| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK14 | MK14_HUMAN | 3LFAA | Q16539 | 4 | 353 | 360.0 | 1N1:361 | Type1 | Inactive | None | 999.0 | 999.0 | None | -119.32, 169.35 | -154.54, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 9.2412 | Saltbr-in | 2.7349 | HRD-in | -67.55, -57.07 | 85.83, -16.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 157.05 | APE8-dihe-out | -85.63, -3.59 | APE8-rot-in | 346.34 | APE67-dihe-in | -59.81, -27.96 | -94.61, -12.54 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.8947 | None | None | None | XRAY | 2.1 | 0.204 | 0.254 | A | 360.0 | 333.0 | 17 | 25 | 10 | 15 | [[24, 308]] | 1.0 | 3lfa | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| OTHER | PKMYT1 | PMYT1_HUMAN | 5VCVA | Q99640 | 75 | 361 | 499.0 | 1N1:60404 | Type1 | Inactive | DFGin | 6.1731 | 14.4679 | BLAminus | -133.17, -164.16 | 53.7, 76.36 | -96.77, 22.58 | 298.04, 107.44 | -64.77, -25.22 | in-in | in | 8.9178 | Saltbr-in | 2.826 | HRD-in | -73.66, -44.65 | 68.1, -0.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8927 | ActLoopCT-out | nonTYR | APEdihe_aaiai | APEdist_iooi | APE10-dihe-na | -65.91, 159.0 | APE9-dihe-na | -91.66, -157.73 | APE8-dihe-in | -52.29, 123.12 | APE8-rot-na | 188.83 | APE67-dihe-in | -60.44, -30.04 | -60.97, -24.44 | APE12-dist-in | 7.9448 | APE11-dist-out | 6.4495 | APE10-dist-out | 9.0797 | APE9-dist-in | 3.1786 | None | TPO260 | TPO260 | XRAY | 1.92 | 0.157 | 0.197 | A | 311.0 | 287.0 | 0 | 27 | 27 | 0 | [[110, 359]] | 1.0 | 5vcv | OTHER_PKMYT1_HUMAN | STE | 9.9e-39 | 139.4 | 1.0 | 255.0 | 255.0 | 250 | 251 | 252 | 254 | 256 | 139 | 157 | 161 | 230 | 232 | 231 | 233.0 | 288 | 277 | 272 | 271 | 270 | 269 | 268 | 267 | 266 | 188 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| STE | STK10 | STK10_HUMAN | 5OWRA | O94804 | 23 | 317 | 968.0 | 1N1:401 | Type1 | Inactive | DFGin | 6.4982 | 16.7221 | BLAminus | -126.18, 173.2 | 57.39, 79.01 | -91.46, 24.21 | 286.72, 77.35 | -53.02, -57.95 | out-out | out | 10.2052 | Saltbr-out | 8.1359 | HRD-in | -70.96, -54.03 | 67.34, 13.9 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.8335 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -61.94, -27.24 | 999.0, -15.2 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.3 | 0.221 | 0.254 | A | 302.0 | 282.0 | 13 | 28 | 21 | 7 | [[36, 294]] | 1.0 | 5owr | STE_STK10_HUMAN | STE | 2e-94 | 321.6 | 1.0 | 257.0 | 257.0 | 174 | 175 | 176 | 178 | 180 | 65 | 81 | 85 | 154 | 156 | 155 | 157.0 | 219 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 111 | Serine/threonine-protein kinase 10 |
| STE | STK24 | STK24_HUMAN | 4QMSA | Q9Y6E0 | 27 | 310 | 443.0 | 1N1:60401 | Type1 | Inactive | DFGin | 7.0296 | 15.2785 | BLAminus | -133.65, 170.4 | 59.12, 88.65 | -100.44, 27.96 | 287.36, 78.03 | -60.48, -24.48 | in-out | in | 9.6308 | Saltbr-out | 4.5468 | HRD-in | -69.75, -48.6 | 69.83, 3.91 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.42, 162.17 | APE9-dihe-na | 128.43, -166.04 | APE8-dihe-in | -119.95, 120.69 | APE8-rot-in | 305.76 | APE67-dihe-in | -58.87, -30.57 | -46.04, -47.24 | APE12-dist-in | 8.2773 | APE11-dist-in | 10.9536 | APE10-dist-in | 5.1134 | APE9-dist-in | 3.3059 | None | TPO190 | TPO190 | XRAY | 1.883 | 0.169 | 0.214 | A | 310.0 | 284.0 | 0 | 28 | 28 | 0 | [[36, 286]] | 1.0 | 4qms | STE_STK24_HUMAN | STE | 3.9e-100 | 340.4 | 1.0 | 257.0 | 257.0 | 173 | 174 | 175 | 177 | 179 | 65 | 82 | 86 | 153 | 155 | 154 | 156.0 | 213 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 112 | Serine/threonine-protein kinase 24 |
| TYR | ABL1 | ABL1_HUMAN | 7N9GB | P00519 | 233 | 498 | 1130.0 | STI:60601,1N1:60602 | Allosteric,Type1 | Active | DFGin | 6.7541 | 13.4449 | BLAminus | -122.97, -168.58 | 58.54, 84.79 | -109.7, 15.38 | 305.77, 104.92 | -56.72, -36.19 | in-in | in | 7.8072 | Saltbr-in | 2.716 | HRD-in | -94.83, -54.73 | 76.06, 6.03 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0408 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -97.97, 124.86 | APE9-dihe-in | -118.42, 152.72 | APE8-dihe-in | -70.17, 95.62 | APE8-rot-na | 28.18 | APE67-dihe-in | -73.36, -13.19 | -53.92, -45.07 | APE12-dist-na | 14.9514 | APE11-dist-na | 10.1213 | APE10-dist-na | 12.2789 | APE9-dist-in | 7.1369 | None | None | None | XRAY | 2.2 | 0.219 | 0.251 | B | 271.0 | 264.0 | 2 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 7n9g | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2GQGA | P00519 | 229 | 500 | 1130.0 | 1N1:60501 | Type1 | Inactive | DFGin | 6.6367 | 14.0391 | BLAminus | -125.87, -162.48 | 50.1, 80.24 | -101.91, 13.59 | 304.08, 105.04 | -55.58, -28.07 | in-in | in | 8.2064 | Saltbr-in | 3.3367 | HRD-in | -94.17, -46.19 | 69.1, 8.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0889 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.45, -178.77 | APE9-dihe-in | -144.75, 146.99 | APE8-dihe-in | -51.41, 101.22 | APE8-rot-na | 30.18 | APE67-dihe-in | -72.33, -8.18 | -47.68, -48.27 | APE12-dist-na | 13.8069 | APE11-dist-na | 10.1551 | APE10-dist-na | 13.162 | APE9-dist-in | 7.0168 | None | PTR393 | PTR393 | XRAY | 2.4 | 0.208 | 0.273 | A | 278.0 | 272.0 | 0 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 2gqg | TYR_ABL1_HUMAN | TYR | 2.4e-100 | 341.1 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2GQGB | P00519 | 229 | 499 | 1130.0 | 1N1:60502 | Type1.5_Back | Active | DFGin | 6.7246 | 13.4066 | BLAminus | -132.96, -163.46 | 57.81, 75.2 | -98.78, 6.6 | 302.62, 104.4 | -52.45, -32.74 | in-in | in | 8.0337 | Saltbr-in | 2.8987 | HRD-in | -101.91, -48.31 | 65.85, 10.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9585 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -100.98, 171.69 | APE9-dihe-in | -137.71, 138.65 | APE8-dihe-in | -58.61, 114.78 | APE8-rot-na | 30.65 | APE67-dihe-in | -71.5, -8.45 | -53.53, -44.9 | APE12-dist-na | 11.2577 | APE11-dist-na | 7.468 | APE10-dist-na | 11.6413 | APE9-dist-in | 6.2756 | None | PTR393 | PTR393 | XRAY | 2.4 | 0.208 | 0.273 | B | 278.0 | 271.0 | 0 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 2gqg | TYR_ABL1_HUMAN | TYR | 2.4e-100 | 341.1 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 4XEYB | P00519 | 122 | 504 | 1130.0 | 1N1:60601 | Type1 | Inactive | DFGinter | 10.0007 | 8.0224 | BABtrans | -71.04, 121.63 | -84.68, 7.52 | -91.76, 101.26 | 207.86, 90.35 | 143.13, -1.76 | in-out | in | 8.918 | Saltbr-out | 8.6427 | HRD-out | -101.25, 126.15 | -79.9, -27.01 | out-out-in | SNCooi | out-in | ActLoopNT-out | 5.4222 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -80.63, 133.07 | APE9-dihe-in | -116.3, 152.74 | APE8-dihe-in | -66.44, 99.47 | APE8-rot-na | 21.89 | APE67-dihe-in | -71.31, -17.26 | -44.98, -48.3 | APE12-dist-na | 18.5596 | APE11-dist-na | 13.9233 | APE10-dist-na | 16.5485 | APE9-dist-in | 6.4285 | None | None | None | XRAY | 2.891 | 0.232 | 0.259 | B | 408.0 | 359.0 | 9 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 4xey | TYR_ABL1_HUMAN | TYR | 8.5e-100 | 339.5 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 7N9GA | P00519 | 233 | 498 | 1130.0 | STI:60601,1N1:60602 | Allosteric,Type1 | Inactive | DFGinter | 10.4212 | 8.1868 | None | -69.43, 136.44 | -123.08, 27.78 | -75.4, -30.96 | 178.85, 77.99 | -98.31, 50.2 | in-out | in | 8.8784 | Saltbr-out | 9.7861 | HRD-out | -92.88, 142.81 | -110.01, 0.88 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.5443 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 170.84 | APE8-dihe-in | -72.01, 95.09 | APE8-rot-na | 30.25 | APE67-dihe-in | -73.75, -10.66 | -54.08, -44.56 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.8503 | None | None | None | XRAY | 2.2 | 0.219 | 0.251 | A | 271.0 | 250.0 | 16 | 29 | 16 | 13 | [[242, 495]] | 1.0 | 7n9g | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 7N9GC | P00519 | 234 | 499 | 1130.0 | STI:60601,1N1:60602 | Allosteric,Type1 | Inactive | DFGinter | 10.016 | 7.7618 | None | -68.53, 140.81 | -120.26, 3.31 | -57.57, -42.4 | 182.82, 108.58 | -86.96, 40.71 | in-none | in | 9.4392 | Saltbr-none | 999.0 | HRD-out | -106.92, 134.12 | -80.26, -30.58 | none-out-none | SNCnon | out-none | ActLoopNT-out | 5.4779 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 96.82 | APE8-dihe-in | -65.53, 99.76 | APE8-rot-na | 23.57 | APE67-dihe-in | -73.61, -20.46 | -60.17, -42.