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| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | PIM1 | PIM1_HUMAN | 5O11A | P11309 | 34 | 305 | 313.0 | 3NG:401 | Type1 | Active | DFGin | 6.128 | 14.611 | BLAminus | -127.88, 174.91 | 62.14, 80.5 | -88.8, 17.09 | 290.86, 80.03 | -61.06, -19.7 | in-in | in | 8.856 | Saltbr-in | 2.607 | HRD-na-A | -68.12, -50.16 | 69.42, 1.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.35, 8.9 | APE9-dihe-na | -86.78, -150.83 | APE8-dihe-in | -93.81, 133.37 | APE8-rot-in | 308.93 | APE67-dihe-in | -69.86, -10.11 | -67.48, -44.09 | APE12-dist-in | 9.742 | APE11-dist-in | 8.73 | APE10-dist-in | 4.861 | APE9-dist-in | 3.817 | None | SEP261 | CME161,SEP261 | XRAY | 2.4 | 0.167 | 0.212 | A | 298 | 270 | 2 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 5o11 | CAMK_PIM1_HUMAN | CAMK | 3.4e-65 | 225.9 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDC | P49759 | 150 | 479 | 484.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.026 | 14.412 | ABAminus | -125.6, -45.1 | -89.27, 107.55 | -111.64, 19.23 | 292.41, 98.32 | -77.1, 0.74 | in-in | in | 8.767 | Saltbr-in | 2.904 | HRD-in | -53.74, -54.41 | 89.98, -20.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.895 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -118.02, -81.8 | APE9-dihe-na | -80.38, 126.35 | APE8-dihe-in | -130.72, 139.1 | APE8-rot-out | 73.02 | APE67-dihe-in | -49.48, -32.44 | -62.98, -36.18 | APE12-dist-in | 13.371 | APE11-dist-in | 9.097 | APE10-dist-out | 11.33 | APE9-dist-out | 7.849 | None | None | None | XRAY | 2.7 | 0.204 | 0.274 | C | 484 | 325 | 5 | 0 | 0 | 0 | [[161, 477]] | 1.0 | 6khd | CMGC_CLK1_HUMAN | CMGC | 8.2e-93 | 317.4 | 1 | 301 | 301 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDB | P49759 | 149 | 482 | 484.0 | 3NG:1000 | Type1 | Inactive | DFGin | 6.908 | 14.076 | BLAminus | -116.48, -175.0 | 67.35, 80.01 | -102.96, 15.9 | 292.23, 100.48 | -53.02, -40.84 | in-in | in | 8.583 | Saltbr-in | 2.636 | HRD-in | -57.21, -57.72 | 79.07, -3.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.918 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -136.88, 104.05 | APE9-dihe-na | 173.26, -145.7 | APE8-dihe-in | -145.78, 56.63 | APE8-rot-in | 325.36 | APE67-dihe-out | -165.57, -36.7 | 24.99, 58.5 | APE12-dist-in | 13.582 | APE11-dist-in | 11.89 | APE10-dist-in | 6.825 | APE9-dist-in | 3.747 | None | None | None | XRAY | 2.7 | 0.204 | 0.274 | B | 484 | 332 | 2 | 0 | 0 | 0 | [[161, 477]] | 1.0 | 6khd | CMGC_CLK1_HUMAN | CMGC | 8.2e-93 | 317.4 | 1 | 301 | 301 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDA | P49759 | 149 | 481 | 484.0 | 3NG:1000 | Type1 | Inactive | DFGin | 6.862 | 14.485 | None | -115.36, -74.37 | -61.99, 112.36 | -110.01, 19.25 | 292.55, 104.1 | -59.59, -27.31 | in-in | in | 8.753 | Saltbr-in | 2.455 | HRD-in | -79.61, -40.92 | 65.39, -11.49 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.98 | ActLoopCT-out | nonTYR | APEdihe_aannn | APEdist_ioon | APE10-dihe-na | -162.31, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -85.78, 10.46 | 999.0, -15.39 | APE12-dist-in | 11.868 | APE11-dist-out | 7.043 | APE10-dist-out | 11.635 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.204 | 0.274 | A | 484 | 322 | 11 | 0 | 0 | 2 | [[161, 477]] | 1.0 | 6khd | CMGC_CLK1_HUMAN | CMGC | 8.2e-93 | 317.4 | 1 | 301 | 301 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYLA | P49760 | 144 | 483 | 499.0 | 3NG:501 | Type1 | Active | DFGin | 7.161 | 14.637 | BLAminus | -119.92, -175.89 | 60.38, 80.92 | -97.43, 16.84 | 290.06, 87.59 | -59.22, -23.17 | in-in | in | 9.054 | Saltbr-in | 2.46 | HRD-in | -71.74, -50.4 | 78.44, -13.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.783 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.7, 169.22 | APE9-dihe-na | 74.63, 150.35 | APE8-dihe-in | -69.34, 134.45 | APE8-rot-in | 299.9 | APE67-dihe-in | -60.04, -23.84 | -27.22, -60.14 | APE12-dist-in | 13.376 | APE11-dist-in | 11.885 | APE10-dist-in | 7.467 | APE9-dist-in | 2.93 | None | None | None | XRAY | 1.95 | 0.19 | 0.213 | A | 363 | 340 | 0 | 0 | 0 | 0 | [[163, 479]] | 1.0 | 6fyl | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1 | 301 | 301 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6KHEA | P49760 | 144 | 485 | 499.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.055 | 14.837 | BLAminus | -131.68, -176.57 | 65.16, 73.84 | -91.75, 19.3 | 289.49, 98.72 | -67.18, -14.55 | in-in | in | 9.186 | Saltbr-in | 2.61 | HRD-out | -72.06, 107.81 | -82.72, -0.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.114 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.6, 166.16 | APE9-dihe-na | 72.38, -179.55 | APE8-dihe-in | -103.99, 128.19 | APE8-rot-in | 299.55 | APE67-dihe-in | -66.25, -31.78 | -33.5, -45.82 | APE12-dist-in | 13.323 | APE11-dist-in | 11.976 | APE10-dist-in | 7.484 | APE9-dist-in | 3.318 | None | None | None | XRAY | 2.8 | 0.203 | 0.261 | A | 499 | 342 | 0 | 0 | 0 | 0 | [[163, 479]] | 1.0 | 6khe | CMGC_CLK2_HUMAN | CMGC | 4.9e-92 | 314.7 | 1 | 301 | 301 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK3 | CLK3_HUMAN | 6FYPA | P49761 | 135 | 482 | 490.0 | 3NG:501 | Type1 | Active | DFGin | 7.371 | 14.517 | BLAminus | -116.73, 177.74 | 60.44, 79.82 | -96.62, 15.47 | 286.13, 83.84 | -75.93, 15.05 | in-in | in | 8.93 | Saltbr-in | 2.503 | HRD-in | -67.5, -54.16 | 75.08, -16.75 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.686 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.43, 170.83 | APE9-dihe-na | 76.46, 148.77 | APE8-dihe-in | -66.24, 143.06 | APE8-rot-in | 302.49 | APE67-dihe-in | -49.68, -26.63 | -51.83, -51.01 | APE12-dist-in | 13.97 | APE11-dist-in | 12.024 | APE10-dist-in | 7.436 | APE9-dist-in | 3.037 | None | None | None | XRAY | 2.29 | 0.23 | 0.267 | A | 360 | 348 | 2 | 0 | 0 | 0 | [[156, 472]] | 1.0 | 6fyp | CMGC_CLK3_HUMAN | CMGC | 1.2e-90 | 309.6 | 1 | 301 | 301 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 6KHFA | P49761 | 142 | 481 | 490.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.15 | 14.219 | BLAminus | -127.11, -179.47 | 56.9, 68.81 | -87.1, 27.16 | 289.67, 76.33 | -67.97, -3.15 | in-in | in | 8.845 | Saltbr-in | 2.725 | HRD-out | -71.79, 130.53 | -107.28, 17.73 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.857 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioi | APE10-dihe-na | -140.37, -24.13 | APE9-dihe-na | -98.19, 177.1 | APE8-dihe-in | -67.74, 125.23 | APE8-rot-in | 310.54 | APE67-dihe-in | -68.95, -22.53 | -32.12, -48.44 | APE12-dist-out | 14.308 | APE11-dist-in | 12.383 | APE10-dist-out | 8.09 | APE9-dist-in | 3.641 | None | None | None | XRAY | 2.598 | 0.229 | 0.284 | A | 490 | 327 | 15 | 0 | 0 | 0 | [[156, 472]] | 1.0 | 6khf | CMGC_CLK3_HUMAN | CMGC | 3.4e-90 | 308.4 | 1 | 301 | 301 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK4 | CLK4_HUMAN | 6FYVA | Q9HAZ1 | 148 | 479 | 481.0 | 3NG:60501 | Type1 | Active | DFGin | 7.194 | 14.312 | BLAminus | -120.78, 176.99 | 65.84, 75.81 | -95.62, 15.62 | 293.79, 91.03 | -57.52, -19.12 | in-in | in | 8.769 | Saltbr-in | 2.784 | HRD-in | -64.07, -51.05 | 77.92, -13.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.05, 170.31 | APE9-dihe-na | 72.69, 148.35 | APE8-dihe-in | -68.0, 139.98 | APE8-rot-in | 290.09 | APE67-dihe-in | -63.52, -22.37 | -39.86, -52.09 | APE12-dist-in | 13.223 | APE11-dist-in | 11.408 | APE10-dist-in | 7.359 | APE9-dist-in | 3.027 | None | None | None | XRAY | 2.46 | 0.204 | 0.223 | A | 337 | 329 | 3 | 0 | 0 | 0 | [[159, 475]] | 1.0 | 6fyv | CMGC_CLK4_HUMAN | CMGC | 8.9e-93 | 316.7 | 1 | 301 | 301 | 322 | 323 | 324 | 326 | 328 | 189 | 204 | 208 | 283 | 285 | 284 | 286 | 359 | 347 | 342 | 341 | 340 | 339 | 338 | 337 | 336 | 240 | Dual specificity protein kinase CLK4 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHA | P68400 | 2 | 333 | 391.0 | SY4:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.477 | 16.394 | BLAminus | -121.68, -179.33 | 58.66, 73.4 | -93.07, 20.44 | 296.95, 80.12 | -72.1, -13.43 | in-in | in | 9.552 | Saltbr-in | 2.705 | HRD-in | -71.8, -47.17 | 67.87, 7.