AGC_GRK1 (Rhodopsin kinase GRK1)

Total number of chains: 2
Active chains: 2
Uniprot: GRK1_HUMAN
Kinase Domain Residues: 190 - 455
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 2 100.0% AF-Q15835-K1A

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GRK1 AF-Q15835-K1A Q15835 182 463 563.0 No_ligand No_ligand Active DFGin 6.2866 12.9823 BLAminus -136.35, -175.46 50.41, 68.56 -84.63, 18.73 288.09, 153.13 -66.15, -19.38 in-in in 8.5389 Saltbr-in 2.6976 HRD-in -79.0, -46.45 64.22, 3.54 in-in-in SNCiii in-in ActLoopNT-in 2.8485 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.64, 146.23 APE9-dihe-na 128.56, 178.92 APE8-dihe-in -91.42, 131.88 APE8-rot-in 297.69 APE67-dihe-inflip 105.02, -24.11 -55.02, 126.46 APE12-dist-in 10.6028 APE11-dist-in 11.2776 APE10-dist-in 5.5393 APE9-dist-in 3.3156 None None None AF2 -1.0 1.0 1.0 A 282.0 282.0 0 28 28 0 [[190, 455]] 1.0 AF-Q15835-K1 AGC_GRK1_HUMAN AGC 4.7e-81 277.6 4.0 260.0 257.0 334 335 336 338 340 219 238 242 314 316 315 317.0 374 362 357 356 355 354 353 352 351 268 Rhodopsin kinase GRK1
GRK1 AF-Q15835-K3A Q15835 182 463 563.0 No_ligand No_ligand Active DFGin 6.2345 12.6731 BLAminus -132.6, -178.51 49.86, 63.45 -76.42, 16.89 298.82, 166.43 -67.25, -17.86 in-in in 8.359 Saltbr-in 2.7065 HRD-in -85.57, -47.78 70.01, -0.82 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.92, 145.73 APE9-dihe-na 125.2, -163.99 APE8-dihe-in -109.07, 130.14 APE8-rot-in 295.51 APE67-dihe-inflip 103.48, -23.56 -54.31, 127.87 APE12-dist-in 10.5262 APE11-dist-in 11.024 APE10-dist-in 5.3332 APE9-dist-in 3.0336 None None None AF2 -1.0 1.0 1.0 A 282.0 282.0 0 28 28 0 [[190, 455]] 1.0 AF-Q15835-K3 AGC_GRK1_HUMAN AGC 4.7e-81 277.6 4.0 260.0 257.0 334 335 336 338 340 219 238 242 314 316 315 317.0 374 362 357 356 355 354 353 352 351 268 Rhodopsin kinase GRK1

AGC_GRK1 (Rhodopsin kinase GRK1)

Total number of chains: 29
Active chains: 19
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 28 96.6% AF-Q15835-K1A
DFGinter None 1 3.4% 3C4YB

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GRK1 GRK1_BOVIN 3T8OA P28327 30 532 561.0 ATP:562 ATPlike Active DFGin 6.784 13.6519 BLAminus -147.61, 176.5 66.51, 86.5 -106.39, 20.07 278.45, 121.96 -78.51, -8.51 in-in in 9.1312 Saltbr-in 2.9462 HRD-in -72.08, -59.57 74.93, 15.13 in-in-in SNCiii in-in ActLoopNT-in 3.0341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.6, 145.4 APE9-dihe-na 140.82, -165.62 APE8-dihe-in -114.33, 123.31 APE8-rot-in 302.45 APE67-dihe-inflip 90.49, -9.25 -48.36, 136.06 APE12-dist-in 10.4193 APE11-dist-in 11.6453 APE10-dist-in 5.7954 APE9-dist-in 4.2758 L166K None None XRAY 2.5 0.209 0.245 A 543.0 493.0 0 28 28 0 [[187, 452]] 1.0 3t8o Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4WA P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 6.5874 13.3137 BLAminus -157.51, 175.0 67.79, 80.23 -106.97, 21.1 277.77, 138.55 -72.95, -18.52 in-in in 8.6705 Saltbr-in 2.6589 HRD-in -67.86, -51.97 60.46, 12.85 in-in-in SNCiii in-in ActLoopNT-in 2.8974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.73, 153.77 APE9-dihe-na 125.45, -175.95 APE8-dihe-in -101.44, 127.92 APE8-rot-in 301.93 APE67-dihe-inflip 97.46, -21.92 -46.81, 133.28 APE12-dist-in 10.0067 APE11-dist-in 11.2485 APE10-dist-in 5.5344 APE9-dist-in 3.5083 None TPO8 TPO8 XRAY 2.7 0.192 999.0 A 543.0 494.0 0 28 28 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4WB P28327 5 533 561.0 ATP:562 ATPlike Active DFGin 5.9629 13.1113 BLAminus -155.04, 178.49 64.64, 79.84 -103.28, 19.03 277.57, 109.21 -72.3, -19.68 in-in in 8.548 Saltbr-in 2.84 HRD-in -67.79, -54.67 64.69, 11.83 in-in-in SNCiii in-in ActLoopNT-in 2.9583 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.45, 154.48 APE9-dihe-na 126.08, -175.35 APE8-dihe-in -101.18, 126.91 APE8-rot-in 300.91 APE67-dihe-inflip 94.23, -17.08 -47.18, 130.86 APE12-dist-in 10.1029 APE11-dist-in 11.2538 APE10-dist-in 5.5445 APE9-dist-in 3.5342 None TPO8 TPO8 XRAY 2.7 0.192 999.0 B 543.0 519.0 0 28 28 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4XA P28327 30 533 561.0 ATP:562 ATPlike Active DFGin 6.3918 13.2944 BLAminus -153.36, -178.73 56.38, 83.66 -101.23, 19.01 282.86, 141.85 -58.01, -33.04 in-in in 8.6227 Saltbr-in 2.8246 HRD-in -65.41, -52.58 62.44, 13.36 in-in-in SNCiii in-in ActLoopNT-in 2.9597 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.48, 144.22 APE9-dihe-na 128.55, -174.69 APE8-dihe-in -103.7, 129.98 APE8-rot-in 314.1 APE67-dihe-inflip 101.04, -22.84 -50.28, 132.61 APE12-dist-in 10.283 APE11-dist-in 11.2374 APE10-dist-in 5.7264 APE9-dist-in 3.8266 None None None XRAY 2.9 0.193 999.0 A 543.0 496.0 0 28 28 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4XB P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 5.9031 13.063 BLAminus -149.62, 174.69 57.3, 76.73 -95.24, 8.98 282.05, 96.12 -51.11, -35.54 in-in in 8.6415 Saltbr-in 2.6755 HRD-in -62.32, -48.48 63.55, 4.44 in-in-in SNCiii in-in ActLoopNT-in 3.0432 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.42, 143.72 APE9-dihe-na 129.46, -175.16 