AGC_GRK1 (Rhodopsin kinase GRK1)

Total number of chains: 2
Active chains: 2
Uniprot: GRK1_HUMAN
Kinase Domain Residues: 190 - 455
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 2 100.0% AF-Q15835-K1A

Download database table as tsv Go to Advanced Page
PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
AF-Q15835-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 182 - 463 0 None None Rhodopsin kinase GRK1
AF-Q15835-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 182 - 463 0 None None Rhodopsin kinase GRK1

AGC_GRK1 (Rhodopsin kinase GRK1)

Total number of chains: 29
Active chains: 19
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 28 96.6% AF-Q15835-K1A
DFGinter None 1 3.4% 3C4YB

Download database table as tsv Go to Advanced Page
UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
GRK1_BOVIN 3T8OA 2.5 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 30 - 532 0 None L166K Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4WA 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 31 - 533 0 TPO8 None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4WB 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 5 - 533 0 TPO8 None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4XA 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4XB 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4ZA 1.84 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C50A 2.6 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C50B 2.6 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C51A 3.55 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C51B 3.55 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9A 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9B 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9C 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9D 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4L9IB 2.32 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 8PR Type1 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4PNIA 1.85 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii KQQ Type1 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MTBG 4.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None S5E,S488E,T489E Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4YA 7.509 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 30 - 532 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4L9IA 2.32 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii 8PR Type1 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOA 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 28 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOB 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOC 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 31 - 531 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOD 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 30 - 531 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MT9G 7.0 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iiio SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MT8G 5.8 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_iiii SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None S5E,S488E,T489E Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MTAG 4.1 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None S5E,S488E,T489E Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4YB 7.509 Inactive DFGinter‑None in-out in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 30 - 532 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_HUMAN AF-Q15835-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 182 - 463 0 None None Rhodopsin kinase GRK1 Homo sapiens
GRK1_HUMAN AF-Q15835-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 182 - 463 0 None None Rhodopsin kinase GRK1 Homo sapiens

AGC_GRK1 (Rhodopsin kinase GRK1)

Total number of chains: 27
Active chains: 17
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 26 96.3% 3C4ZA
DFGinter None 1 3.7% 3C4YB

Download database table as tsv Go to Advanced Page
UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
GRK1_BOVIN 3T8OA 2.5 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 30 - 532 0 None L166K Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4WA 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 31 - 533 0 TPO8 None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4WB 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 5 - 533 0 TPO8 None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4XA 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4XB 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ATP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4ZA 1.84 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C50A 2.6 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C50B 2.6 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C51A 3.55 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C51B 3.55 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9A 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9B 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9C 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3QC9D 2.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ADP ATPlike 31 - 533 0 None T8C,N480C Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4L9IB 2.32 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 8PR Type1 31 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4PNIA 1.85 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii KQQ Type1 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MTBG 4.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None S5E,S488E,T489E Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4YA 7.509 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 30 - 532 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4L9IA 2.32 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii 8PR Type1 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOA 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 28 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOB 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 30 - 533 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOC 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 31 - 531 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 4WBOD 2.81 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ANW Type1 30 - 531 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MT9G 7.0 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iiio SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None None Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MT8G 5.8 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaioi APEdist_iiii SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None S5E,S488E,T489E Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 7MTAG 4.1 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii SGV, SGV, SGV, SGV, SGV, SGV Type1, Type1, Type1, Type1, Type1, Type1 6 - 508 0 None S5E,S488E,T489E Rhodopsin kinase GRK1 Bos taurus
GRK1_BOVIN 3C4YB 7.509 Inactive DFGinter‑None in-out in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 30 - 532 0 None None Rhodopsin kinase GRK1 Bos taurus