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.938 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -131.17, 164.17 | APE9-dihe-na | 70.19, 157.91 | APE8-dihe-in | -73.34, 145.8 | APE8-rot-out | 156.95 | APE67-dihe-in | -65.82, -17.6 | -47.03, -48.02 | APE12-dist-in | 12.626 | APE11-dist-in | 10.464 | APE10-dist-in | 6.133 | APE9-dist-in | 3.368 | None | None | None | XRAY | 1.96 | 0.201 | 0.241 | A | 355 | 332 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hyh | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAA | P68400 | 2 | 332 | 391.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.375 | 16.206 | BLAminus | -109.97, -178.65 | 53.41, 79.28 | -94.14, 17.71 | 296.64, 82.05 | -65.34, -22.88 | in-in | in | 9.136 | Saltbr-in | 2.63 | HRD-in | -74.72, -46.8 | 68.49, 9.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.38, 173.93 | APE9-dihe-na | 62.93, -179.6 | APE8-dihe-in | -105.16, 145.11 | APE8-rot-out | 135.96 | APE67-dihe-in | -65.3, -19.19 | -33.68, -57.22 | APE12-dist-in | 12.574 | APE11-dist-in | 10.393 | APE10-dist-in | 6.071 | APE9-dist-in | 3.094 | None | None | None | XRAY | 2.71 | 0.189 | 0.218 | A | 333 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 3nga | CMGC_CSNK2A1_HUMAN | CMGC | 1.3e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAB | P68400 | 2 | 332 | 391.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.39 | 16.337 | BLAminus | -109.78, -178.98 | 53.4, 79.2 | -94.06, 17.66 | 296.54, 82.9 | -66.35, -22.63 | in-in | in | 9.212 | Saltbr-in | 2.629 | HRD-in | -75.46, -46.47 | 68.49, 7.96 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.89 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -124.41, 174.85 | APE9-dihe-na | 62.34, 178.86 | APE8-dihe-in | -102.65, 148.1 | APE8-rot-out | 136.21 | APE67-dihe-in | -68.17, -20.17 | -36.37, -54.19 | APE12-dist-in | 12.629 | APE11-dist-in | 10.538 | APE10-dist-in | 6.108 | APE9-dist-in | 3.133 | None | None | None | XRAY | 2.71 | 0.189 | 0.218 | B | 333 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 3nga | CMGC_CSNK2A1_HUMAN | CMGC | 1.3e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3PE1A | P68400 | 3 | 329 | 391.0 | 3NG:338 | Type1 | Inactive | DFGin | 7.44 | 16.29 | BLAminus | -112.48, -179.47 | 50.32, 77.23 | -88.93, 20.86 | 296.76, 81.48 | -67.84, -19.52 | in-in | in | 9.203 | Saltbr-in | 2.717 | HRD-in | -76.91, -49.2 | 72.12, 6.33 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.904 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.3, 170.98 | APE9-dihe-na | 65.07, 159.47 | APE8-dihe-in | -81.62, 147.33 | APE8-rot-out | 162.29 | APE67-dihe-in | -67.89, -13.96 | -40.02, -55.24 | APE12-dist-in | 12.724 | APE11-dist-in | 10.359 | APE10-dist-in | 6.157 | APE9-dist-in | 3.234 | None | None | None | XRAY | 1.6 | 0.162 | 0.203 | A | 337 | 327 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 3pe1 | CMGC_CSNK2A1_HUMAN | CMGC | 1.4e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHB | P68400 | 2 | 332 | 391.0 | 3NG:401,SY4:402 | Type1,Allosteric | Inactive | DFGin | 7.455 | 16.686 | BLAminus | -121.17, -179.71 | 60.15, 74.28 | -94.36, 20.01 | 295.53, 80.91 | -72.98, -14.61 | in-in | in | 9.748 | Saltbr-in | 2.802 | HRD-in | -73.27, -48.07 | 68.78, 4.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.887 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.73, 163.63 | APE9-dihe-na | 71.35, 156.53 | APE8-dihe-in | -76.0, 150.02 | APE8-rot-out | 60.35 | APE67-dihe-in | -68.11, -15.2 | -46.02, -50.6 | APE12-dist-in | 12.749 | APE11-dist-in | 10.843 | APE10-dist-in | 6.32 | APE9-dist-in | 3.734 | None | None | None | XRAY | 1.96 | 0.201 | 0.241 | B | 355 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hyh | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHA | P68400 | 2 | 332 | 391.0 | 3NG:403,T9Y:404 | Type1,Allosteric | Inactive | DFGin | 7.383 | 16.565 | BLAminus | -118.8, -178.34 | 55.59, 76.92 | -97.73, 18.91 | 299.34, 78.81 | -65.83, -13.05 | in-in | in | 9.827 | Saltbr-in | 2.873 | HRD-in | -78.42, -45.3 | 64.02, 17.48 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.872 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.04, 164.88 | APE9-dihe-na | 65.11, 156.36 | APE8-dihe-in | -63.07, 152.22 | APE8-rot-out | 172.82 | APE67-dihe-in | -64.56, -17.94 | -58.04, -42.17 | APE12-dist-in | 12.698 | APE11-dist-in | 10.421 | APE10-dist-in | 6.18 | APE9-dist-in | 3.364 | None | None | None | XRAY | 2.07 | 0.216 | 0.256 | A | 355 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hzh | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHB | P68400 | 2 | 332 | 391.0 | 3NG:403,T9Y:404 | Type1,Allosteric | Inactive | DFGin | 7.368 | 16.552 | BLAminus | -119.62, -176.75 | 54.5, 77.97 | -98.25, 23.82 | 298.23, 80.81 | -69.92, -15.41 | in-in | in | 9.779 | Saltbr-in | 2.81 | HRD-in | -71.72, -44.22 | 63.92, 15.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.979 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.6, 164.83 | APE9-dihe-na | 66.55, 154.43 | APE8-dihe-in | -63.65, 152.11 | APE8-rot-out | 176.37 | APE67-dihe-in | -67.11, -13.32 | -56.47, -43.99 | APE12-dist-in | 12.789 | APE11-dist-in | 10.774 | APE10-dist-in | 6.319 | APE9-dist-in | 3.485 | None | None | None | XRAY | 2.07 | 0.216 | 0.256 | B | 355 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hzh | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A2 | CSK22_HUMAN | 8QBUA | P19784 | 6 | 333 | 350.0 | 42J:404,3NG:405 | Allosteric,Type1 | Inactive | DFGin | 7.481 | 16.117 | BLAminus | -115.34, 177.54 | 56.37, 76.99 | -87.29, 16.84 | 296.65, 81.34 | -70.83, -16.25 | in-in | in | 9.243 | Saltbr-in | 2.767 | HRD-in | -74.29, -50.68 | 73.5, 10.15 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.839 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -134.98, 166.78 | APE9-dihe-na | 65.99, 156.92 | APE8-dihe-in | -70.01, 146.12 | APE8-rot-out | 159.04 | APE67-dihe-in | -73.31, -10.45 | -44.42, -45.9 | APE12-dist-in | 12.462 | APE11-dist-in | 10.009 | APE10-dist-in | 6.107 | APE9-dist-in | 3.241 | C336S | None | None | XRAY | 1.09 | 0.16 | 0.179 | A | 364 | 328 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 8qbu | CMGC_CSNK2A2_HUMAN | CMGC | 1e-69 | 241.0 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9IHIA | P19784 | 7 | 333 | 350.0 | SY4:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.415 | 16.026 | BLAminus | -114.42, 178.99 | 58.97, 77.48 | -92.68, 17.89 | 295.72, 83.62 | -70.78, -17.6 | in-in | in | 9.166 | Saltbr-in | 2.815 | HRD-in | -75.11, -48.36 | 72.21, 10.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.841 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.76, 169.32 | APE9-dihe-na | 65.88, 158.62 | APE8-dihe-in | -76.33, 145.23 | APE8-rot-out | 154.92 | APE67-dihe-in | -68.36, -16.5 | -40.48, -52.03 | APE12-dist-in | 12.783 | APE11-dist-in | 10.506 | APE10-dist-in | 6.283 | APE9-dist-in | 3.236 | C336S | None | None | XRAY | 1.23 | 0.136 | 0.166 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9ihi | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9BA | P19784 | 7 | 333 | 350.0 | VN9:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.47 | 16.135 | BLAminus | -114.78, -178.63 | 52.36, 80.6 | -90.66, 23.03 | 297.12, 80.84 | -72.97, -19.45 | in-in | in | 9.164 | Saltbr-in | 2.851 | HRD-in | -75.12, -49.8 | 73.87, 8.