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.8914 | None | None | None | XRAY | 2.2 | 0.219 | 0.251 | C | 271.0 | 233.0 | 33 | 29 | 24 | 5 | [[242, 495]] | 1.0 | 7n9g | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 4XEYA | P00519 | 231 | 503 | 1130.0 | 1N1:60601 | Type1 | Inactive | DFGinter | 9.993 | 7.9273 | None | -70.89, 123.51 | -90.91, 18.27 | -87.3, -11.95 | 199.48, 77.0 | -96.54, 13.69 | in-out | in | 8.9479 | Saltbr-out | 8.6903 | HRD-out | -101.8, 125.8 | -78.66, -28.68 | out-out-in | SNCooi | out-in | ActLoopNT-out | 5.3933 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.59, 140.17 | APE9-dihe-in | -145.27, 142.92 | APE8-dihe-in | -62.13, 98.18 | APE8-rot-na | 23.13 | APE67-dihe-in | -73.29, -19.48 | -49.65, -41.78 | APE12-dist-na | 18.7302 | APE11-dist-na | 14.1077 | APE10-dist-na | 16.5419 | APE9-dist-in | 6.5879 | None | None | None | XRAY | 2.891 | 0.232 | 0.259 | A | 408.0 | 269.0 | 4 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 4xey | TYR_ABL1_HUMAN | TYR | 8.5e-100 | 339.5 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | BMX | BMX_HUMAN | 3SXRA | P51813 | 411 | 671 | 675.0 | 1N1:60001 | Type1 | Inactive | DFGinter | 7.8824 | 8.1671 | BABtrans | -93.57, 121.18 | -103.19, -9.04 | -51.22, 114.45 | 184.77, 74.21 | 62.74, 18.94 | out-out | out | 10.805 | Saltbr-out | 7.5586 | HRD-out | -99.0, 124.02 | -80.22, -7.53 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8353 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -95.14, 119.04 | APE9-dihe-in | -94.0, 160.01 | APE8-dihe-in | -48.96, 127.48 | APE8-rot-na | 331.52 | APE67-dihe-in | -68.66, -11.59 | -65.07, -24.25 | APE12-dist-na | 10.0286 | APE11-dist-na | 7.5492 | APE10-dist-na | 12.0421 | APE9-dist-in | 5.1857 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | A | 268.0 | 257.0 | 4 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 3SXRB | P51813 | 411 | 671 | 675.0 | 1N1:60002 | Type1 | Inactive | DFGinter | 7.7085 | 8.2724 | BABtrans | -92.79, 121.27 | -96.68, -12.13 | -49.05, 115.54 | 186.98, 71.37 | 61.78, 19.24 | out-out | out | 10.8028 | Saltbr-out | 8.0973 | HRD-out | -100.92, 124.05 | -80.64, -7.7 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8449 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.81, 125.57 | APE9-dihe-in | -101.37, 158.16 | APE8-dihe-in | -49.48, 128.1 | APE8-rot-na | 332.21 | APE67-dihe-in | -66.79, -11.14 | -62.63, -27.73 | APE12-dist-na | 9.9457 | APE11-dist-na | 7.4465 | APE10-dist-na | 11.9437 | APE9-dist-in | 5.1904 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | B | 268.0 | 255.0 | 6 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BTK | BTK_HUMAN | 3K54A | Q06187 | 392 | 658 | 659.0 | 1N1:1 | Type1 | Inactive | DFGin | 4.6816 | 13.9981 | BLAplus | -132.68, -179.17 | 50.27, 30.98 | -93.41, -0.42 | 58.12, 86.77 | -82.65, 999.0 | in-out | in | 8.7866 | Saltbr-out | 3.7709 | HRD-in | -69.54, -47.61 | 72.38, -12.01 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 136.06 | APE8-dihe-in | -84.11, 69.82 | APE8-rot-na | 29.89 | APE67-dihe-in | -70.22, -9.36 | -47.67, -47.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.1055 | Y551E | None | None | XRAY | 1.94 | 0.202 | 0.258 | A | 283.0 | 243.0 | 24 | 29 | 12 | 17 | [[402, 653]] | 1.0 | 3k54 | TYR_BTK_HUMAN | TYR | 1.6e-92 | 315.4 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 3OCTA | Q06187 | 394 | 656 | 659.0 | 1N1:663 | Type1 | Inactive | DFGinter | 9.5513 | 8.0475 | BABtrans | -83.49, 139.01 | -103.95, 15.92 | -87.02, 132.92 | 181.28, 97.3 | 77.87, 26.97 | in-out | in | 9.203 | Saltbr-out | 7.7453 | HRD-in | -70.28, -48.13 | 67.57, -13.36 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.3805 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 95.42 | APE8-dihe-in | -60.66, 106.57 | APE8-rot-na | 28.18 | APE67-dihe-in | -77.0, -13.84 | -55.35, -41.2 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.7096 | V555R | None | None | XRAY | 1.95 | 0.199 | 0.251 | A | 265.0 | 244.0 | 19 | 29 | 15 | 14 | [[402, 653]] | 1.0 | 3oct | TYR_BTK_HUMAN | TYR | 2.3e-93 | 318.2 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | DDR1 | DDR1_HUMAN | 6BSDA | Q08345 | 604 | 912 | 913.0 | 1N1:60901 | Type1 | Inactive | DFGinter | 9.9484 | 9.844 | None | -87.87, 155.34 | -64.16, -24.42 | 174.69, 170.82 | 68.3, 89.44 | 55.93, 999.0 | in-in | in | 8.3705 | Saltbr-in | 2.7354 | HRD-in | -61.68, -56.93 | 83.98, -4.33 | in-out-in | SNCioi | out-in | ActLoopNT-out | 19.8476 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -66.74, 115.57 | APE9-dihe-in | -116.16, 127.65 | APE8-dihe-in | -81.76, 68.68 | APE8-rot-na | 34.21 | APE67-dihe-in | -66.93, -20.25 | -61.43, -30.39 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.1458 | None | None | None | XRAY | 2.606 | 0.186 | 0.255 | A | 351.0 | 278.0 | 31 | 30 | 28 | 2 | [[610, 907]] | 1.0 | 6bsd | TYR_DDR1_HUMAN | TYR | 2.3e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 5BVWA | Q08345 | 604 | 911 | 913.0 | 1N1:1009 | Type1 | Inactive | DFGout | 14.538 | 10.296 | None | -113.16, 175.58 | -102.37, -21.68 | 40.34, 118.5 | 221.24, 85.03 | -134.54, 999.0 | in-in | in | 8.3337 | Saltbr-in | 2.775 | HRD-in | -77.35, -46.96 | 73.51, -12.24 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -79.96, 123.56 | APE9-dihe-in | -122.26, 123.59 | APE8-dihe-in | -77.84, 65.49 | APE8-rot-na | 31.29 | APE67-dihe-in | -69.31, -14.79 | -54.53, -34.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.409 | None | None | None | XRAY | 1.94 | 0.186 | 0.234 | A | 324.0 | 274.0 | 34 | 30 | 26 | 4 | [[610, 907]] | 1.0 | 5bvw | TYR_DDR1_HUMAN | TYR | 1.7e-92 | 315.4 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | EPHA2 | EPHA2_HUMAN | 5I9YA | P29317 | 600 | 896 | 976.0 | 1N1:1001 | Type1 | Inactive | DFGin | 6.2223 | 14.973 | BLBminus | -129.12, 177.86 | 73.14, 77.74 | -114.09, 153.37 | 295.9, 102.04 | 147.64, -171.81 | in-in | in | 8.2568 | Saltbr-in | 2.7741 | HRD-in | -75.07, -47.16 | 76.83, -16.24 | in-out-none | SNCion | out-none | ActLoopNT-out | 10.4586 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 139.34 | APE8-rot-na | 36.16 | APE67-dihe-in | -79.28, -3.2 | -53.92, -45.