APE8-dihe-in -98.28, 125.3 APE8-rot-in 312.69 APE67-dihe-inflip 98.15, -18.1 -45.11, 129.51 APE12-dist-in 10.2012 APE11-dist-in 11.2468 APE10-dist-in 5.6099 APE9-dist-in 3.6392 None None None XRAY 2.9 0.193 999.0 B 543.0 475.0 0 28 28 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4ZA P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.9128 13.2351 BLAminus -149.46, 171.26 70.91, 78.39 -108.02, 16.47 270.55, 111.24 -69.43, -16.01 in-in in 8.7363 Saltbr-in 2.7164 HRD-in -71.08, -53.07 69.31, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.8781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.53, 147.45 APE9-dihe-na 134.96, -165.72 APE8-dihe-in -111.39, 128.56 APE8-rot-in 296.58 APE67-dihe-inflip 96.79, -17.75 -54.96, 131.39 APE12-dist-in 10.4298 APE11-dist-in 11.1131 APE10-dist-in 5.4905 APE9-dist-in 3.5422 None None None XRAY 1.84 0.193 999.0 A 543.0 493.0 0 28 28 0 [[187, 452]] 1.0 3c4z Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C50A P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.0752 13.0339 BLAminus -142.59, 172.43 68.85, 78.38 -104.12, 14.36 280.99, 104.76 -67.57, -15.07 in-in in 8.6024 Saltbr-in 2.9252 HRD-in -76.21, -52.36 64.46, 15.62 in-in-in SNCiii in-in ActLoopNT-in 2.7949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.66, 144.27 APE9-dihe-na 130.37, -165.26 APE8-dihe-in -104.68, 131.22 APE8-rot-in 300.48 APE67-dihe-inflip 92.29, -6.18 -56.88, 135.03 APE12-dist-in 10.685 APE11-dist-in 11.4689 APE10-dist-in 5.8763 APE9-dist-in 3.4729 None None None XRAY 2.6 0.19 999.0 A 543.0 499.0 0 28 28 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C50B P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.0782 13.0677 BLAminus -140.52, 175.4 66.53, 77.05 -104.14, 18.55 279.39, 103.87 -67.23, -21.39 in-in in 8.5322 Saltbr-in 2.7211 HRD-in -71.74, -52.34 63.89, 11.32 in-in-in SNCiii in-in ActLoopNT-in 2.8901 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.47, 143.37 APE9-dihe-na 137.53, -168.17 APE8-dihe-in -105.39, 125.32 APE8-rot-in 297.12 APE67-dihe-inflip 95.82, -17.57 -51.32, 135.4 APE12-dist-in 10.1294 APE11-dist-in 11.1147 APE10-dist-in 5.5383 APE9-dist-in 3.4184 None None None XRAY 2.6 0.19 999.0 B 543.0 496.0 0 28 28 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C51A P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.7354 13.2354 BLAminus -156.28, 178.74 57.85, 73.51 -84.14, -2.01 283.03, 106.57 -47.35, -22.99 in-in in 8.7977 Saltbr-in 2.6866 HRD-in -64.41, -45.82 69.5, -19.46 in-in-in SNCiii in-in ActLoopNT-in 2.9155 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.64, 142.5 APE9-dihe-na 155.52, -169.52 APE8-dihe-in -101.5, 135.25 APE8-rot-in 300.99 APE67-dihe-inflip 84.91, 4.53 -59.96, 128.0 APE12-dist-in 10.573 APE11-dist-in 11.5413 APE10-dist-in 6.1515 APE9-dist-in 3.937 None None None XRAY 3.55 0.281 999.0 A 543.0 487.0 0 28 28 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C51B P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.7851 13.1869 BLAminus -156.29, 175.57 58.57, 74.43 -85.29, -1.69 285.99, 107.07 -47.38, -22.91 in-in in 8.696 Saltbr-in 2.7915 HRD-in -66.67, -42.5 63.68, -15.39 in-in-in SNCiii in-in ActLoopNT-in 2.9686 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.05, 141.93 APE9-dihe-na 155.26, -171.96 APE8-dihe-in -101.33, 138.35 APE8-rot-in 299.85 APE67-dihe-inflip 84.6, 5.24 -64.39, 128.67 APE12-dist-in 10.5371 APE11-dist-in 11.5977 APE10-dist-in 6.1564 APE9-dist-in 3.9396 None None None XRAY 3.55 0.281 999.0 B 543.0 461.0 20 28 28 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9A P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.8516 13.4841 BLAminus -151.04, 174.48 70.22, 99.25 -129.57, 18.73 275.22, 99.19 -61.63, -18.96 in-in in 8.9606 Saltbr-in 3.1273 HRD-in -61.98, -58.15 73.37, -3.42 in-in-in SNCiii in-in ActLoopNT-in 2.9166 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.32, 133.82 APE9-dihe-na 142.48, -169.15 APE8-dihe-in -104.33, 125.71 APE8-rot-in 302.67 APE67-dihe-inflip 104.42, -3.83 -50.74, 122.55 APE12-dist-in 10.3557 APE11-dist-in 11.0144 APE10-dist-in 5.5004 APE9-dist-in 3.6645 T8C,N480C None None XRAY 2.7 0.194 0.229 A 543.0 486.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9B P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.8991 13.5043 BLAminus -154.17, 173.67 70.5, 100.81 -132.54, 18.75 276.87, 97.69 -56.57, -24.02 in-in in 8.931 Saltbr-in 3.099 HRD-in -65.24, -58.34 73.4, -2.88 in-in-in SNCiii in-in ActLoopNT-in 2.9339 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -166.53, 132.45 APE9-dihe-na 145.72, -169.79 APE8-dihe-in -103.09, 126.5 APE8-rot-in 303.38 APE67-dihe-inflip 99.94, -4.73 -52.12, 123.93 APE12-dist-in 10.3676 APE11-dist-in 11.0383 APE10-dist-in 5.525 APE9-dist-in 3.6772 T8C,N480C None None XRAY 2.7 0.194 0.229 B 543.0 481.