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.899 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -131.85, 168.61 | APE9-dihe-na | 65.18, 157.14 | APE8-dihe-in | -73.48, 146.48 | APE8-rot-out | 146.34 | APE67-dihe-in | -70.57, -17.74 | -39.27, -49.01 | APE12-dist-in | 12.665 | APE11-dist-in | 10.424 | APE10-dist-in | 6.226 | APE9-dist-in | 3.23 | C336S | None | None | XRAY | 1.84 | 0.168 | 0.206 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9q9b | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QB6A | P19784 | 7 | 333 | 350.0 | RDV:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.4 | 16.015 | BLAminus | -116.09, 178.07 | 58.12, 76.49 | -88.07, 15.69 | 297.72, 81.25 | -71.25, -16.82 | in-in | in | 9.094 | Saltbr-in | 2.784 | HRD-in | -72.64, -51.36 | 73.74, 9.54 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.862 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.78, 169.18 | APE9-dihe-na | 62.18, 162.55 | APE8-dihe-in | -82.53, 146.39 | APE8-rot-out | 147.47 | APE67-dihe-in | -70.59, -14.66 | -39.2, -52.96 | APE12-dist-in | 12.702 | APE11-dist-in | 10.373 | APE10-dist-in | 6.226 | APE9-dist-in | 3.212 | C336S | None | None | XRAY | 1.05 | 0.127 | 0.144 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9qb6 | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QABA | P19784 | 7 | 333 | 350.0 | RA7:401,3NG:402,RA7:403 | Allosteric,Type1,Allosteric | Inactive | DFGin | 7.376 | 16.117 | BLAminus | -113.6, 178.31 | 57.83, 77.52 | -90.77, 14.85 | 296.13, 81.67 | -69.28, -17.99 | in-in | in | 9.175 | Saltbr-in | 2.76 | HRD-in | -72.54, -50.49 | 72.75, 9.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.902 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.24, 170.06 | APE9-dihe-na | 64.96, 162.68 | APE8-dihe-in | -81.37, 147.07 | APE8-rot-out | 150.87 | APE67-dihe-in | -69.81, -15.24 | -39.22, -53.5 | APE12-dist-in | 12.716 | APE11-dist-in | 10.351 | APE10-dist-in | 6.227 | APE9-dist-in | 3.188 | C336S | None | None | XRAY | 0.95 | 0.131 | 0.141 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9qab | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 6HMBA | P19784 | 7 | 334 | 350.0 | 3NG:413 | Type1 | Inactive | DFGin | 7.526 | 16.135 | BLAminus | -111.55, 174.56 | 58.24, 78.46 | -87.65, 16.17 | 297.85, 81.04 | -69.02, -17.39 | in-in | in | 9.184 | Saltbr-in | 2.771 | HRD-in | -73.83, -48.37 | 71.6, 10.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.872 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -135.43, 166.43 | APE9-dihe-na | 65.52, 156.91 | APE8-dihe-in | -69.62, 146.48 | APE8-rot-out | 153.38 | APE67-dihe-in | -70.99, -14.32 | -39.92, -51.06 | APE12-dist-in | 12.572 | APE11-dist-in | 10.14 | APE10-dist-in | 6.125 | APE9-dist-in | 3.269 | C336S | None | None | XRAY | 1.04 | 0.135 | 0.146 | A | 364 | 328 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 6hmb | CMGC_CSNK2A2_HUMAN | CMGC | 1e-69 | 241.0 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9HK5A | P19784 | 7 | 334 | 350.0 | 3NG:402 | Type1 | Inactive | DFGin | 7.542 | 16.208 | BLAminus | -114.65, -179.29 | 53.64, 80.01 | -92.35, 20.62 | 296.39, 82.42 | -74.28, -17.08 | in-in | in | 9.271 | Saltbr-in | 2.826 | HRD-in | -73.22, -49.09 | 72.9, 4.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.899 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -134.78, 167.23 | APE9-dihe-na | 62.78, 157.39 | APE8-dihe-in | -75.16, 149.06 | APE8-rot-out | 147.29 | APE67-dihe-in | -68.84, -16.32 | -43.13, -50.25 | APE12-dist-in | 12.694 | APE11-dist-in | 10.358 | APE10-dist-in | 6.315 | APE9-dist-in | 3.288 | P32V,V83I,T101I,C336S | None | None | XRAY | 1.491 | 0.175 | 0.204 | A | 364 | 328 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9hk5 | CMGC_CSNK2A2_HUMAN | CMGC | 3.1e-70 | 242.7 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9AA | P19784 | 7 | 333 | 350.0 | 3NG:401,A1I4V:402 | Type1,Allosteric | Inactive | DFGin | 7.397 | 16.171 | BLAminus | -114.27, 179.87 | 56.61, 76.76 | -86.69, 17.58 | 298.08, 81.74 | -71.41, -19.01 | in-in | in | 9.247 | Saltbr-in | 2.776 | HRD-in | -75.92, -48.72 | 71.51, 10.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.902 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -131.5, 165.78 | APE9-dihe-na | 68.3, 154.64 | APE8-dihe-in | -67.27, 146.08 | APE8-rot-out | 156.93 | APE67-dihe-in | -69.44, -15.07 | -43.26, -49.96 | APE12-dist-in | 12.724 | APE11-dist-in | 10.389 | APE10-dist-in | 6.234 | APE9-dist-in | 3.275 | C336S | None | None | XRAY | 1.03 | 0.147 | 0.156 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9q9a | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9DA | P19784 | 7 | 332 | 350.0 | 3NG:401,R9G:402 | Type1,Allosteric | Inactive | DFGin | 7.413 | 16.113 | BLAminus | -111.11, 176.5 | 58.97, 76.86 | -90.38, 17.87 | 296.15, 81.91 | -69.6, -18.64 | in-in | in | 9.215 | Saltbr-in | 2.79 | HRD-in | -72.74, -49.53 | 71.25, 10.86 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.74, 169.32 | APE9-dihe-na | 66.15, 161.19 | APE8-dihe-in | -81.94, 147.26 | APE8-rot-out | 152.61 | APE67-dihe-in | -69.62, -15.68 | -40.15, -53.5 | APE12-dist-in | 12.735 | APE11-dist-in | 10.379 | APE10-dist-in | 6.221 | APE9-dist-in | 3.183 | C336S | None | None | XRAY | 0.89 | 0.148 | 0.159 | A | 370 | 326 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9q9d | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QAGA | P19784 | 7 | 333 | 350.0 | 3NG:401,RBJ:402 | Type1,Allosteric | Inactive | DFGin | 7.402 | 16.146 | BLAminus | -113.78, 178.8 | 55.06, 77.97 | -89.73, 16.81 | 296.32, 81.5 | -70.74, -16.11 | in-in | in | 9.239 | Saltbr-in | 2.765 | HRD-in | -72.83, -48.69 | 70.11, 10.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.868 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.87, 167.19 | APE9-dihe-na | 64.82, 157.5 | APE8-dihe-in | -76.42, 146.88 | APE8-rot-out | 148.1 | APE67-dihe-in | -71.68, -14.1 | -39.59, -52.28 | APE12-dist-in | 12.68 | APE11-dist-in | 10.313 | APE10-dist-in | 6.249 | APE9-dist-in | 3.264 | C336S | None | None | XRAY | 1.01 | 0.136 | 0.162 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9qag | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NA | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.332 | 14.774 | BLAminus | -125.89, 175.46 | 60.34, 76.96 | -90.72, 25.89 | 277.64, 75.8 | -70.85, -23.55 | in-in | in | 8.867 | Saltbr-in | 2.627 | HRD-in | -70.94, -45.64 | 77.0, -3.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.65, -35.2 | APE9-dihe-na | -94.12, 169.14 | APE8-dihe-in | -81.45, 135.48 | APE8-rot-in | 271.72 | APE67-dihe-in | -57.78, -21.85 | -42.59, -54.66 | APE12-dist-in | 12.682 | APE11-dist-in | 11.088 | APE10-dist-in | 6.808 | APE9-dist-in | 3.373 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | A | 370 | 346 | 0 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NB | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 6.965 | 15.03 | BLAminus | -121.53, 177.86 | 59.36, 74.88 | -91.0, 24.04 | 284.65, 79.36 | -69.42, -6.51 | in-in | in | 9.072 | Saltbr-in | 2.955 | HRD-in | -65.31, -40.72 | 67.91, 3.75 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.837 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.86, 165.14 | APE9-dihe-na | 70.53, 140.66 | APE8-dihe-in | -62.36, 145.8 | APE8-rot-in | 271.48 | APE67-dihe-in | -55.51, -24.3 | -55.08, -48.98 | APE12-dist-in | 12.652 | APE11-dist-in | 11.24 | APE10-dist-in | 7.392 | APE9-dist-in | 3.193 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | B | 370 | 343 | 3 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NC | Q13627 | 134 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.125 | 14.845 | BLAminus | -127.45, -179.8 | 54.81, 79.63 | -96.7, 25.59 | 287.09, 79.21 | -71.97, -4.29 | in-in | in | 9.218 | Saltbr-in | 2.931 | HRD-in | -65.84, -47.16 | 77.48, 0.17 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.941 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -121.48, 175.3 | APE9-dihe-na | 70.69, 141.68 | APE8-dihe-in | -71.86, 144.08 | APE8-rot-in | 308.65 | APE67-dihe-in | -60.2, -32.88 | -49.5, -49.8 | APE12-dist-in | 13.034 | APE11-dist-in | 11.534 | APE10-dist-in | 7.148 | APE9-dist-in | 3.171 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | C | 370 | 344 | 3 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5ND | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.13 | 14.89 | BLAminus | -128.02, 175.09 | 60.57, 71.33 | -86.84, 26.43 | 281.73, 81.64 | -75.1, -14.91 | in-in | in | 9.081 | Saltbr-in | 2.672 | HRD-in | -60.22, -35.39 | 67.3, 3.