F:406 | Type1 | Active | DFGin | 7.386 | 16.279 | BLAminus | -118.5, 178.76 | 54.91, 76.82 | -86.63, 13.68 | 291.49, 81.55 | -67.5, -20.83 | out-in | out | 10.046 | Saltbr-in | 3.292 | HRD-in | -71.7, -52.07 | 70.7, 14.03 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.882 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.62, 167.98 | APE9-dihe-na | 70.49, 159.89 | APE8-dihe-in | -76.41, 141.74 | APE8-rot-in | 289.66 | APE67-dihe-in | -68.82, -20.3 | -42.56, -42.98 | APE12-dist-in | 12.795 | APE11-dist-in | 10.921 | APE10-dist-in | 6.279 | APE9-dist-in | 3.382 | None | None | None | XRAY | 2.3 | 0.261 | 0.308 | B | 338 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9epw | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.4e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 2ZJWA | P68400 | 1 | 332 | 391.0 | REF:336 | Type1 | Inactive | DFGin | 7.316 | 16.527 | BLAminus | -109.16, -168.7 | 44.38, 76.01 | -90.89, 24.26 | 297.46, 77.89 | -76.15, -7.13 | in-in | in | 9.417 | Saltbr-in | 2.731 | HRD-in | -72.0, -50.11 | 70.44, 13.49 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.907 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -14.58, 161.89 | APE9-dihe-na | 62.59, 163.98 | APE8-dihe-in | -84.5, 146.1 | APE8-rot-out | 153.88 | APE67-dihe-in | -63.0, -17.21 | -40.84, -52.94 | APE12-dist-in | 12.607 | APE11-dist-in | 8.948 | APE10-dist-in | 5.933 | APE9-dist-in | 2.992 | None | None | None | XRAY | 2.4 | 0.222 | 0.274 | A | 340 | 332 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 2zjw | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.4e-69 | 240.5 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 7I8AA | P68400 | 3 | 329 | 391.0 | A1B0F:401 | Type1 | Active | DFGin | 7.457 | 16.071 | BLAminus | -110.77, 179.22 | 49.98, 83.2 | -97.8, 27.66 | 295.37, 80.49 | -74.55, -21.62 | in-in | in | 8.964 | Saltbr-in | 2.748 | HRD-in | -69.35, -49.91 | 66.48, 13.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.27, 172.69 | APE9-dihe-na | 60.01, 160.49 | APE8-dihe-in | -88.34, 150.2 | APE8-rot-in | 298.89 | APE67-dihe-in | -68.6, -15.9 | -36.65, -52.88 | APE12-dist-in | 12.62 | APE11-dist-in | 10.174 | APE10-dist-in | 6.101 | APE9-dist-in | 3.048 | R21S,K74A,K75A,K76A | None | None | XRAY | 1.84 | 0.196 | 0.234 | A | 328 | 323 | 4 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 7i8a | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 8.1e-69 | 238.0 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | DYRK1A | DYR1A_HUMAN | 6A1FA | Q13627 | 134 | 483 | 763.0 | 9OF:807 | Type1 | Active | DFGin | 7.205 | 15.092 | BLAminus | -125.52, 173.04 | 69.56, 79.06 | -100.37, 18.23 | 289.23, 81.85 | -66.74, -28.25 | in-in | in | 8.712 | Saltbr-in | 2.843 | HRD-in | -63.72, -44.37 | 75.39, -2.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.826 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.51, 164.33 | APE9-dihe-na | 78.19, 142.16 | APE8-dihe-in | -71.23, 146.24 | APE8-rot-in | 287.31 | APE67-dihe-in | -64.89, -24.24 | -54.81, -45.1 | APE12-dist-in | 13.001 | APE11-dist-in | 10.937 | APE10-dist-in | 7.397 | APE9-dist-in | 3.189 | None | PTR321 | PTR321 | XRAY | 1.5 | 0.178 | 0.195 | A | 360 | 346 | 4 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 6a1f | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 8.3e-91 | 310.2 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK2 | DYRK2_HUMAN | 7DH9A | Q92630 | 215 | 538 | 601.0 | H7F:601 | Type1 | Inactive | DFGin | 6.955 | 15.393 | BLAminus | -118.25, -176.44 | 52.33, 72.66 | -86.4, 22.32 | 285.5, 71.17 | -68.46, -16.6 | in-in | in | 9.091 | Saltbr-in | 2.818 | HRD-in | -67.52, -48.86 | 77.78, -1.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.826 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.21, 165.64 | APE9-dihe-na | 77.26, 152.01 | APE8-dihe-in | -71.35, 136.19 | APE8-rot-out | 186.16 | APE67-dihe-in | -56.24, -27.47 | -53.15, -48.91 | APE12-dist-in | 13.085 | APE11-dist-in | 11.935 | APE10-dist-in | 7.588 | APE9-dist-in | 3.308 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.194 | 0.19 | 0.218 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dh9 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| CMGC | GSK3B | GSK3B_HUMAN | 9PE9A | P49841 | 36 | 382 | 420.0 | A1CIF:900 | Type1 | Inactive | DFGin | 7.072 | 14.229 | BLAminus | -128.7, -179.96 | 59.31, 84.1 | -97.11, 26.91 | 283.64, 74.63 | -73.69, -18.15 | in-in | in | 8.351 | Saltbr-in | 2.725 | HRD-in | -68.62, -45.57 | 65.7, 16.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.925 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -143.94, 165.33 | APE9-dihe-na | 76.34, 152.28 | APE8-dihe-in | -69.82, 130.62 | APE8-rot-out | 176.66 | APE67-dihe-in | -58.68, -26.71 | -39.69, -56.4 | APE12-dist-in | 13.28 | APE11-dist-in | 11.758 | APE10-dist-in | 7.093 | APE9-dist-in | 3.155 | None | PTR216 | PTR216 | XRAY | 2.11 | 0.221 | 0.247 | A | 359 | 332 | 13 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 9pe9 | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 9PE9B | P49841 | 36 | 382 | 420.0 | A1CIF:900 | Type1 | Inactive | DFGin | 7.058 | 14.218 | BLAminus | -128.76, -179.81 | 59.6, 84.42 | -97.78, 27.09 | 283.79, 74.38 | -73.25, -17.71 | in-in | in | 8.353 | Saltbr-in | 2.713 | HRD-in | -68.49, -44.82 | 64.55, 18.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.94 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -144.27, 163.74 | APE9-dihe-na | 77.64, 152.05 | APE8-dihe-in | -69.14, 130.82 | APE8-rot-out | 177.12 | APE67-dihe-in | -58.92, -26.81 | -39.96, -55.88 | APE12-dist-in | 13.36 | APE11-dist-in | 11.824 | APE10-dist-in | 7.161 | APE9-dist-in | 3.172 | None | PTR216 | PTR216 | XRAY | 2.11 | 0.221 | 0.247 | B | 359 | 332 | 13 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 9pe9 | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 4PTEA | P49841 | 36 | 382 | 420.0 | 2WF:501 | Type1 | Active | DFGin | 6.932 | 14.017 | BLAminus | -141.21, 178.04 | 57.99, 89.39 | -100.23, 24.26 | 286.38, 75.9 | -68.08, -19.02 | in-in | in | 8.716 | Saltbr-in | 2.635 | HRD-in | -73.56, -44.45 | 69.11, 4.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.792 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.74, 175.98 | APE9-dihe-na | 75.98, 148.82 | APE8-dihe-in | -103.79, 152.51 | APE8-rot-in | 295.33 | APE67-dihe-inflip | 95.08, -28.26 | -38.95, 126.56 | APE12-dist-in | 12.979 | APE11-dist-in | 10.89 | APE10-dist-in | 5.883 | APE9-dist-in | 3.088 | None | None | None | XRAY | 2.033 | 0.17 | 0.195 | A | 441 | 341 | 6 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 4pte | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 3.7e-70 | 242.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 4PTEB | P49841 | 36 | 385 | 420.0 | 2WF:501 | Type1 | Active | DFGin | 6.918 | 13.937 | BLAminus | -137.07, 179.43 | 58.52, 88.98 | -101.38, 27.88 | 284.28, 76.88 | -69.85, -20.65 | in-in | in | 8.484 | Saltbr-in | 2.685 | HRD-in | -70.9, -46.61 | 73.05, 2.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.887 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -87.76, 178.59 | APE9-dihe-na | 72.73, 147.77 | APE8-dihe-in | -103.48, 150.66 | APE8-rot-in | 296.89 | APE67-dihe-inflip | 94.67, -27.57 | -36.66, 125.81 | APE12-dist-in | 12.935 | APE11-dist-in | 10.88 | APE10-dist-in | 5.877 | APE9-dist-in | 3.154 | None | None | None | XRAY | 2.033 | 0.17 | 0.195 | B | 441 | 347 | 3 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 4pte | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 3.7e-70 | 242.6 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | MAPK1 | MK01_HUMAN | 5BVDA | P28482 | 9 | 358 | 360.0 | 4VF:60401 | Type1 | None | DFGin | 7.012 | 14.82 | BLAminus | -120.88, -174.96 | 58.49, 83.25 | -99.87, 23.43 | 283.53, 71.8 | -56.85, -34.73 | in-in | in | 9.264 | Saltbr-in | 2.627 | HRD-in | -80.64, -49.81 | 78.16, -6.37 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.72 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 122.19 | APE8-rot-in | 306.38 | APE67-dihe-in | -62.44, -24.22 | -51.26, -49.02 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.9 | 0.172 | 0.207 | A | 361 | 330 | 20 | 0 | 0 | 16 | [[25, 313]] | 1.0 | 5bvd | Homo sapiens | CMGC_MAPK1_HUMAN | CMGC | 9.2e-86 | 293.7 | 1 | 301 | 301 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 8AO6A | P28482 | 11 | 356 | 360.0 | N9F:406 | Type1 | Inactive | DFGin | 6.771 | 16.337 | BLAminus | -129.81, 177.88 | 71.62, 78.81 | -103.22, 23.44 | 283.23, 73.97 | -64.0, -29.38 | out-in | out | 10.371 | Saltbr-in | 2.597 | HRD-in | -72.45, -50.74 | 72.14, 4.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.785 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -96.92, -36.24 | APE9-dihe-na | -66.98, 156.39 | APE8-dihe-in | -51.35, 125.27 | APE8-rot-in | 311.93 | APE67-dihe-in | -64.42, -17.18 | -56.32, -47.54 | APE12-dist-out | 14.414 | APE11-dist-in | 11.107 | APE10-dist-in | 7.103 | APE9-dist-in | 4.264 | None | None | CME127,CME161 | XRAY | 1.811 | 0.175 | 0.222 | A | 368 | 338 | 0 | 0 | 0 | 0 | [[25, 313]] | 1.0 | 8ao6 | Homo sapiens | CMGC_MAPK1_HUMAN | CMGC | 9.9e-86 | 293.6 | 1 | 301 | 301 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_HUMAN | 8AO9A | P28482 | 11 | 356 | 360.0 | N4F:406 | Type1 | Inactive | DFGin | 6.837 | 16.45 | BLAminus | -129.5, 178.83 | 61.88, 81.37 | -96.97, 21.21 | 286.14, 78.83 | -59.7, -30.7 | out-out | out | 10.301 | Saltbr-out | 3.765 | HRD-in | -72.95, -49.65 | 72.84, 3.98 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.854 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -91.06, -44.4 | APE9-dihe-na | -60.28, 156.59 | APE8-dihe-in | -55.09, 130.24 | APE8-rot-in | 307.62 | APE67-dihe-in | -64.58, -17.09 | -62.44, -44.52 | APE12-dist-out | 14.27 | APE11-dist-in | 10.981 | APE10-dist-in | 6.789 | APE9-dist-in | 4.23 | None | None | CME161 | XRAY | 1.624 | 0.184 | 0.232 | A | 368 | 338 | 2 | 0 | 0 | 0 | [[25, 313]] | 1.0 | 8ao9 | Homo sapiens | CMGC_MAPK1_HUMAN | CMGC | 9.9e-86 | 293.6 | 1 | 301 | 301 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK10 | MK10_HUMAN | 3CGFA | P53779 | 45 | 400 | 464.0 | JNF:523 | Type1 | Inactive | DFGin | 3.719 | 14.039 | ABAminus | -89.59, -53.32 | -106.99, -179.49 | -117.03, 20.53 | 309.75, 79.33 | 76.52, -162.79 | in-out | in | 9.602 | Saltbr-out | 3.611 | HRD-in | -43.19, -70.09 | 72.17, 4.64 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -63.93, 178.32 | APE9-dihe-na | -126.54, 145.54 | APE8-dihe-in | -86.07, 133.09 | APE8-rot-in | 307.62 | APE67-dihe-in | -51.07, -34.7 | -123.34, -6.64 | APE12-dist-out | 21.335 | APE11-dist-out | 17.893 | APE10-dist-out | 16.615 | APE9-dist-out | 11.474 | None | None | None | XRAY | 3.0 | 0.225 | 0.317 | A | 365 | 346 | 5 | 0 | 0 | 5 | [[64, 359]] | 1.0 | 3cgf | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.1 | 1 | 301 | 301 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 7YL1A | P53779 | 45 | 400 | 464.0 | J6F:501 | Type1 | Inactive | DFGin | 3.995 | 14.06 | ABAminus | -80.16, -27.18 | -141.36, 174.64 | -114.52, 17.98 | 302.24, 85.17 | 76.51, -161.32 | in-in | in | 9.23 | Saltbr-in | 2.755 | HRD-in | -85.09, -59.15 | 76.16, -2.31 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.441 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -89.31, 134.84 | APE9-dihe-na | -84.54, 138.55 | APE8-dihe-in | -77.28, 127.44 | APE8-rot-in | 291.87 | APE67-dihe-in | -54.76, -19.99 | -106.7, -13.11 | APE12-dist-out | 20.721 | APE11-dist-out | 15.877 | APE10-dist-out | 16.196 | APE9-dist-out | 11.273 | None | None | None | XRAY | 2.48 | 0.208 | 0.294 | A | 464 | 352 | 2 | 0 | 0 | 2 | [[64, 359]] | 1.0 | 7yl1 | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 3e-85 | 292.1 | 1 | 301 | 301 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK14 | MK14_HUMAN | 6ZQSA | Q16539 | 4 | 353 | 360.0 | 3FF:400 | Type1 | Inactive | DFGin | 7.131 | 15.007 | BLAminus | -100.05, 172.92 | 58.72, 89.64 | -100.69, 26.63 | 286.71, 76.86 | -66.14, -26.38 | out-out | out | 10.282 | Saltbr-out | 3.92 | HRD-in | -83.97, -53.39 | 74.81, 10.18 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.23, 173.02 | APE9-dihe-na | 73.87, 161.94 | APE8-dihe-in | -91.46, 139.33 | APE8-rot-in | 294.96 | APE67-dihe-in | -66.05, -18.45 | -53.95, -45.87 | APE12-dist-in | 11.599 | APE11-dist-in | 11.174 | APE10-dist-in | 6.771 | APE9-dist-in | 3.046 | None | TPO180,PTR182 | TPO180,PTR182 | XRAY | 1.95 | 0.178 | 0.223 | A | 362 | 350 | 0 | 0 | 0 | 0 | [[24, 308]] | 1.0 | 6zqs | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 5XYYA | Q16539 | 4 | 352 | 360.0 | P0F:401 | Type1.5_Back | Inactive | DFGin | 8.144 | 16.25 | BLBminus | -111.25, 174.05 | 61.59, 81.71 | -109.03, 145.8 | 286.82, 89.51 | 69.26, 21.62 | in-in | in | 8.942 | Saltbr-in | 2.649 | HRD-in | -68.14, -52.86 | 82.9, -10.64 | in-out-out | SNCioo | out-out | ActLoopNT-out | 11.476 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_oooo | APE10-dihe-na | -136.86, 131.59 | APE9-dihe-na | -62.4, -17.36 | APE8-dihe-out | -62.41, -19.09 | APE8-rot-out | 53.75 | APE67-dihe-in | -64.55, -20.22 | -114.48, -18.89 | APE12-dist-out | 21.139 | APE11-dist-out | 22.895 | APE10-dist-out | 17.093 | APE9-dist-out | 11.759 | None | None | None | XRAY | 1.7 | 0.18 | 0.201 | A | 380 | 343 | 6 | 0 | 0 | 0 | [[24, 308]] | 1.0 | 5xyy | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 7e-85 | 290.9 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 2QD9A | Q16539 | 5 | 352 | 360.0 | LGF:361 | Type1 | Inactive | DFGin | 5.134 | 13.797 | BLBplus | -108.86, 148.96 | 74.79, 24.8 | -73.05, 150.79 | 49.54, 82.76 | 82.07, 6.15 | in-in | in | 9.155 | Saltbr-in | 2.557 | HRD-in | -76.06, -55.95 | 78.8, -20.76 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -59.56, -22.52 | 999.0, -59.62 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.7 | 0.252 | 0.282 | A | 366 | 330 | 18 | 0 | 0 | 13 | [[24, 308]] | 1.0 | 2qd9 | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 6.2e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3QUDA | Q16539 | 4 | 354 | 360.0 | N3F:361 | Type1 | Inactive | DFGin | 10.801 | 12.553 | None | -93.66, 153.34 | -68.51, -47.3 | -136.82, 128.38 | 301.98, 103.1 | -95.02, -166.54 | in-in | in | 9.269 | Saltbr-in | 3.555 | HRD-in | -63.42, -58.28 | 80.41, -12.58 | in-out-out | SNCioo | out-out | ActLoopNT-out | 20.801 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, 112.75 | APE9-dihe-na | -76.37, 136.79 | APE8-dihe-out | -65.47, -38.0 | APE8-rot-in | 295.71 | APE67-dihe-in | -57.05, -26.46 | -56.48, -28.08 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 10.762 | APE9-dist-out | 12.652 | None | None | None | XRAY | 2.0 | 0.234 | 0.278 | A | 360 | 345 | 6 | 0 | 0 | 6 | [[24, 308]] | 1.0 | 3qud | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3QUEA | Q16539 | 5 | 353 | 360.0 | 3FF:362 | Type1 | Inactive | DFGin | 10.642 | 12.339 | None | -82.41, 155.86 | -75.27, -54.23 | -130.98, 134.23 | 308.77, 88.25 | -97.08, -170.31 | in-in | in | 8.96 | Saltbr-in | 2.657 | HRD-in | -64.83, -54.13 | 86.66, -27.06 | in-out-out | SNCioo | out-out | ActLoopNT-out | 21.279 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, 66.84 | APE9-dihe-na | -77.78, 135.56 | APE8-dihe-out | -48.89, -54.16 | APE8-rot-in | 280.74 | APE67-dihe-in | -53.38, -25.8 | -51.95, -34.65 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 9.195 | APE9-dist-out | 11.393 | None | None | None | XRAY | 2.7 | 0.23 | 0.311 | A | 360 | 343 | 6 | 0 | 0 | 6 | [[24, 308]] | 1.0 | 3que | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 4R3CA | Q16539 | 4 | 352 | 360.0 | 3GF:402,3GF:403 | Type1,Allosteric | Inactive | DFGin | 4.924 | 13.134 | None | -118.67, 171.2 | 49.4, 42.48 | -86.86, 999.0 | 38.51, 75.43 | 999.0, 999.0 | in-out | in | 9.543 | Saltbr-out | 3.908 | HRD-in | -66.01, -56.32 | 81.1, -14.57 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 103.85 | APE9-dihe-na | -65.1, 130.86 | APE8-dihe-out | -51.86, -39.46 | APE8-rot-in | 289.55 | APE67-dihe-in | -62.53, -25.36 | -48.44, -37.03 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.264 | None | None | CME162 | XRAY | 2.06 | 0.178 | 0.217 | A | 383 | 336 | 13 | 0 | 0 | 13 | [[24, 308]] | 1.0 | 4r3c | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 7.2e-85 | 290.9 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3L8SA | Q16539 | 4 | 353 | 360.0 | BFF:361 | Type1 | Inactive | DFGout | 15.489 | 11.977 | None | -119.54, 162.4 | -99.13, -16.66 | 31.92, 999.0 | 247.73, 144.9 | 999.0, 999.0 | in-in | in | 9.497 | Saltbr-in | 2.817 | HRD-in | -77.51, -50.13 | 90.87, -25.05 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, 107.11 | APE9-dihe-na | -94.83, 118.78 | APE8-dihe-out | -62.16, -3.07 | APE8-rot-out | 173.18 | APE67-dihe-in | -59.13, -22.21 | -95.45, -15.35 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.2 | C119S,C162S,A172C,F327L | None | None | XRAY | 2.35 | 0.242 | 0.307 | A | 360 | 334 | 16 | 0 | 0 | 13 | [[24, 308]] | 1.0 | 3l8s | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 4.4e-84 | 288.3 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3UVRA | Q16539 | 5 | 351 | 360.0 | 06F:361 | Type2 | Inactive | DFGout | 15.561 | 8.524 | None | -148.63, 178.6 | -133.58, 101.18 | -90.01, -1.78 | 195.55, 17.77 | -54.07, 127.45 | in-in | in | 8.211 | Saltbr-in | 2.627 | HRD-in | -62.71, -55.49 | 83.79, -17.62 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -56.89 | APE8-dihe-out | -51.15, -30.26 | APE8-rot-in | 300.71 | APE67-dihe-in | -70.54, -25.21 | -93.95, -15.4 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.621 | None | None | None | XRAY | 2.1 | 0.204 | 0.245 | A | 360 | 331 | 16 | 0 | 0 | 12 | [[24, 308]] | 1.0 | 3uvr | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK8 | MK08_HUMAN | 8PTAA | P45983 | 8 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.923 | 14.477 | ABAminus | -80.58, -61.37 | -103.85, 165.38 | -100.79, 23.99 | 295.77, 91.74 | 73.84, -149.47 | in-in | in | 9.79 | Saltbr-in | 3.126 | HRD-in | -78.59, -61.53 | 62.23, 7.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.47 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iooo | APE10-dihe-na | -130.45, 138.38 | APE9-dihe-na | -101.99, 109.25 | APE8-dihe-in | -118.89, 112.23 | APE8-rot-out | 53.5 | APE67-dihe-in | -51.79, -30.07 | -95.29, -17.54 | APE12-dist-in | 10.569 | APE11-dist-out | 7.033 | APE10-dist-out | 10.183 | APE9-dist-out | 8.598 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | A | 366 | 354 | 2 | 0 | 0 | 2 | [[26, 321]] | 1.0 | 8pta | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| CMGC | MAPK8 | MK08_HUMAN | 8PTAB | P45983 | 7 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.577 | 13.179 | ABAminus | -81.24, -57.35 | -101.3, 158.61 | -105.36, 14.2 | 308.93, 93.28 | 64.59, -148.13 | in-in | in | 9.366 | Saltbr-in | 3.536 | HRD-in | -77.41, -61.25 | 61.49, 9.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -112.33, 168.25 | APE9-dihe-na | -116.9, 36.67 | APE8-dihe-in | -104.63, 91.0 | APE8-rot-out | 52.55 | APE67-dihe-in | -56.88, -29.41 | -95.02, -21.65 | APE12-dist-in | 11.784 | APE11-dist-in | 9.152 | APE10-dist-out | 11.242 | APE9-dist-out | 10.214 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | B | 366 | 352 | 5 | 0 | 0 | 5 | [[26, 321]] | 1.0 | 8pta | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| CMGC | MAPK8 | MK08_HUMAN | 8PTAC | P45983 | 8 | 361 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.826 | 14.088 | ABAminus | -83.97, -56.35 | -97.04, 154.46 | -105.76, 13.83 | 294.99, 32.04 | 63.79, -147.27 | in-out | in | 9.723 | Saltbr-out | 4.528 | HRD-in | -77.01, -60.9 | 63.25, 7.56 | out-out-out | SNCooo | out-out | ActLoopNT-out | 4.611 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -137.59 | APE9-dihe-na | -94.11, 17.64 | APE8-dihe-in | -81.48, 63.35 | APE8-rot-out | 71.39 | APE67-dihe-in | -58.68, -26.77 | -108.19, -24.77 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 12.467 | APE9-dist-out | 10.78 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | C | 366 | 351 | 3 | 0 | 0 | 3 | [[26, 321]] | 1.0 | 8pta | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| CMGC | MAPK9 | MK09_HUMAN | 3E7OA | P45984 | 9 | 361 | 424.0 | 35F:1 | Type1 | Inactive | DFGin | 4.266 | 14.526 | ABAminus | -84.35, -29.35 | -149.55, 177.24 | -106.27, 9.79 | 301.22, 95.14 | 60.95, -143.01 | in-in | in | 9.439 | Saltbr-in | 2.686 | HRD-in | -64.97, -51.12 | 67.58, -6.1 | in-out-out | SNCioo | out-out | ActLoopNT-out | 5.519 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_oooo | APE10-dihe-na | -84.71, -45.82 | APE9-dihe-na | -76.84, -178.43 | APE8-dihe-in | -88.6, 137.99 | APE8-rot-in | 266.04 | APE67-dihe-out | -72.72, -13.34 | -138.1, 64.96 | APE12-dist-out | 20.29 | APE11-dist-out | 15.686 | APE10-dist-out | 19.328 | APE9-dist-out | 14.665 | C177S,C222S,K250A,K251A,K265A,K270A | None | None | XRAY | 2.14 | 0.219 | 0.25 | A | 360 | 342 | 2 | 0 | 0 | 0 | [[26, 321]] | 1.0 | 3e7o | Homo sapiens | CMGC_MAPK9_HUMAN | CMGC | 2.7e-84 | 288.8 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 9 |
| CMGC | MAPK9 | MK09_HUMAN | 3E7OB | P45984 | 8 | 362 | 424.0 | 35F:2 | Type1 | Inactive | DFGin | 4.276 | 14.318 | ABAminus | -85.32, -37.61 | -133.45, 175.33 | -107.39, 15.94 | 299.45, 88.14 | 90.36, 999.0 | in-in | in | 9.466 | Saltbr-in | 2.801 | HRD-in | -71.07, -57.75 | 72.11, -12.31 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -39.52 | APE8-rot-out | 181.64 | APE67-dihe-in | -65.99, -17.44 | -49.19, -35.22 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | C177S,C222S,K250A,K251A,K265A,K270A | None | None | XRAY | 2.14 | 0.219 | 0.25 | B | 360 | 326 | 19 | 0 | 0 | 16 | [[26, 321]] | 1.0 | 3e7o | Homo sapiens | CMGC_MAPK9_HUMAN | CMGC | 2.7e-84 | 288.8 | 1 | 301 | 301 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 9 |
| OTHER | CDC7 | CDC7_HUMAN | 6YA8A | O00311 | 38 | 572 | 574.0 | ADP:60601,BEF:60603 | ATPlike,Allosteric | None | DFGin | 6.168 | 14.087 | BLAminus | -118.93, 173.08 | 76.34, 83.66 | -102.33, 21.87 | 291.62, 81.2 | -67.07, -22.7 | in-in | in | 8.709 | Saltbr-in | 2.738 | HRD-in | -65.76, -44.2 | 72.35, -4.4 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.755 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | -83.06, -154.71 | APE8-dihe-in | -48.63, 132.1 | APE8-rot-in | 306.86 | APE67-dihe-in | -66.07, -7.37 | -59.08, -35.16 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.888 | None | None | None | XRAY | 1.79 | 0.167 | 0.197 | A | 359 | 338 | 13 | 0 | 0 | 13 | [[58, 569]] | 1.0 | 6ya8 | Homo sapiens | OTHER_CDC7_HUMAN | CMGC | 2e-18 | 137.3 | 1 | 161 | 296 | 195 | 196 | 197 | 199 | 201 | 90 | 104 | 108 | 174 | 176 | 175 | 177 | 396 | 383 | 378 | 377 | 376 | 375 | 0 | 0 | 0 | 135 | Cell division cycle 7-related protein kinase |
| OTHER | GAK | GAK_HUMAN | 4C57A | O14976 | 25 | 334 | 1311.0 | FEF:1340 | Type1 | Inactive | DFGin | 5.754 | 14.141 | ABAminus | -112.53, -37.31 | -102.07, 134.52 | -132.21, 22.67 | 297.88, 98.14 | -59.75, -31.11 | in-out | in | 9.993 | Saltbr-out | 4.057 | HRD-in | -62.14, -51.36 | 70.7, -5.09 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.895 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.34, 3.52 | APE9-dihe-na | -124.99, 156.99 | APE8-dihe-in | -84.98, 122.71 | APE8-rot-in | 297.75 | APE67-dihe-in | -71.57, -19.62 | -46.23, -44.89 | APE12-dist-in | 11.779 | APE11-dist-in | 8.573 | APE10-dist-in | 4.33 | APE9-dist-in | 4.07 | None | None | None | XRAY | 2.55 | 0.18 | 0.228 | A | 340 | 310 | 0 | 0 | 0 | 0 | [[40, 313]] | 1.0 | 4c57 | Homo sapiens | OTHER_GAK_HUMAN | CAMK | 5.3e-44 | 156.7 | 3 | 252 | 250 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | GAK | GAK_HUMAN | 4C57B | O14976 | 27 | 334 | 1311.0 | FEF:1337 | Type1 | Inactive | DFGin | 5.769 | 14.233 | ABAminus | -105.07, -37.59 | -101.51, 133.86 | -130.57, 22.88 | 297.9, 97.48 | -60.27, -26.81 | out-out | out | 10.065 | Saltbr-out | 4.056 | HRD-in | -62.14, -52.49 | 71.3, -9.85 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.891 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.07, 5.67 | APE9-dihe-na | -124.2, 156.66 | APE8-dihe-in | -83.72, 121.96 | APE8-rot-in | 296.0 | APE67-dihe-in | -71.56, -19.42 | -45.7, -45.17 | APE12-dist-in | 11.928 | APE11-dist-in | 8.658 | APE10-dist-in | 4.358 | APE9-dist-in | 4.086 | None | None | None | XRAY | 2.55 | 0.18 | 0.228 | B | 340 | 308 | 0 | 0 | 0 | 0 | [[40, 313]] | 1.0 | 4c57 | Homo sapiens | OTHER_GAK_HUMAN | CAMK | 5.3e-44 | 156.7 | 3 | 252 | 250 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | GAK | GAK_HUMAN | 4C59A | O14976 | 27 | 333 | 1311.0 | FEF:1334 | Type1 | Inactive | DFGin | 5.815 | 13.68 | ABAminus | -134.62, -10.32 | -105.18, 88.43 | -107.04, 23.92 | 300.54, 105.0 | -81.95, -10.0 | in-in | in | 9.093 | Saltbr-in | 2.855 | HRD-in | -82.36, -54.36 | 82.63, -15.13 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.838 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.8 | 0.205 | 0.262 | A | 340 | 266 | 41 | 0 | 0 | 27 | [[40, 313]] | 1.0 | 4c59 | Homo sapiens | OTHER_GAK_HUMAN | CAMK | 5.3e-44 | 156.7 | 3 | 252 | 250 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | HASPIN | HASP_HUMAN | 9FLTA | Q8TF76 | 471 | 798 | 798.0 | A1IDF:801 | Type1 | Active | DFGin | 5.178 | 12.218 | BLAminus | -141.02, 178.95 | 59.99, 70.73 | -81.95, 27.03 | 316.78, 141.24 | -69.29, -28.67 | in-in | in | 8.759 | Saltbr-in | 2.463 | HRD-na-N | -66.6, -53.16 | 75.71, 6.9 | in-in-na | SNCiia | in-na | ActLoopNT-in | 2.905 | ActLoopCT-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | APE10-dihe-na | -131.58, 41.34 | APE9-dihe-na | -102.69, 164.5 | APE8-dihe-na | -162.68, -171.46 | APE8-rot-na | 41.52 | APE67-dihe-na | -134.91, 146.64 | 100.36, -24.97 | APE12-dist-na | 9.64 | APE11-dist-na | 13.509 | APE10-dist-na | 17.247 | APE9-dist-na | 13.279 | None | None | None | XRAY | 2.4 | 0.187 | 0.239 | A | 336 | 320 | 8 | 0 | 0 | 0 | [[484, 797]] | 1.0 | 9flt | Homo sapiens | OTHER_HASPIN_HUMAN | HASP | 1.1e-226 | 756.9 | 1 | 314 | 314 | 686 | 687 | 688 | 690 | 692 | 511 | 535 | 539 | 646 | 648 | 647 | 649 | 741 | 721 | 716 | 715 | 714 | 713 | 712 | 711 | 710 | 604 | Serine/threonine-protein kinase haspin |
| OTHER | TTK | TTK_HUMAN | 4JS8A | P33981 | 515 | 793 | 857.0 | 1PF:801 | Type1 | Inactive | DFGin | 4.246 | 15.018 | ABAminus | -84.57, -49.34 | -133.98, 167.4 | -109.17, 14.51 | 305.07, 151.28 | 67.69, 15.63 | in-out | in | 9.993 | Saltbr-out | 6.699 | HRD-in | -62.96, -52.34 | 70.46, -10.5 | out-out-out | SNCooo | out-out | ActLoopNT-out | 12.036 | ActLoopCT-out | nonTYR | APEdihe_aaini | APEdist_nnoo | APE10-dihe-na | 999.0, 112.01 | APE9-dihe-na | -104.69, -175.56 | APE8-dihe-in | -119.7, 153.55 | APE8-rot-none | 999.0 | APE67-dihe-in | -65.36, -29.34 | -115.57, 0.38 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.198 | APE9-dist-out | 12.111 | None | TPO675,TPO686 | TPO675,TPO686 | XRAY | 1.94 | 0.232 | 0.253 | A | 281 | 261 | 18 | 0 | 0 | 8 | [[525, 791]] | 1.0 | 4js8 | Homo sapiens | OTHER_TTK_HUMAN | CAMK | 5.6e-54 | 189.1 | 1 | 256 | 256 | 663 | 664 | 665 | 667 | 669 | 553 | 571 | 575 | 644 | 646 | 645 | 647 | 716 | 693 | 688 | 687 | 686 | 685 | 684 | 683 | 682 | 603 | Dual specificity protein kinase TTK |
| OTHER | TTK | TTK_HUMAN | 7CHMA | P33981 | 516 | 794 | 857.0 | FZF:801 | Type1 | Inactive | DFGin | 4.413 | 14.608 | None | -111.88, -71.82 | -63.89, 158.67 | -119.5, 9.1 | 283.45, 179.72 | 82.92, -15.75 | in-in | in | 9.56 | Saltbr-in | 3.396 | HRD-in | -57.59, -51.23 | 60.31, 6.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 12.264 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnoo | APE10-dihe-na | 999.0, -62.47 | APE9-dihe-na | 66.11, 172.68 | APE8-dihe-out | -121.28, -175.85 | APE8-rot-none | 999.0 | APE67-dihe-in | -54.56, -33.62 | -132.81, 0.36 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 19.863 | APE9-dist-out | 12.904 | None | TPO675,TPO686 | TPO675,TPO686 | XRAY | 2.65 | 0.212 | 0.253 | A | 281 | 260 | 19 | 0 | 0 | 8 | [[525, 791]] | 1.0 | 7chm | Homo sapiens | OTHER_TTK_HUMAN | CAMK | 5.6e-54 | 189.1 | 1 | 256 | 256 | 663 | 664 | 665 | 667 | 669 | 553 | 571 | 575 | 644 | 646 | 645 | 647 | 716 | 693 | 688 | 687 | 686 | 685 | 684 | 683 | 682 | 603 | Dual specificity protein kinase TTK |
| OTHER | ULK1 | ULK1_HUMAN | 4WNOA | O75385 | 8 | 280 | 1050.0 | 3RF:401 | Type1 | Active | DFGin | 6.889 | 14.949 | BLAminus | -117.94, 169.26 | 64.81, 74.6 | -94.14, 20.86 | 282.18, 71.59 | -63.55, -24.11 | in-in | in | 7.662 | Saltbr-in | 2.77 | HRD-in | -82.57, -51.36 | 80.06, -2.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.966 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -155.03, 162.62 | APE9-dihe-na | 120.91, -162.5 | APE8-dihe-in | -119.54, 124.2 | APE8-rot-in | 305.96 | APE67-dihe-in | -67.71, -19.19 | -53.63, -37.75 | APE12-dist-in | 8.214 | APE11-dist-in | 11.212 | APE10-dist-in | 5.675 | APE9-dist-in | 3.309 | E37A,K38A | TPO180 | TPO180 | XRAY | 1.56 | 0.18 | 0.208 | A | 287 | 273 | 0 | 0 | 0 | 0 | [[14, 278]] | 1.0 | 4wno | Homo sapiens | OTHER_ULK1_HUMAN | ULK | 2.1e-132 | 446.2 | 1 | 256 | 256 | 164 | 165 | 166 | 168 | 170 | 46 | 63 | 67 | 135 | 137 | 136 | 138 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 93 | Serine/threonine-protein kinase ULK1 |