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9C P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.8677 13.481 BLAminus -151.87, 172.48 72.03, 98.62 -128.19, 19.72 276.34, 98.38 -59.47, -19.79 in-in in 8.9508 Saltbr-in 3.1074 HRD-in -62.09, -58.44 72.04, -1.68 in-in-in SNCiii in-in ActLoopNT-in 2.9357 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.26, 134.05 APE9-dihe-na 142.83, -170.11 APE8-dihe-in -104.04, 126.58 APE8-rot-in 301.36 APE67-dihe-inflip 105.14, -2.81 -49.9, 120.73 APE12-dist-in 10.3838 APE11-dist-in 11.0185 APE10-dist-in 5.5081 APE9-dist-in 3.673 T8C,N480C None None XRAY 2.7 0.194 0.229 C 543.0 482.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9D P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.9233 13.5167 BLAminus -151.29, 174.11 71.25, 99.27 -130.54, 20.81 276.77, 98.72 -58.99, -24.3 in-in in 8.9307 Saltbr-in 3.0905 HRD-in -63.44, -57.63 71.87, -0.43 in-in-in SNCiii in-in ActLoopNT-in 2.9269 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.95, 134.69 APE9-dihe-na 141.2, -168.54 APE8-dihe-in -103.28, 126.55 APE8-rot-in 303.76 APE67-dihe-inflip 102.49, -2.5 -51.29, 121.62 APE12-dist-in 10.3966 APE11-dist-in 11.0439 APE10-dist-in 5.5135 APE9-dist-in 3.693 T8C,N480C None None XRAY 2.7 0.194 0.229 D 543.0 486.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4L9IB P28327 31 533 561.0 8PR:601 Type1 Active DFGin 5.7147 13.0643 BLAminus -147.41, -179.95 59.09, 74.76 -90.68, 22.77 285.65, 103.28 -76.71, -12.5 in-in in 8.7578 Saltbr-in 3.1172 HRD-in -77.55, -56.18 71.16, 4.39 in-in-in SNCiii in-in ActLoopNT-in 2.7658 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.45, 143.07 APE9-dihe-na 140.89, -160.87 APE8-dihe-in -115.15, 127.72 APE8-rot-in 297.19 APE67-dihe-inflip 102.74, -33.6 -52.94, 132.06 APE12-dist-in 10.2921 APE11-dist-in 11.2208 APE10-dist-in 5.6416 APE9-dist-in 3.766 None None None XRAY 2.32 0.188 0.231 B 504.0 493.0 0 28 28 0 [[187, 452]] 1.0 4l9i Bos taurus AGC_GRK1_BOVIN AGC 2.5e-80 275.4 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4PNIA P28327 30 533 561.0 KQQ:601 Type1 Active DFGin 5.7355 13.1277 BLAminus -134.98, -179.15 54.91, 73.26 -92.23, 19.47 279.07, 113.0 -67.01, -18.73 in-in in 9.6807 Saltbr-in 3.1063 HRD-in -69.25, -51.31 65.76, 4.71 in-in-in SNCiii in-in ActLoopNT-in 2.9934 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.87, 143.44 APE9-dihe-na 144.11, -165.57 APE8-dihe-in -117.94, 131.85 APE8-rot-in 290.67 APE67-dihe-inflip 103.74, -23.28 -58.63, 131.5 APE12-dist-in 10.3397 APE11-dist-in 11.3538 APE10-dist-in 5.7216 APE9-dist-in 3.6813 None None None XRAY 1.85 0.191 0.23 A 561.0 492.0 0 28 28 0 [[187, 452]] 1.0 4pni Bos taurus AGC_GRK1_BOVIN AGC 3.3e-80 275.0 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MTBG P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Active DFGin 5.4472 13.977 BLAminus -158.7, 161.68 75.49, 110.48 -135.3, 45.5 298.35, 172.26 -102.18, -14.04 in-in in 8.1835 Saltbr-in 3.2327 HRD-in -84.4, -44.53 73.27, 9.15 in-in-in SNCiii in-in ActLoopNT-in 3.0388 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -63.06, 150.99 APE9-dihe-na 114.44, 173.54 APE8-dihe-in -100.2, 123.65 APE8-rot-in 303.1 APE67-dihe-inflip 95.63, -25.77 -41.47, 136.01 APE12-dist-in 10.1039 APE11-dist-in 10.473 APE10-dist-in 4.8138 APE9-dist-in 3.2162 S5E,S488E,T489E None None EM 4.0 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mtb Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4YA P28327 30 532 561.0 No_ligand No_ligand Inactive DFGin 7.6904 11.3511 BLAminus -137.44, 168.27 58.91, 104.81 -126.41, 38.75 308.65, 132.27 -61.68, -52.44 in-out in 9.8329 Saltbr-out 4.3893 HRD-in -106.52, -35.17 66.74, -61.42 out-in-in SNCoii in-in ActLoopNT-in 3.2444 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -178.5, 156.22 APE9-dihe-na 145.3, -132.92 APE8-dihe-in -136.09, 120.97 APE8-rot-in 304.15 APE67-dihe-inflip 122.03, -39.54 -49.39, 107.36 APE12-dist-in 11.4228 APE11-dist-in 12.6652 APE10-dist-in 7.6409 APE9-dist-in 5.7505 None None None XRAY 7.509 0.182 999.0 A 543.0 478.0 2 28 28 0 [[187, 452]] 1.0 3c4y Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4L9IA P28327 30 533 561.0 8PR:601 Type1 Inactive DFGin 5.7724 13.4538 BLAminus -149.91, 178.73 54.74, 79.81 -98.99, 23.91 282.53, 102.36 -68.07, -19.68 in-out in 8.693 Saltbr-out 3.808 HRD-in -75.83, -53.93 68.31, 13.36 out-in-in SNCoii in-in ActLoopNT-in 2.8273 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.8, 142.88 APE9-dihe-na 125.17, -158.26 APE8-dihe-in -112.07, 133.06 APE8-rot-in 301.6 APE67-dihe-inflip 94.99, -2.22 -45.66, 120.79 APE12-dist-in 10.6157 APE11-dist-in 11.3826 APE10-dist-in 5.8078 APE9-dist-in 3.7234 None None None XRAY 2.32 0.188 0.231 A 504.0 504.0 0 28 28 0 [[187, 452]] 1.0 4l9i Bos taurus AGC_GRK1_BOVIN AGC 2.5e-80 275.4 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOA P28327 28 533 561.0 ANW:601 Type1 Inactive DFGin 5.9481 13.2578 BLAminus -146.44, 170.56 64.48, 78.76 -93.1, 25.97 287.19, 103.23 -64.53, -31.02 in-out in 9.4403 Saltbr-out 4.1695 HRD-in -74.57, -52.51 66.08, 11.01 out-in-in SNCoii in-in ActLoopNT-in 2.8138 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.31, 145.0 APE9-dihe-na 138.11, -171.62 APE8-dihe-in -107.94, 132.02 APE8-rot-in 308.16 APE67-dihe-inflip 100.64, -17.52 -51.85, 128.49 APE12-dist-in 10.2576 APE11-dist-in 11.1305 APE10-dist-in 5.5198 APE9-dist-in 3.5303 None None None XRAY 2.81 0.243 0.267 A 541.0 497.