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.228 | 0.164 | 0.179 | A | 306.0 | 287.0 | 10 | 31 | 24 | 7 | [[613, 873]] | 1.0 | 5i9y | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHB4 | EPHB4_HUMAN | 6FNMA | P54760 | 608 | 889 | 987.0 | 1N1:1001 | Type1 | Inactive | DFGin | 5.9609 | 15.7692 | BLBminus | -128.55, -169.2 | 67.78, 75.65 | -110.02, 138.75 | 293.26, 98.41 | 179.12, 146.16 | in-in | in | 8.3255 | Saltbr-in | 3.1793 | HRD-in | -76.03, -51.54 | 81.54, -15.45 | in-out-in | SNCioi | out-in | ActLoopNT-out | 10.0097 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.65, 157.69 | APE9-dihe-in | -64.87, 128.21 | APE8-dihe-in | -78.96, 90.14 | APE8-rot-na | 30.03 | APE67-dihe-in | -61.19, -22.58 | -57.17, -48.0 | APE12-dist-na | 999.0 | APE11-dist-na | 11.3678 | APE10-dist-na | 15.0342 | APE9-dist-in | 6.5764 | Y774E,A803V,V870I | None | None | XRAY | 1.157 | 0.184 | 0.195 | A | 297.0 | 270.0 | 12 | 33 | 21 | 12 | [[615, 876]] | 1.0 | 6fnm | TYR_EPHB4_HUMAN | TYR | 4.2e-105 | 356.7 | 2.0 | 261.0 | 260.0 | 757 | 758 | 759 | 761 | 763 | 647 | 664 | 668 | 737 | 739 | 738 | 740.0 | 802 | 790 | 785 | 784 | 783 | 782 | 781 | 780 | 779 | 694 | Ephrin type-B receptor 4 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UA | Q13882 | 185 | 446 | 451.0 | 1N1:60501 | Type1 | Inactive | DFGin | 5.9983 | 13.4628 | BLBplus | -115.66, 172.2 | 65.44, 13.7 | -58.08, 130.19 | 47.49, 85.54 | 66.94, -1.55 | out-out | out | 14.1683 | Saltbr-out | 16.091 | HRD-in | -72.57, -54.48 | 85.53, -13.44 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.2608 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 72.03, 33.67 | APE9-dihe-out | -55.65, -32.62 | APE8-dihe-out | -63.18, -18.16 | APE8-rot-na | 340.69 | APE67-dihe-in | -82.41, -18.93 | -56.57, -27.65 | APE12-dist-na | 16.3439 | APE11-dist-na | 20.6081 | APE10-dist-na | 18.2629 | APE9-dist-out | 11.0621 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | A | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UB | Q13882 | 185 | 446 | 451.0 | 1N1:60501 | Type1 | Inactive | DFGin | 6.0808 | 13.3427 | BLBplus | -112.62, 168.56 | 69.96, 13.64 | -58.15, 126.09 | 44.9, 88.52 | 70.74, 0.77 | out-out | out | 14.3036 | Saltbr-out | 15.9567 | HRD-in | -65.56, -52.22 | 84.8, -15.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0671 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 67.1, 31.04 | APE9-dihe-out | -51.48, -32.62 | APE8-dihe-out | -56.92, -21.84 | APE8-rot-na | 331.92 | APE67-dihe-in | -82.05, -11.15 | -61.67, -25.37 | APE12-dist-na | 16.2609 | APE11-dist-na | 20.2262 | APE10-dist-na | 17.9045 | APE9-dist-out | 11.0552 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | B | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UC | Q13882 | 185 | 446 | 451.0 | 1N1:60501 | Type1 | Inactive | DFGin | 5.9677 | 13.6341 | BLBplus | -101.49, 165.12 | 71.33, 11.9 | -56.7, 126.68 | 46.28, 85.99 | 72.45, -1.55 | out-out | out | 14.2504 | Saltbr-out | 15.3617 | HRD-in | -69.3, -53.89 | 83.99, -9.53 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.1583 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 66.45, 29.68 | APE9-dihe-out | -47.22, -37.04 | APE8-dihe-out | -58.56, -24.03 | APE8-rot-na | 334.48 | APE67-dihe-in | -84.14, -9.31 | -53.24, -25.76 | APE12-dist-na | 16.3889 | APE11-dist-na | 20.3117 | APE10-dist-na | 17.9592 | APE9-dist-out | 11.0174 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | C | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UD | Q13882 | 185 | 446 | 451.0 | 1N1:60504 | Type1 | Inactive | DFGin | 6.1814 | 13.2695 | BLBplus | -112.73, 164.13 | 73.65, 11.67 | -56.94, 123.73 | 42.41, 88.79 | 73.17, 2.96 | out-out | out | 14.0107 | Saltbr-out | 15.9929 | HRD-in | -70.19, -55.11 | 88.71, -18.22 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.1947 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 72.07, 30.74 | APE9-dihe-out | -48.72, -36.76 | APE8-dihe-out | -61.03, -20.74 | APE8-rot-na | 334.99 | APE67-dihe-in | -84.77, -13.01 | -55.36, -26.11 | APE12-dist-na | 16.3004 | APE11-dist-na | 20.346 | APE10-dist-na | 18.0251 | APE9-dist-out | 11.0324 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | D | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|---|---|---|---|
| DFGin | BLAminus | 13 | 37.1% | 4QMSA |
| DFGinter | BABtrans | 6 | 17.1% | 3SXRA |
| DFGin | BLBplus | 4 | 11.4% | 5H2UA |
| DFGinter | None | 4 | 11.4% | 4XEYA |
| DFGout | None | 3 | 8.6% | 3OHTA |
| DFGin | BLBminus | 2 | 5.7% | 5I9YA |
| DFGin | BLAplus | 1 | 2.9% | 3K54A |
| DFGin | None | 1 | 2.9% | 2Y6OA |
| None | None | 1 | 2.9% | 3LFAA |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SRC | SRC_CHICK | 3QLGA | P00523 | 258 | 533 | 533.0 | 1N1:601 | Type1.5_Back | Inactive | DFGin | 6.5502 | 13.8381 | BLAminus | -128.97, 169.0 | 62.45, 93.12 | -106.99, 6.4 | 306.69, 101.34 | -122.4, 999.0 | in-in | in | 8.7224 | Saltbr-in | 2.9531 | HRD-in | -90.7, -55.87 | 92.28, -19.25 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 140.4 | APE8-dihe-in | -85.59, 52.69 | APE8-rot-na | 6.03 | APE67-dihe-in | -68.2, -8.8 | -50.34, -41.04 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.1548 | L317I | None | None | XRAY | 2.75 | 0.203 | 0.269 | A | 286.0 | 259.0 | 17 | 29 | 12 | 17 | [[267, 518]] | 1.0 | 3qlg | Gallus gallus | TYR_SRC_CHICK | TYR | 7e-94 | 319.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 3QLGB | P00523 | 256 | 533 | 533.0 | 1N1:601 | Type1.5_Back | Inactive | DFGin | 6.2634 | 13.1722 | BLAminus | -132.53, 169.92 | 55.67, 96.64 | -114.48, 23.35 | 323.76, 73.27 | -64.65, -16.14 | in-in | in | 8.523 | Saltbr-in | 2.7156 | HRD-in | -89.78, -56.21 | 92.27, -19.49 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.1877 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 135.14 | APE8-dihe-in | -84.28, 53.37 | APE8-rot-na | 5.94 | APE67-dihe-in | -68.54, -8.95 | -50.64, -40.54 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.0573 | L317I | None | None | XRAY | 2.75 | 0.203 | 0.269 | B | 286.0 | 260.0 | 18 | 29 | 16 | 13 | [[267, 518]] | 1.0 | 3qlg | Gallus gallus | TYR_SRC_CHICK | TYR | 7e-94 | 319.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 3G5DA | P00523 | 257 | 533 | 533.0 | 1N1:1 | Type1.5_Back | None | DFGin | 6.7191 | 14.1749 | BLAminus | -122.29, -173.62 | 52.53, 77.9 | -96.14, 20.03 | 300.27, 89.98 | -55.15, -32.52 | in-in | in | 8.2259 | Saltbr-in | 3.4707 | HRD-in | -89.79, -51.87 | 81.03, -11.33 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.1848 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.62 | APE8-dihe-in | -62.24, 114.12 | APE8-rot-na | 23.22 | APE67-dihe-in | -69.68, -25.09 | -60.39, -25.79 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.7563 | S345C | None | None | XRAY | 2.2 | 0.207 | 0.257 | A | 286.0 | 256.0 | 21 | 29 | 16 | 13 | [[267, 518]] | 1.0 | 3g5d | Gallus gallus | TYR_SRC_CHICK | TYR | 4.5e-94 | 320.5 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 3G5DB | P00523 | 258 | 533 | 533.0 | 1N1:1 | Type1.5_Back | None | DFGin | 6.2754 | 13.5136 | BLAminus | -124.9, 179.31 | 57.13, 77.85 | -97.54, 21.78 | 318.72, 94.26 | -57.84, -11.35 | in-in | in | 8.332 | Saltbr-in | 2.9563 | HRD-in | -82.76, -54.14 | 84.2, -12.02 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.1515 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 141.98 | APE8-dihe-in | -55.02, 101.46 | APE8-rot-na | 16.54 | APE67-dihe-in | -66.6, -25.87 | -58.78, -30.