| STE | MAP2K1 | MP2K1_HUMAN | 7UMBC | Q02750 | 41 | 381 | 393.0 | ANP:401,U9F:402 | ATPlike,Type3 | Inactive | DFGin | 6.169 | 13.767 | BLBplus | -162.24, 171.11 | 70.21, 49.7 | -113.95, 160.88 | 44.65, 94.08 | -79.06, 81.13 | out-out | out | 15.559 | Saltbr-out | 15.273 | HRD-in | -66.12, -48.09 | 76.83, -9.86 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.591 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -127.94, 139.36 | APE9-dihe-na | -138.86, -160.81 | APE8-dihe-out | -82.2, -18.64 | APE8-rot-out | 50.9 | APE67-dihe-out | -106.39, 139.13 | -104.8, 110.61 | APE12-dist-out | 16.699 | APE11-dist-out | 19.666 | APE10-dist-out | 21.57 | APE9-dist-out | 14.915 | None | None | None | XRAY | 3.231 | 0.231 | 0.268 | C | 384 | 303 | 38 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 7umb | Homo sapiens | STE_MAP2K1_HUMAN | STE | 2.3e-97 | 331.4 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K7 | MP2K7_HUMAN | 6YG3A | O14733 | 103 | 400 | 419.0 | 6HF:60510 | Type1 | None | DFGin | 6.195 | 14.549 | BLAminus | -146.55, 178.23 | 54.3, 83.97 | -103.73, 30.03 | 316.89, 91.95 | -57.17, -29.89 | na-na | na | 8.345 | Saltbr-na | 3.36 | HRD-in | -81.36, -52.29 | 76.4, 12.98 | na-in-none | SNCain | in-none | ActLoopNT-in | 2.982 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.05 | 0.191 | 0.235 | A | 307 | 265 | 33 | 0 | 0 | 19 | [[120, 380]] | 1.0 | 6yg3 | Homo sapiens | STE_MAP2K7_HUMAN | STE | 2.4e-80 | 275.5 | 2 | 257 | 256 | 260 | 261 | 262 | 264 | 266 | 149 | 166 | 170 | 240 | 242 | 241 | 243 | 304 | 287 | 282 | 281 | 280 | 279 | 278 | 277 | 276 | 197 | Dual specificity mitogen-activated protein kinase kinase 7 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4A | Q92918 | 4 | 293 | 833.0 | XXF:60401 | Type1 | Inactive | DFGin | 6.846 | 14.475 | BLAminus | -131.99, 171.23 | 62.34, 86.7 | -92.12, 20.1 | 289.3, 88.42 | -59.7, -48.05 | in-in | in | 9.232 | Saltbr-in | 2.734 | HRD-in | -67.47, -51.18 | 67.4, 4.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.199 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -73.65, -44.57 | APE9-dihe-na | 76.29, -171.23 | APE8-dihe-in | -62.48, 141.12 | APE8-rot-out | 34.25 | APE67-dihe-in | -59.58, -27.68 | -102.29, 0.49 | APE12-dist-out | 20.304 | APE11-dist-out | 21.079 | APE10-dist-out | 21.421 | APE9-dist-out | 27.259 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | A | 331 | 290 | 0 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 8fh4 | Homo sapiens | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4B | Q92918 | 6 | 302 | 833.0 | XXF:60402 | Type1 | Inactive | DFGin | 6.551 | 14.294 | BLAminus | -141.43, 174.43 | 62.64, 85.33 | -93.2, 13.55 | 285.99, 85.49 | -57.34, -45.75 | in-in | in | 8.939 | Saltbr-in | 2.697 | HRD-in | -67.85, -50.88 | 67.73, 2.48 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.309 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -67.39, -32.57 | APE9-dihe-na | 75.42, -167.37 | APE8-dihe-in | -61.44, 126.8 | APE8-rot-out | 59.49 | APE67-dihe-in | -56.24, -30.95 | -97.05, -0.91 | APE12-dist-out | 19.464 | APE11-dist-out | 20.586 | APE10-dist-out | 21.665 | APE9-dist-out | 28.047 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | B | 331 | 297 | 0 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 8fh4 | Homo sapiens | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4C | Q92918 | 1 | 292 | 833.0 | XXF:60401 | Type1 | Inactive | DFGin | 6.824 | 14.118 | BLAminus | -136.31, 172.65 | 64.01, 85.1 | -95.02, 19.77 | 288.84, 83.7 | -61.21, -46.39 | in-in | in | 8.967 | Saltbr-in | 2.733 | HRD-in | -69.91, -50.19 | 67.9, 0.86 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.08 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -67.7, -68.85 | APE9-dihe-na | -109.26, -27.15 | APE8-dihe-in | -115.11, 101.44 | APE8-rot-out | 62.11 | APE67-dihe-in | -65.51, -20.35 | -96.81, 16.0 | APE12-dist-out | 19.318 | APE11-dist-out | 20.935 | APE10-dist-out | 23.085 | APE9-dist-out | 28.365 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | C | 331 | 292 | 0 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 8fh4 | Homo sapiens | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8FH4D | Q92918 | 8 | 292 | 833.0 | XXF:60401 | Type1 | Inactive | DFGin | 6.646 | 14.023 | BLAminus | -135.73, 170.9 | 66.66, 83.46 | -93.58, 25.1 | 289.61, 94.72 | -69.05, -41.66 | in-in | in | 9.022 | Saltbr-in | 2.745 | HRD-in | -74.6, -51.27 | 71.89, -5.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.134 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -170.02 | APE8-dihe-in | -67.05, 131.5 | APE8-rot-out | 192.16 | APE67-dihe-in | -57.98, -30.82 | -102.78, -3.16 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 27.427 | T165E,S171E | None | None | XRAY | 1.827 | 0.189 | 0.215 | D | 331 | 276 | 9 | 0 | 0 | 4 | [[17, 274]] | 1.0 | 8fh4 | Homo sapiens | STE_MAP4K1_HUMAN | STE | 6.2e-92 | 313.5 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 9QT6A | Q92918 | 6 | 292 | 833.0 | A1JAF:301 | Type1 | Inactive | DFGin | 6.463 | 13.765 | None | -60.93, -35.58 | -154.04, -176.9 | -79.86, 1.42 | 63.88, 19.01 | 105.02, -157.57 | out-out | out | 13.28 | Saltbr-out | 10.782 | HRD-in | -74.09, -55.53 | 70.27, 5.38 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.582 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioo | APE10-dihe-na | -59.89, -40.77 | APE9-dihe-na | -92.18, -16.28 | APE8-dihe-in | -142.86, 74.69 | APE8-rot-in | 316.27 | APE67-dihe-in | -56.11, -27.62 | -91.41, -1.8 | APE12-dist-in | 9.809 | APE11-dist-in | 11.134 | APE10-dist-out | 15.153 | APE9-dist-out | 12.698 | T165E,S171E | None | None | XRAY | 1.76 | 0.198 | 0.226 | A | 294 | 285 | 2 | 0 | 0 | 0 | [[17, 274]] | 1.0 | 9qt6 | Homo sapiens | STE_MAP4K1_HUMAN | STE | 4.1e-92 | 314.1 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K1 | M4K1_HUMAN | 8CIJA | Q92918 | 14 | 294 | 833.0 | USF:401 | Type1 | Inactive | DFGout | 11.213 | 7.331 | None | -112.58, 122.54 | -96.1, 115.56 | -121.01, 999.0 | 297.98, 106.95 | 999.0, 999.0 | out-out | out | 13.535 | Saltbr-out | 11.8 | HRD-in | -61.67, -48.53 | 69.18, 2.25 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | -87.98, 122.06 | APE9-dihe-na | 145.78, 142.84 | APE8-dihe-in | -120.8, 116.13 | APE8-rot-in | 320.07 | APE67-dihe-in | -58.16, -27.75 | -31.5, -57.68 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.681 | None | None | None | XRAY | 2.821 | 0.239 | 0.266 | A | 307 | 264 | 17 | 0 | 0 | 12 | [[17, 274]] | 1.0 | 8cij | Homo sapiens | STE_MAP4K1_HUMAN | STE | 4.8e-92 | 313.9 | 1 | 256 | 256 | 154 | 155 | 156 | 158 | 160 | 46 | 62 | 66 | 134 | 136 | 135 | 137 | 197 | 182 | 177 | 176 | 175 | 174 | 173 | 172 | 171 | 92 | Mitogen-activated protein kinase kinase kinase kinase 1 |
| STE | MAP4K4 | M4K4_HUMAN | 5DI1A | O95819 | 13 | 309 | 1239.0 | 5DF:4000 | Type1 | Inactive | DFGin | 4.26 | 13.366 | BLBplus | -145.12, 159.02 | 72.53, 52.2 | -89.55, 138.32 | 48.51, 95.38 | -80.62, 999.0 | in-out | in | 9.403 | Saltbr-out | 3.985 | HRD-in | -61.2, -47.09 | 79.65, -23.06 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | -102.21, 124.07 | APE9-dihe-na | -81.57, -147.04 | APE8-dihe-in | -74.95, 131.45 | APE8-rot-out | 195.98 | APE67-dihe-in | -46.35, -33.38 | -85.44, -21.52 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.602 | None | None | None | XRAY | 2.9 | 0.2 | 0.249 | A | 310 | 285 | 12 | 0 | 0 | 12 | [[25, 289]] | 1.0 | 5di1 | Homo sapiens | STE_MAP4K4_HUMAN | STE | 1.3e-102 | 348.4 | 1 | 257 | 257 | 170 | 171 | 172 | 174 | 176 | 54 | 69 | 73 | 150 | 152 | 151 | 153 | 215 | 198 | 193 | 192 | 191 | 190 | 189 | 188 | 187 | 106 | Mitogen-activated protein kinase kinase kinase kinase 4 |
| TKL | ACVR1 | ACVR1_HUMAN | 3MTFA | Q04771 | 203 | 498 | 509.0 | A3F:1 | Type1 | Inactive | DFGin | 7.09 | 13.208 | BLAminus | -126.1, 157.67 | 76.9, 82.69 | -86.05, 21.36 | 306.23, 175.03 | -61.66, -24.97 | in-out | in | 8.331 | Saltbr-out | 4.196 | HRD-in | -82.54, -58.57 | 79.29, -1.49 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.913 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -103.22, 162.67 | APE9-dihe-na | -69.88, 165.81 | APE8-dihe-in | -53.93, 121.99 | APE8-rot-in | 312.82 | APE67-dihe-in | -59.42, -28.32 | -57.34, -37.41 | APE12-dist-in | 10.671 | APE11-dist-out | 6.476 | APE10-dist-out | 9.482 | APE9-dist-in | 4.073 | Q207D | None | None | XRAY | 2.15 | 0.185 | 0.244 | A | 301 | 296 | 0 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 3mtf | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 3MTFB | Q04771 | 202 | 499 | 509.0 | A3F:501 | Type1 | Inactive | DFGin | 7.578 | 13.323 | BLAminus | -114.45, 160.06 | 82.35, 87.49 | -104.83, 25.86 | 291.12, 164.81 | -75.29, -13.54 | in-out | in | 8.5 | Saltbr-out | 4.232 | HRD-in | -82.5, -60.12 | 85.3, -4.39 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.869 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -111.75, 153.3 | APE9-dihe-na | -57.45, 170.81 | APE8-dihe-in | -65.39, 131.64 | APE8-rot-in | 306.28 | APE67-dihe-in | -49.77, -35.33 | -68.1, -43.23 | APE12-dist-in | 10.611 | APE11-dist-out | 6.453 | APE10-dist-out | 9.396 | APE9-dist-in | 4.119 | Q207D | None | None | XRAY | 2.15 | 0.185 | 0.244 | B | 301 | 298 | 0 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 3mtf | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6EIXA | Q04771 | 192 | 503 | 509.0 | A3F:601 | Type1 | Inactive | DFGin | 7.305 | 13.382 | BLAminus | -122.31, 163.89 | 74.01, 85.68 | -98.53, 23.31 | 310.02, 174.96 | -66.89, -23.04 | in-out | in | 9.083 | Saltbr-out | 5.16 | HRD-in | -81.6, -53.66 | 78.97, -2.54 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.023 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -113.45, 165.41 | APE9-dihe-na | -59.94, 163.8 | APE8-dihe-in | -59.76, 126.51 | APE8-rot-in | 307.55 | APE67-dihe-in | -58.05, -30.26 | -58.58, -41.78 | APE12-dist-in | 10.589 | APE11-dist-out | 6.415 | APE10-dist-out | 9.311 | APE9-dist-in | 3.871 | Q207E | None | None | XRAY | 2.3 | 0.191 | 0.249 | A | 340 | 312 | 0 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 6eix | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 2.9e-85 | 292.0 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 8PODA | Q04771 | 172 | 498 | 509.0 | 7IO:60501,F:60502 | Type1,Allosteric | Inactive | DFGin | 7.181 | 13.248 | BLAminus | -129.23, 172.96 | 64.95, 88.23 | -102.11, 21.22 | 307.17, 178.99 | -69.46, -24.05 | in-out | in | 8.75 | Saltbr-out | 5.24 | HRD-in | -77.46, -49.01 | 73.0, -1.63 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.105 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -104.74, 151.99 | APE9-dihe-na | -69.89, 170.49 | APE8-dihe-in | -67.7, 124.46 | APE8-rot-in | 304.29 | APE67-dihe-in | -63.94, -28.35 | -69.6, -32.91 | APE12-dist-in | 10.74 | APE11-dist-out | 6.542 | APE10-dist-out | 9.732 | APE9-dist-in | 4.647 | None | None | None | XRAY | 2.59 | 0.236 | 0.255 | A | 330 | 320 | 1 | 0 | 0 | 0 | [[207, 497]] | 1.0 | 8pod | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 2.6e-85 | 292.1 | 2 | 267 | 266 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | BRAF | BRAF_HUMAN | 4YHTA | P15056 | 449 | 719 | 766.0 | 4EF:61002 | Type1 | Inactive | DFGin | 6.44 | 13.919 | BLAminus | -130.91, -175.71 | 59.89, 88.64 | -101.88, 16.92 | 281.61, 73.69 | -54.19, -26.07 | in-in | in | 8.608 | Saltbr-in | 2.731 | HRD-in | -63.73, -42.35 | 62.62, 3.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.881 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -6.83 | APE8-dihe-in | -100.18, 82.06 | APE8-rot-in | 287.27 | APE67-dihe-in | -63.55, -16.06 | -74.16, -21.42 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.11 | I543T,I544N,I551T,L706T,L716T | None | None | XRAY | 3.05 | 0.2 | 0.233 | A | 272 | 256 | 15 | 0 | 0 | 13 | [[457, 716]] | 1.0 | 4yht | Homo sapiens | TKL_BRAF_HUMAN | TKL | 2.7e-84 | 288.8 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 4YHTB | P15056 | 449 | 720 | 766.0 | 4EF:60802 | Type1 | Inactive | DFGin | 6.405 | 13.921 | BLAminus | -128.69, -172.56 | 54.11, 90.89 | -102.92, 13.66 | 281.86, 71.12 | -49.43, -28.96 | in-in | in | 8.583 | Saltbr-in | 2.701 | HRD-in | -63.82, -42.99 | 62.91, 4.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.864 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -6.59 | APE8-dihe-in | -97.87, 80.96 | APE8-rot-in | 285.28 | APE67-dihe-in | -62.85, -18.47 | -75.71, -20.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.034 | I543T,I544N,I551T,L706T,L716T | None | None | XRAY | 3.05 | 0.2 | 0.233 | B | 272 | 258 | 14 | 0 | 0 | 12 | [[457, 716]] | 1.0 | 4yht | Homo sapiens | TKL_BRAF_HUMAN | TKL | 2.7e-84 | 288.8 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 3Q96A | P15056 | 449 | 722 | 766.0 | 0NF:1 | Type2 | Inactive | DFGout | 12.887 | 10.676 | BBAminus | -160.13, -172.44 | -118.2, 91.86 | -79.01, 12.35 | 294.04, 84.62 | -59.8, 141.31 | in-in | in | 8.392 | Saltbr-in | 2.855 | HRD-in | -57.31, -47.78 | 82.12, -11.82 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -115.71 | APE8-rot-in | 265.02 | APE67-dihe-in | -61.58, -24.04 | -87.09, -36.86 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 3.1 | 0.233 | 0.288 | A | 282 | 253 | 21 | 0 | 0 | 18 | [[457, 716]] | 1.0 | 3q96 | Homo sapiens | TKL_BRAF_HUMAN | TKL | 8e-82 | 280.7 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 3Q96B | P15056 | 449 | 720 | 766.0 | 0NF:1 | Type2 | Inactive | DFGout | 12.338 | 11.655 | BBAminus | -159.06, -168.23 | -117.43, 81.54 | -79.68, 17.57 | 296.0, 82.29 | -26.83, 105.54 | in-in | in | 8.586 | Saltbr-in | 3.176 | HRD-in | -76.92, -42.58 | 73.28, -12.97 | in-out-out | SNCioo | out-out | ActLoopNT-out | 18.49 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 159.44 | APE8-dihe-in | -92.55, 126.53 | APE8-rot-in | 290.06 | APE67-dihe-in | -62.77, -20.3 | -102.35, -28.12 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.232 | None | None | None | XRAY | 3.1 | 0.233 | 0.288 | B | 282 | 262 | 10 | 0 | 0 | 10 | [[457, 716]] | 1.0 | 3q96 | Homo sapiens | TKL_BRAF_HUMAN | TKL | 8e-82 | 280.7 | 4 | 266 | 263 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8A | Q9NWZ3 | 164 | 459 | 460.0 | 4GF:501 | Type1 | Active | DFGin | 6.842 | 14.163 | BLAminus | -130.64, 178.89 | 61.7, 76.88 | -103.53, 25.67 | 310.66, 96.36 | -67.74, -31.55 | in-in | in | 8.778 | Saltbr-in | 3.549 | HRD-in | -57.79, -50.73 | 76.7, -3.