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.821 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -92.57, 171.93 | APE9-dihe-na | 66.97, 156.51 | APE8-dihe-in | -85.5, 144.03 | APE8-rot-in | 283.59 | APE67-dihe-in | -57.76, -18.64 | -49.19, -52.69 | APE12-dist-in | 12.39 | APE11-dist-in | 10.732 | APE10-dist-in | 7.111 | APE9-dist-in | 3.042 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | D | 370 | 338 | 8 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NE | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.188 | 14.841 | BLAminus | -123.41, -179.95 | 58.6, 74.9 | -91.66, 28.87 | 284.52, 74.3 | -74.18, -15.86 | in-in | in | 8.932 | Saltbr-in | 2.599 | HRD-in | -66.53, -45.73 | 70.01, 6.86 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.729 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.5, 169.99 | APE9-dihe-na | 69.78, 136.41 | APE8-dihe-in | -57.94, 135.93 | APE8-rot-in | 298.8 | APE67-dihe-in | -52.87, -33.29 | -49.91, -51.82 | APE12-dist-in | 12.549 | APE11-dist-in | 11.378 | APE10-dist-in | 7.325 | APE9-dist-in | 3.185 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | E | 370 | 340 | 6 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NF | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.268 | 14.5 | BLAminus | -134.01, 179.07 | 56.51, 71.89 | -90.03, 23.99 | 289.58, 70.49 | -65.64, -23.07 | in-in | in | 9.224 | Saltbr-in | 2.867 | HRD-in | -69.65, -42.1 | 76.58, -5.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.88, -177.32 | APE9-dihe-na | 69.42, 90.94 | APE8-dihe-in | -27.36, 123.58 | APE8-rot-in | 265.98 | APE67-dihe-in | -50.43, -31.45 | -50.21, -44.01 | APE12-dist-in | 13.065 | APE11-dist-in | 11.252 | APE10-dist-in | 6.846 | APE9-dist-in | 3.171 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | F | 370 | 346 | 0 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NG | Q13627 | 137 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.344 | 14.781 | BLAminus | -131.27, 177.34 | 58.91, 64.55 | -81.55, 37.12 | 289.02, 78.81 | -81.79, -16.85 | in-in | in | 8.979 | Saltbr-in | 2.629 | HRD-in | -65.23, -49.26 | 77.2, 4.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.719 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.89, 64.11 | APE9-dihe-na | -161.3, 162.4 | APE8-dihe-in | -70.8, 130.74 | APE8-rot-in | 279.54 | APE67-dihe-in | -57.11, -25.99 | -52.9, -46.96 | APE12-dist-in | 12.712 | APE11-dist-in | 11.544 | APE10-dist-in | 6.759 | APE9-dist-in | 3.418 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | G | 370 | 333 | 11 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NH | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | None | DFGin | 6.679 | 14.847 | BLAminus | -128.66, -179.58 | 53.82, 77.25 | -93.05, 20.83 | 280.85, 75.88 | -63.97, -13.6 | in-in | in | 9.075 | Saltbr-in | 3.001 | HRD-in | -63.15, -47.83 | 74.92, 6.9 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.799 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_niii | APE10-dihe-na | -156.21, 166.85 | APE9-dihe-na | 64.29, 161.67 | APE8-dihe-in | -89.72, 140.84 | APE8-rot-none | 999.0 | APE67-dihe-in | -54.39, -32.97 | -48.02, -56.25 | APE12-dist-none | 999.0 | APE11-dist-in | 10.614 | APE10-dist-in | 7.767 | APE9-dist-in | 3.208 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | H | 370 | 307 | 39 | 0 | 0 | 4 | [[159, 479]] | 1.0 | 7z5n | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FA | P49841 | 28 | 383 | 420.0 | 3NG:60401 | Type1 | Inactive | DFGin | 7.172 | 14.387 | BLAminus | -140.61, -172.17 | 56.83, 67.31 | -90.44, 24.59 | 283.96, 78.9 | -70.58, -34.2 | in-in | in | 8.589 | Saltbr-in | 2.706 | HRD-in | -70.71, -48.08 | 68.23, 20.67 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.877 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -121.77, -56.1 | APE9-dihe-na | -73.95, 173.6 | APE8-dihe-in | -71.54, 133.95 | APE8-rot-out | 205.24 | APE67-dihe-in | -54.78, -22.55 | -52.86, -47.6 | APE12-dist-in | 13.711 | APE11-dist-in | 11.921 | APE10-dist-in | 7.257 | APE9-dist-in | 3.478 | None | PTR216 | PTR216 | XRAY | 3.0 | 0.224 | 0.249 | A | 364 | 354 | 2 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 7z1f | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.5 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FB | P49841 | 38 | 382 | 420.0 | 3NG:60401 | Type1 | Inactive | DFGin | 6.87 | 14.469 | BLAminus | -141.12, -171.82 | 52.8, 73.11 | -90.49, 20.89 | 285.47, 81.84 | -62.59, -35.1 | in-in | in | 9.025 | Saltbr-in | 2.763 | HRD-in | -68.41, -52.97 | 70.54, 14.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.039 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -122.34, -53.99 | APE9-dihe-na | -75.88, 165.71 | APE8-dihe-in | -64.92, 136.76 | APE8-rot-out | 179.7 | APE67-dihe-in | -58.44, -19.64 | -54.95, -47.33 | APE12-dist-in | 13.527 | APE11-dist-in | 11.859 | APE10-dist-in | 7.154 | APE9-dist-in | 3.558 | None | PTR216 | PTR216 | XRAY | 3.0 | 0.224 | 0.249 | B | 364 | 321 | 24 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 7z1f | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.5 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1GA | P49841 | 27 | 383 | 420.0 | 3NG:60401 | Type1 | Active | DFGin | 7.272 | 14.699 | BLAminus | -137.45, -179.93 | 52.32, 81.51 | -93.1, 20.22 | 282.75, 78.65 | -65.74, -16.48 | in-in | in | 8.969 | Saltbr-in | 2.771 | HRD-in | -67.62, -47.44 | 74.98, 2.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.926 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -86.67, 177.94 | APE9-dihe-na | 70.81, 142.84 | APE8-dihe-in | -95.23, 170.55 | APE8-rot-in | 305.08 | APE67-dihe-inflip | 72.5, -37.64 | -53.01, 158.1 | APE12-dist-in | 12.785 | APE11-dist-in | 10.847 | APE10-dist-in | 5.858 | APE9-dist-in | 2.984 | None | None | None | XRAY | 2.85 | 0.204 | 0.228 | A | 364 | 355 | 2 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 7z1g | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.5 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | HIPK2 | HIPK2_HUMAN | 6P5SA | Q9H2X6 | 185 | 535 | 1198.0 | 3NG:601 | Type1 | Inactive | DFGin | 7.298 | 14.23 | BLAminus | -121.5, -179.79 | 64.91, 82.62 | -96.84, 22.58 | 294.47, 82.62 | -64.48, -30.53 | in-in | in | 8.971 | Saltbr-in | 2.761 | HRD-in | -77.76, -49.7 | 67.78, 8.12 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.639 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -113.93, 168.02 | APE9-dihe-na | 68.38, 155.05 | APE8-dihe-in | -77.17, 138.14 | APE8-rot-out | 185.94 | APE67-dihe-in | -61.16, -24.2 | -57.86, -43.21 | APE12-dist-in | 10.584 | APE11-dist-in | 11.105 | APE10-dist-in | 7.495 | APE9-dist-in | 3.243 | None | PTR361,SEP441 | PTR361,SEP441 | XRAY | 2.194 | 0.2 | 0.238 | A | 390 | 333 | 18 | 0 | 0 | 6 | [[199, 527]] | 1.0 | 6p5s | CMGC_HIPK2_HUMAN | CMGC | 2.6e-92 | 315.4 | 1 | 301 | 301 | 345 | 346 | 347 | 349 | 351 | 228 | 243 | 247 | 321 | 323 | 322 | 324 | 383 | 371 | 366 | 365 | 364 | 363 | 362 | 361 | 360 | 278 | Homeodomain-interacting protein kinase 2 |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CKA1 | J9VNH4_CRYN9 | 6K3LB | J9VNH4 | 5 | 333 | 338.0 | 3NG:401 | Type1 | Inactive | DFGin | 7.66 | 16.152 | BLAminus | -114.35, -178.61 | 52.93, 78.12 | -89.9, 16.79 | 294.15, 81.47 | -67.97, -25.55 | in-in | in | 9.075 | Saltbr-in | 2.706 | HRD-in | -76.39, -51.63 | 76.4, 5.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.822 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -126.48, 161.19 | APE9-dihe-na | 73.24, 164.99 | APE8-dihe-in | -76.46, 151.58 | APE8-rot-out | 148.39 | APE67-dihe-in | -65.37, -22.86 | -51.07, -48.56 | APE12-dist-in | 12.822 | APE11-dist-in | 10.511 | APE10-dist-in | 6.303 | APE9-dist-in | 3.403 | None | None | None | XRAY | 2.09 | 0.189 | 0.219 | B | 338 | 329 | 0 | 0 | 0 | 0 | [[38, 323]] | 1.0 | 6k3l | Cryptococcus neoformans | CMGC_CKA1_CRYN9 | CMGC | 6e-64 | 222.0 | 1 | 301 | 301 | 173 | 174 | 175 | 177 | 179 | 67 | 80 | 84 | 152 | 154 | 153 | 155 | 213 | 200 | 195 | 194 | 193 | 192 | 191 | 190 | 189 | 113 | Casein kinase II subunit alpha |
