| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| KDR | AF-P35968-K1A | P35968 | 826 | 1170 | 1356.0 | No_ligand | No_ligand | Active | DFGin | 6.724 | 13.7539 | BLAminus | -135.49, -178.07 | 64.31, 58.61 | -79.84, 14.65 | 291.25, 84.84 | -59.67, -29.27 | in-in | in | 7.2738 | Saltbr-in | 2.6536 | HRD-in | -79.81, -44.23 | 66.36, -15.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9851 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.88, 109.91 | APE9-dihe-in | -121.83, 150.33 | APE8-dihe-in | -76.73, 95.83 | APE8-rot-na | 34.09 | APE67-dihe-in | -64.1, -25.24 | -52.96, -31.45 | APE12-dist-na | 14.1753 | APE11-dist-na | 7.9361 | APE10-dist-na | 10.7309 | APE9-dist-in | 6.1962 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 345.0 | 345.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | AF-P35968-K1 | TYR_KDR_HUMAN | TYR | 2.1e-99 | 338.0 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | AF-P35968-K3A | P35968 | 826 | 1170 | 1356.0 | No_ligand | No_ligand | Active | DFGin | 6.4666 | 13.4597 | BLAminus | -139.09, -177.77 | 61.66, 65.38 | -79.85, 17.72 | 289.99, 89.58 | -61.52, -31.06 | in-in | in | 7.8222 | Saltbr-in | 2.7291 | HRD-in | -81.16, -45.43 | 63.07, 4.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9147 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -52.76, 130.74 | APE9-dihe-in | -112.3, 130.74 | APE8-dihe-in | -82.3, 61.23 | APE8-rot-na | 36.08 | APE67-dihe-in | -68.73, -19.78 | -48.02, -36.64 | APE12-dist-na | 13.331 | APE11-dist-na | 7.163 | APE10-dist-na | 8.5381 | APE9-dist-in | 6.7571 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 345.0 | 345.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | AF-P35968-K3 | TYR_KDR_HUMAN | TYR | 2.1e-99 | 338.0 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CJGA | P35968 | 816 | 1168 | 1356.0 | KIM:61167 | Type1 | Inactive | DFGin | 7.412 | 14.1279 | BLAminus | -120.91, -162.35 | 48.63, 86.88 | -107.47, 22.59 | 302.68, 92.72 | -76.12, -15.36 | in-in | in | 7.1793 | Saltbr-in | 2.6808 | HRD-in | -77.13, -50.16 | 74.93, 1.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9769 | ActLoopCT-out | TYR | APEdihe_nnnao | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 19.76 | APE8-rot-na | 1.33 | APE67-dihe-out | -66.63, -12.94 | 74.8, -54.69 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | CSO862,CSO1024 | XRAY | 2.25 | 0.209 | 0.253 | A | 309.0 | 282.0 | 17 | 30 | 16 | 14 | [[834, 1162]] | 1.0 | 3cjg | TYR_KDR_HUMAN | TYR | 4.8e-100 | 340.1 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2P2HA | P35968 | 815 | 1172 | 1356.0 | 994:60501 | Type1 | Inactive | DFGin | 5.7777 | 13.4944 | BLAplus | -120.41, 168.7 | 57.61, 43.27 | -102.94, -14.81 | 60.29, 84.2 | -108.45, 28.25 | in-in | in | 7.3498 | Saltbr-in | 2.5269 | HRD-in | -63.68, -53.12 | 82.34, -19.49 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, 158.7 | APE9-dihe-out | 54.03, 51.67 | APE8-dihe-out | -62.29, -19.22 | APE8-rot-na | 32.86 | APE67-dihe-in | -68.4, -12.54 | -60.9, -27.46 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 19.0397 | APE9-dist-out | 11.1812 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.95 | 0.205 | 0.229 | A | 314.0 | 289.0 | 19 | 30 | 15 | 15 | [[834, 1162]] | 1.0 | 2p2h | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3WZDA | P35968 | 820 | 1167 | 1356.0 | LEV:1201 | Type1 | Inactive | DFGin | 5.4262 | 13.8027 | BLBplus | -131.31, 171.12 | 64.88, 24.46 | -69.96, 136.97 | 45.36, 91.24 | 79.76, 6.08 | in-in | in | 7.3091 | Saltbr-in | 2.9428 | HRD-in | -65.52, -53.13 | 82.13, -20.42 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -70.62 | APE8-dihe-out | -53.22, -31.36 | APE8-rot-na | 22.8 | APE67-dihe-in | -66.02, -15.12 | -58.21, -29.08 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2484 | T940V | None | None | XRAY | 1.57 | 0.184 | 0.212 | A | 309.0 | 278.0 | 20 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 3wzd | TYR_KDR_HUMAN | TYR | 3.7e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3B8RA | P35968 | 818 | 1171 | 1356.0 | 887:60201 | Type1 | Inactive | DFGin | 5.4242 | 13.8708 | BLBplus | -147.04, 169.16 | 57.66, 43.33 | -97.43, 156.79 | 47.05, 78.4 | 59.04, 37.41 | in-in | in | 7.2508 | Saltbr-in | 2.6796 | HRD-in | -59.31, -52.93 | 80.34, -8.78 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 162.25 | APE8-dihe-out | -73.03, -9.68 | APE8-rot-na | 326.59 | APE67-dihe-in | -61.58, -18.77 | -55.36, -31.25 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2594 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.204 | 0.259 | A | 314.0 | 282.0 | 22 | 30 | 13 | 17 | [[834, 1162]] | 1.0 | 3b8r | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3B8RB | P35968 | 821 | 1166 | 1356.0 | 887:60202 | Type1 | Inactive | DFGin | 5.4416 | 13.8855 | BLBplus | -153.23, 176.22 | 49.55, 49.42 | -108.14, 150.46 | 48.31, 72.77 | 69.58, 35.57 | in-in | in | 7.3928 | Saltbr-in | 2.7455 | HRD-in | -68.34, -51.75 | 79.37, -8.5 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.55 | APE8-dihe-out | -62.02, -11.57 | APE8-rot-na | 326.58 | APE67-dihe-in | -65.24, -19.42 | -57.92, -26.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2614 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.204 | 0.259 | B | 314.0 | 267.0 | 29 | 30 | 13 | 17 | [[834, 1162]] | 1.0 | 3b8r | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 1VR2A | P35968 | 820 | 1168 | 1356.0 | No_ligand | No_ligand | Inactive | DFGin | 6.1971 | 12.2007 | None | -132.36, 167.84 | 67.89, 27.54 | -86.08, 999.0 | 49.78, 130.84 | 999.0, 999.0 | in-in | in | 7.7298 | Saltbr-in | 2.9904 | HRD-in | -66.37, -43.4 | 76.06, -15.34 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -137.43, 155.04 | APE9-dihe-in | -108.73, 90.95 | APE8-dihe-out | -47.33, -14.52 | APE8-rot-na | 323.83 | APE67-dihe-in | -64.29, -7.8 | -69.97, -29.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.4665 | E990V | PTR1059 | PTR1059 | XRAY | 2.4 | 0.215 | 999.0 | A | 316.0 | 275.0 | 24 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 1vr2 | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 1Y6AA | P35968 | 820 | 1167 | 1356.0 | AAZ:60201 | Type1 | Inactive | DFGinter | 8.6659 | 8.8381 | None | -73.14, 116.72 | -103.71, 73.1 | -178.89, 999.0 | 25.84, 61.42 | 999.0, 999.0 | in-in | in | 7.4703 | Saltbr-in | 2.8011 | HRD-in | -83.04, -53.13 | 81.96, -16.64 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -20.95 | APE8-rot-na | 328.99 | APE67-dihe-in | -63.85, -16.51 | -63.27, -26.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.1 | 0.196 | 0.217 | A | 366.0 | 261.0 | 87 | 30 | 10 | 20 | [[834, 1162]] | 1.0 | 1y6a | TYR_KDR_HUMAN | TYR | 2.6e-99 | 337.7 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 1Y6BA | P35968 | 819 | 1168 | 1356.0 | AAX:60201 | Type1 | Inactive | DFGinter | 8.9591 | 8.6911 | None | -70.35, 112.74 | -90.68, -29.02 | -42.32, 999.0 | 351.89, 106.67 | 999.0, 999.0 | in-in | in | 7.4818 | Saltbr-in | 2.9568 | HRD-in | -82.96, -58.21 | 87.46, -12.31 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 69.65 | APE8-rot-na | 33.76 | APE67-dihe-in | -65.54, -15.03 | -63.36, -37.08 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.1 | 0.194 | 0.236 | A | 366.0 | 266.0 | 84 | 30 | 10 | 20 | [[834, 1162]] | 1.0 | 1y6b | TYR_KDR_HUMAN | TYR | 2.6e-99 | 337.7 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 4AG8A | P35968 | 816 | 1168 | 1356.0 | AXI:2000 | Type1 | Inactive | DFGout | 16.4966 | 10.362 | BBAminus | -143.7, -179.58 | -144.17, 113.57 | -60.35, -33.13 | 275.19, 77.68 | 54.27, -121.79 | in-in | in | 7.5186 | Saltbr-in | 2.748 | HRD-in | -80.25, -53.16 | 76.08, -12.6 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5659 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.55, 111.08 | APE9-dihe-in | -116.46, 147.01 | APE8-dihe-in | -77.77, 66.25 | APE8-rot-na | 30.85 | APE67-dihe-in | -66.26, -17.06 | -55.96, -37.76 | APE12-dist-na | 16.4565 | APE11-dist-na | 13.5132 | APE10-dist-na | 11.4728 | APE9-dist-in | 7.9832 | E990V | None | None | XRAY | 1.95 | 0.197 | 0.241 | A | 316.0 | 296.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4ag8 | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 4AGDA | P35968 | 802 | 1169 | 1356.0 | B49:2000 | Type1 | Inactive | DFGout | 16.069 | 10.7232 | BBAminus | -138.96, 169.29 | -127.17, 103.68 | -55.8, -25.22 | 266.19, 75.17 | 52.13, -127.76 | in-in | in | 6.7782 | Saltbr-in | 3.0226 | HRD-out | -100.33, 104.42 | -84.72, 20.62 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.8542 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -119.84, 115.98 | APE9-dihe-in | -119.8, 140.98 | APE8-dihe-in | -66.9, 64.41 | APE8-rot-na | 27.14 | APE67-dihe-in | -54.0, -28.9 | -62.45, -38.96 | APE12-dist-na | 16.4726 | APE11-dist-na | 15.6507 | APE10-dist-na | 13.2897 | APE9-dist-in | 7.7775 | E990V | None | None | XRAY | 2.81 | 0.21 | 0.307 | A | 353.0 | 304.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4agd | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CPBB | P35968 | 820 | 1165 | 1356.0 | C92:60002 | Type1 | Inactive | DFGout | 15.47 | 9.8976 | BBAminus | -145.95, -173.33 | -148.66, 122.86 | -90.71, -55.39 | 280.65, 93.5 | 148.13, 999.0 | in-in | in | 7.4662 | Saltbr-in | 2.7434 | HRD-in | -84.85, -49.1 | 84.19, -23.3 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -49.62 | APE8-dihe-out | -64.93, -12.78 | APE8-rot-na | 24.8 | APE67-dihe-in | -63.19, -14.98 | -60.0, -29.22 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3633 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.224 | 0.286 | B | 314.0 | 263.0 | 33 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3cpb | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2XIRA | P35968 | 816 | 1168 | 1356.0 | 00J:2169 | Type1.5_Back | Inactive | DFGout | 15.9719 | 9.922 | BBAminus | -148.97, -178.6 | -143.75, 112.04 | -61.18, -32.48 | 278.24, 81.67 | 54.1, -120.79 | in-in | in | 7.6929 | Saltbr-in | 2.739 | HRD-in | -84.85, -55.21 | 79.77, -10.15 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.7723 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.39, 115.13 | APE9-dihe-in | -121.67, 148.38 | APE8-dihe-in | -77.59, 66.04 | APE8-rot-na | 29.49 | APE67-dihe-in | -66.29, -14.94 | -52.56, -39.25 | APE12-dist-na | 16.9683 | APE11-dist-na | 13.3284 | APE10-dist-na | 11.4596 | APE9-dist-in | 7.9104 | E990V | None | None | XRAY | 1.5 | 0.219 | 0.238 | A | 316.0 | 296.