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.775 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.21, 150.97 | APE9-dihe-na | 140.01, -173.97 | APE8-dihe-in | -103.61, 115.43 | APE8-rot-in | 309.9 | APE67-dihe-in | -66.28, -16.88 | -42.43, -50.13 | APE12-dist-in | 10.008 | APE11-dist-in | 11.614 | APE10-dist-in | 6.326 | APE9-dist-in | 3.918 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | A | 301 | 287 | 9 | 0 | 0 | 4 | [[183, 456]] | 1.0 | 4yp8 | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8B | Q9NWZ3 | 161 | 459 | 460.0 | 4GF:501 | Type1 | Inactive | DFGin | 6.917 | 14.444 | BLAminus | -129.86, 179.56 | 60.17, 77.95 | -104.22, 26.32 | 310.53, 95.0 | -66.78, -33.18 | in-out | in | 8.685 | Saltbr-out | 3.962 | HRD-in | -57.85, -50.75 | 76.66, -4.15 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.853 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.74, 150.82 | APE9-dihe-na | 140.12, -173.75 | APE8-dihe-in | -103.4, 115.49 | APE8-rot-in | 310.63 | APE67-dihe-in | -65.34, -17.03 | -41.64, -51.23 | APE12-dist-in | 10.045 | APE11-dist-in | 11.581 | APE10-dist-in | 6.319 | APE9-dist-in | 3.905 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | B | 301 | 281 | 18 | 0 | 0 | 6 | [[183, 456]] | 1.0 | 4yp8 | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8C | Q9NWZ3 | 164 | 460 | 460.0 | 4GF:501 | Type1 | Inactive | DFGin | 6.821 | 14.409 | BLAminus | -129.81, 179.51 | 59.35, 79.05 | -103.24, 26.6 | 309.61, 96.69 | -66.38, -34.02 | in-out | in | 8.851 | Saltbr-out | 4.684 | HRD-in | -59.31, -50.52 | 77.45, -5.42 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.789 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.88, 150.51 | APE9-dihe-na | 141.79, -174.18 | APE8-dihe-in | -103.25, 114.63 | APE8-rot-in | 311.45 | APE67-dihe-in | -64.61, -17.76 | -41.38, -51.75 | APE12-dist-in | 10.149 | APE11-dist-in | 11.626 | APE10-dist-in | 6.34 | APE9-dist-in | 3.945 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | C | 301 | 290 | 7 | 0 | 0 | 4 | [[183, 456]] | 1.0 | 4yp8 | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 4YP8D | Q9NWZ3 | 164 | 459 | 460.0 | 4GF:501 | Type1 | Inactive | DFGin | 6.854 | 14.319 | BLAminus | -129.62, 178.91 | 61.84, 77.53 | -103.67, 26.43 | 310.15, 95.74 | -66.28, -34.21 | in-out | in | 8.915 | Saltbr-out | 3.802 | HRD-in | -59.75, -49.91 | 75.93, -3.95 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.79 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.59, 153.02 | APE9-dihe-na | 138.42, -174.86 | APE8-dihe-in | -103.4, 114.55 | APE8-rot-in | 310.75 | APE67-dihe-in | -64.11, -17.03 | -41.21, -51.68 | APE12-dist-in | 10.015 | APE11-dist-in | 11.585 | APE10-dist-in | 6.327 | APE9-dist-in | 3.922 | None | TPO342,TPO345,SEP346 | TPO342,TPO345,SEP346 | XRAY | 2.641 | 0.193 | 0.219 | D | 301 | 288 | 8 | 0 | 0 | 4 | [[183, 456]] | 1.0 | 4yp8 | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.1e-84 | 288.2 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYA | Q9NWZ3 | 163 | 458 | 460.0 | EXF:501 | Type1 | Inactive | DFGin | 6.997 | 14.049 | BLAminus | -130.85, 177.02 | 62.25, 85.69 | -105.57, 13.21 | 307.3, 97.03 | -58.17, -30.36 | in-out | in | 8.929 | Saltbr-out | 5.362 | HRD-in | -67.47, -54.1 | 77.02, 0.48 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.819 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.95, 147.66 | APE9-dihe-na | 135.07, -175.38 | APE8-dihe-in | -106.14, 112.07 | APE8-rot-in | 312.29 | APE67-dihe-in | -59.29, -20.88 | -52.35, -43.4 | APE12-dist-in | 10.191 | APE11-dist-in | 11.704 | APE10-dist-in | 6.439 | APE9-dist-in | 4.357 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | A | 305 | 294 | 2 | 0 | 0 | 2 | [[183, 456]] | 1.0 | 6lxy | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYB | Q9NWZ3 | 163 | 459 | 460.0 | EXF:502 | Type1 | None | DFGin | 6.973 | 14.137 | BLAminus | -129.45, 177.84 | 61.74, 86.54 | -106.07, 12.43 | 306.08, 97.48 | -57.61, -29.04 | in-none | in | 9.098 | Saltbr-none | 999.0 | HRD-in | -68.65, -53.21 | 75.68, 1.0 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.807 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.47, 149.33 | APE9-dihe-na | 135.3, -175.41 | APE8-dihe-in | -105.49, 112.4 | APE8-rot-in | 312.11 | APE67-dihe-in | -59.55, -21.17 | -51.5, -42.55 | APE12-dist-in | 10.189 | APE11-dist-in | 11.686 | APE10-dist-in | 6.444 | APE9-dist-in | 4.332 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | B | 305 | 297 | 0 | 0 | 0 | 0 | [[183, 456]] | 1.0 | 6lxy | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYD | Q9NWZ3 | 162 | 459 | 460.0 | EXF:502 | Type1 | Inactive | DFGin | 7.002 | 14.116 | BLAminus | -130.62, 177.55 | 62.4, 85.91 | -106.35, 12.8 | 307.19, 98.16 | -58.64, -30.18 | in-out | in | 8.943 | Saltbr-out | 5.354 | HRD-in | -67.38, -53.42 | 77.14, -1.48 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.786 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.01, 149.8 | APE9-dihe-na | 134.89, -175.28 | APE8-dihe-in | -104.95, 111.45 | APE8-rot-in | 311.34 | APE67-dihe-in | -58.57, -21.72 | -44.58, -48.25 | APE12-dist-in | 10.314 | APE11-dist-in | 11.954 | APE10-dist-in | 6.613 | APE9-dist-in | 4.254 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | D | 305 | 293 | 5 | 0 | 0 | 5 | [[183, 456]] | 1.0 | 6lxy | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6LXYE | Q9NWZ3 | 164 | 458 | 460.0 | EXF:502 | Type1 | Inactive | DFGin | 6.954 | 14.159 | BLAminus | -130.3, 176.57 | 62.62, 85.73 | -105.89, 13.23 | 306.79, 97.59 | -58.45, -29.69 | in-out | in | 8.931 | Saltbr-out | 5.391 | HRD-in | -66.96, -52.89 | 76.03, -0.37 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.795 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.25, 150.73 | APE9-dihe-na | 134.77, -173.9 | APE8-dihe-in | -105.72, 111.9 | APE8-rot-in | 311.85 | APE67-dihe-in | -56.93, -22.86 | -45.56, -48.25 | APE12-dist-in | 10.309 | APE11-dist-in | 11.905 | APE10-dist-in | 6.607 | APE9-dist-in | 4.292 | None | TPO345,SEP346 | TPO345,SEP346 | XRAY | 2.19 | 0.202 | 0.231 | E | 305 | 288 | 7 | 0 | 0 | 7 | [[183, 456]] | 1.0 | 6lxy | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.3e-84 | 288.1 | 5 | 266 | 262 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | MAP3K12 | M3K12_HUMAN | 5CEQA | Q12852 | 117 | 398 | 859.0 | 50F:4000 | Type1 | Inactive | DFGin | 6.285 | 14.143 | BLBplus | -139.34, 175.24 | 65.23, 33.46 | -103.17, 163.52 | 57.07, 90.2 | 71.88, 999.0 | na-na | na | 13.937 | Saltbr-na | 13.245 | HRD-in | -61.44, -57.14 | 79.98, -14.5 | na-none-out | SNCano | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | -71.43, -48.01 | APE9-dihe-na | -72.5, -0.08 | APE8-dihe-out | -118.56, -4.99 | APE8-rot-out | 184.08 | APE67-dihe-in | -55.04, -30.89 | -63.03, -27.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.132 | None | None | None | XRAY | 1.911 | 0.171 | 0.218 | A | 300 | 269 | 13 | 0 | 0 | 13 | [[118, 372]] | 1.0 | 5ceq | Homo sapiens | TKL_MAP3K12_HUMAN | MAP3K123 | 1.5e-137 | 462.8 | 1 | 254 | 254 | 253 | 254 | 255 | 257 | 259 | 152 | 161 | 165 | 233 | 235 | 234 | 236 | 292 | 280 | 275 | 274 | 273 | 272 | 271 | 270 | 269 | 191 | Mitogen-activated protein kinase kinase kinase 12 |
| TKL | MAP3K7 | M3K7_HUMAN | 5J9LA | O43318 | 31 | 496 | 606.0 | 6HF:60501 | Type1 | Inactive | DFGout | 12.964 | 7.575 | None | -126.7, 106.14 | -55.49, -39.75 | -39.65, 999.0 | 105.32, 93.88 | 999.0, 999.0 | in-out | in | 9.619 | Saltbr-out | 4.662 | HRD-in | -64.53, -55.8 | 74.12, -2.79 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 124.52 | APE8-dihe-out | -91.5, 21.0 | APE8-rot-in | 299.75 | APE67-dihe-in | -63.93, -32.31 | -64.12, -36.48 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.7 | None | None | None | XRAY | 2.752 | 0.214 | 0.243 | A | 307 | 253 | 20 | 0 | 0 | 14 | [[36, 286]] | 1.0 | 5j9l | Homo sapiens | TKL_MAP3K7_HUMAN | TKL | 3.7e-74 | 255.5 | 2 | 266 | 265 | 174 | 175 | 176 | 178 | 180 | 63 | 77 | 81 | 153 | 155 | 154 | 156 | 211 | 199 | 194 | 193 | 192 | 191 | 190 | 189 | 188 | 105 | Mitogen-activated protein kinase kinase kinase 7 |
| TKL | RIPK1 | RIPK1_HUMAN | 7FCZA | Q13546 | 10 | 294 | 671.0 | 3IF:301 | Type3 | Inactive | DFGout | 13.865 | 10.379 | BBAminus | -121.61, 171.92 | -133.79, 66.08 | -70.41, -22.3 | 302.99, 177.02 | -85.6, 3.29 | out-out | out | 15.002 | Saltbr-out | 12.85 | HRD-in | -69.8, -48.63 | 73.26, -13.72 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.074 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 77.72 | APE8-dihe-in | -67.19, 127.43 | APE8-rot-in | 294.95 | APE67-dihe-in | -62.33, -29.47 | -101.92, 1.17 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.476 | C34A,C127A,C233A,C240A | None | None | XRAY | 2.21 | 0.236 | 0.257 | A | 297 | 248 | 37 | 0 | 0 | 18 | [[17, 287]] | 1.0 | 7fcz | Homo sapiens | TKL_RIPK1_HUMAN | TKL | 1.3e-72 | 250.5 | 6 | 265 | 260 | 155 | 156 | 157 | 159 | 161 | 45 | 63 | 67 | 135 | 137 | 136 | 138 | 210 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 93 | Receptor-interacting serine/threonine-protein kinase 1 |
| TKL | RIPK1 | RIPK1_HUMAN | 7FCZB | Q13546 | 7 | 294 | 671.0 | 3IF:301 | Type3 | Inactive | DFGout | 13.913 | 10.028 | BBAminus | -118.21, 174.22 | -136.13, 64.53 | -68.29, -24.74 | 303.09, 178.58 | -83.09, -0.43 | out-out | out | 14.189 | Saltbr-out | 12.575 | HRD-in | -73.47, -53.47 | 80.61, -17.48 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.139 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 101.37 | APE8-dihe-in | -64.4, 143.44 | APE8-rot-out | 179.16 | APE67-dihe-in | -62.08, -29.26 | -100.06, -1.15 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.634 | C34A,C127A,C233A,C240A | None | None | XRAY | 2.21 | 0.236 | 0.257 | B | 297 | 263 | 25 | 0 | 0 | 17 | [[17, 287]] | 1.0 | 7fcz | Homo sapiens | TKL_RIPK1_HUMAN | TKL | 1.3e-72 | 250.5 | 6 | 265 | 260 | 155 | 156 | 157 | 159 | 161 | 45 | 63 | 67 | 135 | 137 | 136 | 138 | 210 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 93 | Receptor-interacting serine/threonine-protein kinase 1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 2WOUA | P36897 | 200 | 496 | 503.0 | ZZF:61500 | Type1 | Active | DFGin | 6.124 | 13.039 | BLAminus | -133.49, -169.53 | 51.05, 62.4 | -92.04, 13.34 | 298.31, 178.69 | -62.77, -27.98 | in-in | in | 7.586 | Saltbr-in | 2.752 | HRD-in | -65.52, -56.03 | 81.95, -3.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.039 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.77, -22.31 | APE9-dihe-na | -79.77, -172.15 | APE8-dihe-in | -73.94, 125.36 | APE8-rot-in | 306.35 | APE67-dihe-in | -52.11, -29.79 | -56.64, -45.19 | APE12-dist-in | 13.078 | APE11-dist-in | 11.935 | APE10-dist-in | 6.041 | APE9-dist-in | 3.629 | None | None | None | XRAY | 2.3 | 0.229 | 0.302 | A | 306 | 297 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2wou | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAA | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 5.904 | 13.047 | BLAminus | -165.74, 163.41 | 74.29, 54.12 | -79.67, 24.05 | 317.06, 176.62 | -56.68, -51.28 | in-in | in | 8.001 | Saltbr-in | 2.936 | HRD-in | -45.11, -27.8 | 52.25, 11.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.111 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.43, -171.19 | APE9-dihe-na | 80.03, 171.79 | APE8-dihe-in | -67.98, 121.11 | APE8-rot-in | 302.91 | APE67-dihe-in | -99.71, -73.49 | -46.09, -5.99 | APE12-dist-in | 11.624 | APE11-dist-in | 11.967 | APE10-dist-in | 6.015 | APE9-dist-in | 4.061 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | A | 342 | 328 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAB | P36897 | 171 | 501 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.017 | 13.306 | BLAminus | -136.45, -176.24 | 60.04, 54.86 | -81.47, 12.98 | 307.95, 5.19 | -52.57, -45.29 | in-in | in | 8.1 | Saltbr-in | 3.037 | HRD-in | -75.89, -39.75 | 60.74, 14.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.115 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.32, 175.24 | APE9-dihe-na | 101.52, 166.7 | APE8-dihe-in | -70.87, 127.35 | APE8-rot-in | 315.28 | APE67-dihe-in | -36.34, -44.33 | -43.95, -69.54 | APE12-dist-in | 11.94 | APE11-dist-in | 12.0 | APE10-dist-in | 6.373 | APE9-dist-in | 4.084 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAC | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Inactive | DFGin | 6.142 | 13.141 | BLAminus | -126.27, 176.42 | 50.71, 78.49 | -102.58, 30.06 | 320.3, 19.34 | -66.31, -17.95 | in-in | in | 7.99 | Saltbr-in | 2.662 | HRD-in | -67.56, -21.99 | 46.1, 19.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.947 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -120.66, 131.05 | APE9-dihe-na | 148.7, 175.0 | APE8-dihe-in | -102.93, 87.73 | APE8-rot-in | 305.5 | APE67-dihe-out | -28.83, -55.82 | 5.18, -84.04 | APE12-dist-in | 11.481 | APE11-dist-in | 12.149 | APE10-dist-in | 6.247 | APE9-dist-in | 4.208 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAD | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.26 | 13.168 | BLAminus | -151.5, 176.63 | 62.94, 64.2 | -90.99, 26.98 | 302.19, 4.38 | -66.56, -19.34 | in-in | in | 7.809 | Saltbr-in | 2.745 | HRD-in | -63.44, -55.82 | 78.14, 1.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.86, 174.28 | APE9-dihe-na | 87.09, 173.14 | APE8-dihe-in | -66.87, 116.28 | APE8-rot-in | 325.42 | APE67-dihe-in | -60.47, -38.15 | -48.63, -36.35 | APE12-dist-in | 11.714 | APE11-dist-in | 11.894 | APE10-dist-in | 6.37 | APE9-dist-in | 4.229 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3FAAE | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.355 | 13.366 | BLAminus | -131.48, -168.05 | 37.37, 86.28 | -107.7, 26.02 | 296.92, 176.17 | -65.92, -19.56 | in-in | in | 7.781 | Saltbr-in | 3.095 | HRD-in | -66.77, -57.93 | 79.95, 12.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.85 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.13, 169.87 | APE9-dihe-na | 90.72, 172.5 | APE8-dihe-in | -64.72, 129.04 | APE8-rot-in | 310.98 | APE67-dihe-in | -56.46, -40.64 | -59.57, -42.14 | APE12-dist-in | 11.99 | APE11-dist-in | 12.056 | APE10-dist-in | 6.57 | APE9-dist-in | 3.982 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR2 | TGFR2_HUMAN | 7DV6A | P37173 | 240 | 543 | 567.0 | HJF:9000 | Type1 | Active | DFGin | 7.131 | 13.432 | BLAminus | -156.15, -164.95 | 57.9, 60.45 | -93.44, 15.51 | 294.56, 110.64 | -56.6, -36.89 | in-in | in | 7.444 | Saltbr-in | 2.659 | HRD-in | -60.78, -51.79 | 74.77, -4.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.86 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.14, 141.57 | APE9-dihe-na | 113.33, -173.4 | APE8-dihe-in | -82.04, 128.94 | APE8-rot-in | 303.35 | APE67-dihe-in | -55.96, -36.36 | -60.86, -38.17 | APE12-dist-in | 11.508 | APE11-dist-in | 11.89 | APE10-dist-in | 6.046 | APE9-dist-in | 3.912 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.39 | 0.163 | 0.224 | A | 323 | 304 | 0 | 0 | 0 | 0 | [[244, 540]] | 1.0 | 7dv6 | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 2.1e-77 | 266.2 | 2 | 266 | 265 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TYR | ALK | ALK_HUMAN | 4CCUA | Q9UM73 | 1093 | 1402 | 1620.0 | AWF:1500 | Type1 | Inactive | DFGin | 6.02 | 14.623 | ABAminus | -118.73, -9.8 | -132.17, 139.04 | -133.56, 37.48 | 295.42, 86.35 | -74.53, -27.89 | in-out | in | 8.277 | Saltbr-out | 4.689 | HRD-in | -77.94, -47.73 | 82.62, -10.67 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.803 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.98, -27.23 | APE9-dihe-in | -56.62, 135.11 | APE8-dihe-in | -75.38, 65.75 | APE8-rot-na | 29.29 | APE67-dihe-in | -70.29, -14.23 | -60.1, -29.45 | APE12-dist-na | 14.525 | APE11-dist-na | 15.17 | APE10-dist-na | 10.028 | APE9-dist-in | 7.796 | None | None | None | XRAY | 2.0 | 0.202 | 0.233 | A | 327 | 293 | 17 | 0 | 0 | 6 | [[1116, 1385]] | 1.0 | 4ccu | Homo sapiens | TYR_ALK_HUMAN | TYR | 1.4e-90 | 309.1 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | ALK | ALK_HUMAN | 4FNZA | Q9UM73 | 1093 | 1402 | 1620.0 | NZF:1501 | Type1 | Inactive | DFGin | 5.291 | 12.8 | ABAminus | -135.46, 12.02 | -152.76, 153.63 | -83.97, -38.55 | 283.31, 122.35 | 73.66, 999.0 | in-in | in | 8.5 | Saltbr-in | 2.812 | HRD-in | -72.66, -49.3 | 78.9, -9.45 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -97.65, -24.93 | APE9-dihe-in | -50.61, 132.71 | APE8-dihe-in | -79.34, 69.48 | APE8-rot-na | 27.73 | APE67-dihe-in | -74.42, -13.21 | -56.44, -36.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.83 | C1097S | None | None | XRAY | 2.6 | 0.202 | 0.261 | A | 327 | 287 | 23 | 0 | 0 | 15 | [[1116, 1385]] | 1.0 | 4fnz | Homo sapiens | TYR_ALK_HUMAN | TYR | 1.4e-90 | 309.1 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | ALK | ALK_HUMAN | 4DCEA | Q9UM73 | 1093 | 1402 | 1620.0 | 0JF:1501 | Type1 | Inactive | DFGin | 5.63 | 13.823 | None | -137.27, 16.47 | -161.52, 152.14 | -94.73, 164.26 | 291.72, 122.64 | -76.17, 999.0 | in-in | in | 8.482 | Saltbr-in | 2.883 | HRD-in | -75.4, -48.78 | 85.77, -10.33 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -96.83, -20.84 | APE9-dihe-in | -55.51, 136.7 | APE8-dihe-in | -77.28, 70.08 | APE8-rot-na | 28.6 | APE67-dihe-in | -68.31, -8.92 | -56.77, -41.62 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.974 | C1097S | None | None | XRAY | 2.03 | 0.211 | 0.256 | A | 333 | 288 | 22 | 0 | 0 | 14 | [[1116, 1385]] | 1.0 | 4dce | Homo sapiens | TYR_ALK_HUMAN | TYR | 1.5e-90 | 309.0 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | ALK | ALK_HUMAN | 4DCEB | Q9UM73 | 1094 | 1402 | 1620.0 | 0JF:1501 | Type1 | Inactive | DFGin | 5.747 | 13.628 | None | -141.04, 18.73 | -165.26, 150.02 | -96.5, 167.37 | 286.77, 120.17 | -70.38, 999.0 | in-in | in | 8.563 | Saltbr-in | 2.99 | HRD-in | -72.56, -48.26 | 83.87, -14.3 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -96.41, -12.56 | APE9-dihe-in | -59.98, 136.0 | APE8-dihe-in | -80.48, 64.18 | APE8-rot-na | 31.8 | APE67-dihe-in | -66.1, -14.3 | -52.07, -41.53 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.713 | C1097S | None | None | XRAY | 2.03 | 0.211 | 0.256 | B | 333 | 284 | 25 | 0 | 0 | 15 | [[1116, 1385]] | 1.0 | 4dce | Homo sapiens | TYR_ALK_HUMAN | TYR | 1.5e-90 | 309.0 | 1 | 260 | 260 | 1269 | 1270 | 1271 | 1273 | 1275 | 1150 | 1167 | 1171 | 1246 | 1248 | 1247 | 1249 | 1311 | 1299 | 1294 | 1293 | 1292 | 1291 | 1290 | 1289 | 1288 | 1197 | ALK tyrosine kinase receptor |