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOB P28327 30 533 561.0 ANW:601 Type1 Inactive DFGin 5.9542 13.2886 BLAminus -146.62, 171.17 63.95, 77.64 -91.91, 26.29 286.92, 103.21 -63.89, -32.19 in-out in 9.5168 Saltbr-out 4.1969 HRD-in -74.66, -52.71 66.21, 10.61 out-in-in SNCoii in-in ActLoopNT-in 2.8113 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.36, 145.07 APE9-dihe-na 138.91, -171.46 APE8-dihe-in -107.75, 132.29 APE8-rot-in 308.55 APE67-dihe-inflip 100.74, -17.56 -52.36, 128.88 APE12-dist-in 10.2543 APE11-dist-in 11.1301 APE10-dist-in 5.5133 APE9-dist-in 3.5248 None None None XRAY 2.81 0.243 0.267 B 541.0 495.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOC P28327 31 531 561.0 ANW:601 Type1 Inactive DFGin 5.9556 13.1632 BLAminus -146.21, 170.22 64.35, 78.08 -92.41, 26.2 287.47, 102.96 -63.87, -32.11 in-out in 9.3966 Saltbr-out 3.7689 HRD-in -74.89, -52.54 66.21, 10.58 out-in-in SNCoii in-in ActLoopNT-in 2.8069 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.19, 145.1 APE9-dihe-na 138.92, -171.47 APE8-dihe-in -107.47, 132.18 APE8-rot-in 308.34 APE67-dihe-inflip 100.67, -17.42 -51.93, 128.63 APE12-dist-in 10.2519 APE11-dist-in 11.1292 APE10-dist-in 5.5118 APE9-dist-in 3.5259 None None None XRAY 2.81 0.243 0.267 C 541.0 481.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOD P28327 30 531 561.0 ANW:601 Type1 Inactive DFGin 5.9637 13.2454 BLAminus -146.28, 170.52 64.39, 78.16 -92.93, 26.26 287.26, 103.4 -64.25, -31.88 in-out in 9.4433 Saltbr-out 4.1679 HRD-in -74.7, -52.76 66.23, 10.86 out-in-in SNCoii in-in ActLoopNT-in 2.8047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.01, 145.2 APE9-dihe-na 138.57, -171.52 APE8-dihe-in -107.49, 131.96 APE8-rot-in 308.49 APE67-dihe-inflip 100.73, -17.59 -51.76, 128.57 APE12-dist-in 10.2771 APE11-dist-in 11.157 APE10-dist-in 5.5301 APE9-dist-in 3.529 None None None XRAY 2.81 0.243 0.267 D 541.0 491.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MT9G P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Inactive DFGin 5.6744 13.0596 BLAminus -151.44, 153.5 75.1, 83.16 -101.64, 23.22 308.74, 9.79 -95.55, -5.25 in-out in 8.3758 Saltbr-out 3.7806 HRD-out -84.42, -25.78 58.78, -116.78 out-in-out SNCoio in-out ActLoopNT-in 2.9966 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iiio APE10-dihe-na -156.18, 168.76 APE9-dihe-na 65.79, -175.16 APE8-dihe-in -118.77, 133.16 APE8-rot-in 303.35 APE67-dihe-inflip 85.9, 7.81 -39.32, 131.4 APE12-dist-in 12.4268 APE11-dist-in 12.0285 APE10-dist-in 6.4797 APE9-dist-out 6.7808 None None None EM 7.0 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mt9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MT8G P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Inactive DFGin 5.2778 13.8515 BLAminus -151.24, 148.8 73.0, 121.86 -132.91, 52.67 297.42, 171.65 -103.81, -13.33 in-in in 8.7716 Saltbr-in 3.2791 HRD-in -93.25, -20.41 75.09, -77.24 in-in-out SNCiio in-out ActLoopNT-in 3.0353 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.01, 152.4 APE9-dihe-na 69.43, 177.13 APE8-dihe-in -91.35, 141.08 APE8-rot-out 53.33 APE67-dihe-inflip 95.78, 14.3 -52.12, 148.5 APE12-dist-in 10.7091 APE11-dist-in 10.3507 APE10-dist-in 4.9503 APE9-dist-in 3.4095 S5E,S488E,T489E None None EM 5.8 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mt8 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MTAG P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Inactive DFGin 4.0904 13.8437 BLAminus -167.88, 170.04 60.34, 64.21 -82.37, 97.38 303.24, 179.85 -89.6, -128.64 in-out in 8.6589 Saltbr-out 5.1993 HRD-in -95.2, -46.79 83.22, -60.37 out-in-in SNCoii in-in ActLoopNT-in 3.0912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.79, 133.35 APE9-dihe-na 142.18, 170.18 APE8-dihe-in -78.99, 123.97 APE8-rot-in 304.47 APE67-dihe-inflip 89.96, 4.75 -51.0, 134.99 APE12-dist-in 11.1037 APE11-dist-in 11.0248 APE10-dist-in 5.5893 APE9-dist-in 3.7938 S5E,S488E,T489E None None EM 4.1 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mta Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4YB P28327 30 532 561.0 No_ligand No_ligand Inactive DFGinter 8.0405 10.5531 None -138.64, 168.89 59.27, 104.12 -125.95, 37.77 308.57, 133.4 -61.52, -52.16 in-out in 9.8319 Saltbr-out 4.4166 HRD-in -105.99, -36.37 67.54, -61.73 out-in-in SNCoii in-in ActLoopNT-in 3.2059 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -178.33, 157.76 APE9-dihe-na 144.04, -133.41 APE8-dihe-in -135.26, 121.19 APE8-rot-in 303.52 APE67-dihe-inflip 122.3, -40.41 -49.79, 107.51 APE12-dist-in 11.4257 APE11-dist-in 12.6565 APE10-dist-in 7.6316 APE9-dist-in 5.7888 None None None XRAY 7.509 0.182 999.0 B 543.0 466.0 8 28 28 0 [[187, 452]] 1.0 3c4y Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_HUMAN AF-Q15835-K1A Q15835 182 463 563.0 No_ligand No_ligand Active DFGin 6.2866 12.9823 BLAminus -136.35, -175.46 50.41, 68.56 -84.63, 18.73 288.09, 153.13 -66.15, -19.38 in-in in 8.5389 Saltbr-in 2.6976 HRD-in -79.0, -46.45 64.22, 3.54 in-in-in SNCiii in-in ActLoopNT-in 2.8485 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.64, 146.23 APE9-dihe-na 128.56, 178.92 APE8-dihe-in -91.42, 131.88 APE8-rot-in 297.69 APE67-dihe-inflip 105.02, -24.11 -55.02, 126.46 APE12-dist-in 10.6028 APE11-dist-in 11.2776 APE10-dist-in 5.5393 APE9-dist-in 3.3156 None None None AF2 -1.0 1.0 1.0 A 282.0 282.0 0 28 28 0 [[190, 455]] 1.0 AF-Q15835-K1 Homo sapiens AGC_GRK1_HUMAN AGC 4.7e-81 277.6 4.0 260.0 257.0 334 335 336 338 340 219 238 242 314 316 315 317.0 374 362 357 356 355 354 353 352 351 268 Rhodopsin kinase GRK1