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.0801 | S345C | None | None | XRAY | 2.2 | 0.207 | 0.257 | B | 286.0 | 257.0 | 19 | 29 | 16 | 13 | [[267, 518]] | 1.0 | 3g5d | Gallus gallus | TYR_SRC_CHICK | TYR | 4.5e-94 | 320.5 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| CMGC | MAPK14 | MK14_HUMAN | 3LFAA | Q16539 | 4 | 353 | 360.0 | 1N1:361 | Type1 | Inactive | None | 999.0 | 999.0 | None | -119.32, 169.35 | -154.54, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-in | in | 9.2412 | Saltbr-in | 2.7349 | HRD-in | -67.55, -57.07 | 85.83, -16.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 157.05 | APE8-dihe-out | -85.63, -3.59 | APE8-rot-in | 346.34 | APE67-dihe-in | -59.81, -27.96 | -94.61, -12.54 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.8947 | None | None | None | XRAY | 2.1 | 0.204 | 0.254 | A | 360.0 | 333.0 | 17 | 25 | 10 | 15 | [[24, 308]] | 1.0 | 3lfa | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| OTHER | PKMYT1 | PMYT1_HUMAN | 5VCVA | Q99640 | 75 | 361 | 499.0 | 1N1:60404 | Type1 | Inactive | DFGin | 6.1731 | 14.4679 | BLAminus | -133.17, -164.16 | 53.7, 76.36 | -96.77, 22.58 | 298.04, 107.44 | -64.77, -25.22 | in-in | in | 8.9178 | Saltbr-in | 2.826 | HRD-in | -73.66, -44.65 | 68.1, -0.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8927 | ActLoopCT-out | nonTYR | APEdihe_aaiai | APEdist_iooi | APE10-dihe-na | -65.91, 159.0 | APE9-dihe-na | -91.66, -157.73 | APE8-dihe-in | -52.29, 123.12 | APE8-rot-na | 188.83 | APE67-dihe-in | -60.44, -30.04 | -60.97, -24.44 | APE12-dist-in | 7.9448 | APE11-dist-out | 6.4495 | APE10-dist-out | 9.0797 | APE9-dist-in | 3.1786 | None | TPO260 | TPO260 | XRAY | 1.92 | 0.157 | 0.197 | A | 311.0 | 287.0 | 0 | 27 | 27 | 0 | [[110, 359]] | 1.0 | 5vcv | Homo sapiens | OTHER_PKMYT1_HUMAN | STE | 9.9e-39 | 139.4 | 1.0 | 255.0 | 255.0 | 250 | 251 | 252 | 254 | 256 | 139 | 157 | 161 | 230 | 232 | 231 | 233.0 | 288 | 277 | 272 | 271 | 270 | 269 | 268 | 267 | 266 | 188 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| STE | STK10 | STK10_HUMAN | 5OWRA | O94804 | 23 | 317 | 968.0 | 1N1:401 | Type1 | Inactive | DFGin | 6.4982 | 16.7221 | BLAminus | -126.18, 173.2 | 57.39, 79.01 | -91.46, 24.21 | 286.72, 77.35 | -53.02, -57.95 | out-out | out | 10.2052 | Saltbr-out | 8.1359 | HRD-in | -70.96, -54.03 | 67.34, 13.9 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.8335 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -61.94, -27.24 | 999.0, -15.2 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.3 | 0.221 | 0.254 | A | 302.0 | 282.0 | 13 | 28 | 21 | 7 | [[36, 294]] | 1.0 | 5owr | Homo sapiens | STE_STK10_HUMAN | STE | 2e-94 | 321.6 | 1.0 | 257.0 | 257.0 | 174 | 175 | 176 | 178 | 180 | 65 | 81 | 85 | 154 | 156 | 155 | 157.0 | 219 | 202 | 197 | 196 | 195 | 194 | 193 | 192 | 191 | 111 | Serine/threonine-protein kinase 10 |
| STE | STK24 | STK24_HUMAN | 4QMSA | Q9Y6E0 | 27 | 310 | 443.0 | 1N1:60401 | Type1 | Inactive | DFGin | 7.0296 | 15.2785 | BLAminus | -133.65, 170.4 | 59.12, 88.65 | -100.44, 27.96 | 287.36, 78.03 | -60.48, -24.48 | in-out | in | 9.6308 | Saltbr-out | 4.5468 | HRD-in | -69.75, -48.6 | 69.83, 3.91 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.42, 162.17 | APE9-dihe-na | 128.43, -166.04 | APE8-dihe-in | -119.95, 120.69 | APE8-rot-in | 305.76 | APE67-dihe-in | -58.87, -30.57 | -46.04, -47.24 | APE12-dist-in | 8.2773 | APE11-dist-in | 10.9536 | APE10-dist-in | 5.1134 | APE9-dist-in | 3.3059 | None | TPO190 | TPO190 | XRAY | 1.883 | 0.169 | 0.214 | A | 310.0 | 284.0 | 0 | 28 | 28 | 0 | [[36, 286]] | 1.0 | 4qms | Homo sapiens | STE_STK24_HUMAN | STE | 3.9e-100 | 340.4 | 1.0 | 257.0 | 257.0 | 173 | 174 | 175 | 177 | 179 | 65 | 82 | 86 | 153 | 155 | 154 | 156.0 | 213 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 112 | Serine/threonine-protein kinase 24 |
| TYR | ABL1 | ABL1_HUMAN | 7N9GB | P00519 | 233 | 498 | 1130.0 | STI:60601,1N1:60602 | Allosteric,Type1 | Active | DFGin | 6.7541 | 13.4449 | BLAminus | -122.97, -168.58 | 58.54, 84.79 | -109.7, 15.38 | 305.77, 104.92 | -56.72, -36.19 | in-in | in | 7.8072 | Saltbr-in | 2.716 | HRD-in | -94.83, -54.73 | 76.06, 6.03 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0408 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -97.97, 124.86 | APE9-dihe-in | -118.42, 152.72 | APE8-dihe-in | -70.17, 95.62 | APE8-rot-na | 28.18 | APE67-dihe-in | -73.36, -13.19 | -53.92, -45.07 | APE12-dist-na | 14.9514 | APE11-dist-na | 10.1213 | APE10-dist-na | 12.2789 | APE9-dist-in | 7.1369 | None | None | None | XRAY | 2.2 | 0.219 | 0.251 | B | 271.0 | 264.0 | 2 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 7n9g | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2GQGA | P00519 | 229 | 500 | 1130.0 | 1N1:60501 | Type1 | Inactive | DFGin | 6.6367 | 14.0391 | BLAminus | -125.87, -162.48 | 50.1, 80.24 | -101.91, 13.59 | 304.08, 105.04 | -55.58, -28.07 | in-in | in | 8.2064 | Saltbr-in | 3.3367 | HRD-in | -94.17, -46.19 | 69.1, 8.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0889 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.45, -178.77 | APE9-dihe-in | -144.75, 146.99 | APE8-dihe-in | -51.41, 101.22 | APE8-rot-na | 30.18 | APE67-dihe-in | -72.33, -8.18 | -47.68, -48.27 | APE12-dist-na | 13.8069 | APE11-dist-na | 10.1551 | APE10-dist-na | 13.162 | APE9-dist-in | 7.0168 | None | PTR393 | PTR393 | XRAY | 2.4 | 0.208 | 0.273 | A | 278.0 | 272.0 | 0 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 2gqg | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.4e-100 | 341.1 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2GQGB | P00519 | 229 | 499 | 1130.0 | 1N1:60502 | Type1.5_Back | Active | DFGin | 6.7246 | 13.4066 | BLAminus | -132.96, -163.46 | 57.81, 75.2 | -98.78, 6.6 | 302.62, 104.4 | -52.45, -32.74 | in-in | in | 8.0337 | Saltbr-in | 2.8987 | HRD-in | -101.91, -48.31 | 65.85, 10.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9585 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -100.98, 171.69 | APE9-dihe-in | -137.71, 138.65 | APE8-dihe-in | -58.61, 114.78 | APE8-rot-na | 30.65 | APE67-dihe-in | -71.5, -8.45 | -53.53, -44.9 | APE12-dist-na | 11.2577 | APE11-dist-na | 7.468 | APE10-dist-na | 11.6413 | APE9-dist-in | 6.2756 | None | PTR393 | PTR393 | XRAY | 2.4 | 0.208 | 0.273 | B | 278.0 | 271.0 | 0 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 2gqg | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.4e-100 | 341.1 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 4XEYB | P00519 | 122 | 504 | 1130.0 | 1N1:60601 | Type1 | Inactive | DFGinter | 10.0007 | 8.0224 | BABtrans | -71.04, 121.63 | -84.68, 7.52 | -91.76, 101.26 | 207.86, 90.35 | 143.13, -1.76 | in-out | in | 8.918 | Saltbr-out | 8.6427 | HRD-out | -101.25, 126.15 | -79.9, -27.01 | out-out-in | SNCooi | out-in | ActLoopNT-out | 5.4222 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -80.63, 133.07 | APE9-dihe-in | -116.3, 152.74 | APE8-dihe-in | -66.44, 99.47 | APE8-rot-na | 21.89 | APE67-dihe-in | -71.31, -17.26 | -44.98, -48.3 | APE12-dist-na | 18.5596 | APE11-dist-na | 13.9233 | APE10-dist-na | 16.5485 | APE9-dist-in | 6.4285 | None | None | None | XRAY | 2.891 | 0.232 | 0.259 | B | 408.0 | 359.0 | 9 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 4xey | Homo sapiens | TYR_ABL1_HUMAN | TYR | 8.5e-100 | 339.5 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 7N9GA | P00519 | 233 | 498 | 1130.0 | STI:60601,1N1:60602 | Allosteric,Type1 | Inactive | DFGinter | 10.4212 | 8.1868 | None | -69.43, 136.44 | -123.08, 