| TYR | BTK | BTK_HUMAN | 5FBNC | Q06187 | 395 | 658 | 659.0 | 5WF:701,5WE:702 | Type1.5_Front,Allosteric | Inactive | DFGin | 6.234 | 13.485 | BLBplus | -138.97, 172.93 | 64.41, 21.2 | -64.91, 134.85 | 43.34, 89.93 | 78.28, -17.1 | out-out | out | 15.007 | Saltbr-out | 15.714 | HRD-in | -67.81, -54.89 | 86.66, -24.42 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.194 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | 143.31, -31.01 | APE9-dihe-in | -63.12, 135.49 | APE8-dihe-in | -76.38, 65.1 | APE8-rot-na | 32.35 | APE67-dihe-in | -72.98, -10.12 | -50.46, -47.16 | APE12-dist-na | 999.0 | APE11-dist-na | 17.831 | APE10-dist-na | 12.608 | APE9-dist-out | 8.181 | None | None | None | XRAY | 1.8 | 0.182 | 0.226 | C | 271 | 256 | 8 | 0 | 0 | 8 | [[402, 653]] | 1.0 | 5fbn | Homo sapiens | TYR_BTK_HUMAN | TYR | 6e-93 | 316.8 | 1 | 258 | 258 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 5FBND | Q06187 | 394 | 658 | 659.0 | 5WF:702,5WE:703,5WE:704,5WE:705 | Type1.5_Front,Allosteric,Allosteric,Allosteric | Inactive | DFGin | 6.25 | 13.472 | BLBplus | -137.76, 172.64 | 65.66, 19.16 | -62.24, 135.48 | 45.56, 88.91 | 74.32, -16.76 | out-out | out | 15.056 | Saltbr-out | 15.752 | HRD-in | -65.32, -54.88 | 86.04, -26.38 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.195 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 136.18 | APE8-dihe-in | -78.24, 64.6 | APE8-rot-na | 31.95 | APE67-dihe-in | -74.36, -8.3 | -50.81, -46.27 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.898 | None | None | None | XRAY | 1.8 | 0.182 | 0.226 | D | 271 | 255 | 10 | 0 | 0 | 10 | [[402, 653]] | 1.0 | 5fbn | Homo sapiens | TYR_BTK_HUMAN | TYR | 6e-93 | 316.8 | 1 | 258 | 258 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | DDR1 | DDR1_HUMAN | 5SAUA | Q08345 | 604 | 912 | 913.0 | 1IF:61000 | Type2 | Inactive | DFGout | 12.628 | 9.672 | BBAminus | -137.39, -170.54 | -153.95, 108.1 | -100.48, 5.9 | 289.81, 101.12 | 83.39, -174.73 | in-in | in | 8.355 | Saltbr-in | 2.869 | HRD-in | -71.66, -48.67 | 82.15, -10.52 | in-out-in | SNCioi | out-in | ActLoopNT-out | 18.139 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.56, 139.94 | APE9-dihe-in | -129.66, 123.98 | APE8-dihe-in | -80.56, 70.77 | APE8-rot-na | 35.49 | APE67-dihe-in | -73.85, -9.33 | -63.13, -31.85 | APE12-dist-na | 13.331 | APE11-dist-na | 10.312 | APE10-dist-na | 5.884 | APE9-dist-in | 7.555 | None | None | None | XRAY | 1.8 | 0.201 | 0.231 | A | 321 | 287 | 16 | 0 | 0 | 0 | [[610, 907]] | 1.0 | 5sau | Homo sapiens | TYR_DDR1_HUMAN | TYR | 1.4e-92 | 315.7 | 1 | 260 | 260 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | EPHA2 | EPHA2_HUMAN | 8BOCA | P29317 | 605 | 888 | 976.0 | QUF:1001 | Type2 | Inactive | DFGout | 13.583 | 10.813 | BBAminus | -139.62, -179.28 | -151.24, 106.28 | -78.98, -6.2 | 302.64, 171.21 | 84.05, 5.79 | in-in | in | 8.869 | Saltbr-in | 3.501 | HRD-in | -70.68, -54.7 | 83.35, -19.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 12.248 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.53, 160.37 | APE9-dihe-in | -116.01, 148.45 | APE8-dihe-in | -79.02, 97.78 | APE8-rot-na | 34.23 | APE67-dihe-in | -77.84, -8.8 | -56.96, -40.4 | APE12-dist-na | 12.844 | APE11-dist-na | 9.325 | APE10-dist-na | 7.892 | APE9-dist-in | 5.837 | None | None | None | XRAY | 1.9 | 0.248 | 0.286 | A | 306 | 271 | 13 | 0 | 0 | 0 | [[613, 873]] | 1.0 | 8boc | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2 | 261 | 260 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHB4 | EPHB4_HUMAN | 2X9FA | P54760 | 608 | 888 | 987.0 | X9F:1889 | Type1 | Inactive | DFGin | 6.208 | 14.33 | BLBminus | -134.1, -172.08 | 65.01, 71.96 | -106.66, 162.22 | 301.36, 107.12 | 163.16, 158.85 | in-in | in | 7.543 | Saltbr-in | 2.703 | HRD-in | -73.92, -48.13 | 77.71, -16.54 | in-out-in | SNCioi | out-in | ActLoopNT-out | 9.79 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -102.56, 149.08 | APE9-dihe-in | -55.67, 129.32 | APE8-dihe-in | -83.14, 89.74 | APE8-rot-na | 29.6 | APE67-dihe-in | -62.34, -22.56 | -52.45, -48.78 | APE12-dist-na | 8.363 | APE11-dist-na | 11.417 | APE10-dist-na | 15.416 | APE9-dist-in | 6.34 | Y774E | None | None | XRAY | 1.75 | 0.159 | 0.194 | A | 302 | 265 | 16 | 0 | 0 | 13 | [[615, 876]] | 1.0 | 2x9f | Homo sapiens | TYR_EPHB4_HUMAN | TYR | 3.9e-104 | 353.5 | 2 | 261 | 260 | 757 | 758 | 759 | 761 | 763 | 647 | 664 | 668 | 737 | 739 | 738 | 740 | 802 | 790 | 785 | 784 | 783 | 782 | 781 | 780 | 779 | 694 | Ephrin type-B receptor 4 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIA | P11362 | 458 | 764 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.058 | 13.436 | BLAplus | -111.91, 163.26 | 62.65, 26.85 | -80.22, -19.74 | 58.59, 88.0 | -94.12, 4.52 | in-in | in | 8.251 | Saltbr-in | 2.888 | HRD-in | -74.14, -50.3 | 78.02, -11.1 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.511 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -88.77, 149.44 | APE9-dihe-in | -108.01, 98.39 | APE8-dihe-out | -63.46, -15.87 | APE8-rot-na | 3.35 | APE67-dihe-in | -71.69, -10.38 | -55.45, -26.93 | APE12-dist-na | 17.216 | APE11-dist-na | 19.672 | APE10-dist-na | 16.685 | APE9-dist-out | 11.083 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | A | 310 | 307 | 0 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 9uhi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIB | P11362 | 458 | 763 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.213 | 12.738 | BLAplus | -108.15, 164.77 | 66.41, 24.28 | -84.34, -17.16 | 58.96, 83.83 | -89.87, -8.4 | in-in | in | 7.768 | Saltbr-in | 3.449 | HRD-in | -77.39, -52.67 | 76.89, -15.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -74.45, 132.66 | APE9-dihe-in | -102.74, 93.19 | APE8-dihe-out | -60.68, -21.29 | APE8-rot-na | 332.28 | APE67-dihe-in | -72.11, -2.38 | -56.87, -27.58 | APE12-dist-na | 17.352 | APE11-dist-na | 20.682 | APE10-dist-na | 16.965 | APE9-dist-out | 11.364 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | B | 310 | 286 | 20 | 0 | 0 | 7 | [[478, 756]] | 1.0 | 9uhi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FA | P11362 | 464 | 765 | 822.0 | C4F:1 | Type1.5_Back | Inactive | DFGin | 5.114 | 13.318 | BLAplus | -110.44, 159.78 | 58.59, 34.58 | -81.02, -11.31 | 51.22, 81.2 | -119.48, 23.64 | in-out | in | 7.866 | Saltbr-out | 4.632 | HRD-in | -67.82, -57.48 | 84.79, -17.47 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.069 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.31, 173.6 | APE9-dihe-in | -111.71, 110.92 | APE8-dihe-out | -49.57, -28.9 | APE8-rot-na | 335.93 | APE67-dihe-in | -76.49, -6.67 | -57.78, -16.15 | APE12-dist-na | 19.292 | APE11-dist-na | 21.121 | APE10-dist-na | 19.395 | APE9-dist-out | 11.757 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | A | 302 | 290 | 12 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 3c4f | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FB | P11362 | 464 | 765 | 822.0 | C4F:2 | Type1.5_Back | Inactive | DFGin | 5.186 | 13.096 | BLAplus | -113.87, 161.2 | 54.21, 44.76 | -88.95, -14.38 | 49.14, 89.01 | -114.94, 24.21 | in-in | in | 7.831 | Saltbr-in | 3.248 | HRD-in | -69.91, -54.09 | 86.4, -33.67 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.934 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.54, 164.12 | APE9-dihe-in | -103.97, 111.75 | APE8-dihe-out | -49.46, -30.24 | APE8-rot-na | 330.07 | APE67-dihe-in | -74.8, -7.14 | -56.82, -17.81 | APE12-dist-na | 19.37 | APE11-dist-na | 21.296 | APE10-dist-na | 19.671 | APE9-dist-out | 11.643 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | B | 302 | 290 | 12 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 3c4f | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5EW8A | P11362 | 464 | 765 | 822.0 | 5SF:803 | Type1.5_Back | Inactive | DFGin | 4.948 | 13.265 | BLAplus | -106.94, 161.6 | 53.73, 34.99 | -75.93, -13.84 | 56.0, 83.89 | -112.21, 7.75 | in-in | in | 7.954 | Saltbr-in | 2.801 | HRD-in | -68.23, -51.53 | 79.48, -14.26 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.067 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.87, 162.8 | APE9-dihe-in | -100.01, 112.78 | APE8-dihe-out | -57.6, -21.18 | APE8-rot-na | 333.77 | APE67-dihe-in | -70.4, -6.07 | -56.33, -25.26 | APE12-dist-na | 19.37 | APE11-dist-na | 20.743 | APE10-dist-na | 19.216 | APE9-dist-out | 11.882 | None | None | None | XRAY | 1.63 | 0.186 | 0.206 | A | 309 | 291 | 11 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 5ew8 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5EW8B | P11362 | 461 | 765 | 822.0 | 5SF:802 | Type1.5_Back | Inactive | DFGin | 5.002 | 13.124 | BLAplus | -109.75, 160.16 | 55.05, 34.73 | -78.35, -12.87 | 54.65, 85.31 | -106.64, 12.94 | in-in | in | 7.88 | Saltbr-in | 2.807 | HRD-in | -67.52, -52.32 | 78.89, -12.97 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.38 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.81, 162.42 | APE9-dihe-in | -99.2, 111.94 | APE8-dihe-out | -57.42, -21.49 | APE8-rot-na | 334.53 | APE67-dihe-in | -69.99, -6.88 | -56.65, -24.13 | APE12-dist-na | 19.902 | APE11-dist-na | 21.169 | APE10-dist-na | 19.654 | APE9-dist-out | 11.767 | None | None | None | XRAY | 1.63 | 0.186 | 0.206 | B | 309 | 290 | 15 | 0 | 0 | 2 | [[478, 756]] | 1.0 | 5ew8 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7WCLA | P11362 | 459 | 764 | 822.0 | 8ZF:60801 | Type1.5_Back | Inactive | DFGin | 5.032 | 13.511 | BLAplus | -110.65, 158.43 | 54.71, 42.71 | -89.1, -11.93 | 53.54, 87.56 | -114.63, 26.86 | in-in | in | 8.234 | Saltbr-in | 2.943 | HRD-in | -65.51, -45.04 | 70.13, -0.28 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.98 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.05, 142.67 | APE9-dihe-in | -99.82, 98.85 | APE8-dihe-out | -66.04, -10.56 | APE8-rot-na | 23.45 | APE67-dihe-in | -75.78, -2.11 | -60.96, -29.19 | APE12-dist-na | 16.725 | APE11-dist-na | 19.067 | APE10-dist-na | 16.226 | APE9-dist-out | 11.223 | C584S | None | None | XRAY | 2.495 | 0.195 | 0.23 | A | 310 | 306 | 0 | 0 | 0 | 0 | [[478, 756]] | 1.0 | 7wcl | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7WCLB | P11362 | 458 | 763 | 822.0 | 8ZF:60801 | Type1.5_Back | Inactive | DFGin | 5.686 | 13.297 | BLAplus | -116.0, 164.36 | 53.53, 38.11 | -89.51, -19.74 | 50.41, 88.95 | -102.65, 11.92 | in-in | in | 8.381 | Saltbr-in | 2.804 | HRD-in | -77.55, -44.61 | 69.5, -1.67 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -124.03, 166.88 | APE9-dihe-in | -112.63, 116.79 | APE8-dihe-out | -58.21, -18.36 | APE8-rot-na | 340.54 | APE67-dihe-in | -81.23, 2.92 | -65.55, -20.31 | APE12-dist-na | 18.6 | APE11-dist-na | 21.605 | APE10-dist-na | 19.498 | APE9-dist-out | 11.402 | C584S | None | None | XRAY | 2.495 | 0.195 | 0.23 | B | 310 | 285 | 21 | 0 | 0 | 8 | [[478, 756]] | 1.0 | 7wcl | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1 | 260 | 260 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDTA | P22607 | 457 | 756 | 806.0 | MLT:61001,MLT:61002,WGF:61003 | Allosteric,Allosteric,Type1.5_Front | Inactive | DFGin | 5.441 | 13.493 | BLAplus | -114.8, 158.79 | 55.69, 43.2 | -82.19, -34.37 | 42.84, 89.08 | -83.27, -4.41 | in-out | in | 8.383 | Saltbr-out | 5.287 | HRD-in | -68.34, -46.54 | 75.89, -9.4 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.921 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 112.29 | APE8-dihe-out | -63.06, -32.23 | APE8-rot-na | 340.92 | APE67-dihe-in | -68.35, -26.42 | -62.13, -28.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.198 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | A | 297 | 284 | 4 | 0 | 0 | 4 | [[472, 750]] | 1.0 | 8udt | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1 | 260 | 260 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDTB | P22607 | 457 | 754 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.258 | 13.71 | BLAplus | -108.64, 157.87 | 56.15, 40.62 | -79.39, -35.54 | 45.72, 88.06 | -80.67, 0.1 | in-out | in | 8.445 | Saltbr-out | 5.398 | HRD-in | -67.98, -43.8 | 74.91, -8.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.867 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -64.67 | APE9-dihe-out | -68.82, -39.67 | APE8-dihe-out | -56.45, -17.85 | APE8-rot-na | 337.42 | APE67-dihe-in | -61.76, -27.35 | -59.02, -40.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.666 | APE9-dist-out | 10.854 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | B | 297 | 283 | 3 | 0 | 0 | 3 | [[472, 750]] | 1.0 | 8udt | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1 | 260 | 260 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDTC | P22607 | 457 | 756 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.258 | 13.824 | BLAplus | -109.74, 157.08 | 55.91, 40.67 | -78.94, -35.79 | 45.97, 87.77 | -81.04, -4.46 | in-out | in | 8.545 | Saltbr-out | 4.103 | HRD-in | -68.09, -46.3 | 75.11, -4.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.87 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -150.08 | APE9-dihe-out | -67.3, -42.56 | APE8-dihe-out | -46.98, -31.66 | APE8-rot-na | 333.46 | APE67-dihe-in | -60.08, -29.46 | -58.03, -43.