Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 7 | 6AAMA |
DFGin | ABAminus | 2 | 6AAHA |
Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|
TYR | JAK1 | JAK1_HUMAN | Tyrosine-protein kinase JAK1 | 6AAHA | 1.83 | Inactive | DFGin | ABAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK1 | JAK1_HUMAN | Tyrosine-protein kinase JAK1 | 6AAHB | 1.83 | Inactive | DFGin | ABAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 6AAJA | 2.37 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 6AAJB | 2.37 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKA | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKB | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKC | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKD | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
TYR | TYK2 | TYK2_HUMAN | Non-receptor tyrosine-protein kinase TYK2 | 6AAMA | 1.98 | None | DFGin | BLAminus | in-in | in-none | 9T6 | Type1 |
Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 7 | 6AAMA |
DFGin | ABAminus | 2 | 6AAHA |
Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Homo sapiens | TYR | JAK1 | JAK1_HUMAN | Tyrosine-protein kinase JAK1 | 6AAHA | 1.83 | Inactive | DFGin | ABAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK1 | JAK1_HUMAN | Tyrosine-protein kinase JAK1 | 6AAHB | 1.83 | Inactive | DFGin | ABAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 6AAJA | 2.37 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 6AAJB | 2.37 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKA | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKB | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKC | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | JAK3 | JAK3_HUMAN | Tyrosine-protein kinase JAK3 | 6AAKD | 2.67 | Active | DFGin | BLAminus | in-in | in-in | 9T6 | Type1 |
Homo sapiens | TYR | TYK2 | TYK2_HUMAN | Non-receptor tyrosine-protein kinase TYK2 | 6AAMA | 1.98 | None | DFGin | BLAminus | in-in | in-none | 9T6 | Type1 |
Spatial | Dihedral | Chains | Representative |
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Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
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