27.78 | -75.4, -30.96 | 178.85, 77.99 | -98.31, 50.2 | in-out | in | 8.8784 | Saltbr-out | 9.7861 | HRD-out | -92.88, 142.81 | -110.01, 0.88 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.5443 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 170.84 | APE8-dihe-in | -72.01, 95.09 | APE8-rot-na | 30.25 | APE67-dihe-in | -73.75, -10.66 | -54.08, -44.56 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.8503 | None | None | None | XRAY | 2.2 | 0.219 | 0.251 | A | 271.0 | 250.0 | 16 | 29 | 16 | 13 | [[242, 495]] | 1.0 | 7n9g | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 7N9GC | P00519 | 234 | 499 | 1130.0 | STI:60601,1N1:60602 | Allosteric,Type1 | Inactive | DFGinter | 10.016 | 7.7618 | None | -68.53, 140.81 | -120.26, 3.31 | -57.57, -42.4 | 182.82, 108.58 | -86.96, 40.71 | in-none | in | 9.4392 | Saltbr-none | 999.0 | HRD-out | -106.92, 134.12 | -80.26, -30.58 | none-out-none | SNCnon | out-none | ActLoopNT-out | 5.4779 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 96.82 | APE8-dihe-in | -65.53, 99.76 | APE8-rot-na | 23.57 | APE67-dihe-in | -73.61, -20.46 | -60.17, -42.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.8914 | None | None | None | XRAY | 2.2 | 0.219 | 0.251 | C | 271.0 | 233.0 | 33 | 29 | 24 | 5 | [[242, 495]] | 1.0 | 7n9g | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 4XEYA | P00519 | 231 | 503 | 1130.0 | 1N1:60601 | Type1 | Inactive | DFGinter | 9.993 | 7.9273 | None | -70.89, 123.51 | -90.91, 18.27 | -87.3, -11.95 | 199.48, 77.0 | -96.54, 13.69 | in-out | in | 8.9479 | Saltbr-out | 8.6903 | HRD-out | -101.8, 125.8 | -78.66, -28.68 | out-out-in | SNCooi | out-in | ActLoopNT-out | 5.3933 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.59, 140.17 | APE9-dihe-in | -145.27, 142.92 | APE8-dihe-in | -62.13, 98.18 | APE8-rot-na | 23.13 | APE67-dihe-in | -73.29, -19.48 | -49.65, -41.78 | APE12-dist-na | 18.7302 | APE11-dist-na | 14.1077 | APE10-dist-na | 16.5419 | APE9-dist-in | 6.5879 | None | None | None | XRAY | 2.891 | 0.232 | 0.259 | A | 408.0 | 269.0 | 4 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 4xey | Homo sapiens | TYR_ABL1_HUMAN | TYR | 8.5e-100 | 339.5 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | BMX | BMX_HUMAN | 3SXRA | P51813 | 411 | 671 | 675.0 | 1N1:60001 | Type1 | Inactive | DFGinter | 7.8824 | 8.1671 | BABtrans | -93.57, 121.18 | -103.19, -9.04 | -51.22, 114.45 | 184.77, 74.21 | 62.74, 18.94 | out-out | out | 10.805 | Saltbr-out | 7.5586 | HRD-out | -99.0, 124.02 | -80.22, -7.53 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8353 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -95.14, 119.04 | APE9-dihe-in | -94.0, 160.01 | APE8-dihe-in | -48.96, 127.48 | APE8-rot-na | 331.52 | APE67-dihe-in | -68.66, -11.59 | -65.07, -24.25 | APE12-dist-na | 10.0286 | APE11-dist-na | 7.5492 | APE10-dist-na | 12.0421 | APE9-dist-in | 5.1857 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | A | 268.0 | 257.0 | 4 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | Homo sapiens | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 3SXRB | P51813 | 411 | 671 | 675.0 | 1N1:60002 | Type1 | Inactive | DFGinter | 7.7085 | 8.2724 | BABtrans | -92.79, 121.27 | -96.68, -12.13 | -49.05, 115.54 | 186.98, 71.37 | 61.78, 19.24 | out-out | out | 10.8028 | Saltbr-out | 8.0973 | HRD-out | -100.92, 124.05 | -80.64, -7.7 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8449 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.81, 125.57 | APE9-dihe-in | -101.37, 158.16 | APE8-dihe-in | -49.48, 128.1 | APE8-rot-na | 332.21 | APE67-dihe-in | -66.79, -11.14 | -62.63, -27.73 | APE12-dist-na | 9.9457 | APE11-dist-na | 7.4465 | APE10-dist-na | 11.9437 | APE9-dist-in | 5.1904 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | B | 268.0 | 255.0 | 6 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | Homo sapiens | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BTK | BTK_HUMAN | 3K54A | Q06187 | 392 | 658 | 659.0 | 1N1:1 | Type1 | Inactive | DFGin | 4.6816 | 13.9981 | BLAplus | -132.68, -179.17 | 50.27, 30.98 | -93.41, -0.42 | 58.12, 86.77 | -82.65, 999.0 | in-out | in | 8.7866 | Saltbr-out | 3.7709 | HRD-in | -69.54, -47.61 | 72.38, -12.01 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 136.06 | APE8-dihe-in | -84.11, 69.82 | APE8-rot-na | 29.89 | APE67-dihe-in | -70.22, -9.36 | -47.67, -47.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.1055 | Y551E | None | None | XRAY | 1.94 | 0.202 | 0.258 | A | 283.0 | 243.0 | 24 | 29 | 12 | 17 | [[402, 653]] | 1.0 | 3k54 | Homo sapiens | TYR_BTK_HUMAN | TYR | 1.6e-92 | 315.4 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_HUMAN | 3OCTA | Q06187 | 394 | 656 | 659.0 | 1N1:663 | Type1 | Inactive | DFGinter | 9.5513 | 8.0475 | BABtrans | -83.49, 139.01 | -103.95, 15.92 | -87.02, 132.92 | 181.28, 97.3 | 77.87, 26.97 | in-out | in | 9.203 | Saltbr-out | 7.7453 | HRD-in | -70.28, -48.13 | 67.57, -13.36 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.3805 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 95.42 | APE8-dihe-in | -60.66, 106.57 | APE8-rot-na | 28.18 | APE67-dihe-in | -77.0, -13.84 | -55.35, -41.2 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.7096 | V555R | None | None | XRAY | 1.95 | 0.199 | 0.251 | A | 265.0 | 244.0 | 19 | 29 | 15 | 14 | [[402, 653]] | 1.0 | 3oct | Homo sapiens | TYR_BTK_HUMAN | TYR | 2.3e-93 | 318.2 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | DDR1 | DDR1_HUMAN | 6BSDA | Q08345 | 604 | 912 | 913.0 | 1N1:60901 | Type1 | Inactive | DFGinter | 9.9484 | 9.844 | None | -87.87, 155.34 | -64.16, -24.42 | 174.69, 170.82 | 68.3, 89.44 | 55.93, 999.0 | in-in | in | 8.3705 | Saltbr-in | 2.7354 | HRD-in | -61.68, -56.93 | 83.98, -4.33 | in-out-in | SNCioi | out-in | ActLoopNT-out | 19.8476 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -66.74, 115.57 | APE9-dihe-in | -116.16, 127.65 | APE8-dihe-in | -81.76, 68.68 | APE8-rot-na | 34.21 | APE67-dihe-in | -66.93, -20.25 | -61.43, -30.39 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.1458 | None | None | None | XRAY | 2.606 | 0.186 | 0.255 | A | 351.0 | 278.0 | 31 | 30 | 28 | 2 | [[610, 907]] | 1.0 | 6bsd | Homo sapiens | TYR_DDR1_HUMAN | TYR | 2.3e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 5BVWA | Q08345 | 604 | 911 | 913.0 | 1N1:1009 | Type1 | Inactive | DFGout | 14.538 | 10.296 | None | -113.16, 175.58 | -102.37, -21.68 | 40.34, 118.5 | 221.24, 85.03 | -134.54, 999.0 | in-in | in | 8.3337 | Saltbr-in | 2.775 | HRD-in | -77.35, -46.96 | 73.51, -12.24 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -79.96, 123.56 | APE9-dihe-in | -122.26, 123.59 | APE8-dihe-in | -77.84, 65.49 | APE8-rot-na | 31.29 | APE67-dihe-in | -69.31, -14.79 | -54.53, -34.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.409 | None | None | None | XRAY | 1.94 | 0.186 | 0.234 | A | 324.0 | 274.0 | 34 | 30 | 26 | 4 | [[610, 907]] | 1.0 | 5bvw | Homo sapiens | TYR_DDR1_HUMAN | TYR | 1.7e-92 | 315.4 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | EPHA2 | EPHA2_HUMAN | 5I9YA | P29317 | 600 | 896 | 976.0 | 1N1:1001 | Type1 | Inactive | DFGin | 6.2223 | 14.973 | BLBminus | -129.12, 177.86 | 73.14, 77.74 | -114.09, 153.37 | 295.9, 102.04 | 147.64, -171.81 | in-in | in | 8.2568 | Saltbr-in | 2.7741 | HRD-in | -75.07, -47.16 | 76.83, -16.24 | in-out-none | SNCion | out-none | ActLoopNT-out | 10.4586 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 139.34 | APE8-rot-na | 36.16 | APE67-dihe-in | -79.28, -3.2 | -53.92, -45.