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.405 | APE9-dist-out | 11.049 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | C | 297 | 284 | 4 | 0 | 0 | 4 | [[472, 750]] | 1.0 | 8udt | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1 | 260 | 260 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR4 | FGFR4_HUMAN | 7WCXA | P22455 | 453 | 752 | 802.0 | 90F:801 | Type1 | Inactive | DFGin | 5.263 | 13.141 | BLAplus | -114.81, 160.0 | 54.39, 48.08 | -89.68, -16.38 | 44.55, 83.39 | -109.65, 26.27 | in-in | in | 7.792 | Saltbr-in | 2.511 | HRD-in | -76.2, -43.73 | 72.01, -8.39 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.644 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -80.24, 137.24 | APE9-dihe-in | -109.54, 93.42 | APE8-dihe-out | -57.65, -19.77 | APE8-rot-na | 335.57 | APE67-dihe-in | -71.93, -5.42 | -64.19, -25.82 | APE12-dist-na | 19.074 | APE11-dist-na | 20.85 | APE10-dist-na | 16.822 | APE9-dist-out | 11.904 | C477A,R664E | None | None | XRAY | 2.175 | 0.173 | 0.221 | A | 309 | 300 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 7wcx | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 7e-101 | 342.8 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7WCWA | P22455 | 453 | 752 | 802.0 | 90F:801 | Type1 | Inactive | DFGin | 5.839 | 13.063 | BLAplus | -123.48, 161.59 | 54.95, 50.1 | -96.76, -24.53 | 39.59, 83.16 | -101.63, 31.89 | in-in | in | 7.582 | Saltbr-in | 3.4 | HRD-in | -77.43, -45.16 | 72.65, -7.54 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.633 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -81.49, 135.61 | APE9-dihe-in | -107.87, 94.77 | APE8-dihe-out | -59.45, -18.22 | APE8-rot-na | 336.81 | APE67-dihe-in | -74.15, -1.22 | -67.3, -23.03 | APE12-dist-na | 19.435 | APE11-dist-na | 20.996 | APE10-dist-na | 16.929 | APE9-dist-out | 11.84 | C477A,R664E | None | None | XRAY | 2.317 | 0.179 | 0.221 | A | 309 | 300 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 7wcw | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.9e-100 | 341.4 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 6JPJA | P22455 | 454 | 752 | 802.0 | FGF:800 | Type1 | Inactive | DFGin | 5.301 | 12.658 | BLAplus | -117.71, 161.57 | 53.08, 42.72 | -89.02, -4.4 | 50.47, 87.12 | -117.52, 24.43 | in-in | in | 7.247 | Saltbr-in | 2.318 | HRD-out | -71.89, 98.16 | -78.45, 15.53 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.002 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -85.03, 139.81 | APE9-dihe-in | -112.83, 87.62 | APE8-dihe-out | -50.76, -19.28 | APE8-rot-na | 332.54 | APE67-dihe-in | -80.03, 5.83 | -68.35, -18.64 | APE12-dist-na | 19.294 | APE11-dist-na | 21.068 | APE10-dist-na | 17.129 | APE9-dist-out | 12.054 | C477A,R664E | None | None | XRAY | 2.638 | 0.198 | 0.243 | A | 311 | 299 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 6jpj | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.3e-100 | 341.9 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7VJLA | P22455 | 454 | 753 | 802.0 | 7IF:801 | Type1 | Inactive | DFGin | 5.301 | 12.42 | BLAplus | -114.78, 170.3 | 57.71, 40.42 | -94.32, 21.48 | 55.77, 90.38 | -107.29, 999.0 | in-in | in | 7.485 | Saltbr-in | 2.904 | HRD-out | -79.19, -58.83 | -98.34, 2.36 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 2.26 | APE8-rot-na | 31.94 | APE67-dihe-in | -59.38, -20.97 | -56.11, -39.64 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.9 | 0.212 | 0.273 | A | 301 | 263 | 37 | 0 | 0 | 19 | [[467, 745]] | 1.0 | 7vjl | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.1e-100 | 342.2 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7VJLB | P22455 | 453 | 753 | 802.0 | 7IF:801 | Type1 | Inactive | DFGin | 5.405 | 13.204 | BLAplus | -123.58, 175.88 | 60.77, 35.86 | -95.6, 5.83 | 48.51, 81.65 | -122.94, 999.0 | in-in | in | 7.876 | Saltbr-in | 2.665 | HRD-out | -72.76, -57.66 | -103.85, -18.8 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 6.57 | APE8-rot-na | 30.25 | APE67-dihe-in | -55.58, -34.43 | -70.09, -36.28 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.9 | 0.212 | 0.273 | B | 301 | 266 | 35 | 0 | 0 | 19 | [[467, 745]] | 1.0 | 7vjl | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.1e-100 | 342.2 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 6YI8A | P22455 | 453 | 753 | 802.0 | FGF:801 | Type1 | Inactive | DFGin | 5.052 | 12.585 | BLAplus | -114.37, 162.1 | 61.01, 37.7 | -86.22, -22.44 | 57.75, 86.82 | -88.83, -1.63 | in-in | in | 7.21 | Saltbr-in | 2.807 | HRD-in | -68.35, -54.97 | 79.66, -18.38 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 137.99 | APE9-dihe-in | -91.08, 144.79 | APE8-dihe-in | -80.88, 56.75 | APE8-rot-na | 32.63 | APE67-dihe-in | -69.74, -13.54 | -50.67, -37.69 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 19.129 | APE9-dist-out | 9.562 | None | None | None | XRAY | 2.13 | 0.198 | 0.231 | A | 307 | 277 | 24 | 0 | 0 | 15 | [[467, 745]] | 1.0 | 6yi8 | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.1 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 6YI8B | P22455 | 451 | 752 | 802.0 | FGF:801 | Type1 | Inactive | DFGin | 5.551 | 13.074 | BLAplus | -114.83, 168.14 | 49.73, 54.77 | -99.35, -32.03 | 46.0, 89.99 | -71.98, 999.0 | in-in | in | 7.399 | Saltbr-in | 2.814 | HRD-in | -67.69, -51.4 | 79.31, -36.01 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 133.49 | APE8-dihe-in | -88.73, 63.1 | APE8-rot-na | 25.93 | APE67-dihe-in | -70.74, -12.22 | -53.82, -35.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.081 | None | None | None | XRAY | 2.13 | 0.198 | 0.231 | B | 307 | 270 | 32 | 0 | 0 | 18 | [[467, 745]] | 1.0 | 6yi8 | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.1 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 7WCTA | P22455 | 453 | 752 | 802.0 | 90F:801 | Type1 | Inactive | DFGin | 5.499 | 13.008 | BLAplus | -115.75, 158.15 | 54.59, 44.67 | -82.33, -22.35 | 42.51, 87.35 | -106.03, 33.12 | in-in | in | 7.476 | Saltbr-in | 2.881 | HRD-in | -76.31, -44.07 | 70.33, -3.05 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.497 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -84.18, 139.68 | APE9-dihe-in | -111.32, 93.14 | APE8-dihe-out | -55.09, -20.87 | APE8-rot-na | 333.3 | APE67-dihe-in | -74.74, -3.5 | -65.15, -23.14 | APE12-dist-na | 19.463 | APE11-dist-na | 21.045 | APE10-dist-na | 17.074 | APE9-dist-out | 11.772 | R664E | None | None | XRAY | 2.106 | 0.184 | 0.217 | A | 311 | 300 | 0 | 0 | 0 | 0 | [[467, 745]] | 1.0 | 7wct | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.9e-100 | 341.4 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 5XFJA | P22455 | 453 | 750 | 802.0 | 6LF:801 | Type1 | Inactive | DFGin | 5.021 | 13.251 | None | -115.6, 133.16 | 70.83, 138.96 | -157.69, 175.22 | 19.16, 82.91 | -161.9, 174.05 | in-out | in | 8.31 | Saltbr-out | 4.274 | HRD-out | -142.96, 112.57 | -85.34, -51.29 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -47.84 | APE8-dihe-in | -93.04, 75.41 | APE8-rot-na | 34.31 | APE67-dihe-in | -59.81, -17.88 | -81.83, -32.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.229 | V550M | None | None | XRAY | 3.25 | 0.284 | 0.336 | A | 311 | 266 | 32 | 0 | 0 | 17 | [[467, 745]] | 1.0 | 5xfj | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 4.5e-101 | 343.4 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 5XFFA | P22455 | 453 | 750 | 802.0 | 6LF:801 | Type1 | Inactive | DFGin | 7.251 | 13.8 | None | -91.81, 157.14 | 71.12, 141.83 | -151.53, 140.75 | 303.34, 100.5 | -174.03, 158.26 | in-in | in | 7.907 | Saltbr-in | 3.562 | HRD-out | -144.83, 101.6 | -75.14, -41.6 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -18.13 | APE8-dihe-in | -83.47, 67.75 | APE8-rot-na | 31.32 | APE67-dihe-in | -75.73, 1.3 | -73.66, -27.62 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.541 | V550L | None | None | XRAY | 2.7 | 0.27 | 0.32 | A | 311 | 269 | 29 | 0 | 0 | 17 | [[467, 745]] | 1.0 | 5xff | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.0 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 5JKGA | P22455 | 453 | 750 | 802.0 | 6LF:801 | Type1 | Inactive | DFGin | 4.645 | 13.415 | None | -80.35, 138.57 | 42.13, 154.03 | -151.26, -44.79 | 29.5, 89.83 | 59.57, 154.84 | in-in | in | 7.788 | Saltbr-in | 2.748 | HRD-out | -157.35, 80.6 | -45.38, -51.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -51.98 | APE8-dihe-in | -77.75, 74.49 | APE8-rot-na | 28.85 | APE67-dihe-in | -78.7, 0.61 | -72.33, -28.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.405 | None | None | None | XRAY | 2.352 | 0.237 | 0.277 | A | 311 | 266 | 32 | 0 | 0 | 17 | [[467, 745]] | 1.0 | 5jkg | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 8.4e-101 | 342.6 | 1 | 261 | 261 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FLT3 | FLT3_HUMAN | 6JQRA | P36888 | 571 | 951 | 993.0 | C6F:1001 | Type1 | Inactive | DFGout | 15.394 | 10.885 | None | -119.73, 157.71 | -104.23, 115.68 | 77.2, 999.0 | 255.94, 91.42 | 999.0, 999.0 | in-in | in | 8.326 | Saltbr-in | 2.804 | HRD-out | -98.26, 117.82 | -85.48, 11.47 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.05, 100.76 | APE9-dihe-in | -103.87, 123.04 | APE8-dihe-in | -78.74, 70.62 | APE8-rot-na | 34.5 | APE67-dihe-in | -69.1, -11.06 | -54.04, -46.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.223 | None | None | None | XRAY | 2.2 | 0.181 | 0.213 | A | 330 | 301 | 29 | 0 | 0 | 6 | [[610, 945]] | 1.0 | 6jqr | Homo sapiens | TYR_FLT3_HUMAN | TYR | 8.5e-103 | 349.1 | 1 | 259 | 259 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| TYR | HCK | HCK_HUMAN | 3VS4A | P08631 | 81 | 526 | 526.0 | VSF:60603 | Type1.5_Back | Inactive | DFGin | 5.296 | 12.617 | BLBplus | -129.05, 156.5 | 78.18, 7.28 | -55.31, 122.08 | 48.34, 94.72 | 91.65, -36.18 | out-out | out | 13.53 | Saltbr-out | 14.391 | HRD-in | -89.51, -57.9 | 84.08, -11.13 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.875 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 47.3 | APE8-dihe-in | -93.7, 67.91 | APE8-rot-na | 28.82 | APE67-dihe-in | -68.45, -16.47 | -64.44, -22.55 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.697 | Q523E,Q524E,Q525I | PTR522 | PTR522 | XRAY | 2.747 | 0.265 | 0.265 | A | 454 | 429 | 11 | 0 | 0 | 11 | [[262, 513]] | 1.0 | 3vs4 | Homo sapiens | TYR_HCK_HUMAN | TYR | 1.4e-95 | 325.6 | 1 | 260 | 260 | 398 | 399 | 400 | 402 | 404 | 290 | 305 | 309 | 378 | 380 | 379 | 381 | 439 | 427 | 422 | 421 | 420 | 419 | 418 | 417 | 416 | 334 | Tyrosine-protein kinase HCK |
| TYR | HCK | HCK_HUMAN | 3VS4B | P08631 | 81 | 526 | 526.0 | VSF:60603 | Type1.5_Back | Inactive | DFGin | 5.285 | 12.665 | BLBplus | -120.89, 167.83 | 61.49, 15.86 | -62.02, 121.53 | 47.24, 95.4 | 75.03, 10.7 | out-out | out | 13.766 | Saltbr-out | 15.042 | HRD-in | -94.45, -46.27 | 74.87, -7.2 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.135 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 48.23 | APE8-dihe-in | -84.31, 74.96 | APE8-rot-na | 34.0 | APE67-dihe-in | -71.24, -2.76 | -88.69, -13.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.595 | Q523E,Q524E,Q525I | PTR522 | PTR522 | XRAY | 2.747 | 0.265 | 0.265 | B | 454 | 434 | 12 | 0 | 0 | 12 | [[262, 513]] | 1.0 | 3vs4 | Homo sapiens | TYR_HCK_HUMAN | TYR | 1.4e-95 | 325.6 | 1 | 260 | 260 | 398 | 399 | 400 | 402 | 404 | 290 | 305 | 309 | 378 | 380 | 379 | 381 | 439 | 427 | 422 | 421 | 420 | 419 | 418 | 417 | 416 | 334 | Tyrosine-protein kinase HCK |
| TYR | JAK2-1 | JAK2_HUMAN | 8B9EA | O60674 | 536 | 809 | 1132.0 | Q7F:1003 | Type1 | Pseudo | DFGin | 5.769 | 13.226 | None | -72.27, 175.04 | -67.31, 162.54 | -76.41, -26.42 | 340.6, 33.67 | 78.05, -163.23 | out-na | out | 11.726 | Saltbr-na | 999.0 | HRD-in | -83.9, -60.17 | 88.41, -6.41 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 8.95 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -67.18, -39.02 | APE9-dihe-out | -59.74, -28.13 | APE8-dihe-out | -86.36, 6.28 | APE8-rot-na | 284.57 | APE67-dihe-out | -105.41, 26.85 | -68.63, 134.78 | APE12-dist-na | 9.613 | APE11-dist-na | 11.316 | APE10-dist-na | 15.854 | APE9-dist-out | 12.106 | W777A,F794H | None | None | XRAY | 1.5 | 0.17 | 0.194 | A | 289 | 274 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 8b9e | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 6.4e-64 | 221.7 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 8B9HA | O60674 | 536 | 809 | 1132.0 | Q7F:901 | Type1 | Pseudo | DFGin | 6.01 | 13.307 | None | -84.93, -177.89 | -74.12, 157.3 | -67.76, -31.57 | 343.4, 32.07 | 81.26, -168.8 | out-na | out | 12.097 | Saltbr-na | 999.0 | HRD-in | -82.25, -60.3 | 91.76, -5.32 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.143 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -65.85, -39.85 | APE9-dihe-out | -62.27, -26.85 | APE8-dihe-out | -86.04, 1.76 | APE8-rot-na | 292.25 | APE67-dihe-out | -100.68, 23.58 | -62.84, 136.16 | APE12-dist-na | 9.712 | APE11-dist-na | 11.434 | APE10-dist-na | 15.933 | APE9-dist-out | 12.428 | W659A,W777A,F794H | None | None | XRAY | 1.5 | 0.182 | 0.208 | A | 289 | 274 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 8b9h | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 1.9e-64 | 223.4 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | KDR | VGFR2_HUMAN | 3VO3A | P35968 | 812 | 1168 | 1356.0 | 0KF:2001 | Type2 | Inactive | DFGout | 16.448 | 8.215 | None | -125.16, 179.81 | -141.05, 99.79 | -70.03, -34.74 | 215.55, 55.41 | 59.77, -120.61 | in-in | in | 7.357 | Saltbr-in | 2.898 | HRD-in | -84.45, -53.71 | 76.95, -3.4 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.477 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.91, 109.54 | APE9-dihe-in | -120.7, 147.5 | APE8-dihe-in | -78.09, 65.8 | APE8-rot-na | 32.33 | APE67-dihe-in | -67.73, -12.3 | -53.4, -39.21 | APE12-dist-na | 17.03 | APE11-dist-na | 14.067 | APE10-dist-na | 11.393 | APE9-dist-in | 7.997 | None | None | None | XRAY | 1.52 | 0.162 | 0.182 | A | 318 | 303 | 4 | 0 | 0 | 0 | [[834, 1162]] | 1.0 | 3vo3 | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.2e-100 | 340.3 | 1 | 260 | 260 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| TYR | KDR | VGFR2_HUMAN | 1YWNA | P35968 | 820 | 1171 | 1356.0 | LIF:60301 | Type1 | Inactive | None | 999.0 | 999.0 | None | -128.91, 171.96 | -143.62, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 7.21 | Saltbr-in | 2.725 | HRD-in | -77.88, -50.07 | 82.87, -17.6 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -141.39, 161.44 | APE9-dihe-in | -104.18, 100.32 | APE8-dihe-out | -56.09, -24.71 | APE8-rot-na | 336.02 | APE67-dihe-in | -70.59, -14.0 | -51.58, -32.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.239 | E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.71 | 0.206 | 0.23 | A | 316 | 281 | 21 | 0 | 0 | 6 | [[834, 1162]] | 1.0 | 1ywn | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1 | 260 | 260 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| TYR | LCK | LCK_HUMAN | 2ZM1A | P06239 | 231 | 501 | 509.0 | KSF:513 | Type1 | Active | DFGin | 6.499 | 14.193 | BLAminus | -132.48, -160.42 | 31.13, 88.01 | -99.25, 22.14 | 293.45, 97.67 | -69.47, -32.89 | in-in | in | 8.512 | Saltbr-in | 2.933 | HRD-in | -100.89, -51.07 | 73.44, -7.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.929 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.43, 148.33 | APE9-dihe-in | -138.82, 152.04 | APE8-dihe-in | -57.54, 117.05 | APE8-rot-na | 333.13 | APE67-dihe-in | -71.51, -24.6 | -61.57, -39.74 | APE12-dist-na | 15.101 | APE11-dist-na | 10.35 | APE10-dist-na | 13.014 | APE9-dist-in | 6.822 | None | PTR394 | PTR394 | XRAY | 2.1 | 0.172 | 0.232 | A | 285 | 271 | 0 | 0 | 0 | 0 | [[245, 496]] | 1.0 | 2zm1 | Homo sapiens | TYR_LCK_HUMAN | TYR | 1.5e-94 | 322.1 | 1 | 260 | 260 | 381 | 382 | 383 | 385 | 387 | 273 | 288 | 292 | 361 | 363 | 362 | 364 | 422 | 410 | 405 | 404 | 403 | 402 | 401 | 400 | 399 | 317 | Tyrosine-protein kinase Lck |