GRK1 GRK1_HUMAN AF-Q15835-K3A Q15835 182 463 563.0 No_ligand No_ligand Active DFGin 6.2345 12.6731 BLAminus -132.6, -178.51 49.86, 63.45 -76.42, 16.89 298.82, 166.43 -67.25, -17.86 in-in in 8.359 Saltbr-in 2.7065 HRD-in -85.57, -47.78 70.01, -0.82 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.92, 145.73 APE9-dihe-na 125.2, -163.99 APE8-dihe-in -109.07, 130.14 APE8-rot-in 295.51 APE67-dihe-inflip 103.48, -23.56 -54.31, 127.87 APE12-dist-in 10.5262 APE11-dist-in 11.024 APE10-dist-in 5.3332 APE9-dist-in 3.0336 None None None AF2 -1.0 1.0 1.0 A 282.0 282.0 0 28 28 0 [[190, 455]] 1.0 AF-Q15835-K3 Homo sapiens AGC_GRK1_HUMAN AGC 4.7e-81 277.6 4.0 260.0 257.0 334 335 336 338 340 219 238 242 314 316 315 317.0 374 362 357 356 355 354 353 352 351 268 Rhodopsin kinase GRK1

AGC_GRK1 (Rhodopsin kinase GRK1)

Total number of chains: 27
Active chains: 17
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 26 96.3% 3C4ZA
DFGinter None 1 3.7% 3C4YB

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GRK1 GRK1_BOVIN 3T8OA P28327 30 532 561.0 ATP:562 ATPlike Active DFGin 6.784 13.6519 BLAminus -147.61, 176.5 66.51, 86.5 -106.39, 20.07 278.45, 121.96 -78.51, -8.51 in-in in 9.1312 Saltbr-in 2.9462 HRD-in -72.08, -59.57 74.93, 15.13 in-in-in SNCiii in-in ActLoopNT-in 3.0341 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.6, 145.4 APE9-dihe-na 140.82, -165.62 APE8-dihe-in -114.33, 123.31 APE8-rot-in 302.45 APE67-dihe-inflip 90.49, -9.25 -48.36, 136.06 APE12-dist-in 10.4193 APE11-dist-in 11.6453 APE10-dist-in 5.7954 APE9-dist-in 4.2758 L166K None None XRAY 2.5 0.209 0.245 A 543.0 493.0 0 28 28 0 [[187, 452]] 1.0 3t8o Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4WA P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 6.5874 13.3137 BLAminus -157.51, 175.0 67.79, 80.23 -106.97, 21.1 277.77, 138.55 -72.95, -18.52 in-in in 8.6705 Saltbr-in 2.6589 HRD-in -67.86, -51.97 60.46, 12.85 in-in-in SNCiii in-in ActLoopNT-in 2.8974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.73, 153.77 APE9-dihe-na 125.45, -175.95 APE8-dihe-in -101.44, 127.92 APE8-rot-in 301.93 APE67-dihe-inflip 97.46, -21.92 -46.81, 133.28 APE12-dist-in 10.0067 APE11-dist-in 11.2485 APE10-dist-in 5.5344 APE9-dist-in 3.5083 None TPO8 TPO8 XRAY 2.7 0.192 999.0 A 543.0 494.0 0 28 28 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4WB P28327 5 533 561.0 ATP:562 ATPlike Active DFGin 5.9629 13.1113 BLAminus -155.04, 178.49 64.64, 79.84 -103.28, 19.03 277.57, 109.21 -72.3, -19.68 in-in in 8.548 Saltbr-in 2.84 HRD-in -67.79, -54.67 64.69, 11.83 in-in-in SNCiii in-in ActLoopNT-in 2.9583 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.45, 154.48 APE9-dihe-na 126.08, -175.35 APE8-dihe-in -101.18, 126.91 APE8-rot-in 300.91 APE67-dihe-inflip 94.23, -17.08 -47.18, 130.86 APE12-dist-in 10.1029 APE11-dist-in 11.2538 APE10-dist-in 5.5445 APE9-dist-in 3.5342 None TPO8 TPO8 XRAY 2.7 0.192 999.0 B 543.0 519.0 0 28 28 0 [[187, 452]] 1.0 3c4w Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4XA P28327 30 533 561.0 ATP:562 ATPlike Active DFGin 6.3918 13.2944 BLAminus -153.36, -178.73 56.38, 83.66 -101.23, 19.01 282.86, 141.85 -58.01, -33.04 in-in in 8.6227 Saltbr-in 2.8246 HRD-in -65.41, -52.58 62.44, 13.36 in-in-in SNCiii in-in ActLoopNT-in 2.9597 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.48, 144.22 APE9-dihe-na 128.55, -174.69 APE8-dihe-in -103.7, 129.98 APE8-rot-in 314.1 APE67-dihe-inflip 101.04, -22.84 -50.28, 132.61 APE12-dist-in 10.283 APE11-dist-in 11.2374 APE10-dist-in 5.7264 APE9-dist-in 3.8266 None None None XRAY 2.9 0.193 999.0 A 543.0 496.0 0 28 28 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4XB P28327 31 533 561.0 ATP:562 ATPlike Active DFGin 5.9031 13.063 BLAminus -149.62, 174.69 57.3, 76.73 -95.24, 8.98 282.05, 96.12 -51.11, -35.54 in-in in 8.6415 Saltbr-in 2.6755 HRD-in -62.32, -48.48 63.55, 4.44 in-in-in SNCiii in-in ActLoopNT-in 3.0432 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.42, 143.72 APE9-dihe-na 129.46, -175.16 APE8-dihe-in -98.28, 125.3 APE8-rot-in 312.69 APE67-dihe-inflip 98.15, -18.1 -45.11, 129.51 APE12-dist-in 10.2012 APE11-dist-in 11.2468 APE10-dist-in 5.6099 APE9-dist-in 3.6392 None None None XRAY 2.9 0.193 999.0 B 543.0 475.0 0 28 28 0 [[187, 452]] 1.0 3c4x Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4ZA P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.9128 13.2351 BLAminus -149.46, 171.26 70.91, 78.39 -108.02, 16.47 270.55, 111.24 -69.43, -16.01 in-in in 8.7363 Saltbr-in 2.7164 HRD-in -71.08, -53.07 69.31, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.8781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.53, 147.45 APE9-dihe-na 134.96, -165.72 APE8-dihe-in -111.39, 128.56 APE8-rot-in 296.58 APE67-dihe-inflip 96.79, -17.75 -54.96, 131.39 APE12-dist-in 10.4298 APE11-dist-in 11.1131 APE10-dist-in 5.4905 APE9-dist-in 3.5422 None None None XRAY 1.84 0.193 999.0 A 543.0 493.0 0 28 28 0 [[187, 452]] 1.0 3c4z Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C50A P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.0752 13.0339 BLAminus -142.59, 172.43 68.85, 78.38 -104.12, 14.36 280.99, 104.76 -67.57, -15.07 in-in in 8.6024 Saltbr-in 2.9252 HRD-in -76.21, -52.36 64.46, 15.62 in-in-in SNCiii in-in ActLoopNT-in 2.7949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.66, 144.27 APE9-dihe-na 130.37, -165.26 APE8-dihe-in -104.68, 131.22 APE8-rot-in 300.48 APE67-dihe-inflip 92.29, -6.18 -56.88, 135.03 APE12-dist-in 10.685 APE11-dist-in 11.4689 APE10-dist-in 5.8763 APE9-dist-in 3.4729 None None None XRAY 2.6 0.19 999.0 A 543.0 499.0 0 28 28 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C50B P28327 30 533 561.0 ADP:562 ATPlike Active DFGin 6.0782 13.0677 BLAminus -140.52, 175.4 66.53, 77.05 -104.14, 18.55 279.39, 103.87 -67.23, -21.39 in-in in 8.5322 Saltbr-in 2.7211 HRD-in -71.74, -52.34 63.89, 11.32 in-in-in SNCiii in-in ActLoopNT-in 2.8901 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -161.47, 143.37 APE9-dihe-na 137.53, -168.17 APE8-dihe-in -105.39, 125.32 APE8-rot-in 297.12 APE67-dihe-inflip 95.82, -17.57 -51.32, 135.4 APE12-dist-in 10.1294 APE11-dist-in 11.1147 APE10-dist-in 5.5383 APE9-dist-in 3.4184 None None None XRAY 2.6 0.19 999.0 B 543.0 496.0 0 28 28 0 [[187, 452]] 1.0 3c50 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C51A P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.7354 13.2354 BLAminus -156.28, 178.74 57.85, 73.51 -84.14, -2.01 283.03, 106.57 -47.35, -22.99 in-in in 8.7977 Saltbr-in 2.6866 HRD-in -64.41, -45.82 69.5, -19.46 in-in-in SNCiii in-in ActLoopNT-in 2.9155 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.64, 142.5 APE9-dihe-na 155.52, -169.52 APE8-dihe-in -101.5, 135.25 APE8-rot-in 300.99 APE67-dihe-inflip 84.91, 4.53 -59.96, 128.0 APE12-dist-in 10.573 APE11-dist-in 11.5413 APE10-dist-in 6.1515 APE9-dist-in 3.937 None None None XRAY 3.55 0.281 999.0 A 543.0 487.0 0 28 28 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C51B P28327 31 533 561.0 ADP:562 ATPlike Active DFGin 5.7851 13.1869 BLAminus -156.29, 175.57 58.57, 74.43 -85.29, -1.69 285.99, 107.07 -47.38, -22.91 in-in in 8.696 Saltbr-in 2.7915 HRD-in -66.67, -42.5 63.68, -15.39 in-in-in SNCiii in-in ActLoopNT-in 2.9686 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -176.05, 141.93 APE9-dihe-na 155.26, -171.96 APE8-dihe-in -101.33, 138.35 APE8-rot-in 299.85 APE67-dihe-inflip 84.6, 5.24 -64.39, 128.67 APE12-dist-in 10.5371 APE11-dist-in 11.5977 APE10-dist-in 6.1564 APE9-dist-in 3.9396 None None None XRAY 3.55 0.281 999.0 B 543.0 461.0 20 28 28 0 [[187, 452]] 1.0 3c51 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9A P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.8516 13.4841 BLAminus -151.04, 174.48 70.22, 99.25 -129.57, 18.73 275.22, 99.19 -61.63, -18.96 in-in in 8.9606 Saltbr-in 3.1273 HRD-in -61.98, -58.15 73.37, -3.42 in-in-in SNCiii in-in ActLoopNT-in 2.9166 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -167.32, 133.82 APE9-dihe-na 142.48, -169.15 APE8-dihe-in -104.33, 125.71 APE8-rot-in 302.67 APE67-dihe-inflip 104.42, -3.83 -50.74, 122.55 APE12-dist-in 10.3557 APE11-dist-in 11.0144 APE10-dist-in 5.5004 APE9-dist-in 3.6645 T8C,N480C None None XRAY 2.7 0.194 0.229 A 543.0 486.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9B P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.8991 13.5043 BLAminus -154.17, 173.67 70.5, 100.81 -132.54, 18.75 276.87, 97.69 -56.57, -24.02 in-in in 8.931 Saltbr-in 3.099 HRD-in -65.24, -58.34 73.4, -2.88 in-in-in SNCiii in-in ActLoopNT-in 2.9339 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -166.53, 132.45 APE9-dihe-na 145.72, -169.79 APE8-dihe-in -103.09, 126.5 APE8-rot-in 303.38 APE67-dihe-inflip 99.94, -4.73 -52.12, 123.93 APE12-dist-in 10.3676 APE11-dist-in 11.0383 APE10-dist-in 5.525 APE9-dist-in 3.6772 T8C,N480C None None XRAY 2.7 0.194 0.229 B 543.0 481.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9C P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.8677 13.481 BLAminus -151.87, 172.48 72.03, 98.62 -128.19, 19.72 276.34, 98.38 -59.47, -19.79 in-in in 8.9508 Saltbr-in 3.1074 HRD-in -62.09, -58.44 72.04, -1.68 in-in-in SNCiii in-in ActLoopNT-in 2.9357 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -168.26, 134.05 APE9-dihe-na 142.83, -170.11 APE8-dihe-in -104.04, 126.58 APE8-rot-in 301.36 APE67-dihe-inflip 105.14, -2.81 -49.9, 120.73 APE12-dist-in 10.3838 APE11-dist-in 11.0185 APE10-dist-in 5.5081 APE9-dist-in 3.673 T8C,N480C None None XRAY 2.7 0.194 0.229 C 543.0 482.