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.228 | 0.164 | 0.179 | A | 306.0 | 287.0 | 10 | 31 | 24 | 7 | [[613, 873]] | 1.0 | 5i9y | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHB4 | EPHB4_HUMAN | 6FNMA | P54760 | 608 | 889 | 987.0 | 1N1:1001 | Type1 | Inactive | DFGin | 5.9609 | 15.7692 | BLBminus | -128.55, -169.2 | 67.78, 75.65 | -110.02, 138.75 | 293.26, 98.41 | 179.12, 146.16 | in-in | in | 8.3255 | Saltbr-in | 3.1793 | HRD-in | -76.03, -51.54 | 81.54, -15.45 | in-out-in | SNCioi | out-in | ActLoopNT-out | 10.0097 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.65, 157.69 | APE9-dihe-in | -64.87, 128.21 | APE8-dihe-in | -78.96, 90.14 | APE8-rot-na | 30.03 | APE67-dihe-in | -61.19, -22.58 | -57.17, -48.0 | APE12-dist-na | 999.0 | APE11-dist-na | 11.3678 | APE10-dist-na | 15.0342 | APE9-dist-in | 6.5764 | Y774E,A803V,V870I | None | None | XRAY | 1.157 | 0.184 | 0.195 | A | 297.0 | 270.0 | 12 | 33 | 21 | 12 | [[615, 876]] | 1.0 | 6fnm | Homo sapiens | TYR_EPHB4_HUMAN | TYR | 4.2e-105 | 356.7 | 2.0 | 261.0 | 260.0 | 757 | 758 | 759 | 761 | 763 | 647 | 664 | 668 | 737 | 739 | 738 | 740.0 | 802 | 790 | 785 | 784 | 783 | 782 | 781 | 780 | 779 | 694 | Ephrin type-B receptor 4 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UA | Q13882 | 185 | 446 | 451.0 | 1N1:60501 | Type1 | Inactive | DFGin | 5.9983 | 13.4628 | BLBplus | -115.66, 172.2 | 65.44, 13.7 | -58.08, 130.19 | 47.49, 85.54 | 66.94, -1.55 | out-out | out | 14.1683 | Saltbr-out | 16.091 | HRD-in | -72.57, -54.48 | 85.53, -13.44 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.2608 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 72.03, 33.67 | APE9-dihe-out | -55.65, -32.62 | APE8-dihe-out | -63.18, -18.16 | APE8-rot-na | 340.69 | APE67-dihe-in | -82.41, -18.93 | -56.57, -27.65 | APE12-dist-na | 16.3439 | APE11-dist-na | 20.6081 | APE10-dist-na | 18.2629 | APE9-dist-out | 11.0621 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | A | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | Homo sapiens | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UB | Q13882 | 185 | 446 | 451.0 | 1N1:60501 | Type1 | Inactive | DFGin | 6.0808 | 13.3427 | BLBplus | -112.62, 168.56 | 69.96, 13.64 | -58.15, 126.09 | 44.9, 88.52 | 70.74, 0.77 | out-out | out | 14.3036 | Saltbr-out | 15.9567 | HRD-in | -65.56, -52.22 | 84.8, -15.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0671 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 67.1, 31.04 | APE9-dihe-out | -51.48, -32.62 | APE8-dihe-out | -56.92, -21.84 | APE8-rot-na | 331.92 | APE67-dihe-in | -82.05, -11.15 | -61.67, -25.37 | APE12-dist-na | 16.2609 | APE11-dist-na | 20.2262 | APE10-dist-na | 17.9045 | APE9-dist-out | 11.0552 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | B | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | Homo sapiens | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UC | Q13882 | 185 | 446 | 451.0 | 1N1:60501 | Type1 | Inactive | DFGin | 5.9677 | 13.6341 | BLBplus | -101.49, 165.12 | 71.33, 11.9 | -56.7, 126.68 | 46.28, 85.99 | 72.45, -1.55 | out-out | out | 14.2504 | Saltbr-out | 15.3617 | HRD-in | -69.3, -53.89 | 83.99, -9.53 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.1583 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 66.45, 29.68 | APE9-dihe-out | -47.22, -37.04 | APE8-dihe-out | -58.56, -24.03 | APE8-rot-na | 334.48 | APE67-dihe-in | -84.14, -9.31 | -53.24, -25.76 | APE12-dist-na | 16.3889 | APE11-dist-na | 20.3117 | APE10-dist-na | 17.9592 | APE9-dist-out | 11.0174 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | C | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | Homo sapiens | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | PTK6 | PTK6_HUMAN | 5H2UD | Q13882 | 185 | 446 | 451.0 | 1N1:60504 | Type1 | Inactive | DFGin | 6.1814 | 13.2695 | BLBplus | -112.73, 164.13 | 73.65, 11.67 | -56.94, 123.73 | 42.41, 88.79 | 73.17, 2.96 | out-out | out | 14.0107 | Saltbr-out | 15.9929 | HRD-in | -70.19, -55.11 | 88.71, -18.22 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.1947 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | 72.07, 30.74 | APE9-dihe-out | -48.72, -36.76 | APE8-dihe-out | -61.03, -20.74 | APE8-rot-na | 334.99 | APE67-dihe-in | -84.77, -13.01 | -55.36, -26.11 | APE12-dist-na | 16.3004 | APE11-dist-na | 20.346 | APE10-dist-na | 18.0251 | APE9-dist-out | 11.0324 | C433T | None | None | XRAY | 2.24 | 0.208 | 0.26 | D | 267.0 | 261.0 | 1 | 28 | 28 | 0 | [[191, 443]] | 1.0 | 5h2u | Homo sapiens | TYR_PTK6_HUMAN | TYR | 9.8e-89 | 303.0 | 2.0 | 260.0 | 259.0 | 329 | 330 | 331 | 333 | 335 | 219 | 235 | 239 | 309 | 311 | 310 | 312.0 | 369 | 357 | 352 | 351 | 350 | 349 | 348 | 347 | 346 | 265 | Protein-tyrosine kinase 6 |
| TYR | ABL2 | ABL2_MOUSE | 4XLIA | Q4JIM5 | 279 | 546 | 1182.0 | 1N1:601 | Type1.5_Back | Inactive | DFGin | 6.5075 | 13.6034 | BLAminus | -146.93, -165.44 | 45.19, 75.22 | -96.7, 24.95 | 303.43, 100.32 | -77.67, 1.06 | in-out | in | 8.1979 | Saltbr-out | 4.2161 | HRD-in | -89.85, -46.08 | 70.33, 6.25 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9692 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.74, 141.9 | APE9-dihe-in | -130.79, 158.17 | APE8-dihe-in | -65.12, 108.35 | APE8-rot-na | 22.1 | APE67-dihe-in | -73.67, -11.6 | -58.5, -43.4 | APE12-dist-na | 15.3379 | APE11-dist-na | 10.7818 | APE10-dist-na | 13.3164 | APE9-dist-in | 7.1309 | None | None | None | XRAY | 2.5 | 0.157 | 0.205 | A | 268.0 | 264.0 | 4 | 29 | 29 | 0 | [[288, 541]] | 1.0 | 4xli | Mus musculus | TYR_ABL2_MOUSE | TYR | 2e-98 | 334.8 | 1.0 | 260.0 | 260.0 | 426 | 427 | 428 | 430 | 432 | 317 | 332 | 336 | 406 | 408 | 407 | 409.0 | 467 | 455 | 450 | 449 | 448 | 447 | 446 | 445 | 444 | 362 | Tyrosine-protein kinase ABL2 |
| TYR | ABL2 | ABL2_MOUSE | 4XLIB | Q4JIM5 | 279 | 546 | 1182.0 | 1N1:600 | Type1.5_Back | Active | DFGin | 6.3912 | 13.6381 | BLAminus | -131.7, -165.09 | 47.95, 80.18 | -101.55, 32.58 | 307.48, 89.21 | -70.05, -27.33 | in-in | in | 8.2287 | Saltbr-in | 2.5374 | HRD-in | -85.97, -54.42 | 80.41, 14.17 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -119.09, 129.65 | APE9-dihe-in | -110.16, 158.75 | APE8-dihe-in | -72.12, 103.04 | APE8-rot-na | 29.85 | APE67-dihe-in | -62.36, -22.19 | -57.39, -43.34 | APE12-dist-na | 15.0495 | APE11-dist-na | 10.2063 | APE10-dist-na | 12.5948 | APE9-dist-in | 7.0962 | None | None | None | XRAY | 2.5 | 0.157 | 0.205 | B | 268.0 | 264.0 | 4 | 29 | 29 | 0 | [[288, 541]] | 1.0 | 4xli | Mus musculus | TYR_ABL2_MOUSE | TYR | 2e-98 | 334.8 | 1.0 | 260.0 | 260.0 | 426 | 427 | 428 | 430 | 432 | 317 | 332 | 336 | 406 | 408 | 407 | 409.0 | 467 | 455 | 450 | 449 | 448 | 447 | 446 | 445 | 444 | 362 | Tyrosine-protein kinase ABL2 |
| TYR | BTK | BTK_MOUSE | 8S9FA | P35991 | 392 | 659 | 659.0 | 1N1:801 | Type1 | Inactive | DFGinter | 9.7383 | 8.4773 | BABtrans | -103.75, 162.9 | -98.62, -12.56 | -74.46, 134.73 | 203.6, 82.29 | 75.53, 30.46 | out-out | out | 11.3245 | Saltbr-out | 8.457 | HRD-out | -78.16, 120.76 | -71.26, -27.71 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.4638 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 89.3 | APE8-rot-na | 354.27 | APE67-dihe-in | -88.28, 1.83 | -66.03, -37.53 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | L390G,Y551E,Y617P | None | None | XRAY | 2.6 | 0.244 | 0.284 | A | 279.0 | 254.0 | 14 | 29 | 15 | 14 | [[402, 653]] | 1.0 | 8s9f | Mus musculus | TYR_BTK_MOUSE | TYR | 1.3e-92 | 315.7 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_MOUSE | 8S9FB | P35991 | 392 | 659 | 659.0 | 1N1:801 | Type1 | Inactive | DFGinter | 9.5087 | 8.4716 | BABtrans | -108.61, 149.63 | -109.15, 7.92 | -82.22, 131.91 | 185.43, 98.64 | 78.7, 27.48 | out-out | out | 11.0192 | Saltbr-out | 10.3295 | HRD-out | -91.58, 112.75 | -69.14, -29.29 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.6813 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 166.92 | APE9-dihe-in | -91.32, 115.75 | APE8-dihe-in | -71.7, 107.6 | APE8-rot-na | 25.58 | APE67-dihe-in | -83.25, -12.58 | -54.13, -30.99 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 16.1492 | APE9-dist-out | 18.604 | L390G,Y551E,Y617P | None | None | XRAY | 2.6 | 0.244 | 0.284 | B | 279.0 | 255.0 | 13 | 29 | 17 | 12 | [[402, 653]] | 1.0 | 8s9f | Mus musculus | TYR_BTK_MOUSE | TYR | 1.3e-92 | 315.7 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | EPHA4 | EPHA4_MOUSE | 2Y6OA | Q03137 | 609 | 891 | 986.0 | 1N1:1892 | Type1 | Inactive | DFGin | 6.5237 | 15.3156 | None | -125.69, -163.2 | 68.45, 65.65 | -111.22, 999.0 | 295.37, 106.51 | 999.0, 999.0 | in-in | in | 8.2042 | Saltbr-in | 2.6896 | HRD-in | -74.99, -48.94 | 76.82, -16.04 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 122.47 | APE8-dihe-in | -69.65, 86.1 | APE8-rot-na | 27.26 | APE67-dihe-in | -78.79, 0.73 | -48.0, -50.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.6377 | None | None | None | XRAY | 1.543 | 0.181 | 0.201 | A | 291.0 | 263.0 | 20 | 31 | 11 | 20 | [[621, 880]] | 1.0 | 2y6o | Mus musculus | TYR_EPHA4_MOUSE | TYR | 1.6e-109 | 371.2 | 1.0 | 261.0 | 261.0 | 763 | 764 | 765 | 767 | 769 | 653 | 670 | 674 | 743 | 745 | 744 | 746.0 | 806 | 794 | 789 | 788 | 787 | 786 | 785 | 784 | 783 | 700 | Ephrin type-A receptor 4 |
| TYR | LYN | LYN_MOUSE | 2ZVAA | P25911 | 239 | 502 | 512.0 | 1N1:60513 | Type1.5_Back | Inactive | DFGin | 6.4453 | 13.8753 | BLAminus | -120.49, -171.3 | 46.11, 83.42 | -100.41, 24.42 | 303.87, 89.77 | -59.23, -40.1 | in-in | in | 8.3149 | Saltbr-in | 2.7526 | HRD-naN | -93.32, -50.56 | 73.54, -8.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7284 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 87.79, 115.97 | APE9-dihe-in | -82.02, 152.26 | APE8-dihe-in | -82.89, 88.6 | APE8-rot-na | 28.7 | APE67-dihe-in | -67.8, -12.1 | -43.08, -51.75 | APE12-dist-na | 10.4403 | APE11-dist-na | 6.3096 | APE10-dist-na | 9.4506 | APE9-dist-in | 5.3495 | None | None | None | XRAY | 2.6 | 0.199 | 0.231 | A | 279.0 | 260.0 | 4 | 29 | 25 | 4 | [[247, 499]] | 1.0 | 2zva | Mus musculus | TYR_LYN_MOUSE | TYR | 4.1e-95 | 323.9 | 1.0 | 260.0 | 260.0 | 384 | 385 | 386 | 388 | 390 | 275 | 290 | 294 | 364 | 366 | 365 | 367.0 | 425 | 413 | 408 | 407 | 406 | 405 | 404 | 403 | 402 | 320 | Tyrosine-protein kinase Lyn |
| CMGC | P38A | A9UJZ9_SALSA | 3OHTA | A9UJZ9 | 5 | 352 | 361.0 | 1N1:1000,1N1:2000 | Type1.5_Back,Allosteric | Inactive | DFGout | 13.5799 | 9.5849 | None | -78.92, -176.24 | -106.96, 26.33 | -169.7, 165.77 | 77.85, 98.84 | 145.96, 999.0 | in-in | in | 9.1763 | Saltbr-in | 2.7252 | HRD-out | -88.45, 143.68 | -105.73, 98.3 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.235 | 0.289 | A | 389.0 | 331.0 | 17 | 25 | 8 | 17 | [[25, 309]] | 1.0 | 3oht | Salmo salar | CMGC_P38A_SALSA | CMGC | 2.1e-83 | 286.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 54 | 72 | 76 | 148 | 150 | 149 | 151.0 | 206 | 193 | 188 | 187 | 186 | 185 | 184 | 183 | 182 | 108 | mitogen-activated protein kinase |
| CMGC | P38A | A9UJZ9_SALSA | 3OHTB | A9UJZ9 | 5 | 352 | 361.0 | 1N1:1000,1N1:2000 | Type1.5_Back,Allosteric | Inactive | DFGout | 13.3516 | 9.2901 | None | -90.67, 172.5 | -94.08, 34.32 | -176.15, 166.37 | 74.91, 100.91 | -151.94, 999.0 | in-in | in | 9.1457 | Saltbr-in | 2.7005 | HRD-out | -93.8, 126.44 | -88.56, 105.72 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.235 | 0.289 | B | 389.0 | 331.0 | 17 | 25 | 8 | 17 | [[25, 309]] | 1.0 | 3oht | Salmo salar | CMGC_P38A_SALSA | CMGC | 2.1e-83 | 286.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 54 | 72 | 76 | 148 | 150 | 149 | 151.0 | 206 | 193 | 188 | 187 | 186 | 185 | 184 | 183 | 182 | 108 | mitogen-activated protein kinase |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SRC | SRC_CHICK | 3QLGA | P00523 | 258 | 533 | 533.0 | 1N1:601 | Type1.5_Back | Inactive | DFGin | 6.5502 | 13.8381 | BLAminus | -128.97, 169.0 | 62.45, 93.12 | -106.99, 6.4 | 306.69, 101.34 | -122.4, 999.0 | in-in | in | 8.7224 | Saltbr-in | 2.9531 | HRD-in | -90.7, -55.87 | 92.28, -19.25 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 140.4 | APE8-dihe-in | -85.59, 52.69 | APE8-rot-na | 6.03 | APE67-dihe-in | -68.2, -8.8 | -50.34, -41.04 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.1548 | L317I | None | None | XRAY | 2.75 | 0.203 | 0.269 | A | 286.0 | 259.0 | 17 | 29 | 12 | 17 | [[267, 518]] | 1.0 | 3qlg | Gallus gallus | TYR_SRC_CHICK | TYR | 7e-94 | 319.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 3QLGB | P00523 | 256 | 533 | 533.0 | 1N1:601 | Type1.5_Back | Inactive | DFGin | 6.2634 | 13.1722 | BLAminus | -132.53, 169.92 | 55.67, 96.64 | -114.48, 23.35 | 323.76, 73.27 | -64.65, -16.14 | in-in | in | 8.523 | Saltbr-in | 2.7156 | HRD-in | -89.78, -56.21 | 92.27, -19.49 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.1877 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 135.14 | APE8-dihe-in | -84.28, 53.37 | APE8-rot-na | 5.94 | APE67-dihe-in | -68.54, -8.95 | -50.64, -40.54 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.0573 | L317I | None | None | XRAY | 2.75 | 0.203 | 0.269 | B | 286.0 | 260.0 | 18 | 29 | 16 | 13 | [[267, 518]] | 1.0 | 3qlg | Gallus gallus | TYR_SRC_CHICK | TYR | 7e-94 | 319.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 3G5DA | P00523 | 257 | 533 | 533.0 | 1N1:1 | Type1.5_Back | None | DFGin | 6.7191 | 14.1749 | BLAminus | -122.29, -173.62 | 52.53, 77.9 | -96.14, 20.03 | 300.27, 89.98 | -55.15, -32.52 | in-in | in | 8.2259 | Saltbr-in | 3.4707 | HRD-in | -89.79, -51.87 | 81.03, -11.33 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.1848 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.62 | APE8-dihe-in | -62.24, 114.12 | APE8-rot-na | 23.22 | APE67-dihe-in | -69.68, -25.09 | -60.39, -25.79 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.7563 | S345C | None | None | XRAY | 2.2 | 0.207 | 0.257 | A | 286.0 | 256.0 | 21 | 29 | 16 | 13 | [[267, 518]] | 1.0 | 3g5d | Gallus gallus | TYR_SRC_CHICK | TYR | 4.5e-94 | 320.5 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 3G5DB | P00523 | 258 | 533 | 533.0 | 1N1:1 | Type1.5_Back | None | DFGin | 6.2754 | 13.5136 | BLAminus | -124.9, 179.31 | 57.13, 77.85 | -97.54, 21.78 | 318.72, 94.26 | -57.84, -11.35 | in-in | in | 8.332 | Saltbr-in | 2.9563 | HRD-in | -82.76, -54.14 | 84.2, -12.02 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.1515 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 141.98 | APE8-dihe-in | -55.02, 101.46 | APE8-rot-na | 16.54 | APE67-dihe-in | -66.6, -25.87 | -58.78, -30.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.0801 | S345C | None | None | XRAY | 2.2 | 0.207 | 0.257 | B | 286.0 | 257.0 | 19 | 29 | 16 | 13 | [[267, 518]] | 1.0 | 3g5d | Gallus gallus | TYR_SRC_CHICK | TYR | 4.5e-94 | 320.5 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | ABL2 | ABL2_MOUSE | 4XLIA | Q4JIM5 | 279 | 546 | 1182.0 | 1N1:601 | Type1.5_Back | Inactive | DFGin | 6.5075 | 13.6034 | BLAminus | -146.93, -165.44 | 45.19, 75.22 | -96.7, 24.95 | 303.43, 100.32 | -77.67, 1.06 | in-out | in | 8.1979 | Saltbr-out | 4.2161 | HRD-in | -89.85, -46.08 | 70.33, 6.25 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9692 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.74, 141.9 | APE9-dihe-in | -130.79, 158.17 | APE8-dihe-in | -65.12, 108.35 | APE8-rot-na | 22.1 | APE67-dihe-in | -73.67, -11.6 | -58.5, -43.4 | APE12-dist-na | 15.3379 | APE11-dist-na | 10.7818 | APE10-dist-na | 13.3164 | APE9-dist-in | 7.1309 | None | None | None | XRAY | 2.5 | 0.157 | 0.205 | A | 268.0 | 264.0 | 4 | 29 | 29 | 0 | [[288, 541]] | 1.0 | 4xli | Mus musculus | TYR_ABL2_MOUSE | TYR | 2e-98 | 334.8 | 1.0 | 260.0 | 260.0 | 426 | 427 | 428 | 430 | 432 | 317 | 332 | 336 | 406 | 408 | 407 | 409.0 | 467 | 455 | 450 | 449 | 448 | 447 | 446 | 445 | 444 | 362 | Tyrosine-protein kinase ABL2 |
| TYR | ABL2 | ABL2_MOUSE | 4XLIB | Q4JIM5 | 279 | 546 | 1182.0 | 1N1:600 | Type1.5_Back | Active | DFGin | 6.3912 | 13.6381 | BLAminus | -131.7, -165.09 | 47.95, 80.18 | -101.55, 32.58 | 307.48, 89.21 | -70.05, -27.33 | in-in | in | 8.2287 | Saltbr-in | 2.5374 | HRD-in | -85.97, -54.42 | 80.41, 14.17 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -119.09, 129.65 | APE9-dihe-in | -110.16, 158.75 | APE8-dihe-in | -72.12, 103.04 | APE8-rot-na | 29.85 | APE67-dihe-in | -62.36, -22.19 | -57.39, -43.34 | APE12-dist-na | 15.0495 | APE11-dist-na | 10.2063 | APE10-dist-na | 12.5948 | APE9-dist-in | 7.0962 | None | None | None | XRAY | 2.5 | 0.157 | 0.205 | B | 268.0 | 264.0 | 4 | 29 | 29 | 0 | [[288, 541]] | 1.0 | 4xli | Mus musculus | TYR_ABL2_MOUSE | TYR | 2e-98 | 334.8 | 1.0 | 260.0 | 260.0 | 426 | 427 | 428 | 430 | 432 | 317 | 332 | 336 | 406 | 408 | 407 | 409.0 | 467 | 455 | 450 | 449 | 448 | 447 | 446 | 445 | 444 | 362 | Tyrosine-protein kinase ABL2 |
| TYR | BTK | BTK_MOUSE | 8S9FA | P35991 | 392 | 659 | 659.0 | 1N1:801 | Type1 | Inactive | DFGinter | 9.7383 | 8.4773 | BABtrans | -103.75, 162.9 | -98.62, -12.56 | -74.46, 134.73 | 203.6, 82.29 | 75.53, 30.46 | out-out | out | 11.3245 | Saltbr-out | 8.457 | HRD-out | -78.16, 120.76 | -71.26, -27.71 | out-out-none | SNCoon | out-none | ActLoopNT-out | 5.4638 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 89.3 | APE8-rot-na | 354.27 | APE67-dihe-in | -88.28, 1.83 | -66.03, -37.53 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | L390G,Y551E,Y617P | None | None | XRAY | 2.6 | 0.244 | 0.284 | A | 279.0 | 254.0 | 14 | 29 | 15 | 14 | [[402, 653]] | 1.0 | 8s9f | Mus musculus | TYR_BTK_MOUSE | TYR | 1.3e-92 | 315.7 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | BTK | BTK_MOUSE | 8S9FB | P35991 | 392 | 659 | 659.0 | 1N1:801 | Type1 | Inactive | DFGinter | 9.5087 | 8.4716 | BABtrans | -108.61, 149.63 | -109.15, 7.92 | -82.22, 131.91 | 185.43, 98.64 | 78.7, 27.48 | out-out | out | 11.0192 | Saltbr-out | 10.3295 | HRD-out | -91.58, 112.75 | -69.14, -29.29 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.6813 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 166.92 | APE9-dihe-in | -91.32, 115.75 | APE8-dihe-in | -71.7, 107.6 | APE8-rot-na | 25.58 | APE67-dihe-in | -83.25, -12.58 | -54.13, -30.99 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 16.1492 | APE9-dist-out | 18.604 | L390G,Y551E,Y617P | None | None | XRAY | 2.6 | 0.244 | 0.284 | B | 279.0 | 255.0 | 13 | 29 | 17 | 12 | [[402, 653]] | 1.0 | 8s9f | Mus musculus | TYR_BTK_MOUSE | TYR | 1.3e-92 | 315.7 | 1.0 | 258.0 | 258.0 | 538 | 539 | 540 | 542 | 544 | 430 | 445 | 449 | 518 | 520 | 519 | 521.0 | 579 | 567 | 562 | 561 | 560 | 559 | 558 | 557 | 556 | 475 | Tyrosine-protein kinase BTK |
| TYR | EPHA4 | EPHA4_MOUSE | 2Y6OA | Q03137 | 609 | 891 | 986.0 | 1N1:1892 | Type1 | Inactive | DFGin | 6.5237 | 15.3156 | None | -125.69, -163.2 | 68.45, 65.65 | -111.22, 999.0 | 295.37, 106.51 | 999.0, 999.0 | in-in | in | 8.2042 | Saltbr-in | 2.6896 | HRD-in | -74.99, -48.94 | 76.82, -16.04 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 122.47 | APE8-dihe-in | -69.65, 86.1 | APE8-rot-na | 27.26 | APE67-dihe-in | -78.79, 0.73 | -48.0, -50.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.6377 | None | None | None | XRAY | 1.543 | 0.181 | 0.201 | A | 291.0 | 263.0 | 20 | 31 | 11 | 20 | [[621, 880]] | 1.0 | 2y6o | Mus musculus | TYR_EPHA4_MOUSE | TYR | 1.6e-109 | 371.2 | 1.0 | 261.0 | 261.0 | 763 | 764 | 765 | 767 | 769 | 653 | 670 | 674 | 743 | 745 | 744 | 746.0 | 806 | 794 | 789 | 788 | 787 | 786 | 785 | 784 | 783 | 700 | Ephrin type-A receptor 4 |
| TYR | LYN | LYN_MOUSE | 2ZVAA | P25911 | 239 | 502 | 512.0 | 1N1:60513 | Type1.5_Back | Inactive | DFGin | 6.4453 | 13.8753 | BLAminus | -120.49, -171.3 | 46.11, 83.42 | -100.41, 24.42 | 303.87, 89.77 | -59.23, -40.1 | in-in | in | 8.3149 | Saltbr-in | 2.7526 | HRD-naN | -93.32, -50.56 | 73.54, -8.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7284 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 87.79, 115.97 | APE9-dihe-in | -82.02, 152.26 | APE8-dihe-in | -82.89, 88.6 | APE8-rot-na | 28.7 | APE67-dihe-in | -67.8, -12.1 | -43.08, -51.75 | APE12-dist-na | 10.4403 | APE11-dist-na | 6.3096 | APE10-dist-na | 9.4506 | APE9-dist-in | 5.3495 | None | None | None | XRAY | 2.6 | 0.199 | 0.231 | A | 279.0 | 260.0 | 4 | 29 | 25 | 4 | [[247, 499]] | 1.0 | 2zva | Mus musculus | TYR_LYN_MOUSE | TYR | 4.1e-95 | 323.9 | 1.0 | 260.0 | 260.0 | 384 | 385 | 386 | 388 | 390 | 275 | 290 | 294 | 364 | 366 | 365 | 367.0 | 425 | 413 | 408 | 407 | 406 | 405 | 404 | 403 | 402 | 320 | Tyrosine-protein kinase Lyn |
| CMGC | P38A | A9UJZ9_SALSA | 3OHTA | A9UJZ9 | 5 | 352 | 361.0 | 1N1:1000,1N1:2000 | Type1.5_Back,Allosteric | Inactive | DFGout | 13.5799 | 9.5849 | None | -78.92, -176.24 | -106.96, 26.33 | -169.7, 165.77 | 77.85, 98.84 | 145.96, 999.0 | in-in | in | 9.1763 | Saltbr-in | 2.7252 | HRD-out | -88.45, 143.68 | -105.73, 98.3 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.235 | 0.289 | A | 389.0 | 331.0 | 17 | 25 | 8 | 17 | [[25, 309]] | 1.0 | 3oht | Salmo salar | CMGC_P38A_SALSA | CMGC | 2.1e-83 | 286.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 54 | 72 | 76 | 148 | 150 | 149 | 151.0 | 206 | 193 | 188 | 187 | 186 | 185 | 184 | 183 | 182 | 108 | mitogen-activated protein kinase |
| CMGC | P38A | A9UJZ9_SALSA | 3OHTB | A9UJZ9 | 5 | 352 | 361.0 | 1N1:1000,1N1:2000 | Type1.5_Back,Allosteric | Inactive | DFGout | 13.3516 | 9.2901 | None | -90.67, 172.5 | -94.08, 34.32 | -176.15, 166.37 | 74.91, 100.91 | -151.94, 999.0 | in-in | in | 9.1457 | Saltbr-in | 2.7005 | HRD-out | -93.8, 126.44 | -88.56, 105.72 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, 999.0 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.235 | 0.289 | B | 389.0 | 331.0 | 17 | 25 | 8 | 17 | [[25, 309]] | 1.0 | 3oht | Salmo salar | CMGC_P38A_SALSA | CMGC | 2.1e-83 | 286.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 54 | 72 | 76 | 148 | 150 | 149 | 151.0 | 206 | 193 | 188 | 187 | 186 | 185 | 184 | 183 | 182 | 108 | mitogen-activated protein kinase |