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 2xir | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 4AGCA | P35968 | 801 | 1169 | 1356.0 | AXI:2000 | Type1.5_Back | Inactive | DFGout | 16.3416 | 10.4506 | BBAminus | -142.09, -174.91 | -148.19, 116.12 | -63.13, -37.04 | 279.42, 73.43 | 58.39, -117.25 | in-in | in | 7.3471 | Saltbr-in | 2.6694 | HRD-out | -119.32, 107.11 | -77.42, 1.81 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5253 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.04, 119.4 | APE9-dihe-in | -126.34, 146.64 | APE8-dihe-in | -75.44, 63.67 | APE8-rot-na | 28.57 | APE67-dihe-in | -65.72, -15.94 | -53.26, -41.15 | APE12-dist-na | 16.7577 | APE11-dist-na | 14.4263 | APE10-dist-na | 12.2303 | APE9-dist-in | 7.621 | E990V | None | None | XRAY | 2.0 | 0.204 | 0.251 | A | 353.0 | 305.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4agc | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3WZEA | P35968 | 815 | 1167 | 1356.0 | BAX:1201 | Type2 | Inactive | DFGout | 15.4233 | 9.7241 | BBAminus | -149.68, 178.07 | -142.38, 105.98 | -66.68, -30.19 | 278.49, 88.73 | 48.89, -116.05 | in-in | in | 7.489 | Saltbr-in | 2.7908 | HRD-in | -80.41, -52.96 | 79.37, -11.85 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.6579 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -114.24, 115.23 | APE9-dihe-in | -125.6, 147.79 | APE8-dihe-in | -77.19, 70.99 | APE8-rot-na | 33.48 | APE67-dihe-in | -66.14, -18.73 | -60.64, -36.14 | APE12-dist-na | 999.0 | APE11-dist-na | 13.6996 | APE10-dist-na | 11.3421 | APE9-dist-out | 8.0812 | T940V | None | None | XRAY | 1.9 | 0.188 | 0.224 | A | 309.0 | 298.0 | 5 | 30 | 29 | 1 | [[834, 1162]] | 1.0 | 3wze | TYR_KDR_HUMAN | TYR | 3.7e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2OH4A | P35968 | 816 | 1171 | 1356.0 | GIG:60303 | Type2 | Inactive | DFGout | 15.0312 | 10.8963 | BBAminus | -143.49, 178.34 | -145.54, 97.19 | -58.33, -39.73 | 283.57, 84.4 | 57.49, 37.59 | in-in | in | 7.3557 | Saltbr-in | 2.6339 | HRD-in | -73.75, -53.05 | 85.59, -23.47 | in-out-out | SNCioo | out-out | ActLoopNT-out | 17.8549 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -140.49, 159.6 | APE9-dihe-in | -103.67, 100.95 | APE8-dihe-out | -54.41, -26.49 | APE8-rot-na | 335.24 | APE67-dihe-in | -67.64, -14.75 | -51.43, -34.8 | APE12-dist-na | 13.3074 | APE11-dist-na | 12.7942 | APE10-dist-na | 13.546 | APE9-dist-out | 11.2059 | None | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.05 | 0.189 | 0.231 | A | 316.0 | 299.0 | 6 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 2oh4 | TYR_KDR_HUMAN | TYR | 5.6e-100 | 339.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2P2IA | P35968 | 817 | 1172 | 1356.0 | 608:60501 | Type2 | Inactive | DFGout | 16.6465 | 10.4202 | BBAminus | -140.93, -165.49 | -165.76, 112.99 | -76.4, -20.94 | 281.97, 76.28 | -89.36, -168.3 | in-in | in | 7.4872 | Saltbr-in | 2.8784 | HRD-in | -67.84, -45.58 | 77.98, -15.16 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 145.47 | APE8-dihe-in | -74.22, 56.93 | APE8-rot-na | 34.49 | APE67-dihe-in | -67.46, -12.22 | -54.19, -35.12 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.6503 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.222 | 0.266 | A | 314.0 | 283.0 | 23 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 2p2i | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3EFLA | P35968 | 817 | 1171 | 1356.0 | 706:60501 | Type2 | Inactive | DFGout | 16.1802 | 10.559 | BBAminus | -138.71, -172.72 | -156.17, 97.27 | -59.6, -16.87 | 285.84, 75.59 | 69.09, 999.0 | in-in | in | 7.3332 | Saltbr-in | 2.8225 | HRD-in | -65.88, -53.9 | 89.41, -28.23 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 54.05 | APE8-rot-na | 34.8 | APE67-dihe-in | -59.53, -20.45 | -52.35, -30.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | A | 314.0 | 279.0 | 26 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3efl | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3EFLB | P35968 | 821 | 1165 | 1356.0 | 706:60502 | Type2 | Inactive | DFGout | 16.1133 | 10.2301 | BBAminus | -141.16, -175.15 | -153.12, 108.94 | -69.6, -34.74 | 280.14, 78.23 | 138.83, 999.0 | in-in | in | 7.0963 | Saltbr-in | 3.2421 | HRD-in | -62.3, -53.81 | 81.7, -4.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.71 | APE8-dihe-out | -39.02, -20.75 | APE8-rot-na | 27.77 | APE67-dihe-in | -68.47, -11.11 | -59.68, -39.14 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.8201 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | B | 314.0 | 263.0 | 32 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3efl | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 5EW3A | P35968 | 821 | 1168 | 1356.0 | 5T2:1201 | Type2 | Inactive | DFGout | 15.8796 | 10.0816 | BBAminus | -139.44, -178.76 | -147.6, 111.79 | -72.49, -35.99 | 276.01, 89.46 | -76.06, 999.0 | in-in | in | 7.4229 | Saltbr-in | 2.9636 | HRD-in | -64.57, -50.86 | 83.75, -23.1 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -57.13 | APE8-dihe-in | -81.64, 66.53 | APE8-rot-na | 27.98 | APE67-dihe-in | -64.62, -30.42 | -51.68, -35.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.717 | None | None | None | XRAY | 2.5 | 0.219 | 0.254 | A | 316.0 | 274.0 | 24 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 5ew3 | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 5EW3B | P35968 | 820 | 1165 | 1356.0 | 5T2:1201 | Type2 | Inactive | DFGout | 15.8616 | 10.1067 | BBAminus | -138.44, -179.7 | -148.59, 111.71 | -71.05, -37.05 | 275.98, 95.16 | -74.59, 999.0 | in-in | in | 7.2167 | Saltbr-in | 2.9045 | HRD-in | -64.78, -51.26 | 84.58, -25.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 135.03 | APE8-dihe-in | -87.05, 66.83 | APE8-rot-na | 29.69 | APE67-dihe-in | -64.72, -30.16 | -52.26, -35.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.6647 | None | None | None | XRAY | 2.5 | 0.219 | 0.254 | B | 316.0 | 266.0 | 30 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 5ew3 | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 6GQOA | P35968 | 811 | 1168 | 1356.0 | F82:61201 | Type2 | Inactive | DFGout | 15.5097 | 9.872 | BBAminus | -137.41, -174.48 | -148.75, 103.09 | -62.92, -33.23 | 281.85, 85.18 | 53.53, -124.22 | in-in | in | 7.6522 | Saltbr-in | 2.8423 | HRD-in | -77.93, -60.11 | 81.09, -6.45 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4783 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.71, 109.7 | APE9-dihe-in | -116.16, 147.79 | APE8-dihe-in | -80.04, 70.94 | APE8-rot-na | 31.31 | APE67-dihe-in | -64.81, -13.7 | -51.33, -43.39 | APE12-dist-na | 16.3984 | APE11-dist-na | 13.2123 | APE10-dist-na | 11.0908 | APE9-dist-in | 7.9513 | None | None | None | XRAY | 1.87 | 0.174 | 0.207 | A | 322.0 | 307.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6gqo | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 6GQPA | P35968 | 821 | 1168 | 1356.0 | F88:61201 | Type2 | Inactive | DFGout | 16.0412 | 9.8283 | BBAminus | -137.29, -179.39 | -147.6, 105.82 | -66.11, -30.27 | 279.44, 81.63 | 58.93, -133.79 | in-in | in | 7.7844 | Saltbr-in | 3.1604 | HRD-in | -72.29, -59.65 | 82.33, -13.78 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.7865 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -109.31, 108.64 | APE9-dihe-in | -119.08, 147.18 | APE8-dihe-in | -76.82, 68.93 | APE8-rot-na | 29.84 | APE67-dihe-in | -64.0, -17.44 | -48.7, -44.35 | APE12-dist-na | 16.2799 | APE11-dist-na | 13.0288 | APE10-dist-na | 10.463 | APE9-dist-out | 8.0203 | None | None | None | XRAY | 2.09 | 0.201 | 0.234 | A | 322.0 | 298.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6gqp | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 6GQQA | P35968 | 813 | 1167 | 1356.0 | F8B:61201 | Type2 | Inactive | DFGout | 16.3179 | 9.8934 | BBAminus | -140.35, 179.68 | -146.82, 105.0 | -62.58, -33.91 | 278.73, 81.84 | 52.08, -122.03 | in-in | in | 7.8551 | Saltbr-in | 2.8701 | HRD-in | -79.41, -58.06 | 81.99, -7.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.6419 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -102.87, 113.66 | APE9-dihe-in | -116.65, 151.24 | APE8-dihe-in | -82.45, 66.44 | APE8-rot-na | 31.58 | APE67-dihe-in | -64.76, -12.48 | -47.19, -45.1 | APE12-dist-na | 16.8675 | APE11-dist-na | 13.2075 | APE10-dist-na | 11.6327 | APE9-dist-out | 8.0466 | None | None | None | XRAY | 1.52 | 0.178 | 0.204 | A | 322.0 | 304.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6gqq | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 6XVJA | P35968 | 813 | 1167 | 1356.0 | O35:1201 | Type2 | Inactive | DFGout | 15.7966 | 9.8597 | BBAminus | -132.46, -168.17 | -160.35, 90.75 | -54.1, -41.9 | 283.85, 84.23 | 55.21, -117.78 | in-in | in | 7.7129 | Saltbr-in | 2.862 | HRD-in | -84.82, -59.51 | 82.99, -12.32 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.6823 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -99.56, 109.17 | APE9-dihe-in | -116.73, 149.21 | APE8-dihe-in | -78.94, 66.26 | APE8-rot-na | 30.73 | APE67-dihe-in | -62.92, -14.21 | -46.08, -45.25 | APE12-dist-na | 17.103 | APE11-dist-na | 13.5038 | APE10-dist-na | 11.3446 | APE9-dist-in | 7.9918 | E990V | None | None | XRAY | 1.78 | 0.18 | 0.215 | A | 322.0 | 305.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6xvj | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 6XVKA | P35968 | 821 | 1168 | 1356.0 | O3E:1201 | Type2 | Inactive | DFGout | 16.107 | 9.9746 | BBAminus | -141.36, -173.76 | -156.84, 95.12 | -54.67, -41.12 | 280.3, 80.99 | 54.89, -110.87 | in-in | in | 7.6818 | Saltbr-in | 2.8161 | HRD-in | -73.74, -55.3 | 80.84, -9.06 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.6059 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -105.81, 104.06 | APE9-dihe-in | -104.53, 149.15 | APE8-dihe-in | -78.71, 70.31 | APE8-rot-na | 29.7 | APE67-dihe-in | -63.75, -14.49 | -47.12, -46.79 | APE12-dist-na | 16.7775 | APE11-dist-na | 12.9611 | APE10-dist-na | 11.3811 | APE9-dist-in | 7.6764 | E990V | None | None | XRAY | 1.99 | 0.208 | 0.244 | A | 322.0 | 298.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6xvk | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 4ASDA | P35968 | 807 | 1168 | 1356.0 | BAX:1500 | Type2 | Inactive | DFGout | 15.5976 | 9.5654 | BBAminus | -143.46, -179.3 | -143.72, 107.55 | -61.84, -34.25 | 277.42, 87.13 | 55.65, -120.32 | in-in | in | 7.5842 | Saltbr-in | 2.9145 | HRD-in | -94.7, -57.23 | 78.86, -11.11 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5646 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.01, 114.08 | APE9-dihe-in | -124.4, 147.41 | APE8-dihe-in | -79.65, 63.41 | APE8-rot-na | 32.33 | APE67-dihe-in | -69.55, -12.31 | -53.55, -35.42 | APE12-dist-na | 16.0444 | APE11-dist-na | 13.4306 | APE10-dist-na | 11.4557 | APE9-dist-in | 7.9757 | E990V | None | None | XRAY | 2.03 | 0.178 | 0.23 | A | 353.0 | 305.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4asd | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 4ASEA | P35968 | 807 | 1169 | 1356.0 | AV9:3169 | Type2 | Inactive | DFGout | 15.5083 | 9.6214 | BBAminus | -131.22, 172.65 | -143.22, 109.66 | -69.47, -29.54 | 275.37, 90.83 | 50.61, -120.83 | in-in | in | 7.6836 | Saltbr-in | 3.0518 | HRD-in | -82.51, -52.61 | 76.99, -4.03 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4515 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.53, 119.23 | APE9-dihe-in | -120.88, 143.86 | APE8-dihe-in | -75.11, 65.17 | APE8-rot-na | 28.66 | APE67-dihe-in | -64.27, -9.66 | -54.44, -43.05 | APE12-dist-na | 16.1551 | APE11-dist-na | 13.7976 | APE10-dist-na | 11.6525 | APE9-dist-in | 7.9754 | E990V | None | None | XRAY | 1.83 | 0.207 | 0.231 | A | 353.0 | 307.0 | 6 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4ase | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3VHEA | P35968 | 811 | 1169 | 1356.0 | 42Q:1170 | Type2 | Inactive | DFGout | 15.9847 | 10.209 | BBAminus | -150.75, 179.81 | -145.06, 104.72 | -59.59, -35.08 | 275.44, 63.4 | 53.57, -124.69 | in-in | in | 7.5456 | Saltbr-in | 2.811 | HRD-in | -83.47, -54.75 | 79.34, -6.09 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.7061 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -104.74, 113.79 | APE9-dihe-in | -123.79, 149.45 | APE8-dihe-in | -81.9, 62.59 | APE8-rot-na | 35.67 | APE67-dihe-in | -65.86, -15.29 | -45.47, -41.75 | APE12-dist-na | 999.0 | APE11-dist-na | 15.5547 | APE10-dist-na | 11.5571 | APE9-dist-out | 8.0431 | None | None | None | XRAY | 1.55 | 0.186 | 0.209 | A | 359.0 | 303.0 | 56 | 30 | 28 | 2 | [[834, 1162]] | 1.0 | 3vhe | TYR_KDR_HUMAN | TYR | 2.4e-99 | 337.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3VHKA | P35968 | 814 | 1168 | 1356.0 | BPK:2001 | Type2 | Inactive | DFGout | 16.4972 | 9.9697 | BBAminus | -142.42, -168.12 | -154.13, 113.05 | -66.9, -34.19 | 279.52, 80.67 | 55.02, -115.26 | in-in | in | 7.7317 | Saltbr-in | 2.6852 | HRD-in | -85.63, -50.5 | 78.47, -9.06 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.6338 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -101.84, 113.0 | APE9-dihe-in | -119.22, 139.89 | APE8-dihe-in | -75.91, 70.12 | APE8-rot-na | 29.63 | APE67-dihe-in | -67.23, -15.54 | -56.62, -35.16 | APE12-dist-na | 999.0 | APE11-dist-na | 13.3761 | APE10-dist-na | 11.0032 | APE9-dist-out | 8.1076 | None | None | None | XRAY | 2.49 | 0.21 | 0.262 | A | 368.0 | 297.0 | 58 | 30 | 28 | 2 | [[834, 1162]] | 1.0 | 3vhk | TYR_KDR_HUMAN | TYR | 2.6e-99 | 337.7 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2QU5A | P35968 | 816 | 1170 | 1356.0 | 276:501 | Type2 | Inactive | DFGout | 15.957 | 9.8302 | BBAminus | -148.46, -172.65 | -150.45, 108.8 | -78.65, -16.42 | 280.25, 86.88 | -99.11, -166.35 | in-in | in | 7.8737 | Saltbr-in | 2.7519 | HRD-in | -80.82, -52.31 | 94.02, -25.74 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -87.63, 5.51 | APE9-dihe-out | 37.61, 55.41 | APE8-dihe-out | -52.54, -22.13 | APE8-rot-na | 25.49 | APE67-dihe-in | -67.04, -17.69 | -59.89, -24.68 | APE12-dist-na | 10.2791 | APE11-dist-na | 14.2242 | APE10-dist-na | 11.1098 | APE9-dist-out | 11.3224 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.95 | 0.213 | 0.251 | A | 314.0 | 292.0 | 13 | 30 | 17 | 13 | [[834, 1162]] | 1.0 | 2qu5 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2QU6A | P35968 | 817 | 1171 | 1356.0 | 857:60501 | Type2 | Inactive | DFGout | 15.9424 | 9.8172 | BBAminus | -132.31, -170.97 | -155.67, 103.74 | -71.24, -21.04 | 287.6, 86.95 | -49.98, 999.0 | in-in | in | 7.8367 | Saltbr-in | 3.056 | HRD-in | -61.86, -49.75 | 81.1, -16.44 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 40.43 | APE8-rot-na | 31.68 | APE67-dihe-in | -68.37, -13.6 | -54.82, -35.61 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.1 | 0.242 | 0.272 | A | 314.0 | 276.0 | 29 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 2qu6 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2RL5A | P35968 | 815 | 1171 | 1356.0 | 2RL:60501 | Type2 | Inactive | DFGout | 15.3924 | 11.07 | BBAminus | -145.48, -175.23 | -148.97, 113.05 | -80.1, -11.01 | 289.69, 95.02 | 69.28, 57.0 | in-in | in | 7.8261 | Saltbr-in | 2.6984 | HRD-in | -65.08, -49.32 | 80.71, -16.94 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -86.71, -13.59 | APE9-dihe-out | 45.53, 52.75 | APE8-dihe-out | -54.88, -21.97 | APE8-rot-na | 32.05 | APE67-dihe-in | -73.02, -12.93 | -62.39, -23.08 | APE12-dist-na | 7.9303 | APE11-dist-na | 10.6315 | APE10-dist-na | 6.7426 | APE9-dist-out | 11.661 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.65 | 0.199 | 0.233 | A | 314.0 | 290.0 | 17 | 30 | 16 | 14 | [[834, 1162]] | 1.0 | 2rl5 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3B8QB | P35968 | 820 | 1166 | 1356.0 | 900:60502 | Type2 | Inactive | DFGout | 15.4044 | 10.0777 | BBAminus | -136.11, -171.43 | -160.46, 118.31 | -80.85, -45.83 | 290.91, 83.9 | 123.21, 999.0 | in-in | in | 7.8977 | Saltbr-in | 2.9027 | HRD-in | -68.36, -46.63 | 75.78, -5.88 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 155.56 | APE8-dihe-out | -60.35, -14.62 | APE8-rot-na | 30.93 | APE67-dihe-in | -68.62, -6.92 | -55.79, -32.87 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2967 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.75 | 0.218 | 0.276 | B | 314.0 | 271.0 | 26 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3b8q | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3BE2A | P35968 | 815 | 1171 | 1356.0 | RAJ:60501 | Type2 | Inactive | DFGout | 14.1127 | 11.0427 | BBAminus | -134.72, 177.84 | -152.38, 97.13 | -77.52, -8.1 | 302.77, 127.65 | 76.19, 999.0 | in-in | in | 7.941 | Saltbr-in | 2.7693 | HRD-in | -67.93, -53.26 | 79.3, -9.77 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 56.48 | APE8-rot-na | 341.32 | APE67-dihe-in | -65.72, -14.43 | -46.07, -42.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.75 | 0.197 | 0.226 | A | 314.0 | 285.0 | 22 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3be2 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CP9A | P35968 | 817 | 1171 | 1356.0 | C19:60501 | Type2 | Inactive | DFGout | 16.6202 | 10.2751 | BBAminus | -128.38, -176.57 | -155.05, 99.17 | -63.66, -9.88 | 278.68, 88.56 | -54.74, 999.0 | in-in | in | 7.7333 | Saltbr-in | 2.6364 | HRD-in | -61.14, -53.92 | 79.09, -9.79 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 101.57 | APE8-dihe-out | -50.34, -15.58 | APE8-rot-na | 28.54 | APE67-dihe-in | -69.67, -13.51 | -65.76, -26.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.5778 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.5 | 0.211 | 0.263 | A | 314.0 | 281.0 | 24 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3cp9 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CP9B | P35968 | 819 | 1165 | 1356.0 | C19:60502 | Type2 | Inactive | DFGout | 16.8412 | 10.4044 | BBAminus | -132.75, -171.12 | -162.18, 105.04 | -62.12, -28.88 | 281.99, 80.12 | 49.45, -86.0 | in-in | in | 7.6456 | Saltbr-in | 3.0483 | HRD-in | -88.31, -43.32 | 78.52, -15.92 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -57.69 | APE8-dihe-out | -39.24, -27.85 | APE8-rot-na | 24.86 | APE67-dihe-in | -68.9, -8.27 | -59.68, -31.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.4403 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.5 | 0.211 | 0.263 | B | 314.0 | 269.0 | 28 | 30 | 13 | 17 | [[834, 1162]] | 1.0 | 3cp9 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CPCB | P35968 | 820 | 1165 | 1356.0 | C52:60002 | Type2 | Inactive | DFGout | 16.6391 | 10.3787 | BBAminus | -131.82, -178.95 | -148.17, 107.11 | -69.23, -53.88 | 273.75, 87.39 | 111.77, 999.0 | in-in | in | 7.4849 | Saltbr-in | 2.706 | HRD-in | -75.42, -46.4 | 80.7, -16.54 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -53.89 | APE8-dihe-out | -53.45, -16.48 | APE8-rot-na | 17.35 | APE67-dihe-in | -69.92, -17.21 | -63.01, -26.25 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3843 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.221 | 0.272 | B | 314.0 | 262.0 | 34 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3cpc | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3DTWB | P35968 | 820 | 1166 | 1356.0 | A96:60502 | Type2 | Inactive | DFGout | 15.0355 | 10.1682 | BBAminus | -136.42, -166.86 | -159.08, 106.24 | -84.37, -81.02 | 295.18, 95.96 | 174.82, 139.27 | in-in | in | 8.1766 | Saltbr-in | 2.9571 | HRD-in | -66.59, -51.66 | 77.85, -16.94 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, 31.74 | APE9-dihe-out | -53.82, -56.19 | APE8-dihe-out | -45.11, -17.45 | APE8-rot-na | 28.36 | APE67-dihe-in | -71.35, -4.04 | -72.8, -21.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.2914 | APE9-dist-out | 11.5266 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.9 | 0.215 | 0.279 | B | 314.0 | 269.0 | 28 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 3dtw | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3EWHA | P35968 | 815 | 1171 | 1356.0 | K11:60001 | Type2 | Inactive | DFGout | 15.139 | 11.4202 | BBAminus | -133.49, -179.18 | -135.71, 102.66 | -69.48, -9.86 | 280.78, 102.57 | 67.93, 33.26 | in-in | in | 7.9373 | Saltbr-in | 3.0791 | HRD-in | -71.49, -51.89 | 78.14, -10.7 | in-out-none | SNCion | out-none | ActLoopNT-out | 12.9444 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 130.93 | APE8-dihe-in | -76.46, 69.83 | APE8-rot-na | 30.0 | APE67-dihe-in | -66.36, -17.49 | -56.88, -35.11 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.9722 | C817A,V916T,E990V | None | None | XRAY | 1.6 | 0.208 | 0.234 | A | 314.0 | 295.0 | 12 | 30 | 21 | 9 | [[834, 1162]] | 1.0 | 3ewh | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3U6JA | P35968 | 815 | 1171 | 1356.0 | 03X:60001 | Type2 | Inactive | DFGout | 14.9795 | 10.356 | BBAminus | -144.73, -178.41 | -146.44, 121.96 | -64.93, -27.75 | 282.37, 79.48 | 52.91, -122.32 | in-in | in | 7.455 | Saltbr-in | 2.8674 | HRD-in | -74.57, -56.02 | 80.88, -14.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.1328 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -99.27, 117.84 | APE9-dihe-in | -122.3, 141.03 | APE8-dihe-in | -77.42, 64.76 | APE8-rot-na | 30.56 | APE67-dihe-in | -69.06, -14.4 | -51.48, -37.1 | APE12-dist-na | 17.3677 | APE11-dist-na | 14.2143 | APE10-dist-na | 12.3875 | APE9-dist-in | 7.7332 | V916T,E990V | None | None | XRAY | 2.15 | 0.196 | 0.23 | A | 314.0 | 305.0 | 2 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 3u6j | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3C7QA | P35968 | 819 | 1171 | 1356.0 | XIN:1172 | Type1 | Inactive | DFGout | 15.7851 | 9.7942 | None | -118.96, 138.15 | -110.64, 113.79 | -73.47, 999.0 | 192.45, 128.99 | 999.0, 999.0 | in-in | in | 7.2832 | Saltbr-in | 2.6084 | HRD-in | -83.9, -48.68 | 82.47, -6.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -147.17, 145.76 | APE9-dihe-in | -104.98, 98.81 | APE8-dihe-out | -50.37, -26.53 | APE8-rot-na | 330.15 | APE67-dihe-in | -62.19, -10.0 | -56.65, -35.85 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.1746 | None | PTR1054,PTR1059 | CME862,CME1007,CME1024,PTR1054,PTR1059 | XRAY | 2.1 | 0.221 | 0.279 | A | 316.0 | 291.0 | 10 | 30 | 26 | 4 | [[834, 1162]] | 1.0 | 3c7q | TYR_KDR_HUMAN | TYR | 3.9e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2P2IB | P35968 | 820 | 1168 | 1356.0 | 608:60502 | Type1 | Inactive | DFGout | 16.2739 | 10.2035 | None | -141.39, -171.24 | -157.47, 119.0 | -85.08, 999.0 | 285.18, 81.66 | 999.0, 999.0 | in-in | in | 7.1432 | Saltbr-in | 3.2708 | HRD-in | -71.95, -45.89 | 71.89, -7.38 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 36.68 | APE8-rot-na | 31.31 | APE67-dihe-in | -54.41, -18.08 | -58.67, -41.73 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.222 | 0.266 | B | 314.0 | 263.0 | 36 | 30 | 10 | 20 | [[834, 1162]] | 1.0 | 2p2i | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3VNTA | P35968 | 812 | 1168 | 1356.0 | 0JA:2001 | Type2 | Inactive | DFGout | 16.7639 | 8.3863 | None | -132.49, -178.83 | -142.53, 104.52 | -68.92, -32.97 | 219.02, 49.93 | 58.07, -122.23 | in-in | in | 7.4677 | Saltbr-in | 2.7462 | HRD-in | -79.08, -51.8 | 75.79, -7.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5421 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.01, 111.64 | APE9-dihe-in | -121.89, 148.7 | APE8-dihe-in | -79.2, 68.13 | APE8-rot-na | 30.95 | APE67-dihe-in | -64.82, -12.79 | -56.01, -39.41 | APE12-dist-na | 16.8255 | APE11-dist-na | 13.4544 | APE10-dist-na | 11.2921 | APE9-dist-in | 7.8693 | None | None | None | XRAY | 1.64 | 0.153 | 0.192 | A | 318.0 | 301.0 | 6 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 3vnt | TYR_KDR_HUMAN | TYR | 4.2e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3VO3A | P35968 | 812 | 1168 | 1356.0 | 0KF:2001 | Type2 | Inactive | DFGout | 16.4477 | 8.2146 | None | -125.16, 179.81 | -141.05, 99.79 | -70.03, -34.74 | 215.55, 55.41 | 59.77, -120.61 | in-in | in | 7.3573 | Saltbr-in | 2.8979 | HRD-in | -84.45, -53.71 | 76.95, -3.4 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4768 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.91, 109.54 | APE9-dihe-in | -120.7, 147.5 | APE8-dihe-in | -78.09, 65.8 | APE8-rot-na | 32.33 | APE67-dihe-in | -67.73, -12.3 | -53.4, -39.21 | APE12-dist-na | 17.0304 | APE11-dist-na | 14.0671 | APE10-dist-na | 11.3935 | APE9-dist-in | 7.9974 | None | None | None | XRAY | 1.52 | 0.162 | 0.182 | A | 318.0 | 303.0 | 4 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 3vo3 | TYR_KDR_HUMAN | TYR | 4.2e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 2QU6B | P35968 | 822 | 1165 | 1356.0 | 857:60502 | Type2 | Inactive | DFGout | 15.9633 | 9.5409 | None | -133.96, -169.17 | -160.0, 100.56 | -72.82, 999.0 | 288.62, 90.71 | 999.0, 999.0 | in-in | in | 7.9527 | Saltbr-in | 3.0946 | HRD-in | -62.66, -51.11 | 76.69, -2.42 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 122.74 | APE8-dihe-in | -72.44, 73.71 | APE8-rot-na | 32.18 | APE67-dihe-in | -66.59, -17.43 | -56.47, -30.13 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.2922 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.1 | 0.242 | 0.272 | B | 314.0 | 260.0 | 34 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 2qu6 | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3B8QA | P35968 | 818 | 1171 | 1356.0 | 900:60501 | Type2 | Inactive | DFGout | 15.4672 | 9.913 | None | -131.74, -168.2 | -159.75, 118.5 | -86.72, 999.0 | 284.22, 100.5 | 999.0, 999.0 | in-in | in | 7.7591 | Saltbr-in | 2.7653 | HRD-in | -57.53, -50.67 | 79.88, -14.29 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 160.03 | APE8-dihe-out | -77.48, -12.97 | APE8-rot-na | 36.4 | APE67-dihe-in | -68.93, -8.62 | -57.21, -28.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.0722 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.75 | 0.218 | 0.276 | A | 314.0 | 285.0 | 19 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3b8q | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CPBA | P35968 | 819 | 1171 | 1356.0 | C92:60001 | Type2 | Inactive | DFGout | 15.3326 | 9.7507 | None | -143.96, -172.89 | -147.19, 119.38 | -89.94, 999.0 | 278.49, 101.53 | 999.0, 999.0 | in-in | in | 7.7633 | Saltbr-in | 3.5846 | HRD-in | -60.85, -44.16 | 62.59, 3.77 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 128.93 | APE8-dihe-out | -45.12, -28.83 | APE8-rot-na | 328.95 | APE67-dihe-in | -65.36, -7.17 | -53.29, -33.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.351 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.224 | 0.286 | A | 314.0 | 278.0 | 25 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3cpb | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CPCA | P35968 | 820 | 1171 | 1356.0 | C52:60001 | Type2 | Inactive | DFGout | 16.8028 | 10.3818 | None | -127.27, -176.88 | -144.84, 92.18 | -66.45, 999.0 | 268.44, 99.63 | 999.0, 999.0 | in-out | in | 8.0268 | Saltbr-out | 3.9767 | HRD-in | -74.56, -44.56 | 79.03, -21.68 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.84 | APE8-dihe-out | -45.97, -30.08 | APE8-rot-na | 328.28 | APE67-dihe-in | -73.13, -9.14 | -56.02, -29.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3564 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.221 | 0.272 | A | 314.0 | 277.0 | 25 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3cpc | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3DTWA | P35968 | 818 | 1171 | 1356.0 | A96:60501 | Type2 | Inactive | DFGout | 15.1581 | 10.0994 | None | -129.54, -170.94 | -153.49, 103.32 | -82.68, 999.0 | 294.21, 96.03 | 999.0, 999.0 | in-in | in | 8.0061 | Saltbr-in | 2.6405 | HRD-in | -53.04, -53.77 | 79.82, -12.25 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.1 | APE8-dihe-out | -46.34, -20.16 | APE8-rot-na | 23.94 | APE67-dihe-in | -60.71, -7.92 | -57.08, -38.78 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2341 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.9 | 0.215 | 0.279 | A | 314.0 | 281.0 | 23 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3dtw | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3CJFA | P35968 | 817 | 1168 | 1356.0 | SAV:61167 | Type1 | Inactive | None | 999.0 | 999.0 | None | -83.44, 111.78 | -118.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-out | in | 7.8208 | Saltbr-out | 5.2231 | HRD-out | -105.6, 121.11 | -71.37, -10.71 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.8895 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 48.59 | APE8-rot-na | 25.36 | APE67-dihe-in | -69.88, -14.36 | -60.34, -37.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | CSO862,CSO1007,CSO1024,CSO1045,CSO1116 | XRAY | 2.15 | 0.205 | 0.258 | A | 309.0 | 281.0 | 17 | 30 | 16 | 14 | [[834, 1162]] | 1.0 | 3cjf | TYR_KDR_HUMAN | TYR | 4.8e-100 | 340.1 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 1YWNA | P35968 | 820 | 1171 | 1356.0 | LIF:60301 | Type1 | Inactive | None | 999.0 | 999.0 | None | -128.91, 171.96 | -143.62, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 7.2102 | Saltbr-in | 2.725 | HRD-in | -77.88, -50.07 | 82.87, -17.6 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -141.39, 161.44 | APE9-dihe-in | -104.18, 100.32 | APE8-dihe-out | -56.09, -24.71 | APE8-rot-na | 336.02 | APE67-dihe-in | -70.59, -14.0 | -51.58, -32.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2392 | E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.71 | 0.206 | 0.23 | A | 316.0 | 281.0 | 21 | 30 | 24 | 6 | [[834, 1162]] | 1.0 | 1ywn | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | 3VIDA | P35968 | 813 | 1168 | 1356.0 | 4TT:2001 | Type1 | Inactive | None | 999.0 | 999.0 | None | -128.64, 167.68 | -132.79, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 7.3263 | Saltbr-in | 2.9803 | HRD-in | -77.53, -50.55 | 79.3, -13.28 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -152.12, 159.09 | APE9-dihe-in | -96.12, 109.5 | APE8-dihe-out | -66.36, -14.96 | APE8-rot-na | 337.32 | APE67-dihe-in | -69.61, -3.71 | -60.46, -30.42 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3777 | None | None | None | XRAY | 2.3 | 0.247 | 0.281 | A | 356.0 | 299.0 | 57 | 30 | 23 | 7 | [[834, 1162]] | 1.0 | 3vid | TYR_KDR_HUMAN | TYR | 2.3e-99 | 337.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| KDR | VGFR2_HUMAN | AF-P35968-K1A | P35968 | 826 | 1170 | 1356.0 | No_ligand | No_ligand | Active | DFGin | 6.724 | 13.7539 | BLAminus | -135.49, -178.07 | 64.31, 58.61 | -79.84, 14.65 | 291.25, 84.84 | -59.67, -29.27 | in-in | in | 7.2738 | Saltbr-in | 2.6536 | HRD-in | -79.81, -44.23 | 66.36, -15.