TYR_KDR (Vascular endothelial growth factor receptor 2)

Total number of chains: 54
Active chains: 2
Uniprot: VGFR2_HUMAN
Kinase Domain Residues: 834 - 1162
Spatial label Dihedral label Number of Chains Percent Representative
DFGout BBAminus 32 59.3% 6GQQA
DFGout None 9 16.7% 3VO3A
DFGin BLAminus 3 5.6% AF-P35968-K1A
DFGin BLBplus 3 5.6% 3WZDA
None None 3 5.6% 3CJFA
DFGinter None 2 3.7% 1Y6BA
DFGin BLAplus 1 1.9% 2P2HA
DFGin None 1 1.9% 1VR2A

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PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
AF-P35968-K1A -1.0 Active DFGin‑BLAminus in-in in-in TYR APEdihe_iiiai APEdist_aaai No_ligand No_ligand 826 - 1170 0 None None Vascular endothelial growth factor receptor 2
AF-P35968-K3A -1.0 Active DFGin‑BLAminus in-in in-in TYR APEdihe_iiiai APEdist_aaai No_ligand No_ligand 826 - 1170 0 None None Vascular endothelial growth factor receptor 2
3CJGA 2.25 Inactive DFGin‑BLAminus in-in in-out TYR APEdihe_nnnao APEdist_aaan KIM Type1 816 - 1168 0 None None Vascular endothelial growth factor receptor 2
2P2HA 1.95 Inactive DFGin‑BLAplus in-in none-out TYR APEdihe_nooai APEdist_aaao 994 Type1 815 - 1172 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3WZDA 1.57 Inactive DFGin‑BLBplus in-in none-out TYR APEdihe_nnoai APEdist_aaao LEV Type1 820 - 1167 0 None T940V Vascular endothelial growth factor receptor 2
3B8RA 2.7 Inactive DFGin‑BLBplus in-in none-out TYR APEdihe_nnoai APEdist_aaao 887 Type1 818 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3B8RB 2.7 Inactive DFGin‑BLBplus in-in none-out TYR APEdihe_nnoai APEdist_aaao 887 Type1 821 - 1166 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
1VR2A 2.4 Inactive DFGin‑None in-in none-out TYR APEdihe_iioai APEdist_aaao No_ligand No_ligand 820 - 1168 0 PTR1059 E990V Vascular endothelial growth factor receptor 2
1Y6AA 2.1 Inactive DFGinter‑None in-in none-none TYR APEdihe_nnnai APEdist_aaan AAZ Type1 820 - 1167 0 None None Vascular endothelial growth factor receptor 2
1Y6BA 2.1 Inactive DFGinter‑None in-in none-none TYR APEdihe_nnnai APEdist_aaan AAX Type1 819 - 1168 0 None None Vascular endothelial growth factor receptor 2
4AG8A 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai AXI Type1 816 - 1168 0 None E990V Vascular endothelial growth factor receptor 2
4AGDA 2.81 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai B49 Type1 802 - 1169 0 None E990V Vascular endothelial growth factor receptor 2
3CPBB 2.7 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C92 Type1 820 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
2XIRA 1.5 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai 00J Type1.5_Back 816 - 1168 0 None E990V Vascular endothelial growth factor receptor 2
4AGCA 2.0 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai AXI Type1.5_Back 801 - 1169 0 None E990V Vascular endothelial growth factor receptor 2
3WZEA 1.9 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao BAX Type2 815 - 1167 0 None T940V Vascular endothelial growth factor receptor 2
2OH4A 2.05 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iioai APEdist_aaao GIG Type2 816 - 1171 0 PTR1054,PTR1059 None Vascular endothelial growth factor receptor 2
2P2IA 2.4 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao 608 Type2 817 - 1172 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2
3EFLA 2.2 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nnnai APEdist_aaan 706 Type2 817 - 1171 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2
3EFLB 2.2 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao 706 Type2 821 - 1165 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2
5EW3A 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao 5T2 Type2 821 - 1168 0 None None Vascular endothelial growth factor receptor 2
5EW3B 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao 5T2 Type2 820 - 1165 0 None None Vascular endothelial growth factor receptor 2
6GQOA 1.87 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai F82 Type2 811 - 1168 0 None None Vascular endothelial growth factor receptor 2
6GQPA 2.09 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao F88 Type2 821 - 1168 0 None None Vascular endothelial growth factor receptor 2
6GQQA 1.52 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao F8B Type2 813 - 1167 0 None None Vascular endothelial growth factor receptor 2