| CAMK | PIM1 | PIM1_HUMAN | 5O11A | P11309 | 34 | 305 | 313.0 | 3NG:401 | Type1 | Active | DFGin | 6.128 | 14.611 | BLAminus | -127.88, 174.91 | 62.14, 80.5 | -88.8, 17.09 | 290.86, 80.03 | -61.06, -19.7 | in-in | in | 8.856 | Saltbr-in | 2.607 | HRD-na-A | -68.12, -50.16 | 69.42, 1.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.35, 8.9 | APE9-dihe-na | -86.78, -150.83 | APE8-dihe-in | -93.81, 133.37 | APE8-rot-in | 308.93 | APE67-dihe-in | -69.86, -10.11 | -67.48, -44.09 | APE12-dist-in | 9.742 | APE11-dist-in | 8.73 | APE10-dist-in | 4.861 | APE9-dist-in | 3.817 | None | SEP261 | CME161,SEP261 | XRAY | 2.4 | 0.167 | 0.212 | A | 298 | 270 | 2 | 0 | 0 | 0 | [[38, 290]] | 1.0 | 5o11 | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 3.4e-65 | 225.9 | 1 | 256 | 256 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDC | P49759 | 150 | 479 | 484.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.026 | 14.412 | ABAminus | -125.6, -45.1 | -89.27, 107.55 | -111.64, 19.23 | 292.41, 98.32 | -77.1, 0.74 | in-in | in | 8.767 | Saltbr-in | 2.904 | HRD-in | -53.74, -54.41 | 89.98, -20.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.895 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -118.02, -81.8 | APE9-dihe-na | -80.38, 126.35 | APE8-dihe-in | -130.72, 139.1 | APE8-rot-out | 73.02 | APE67-dihe-in | -49.48, -32.44 | -62.98, -36.18 | APE12-dist-in | 13.371 | APE11-dist-in | 9.097 | APE10-dist-out | 11.33 | APE9-dist-out | 7.849 | None | None | None | XRAY | 2.7 | 0.204 | 0.274 | C | 484 | 325 | 5 | 0 | 0 | 0 | [[161, 477]] | 1.0 | 6khd | Homo sapiens | CMGC_CLK1_HUMAN | CMGC | 8.2e-93 | 317.4 | 1 | 301 | 301 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDB | P49759 | 149 | 482 | 484.0 | 3NG:1000 | Type1 | Inactive | DFGin | 6.908 | 14.076 | BLAminus | -116.48, -175.0 | 67.35, 80.01 | -102.96, 15.9 | 292.23, 100.48 | -53.02, -40.84 | in-in | in | 8.583 | Saltbr-in | 2.636 | HRD-in | -57.21, -57.72 | 79.07, -3.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.918 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -136.88, 104.05 | APE9-dihe-na | 173.26, -145.7 | APE8-dihe-in | -145.78, 56.63 | APE8-rot-in | 325.36 | APE67-dihe-out | -165.57, -36.7 | 24.99, 58.5 | APE12-dist-in | 13.582 | APE11-dist-in | 11.89 | APE10-dist-in | 6.825 | APE9-dist-in | 3.747 | None | None | None | XRAY | 2.7 | 0.204 | 0.274 | B | 484 | 332 | 2 | 0 | 0 | 0 | [[161, 477]] | 1.0 | 6khd | Homo sapiens | CMGC_CLK1_HUMAN | CMGC | 8.2e-93 | 317.4 | 1 | 301 | 301 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6KHDA | P49759 | 149 | 481 | 484.0 | 3NG:1000 | Type1 | Inactive | DFGin | 6.862 | 14.485 | None | -115.36, -74.37 | -61.99, 112.36 | -110.01, 19.25 | 292.55, 104.1 | -59.59, -27.31 | in-in | in | 8.753 | Saltbr-in | 2.455 | HRD-in | -79.61, -40.92 | 65.39, -11.49 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.98 | ActLoopCT-out | nonTYR | APEdihe_aannn | APEdist_ioon | APE10-dihe-na | -162.31, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -85.78, 10.46 | 999.0, -15.39 | APE12-dist-in | 11.868 | APE11-dist-out | 7.043 | APE10-dist-out | 11.635 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.204 | 0.274 | A | 484 | 322 | 11 | 0 | 0 | 2 | [[161, 477]] | 1.0 | 6khd | Homo sapiens | CMGC_CLK1_HUMAN | CMGC | 8.2e-93 | 317.4 | 1 | 301 | 301 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYLA | P49760 | 144 | 483 | 499.0 | 3NG:501 | Type1 | Active | DFGin | 7.161 | 14.637 | BLAminus | -119.92, -175.89 | 60.38, 80.92 | -97.43, 16.84 | 290.06, 87.59 | -59.22, -23.17 | in-in | in | 9.054 | Saltbr-in | 2.46 | HRD-in | -71.74, -50.4 | 78.44, -13.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.783 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.7, 169.22 | APE9-dihe-na | 74.63, 150.35 | APE8-dihe-in | -69.34, 134.45 | APE8-rot-in | 299.9 | APE67-dihe-in | -60.04, -23.84 | -27.22, -60.14 | APE12-dist-in | 13.376 | APE11-dist-in | 11.885 | APE10-dist-in | 7.467 | APE9-dist-in | 2.93 | None | None | None | XRAY | 1.95 | 0.19 | 0.213 | A | 363 | 340 | 0 | 0 | 0 | 0 | [[163, 479]] | 1.0 | 6fyl | Homo sapiens | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1 | 301 | 301 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6KHEA | P49760 | 144 | 485 | 499.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.055 | 14.837 | BLAminus | -131.68, -176.57 | 65.16, 73.84 | -91.75, 19.3 | 289.49, 98.72 | -67.18, -14.55 | in-in | in | 9.186 | Saltbr-in | 2.61 | HRD-out | -72.06, 107.81 | -82.72, -0.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.114 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.6, 166.16 | APE9-dihe-na | 72.38, -179.55 | APE8-dihe-in | -103.99, 128.19 | APE8-rot-in | 299.55 | APE67-dihe-in | -66.25, -31.78 | -33.5, -45.82 | APE12-dist-in | 13.323 | APE11-dist-in | 11.976 | APE10-dist-in | 7.484 | APE9-dist-in | 3.318 | None | None | None | XRAY | 2.8 | 0.203 | 0.261 | A | 499 | 342 | 0 | 0 | 0 | 0 | [[163, 479]] | 1.0 | 6khe | Homo sapiens | CMGC_CLK2_HUMAN | CMGC | 4.9e-92 | 314.7 | 1 | 301 | 301 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK3 | CLK3_HUMAN | 6FYPA | P49761 | 135 | 482 | 490.0 | 3NG:501 | Type1 | Active | DFGin | 7.371 | 14.517 | BLAminus | -116.73, 177.74 | 60.44, 79.82 | -96.62, 15.47 | 286.13, 83.84 | -75.93, 15.05 | in-in | in | 8.93 | Saltbr-in | 2.503 | HRD-in | -67.5, -54.16 | 75.08, -16.75 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.686 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.43, 170.83 | APE9-dihe-na | 76.46, 148.77 | APE8-dihe-in | -66.24, 143.06 | APE8-rot-in | 302.49 | APE67-dihe-in | -49.68, -26.63 | -51.83, -51.01 | APE12-dist-in | 13.97 | APE11-dist-in | 12.024 | APE10-dist-in | 7.436 | APE9-dist-in | 3.037 | None | None | None | XRAY | 2.29 | 0.23 | 0.267 | A | 360 | 348 | 2 | 0 | 0 | 0 | [[156, 472]] | 1.0 | 6fyp | Homo sapiens | CMGC_CLK3_HUMAN | CMGC | 1.2e-90 | 309.6 | 1 | 301 | 301 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 6KHFA | P49761 | 142 | 481 | 490.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.15 | 14.219 | BLAminus | -127.11, -179.47 | 56.9, 68.81 | -87.1, 27.16 | 289.67, 76.33 | -67.97, -3.15 | in-in | in | 8.845 | Saltbr-in | 2.725 | HRD-out | -71.79, 130.53 | -107.28, 17.73 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.857 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioi | APE10-dihe-na | -140.37, -24.13 | APE9-dihe-na | -98.19, 177.1 | APE8-dihe-in | -67.74, 125.23 | APE8-rot-in | 310.54 | APE67-dihe-in | -68.95, -22.53 | -32.12, -48.44 | APE12-dist-out | 14.308 | APE11-dist-in | 12.383 | APE10-dist-out | 8.09 | APE9-dist-in | 3.641 | None | None | None | XRAY | 2.598 | 0.229 | 0.284 | A | 490 | 327 | 15 | 0 | 0 | 0 | [[156, 472]] | 1.0 | 6khf | Homo sapiens | CMGC_CLK3_HUMAN | CMGC | 3.4e-90 | 308.4 | 1 | 301 | 301 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK4 | CLK4_HUMAN | 6FYVA | Q9HAZ1 | 148 | 479 | 481.0 | 3NG:60501 | Type1 | Active | DFGin | 7.194 | 14.312 | BLAminus | -120.78, 176.99 | 65.84, 75.81 | -95.62, 15.62 | 293.79, 91.03 | -57.52, -19.12 | in-in | in | 8.769 | Saltbr-in | 2.784 | HRD-in | -64.07, -51.05 | 77.92, -13.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.05, 170.31 | APE9-dihe-na | 72.69, 148.35 | APE8-dihe-in | -68.0, 139.98 | APE8-rot-in | 290.09 | APE67-dihe-in | -63.52, -22.37 | -39.86, -52.09 | APE12-dist-in | 13.223 | APE11-dist-in | 11.408 | APE10-dist-in | 7.359 | APE9-dist-in | 3.027 | None | None | None | XRAY | 2.46 | 0.204 | 0.223 | A | 337 | 329 | 3 | 0 | 0 | 0 | [[159, 475]] | 1.0 | 6fyv | Homo sapiens | CMGC_CLK4_HUMAN | CMGC | 8.9e-93 | 316.7 | 1 | 301 | 301 | 322 | 323 | 324 | 326 | 328 | 189 | 204 | 208 | 283 | 285 | 284 | 286 | 359 | 347 | 342 | 341 | 340 | 339 | 338 | 337 | 336 | 240 | Dual specificity protein kinase CLK4 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHA | P68400 | 2 | 333 | 391.0 | SY4:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.477 | 16.394 | BLAminus | -121.68, -179.33 | 58.66, 73.4 | -93.07, 20.44 | 296.95, 80.12 | -72.1, -13.43 | in-in | in | 9.552 | Saltbr-in | 2.705 | HRD-in | -71.8, -47.17 | 67.87, 7.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.938 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -131.17, 164.17 | APE9-dihe-na | 70.19, 157.91 | APE8-dihe-in | -73.34, 145.8 | APE8-rot-out | 156.95 | APE67-dihe-in | -65.82, -17.6 | -47.03, -48.02 | APE12-dist-in | 12.626 | APE11-dist-in | 10.464 | APE10-dist-in | 6.133 | APE9-dist-in | 3.368 | None | None | None | XRAY | 1.96 | 0.201 | 0.241 | A | 355 | 332 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hyh | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAA | P68400 | 2 | 332 | 391.