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3QC9D P28327 31 533 561.0 ADP:700 ATPlike Active DFGin 6.9233 13.5167 BLAminus -151.29, 174.11 71.25, 99.27 -130.54, 20.81 276.77, 98.72 -58.99, -24.3 in-in in 8.9307 Saltbr-in 3.0905 HRD-in -63.44, -57.63 71.87, -0.43 in-in-in SNCiii in-in ActLoopNT-in 2.9269 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -165.95, 134.69 APE9-dihe-na 141.2, -168.54 APE8-dihe-in -103.28, 126.55 APE8-rot-in 303.76 APE67-dihe-inflip 102.49, -2.5 -51.29, 121.62 APE12-dist-in 10.3966 APE11-dist-in 11.0439 APE10-dist-in 5.5135 APE9-dist-in 3.693 T8C,N480C None None XRAY 2.7 0.194 0.229 D 543.0 486.0 0 28 28 0 [[187, 452]] 1.0 3qc9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4L9IB P28327 31 533 561.0 8PR:601 Type1 Active DFGin 5.7147 13.0643 BLAminus -147.41, -179.95 59.09, 74.76 -90.68, 22.77 285.65, 103.28 -76.71, -12.5 in-in in 8.7578 Saltbr-in 3.1172 HRD-in -77.55, -56.18 71.16, 4.39 in-in-in SNCiii in-in ActLoopNT-in 2.7658 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.45, 143.07 APE9-dihe-na 140.89, -160.87 APE8-dihe-in -115.15, 127.72 APE8-rot-in 297.19 APE67-dihe-inflip 102.74, -33.6 -52.94, 132.06 APE12-dist-in 10.2921 APE11-dist-in 11.2208 APE10-dist-in 5.6416 APE9-dist-in 3.766 None None None XRAY 2.32 0.188 0.231 B 504.0 493.0 0 28 28 0 [[187, 452]] 1.0 4l9i Bos taurus AGC_GRK1_BOVIN AGC 2.5e-80 275.4 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4PNIA P28327 30 533 561.0 KQQ:601 Type1 Active DFGin 5.7355 13.1277 BLAminus -134.98, -179.15 54.91, 73.26 -92.23, 19.47 279.07, 113.0 -67.01, -18.73 in-in in 9.6807 Saltbr-in 3.1063 HRD-in -69.25, -51.31 65.76, 4.71 in-in-in SNCiii in-in ActLoopNT-in 2.9934 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.87, 143.44 APE9-dihe-na 144.11, -165.57 APE8-dihe-in -117.94, 131.85 APE8-rot-in 290.67 APE67-dihe-inflip 103.74, -23.28 -58.63, 131.5 APE12-dist-in 10.3397 APE11-dist-in 11.3538 APE10-dist-in 5.7216 APE9-dist-in 3.6813 None None None XRAY 1.85 0.191 0.23 A 561.0 492.0 0 28 28 0 [[187, 452]] 1.0 4pni Bos taurus AGC_GRK1_BOVIN AGC 3.3e-80 275.0 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MTBG P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Active DFGin 5.4472 13.977 BLAminus -158.7, 161.68 75.49, 110.48 -135.3, 45.5 298.35, 172.26 -102.18, -14.04 in-in in 8.1835 Saltbr-in 3.2327 HRD-in -84.4, -44.53 73.27, 9.15 in-in-in SNCiii in-in ActLoopNT-in 3.0388 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -63.06, 150.99 APE9-dihe-na 114.44, 173.54 APE8-dihe-in -100.2, 123.65 APE8-rot-in 303.1 APE67-dihe-inflip 95.63, -25.77 -41.47, 136.01 APE12-dist-in 10.1039 APE11-dist-in 10.473 APE10-dist-in 4.8138 APE9-dist-in 3.2162 S5E,S488E,T489E None None EM 4.0 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mtb Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4YA P28327 30 532 561.0 No_ligand No_ligand Inactive DFGin 7.6904 11.3511 BLAminus -137.44, 168.27 58.91, 104.81 -126.41, 38.75 308.65, 132.27 -61.68, -52.44 in-out in 9.8329 Saltbr-out 4.3893 HRD-in -106.52, -35.17 66.74, -61.42 out-in-in SNCoii in-in ActLoopNT-in 3.2444 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -178.5, 156.22 APE9-dihe-na 145.3, -132.92 APE8-dihe-in -136.09, 120.97 APE8-rot-in 304.15 APE67-dihe-inflip 122.03, -39.54 -49.39, 107.36 APE12-dist-in 11.4228 APE11-dist-in 12.6652 APE10-dist-in 7.6409 APE9-dist-in 5.7505 None None None XRAY 7.509 0.182 999.0 A 543.0 478.0 2 28 28 0 [[187, 452]] 1.0 3c4y Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4L9IA P28327 30 533 561.0 8PR:601 Type1 Inactive DFGin 5.7724 13.4538 BLAminus -149.91, 178.73 54.74, 79.81 -98.99, 23.91 282.53, 102.36 -68.07, -19.68 in-out in 8.693 Saltbr-out 3.808 HRD-in -75.83, -53.93 68.31, 13.36 out-in-in SNCoii in-in ActLoopNT-in 2.8273 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.8, 142.88 APE9-dihe-na 125.17, -158.26 APE8-dihe-in -112.07, 133.06 APE8-rot-in 301.6 APE67-dihe-inflip 94.99, -2.22 -45.66, 120.79 APE12-dist-in 10.6157 APE11-dist-in 11.3826 APE10-dist-in 5.8078 APE9-dist-in 3.7234 None None None XRAY 2.32 0.188 0.231 A 504.0 504.0 0 28 28 0 [[187, 452]] 1.0 4l9i Bos taurus AGC_GRK1_BOVIN AGC 2.5e-80 275.4 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOA P28327 28 533 561.0 ANW:601 Type1 Inactive DFGin 5.9481 13.2578 BLAminus -146.44, 170.56 64.48, 78.76 -93.1, 25.97 287.19, 103.23 -64.53, -31.02 in-out in 9.4403 Saltbr-out 4.1695 HRD-in -74.57, -52.51 66.08, 11.01 out-in-in SNCoii in-in ActLoopNT-in 2.8138 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.31, 145.0 APE9-dihe-na 138.11, -171.62 APE8-dihe-in -107.94, 132.02 APE8-rot-in 308.16 APE67-dihe-inflip 100.64, -17.52 -51.85, 128.49 APE12-dist-in 10.2576 APE11-dist-in 11.1305 APE10-dist-in 5.5198 APE9-dist-in 3.5303 None None None XRAY 2.81 0.243 0.267 A 541.0 497.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOB P28327 30 533 561.0 ANW:601 Type1 Inactive DFGin 5.9542 13.2886 BLAminus -146.62, 171.17 63.95, 77.64 -91.91, 26.29 286.92, 103.21 -63.89, -32.19 in-out in 9.5168 Saltbr-out 4.1969 HRD-in -74.66, -52.71 66.21, 10.61 out-in-in SNCoii in-in ActLoopNT-in 2.8113 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.36, 145.07 APE9-dihe-na 138.91, -171.46 APE8-dihe-in -107.75, 132.29 APE8-rot-in 308.55 APE67-dihe-inflip 100.74, -17.56 -52.36, 128.88 APE12-dist-in 10.2543 APE11-dist-in 11.1301 APE10-dist-in 5.5133 APE9-dist-in 3.5248 None None None XRAY 2.81 0.243 0.267 B 541.0 495.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOC P28327 31 531 561.0 ANW:601 Type1 Inactive DFGin 5.9556 13.1632 BLAminus -146.21, 170.22 64.35, 78.08 -92.41, 26.2 287.47, 102.96 -63.87, -32.11 in-out in 9.3966 Saltbr-out 3.7689 HRD-in -74.89, -52.54 66.21, 10.58 out-in-in SNCoii in-in ActLoopNT-in 2.8069 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.19, 145.1 APE9-dihe-na 138.92, -171.47 APE8-dihe-in -107.47, 132.18 APE8-rot-in 308.34 APE67-dihe-inflip 100.67, -17.42 -51.93, 128.63 APE12-dist-in 10.2519 APE11-dist-in 11.1292 APE10-dist-in 5.5118 APE9-dist-in 3.5259 None None None XRAY 2.81 0.243 0.267 C 541.0 481.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 4WBOD P28327 30 531 561.0 ANW:601 Type1 Inactive DFGin 5.9637 13.2454 BLAminus -146.28, 170.52 64.39, 78.16 -92.93, 26.26 287.26, 103.4 -64.25, -31.88 in-out in 9.4433 Saltbr-out 4.1679 HRD-in -74.7, -52.76 66.23, 10.86 out-in-in SNCoii in-in ActLoopNT-in 2.8047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.01, 145.2 APE9-dihe-na 138.57, -171.52 APE8-dihe-in -107.49, 131.96 APE8-rot-in 308.49 APE67-dihe-inflip 100.73, -17.59 -51.76, 128.57 APE12-dist-in 10.2771 APE11-dist-in 11.157 APE10-dist-in 5.5301 APE9-dist-in 3.529 None None None XRAY 2.81 0.243 0.267 D 541.0 491.0 0 28 28 0 [[187, 452]] 1.0 4wbo Bos taurus AGC_GRK1_BOVIN AGC 3e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MT9G P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Inactive DFGin 5.6744 13.0596 BLAminus -151.44, 153.5 75.1, 83.16 -101.64, 23.22 308.74, 9.79 -95.55, -5.25 in-out in 8.3758 Saltbr-out 3.7806 HRD-out -84.42, -25.78 58.78, -116.78 out-in-out SNCoio in-out ActLoopNT-in 2.9966 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iiio APE10-dihe-na -156.18, 168.76 APE9-dihe-na 65.79, -175.16 APE8-dihe-in -118.77, 133.16 APE8-rot-in 303.35 APE67-dihe-inflip 85.9, 7.81 -39.32, 131.4 APE12-dist-in 12.4268 APE11-dist-in 12.0285 APE10-dist-in 6.4797 APE9-dist-out 6.7808 None None None EM 7.0 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mt9 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MT8G P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Inactive DFGin 5.2778 13.8515 BLAminus -151.24, 148.8 73.0, 121.86 -132.91, 52.67 297.42, 171.65 -103.81, -13.33 in-in in 8.7716 Saltbr-in 3.2791 HRD-in -93.25, -20.41 75.09, -77.24 in-in-out SNCiio in-out ActLoopNT-in 3.0353 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.01, 152.4 APE9-dihe-na 69.43, 177.13 APE8-dihe-in -91.35, 141.08 APE8-rot-out 53.33 APE67-dihe-inflip 95.78, 14.3 -52.12, 148.5 APE12-dist-in 10.7091 APE11-dist-in 10.3507 APE10-dist-in 4.9503 APE9-dist-in 3.4095 S5E,S488E,T489E None None EM 5.8 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mt8 Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 7MTAG P28327 6 508 561.0 SGV:601,SGV:601,SGV:601,SGV:601,SGV:601,SGV:601 Type1,Type1,Type1,Type1,Type1,Type1 Inactive DFGin 4.0904 13.8437 BLAminus -167.88, 170.04 60.34, 64.21 -82.37, 97.38 303.24, 179.85 -89.6, -128.64 in-out in 8.6589 Saltbr-out 5.1993 HRD-in -95.2, -46.79 83.22, -60.37 out-in-in SNCoii in-in ActLoopNT-in 3.0912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.79, 133.35 APE9-dihe-na 142.18, 170.18 APE8-dihe-in -78.99, 123.97 APE8-rot-in 304.47 APE67-dihe-inflip 89.96, 4.75 -51.0, 134.99 APE12-dist-in 11.1037 APE11-dist-in 11.0248 APE10-dist-in 5.5893 APE9-dist-in 3.7938 S5E,S488E,T489E None None EM 4.1 999.0 999.0 G 543.0 346.0 0 28 28 0 [[187, 452]] 1.0 7mta Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1
GRK1 GRK1_BOVIN 3C4YB P28327 30 532 561.0 No_ligand No_ligand Inactive DFGinter 8.0405 10.5531 None -138.64, 168.89 59.27, 104.12 -125.95, 37.77 308.57, 133.4 -61.52, -52.16 in-out in 9.8319 Saltbr-out 4.4166 HRD-in -105.99, -36.37 67.54, -61.73 out-in-in SNCoii in-in ActLoopNT-in 3.2059 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -178.33, 157.76 APE9-dihe-na 144.04, -133.41 APE8-dihe-in -135.26, 121.19 APE8-rot-in 303.52 APE67-dihe-inflip 122.3, -40.41 -49.79, 107.51 APE12-dist-in 11.4257 APE11-dist-in 12.6565 APE10-dist-in 7.6316 APE9-dist-in 5.7888 None None None XRAY 7.509 0.182 999.0 B 543.0 466.0 8 28 28 0 [[187, 452]] 1.0 3c4y Bos taurus AGC_GRK1_BOVIN AGC 3.1e-80 275.1 4.0 260.0 257.0 331 332 333 335 337 216 235 239 311 313 312 314.0 371 359 354 353 352 351 350 349 348 265 Rhodopsin kinase GRK1