6XVJA 1.78 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai O35 Type2 813 - 1167 0 None E990V Vascular endothelial growth factor receptor 2
6XVKA 1.99 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai O3E Type2 821 - 1168 0 None E990V Vascular endothelial growth factor receptor 2
4ASDA 2.03 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai BAX Type2 807 - 1168 0 None E990V Vascular endothelial growth factor receptor 2
4ASEA 1.83 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai AV9 Type2 807 - 1169 0 None E990V Vascular endothelial growth factor receptor 2
3VHEA 1.55 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao 42Q Type2 811 - 1169 0 None None Vascular endothelial growth factor receptor 2
3VHKA 2.49 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao BPK Type2 814 - 1168 0 None None Vascular endothelial growth factor receptor 2
2QU5A 2.95 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_oooai APEdist_aaao 276 Type2 816 - 1170 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
2QU6A 2.1 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nnnai APEdist_aaan 857 Type2 817 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
2RL5A 2.65 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_oooai APEdist_aaao 2RL Type2 815 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3B8QB 2.75 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao 900 Type2 820 - 1166 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3BE2A 1.75 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nnnai APEdist_aaan RAJ Type2 815 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3CP9A 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C19 Type2 817 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3CP9B 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C19 Type2 819 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3CPCB 2.4 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C52 Type2 820 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3DTWB 2.9 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nooai APEdist_aaao A96 Type2 820 - 1166 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3EWHA 1.6 Inactive DFGout‑BBAminus in-in out-none TYR APEdihe_nniai APEdist_aaai K11 Type2 815 - 1171 0 None C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3U6JA 2.15 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai 03X Type2 815 - 1171 0 None V916T,E990V Vascular endothelial growth factor receptor 2
3C7QA 2.1 Inactive DFGout‑None in-in none-out TYR APEdihe_iioai APEdist_aaao XIN Type1 819 - 1171 0 PTR1054,PTR1059 None Vascular endothelial growth factor receptor 2
2P2IB 2.4 Inactive DFGout‑None in-in none-none TYR APEdihe_nnnai APEdist_aaan 608 Type1 820 - 1168 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2
3VNTA 1.64 Inactive DFGout‑None in-in out-in TYR APEdihe_iiiai APEdist_aaai 0JA Type2 812 - 1168 0 None None Vascular endothelial growth factor receptor 2
3VO3A 1.52 Inactive DFGout‑None in-in out-in TYR APEdihe_iiiai APEdist_aaai 0KF Type2 812 - 1168 0 None None Vascular endothelial growth factor receptor 2
2QU6B 2.1 Inactive DFGout‑None in-in none-out TYR APEdihe_nniai APEdist_aaao 857 Type2 822 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3B8QA 2.75 Inactive DFGout‑None in-in none-out TYR APEdihe_nnoai APEdist_aaao 900 Type2 818 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3CPBA 2.7 Inactive DFGout‑None in-in none-out TYR APEdihe_nnoai APEdist_aaao C92 Type2 819 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3CPCA 2.4 Inactive DFGout‑None in-out none-out TYR APEdihe_nnoai APEdist_aaao C52 Type2 820 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3DTWA 2.9 Inactive DFGout‑None in-in none-out TYR APEdihe_nnoai APEdist_aaao A96 Type2 818 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2
3CJFA 2.15 Inactive None‑None in-out in-none TYR APEdihe_nnnai APEdist_aaan SAV Type1 817 - 1168 0 None None Vascular endothelial growth factor receptor 2
1YWNA 1.71 Inactive None‑None in-in none-out TYR APEdihe_iioai APEdist_aaao LIF Type1 820 - 1171 0 PTR1054,PTR1059 E990V Vascular endothelial growth factor receptor 2
3VIDA 2.3 Inactive None‑None in-in none-out TYR APEdihe_iioai APEdist_aaao 4TT Type1 813 - 1168 0 None None Vascular endothelial growth factor receptor 2