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9851 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.88, 109.91 | APE9-dihe-in | -121.83, 150.33 | APE8-dihe-in | -76.73, 95.83 | APE8-rot-na | 34.09 | APE67-dihe-in | -64.1, -25.24 | -52.96, -31.45 | APE12-dist-na | 14.1753 | APE11-dist-na | 7.9361 | APE10-dist-na | 10.7309 | APE9-dist-in | 6.1962 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 345.0 | 345.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | AF-P35968-K1 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.1e-99 | 338.0 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | AF-P35968-K3A | P35968 | 826 | 1170 | 1356.0 | No_ligand | No_ligand | Active | DFGin | 6.4666 | 13.4597 | BLAminus | -139.09, -177.77 | 61.66, 65.38 | -79.85, 17.72 | 289.99, 89.58 | -61.52, -31.06 | in-in | in | 7.8222 | Saltbr-in | 2.7291 | HRD-in | -81.16, -45.43 | 63.07, 4.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9147 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -52.76, 130.74 | APE9-dihe-in | -112.3, 130.74 | APE8-dihe-in | -82.3, 61.23 | APE8-rot-na | 36.08 | APE67-dihe-in | -68.73, -19.78 | -48.02, -36.64 | APE12-dist-na | 13.331 | APE11-dist-na | 7.163 | APE10-dist-na | 8.5381 | APE9-dist-in | 6.7571 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 345.0 | 345.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | AF-P35968-K3 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.1e-99 | 338.0 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CJGA | P35968 | 816 | 1168 | 1356.0 | KIM:61167 | Type1 | Inactive | DFGin | 7.412 | 14.1279 | BLAminus | -120.91, -162.35 | 48.63, 86.88 | -107.47, 22.59 | 302.68, 92.72 | -76.12, -15.36 | in-in | in | 7.1793 | Saltbr-in | 2.6808 | HRD-in | -77.13, -50.16 | 74.93, 1.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9769 | ActLoopCT-out | TYR | APEdihe_nnnao | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 19.76 | APE8-rot-na | 1.33 | APE67-dihe-out | -66.63, -12.94 | 74.8, -54.69 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | CSO862,CSO1024 | XRAY | 2.25 | 0.209 | 0.253 | A | 309.0 | 282.0 | 17 | 30 | 16 | 14 | [[834, 1162]] | 1.0 | 3cjg | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.8e-100 | 340.1 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2P2HA | P35968 | 815 | 1172 | 1356.0 | 994:60501 | Type1 | Inactive | DFGin | 5.7777 | 13.4944 | BLAplus | -120.41, 168.7 | 57.61, 43.27 | -102.94, -14.81 | 60.29, 84.2 | -108.45, 28.25 | in-in | in | 7.3498 | Saltbr-in | 2.5269 | HRD-in | -63.68, -53.12 | 82.34, -19.49 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, 158.7 | APE9-dihe-out | 54.03, 51.67 | APE8-dihe-out | -62.29, -19.22 | APE8-rot-na | 32.86 | APE67-dihe-in | -68.4, -12.54 | -60.9, -27.46 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 19.0397 | APE9-dist-out | 11.1812 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.95 | 0.205 | 0.229 | A | 314.0 | 289.0 | 19 | 30 | 15 | 15 | [[834, 1162]] | 1.0 | 2p2h | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3WZDA | P35968 | 820 | 1167 | 1356.0 | LEV:1201 | Type1 | Inactive | DFGin | 5.4262 | 13.8027 | BLBplus | -131.31, 171.12 | 64.88, 24.46 | -69.96, 136.97 | 45.36, 91.24 | 79.76, 6.08 | in-in | in | 7.3091 | Saltbr-in | 2.9428 | HRD-in | -65.52, -53.13 | 82.13, -20.42 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -70.62 | APE8-dihe-out | -53.22, -31.36 | APE8-rot-na | 22.8 | APE67-dihe-in | -66.02, -15.12 | -58.21, -29.08 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2484 | T940V | None | None | XRAY | 1.57 | 0.184 | 0.212 | A | 309.0 | 278.0 | 20 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 3wzd | Homo sapiens | TYR_KDR_HUMAN | TYR | 3.7e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3B8RA | P35968 | 818 | 1171 | 1356.0 | 887:60201 | Type1 | Inactive | DFGin | 5.4242 | 13.8708 | BLBplus | -147.04, 169.16 | 57.66, 43.33 | -97.43, 156.79 | 47.05, 78.4 | 59.04, 37.41 | in-in | in | 7.2508 | Saltbr-in | 2.6796 | HRD-in | -59.31, -52.93 | 80.34, -8.78 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 162.25 | APE8-dihe-out | -73.03, -9.68 | APE8-rot-na | 326.59 | APE67-dihe-in | -61.58, -18.77 | -55.36, -31.25 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2594 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.204 | 0.259 | A | 314.0 | 282.0 | 22 | 30 | 13 | 17 | [[834, 1162]] | 1.0 | 3b8r | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3B8RB | P35968 | 821 | 1166 | 1356.0 | 887:60202 | Type1 | Inactive | DFGin | 5.4416 | 13.8855 | BLBplus | -153.23, 176.22 | 49.55, 49.42 | -108.14, 150.46 | 48.31, 72.77 | 69.58, 35.57 | in-in | in | 7.3928 | Saltbr-in | 2.7455 | HRD-in | -68.34, -51.75 | 79.37, -8.5 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.55 | APE8-dihe-out | -62.02, -11.57 | APE8-rot-na | 326.58 | APE67-dihe-in | -65.24, -19.42 | -57.92, -26.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2614 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.204 | 0.259 | B | 314.0 | 267.0 | 29 | 30 | 13 | 17 | [[834, 1162]] | 1.0 | 3b8r | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 1VR2A | P35968 | 820 | 1168 | 1356.0 | No_ligand | No_ligand | Inactive | DFGin | 6.1971 | 12.2007 | None | -132.36, 167.84 | 67.89, 27.54 | -86.08, 999.0 | 49.78, 130.84 | 999.0, 999.0 | in-in | in | 7.7298 | Saltbr-in | 2.9904 | HRD-in | -66.37, -43.4 | 76.06, -15.34 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -137.43, 155.04 | APE9-dihe-in | -108.73, 90.95 | APE8-dihe-out | -47.33, -14.52 | APE8-rot-na | 323.83 | APE67-dihe-in | -64.29, -7.8 | -69.97, -29.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.4665 | E990V | PTR1059 | PTR1059 | XRAY | 2.4 | 0.215 | 999.0 | A | 316.0 | 275.0 | 24 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 1vr2 | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 1Y6AA | P35968 | 820 | 1167 | 1356.0 | AAZ:60201 | Type1 | Inactive | DFGinter | 8.6659 | 8.8381 | None | -73.14, 116.72 | -103.71, 73.1 | -178.89, 999.0 | 25.84, 61.42 | 999.0, 999.0 | in-in | in | 7.4703 | Saltbr-in | 2.8011 | HRD-in | -83.04, -53.13 | 81.96, -16.64 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -20.95 | APE8-rot-na | 328.99 | APE67-dihe-in | -63.85, -16.51 | -63.27, -26.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.1 | 0.196 | 0.217 | A | 366.0 | 261.0 | 87 | 30 | 10 | 20 | [[834, 1162]] | 1.0 | 1y6a | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.6e-99 | 337.7 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 1Y6BA | P35968 | 819 | 1168 | 1356.0 | AAX:60201 | Type1 | Inactive | DFGinter | 8.9591 | 8.6911 | None | -70.35, 112.74 | -90.68, -29.02 | -42.32, 999.0 | 351.89, 106.67 | 999.0, 999.0 | in-in | in | 7.4818 | Saltbr-in | 2.9568 | HRD-in | -82.96, -58.21 | 87.46, -12.31 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 69.65 | APE8-rot-na | 33.76 | APE67-dihe-in | -65.54, -15.03 | -63.36, -37.08 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.1 | 0.194 | 0.236 | A | 366.0 | 266.0 | 84 | 30 | 10 | 20 | [[834, 1162]] | 1.0 | 1y6b | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.6e-99 | 337.7 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 4AG8A | P35968 | 816 | 1168 | 1356.0 | AXI:2000 | Type1 | Inactive | DFGout | 16.4966 | 10.362 | BBAminus | -143.7, -179.58 | -144.17, 113.57 | -60.35, -33.13 | 275.19, 77.68 | 54.27, -121.79 | in-in | in | 7.5186 | Saltbr-in | 2.748 | HRD-in | -80.25, -53.16 | 76.08, -12.6 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5659 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.55, 111.08 | APE9-dihe-in | -116.46, 147.01 | APE8-dihe-in | -77.77, 66.25 | APE8-rot-na | 30.85 | APE67-dihe-in | -66.26, -17.06 | -55.96, -37.76 | APE12-dist-na | 16.4565 | APE11-dist-na | 13.5132 | APE10-dist-na | 11.4728 | APE9-dist-in | 7.9832 | E990V | None | None | XRAY | 1.95 | 0.197 | 0.241 | A | 316.0 | 296.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4ag8 | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 4AGDA | P35968 | 802 | 1169 | 1356.0 | B49:2000 | Type1 | Inactive | DFGout | 16.069 | 10.7232 | BBAminus | -138.96, 169.29 | -127.17, 103.68 | -55.8, -25.22 | 266.19, 75.17 | 52.13, -127.76 | in-in | in | 6.7782 | Saltbr-in | 3.0226 | HRD-out | -100.33, 104.42 | -84.72, 20.62 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.8542 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -119.84, 115.98 | APE9-dihe-in | -119.8, 140.98 | APE8-dihe-in | -66.9, 64.41 | APE8-rot-na | 27.14 | APE67-dihe-in | -54.0, -28.9 | -62.45, -38.96 | APE12-dist-na | 16.4726 | APE11-dist-na | 15.6507 | APE10-dist-na | 13.2897 | APE9-dist-in | 7.7775 | E990V | None | None | XRAY | 2.81 | 0.21 | 0.307 | A | 353.0 | 304.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4agd | Homo sapiens | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CPBB | P35968 | 820 | 1165 | 1356.0 | C92:60002 | Type1 | Inactive | DFGout | 15.47 | 9.8976 | BBAminus | -145.95, -173.33 | -148.66, 122.86 | -90.71, -55.39 | 280.65, 93.5 | 148.13, 999.0 | in-in | in | 7.4662 | Saltbr-in | 2.7434 | HRD-in | -84.85, -49.1 | 84.19, -23.3 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -49.62 | APE8-dihe-out | -64.93, -12.78 | APE8-rot-na | 24.8 | APE67-dihe-in | -63.19, -14.98 | -60.0, -29.22 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3633 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.224 | 0.286 | B | 314.0 | 263.0 | 33 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3cpb | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2XIRA | P35968 | 816 | 1168 | 1356.0 | 00J:2169 | Type1.5_Back | Inactive | DFGout | 15.9719 | 9.922 | BBAminus | -148.97, -178.6 | -143.75, 112.04 | -61.18, -32.48 | 278.24, 81.67 | 54.1, -120.79 | in-in | in | 7.6929 | Saltbr-in | 2.739 | HRD-in | -84.85, -55.21 | 79.77, -10.15 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.7723 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.39, 115.13 | APE9-dihe-in | -121.67, 148.38 | APE8-dihe-in | -77.59, 66.04 | APE8-rot-na | 29.49 | APE67-dihe-in | -66.29, -14.94 | -52.56, -39.25 | APE12-dist-na | 16.9683 | APE11-dist-na | 13.3284 | APE10-dist-na | 11.4596 | APE9-dist-in | 7.9104 | E990V | None | None | XRAY | 1.5 | 0.219 | 0.238 | A | 316.0 | 296.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 2xir | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 4AGCA | P35968 | 801 | 1169 | 1356.0 | AXI:2000 | Type1.5_Back | Inactive | DFGout | 16.3416 | 10.4506 | BBAminus | -142.09, -174.91 | -148.19, 116.12 | -63.13, -37.04 | 279.42, 73.43 | 58.39, -117.25 | in-in | in | 7.3471 | Saltbr-in | 2.6694 | HRD-out | -119.32, 107.11 | -77.42, 1.81 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5253 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.04, 119.4 | APE9-dihe-in | -126.34, 146.64 | APE8-dihe-in | -75.44, 63.67 | APE8-rot-na | 28.57 | APE67-dihe-in | -65.72, -15.94 | -53.26, -41.15 | APE12-dist-na | 16.7577 | APE11-dist-na | 14.4263 | APE10-dist-na | 12.2303 | APE9-dist-in | 7.621 | E990V | None | None | XRAY | 2.0 | 0.204 | 0.251 | A | 353.0 | 305.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4agc | Homo sapiens | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3WZEA | P35968 | 815 | 1167 | 1356.0 | BAX:1201 | Type2 | Inactive | DFGout | 15.4233 | 9.7241 | BBAminus | -149.68, 178.07 | -142.38, 105.98 | -66.68, -30.19 | 278.49, 88.73 | 48.89, -116.05 | in-in | in | 7.489 | Saltbr-in | 2.7908 | HRD-in | -80.41, -52.96 | 79.37, -11.85 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.6579 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -114.24, 115.23 | APE9-dihe-in | -125.6, 147.79 | APE8-dihe-in | -77.19, 70.99 | APE8-rot-na | 33.48 | APE67-dihe-in | -66.14, -18.73 | -60.64, -36.14 | APE12-dist-na | 999.0 | APE11-dist-na | 13.6996 | APE10-dist-na | 11.3421 | APE9-dist-out | 8.0812 | T940V | None | None | XRAY | 1.9 | 0.188 | 0.224 | A | 309.0 | 298.0 | 5 | 30 | 29 | 1 | [[834, 1162]] | 1.0 | 3wze | Homo sapiens | TYR_KDR_HUMAN | TYR | 3.7e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2OH4A | P35968 | 816 | 1171 | 1356.0 | GIG:60303 | Type2 | Inactive | DFGout | 15.0312 | 10.8963 | BBAminus | -143.49, 178.34 | -145.54, 97.19 | -58.33, -39.73 | 283.57, 84.4 | 57.49, 37.59 | in-in | in | 7.3557 | Saltbr-in | 2.6339 | HRD-in | -73.75, -53.05 | 85.59, -23.47 | in-out-out | SNCioo | out-out | ActLoopNT-out | 17.8549 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -140.49, 159.6 | APE9-dihe-in | -103.67, 100.95 | APE8-dihe-out | -54.41, -26.49 | APE8-rot-na | 335.24 | APE67-dihe-in | -67.64, -14.75 | -51.43, -34.8 | APE12-dist-na | 13.3074 | APE11-dist-na | 12.7942 | APE10-dist-na | 13.546 | APE9-dist-out | 11.2059 | None | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.05 | 0.189 | 0.231 | A | 316.0 | 299.0 | 6 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 2oh4 | Homo sapiens | TYR_KDR_HUMAN | TYR | 5.6e-100 | 339.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2P2IA | P35968 | 817 | 1172 | 1356.0 | 608:60501 | Type2 | Inactive | DFGout | 16.6465 | 10.4202 | BBAminus | -140.93, -165.49 | -165.76, 112.99 | -76.4, -20.94 | 281.97, 76.28 | -89.36, -168.3 | in-in | in | 7.4872 | Saltbr-in | 2.8784 | HRD-in | -67.84, -45.58 | 77.98, -15.16 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 145.47 | APE8-dihe-in | -74.22, 56.93 | APE8-rot-na | 34.49 | APE67-dihe-in | -67.46, -12.22 | -54.19, -35.12 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.6503 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.222 | 0.266 | A | 314.0 | 283.0 | 23 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 2p2i | Homo sapiens | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3EFLA | P35968 | 817 | 1171 | 1356.0 | 706:60501 | Type2 | Inactive | DFGout | 16.1802 | 10.559 | BBAminus | -138.71, -172.72 | -156.17, 97.27 | -59.6, -16.87 | 285.84, 75.59 | 69.09, 999.0 | in-in | in | 7.3332 | Saltbr-in | 2.8225 | HRD-in | -65.88, -53.9 | 89.41, -28.23 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 54.05 | APE8-rot-na | 34.8 | APE67-dihe-in | -59.53, -20.45 | -52.35, -30.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | A | 314.0 | 279.0 | 26 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3efl | Homo sapiens | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3EFLB | P35968 | 821 | 1165 | 1356.0 | 706:60502 | Type2 | Inactive | DFGout | 16.1133 | 10.2301 | BBAminus | -141.16, -175.15 | -153.12, 108.94 | -69.6, -34.74 | 280.14, 78.23 | 138.83, 999.0 | in-in | in | 7.0963 | Saltbr-in | 3.2421 | HRD-in | -62.3, -53.81 | 81.7, -4.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.71 | APE8-dihe-out | -39.02, -20.75 | APE8-rot-na | 27.77 | APE67-dihe-in | -68.47, -11.11 | -59.68, -39.14 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.8201 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | B | 314.0 | 263.0 | 32 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3efl | Homo sapiens | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 5EW3A | P35968 | 821 | 1168 | 1356.0 | 5T2:1201 | Type2 | Inactive | DFGout | 15.8796 | 10.0816 | BBAminus | -139.44, -178.76 | -147.6, 111.79 | -72.49, -35.99 | 276.01, 89.46 | -76.06, 999.0 | in-in | in | 7.4229 | Saltbr-in | 2.9636 | HRD-in | -64.57, -50.86 | 83.75, -23.1 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -57.13 | APE8-dihe-in | -81.64, 66.53 | APE8-rot-na | 27.98 | APE67-dihe-in | -64.62, -30.42 | -51.68, -35.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.717 | None | None | None | XRAY | 2.5 | 0.219 | 0.254 | A | 316.0 | 274.0 | 24 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 5ew3 | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 5EW3B | P35968 | 820 | 1165 | 1356.0 | 5T2:1201 | Type2 | Inactive | DFGout | 15.8616 | 10.1067 | BBAminus | -138.44, -179.7 | -148.59, 111.71 | -71.05, -37.05 | 275.98, 95.16 | -74.59, 999.0 | in-in | in | 7.2167 | Saltbr-in | 2.9045 | HRD-in | -64.78, -51.26 | 84.58, -25.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 135.03 | APE8-dihe-in | -87.05, 66.83 | APE8-rot-na | 29.69 | APE67-dihe-in | -64.72, -30.16 | -52.26, -35.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.6647 | None | None | None | XRAY | 2.5 | 0.219 | 0.254 | B | 316.0 | 266.0 | 30 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 5ew3 | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 6GQOA | P35968 | 811 | 1168 | 1356.0 | F82:61201 | Type2 | Inactive | DFGout | 15.5097 | 9.872 | BBAminus | -137.41, -174.48 | -148.75, 103.09 | -62.92, -33.23 | 281.85, 85.18 | 53.53, -124.22 | in-in | in | 7.6522 | Saltbr-in | 2.8423 | HRD-in | -77.93, -60.11 | 81.09, -6.45 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4783 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.71, 109.7 | APE9-dihe-in | -116.16, 147.79 | APE8-dihe-in | -80.04, 70.94 | APE8-rot-na | 31.31 | APE67-dihe-in | -64.81, -13.7 | -51.33, -43.39 | APE12-dist-na | 16.3984 | APE11-dist-na | 13.2123 | APE10-dist-na | 11.0908 | APE9-dist-in | 7.9513 | None | None | None | XRAY | 1.87 | 0.174 | 0.207 | A | 322.0 | 307.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6gqo | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 6GQPA | P35968 | 821 | 1168 | 1356.0 | F88:61201 | Type2 | Inactive | DFGout | 16.0412 | 9.8283 | BBAminus | -137.29, -179.39 | -147.6, 105.82 | -66.11, -30.27 | 279.44, 81.63 | 58.93, -133.79 | in-in | in | 7.7844 | Saltbr-in | 3.1604 | HRD-in | -72.29, -59.65 | 82.33, -13.78 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.7865 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -109.31, 108.64 | APE9-dihe-in | -119.08, 147.18 | APE8-dihe-in | -76.82, 68.93 | APE8-rot-na | 29.84 | APE67-dihe-in | -64.0, -17.44 | -48.7, -44.35 | APE12-dist-na | 16.2799 | APE11-dist-na | 13.0288 | APE10-dist-na | 10.463 | APE9-dist-out | 8.0203 | None | None | None | XRAY | 2.09 | 0.201 | 0.234 | A | 322.0 | 298.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6gqp | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 6GQQA | P35968 | 813 | 1167 | 1356.0 | F8B:61201 | Type2 | Inactive | DFGout | 16.3179 | 9.8934 | BBAminus | -140.35, 179.68 | -146.82, 105.0 | -62.58, -33.91 | 278.73, 81.84 | 52.08, -122.03 | in-in | in | 7.8551 | Saltbr-in | 2.8701 | HRD-in | -79.41, -58.06 | 81.99, -7.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.6419 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -102.87, 113.66 | APE9-dihe-in | -116.65, 151.24 | APE8-dihe-in | -82.45, 66.44 | APE8-rot-na | 31.58 | APE67-dihe-in | -64.76, -12.48 | -47.19, -45.1 | APE12-dist-na | 16.8675 | APE11-dist-na | 13.2075 | APE10-dist-na | 11.6327 | APE9-dist-out | 8.0466 | None | None | None | XRAY | 1.52 | 0.178 | 0.204 | A | 322.0 | 304.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6gqq | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 6XVJA | P35968 | 813 | 1167 | 1356.0 | O35:1201 | Type2 | Inactive | DFGout | 15.7966 | 9.8597 | BBAminus | -132.46, -168.17 | -160.35, 90.75 | -54.1, -41.9 | 283.85, 84.23 | 55.21, -117.78 | in-in | in | 7.7129 | Saltbr-in | 2.862 | HRD-in | -84.82, -59.51 | 82.99, -12.32 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.6823 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -99.56, 109.17 | APE9-dihe-in | -116.73, 149.21 | APE8-dihe-in | -78.94, 66.26 | APE8-rot-na | 30.73 | APE67-dihe-in | -62.92, -14.21 | -46.08, -45.25 | APE12-dist-na | 17.103 | APE11-dist-na | 13.5038 | APE10-dist-na | 11.3446 | APE9-dist-in | 7.9918 | E990V | None | None | XRAY | 1.78 | 0.18 | 0.215 | A | 322.0 | 305.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6xvj | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 6XVKA | P35968 | 821 | 1168 | 1356.0 | O3E:1201 | Type2 | Inactive | DFGout | 16.107 | 9.9746 | BBAminus | -141.36, -173.76 | -156.84, 95.12 | -54.67, -41.12 | 280.3, 80.99 | 54.89, -110.87 | in-in | in | 7.6818 | Saltbr-in | 2.8161 | HRD-in | -73.74, -55.3 | 80.84, -9.06 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.6059 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -105.81, 104.06 | APE9-dihe-in | -104.53, 149.15 | APE8-dihe-in | -78.71, 70.31 | APE8-rot-na | 29.7 | APE67-dihe-in | -63.75, -14.49 | -47.12, -46.79 | APE12-dist-na | 16.7775 | APE11-dist-na | 12.9611 | APE10-dist-na | 11.3811 | APE9-dist-in | 7.6764 | E990V | None | None | XRAY | 1.99 | 0.208 | 0.244 | A | 322.0 | 298.0 | 0 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 6xvk | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.4e-100 | 340.2 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 4ASDA | P35968 | 807 | 1168 | 1356.0 | BAX:1500 | Type2 | Inactive | DFGout | 15.5976 | 9.5654 | BBAminus | -143.46, -179.3 | -143.72, 107.55 | -61.84, -34.25 | 277.42, 87.13 | 55.65, -120.32 | in-in | in | 7.5842 | Saltbr-in | 2.9145 | HRD-in | -94.7, -57.23 | 78.86, -11.11 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5646 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.01, 114.08 | APE9-dihe-in | -124.4, 147.41 | APE8-dihe-in | -79.65, 63.41 | APE8-rot-na | 32.33 | APE67-dihe-in | -69.55, -12.31 | -53.55, -35.42 | APE12-dist-na | 16.0444 | APE11-dist-na | 13.4306 | APE10-dist-na | 11.4557 | APE9-dist-in | 7.9757 | E990V | None | None | XRAY | 2.03 | 0.178 | 0.23 | A | 353.0 | 305.0 | 7 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4asd | Homo sapiens | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 4ASEA | P35968 | 807 | 1169 | 1356.0 | AV9:3169 | Type2 | Inactive | DFGout | 15.5083 | 9.6214 | BBAminus | -131.22, 172.65 | -143.22, 109.66 | -69.47, -29.54 | 275.37, 90.83 | 50.61, -120.83 | in-in | in | 7.6836 | Saltbr-in | 3.0518 | HRD-in | -82.51, -52.61 | 76.99, -4.03 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4515 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.53, 119.23 | APE9-dihe-in | -120.88, 143.86 | APE8-dihe-in | -75.11, 65.17 | APE8-rot-na | 28.66 | APE67-dihe-in | -64.27, -9.66 | -54.44, -43.05 | APE12-dist-na | 16.1551 | APE11-dist-na | 13.7976 | APE10-dist-na | 11.6525 | APE9-dist-in | 7.9754 | E990V | None | None | XRAY | 1.83 | 0.207 | 0.231 | A | 353.0 | 307.0 | 6 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 4ase | Homo sapiens | TYR_KDR_HUMAN | TYR | 6e-100 | 339.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3VHEA | P35968 | 811 | 1169 | 1356.0 | 42Q:1170 | Type2 | Inactive | DFGout | 15.9847 | 10.209 | BBAminus | -150.75, 179.81 | -145.06, 104.72 | -59.59, -35.08 | 275.44, 63.4 | 53.57, -124.69 | in-in | in | 7.5456 | Saltbr-in | 2.811 | HRD-in | -83.47, -54.75 | 79.34, -6.09 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.7061 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -104.74, 113.79 | APE9-dihe-in | -123.79, 149.45 | APE8-dihe-in | -81.9, 62.59 | APE8-rot-na | 35.67 | APE67-dihe-in | -65.86, -15.29 | -45.47, -41.75 | APE12-dist-na | 999.0 | APE11-dist-na | 15.5547 | APE10-dist-na | 11.5571 | APE9-dist-out | 8.0431 | None | None | None | XRAY | 1.55 | 0.186 | 0.209 | A | 359.0 | 303.0 | 56 | 30 | 28 | 2 | [[834, 1162]] | 1.0 | 3vhe | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.4e-99 | 337.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3VHKA | P35968 | 814 | 1168 | 1356.0 | BPK:2001 | Type2 | Inactive | DFGout | 16.4972 | 9.9697 | BBAminus | -142.42, -168.12 | -154.13, 113.05 | -66.9, -34.19 | 279.52, 80.67 | 55.02, -115.26 | in-in | in | 7.7317 | Saltbr-in | 2.6852 | HRD-in | -85.63, -50.5 | 78.47, -9.06 | in-out-out | SNCioo | out-out | ActLoopNT-out | 16.6338 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -101.84, 113.0 | APE9-dihe-in | -119.22, 139.89 | APE8-dihe-in | -75.91, 70.12 | APE8-rot-na | 29.63 | APE67-dihe-in | -67.23, -15.54 | -56.62, -35.16 | APE12-dist-na | 999.0 | APE11-dist-na | 13.3761 | APE10-dist-na | 11.0032 | APE9-dist-out | 8.1076 | None | None | None | XRAY | 2.49 | 0.21 | 0.262 | A | 368.0 | 297.0 | 58 | 30 | 28 | 2 | [[834, 1162]] | 1.0 | 3vhk | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.6e-99 | 337.7 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2QU5A | P35968 | 816 | 1170 | 1356.0 | 276:501 | Type2 | Inactive | DFGout | 15.957 | 9.8302 | BBAminus | -148.46, -172.65 | -150.45, 108.8 | -78.65, -16.42 | 280.25, 86.88 | -99.11, -166.35 | in-in | in | 7.8737 | Saltbr-in | 2.7519 | HRD-in | -80.82, -52.31 | 94.02, -25.74 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -87.63, 5.51 | APE9-dihe-out | 37.61, 55.41 | APE8-dihe-out | -52.54, -22.13 | APE8-rot-na | 25.49 | APE67-dihe-in | -67.04, -17.69 | -59.89, -24.68 | APE12-dist-na | 10.2791 | APE11-dist-na | 14.2242 | APE10-dist-na | 11.1098 | APE9-dist-out | 11.3224 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.95 | 0.213 | 0.251 | A | 314.0 | 292.0 | 13 | 30 | 17 | 13 | [[834, 1162]] | 1.0 | 2qu5 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2QU6A | P35968 | 817 | 1171 | 1356.0 | 857:60501 | Type2 | Inactive | DFGout | 15.9424 | 9.8172 | BBAminus | -132.31, -170.97 | -155.67, 103.74 | -71.24, -21.04 | 287.6, 86.95 | -49.98, 999.0 | in-in | in | 7.8367 | Saltbr-in | 3.056 | HRD-in | -61.86, -49.75 | 81.1, -16.44 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 40.43 | APE8-rot-na | 31.68 | APE67-dihe-in | -68.37, -13.6 | -54.82, -35.61 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.1 | 0.242 | 0.272 | A | 314.0 | 276.0 | 29 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 2qu6 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2RL5A | P35968 | 815 | 1171 | 1356.0 | 2RL:60501 | Type2 | Inactive | DFGout | 15.3924 | 11.07 | BBAminus | -145.48, -175.23 | -148.97, 113.05 | -80.1, -11.01 | 289.69, 95.02 | 69.28, 57.0 | in-in | in | 7.8261 | Saltbr-in | 2.6984 | HRD-in | -65.08, -49.32 | 80.71, -16.94 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -86.71, -13.59 | APE9-dihe-out | 45.53, 52.75 | APE8-dihe-out | -54.88, -21.97 | APE8-rot-na | 32.05 | APE67-dihe-in | -73.02, -12.93 | -62.39, -23.08 | APE12-dist-na | 7.9303 | APE11-dist-na | 10.6315 | APE10-dist-na | 6.7426 | APE9-dist-out | 11.661 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.65 | 0.199 | 0.233 | A | 314.0 | 290.0 | 17 | 30 | 16 | 14 | [[834, 1162]] | 1.0 | 2rl5 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3B8QB | P35968 | 820 | 1166 | 1356.0 | 900:60502 | Type2 | Inactive | DFGout | 15.4044 | 10.0777 | BBAminus | -136.11, -171.43 | -160.46, 118.31 | -80.85, -45.83 | 290.91, 83.9 | 123.21, 999.0 | in-in | in | 7.8977 | Saltbr-in | 2.9027 | HRD-in | -68.36, -46.63 | 75.78, -5.88 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 155.56 | APE8-dihe-out | -60.35, -14.62 | APE8-rot-na | 30.93 | APE67-dihe-in | -68.62, -6.92 | -55.79, -32.87 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2967 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.75 | 0.218 | 0.276 | B | 314.0 | 271.0 | 26 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3b8q | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3BE2A | P35968 | 815 | 1171 | 1356.0 | RAJ:60501 | Type2 | Inactive | DFGout | 14.1127 | 11.0427 | BBAminus | -134.72, 177.84 | -152.38, 97.13 | -77.52, -8.1 | 302.77, 127.65 | 76.19, 999.0 | in-in | in | 7.941 | Saltbr-in | 2.7693 | HRD-in | -67.93, -53.26 | 79.3, -9.77 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 56.48 | APE8-rot-na | 341.32 | APE67-dihe-in | -65.72, -14.43 | -46.07, -42.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.75 | 0.197 | 0.226 | A | 314.0 | 285.0 | 22 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3be2 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CP9A | P35968 | 817 | 1171 | 1356.0 | C19:60501 | Type2 | Inactive | DFGout | 16.6202 | 10.2751 | BBAminus | -128.38, -176.57 | -155.05, 99.17 | -63.66, -9.88 | 278.68, 88.56 | -54.74, 999.0 | in-in | in | 7.7333 | Saltbr-in | 2.6364 | HRD-in | -61.14, -53.92 | 79.09, -9.79 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 101.57 | APE8-dihe-out | -50.34, -15.58 | APE8-rot-na | 28.54 | APE67-dihe-in | -69.67, -13.51 | -65.76, -26.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.5778 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.5 | 0.211 | 0.263 | A | 314.0 | 281.0 | 24 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3cp9 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CP9B | P35968 | 819 | 1165 | 1356.0 | C19:60502 | Type2 | Inactive | DFGout | 16.8412 | 10.4044 | BBAminus | -132.75, -171.12 | -162.18, 105.04 | -62.12, -28.88 | 281.99, 80.12 | 49.45, -86.0 | in-in | in | 7.6456 | Saltbr-in | 3.0483 | HRD-in | -88.31, -43.32 | 78.52, -15.92 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -57.69 | APE8-dihe-out | -39.24, -27.85 | APE8-rot-na | 24.86 | APE67-dihe-in | -68.9, -8.27 | -59.68, -31.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.4403 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.5 | 0.211 | 0.263 | B | 314.0 | 269.0 | 28 | 30 | 13 | 17 | [[834, 1162]] | 1.0 | 3cp9 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CPCB | P35968 | 820 | 1165 | 1356.0 | C52:60002 | Type2 | Inactive | DFGout | 16.6391 | 10.3787 | BBAminus | -131.82, -178.95 | -148.17, 107.11 | -69.23, -53.88 | 273.75, 87.39 | 111.77, 999.0 | in-in | in | 7.4849 | Saltbr-in | 2.706 | HRD-in | -75.42, -46.4 | 80.7, -16.54 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -53.89 | APE8-dihe-out | -53.45, -16.48 | APE8-rot-na | 17.35 | APE67-dihe-in | -69.92, -17.21 | -63.01, -26.25 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3843 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.221 | 0.272 | B | 314.0 | 262.0 | 34 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3cpc | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3DTWB | P35968 | 820 | 1166 | 1356.0 | A96:60502 | Type2 | Inactive | DFGout | 15.0355 | 10.1682 | BBAminus | -136.42, -166.86 | -159.08, 106.24 | -84.37, -81.02 | 295.18, 95.96 | 174.82, 139.27 | in-in | in | 8.1766 | Saltbr-in | 2.9571 | HRD-in | -66.59, -51.66 | 77.85, -16.94 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, 31.74 | APE9-dihe-out | -53.82, -56.19 | APE8-dihe-out | -45.11, -17.45 | APE8-rot-na | 28.36 | APE67-dihe-in | -71.35, -4.04 | -72.8, -21.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.2914 | APE9-dist-out | 11.5266 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.9 | 0.215 | 0.279 | B | 314.0 | 269.0 | 28 | 30 | 14 | 16 | [[834, 1162]] | 1.0 | 3dtw | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3EWHA | P35968 | 815 | 1171 | 1356.0 | K11:60001 | Type2 | Inactive | DFGout | 15.139 | 11.4202 | BBAminus | -133.49, -179.18 | -135.71, 102.66 | -69.48, -9.86 | 280.78, 102.57 | 67.93, 33.26 | in-in | in | 7.9373 | Saltbr-in | 3.0791 | HRD-in | -71.49, -51.89 | 78.14, -10.7 | in-out-none | SNCion | out-none | ActLoopNT-out | 12.9444 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 130.93 | APE8-dihe-in | -76.46, 69.83 | APE8-rot-na | 30.0 | APE67-dihe-in | -66.36, -17.49 | -56.88, -35.11 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.9722 | C817A,V916T,E990V | None | None | XRAY | 1.6 | 0.208 | 0.234 | A | 314.0 | 295.0 | 12 | 30 | 21 | 9 | [[834, 1162]] | 1.0 | 3ewh | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3U6JA | P35968 | 815 | 1171 | 1356.0 | 03X:60001 | Type2 | Inactive | DFGout | 14.9795 | 10.356 | BBAminus | -144.73, -178.41 | -146.44, 121.96 | -64.93, -27.75 | 282.37, 79.48 | 52.91, -122.32 | in-in | in | 7.455 | Saltbr-in | 2.8674 | HRD-in | -74.57, -56.02 | 80.88, -14.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.1328 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -99.27, 117.84 | APE9-dihe-in | -122.3, 141.03 | APE8-dihe-in | -77.42, 64.76 | APE8-rot-na | 30.56 | APE67-dihe-in | -69.06, -14.4 | -51.48, -37.1 | APE12-dist-na | 17.3677 | APE11-dist-na | 14.2143 | APE10-dist-na | 12.3875 | APE9-dist-in | 7.7332 | V916T,E990V | None | None | XRAY | 2.15 | 0.196 | 0.23 | A | 314.0 | 305.0 | 2 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 3u6j | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3C7QA | P35968 | 819 | 1171 | 1356.0 | XIN:1172 | Type1 | Inactive | DFGout | 15.7851 | 9.7942 | None | -118.96, 138.15 | -110.64, 113.79 | -73.47, 999.0 | 192.45, 128.99 | 999.0, 999.0 | in-in | in | 7.2832 | Saltbr-in | 2.6084 | HRD-in | -83.9, -48.68 | 82.47, -6.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -147.17, 145.76 | APE9-dihe-in | -104.98, 98.81 | APE8-dihe-out | -50.37, -26.53 | APE8-rot-na | 330.15 | APE67-dihe-in | -62.19, -10.0 | -56.65, -35.85 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.1746 | None | PTR1054,PTR1059 | CME862,CME1007,CME1024,PTR1054,PTR1059 | XRAY | 2.1 | 0.221 | 0.279 | A | 316.0 | 291.0 | 10 | 30 | 26 | 4 | [[834, 1162]] | 1.0 | 3c7q | Homo sapiens | TYR_KDR_HUMAN | TYR | 3.9e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2P2IB | P35968 | 820 | 1168 | 1356.0 | 608:60502 | Type1 | Inactive | DFGout | 16.2739 | 10.2035 | None | -141.39, -171.24 | -157.47, 119.0 | -85.08, 999.0 | 285.18, 81.66 | 999.0, 999.0 | in-in | in | 7.1432 | Saltbr-in | 3.2708 | HRD-in | -71.95, -45.89 | 71.89, -7.38 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 36.68 | APE8-rot-na | 31.31 | APE67-dihe-in | -54.41, -18.08 | -58.67, -41.73 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.222 | 0.266 | B | 314.0 | 263.0 | 36 | 30 | 10 | 20 | [[834, 1162]] | 1.0 | 2p2i | Homo sapiens | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3VNTA | P35968 | 812 | 1168 | 1356.0 | 0JA:2001 | Type2 | Inactive | DFGout | 16.7639 | 8.3863 | None | -132.49, -178.83 | -142.53, 104.52 | -68.92, -32.97 | 219.02, 49.93 | 58.07, -122.23 | in-in | in | 7.4677 | Saltbr-in | 2.7462 | HRD-in | -79.08, -51.8 | 75.79, -7.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5421 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.01, 111.64 | APE9-dihe-in | -121.89, 148.7 | APE8-dihe-in | -79.2, 68.13 | APE8-rot-na | 30.95 | APE67-dihe-in | -64.82, -12.79 | -56.01, -39.41 | APE12-dist-na | 16.8255 | APE11-dist-na | 13.4544 | APE10-dist-na | 11.2921 | APE9-dist-in | 7.8693 | None | None | None | XRAY | 1.64 | 0.153 | 0.192 | A | 318.0 | 301.0 | 6 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 3vnt | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.2e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3VO3A | P35968 | 812 | 1168 | 1356.0 | 0KF:2001 | Type2 | Inactive | DFGout | 16.4477 | 8.2146 | None | -125.16, 179.81 | -141.05, 99.79 | -70.03, -34.74 | 215.55, 55.41 | 59.77, -120.61 | in-in | in | 7.3573 | Saltbr-in | 2.8979 | HRD-in | -84.45, -53.71 | 76.95, -3.4 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4768 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.91, 109.54 | APE9-dihe-in | -120.7, 147.5 | APE8-dihe-in | -78.09, 65.8 | APE8-rot-na | 32.33 | APE67-dihe-in | -67.73, -12.3 | -53.4, -39.21 | APE12-dist-na | 17.0304 | APE11-dist-na | 14.0671 | APE10-dist-na | 11.3935 | APE9-dist-in | 7.9974 | None | None | None | XRAY | 1.52 | 0.162 | 0.182 | A | 318.0 | 303.0 | 4 | 30 | 30 | 0 | [[834, 1162]] | 1.0 | 3vo3 | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.2e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 2QU6B | P35968 | 822 | 1165 | 1356.0 | 857:60502 | Type2 | Inactive | DFGout | 15.9633 | 9.5409 | None | -133.96, -169.17 | -160.0, 100.56 | -72.82, 999.0 | 288.62, 90.71 | 999.0, 999.0 | in-in | in | 7.9527 | Saltbr-in | 3.0946 | HRD-in | -62.66, -51.11 | 76.69, -2.42 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 122.74 | APE8-dihe-in | -72.44, 73.71 | APE8-rot-na | 32.18 | APE67-dihe-in | -66.59, -17.43 | -56.47, -30.13 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.2922 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.1 | 0.242 | 0.272 | B | 314.0 | 260.0 | 34 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 2qu6 | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3B8QA | P35968 | 818 | 1171 | 1356.0 | 900:60501 | Type2 | Inactive | DFGout | 15.4672 | 9.913 | None | -131.74, -168.2 | -159.75, 118.5 | -86.72, 999.0 | 284.22, 100.5 | 999.0, 999.0 | in-in | in | 7.7591 | Saltbr-in | 2.7653 | HRD-in | -57.53, -50.67 | 79.88, -14.29 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 160.03 | APE8-dihe-out | -77.48, -12.97 | APE8-rot-na | 36.4 | APE67-dihe-in | -68.93, -8.62 | -57.21, -28.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.0722 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.75 | 0.218 | 0.276 | A | 314.0 | 285.0 | 19 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3b8q | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CPBA | P35968 | 819 | 1171 | 1356.0 | C92:60001 | Type2 | Inactive | DFGout | 15.3326 | 9.7507 | None | -143.96, -172.89 | -147.19, 119.38 | -89.94, 999.0 | 278.49, 101.53 | 999.0, 999.0 | in-in | in | 7.7633 | Saltbr-in | 3.5846 | HRD-in | -60.85, -44.16 | 62.59, 3.77 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 128.93 | APE8-dihe-out | -45.12, -28.83 | APE8-rot-na | 328.95 | APE67-dihe-in | -65.36, -7.17 | -53.29, -33.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.351 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.7 | 0.224 | 0.286 | A | 314.0 | 278.0 | 25 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3cpb | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CPCA | P35968 | 820 | 1171 | 1356.0 | C52:60001 | Type2 | Inactive | DFGout | 16.8028 | 10.3818 | None | -127.27, -176.88 | -144.84, 92.18 | -66.45, 999.0 | 268.44, 99.63 | 999.0, 999.0 | in-out | in | 8.0268 | Saltbr-out | 3.9767 | HRD-in | -74.56, -44.56 | 79.03, -21.68 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.84 | APE8-dihe-out | -45.97, -30.08 | APE8-rot-na | 328.28 | APE67-dihe-in | -73.13, -9.14 | -56.02, -29.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3564 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.4 | 0.221 | 0.272 | A | 314.0 | 277.0 | 25 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3cpc | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3DTWA | P35968 | 818 | 1171 | 1356.0 | A96:60501 | Type2 | Inactive | DFGout | 15.1581 | 10.0994 | None | -129.54, -170.94 | -153.49, 103.32 | -82.68, 999.0 | 294.21, 96.03 | 999.0, 999.0 | in-in | in | 8.0061 | Saltbr-in | 2.6405 | HRD-in | -53.04, -53.77 | 79.82, -12.25 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.1 | APE8-dihe-out | -46.34, -20.16 | APE8-rot-na | 23.94 | APE67-dihe-in | -60.71, -7.92 | -57.08, -38.78 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2341 | C817A,V916T,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.9 | 0.215 | 0.279 | A | 314.0 | 281.0 | 23 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3dtw | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.8e-100 | 340.9 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3CJFA | P35968 | 817 | 1168 | 1356.0 | SAV:61167 | Type1 | Inactive | None | 999.0 | 999.0 | None | -83.44, 111.78 | -118.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-out | in | 7.8208 | Saltbr-out | 5.2231 | HRD-out | -105.6, 121.11 | -71.37, -10.71 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.8895 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 48.59 | APE8-rot-na | 25.36 | APE67-dihe-in | -69.88, -14.36 | -60.34, -37.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | CSO862,CSO1007,CSO1024,CSO1045,CSO1116 | XRAY | 2.15 | 0.205 | 0.258 | A | 309.0 | 281.0 | 17 | 30 | 16 | 14 | [[834, 1162]] | 1.0 | 3cjf | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.8e-100 | 340.1 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 1YWNA | P35968 | 820 | 1171 | 1356.0 | LIF:60301 | Type1 | Inactive | None | 999.0 | 999.0 | None | -128.91, 171.96 | -143.62, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 7.2102 | Saltbr-in | 2.725 | HRD-in | -77.88, -50.07 | 82.87, -17.6 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -141.39, 161.44 | APE9-dihe-in | -104.18, 100.32 | APE8-dihe-out | -56.09, -24.71 | APE8-rot-na | 336.02 | APE67-dihe-in | -70.59, -14.0 | -51.58, -32.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2392 | E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 1.71 | 0.206 | 0.23 | A | 316.0 | 281.0 | 21 | 30 | 24 | 6 | [[834, 1162]] | 1.0 | 1ywn | Homo sapiens | TYR_KDR_HUMAN | TYR | 4.1e-100 | 340.3 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| KDR | VGFR2_HUMAN | 3VIDA | P35968 | 813 | 1168 | 1356.0 | 4TT:2001 | Type1 | Inactive | None | 999.0 | 999.0 | None | -128.64, 167.68 | -132.79, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 7.3263 | Saltbr-in | 2.9803 | HRD-in | -77.53, -50.55 | 79.3, -13.28 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -152.12, 159.09 | APE9-dihe-in | -96.12, 109.5 | APE8-dihe-out | -66.36, -14.96 | APE8-rot-na | 337.32 | APE67-dihe-in | -69.61, -3.71 | -60.46, -30.42 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3777 | None | None | None | XRAY | 2.3 | 0.247 | 0.281 | A | 356.0 | 299.0 | 57 | 30 | 23 | 7 | [[834, 1162]] | 1.0 | 3vid | Homo sapiens | TYR_KDR_HUMAN | TYR | 2.3e-99 | 337.8 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|