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.375 | 16.206 | BLAminus | -109.97, -178.65 | 53.41, 79.28 | -94.14, 17.71 | 296.64, 82.05 | -65.34, -22.88 | in-in | in | 9.136 | Saltbr-in | 2.63 | HRD-in | -74.72, -46.8 | 68.49, 9.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.38, 173.93 | APE9-dihe-na | 62.93, -179.6 | APE8-dihe-in | -105.16, 145.11 | APE8-rot-out | 135.96 | APE67-dihe-in | -65.3, -19.19 | -33.68, -57.22 | APE12-dist-in | 12.574 | APE11-dist-in | 10.393 | APE10-dist-in | 6.071 | APE9-dist-in | 3.094 | None | None | None | XRAY | 2.71 | 0.189 | 0.218 | A | 333 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 3nga | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.3e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3NGAB | P68400 | 2 | 332 | 391.0 | 3NG:1000 | Type1 | Inactive | DFGin | 7.39 | 16.337 | BLAminus | -109.78, -178.98 | 53.4, 79.2 | -94.06, 17.66 | 296.54, 82.9 | -66.35, -22.63 | in-in | in | 9.212 | Saltbr-in | 2.629 | HRD-in | -75.46, -46.47 | 68.49, 7.96 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.89 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -124.41, 174.85 | APE9-dihe-na | 62.34, 178.86 | APE8-dihe-in | -102.65, 148.1 | APE8-rot-out | 136.21 | APE67-dihe-in | -68.17, -20.17 | -36.37, -54.19 | APE12-dist-in | 12.629 | APE11-dist-in | 10.538 | APE10-dist-in | 6.108 | APE9-dist-in | 3.133 | None | None | None | XRAY | 2.71 | 0.189 | 0.218 | B | 333 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 3nga | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.3e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 3PE1A | P68400 | 3 | 329 | 391.0 | 3NG:338 | Type1 | Inactive | DFGin | 7.44 | 16.29 | BLAminus | -112.48, -179.47 | 50.32, 77.23 | -88.93, 20.86 | 296.76, 81.48 | -67.84, -19.52 | in-in | in | 9.203 | Saltbr-in | 2.717 | HRD-in | -76.91, -49.2 | 72.12, 6.33 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.904 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.3, 170.98 | APE9-dihe-na | 65.07, 159.47 | APE8-dihe-in | -81.62, 147.33 | APE8-rot-out | 162.29 | APE67-dihe-in | -67.89, -13.96 | -40.02, -55.24 | APE12-dist-in | 12.724 | APE11-dist-in | 10.359 | APE10-dist-in | 6.157 | APE9-dist-in | 3.234 | None | None | None | XRAY | 1.6 | 0.162 | 0.203 | A | 337 | 327 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 3pe1 | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.4e-69 | 240.6 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HYHB | P68400 | 2 | 332 | 391.0 | 3NG:401,SY4:402 | Type1,Allosteric | Inactive | DFGin | 7.455 | 16.686 | BLAminus | -121.17, -179.71 | 60.15, 74.28 | -94.36, 20.01 | 295.53, 80.91 | -72.98, -14.61 | in-in | in | 9.748 | Saltbr-in | 2.802 | HRD-in | -73.27, -48.07 | 68.78, 4.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.887 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.73, 163.63 | APE9-dihe-na | 71.35, 156.53 | APE8-dihe-in | -76.0, 150.02 | APE8-rot-out | 60.35 | APE67-dihe-in | -68.11, -15.2 | -46.02, -50.6 | APE12-dist-in | 12.749 | APE11-dist-in | 10.843 | APE10-dist-in | 6.32 | APE9-dist-in | 3.734 | None | None | None | XRAY | 1.96 | 0.201 | 0.241 | B | 355 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hyh | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHA | P68400 | 2 | 332 | 391.0 | 3NG:403,T9Y:404 | Type1,Allosteric | Inactive | DFGin | 7.383 | 16.565 | BLAminus | -118.8, -178.34 | 55.59, 76.92 | -97.73, 18.91 | 299.34, 78.81 | -65.83, -13.05 | in-in | in | 9.827 | Saltbr-in | 2.873 | HRD-in | -78.42, -45.3 | 64.02, 17.48 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.872 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.04, 164.88 | APE9-dihe-na | 65.11, 156.36 | APE8-dihe-in | -63.07, 152.22 | APE8-rot-out | 172.82 | APE67-dihe-in | -64.56, -17.94 | -58.04, -42.17 | APE12-dist-in | 12.698 | APE11-dist-in | 10.421 | APE10-dist-in | 6.18 | APE9-dist-in | 3.364 | None | None | None | XRAY | 2.07 | 0.216 | 0.256 | A | 355 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hzh | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 9HZHB | P68400 | 2 | 332 | 391.0 | 3NG:403,T9Y:404 | Type1,Allosteric | Inactive | DFGin | 7.368 | 16.552 | BLAminus | -119.62, -176.75 | 54.5, 77.97 | -98.25, 23.82 | 298.23, 80.81 | -69.92, -15.41 | in-in | in | 9.779 | Saltbr-in | 2.81 | HRD-in | -71.72, -44.22 | 63.92, 15.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.979 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.6, 164.83 | APE9-dihe-na | 66.55, 154.43 | APE8-dihe-in | -63.65, 152.11 | APE8-rot-out | 176.37 | APE67-dihe-in | -67.11, -13.32 | -56.47, -43.99 | APE12-dist-in | 12.789 | APE11-dist-in | 10.774 | APE10-dist-in | 6.319 | APE9-dist-in | 3.485 | None | None | None | XRAY | 2.07 | 0.216 | 0.256 | B | 355 | 331 | 0 | 0 | 0 | 0 | [[39, 324]] | 1.0 | 9hzh | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 1.6e-69 | 240.3 | 1 | 301 | 301 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A2 | CSK22_HUMAN | 8QBUA | P19784 | 6 | 333 | 350.0 | 42J:404,3NG:405 | Allosteric,Type1 | Inactive | DFGin | 7.481 | 16.117 | BLAminus | -115.34, 177.54 | 56.37, 76.99 | -87.29, 16.84 | 296.65, 81.34 | -70.83, -16.25 | in-in | in | 9.243 | Saltbr-in | 2.767 | HRD-in | -74.29, -50.68 | 73.5, 10.15 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.839 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -134.98, 166.78 | APE9-dihe-na | 65.99, 156.92 | APE8-dihe-in | -70.01, 146.12 | APE8-rot-out | 159.04 | APE67-dihe-in | -73.31, -10.45 | -44.42, -45.9 | APE12-dist-in | 12.462 | APE11-dist-in | 10.009 | APE10-dist-in | 6.107 | APE9-dist-in | 3.241 | C336S | None | None | XRAY | 1.09 | 0.16 | 0.179 | A | 364 | 328 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 8qbu | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1e-69 | 241.0 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9IHIA | P19784 | 7 | 333 | 350.0 | SY4:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.415 | 16.026 | BLAminus | -114.42, 178.99 | 58.97, 77.48 | -92.68, 17.89 | 295.72, 83.62 | -70.78, -17.6 | in-in | in | 9.166 | Saltbr-in | 2.815 | HRD-in | -75.11, -48.36 | 72.21, 10.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.841 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.76, 169.32 | APE9-dihe-na | 65.88, 158.62 | APE8-dihe-in | -76.33, 145.23 | APE8-rot-out | 154.92 | APE67-dihe-in | -68.36, -16.5 | -40.48, -52.03 | APE12-dist-in | 12.783 | APE11-dist-in | 10.506 | APE10-dist-in | 6.283 | APE9-dist-in | 3.236 | C336S | None | None | XRAY | 1.23 | 0.136 | 0.166 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9ihi | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9BA | P19784 | 7 | 333 | 350.0 | VN9:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.47 | 16.135 | BLAminus | -114.78, -178.63 | 52.36, 80.6 | -90.66, 23.03 | 297.12, 80.84 | -72.97, -19.45 | in-in | in | 9.164 | Saltbr-in | 2.851 | HRD-in | -75.12, -49.8 | 73.87, 8.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.899 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -131.85, 168.61 | APE9-dihe-na | 65.18, 157.14 | APE8-dihe-in | -73.48, 146.48 | APE8-rot-out | 146.34 | APE67-dihe-in | -70.57, -17.74 | -39.27, -49.01 | APE12-dist-in | 12.665 | APE11-dist-in | 10.424 | APE10-dist-in | 6.226 | APE9-dist-in | 3.23 | C336S | None | None | XRAY | 1.84 | 0.168 | 0.206 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9q9b | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QB6A | P19784 | 7 | 333 | 350.0 | RDV:401,3NG:402 | Allosteric,Type1 | Inactive | DFGin | 7.4 | 16.015 | BLAminus | -116.09, 178.07 | 58.12, 76.49 | -88.07, 15.69 | 297.72, 81.25 | -71.25, -16.82 | in-in | in | 9.094 | Saltbr-in | 2.784 | HRD-in | -72.64, -51.36 | 73.74, 9.54 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.862 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.78, 169.18 | APE9-dihe-na | 62.18, 162.55 | APE8-dihe-in | -82.53, 146.39 | APE8-rot-out | 147.47 | APE67-dihe-in | -70.59, -14.66 | -39.2, -52.96 | APE12-dist-in | 12.702 | APE11-dist-in | 10.373 | APE10-dist-in | 6.226 | APE9-dist-in | 3.212 | C336S | None | None | XRAY | 1.05 | 0.127 | 0.144 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9qb6 | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QABA | P19784 | 7 | 333 | 350.0 | RA7:401,3NG:402,RA7:403 | Allosteric,Type1,Allosteric | Inactive | DFGin | 7.376 | 16.117 | BLAminus | -113.6, 178.31 | 57.83, 77.52 | -90.77, 14.85 | 296.13, 81.67 | -69.28, -17.99 | in-in | in | 9.175 | Saltbr-in | 2.76 | HRD-in | -72.54, -50.49 | 72.75, 9.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.902 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.24, 170.06 | APE9-dihe-na | 64.96, 162.68 | APE8-dihe-in | -81.37, 147.07 | APE8-rot-out | 150.87 | APE67-dihe-in | -69.81, -15.24 | -39.22, -53.5 | APE12-dist-in | 12.716 | APE11-dist-in | 10.351 | APE10-dist-in | 6.227 | APE9-dist-in | 3.188 | C336S | None | None | XRAY | 0.95 | 0.131 | 0.141 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9qab | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 6HMBA | P19784 | 7 | 334 | 350.0 | 3NG:413 | Type1 | Inactive | DFGin | 7.526 | 16.135 | BLAminus | -111.55, 174.56 | 58.24, 78.46 | -87.65, 16.17 | 297.85, 81.04 | -69.02, -17.39 | in-in | in | 9.184 | Saltbr-in | 2.771 | HRD-in | -73.83, -48.37 | 71.6, 10.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.872 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -135.43, 166.43 | APE9-dihe-na | 65.52, 156.91 | APE8-dihe-in | -69.62, 146.48 | APE8-rot-out | 153.38 | APE67-dihe-in | -70.99, -14.32 | -39.92, -51.06 | APE12-dist-in | 12.572 | APE11-dist-in | 10.14 | APE10-dist-in | 6.125 | APE9-dist-in | 3.269 | C336S | None | None | XRAY | 1.04 | 0.135 | 0.146 | A | 364 | 328 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 6hmb | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1e-69 | 241.0 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9HK5A | P19784 | 7 | 334 | 350.0 | 3NG:402 | Type1 | Inactive | DFGin | 7.542 | 16.208 | BLAminus | -114.65, -179.29 | 53.64, 80.01 | -92.35, 20.62 | 296.39, 82.42 | -74.28, -17.08 | in-in | in | 9.271 | Saltbr-in | 2.826 | HRD-in | -73.22, -49.09 | 72.9, 4.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.899 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -134.78, 167.23 | APE9-dihe-na | 62.78, 157.39 | APE8-dihe-in | -75.16, 149.06 | APE8-rot-out | 147.29 | APE67-dihe-in | -68.84, -16.32 | -43.13, -50.25 | APE12-dist-in | 12.694 | APE11-dist-in | 10.358 | APE10-dist-in | 6.315 | APE9-dist-in | 3.288 | P32V,V83I,T101I,C336S | None | None | XRAY | 1.491 | 0.175 | 0.204 | A | 364 | 328 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9hk5 | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 3.1e-70 | 242.7 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9AA | P19784 | 7 | 333 | 350.0 | 3NG:401,A1I4V:402 | Type1,Allosteric | Inactive | DFGin | 7.397 | 16.171 | BLAminus | -114.27, 179.87 | 56.61, 76.76 | -86.69, 17.58 | 298.08, 81.74 | -71.41, -19.01 | in-in | in | 9.247 | Saltbr-in | 2.776 | HRD-in | -75.92, -48.72 | 71.51, 10.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.902 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -131.5, 165.78 | APE9-dihe-na | 68.3, 154.64 | APE8-dihe-in | -67.27, 146.08 | APE8-rot-out | 156.93 | APE67-dihe-in | -69.44, -15.07 | -43.26, -49.96 | APE12-dist-in | 12.724 | APE11-dist-in | 10.389 | APE10-dist-in | 6.234 | APE9-dist-in | 3.275 | C336S | None | None | XRAY | 1.03 | 0.147 | 0.156 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9q9a | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9Q9DA | P19784 | 7 | 332 | 350.0 | 3NG:401,R9G:402 | Type1,Allosteric | Inactive | DFGin | 7.413 | 16.113 | BLAminus | -111.11, 176.5 | 58.97, 76.86 | -90.38, 17.87 | 296.15, 81.91 | -69.6, -18.64 | in-in | in | 9.215 | Saltbr-in | 2.79 | HRD-in | -72.74, -49.53 | 71.25, 10.86 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.74, 169.32 | APE9-dihe-na | 66.15, 161.19 | APE8-dihe-in | -81.94, 147.26 | APE8-rot-out | 152.61 | APE67-dihe-in | -69.62, -15.68 | -40.15, -53.5 | APE12-dist-in | 12.735 | APE11-dist-in | 10.379 | APE10-dist-in | 6.221 | APE9-dist-in | 3.183 | C336S | None | None | XRAY | 0.89 | 0.148 | 0.159 | A | 370 | 326 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9q9d | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | CSNK2A2 | CSK22_HUMAN | 9QAGA | P19784 | 7 | 333 | 350.0 | 3NG:401,RBJ:402 | Type1,Allosteric | Inactive | DFGin | 7.402 | 16.146 | BLAminus | -113.78, 178.8 | 55.06, 77.97 | -89.73, 16.81 | 296.32, 81.5 | -70.74, -16.11 | in-in | in | 9.239 | Saltbr-in | 2.765 | HRD-in | -72.83, -48.69 | 70.11, 10.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.868 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.87, 167.19 | APE9-dihe-na | 64.82, 157.5 | APE8-dihe-in | -76.42, 146.88 | APE8-rot-out | 148.1 | APE67-dihe-in | -71.68, -14.1 | -39.59, -52.28 | APE12-dist-in | 12.68 | APE11-dist-in | 10.313 | APE10-dist-in | 6.249 | APE9-dist-in | 3.264 | C336S | None | None | XRAY | 1.01 | 0.136 | 0.162 | A | 370 | 327 | 0 | 0 | 0 | 0 | [[40, 325]] | 1.0 | 9qag | Homo sapiens | CMGC_CSNK2A2_HUMAN | CMGC | 1.1e-69 | 240.9 | 1 | 301 | 301 | 175 | 176 | 177 | 179 | 181 | 69 | 82 | 86 | 154 | 156 | 155 | 157 | 215 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 115 | Casein kinase II subunit alpha' |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NA | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.332 | 14.774 | BLAminus | -125.89, 175.46 | 60.34, 76.96 | -90.72, 25.89 | 277.64, 75.8 | -70.85, -23.55 | in-in | in | 8.867 | Saltbr-in | 2.627 | HRD-in | -70.94, -45.64 | 77.0, -3.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.65, -35.2 | APE9-dihe-na | -94.12, 169.14 | APE8-dihe-in | -81.45, 135.48 | APE8-rot-in | 271.72 | APE67-dihe-in | -57.78, -21.85 | -42.59, -54.66 | APE12-dist-in | 12.682 | APE11-dist-in | 11.088 | APE10-dist-in | 6.808 | APE9-dist-in | 3.373 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | A | 370 | 346 | 0 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NB | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 6.965 | 15.03 | BLAminus | -121.53, 177.86 | 59.36, 74.88 | -91.0, 24.04 | 284.65, 79.36 | -69.42, -6.51 | in-in | in | 9.072 | Saltbr-in | 2.955 | HRD-in | -65.31, -40.72 | 67.91, 3.75 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.837 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.86, 165.14 | APE9-dihe-na | 70.53, 140.66 | APE8-dihe-in | -62.36, 145.8 | APE8-rot-in | 271.48 | APE67-dihe-in | -55.51, -24.3 | -55.08, -48.98 | APE12-dist-in | 12.652 | APE11-dist-in | 11.24 | APE10-dist-in | 7.392 | APE9-dist-in | 3.193 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | B | 370 | 343 | 3 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NC | Q13627 | 134 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.125 | 14.845 | BLAminus | -127.45, -179.8 | 54.81, 79.63 | -96.7, 25.59 | 287.09, 79.21 | -71.97, -4.29 | in-in | in | 9.218 | Saltbr-in | 2.931 | HRD-in | -65.84, -47.16 | 77.48, 0.17 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.941 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -121.48, 175.3 | APE9-dihe-na | 70.69, 141.68 | APE8-dihe-in | -71.86, 144.08 | APE8-rot-in | 308.65 | APE67-dihe-in | -60.2, -32.88 | -49.5, -49.8 | APE12-dist-in | 13.034 | APE11-dist-in | 11.534 | APE10-dist-in | 7.148 | APE9-dist-in | 3.171 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | C | 370 | 344 | 3 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5ND | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.13 | 14.89 | BLAminus | -128.02, 175.09 | 60.57, 71.33 | -86.84, 26.43 | 281.73, 81.64 | -75.1, -14.91 | in-in | in | 9.081 | Saltbr-in | 2.672 | HRD-in | -60.22, -35.39 | 67.3, 3.