TYR_KDR (Vascular endothelial growth factor receptor 2)

Total number of chains: 54
Active chains: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGout BBAminus 32 59.3% 6GQQA
DFGout None 9 16.7% 3VO3A
DFGin BLAminus 3 5.6% AF-P35968-K1A
DFGin BLBplus 3 5.6% 3WZDA
None None 3 5.6% 3CJFA
DFGinter None 2 3.7% 1Y6BA
DFGin BLAplus 1 1.9% 2P2HA
DFGin None 1 1.9% 1VR2A

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
VGFR2_HUMAN AF-P35968-K1A -1.0 Active DFGin‑BLAminus in-in in-in TYR APEdihe_iiiai APEdist_aaai No_ligand No_ligand 826 - 1170 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN AF-P35968-K3A -1.0 Active DFGin‑BLAminus in-in in-in TYR APEdihe_iiiai APEdist_aaai No_ligand No_ligand 826 - 1170 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CJGA 2.25 Inactive DFGin‑BLAminus in-in in-out TYR APEdihe_nnnao APEdist_aaan KIM Type1 816 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2P2HA 1.95 Inactive DFGin‑BLAplus in-in none-out TYR APEdihe_nooai APEdist_aaao 994 Type1 815 - 1172 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3WZDA 1.57 Inactive DFGin‑BLBplus in-in none-out TYR APEdihe_nnoai APEdist_aaao LEV Type1 820 - 1167 0 None T940V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3B8RA 2.7 Inactive DFGin‑BLBplus in-in none-out TYR APEdihe_nnoai APEdist_aaao 887 Type1 818 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3B8RB 2.7 Inactive DFGin‑BLBplus in-in none-out TYR APEdihe_nnoai APEdist_aaao 887 Type1 821 - 1166 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 1VR2A 2.4 Inactive DFGin‑None in-in none-out TYR APEdihe_iioai APEdist_aaao No_ligand No_ligand 820 - 1168 0 PTR1059 E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 1Y6AA 2.1 Inactive DFGinter‑None in-in none-none TYR APEdihe_nnnai APEdist_aaan AAZ Type1 820 - 1167 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 1Y6BA 2.1 Inactive DFGinter‑None in-in none-none TYR APEdihe_nnnai APEdist_aaan AAX Type1 819 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 4AG8A 1.95 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai AXI Type1 816 - 1168 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 4AGDA 2.81 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai B49 Type1 802 - 1169 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CPBB 2.7 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C92 Type1 820 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2XIRA 1.5 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai 00J Type1.5_Back 816 - 1168 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 4AGCA 2.0 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai AXI Type1.5_Back 801 - 1169 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3WZEA 1.9 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao BAX Type2 815 - 1167 0 None T940V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2OH4A 2.05 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iioai APEdist_aaao GIG Type2 816 - 1171 0 PTR1054,PTR1059 None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2P2IA 2.4 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao 608 Type2 817 - 1172 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3EFLA 2.2 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nnnai APEdist_aaan 706 Type2 817 - 1171 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3EFLB 2.2 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao 706 Type2 821 - 1165 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 5EW3A 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao 5T2 Type2 821 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 5EW3B 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nniai APEdist_aaao 5T2 Type2 820 - 1165 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 6GQOA 1.87 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai F82 Type2 811 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 6GQPA 2.09 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao F88 Type2 821 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 6GQQA 1.52 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao F8B Type2 813 - 1167 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 6XVJA 1.78 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai O35 Type2 813 - 1167 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 6XVKA 1.99 