| TYR | MERTK | MERTK_HUMAN | 9BHIA | Q12866 | 578 | 864 | 999.0 | A1APF:60901 | Type1.5_Front | Inactive | DFGin | 6.992 | 12.805 | BLAminus | -138.66, -158.87 | 44.96, 74.5 | -90.39, 18.73 | 305.52, 137.7 | -55.48, -30.3 | out-out | out | 13.615 | Saltbr-out | 13.031 | HRD-in | -81.75, -51.8 | 68.35, 6.62 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.82 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.15, 11.33 | APE9-dihe-in | -72.53, 150.77 | APE8-dihe-in | -64.75, 117.67 | APE8-rot-na | 25.92 | APE67-dihe-in | -73.91, -0.64 | -53.67, -34.29 | APE12-dist-na | 7.154 | APE11-dist-na | 12.056 | APE10-dist-na | 11.657 | APE9-dist-in | 6.71 | None | None | None | XRAY | 2.07 | 0.211 | 0.23 | A | 323 | 278 | 9 | 0 | 0 | 2 | [[587, 856]] | 1.0 | 9bhi | Homo sapiens | TYR_MERTK_HUMAN | TYR | 1.6e-92 | 315.5 | 2 | 261 | 260 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| TYR | MERTK | MERTK_HUMAN | 7AB1A | Q12866 | 571 | 862 | 999.0 | C6F:60901 | Type1 | Inactive | DFGin | 5.872 | 13.527 | None | -150.27, 178.21 | 48.78, 48.66 | -107.87, 999.0 | 41.9, 85.18 | 999.0, 999.0 | out-out | out | 12.844 | Saltbr-out | 9.566 | HRD-in | -84.92, -52.07 | 85.67, -41.55 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 62.29 | APE8-rot-na | 36.31 | APE67-dihe-in | -65.53, -14.5 | -57.08, -42.11 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | K591R,K693R,K702R,K856R | None | None | XRAY | 1.93 | 0.237 | 0.298 | A | 298 | 267 | 25 | 0 | 0 | 20 | [[587, 856]] | 1.0 | 7ab1 | Homo sapiens | TYR_MERTK_HUMAN | TYR | 2.3e-92 | 314.9 | 2 | 260 | 259 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| TYR | MET | MET_HUMAN | 3ZCLA | P08581 | 1052 | 1345 | 1390.0 | 5TF:1 | Type1 | Inactive | DFGin | 5.341 | 14.033 | BLBplus | -130.37, -159.34 | 48.43, 53.41 | -147.61, 165.56 | 74.15, 92.01 | 59.61, -131.84 | out-out | out | 14.636 | Saltbr-out | 12.785 | HRD-in | -76.45, -51.81 | 82.5, -13.86 | out-out-in | SNCooi | out-in | ActLoopNT-out | 10.735 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.5, 109.91 | APE9-dihe-in | -127.18, 152.9 | APE8-dihe-in | -78.54, 68.73 | APE8-rot-na | 30.54 | APE67-dihe-in | -82.79, -0.65 | -60.11, -28.04 | APE12-dist-na | 22.937 | APE11-dist-na | 18.131 | APE10-dist-na | 17.771 | APE9-dist-in | 7.357 | None | None | None | XRAY | 1.4 | 0.194 | 0.211 | A | 306 | 291 | 3 | 0 | 0 | 0 | [[1078, 1339]] | 1.0 | 3zcl | Homo sapiens | TYR_MET_HUMAN | TYR | 6.7e-92 | 313.6 | 2 | 260 | 259 | 1221 | 1222 | 1223 | 1225 | 1227 | 1110 | 1127 | 1131 | 1201 | 1203 | 1202 | 1204 | 1265 | 1253 | 1248 | 1247 | 1246 | 1245 | 1244 | 1243 | 1242 | 1158 | Hepatocyte growth factor receptor |
| TYR | MET | MET_HUMAN | 4MXCA | P08581 | 1052 | 1346 | 1390.0 | DWF:1401 | Type2 | Inactive | DFGout | 14.41 | 10.337 | BBAminus | -151.35, -174.18 | -156.99, 122.43 | -67.95, -16.78 | 287.52, 70.23 | 58.23, -116.98 | in-in | in | 8.929 | Saltbr-in | 3.515 | HRD-in | -73.25, -51.06 | 80.68, -17.87 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.287 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -88.68, 108.68 | APE9-dihe-in | -118.71, 133.81 | APE8-dihe-in | -79.71, 72.93 | APE8-rot-na | 28.81 | APE67-dihe-in | -75.71, -5.79 | -60.94, -31.89 | APE12-dist-na | 999.0 | APE11-dist-na | 13.628 | APE10-dist-na | 10.273 | APE9-dist-in | 7.344 | None | None | None | XRAY | 1.632 | 0.18 | 0.207 | A | 319 | 290 | 5 | 0 | 0 | 5 | [[1078, 1339]] | 1.0 | 4mxc | Homo sapiens | TYR_MET_HUMAN | TYR | 7.7e-92 | 313.7 | 2 | 260 | 259 | 1221 | 1222 | 1223 | 1225 | 1227 | 1110 | 1127 | 1131 | 1201 | 1203 | 1202 | 1204 | 1265 | 1253 | 1248 | 1247 | 1246 | 1245 | 1244 | 1243 | 1242 | 1158 | Hepatocyte growth factor receptor |
| TYR | NTRK1 | NTRK1_HUMAN | 5H3QA | P04629 | 484 | 796 | 796.0 | 7HF:1001 | Type1 | Inactive | DFGout | 12.708 | 6.583 | BBAminus | 172.54, 156.19 | -157.42, 160.24 | -99.39, 17.97 | 295.12, 97.4 | 79.34, 29.52 | in-out | in | 9.447 | Saltbr-out | 5.851 | HRD-in | -81.9, -52.58 | 77.47, -12.71 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.801 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -128.94, 112.39 | APE9-dihe-in | -107.73, 133.13 | APE8-dihe-in | -79.15, 63.42 | APE8-rot-na | 34.45 | APE67-dihe-in | -63.33, -18.08 | -61.61, -34.65 | APE12-dist-na | 13.748 | APE11-dist-na | 15.2 | APE10-dist-na | 10.681 | APE9-dist-in | 7.568 | None | None | None | XRAY | 2.1 | 0.19 | 0.215 | A | 324 | 303 | 10 | 0 | 0 | 0 | [[510, 783]] | 1.0 | 5h3q | Homo sapiens | TYR_NTRK1_HUMAN | TYR | 2.4e-100 | 341.1 | 2 | 260 | 259 | 667 | 668 | 669 | 671 | 673 | 544 | 560 | 564 | 647 | 649 | 648 | 650 | 709 | 697 | 692 | 691 | 690 | 689 | 688 | 687 | 686 | 590 | High affinity nerve growth factor receptor |
| TYR | NTRK1 | NTRK1_HUMAN | 5KMJA | P04629 | 486 | 795 | 796.0 | 6UF:901 | Type3 | Inactive | DFGout | 12.074 | 7.602 | None | 156.98, 152.76 | -155.56, 161.93 | -106.33, 28.22 | 308.11, 127.92 | 67.17, 26.59 | in-in | in | 9.714 | Saltbr-in | 2.772 | HRD-in | -79.87, -55.53 | 78.72, -12.42 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.107 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -122.86, 120.05 | APE9-dihe-in | -107.69, 130.38 | APE8-dihe-in | -83.48, 63.94 | APE8-rot-na | 32.0 | APE67-dihe-in | -63.64, -21.11 | -52.37, -37.83 | APE12-dist-na | 15.016 | APE11-dist-na | 15.494 | APE10-dist-na | 11.096 | APE9-dist-in | 7.6 | None | None | None | XRAY | 2.04 | 0.196 | 0.226 | A | 329 | 300 | 6 | 0 | 0 | 0 | [[510, 783]] | 1.0 | 5kmj | Homo sapiens | TYR_NTRK1_HUMAN | TYR | 2.5e-100 | 341.0 | 2 | 260 | 259 | 667 | 668 | 669 | 671 | 673 | 544 | 560 | 564 | 647 | 649 | 648 | 650 | 709 | 697 | 692 | 691 | 690 | 689 | 688 | 687 | 686 | 590 | High affinity nerve growth factor receptor |
| TYR | PTK2 | FAK1_HUMAN | 4EBWA | Q05397 | 411 | 686 | 1052.0 | 0PF:700 | Type1 | Inactive | DFGinter | 10.52 | 8.023 | None | -156.77, 167.19 | -119.55, 38.35 | -154.8, 160.1 | 57.14, 97.67 | -105.09, 155.15 | in-in | in | 7.232 | Saltbr-in | 3.021 | HRD-out | -85.85, 108.83 | -92.42, -13.42 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 105.2 | APE9-dihe-in | -103.42, 143.85 | APE8-dihe-in | -74.96, 72.04 | APE8-rot-na | 29.05 | APE67-dihe-in | -70.29, -24.24 | -52.29, -39.56 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 17.857 | APE9-dist-out | 9.391 | None | None | None | XRAY | 2.65 | 0.186 | 0.273 | A | 304 | 259 | 17 | 0 | 0 | 15 | [[422, 678]] | 1.0 | 4ebw | Homo sapiens | TYR_PTK2_HUMAN | TYR | 4.7e-93 | 317.2 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | SYK | KSYK_HUMAN | 5LMBA | P43405 | 364 | 634 | 635.0 | 6ZF:701 | Type1 | Active | DFGin | 6.448 | 14.283 | BLAminus | -131.02, -173.87 | 62.28, 69.39 | -93.16, 19.0 | 290.08, 82.25 | -59.68, -28.46 | in-in | in | 7.696 | Saltbr-in | 2.454 | HRD-in | -78.06, -53.9 | 76.38, 4.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.963 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.66, 104.96 | APE9-dihe-in | -108.73, 152.4 | APE8-dihe-in | -79.7, 70.25 | APE8-rot-na | 31.84 | APE67-dihe-in | -69.34, -16.13 | -51.43, -34.69 | APE12-dist-na | 13.073 | APE11-dist-na | 10.546 | APE10-dist-na | 11.448 | APE9-dist-in | 6.959 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | A | 277 | 265 | 6 | 0 | 0 | 0 | [[370, 628]] | 1.0 | 5lmb | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 5LMBB | P43405 | 364 | 630 | 635.0 | 6ZF:701 | Type1 | None | DFGin | 6.542 | 14.207 | BLAminus | -133.05, -174.7 | 62.98, 72.21 | -97.02, 21.38 | 290.54, 88.36 | -62.52, -32.46 | in-in | in | 7.737 | Saltbr-in | 2.556 | HRD-in | -77.26, -52.74 | 74.6, 8.57 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.872 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 129.43 | APE8-dihe-in | -80.7, 73.18 | APE8-rot-na | 30.16 | APE67-dihe-in | -64.42, -18.25 | -49.18, -37.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.948 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | B | 277 | 262 | 5 | 0 | 0 | 5 | [[370, 628]] | 1.0 | 5lmb | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 4YJOA | P43405 | 363 | 632 | 635.0 | 4DF:701 | Type1 | Active | DFGin | 7.151 | 15.404 | BLAminus | -136.57, 178.57 | 59.58, 80.7 | -95.16, 22.65 | 286.36, 75.19 | -55.96, -31.16 | in-in | in | 8.32 | Saltbr-in | 3.044 | HRD-in | -80.48, -52.4 | 72.29, 6.84 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.957 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -56.5, 127.44 | APE9-dihe-in | -144.08, 83.31 | APE8-dihe-in | -75.74, 70.97 | APE8-rot-na | 33.07 | APE67-dihe-in | -63.43, -16.56 | -52.99, -37.5 | APE12-dist-na | 999.0 | APE11-dist-na | 10.63 | APE10-dist-na | 7.9 | APE9-dist-in | 7.507 | None | None | None | XRAY | 1.6 | 0.186 | 0.23 | A | 281 | 267 | 3 | 0 | 0 | 3 | [[370, 628]] | 1.0 | 4yjo | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.8e-90 | 307.3 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 5TT7A | P43405 | 358 | 635 | 635.0 | 7KF:60901 | Type1 | Active | DFGin | 6.311 | 14.341 | BLAminus | -130.62, -177.29 | 62.11, 72.82 | -94.96, 21.67 | 289.95, 80.8 | -60.6, -26.94 | in-in | in | 7.709 | Saltbr-in | 2.84 | HRD-in | -77.7, -52.28 | 69.96, 13.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.878 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.65, 88.09 | APE9-dihe-in | -107.14, 140.48 | APE8-dihe-in | -78.3, 78.38 | APE8-rot-na | 32.04 | APE67-dihe-in | -64.56, -15.37 | -56.64, -35.35 | APE12-dist-na | 13.888 | APE11-dist-na | 10.557 | APE10-dist-na | 10.342 | APE9-dist-in | 6.849 | None | None | None | XRAY | 1.77 | 0.208 | 0.234 | A | 289 | 270 | 8 | 0 | 0 | 0 | [[370, 628]] | 1.0 | 5tt7 | Homo sapiens | TYR_SYK_HUMAN | TYR | 5.4e-90 | 307.1 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 4FYOA | P43405 | 363 | 635 | 635.0 | 0VF:60701 | Type1 | None | DFGin | 6.527 | 14.676 | BLAminus | -132.65, -177.95 | 62.23, 72.42 | -93.99, 21.12 | 289.45, 90.18 | -61.07, -25.58 | in-in | in | 7.75 | Saltbr-in | 2.757 | HRD-in | -74.26, -50.97 | 72.76, 4.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.952 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 140.05 | APE9-dihe-in | -108.11, 144.2 | APE8-dihe-in | -76.07, 73.27 | APE8-rot-na | 27.85 | APE67-dihe-in | -65.29, -14.44 | -52.41, -38.79 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.947 | APE9-dist-in | 7.308 | None | None | None | XRAY | 1.4 | 0.22 | 0.24 | A | 291 | 263 | 10 | 0 | 0 | 4 | [[370, 628]] | 1.0 | 4fyo | Homo sapiens | TYR_SYK_HUMAN | TYR | 5.5e-90 | 307.1 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 4GFGA | P43405 | 363 | 635 | 635.0 | 0XF:60701 | Type1 | Active | DFGin | 6.382 | 14.706 | BLAminus | -133.41, -165.6 | 61.44, 68.78 | -94.44, 29.51 | 290.84, 74.86 | -64.09, -30.1 | in-in | in | 8.551 | Saltbr-in | 3.497 | HRD-in | -86.12, -47.8 | 68.36, 5.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.866 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -53.12, 138.6 | APE9-dihe-in | -110.15, 137.21 | APE8-dihe-in | -65.63, 68.92 | APE8-rot-na | 25.72 | APE67-dihe-in | -68.08, -17.47 | -52.98, -35.53 | APE12-dist-na | 9.582 | APE11-dist-na | 10.629 | APE10-dist-na | 11.706 | APE9-dist-in | 7.231 | None | None | None | XRAY | 2.35 | 0.221 | 0.246 | A | 291 | 273 | 0 | 0 | 0 | 0 | [[370, 628]] | 1.0 | 4gfg | Homo sapiens | TYR_SYK_HUMAN | TYR | 5.5e-90 | 307.1 | 5 | 260 | 256 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| CMGC | MAPK14 | MK14_MOUSE | 5R9OA | P47811 | 5 | 352 | 360.0 | 54F:401 | Allosteric | Inactive | DFGin | 7.673 | 17.211 | BLBminus | -136.39, -176.43 | 54.27, 60.09 | -56.75, 144.98 | 283.51, 68.16 | -67.8, 120.41 | in-in | in | 9.802 | Saltbr-in | 2.875 | HRD-in | -68.65, -55.19 | 86.09, -8.85 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.312 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_oooo | APE10-dihe-na | -136.85, 133.85 | APE9-dihe-na | -63.65, -21.53 | APE8-dihe-out | -61.93, -15.63 | APE8-rot-out | 53.56 | APE67-dihe-in | -63.52, -19.95 | -117.35, -20.3 | APE12-dist-out | 21.981 | APE11-dist-out | 24.156 | APE10-dist-out | 18.374 | APE9-dist-out | 11.868 | None | None | None | XRAY | 1.6 | 0.18 | 0.196 | A | 360 | 348 | 0 | 0 | 0 | 0 | [[24, 308]] | 1.0 | 5r9o | Mus musculus | CMGC_MAPK14_MOUSE | CMGC | 1.9e-85 | 292.7 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| TKL | RIPK3 | RIPK3_MOUSE | 9LVHA | Q9QZL0 | 13 | 312 | 486.0 | MYF:401 | Type1 | None | DFGin | 6.25 | 14.259 | BLAminus | -136.98, 168.96 | 62.75, 89.32 | -105.42, 15.63 | 293.79, 91.31 | -62.49, -27.0 | in-in | in | 8.376 | Saltbr-in | 2.879 | HRD-in | -72.81, -50.94 | 74.54, 2.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.778 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -60.25, -26.93 | 999.0, -1.12 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.38 | 0.251 | 0.271 | A | 325 | 263 | 37 | 0 | 0 | 19 | [[20, 290]] | 1.0 | 9lvh | Mus musculus | TKL_RIPK3_MOUSE | TKL | 5e-60 | 209.3 | 3 | 265 | 263 | 160 | 161 | 162 | 164 | 166 | 51 | 61 | 65 | 140 | 142 | 141 | 143 | 208 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 96 | Receptor-interacting serine/threonine-protein kinase 3 |
| TKL | RIPK3 | RIPK3_MOUSE | 9LVHB | Q9QZL0 | 13 | 312 | 486.0 | MYF:401 | Type1 | None | DFGin | 6.144 | 14.058 | BLAminus | -139.36, 174.01 | 57.76, 83.37 | -93.9, 23.89 | 297.93, 87.69 | -58.87, -31.82 | in-in | in | 8.581 | Saltbr-in | 2.817 | HRD-in | -67.48, -56.31 | 78.93, 2.25 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.713 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 138.93 | APE8-rot-in | 302.42 | APE67-dihe-in | -61.51, -26.08 | -64.96, -15.97 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.38 | 0.251 | 0.271 | B | 325 | 266 | 34 | 0 | 0 | 18 | [[20, 290]] | 1.0 | 9lvh | Mus musculus | TKL_RIPK3_MOUSE | TKL | 5e-60 | 209.3 | 3 | 265 | 263 | 160 | 161 | 162 | 164 | 166 | 51 | 61 | 65 | 140 | 142 | 141 | 143 | 208 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 96 | Receptor-interacting serine/threonine-protein kinase 3 |
| OTHER | CDC7 | CDC7_YEAST | 7PT78 | P06243 | 10 | 475 | 507.0 | ADP:1001,BEF:1003 | ATPlike,Allosteric | Inactive | DFGin | 7.05 | 14.828 | ABAminus | -125.48, -62.19 | -62.72, 136.55 | -132.76, 24.05 | 270.26, 81.1 | -56.4, -43.64 | in-out | in | 8.956 | Saltbr-out | 6.838 | HRD-out | -95.15, 91.19 | -59.72, -45.2 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.418 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -63.65, 141.8 | APE9-dihe-na | 169.57, -141.23 | APE8-dihe-in | -138.07, 164.32 | APE8-rot-in | 301.9 | APE67-dihe-out | 82.72, -175.36 | -64.25, 106.81 | APE12-dist-in | 8.854 | APE11-dist-in | 11.015 | APE10-dist-in | 5.043 | APE9-dist-in | 4.626 | None | None | None | EM | 3.8 | 999.0 | 999.0 | 8 | 507 | 402 | 64 | 0 | 0 | 46 | [[33, 469]] | 1.0 | 7pt7 | Saccharomyces cerevisiae | OTHER_CDC7_YEAST | CMGC | 4e-17 | 121.0 | 1 | 158 | 260 | 181 | 182 | 183 | 185 | 187 | 76 | 90 | 94 | 160 | 162 | 161 | 163 | 301 | 288 | 283 | 282 | 281 | 280 | 279 | 278 | 277 | 121 | Cell division control protein 7 |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HVXA | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60401 | Type1 | Inactive | DFGin | 6.812 | 13.739 | BLAminus | -151.79, -170.99 | 58.28, 71.83 | -90.67, 23.31 | 282.96, 81.43 | -68.24, -23.58 | in-in | in | 7.973 | Saltbr-in | 2.67 | HRD-in | -79.27, -44.62 | 69.75, 6.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.916 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.04, -39.68 | APE9-dihe-na | -85.38, 168.26 | APE8-dihe-in | -65.75, 139.05 | APE8-rot-out | 179.82 | APE67-dihe-in | -62.31, -27.06 | -57.82, -44.69 | APE12-dist-in | 13.505 | APE11-dist-in | 11.868 | APE10-dist-in | 7.371 | APE9-dist-in | 3.499 | None | PTR211 | PTR211 | XRAY | 2.1 | 0.203 | 0.25 | A | 350 | 323 | 16 | 0 | 0 | 0 | [[47, 344]] | 1.0 | 9hvx | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 6.4e-71 | 244.9 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6A | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60401 | Type1 | Inactive | DFGin | 6.554 | 13.514 | BLAminus | -159.29, -172.81 | 63.26, 75.9 | -98.23, 18.12 | 289.64, 83.03 | -60.9, -17.5 | in-in | in | 8.248 | Saltbr-in | 2.913 | HRD-in | -74.22, -42.3 | 70.91, -2.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.779 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_niio | APE10-dihe-na | -107.29, 145.01 | APE9-dihe-na | -102.07, 19.34 | APE8-dihe-in | -80.82, 138.15 | APE8-rot-out | 53.99 | APE67-dihe-in | -80.29, -18.75 | -104.8, -54.34 | APE12-dist-none | 999.0 | APE11-dist-in | 10.111 | APE10-dist-in | 7.183 | APE9-dist-out | 8.805 | None | PTR211,SEP257 | PTR211,SEP257 | XRAY | 2.9 | 0.207 | 0.26 | A | 373 | 332 | 7 | 0 | 0 | 3 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6B | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60402 | Type1 | Inactive | DFGin | 6.969 | 13.759 | BLAminus | -158.71, -175.52 | 61.04, 75.48 | -97.8, 20.68 | 289.3, 83.48 | -61.51, -18.44 | in-in | in | 8.34 | Saltbr-in | 2.533 | HRD-in | -73.25, -38.58 | 70.21, -4.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.957 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnio | APE10-dihe-na | 999.0, 137.93 | APE9-dihe-na | -128.88, -94.97 | APE8-dihe-out | 8.76, 102.73 | APE8-rot-out | 52.93 | APE67-dihe-in | -72.89, -15.66 | -99.47, -15.26 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 6.673 | APE9-dist-out | 7.874 | None | PTR211 | PTR211 | XRAY | 2.9 | 0.207 | 0.26 | B | 373 | 332 | 7 | 0 | 0 | 6 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6D | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60402 | Type1 | Inactive | DFGin | 6.752 | 13.545 | BLAminus | -157.98, -176.25 | 63.15, 72.4 | -94.88, 18.71 | 288.21, 86.06 | -60.77, -17.66 | in-in | in | 8.448 | Saltbr-in | 3.001 | HRD-in | -74.85, -41.94 | 71.3, -1.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.853 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_nnio | APE10-dihe-na | 999.0, -28.71 | APE9-dihe-na | 70.23, 60.42 | APE8-dihe-out | -136.17, -56.82 | APE8-rot-out | 132.32 | APE67-dihe-out | -77.45, -28.23 | 69.46, -39.41 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 7.077 | APE9-dist-out | 8.582 | None | PTR211,SEP257 | PTR211,SEP257 | XRAY | 2.9 | 0.207 | 0.26 | D | 373 | 327 | 12 | 0 | 0 | 9 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6F | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60401 | Type1 | Inactive | DFGin | 6.98 | 13.82 | BLAminus | -156.62, -174.56 | 59.51, 71.39 | -97.24, 16.48 | 288.27, 84.06 | -60.16, -18.79 | in-in | in | 8.206 | Saltbr-in | 2.735 | HRD-in | -76.38, -41.74 | 71.66, -4.7 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.744 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_niio | APE10-dihe-na | -146.52, 154.45 | APE9-dihe-na | -92.11, 49.24 | APE8-dihe-in | -83.14, 134.37 | APE8-rot-out | 54.49 | APE67-dihe-in | -77.45, -15.85 | -109.34, -69.31 | APE12-dist-none | 999.0 | APE11-dist-in | 9.936 | APE10-dist-in | 6.674 | APE9-dist-out | 9.042 | None | PTR211 | PTR211 | XRAY | 2.9 | 0.207 | 0.26 | F | 373 | 325 | 14 | 0 | 0 | 6 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_CRIGR | 7PIEA | P25321 | 1 | 351 | 351.0 | 7QF:60401 | Type1 | Inactive | DFGin | 6.437 | 14.708 | ABAminus | -120.2, -32.0 | -97.5, 116.46 | -117.79, 21.67 | 284.38, 87.37 | -67.96, -24.99 | in-in | in | 9.018 | Saltbr-in | 2.947 | HRD-in | -90.08, -55.75 | 70.92, 8.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.9, 155.75 | APE9-dihe-na | 129.48, -166.45 | APE8-dihe-in | -116.19, 135.64 | APE8-rot-in | 298.32 | APE67-dihe-in | -59.08, -26.0 | -47.12, -51.73 | APE12-dist-in | 8.298 | APE11-dist-in | 11.483 | APE10-dist-in | 5.921 | APE9-dist-in | 3.894 | None | SEP11,SEP140,TPO198,SEP339 | SEP11,SEP140,TPO198,SEP339 | XRAY | 1.427 | 0.137 | 0.158 | A | 353 | 350 | 0 | 0 | 0 | 0 | [[44, 298]] | 1.0 | 7pie | Cricetulus griseus | AGC_PRKACA_CRIGR | AGC | 6.6e-95 | 323.2 | 1 | 260 | 260 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_CRIGR | 9RETA | P25321 | 13 | 351 | 351.0 | A1JEF:60404 | Allosteric | Active | DFGin | 6.503 | 14.919 | BLAminus | -121.64, 161.02 | 79.66, 89.44 | -97.28, 25.84 | 271.42, 57.67 | -59.32, -29.98 | in-in | in | 9.058 | Saltbr-in | 2.688 | HRD-in | -91.57, -50.28 | 65.7, 14.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.961 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.82, 155.57 | APE9-dihe-na | 119.38, 155.92 | APE8-dihe-in | -73.83, 138.5 | APE8-rot-in | 315.72 | APE67-dihe-in | -57.32, -25.4 | -54.39, -42.36 | APE12-dist-in | 8.186 | APE11-dist-in | 11.402 | APE10-dist-in | 5.952 | APE9-dist-in | 4.241 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 1.75 | 0.193 | 0.227 | A | 353 | 339 | 0 | 0 | 0 | 0 | [[44, 298]] | 1.0 | 9ret | Cricetulus griseus | AGC_PRKACA_CRIGR | AGC | 6.6e-95 | 323.2 | 1 | 260 | 260 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| TYR | SRC | SRC_CHICK | 5SYSA | P00523 | 258 | 533 | 533.0 | 72F:600 | Type2 | Inactive | DFGout | 13.354 | 9.801 | BBAminus | -126.48, -173.83 | -168.38, 115.62 | -104.78, -47.96 | 311.28, 146.33 | 163.56, 999.0 | in-in | in | 8.579 | Saltbr-in | 3.03 | HRD-in | -86.37, -44.08 | 72.1, 11.73 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -16.31 | APE8-rot-na | 5.39 | APE67-dihe-in | -61.6, -39.03 | -88.61, -20.33 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | V281C | None | None | XRAY | 2.8 | 0.288 | 0.334 | A | 286 | 258 | 18 | 0 | 0 | 18 | [[267, 518]] | 1.0 | 5sys | Gallus gallus | TYR_SRC_CHICK | TYR | 4.2e-93 | 317.3 | 1 | 260 | 260 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 5SYSB | P00523 | 258 | 533 | 533.0 | 72F:600 | Type2 | Inactive | DFGout | 13.413 | 10.163 | BBAminus | -126.31, -175.1 | -166.31, 115.77 | -103.34, -47.57 | 306.63, 130.98 | 67.96, 999.0 | in-in | in | 8.321 | Saltbr-in | 3.044 | HRD-in | -86.54, -44.23 | 72.2, 11.45 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -18.84 | APE8-rot-na | 6.43 | APE67-dihe-in | -61.0, -39.73 | -89.58, -19.88 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | V281C | None | None | XRAY | 2.8 | 0.288 | 0.334 | B | 286 | 258 | 18 | 0 | 0 | 18 | [[267, 518]] | 1.0 | 5sys | Gallus gallus | TYR_SRC_CHICK | TYR | 4.2e-93 | 317.3 | 1 | 260 | 260 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| CMGC | MAPK14 | MK14_MOUSE | 5R9OA | P47811 | 5 | 352 | 360.0 | 54F:401 | Allosteric | Inactive | DFGin | 7.673 | 17.211 | BLBminus | -136.39, -176.43 | 54.27, 60.09 | -56.75, 144.98 | 283.51, 68.16 | -67.8, 120.41 | in-in | in | 9.802 | Saltbr-in | 2.875 | HRD-in | -68.65, -55.19 | 86.09, -8.85 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.312 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_oooo | APE10-dihe-na | -136.85, 133.85 | APE9-dihe-na | -63.65, -21.53 | APE8-dihe-out | -61.93, -15.63 | APE8-rot-out | 53.56 | APE67-dihe-in | -63.52, -19.95 | -117.35, -20.3 | APE12-dist-out | 21.981 | APE11-dist-out | 24.156 | APE10-dist-out | 18.374 | APE9-dist-out | 11.868 | None | None | None | XRAY | 1.6 | 0.18 | 0.196 | A | 360 | 348 | 0 | 0 | 0 | 0 | [[24, 308]] | 1.0 | 5r9o | Mus musculus | CMGC_MAPK14_MOUSE | CMGC | 1.9e-85 | 292.7 | 1 | 301 | 301 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| TKL | RIPK3 | RIPK3_MOUSE | 9LVHA | Q9QZL0 | 13 | 312 | 486.0 | MYF:401 | Type1 | None | DFGin | 6.25 | 14.259 | BLAminus | -136.98, 168.96 | 62.75, 89.32 | -105.42, 15.63 | 293.79, 91.31 | -62.49, -27.0 | in-in | in | 8.376 | Saltbr-in | 2.879 | HRD-in | -72.81, -50.94 | 74.54, 2.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.778 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -60.25, -26.93 | 999.0, -1.12 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.38 | 0.251 | 0.271 | A | 325 | 263 | 37 | 0 | 0 | 19 | [[20, 290]] | 1.0 | 9lvh | Mus musculus | TKL_RIPK3_MOUSE | TKL | 5e-60 | 209.3 | 3 | 265 | 263 | 160 | 161 | 162 | 164 | 166 | 51 | 61 | 65 | 140 | 142 | 141 | 143 | 208 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 96 | Receptor-interacting serine/threonine-protein kinase 3 |
| TKL | RIPK3 | RIPK3_MOUSE | 9LVHB | Q9QZL0 | 13 | 312 | 486.0 | MYF:401 | Type1 | None | DFGin | 6.144 | 14.058 | BLAminus | -139.36, 174.01 | 57.76, 83.37 | -93.9, 23.89 | 297.93, 87.69 | -58.87, -31.82 | in-in | in | 8.581 | Saltbr-in | 2.817 | HRD-in | -67.48, -56.31 | 78.93, 2.25 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.713 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 138.93 | APE8-rot-in | 302.42 | APE67-dihe-in | -61.51, -26.08 | -64.96, -15.97 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.38 | 0.251 | 0.271 | B | 325 | 266 | 34 | 0 | 0 | 18 | [[20, 290]] | 1.0 | 9lvh | Mus musculus | TKL_RIPK3_MOUSE | TKL | 5e-60 | 209.3 | 3 | 265 | 263 | 160 | 161 | 162 | 164 | 166 | 51 | 61 | 65 | 140 | 142 | 141 | 143 | 208 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 96 | Receptor-interacting serine/threonine-protein kinase 3 |
| OTHER | CDC7 | CDC7_YEAST | 7PT78 | P06243 | 10 | 475 | 507.0 | ADP:1001,BEF:1003 | ATPlike,Allosteric | Inactive | DFGin | 7.05 | 14.828 | ABAminus | -125.48, -62.19 | -62.72, 136.55 | -132.76, 24.05 | 270.26, 81.1 | -56.4, -43.64 | in-out | in | 8.956 | Saltbr-out | 6.838 | HRD-out | -95.15, 91.19 | -59.72, -45.2 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.418 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -63.65, 141.8 | APE9-dihe-na | 169.57, -141.23 | APE8-dihe-in | -138.07, 164.32 | APE8-rot-in | 301.9 | APE67-dihe-out | 82.72, -175.36 | -64.25, 106.81 | APE12-dist-in | 8.854 | APE11-dist-in | 11.015 | APE10-dist-in | 5.043 | APE9-dist-in | 4.626 | None | None | None | EM | 3.8 | 999.0 | 999.0 | 8 | 507 | 402 | 64 | 0 | 0 | 46 | [[33, 469]] | 1.0 | 7pt7 | Saccharomyces cerevisiae | OTHER_CDC7_YEAST | CMGC | 4e-17 | 121.0 | 1 | 158 | 260 | 181 | 182 | 183 | 185 | 187 | 76 | 90 | 94 | 160 | 162 | 161 | 163 | 301 | 288 | 283 | 282 | 281 | 280 | 279 | 278 | 277 | 121 | Cell division control protein 7 |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HVXA | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60401 | Type1 | Inactive | DFGin | 6.812 | 13.739 | BLAminus | -151.79, -170.99 | 58.28, 71.83 | -90.67, 23.31 | 282.96, 81.43 | -68.24, -23.58 | in-in | in | 7.973 | Saltbr-in | 2.67 | HRD-in | -79.27, -44.62 | 69.75, 6.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.916 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.04, -39.68 | APE9-dihe-na | -85.38, 168.26 | APE8-dihe-in | -65.75, 139.05 | APE8-rot-out | 179.82 | APE67-dihe-in | -62.31, -27.06 | -57.82, -44.69 | APE12-dist-in | 13.505 | APE11-dist-in | 11.868 | APE10-dist-in | 7.371 | APE9-dist-in | 3.499 | None | PTR211 | PTR211 | XRAY | 2.1 | 0.203 | 0.25 | A | 350 | 323 | 16 | 0 | 0 | 0 | [[47, 344]] | 1.0 | 9hvx | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 6.4e-71 | 244.9 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6A | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60401 | Type1 | Inactive | DFGin | 6.554 | 13.514 | BLAminus | -159.29, -172.81 | 63.26, 75.9 | -98.23, 18.12 | 289.64, 83.03 | -60.9, -17.5 | in-in | in | 8.248 | Saltbr-in | 2.913 | HRD-in | -74.22, -42.3 | 70.91, -2.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.779 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_niio | APE10-dihe-na | -107.29, 145.01 | APE9-dihe-na | -102.07, 19.34 | APE8-dihe-in | -80.82, 138.15 | APE8-rot-out | 53.99 | APE67-dihe-in | -80.29, -18.75 | -104.8, -54.34 | APE12-dist-none | 999.0 | APE11-dist-in | 10.111 | APE10-dist-in | 7.183 | APE9-dist-out | 8.805 | None | PTR211,SEP257 | PTR211,SEP257 | XRAY | 2.9 | 0.207 | 0.26 | A | 373 | 332 | 7 | 0 | 0 | 3 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6B | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60402 | Type1 | Inactive | DFGin | 6.969 | 13.759 | BLAminus | -158.71, -175.52 | 61.04, 75.48 | -97.8, 20.68 | 289.3, 83.48 | -61.51, -18.44 | in-in | in | 8.34 | Saltbr-in | 2.533 | HRD-in | -73.25, -38.58 | 70.21, -4.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.957 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnio | APE10-dihe-na | 999.0, 137.93 | APE9-dihe-na | -128.88, -94.97 | APE8-dihe-out | 8.76, 102.73 | APE8-rot-out | 52.93 | APE67-dihe-in | -72.89, -15.66 | -99.47, -15.26 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 6.673 | APE9-dist-out | 7.874 | None | PTR211 | PTR211 | XRAY | 2.9 | 0.207 | 0.26 | B | 373 | 332 | 7 | 0 | 0 | 6 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6D | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60402 | Type1 | Inactive | DFGin | 6.752 | 13.545 | BLAminus | -157.98, -176.25 | 63.15, 72.4 | -94.88, 18.71 | 288.21, 86.06 | -60.77, -17.66 | in-in | in | 8.448 | Saltbr-in | 3.001 | HRD-in | -74.85, -41.94 | 71.3, -1.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.853 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_nnio | APE10-dihe-na | 999.0, -28.71 | APE9-dihe-na | 70.23, 60.42 | APE8-dihe-out | -136.17, -56.82 | APE8-rot-out | 132.32 | APE67-dihe-out | -77.45, -28.23 | 69.46, -39.41 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 7.077 | APE9-dist-out | 8.582 | None | PTR211,SEP257 | PTR211,SEP257 | XRAY | 2.9 | 0.207 | 0.26 | D | 373 | 327 | 12 | 0 | 0 | 9 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |
| CMGC | GSK3B | A0A125YY75_TOXGG | 9HW6F | A0A125YY75 | 46 | 384 | 394.0 | A1IYF:60401 | Type1 | Inactive | DFGin | 6.98 | 13.82 | BLAminus | -156.62, -174.56 | 59.51, 71.39 | -97.24, 16.48 | 288.27, 84.06 | -60.16, -18.79 | in-in | in | 8.206 | Saltbr-in | 2.735 | HRD-in | -76.38, -41.74 | 71.66, -4.7 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.744 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_niio | APE10-dihe-na | -146.52, 154.45 | APE9-dihe-na | -92.11, 49.24 | APE8-dihe-in | -83.14, 134.37 | APE8-rot-out | 54.49 | APE67-dihe-in | -77.45, -15.85 | -109.34, -69.31 | APE12-dist-none | 999.0 | APE11-dist-in | 9.936 | APE10-dist-in | 6.674 | APE9-dist-out | 9.042 | None | PTR211 | PTR211 | XRAY | 2.9 | 0.207 | 0.26 | F | 373 | 325 | 14 | 0 | 0 | 6 | [[47, 344]] | 1.0 | 9hw6 | Toxoplasma gondii | CMGC_GSK3B_TOXGG | CMGC | 8e-71 | 244.6 | 1 | 301 | 301 | 194 | 195 | 196 | 198 | 200 | 76 | 88 | 92 | 173 | 175 | 174 | 176 | 234 | 221 | 216 | 215 | 214 | 213 | 212 | 211 | 210 | 128 | Putative cell-cycle-associated protein kinase GSK |