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.821 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -92.57, 171.93 | APE9-dihe-na | 66.97, 156.51 | APE8-dihe-in | -85.5, 144.03 | APE8-rot-in | 283.59 | APE67-dihe-in | -57.76, -18.64 | -49.19, -52.69 | APE12-dist-in | 12.39 | APE11-dist-in | 10.732 | APE10-dist-in | 7.111 | APE9-dist-in | 3.042 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | D | 370 | 338 | 8 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NE | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.188 | 14.841 | BLAminus | -123.41, -179.95 | 58.6, 74.9 | -91.66, 28.87 | 284.52, 74.3 | -74.18, -15.86 | in-in | in | 8.932 | Saltbr-in | 2.599 | HRD-in | -66.53, -45.73 | 70.01, 6.86 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.729 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.5, 169.99 | APE9-dihe-na | 69.78, 136.41 | APE8-dihe-in | -57.94, 135.93 | APE8-rot-in | 298.8 | APE67-dihe-in | -52.87, -33.29 | -49.91, -51.82 | APE12-dist-in | 12.549 | APE11-dist-in | 11.378 | APE10-dist-in | 7.325 | APE9-dist-in | 3.185 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | E | 370 | 340 | 6 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NF | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.268 | 14.5 | BLAminus | -134.01, 179.07 | 56.51, 71.89 | -90.03, 23.99 | 289.58, 70.49 | -65.64, -23.07 | in-in | in | 9.224 | Saltbr-in | 2.867 | HRD-in | -69.65, -42.1 | 76.58, -5.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.88, -177.32 | APE9-dihe-na | 69.42, 90.94 | APE8-dihe-in | -27.36, 123.58 | APE8-rot-in | 265.98 | APE67-dihe-in | -50.43, -31.45 | -50.21, -44.01 | APE12-dist-in | 13.065 | APE11-dist-in | 11.252 | APE10-dist-in | 6.846 | APE9-dist-in | 3.171 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | F | 370 | 346 | 0 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NG | Q13627 | 137 | 480 | 763.0 | 3NG:501 | Type1 | Active | DFGin | 7.344 | 14.781 | BLAminus | -131.27, 177.34 | 58.91, 64.55 | -81.55, 37.12 | 289.02, 78.81 | -81.79, -16.85 | in-in | in | 8.979 | Saltbr-in | 2.629 | HRD-in | -65.23, -49.26 | 77.2, 4.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.719 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.89, 64.11 | APE9-dihe-na | -161.3, 162.4 | APE8-dihe-in | -70.8, 130.74 | APE8-rot-in | 279.54 | APE67-dihe-in | -57.11, -25.99 | -52.9, -46.96 | APE12-dist-in | 12.712 | APE11-dist-in | 11.544 | APE10-dist-in | 6.759 | APE9-dist-in | 3.418 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | G | 370 | 333 | 11 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 7Z5NH | Q13627 | 135 | 480 | 763.0 | 3NG:501 | Type1 | None | DFGin | 6.679 | 14.847 | BLAminus | -128.66, -179.58 | 53.82, 77.25 | -93.05, 20.83 | 280.85, 75.88 | -63.97, -13.6 | in-in | in | 9.075 | Saltbr-in | 3.001 | HRD-in | -63.15, -47.83 | 74.92, 6.9 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.799 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_niii | APE10-dihe-na | -156.21, 166.85 | APE9-dihe-na | 64.29, 161.67 | APE8-dihe-in | -89.72, 140.84 | APE8-rot-none | 999.0 | APE67-dihe-in | -54.39, -32.97 | -48.02, -56.25 | APE12-dist-none | 999.0 | APE11-dist-in | 10.614 | APE10-dist-in | 7.767 | APE9-dist-in | 3.208 | None | PTR321 | PTR321 | XRAY | 2.77 | 0.207 | 0.252 | H | 370 | 307 | 39 | 0 | 0 | 4 | [[159, 479]] | 1.0 | 7z5n | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 9.2e-91 | 310.1 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FA | P49841 | 28 | 383 | 420.0 | 3NG:60401 | Type1 | Inactive | DFGin | 7.172 | 14.387 | BLAminus | -140.61, -172.17 | 56.83, 67.31 | -90.44, 24.59 | 283.96, 78.9 | -70.58, -34.2 | in-in | in | 8.589 | Saltbr-in | 2.706 | HRD-in | -70.71, -48.08 | 68.23, 20.67 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.877 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -121.77, -56.1 | APE9-dihe-na | -73.95, 173.6 | APE8-dihe-in | -71.54, 133.95 | APE8-rot-out | 205.24 | APE67-dihe-in | -54.78, -22.55 | -52.86, -47.6 | APE12-dist-in | 13.711 | APE11-dist-in | 11.921 | APE10-dist-in | 7.257 | APE9-dist-in | 3.478 | None | PTR216 | PTR216 | XRAY | 3.0 | 0.224 | 0.249 | A | 364 | 354 | 2 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 7z1f | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.5 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1FB | P49841 | 38 | 382 | 420.0 | 3NG:60401 | Type1 | Inactive | DFGin | 6.87 | 14.469 | BLAminus | -141.12, -171.82 | 52.8, 73.11 | -90.49, 20.89 | 285.47, 81.84 | -62.59, -35.1 | in-in | in | 9.025 | Saltbr-in | 2.763 | HRD-in | -68.41, -52.97 | 70.54, 14.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.039 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -122.34, -53.99 | APE9-dihe-na | -75.88, 165.71 | APE8-dihe-in | -64.92, 136.76 | APE8-rot-out | 179.7 | APE67-dihe-in | -58.44, -19.64 | -54.95, -47.33 | APE12-dist-in | 13.527 | APE11-dist-in | 11.859 | APE10-dist-in | 7.154 | APE9-dist-in | 3.558 | None | PTR216 | PTR216 | XRAY | 3.0 | 0.224 | 0.249 | B | 364 | 321 | 24 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 7z1f | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.5 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | GSK3B | GSK3B_HUMAN | 7Z1GA | P49841 | 27 | 383 | 420.0 | 3NG:60401 | Type1 | Active | DFGin | 7.272 | 14.699 | BLAminus | -137.45, -179.93 | 52.32, 81.51 | -93.1, 20.22 | 282.75, 78.65 | -65.74, -16.48 | in-in | in | 8.969 | Saltbr-in | 2.771 | HRD-in | -67.62, -47.44 | 74.98, 2.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.926 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -86.67, 177.94 | APE9-dihe-na | 70.81, 142.84 | APE8-dihe-in | -95.23, 170.55 | APE8-rot-in | 305.08 | APE67-dihe-inflip | 72.5, -37.64 | -53.01, 158.1 | APE12-dist-in | 12.785 | APE11-dist-in | 10.847 | APE10-dist-in | 5.858 | APE9-dist-in | 2.984 | None | None | None | XRAY | 2.85 | 0.204 | 0.228 | A | 364 | 355 | 2 | 0 | 0 | 0 | [[56, 340]] | 1.0 | 7z1g | Homo sapiens | CMGC_GSK3B_HUMAN | CMGC | 2e-70 | 243.5 | 1 | 301 | 301 | 199 | 200 | 201 | 203 | 205 | 85 | 97 | 101 | 178 | 180 | 179 | 181 | 239 | 226 | 221 | 220 | 219 | 218 | 217 | 216 | 215 | 133 | Glycogen synthase kinase-3 beta |
| CMGC | HIPK2 | HIPK2_HUMAN | 6P5SA | Q9H2X6 | 185 | 535 | 1198.0 | 3NG:601 | Type1 | Inactive | DFGin | 7.298 | 14.23 | BLAminus | -121.5, -179.79 | 64.91, 82.62 | -96.84, 22.58 | 294.47, 82.62 | -64.48, -30.53 | in-in | in | 8.971 | Saltbr-in | 2.761 | HRD-in | -77.76, -49.7 | 67.78, 8.12 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.639 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -113.93, 168.02 | APE9-dihe-na | 68.38, 155.05 | APE8-dihe-in | -77.17, 138.14 | APE8-rot-out | 185.94 | APE67-dihe-in | -61.16, -24.2 | -57.86, -43.21 | APE12-dist-in | 10.584 | APE11-dist-in | 11.105 | APE10-dist-in | 7.495 | APE9-dist-in | 3.243 | None | PTR361,SEP441 | PTR361,SEP441 | XRAY | 2.194 | 0.2 | 0.238 | A | 390 | 333 | 18 | 0 | 0 | 6 | [[199, 527]] | 1.0 | 6p5s | Homo sapiens | CMGC_HIPK2_HUMAN | CMGC | 2.6e-92 | 315.4 | 1 | 301 | 301 | 345 | 346 | 347 | 349 | 351 | 228 | 243 | 247 | 321 | 323 | 322 | 324 | 383 | 371 | 366 | 365 | 364 | 363 | 362 | 361 | 360 | 278 | Homeodomain-interacting protein kinase 2 |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CKA1 | J9VNH4_CRYN9 | 6K3LB | J9VNH4 | 5 | 333 | 338.0 | 3NG:401 | Type1 | Inactive | DFGin | 7.66 | 16.152 | BLAminus | -114.35, -178.61 | 52.93, 78.12 | -89.9, 16.79 | 294.15, 81.47 | -67.97, -25.55 | in-in | in | 9.075 | Saltbr-in | 2.706 | HRD-in | -76.39, -51.63 | 76.4, 5.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.822 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -126.48, 161.19 | APE9-dihe-na | 73.24, 164.99 | APE8-dihe-in | -76.46, 151.58 | APE8-rot-out | 148.39 | APE67-dihe-in | -65.37, -22.86 | -51.07, -48.56 | APE12-dist-in | 12.822 | APE11-dist-in | 10.511 | APE10-dist-in | 6.303 | APE9-dist-in | 3.403 | None | None | None | XRAY | 2.09 | 0.189 | 0.219 | B | 338 | 329 | 0 | 0 | 0 | 0 | [[38, 323]] | 1.0 | 6k3l | Cryptococcus neoformans | CMGC_CKA1_CRYN9 | CMGC | 6e-64 | 222.0 | 1 | 301 | 301 | 173 | 174 | 175 | 177 | 179 | 67 | 80 | 84 | 152 | 154 | 153 | 155 | 213 | 200 | 195 | 194 | 193 | 192 | 191 | 190 | 189 | 113 | Casein kinase II subunit alpha |