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai O3E Type2 821 - 1168 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 4ASDA 2.03 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai BAX Type2 807 - 1168 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 4ASEA 1.83 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai AV9 Type2 807 - 1169 0 None E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3VHEA 1.55 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao 42Q Type2 811 - 1169 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3VHKA 2.49 Inactive DFGout‑BBAminus in-in out-out TYR APEdihe_iiiai APEdist_aaao BPK Type2 814 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2QU5A 2.95 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_oooai APEdist_aaao 276 Type2 816 - 1170 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2QU6A 2.1 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nnnai APEdist_aaan 857 Type2 817 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2RL5A 2.65 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_oooai APEdist_aaao 2RL Type2 815 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3B8QB 2.75 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao 900 Type2 820 - 1166 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3BE2A 1.75 Inactive DFGout‑BBAminus in-in none-none TYR APEdihe_nnnai APEdist_aaan RAJ Type2 815 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CP9A 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C19 Type2 817 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CP9B 2.5 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C19 Type2 819 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CPCB 2.4 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nnoai APEdist_aaao C52 Type2 820 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3DTWB 2.9 Inactive DFGout‑BBAminus in-in none-out TYR APEdihe_nooai APEdist_aaao A96 Type2 820 - 1166 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3EWHA 1.6 Inactive DFGout‑BBAminus in-in out-none TYR APEdihe_nniai APEdist_aaai K11 Type2 815 - 1171 0 None C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3U6JA 2.15 Inactive DFGout‑BBAminus in-in out-in TYR APEdihe_iiiai APEdist_aaai 03X Type2 815 - 1171 0 None V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3C7QA 2.1 Inactive DFGout‑None in-in none-out TYR APEdihe_iioai APEdist_aaao XIN Type1 819 - 1171 0 PTR1054,PTR1059 None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2P2IB 2.4 Inactive DFGout‑None in-in none-none TYR APEdihe_nnnai APEdist_aaan 608 Type1 820 - 1168 0 PTR1054,PTR1059 C817A,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3VNTA 1.64 Inactive DFGout‑None in-in out-in TYR APEdihe_iiiai APEdist_aaai 0JA Type2 812 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3VO3A 1.52 Inactive DFGout‑None in-in out-in TYR APEdihe_iiiai APEdist_aaai 0KF Type2 812 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 2QU6B 2.1 Inactive DFGout‑None in-in none-out TYR APEdihe_nniai APEdist_aaao 857 Type2 822 - 1165 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3B8QA 2.75 Inactive DFGout‑None in-in none-out TYR APEdihe_nnoai APEdist_aaao 900 Type2 818 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CPBA 2.7 Inactive DFGout‑None in-in none-out TYR APEdihe_nnoai APEdist_aaao C92 Type2 819 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CPCA 2.4 Inactive DFGout‑None in-out none-out TYR APEdihe_nnoai APEdist_aaao C52 Type2 820 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3DTWA 2.9 Inactive DFGout‑None in-in none-out TYR APEdihe_nnoai APEdist_aaao A96 Type2 818 - 1171 0 PTR1054,PTR1059 C817A,V916T,E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3CJFA 2.15 Inactive None‑None in-out in-none TYR APEdihe_nnnai APEdist_aaan SAV Type1 817 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 1YWNA 1.71 Inactive None‑None in-in none-out TYR APEdihe_iioai APEdist_aaao LIF Type1 820 - 1171 0 PTR1054,PTR1059 E990V Vascular endothelial growth factor receptor 2 Homo sapiens
VGFR2_HUMAN 3VIDA 2.3 Inactive None‑None in-in none-out TYR APEdihe_iioai APEdist_aaao 4TT Type1 813 - 1168 0 None None Vascular endothelial growth factor receptor 2 Homo sapiens

TYR_KDR (Vascular endothelial growth factor receptor 2)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism