| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| RAF1 | AF-P04049-K1A | P04049 | 341 | 616 | 648.0 | No_ligand | No_ligand | Active | DFGin | 6.5203 | 13.7817 | BLAminus | -132.07, -167.34 | 50.52, 81.79 | -93.0, 17.5 | 287.63, 84.75 | -60.82, -26.68 | in-in | in | 8.771 | Saltbr-in | 2.7908 | HRD-in | -75.2, -41.77 | 65.71, -17.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.891 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -82.32, 124.86 | APE9-dihe-na | 150.0, -177.65 | APE8-dihe-in | -88.86, 110.11 | APE8-rot-in | 297.22 | APE67-dihe-in | -59.64, -29.86 | -48.29, -38.25 | APE12-dist-in | 13.3725 | APE11-dist-in | 11.5758 | APE10-dist-in | 7.2465 | APE9-dist-in | 5.6357 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | AF-P04049-K1 | TKL_RAF1_HUMAN | TKL | 2.5e-81 | 279.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | AF-P04049-K3A | P04049 | 341 | 616 | 648.0 | No_ligand | No_ligand | Active | DFGin | 6.6956 | 13.8203 | BLAminus | -127.79, -164.94 | 51.29, 73.3 | -87.25, 15.65 | 292.37, 90.99 | -61.36, -23.57 | in-in | in | 9.3042 | Saltbr-in | 2.9127 | HRD-in | -75.32, -37.72 | 66.17, -19.03 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9047 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.73, 136.21 | APE9-dihe-na | 118.54, -171.69 | APE8-dihe-in | -96.47, 111.5 | APE8-rot-in | 306.19 | APE67-dihe-in | -65.71, -24.96 | -56.51, -31.57 | APE12-dist-in | 12.8315 | APE11-dist-in | 12.1084 | APE10-dist-in | 6.6368 | APE9-dist-in | 4.1332 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | AF-P04049-K3 | TKL_RAF1_HUMAN | TKL | 2.5e-81 | 279.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AYAA | P04049 | 342 | 614 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.3662 | 14.2668 | BLAminus | -136.12, -165.85 | 49.32, 86.99 | -103.48, 21.74 | 291.83, 76.13 | -59.74, -18.47 | in-none | in | 9.0808 | Saltbr-none | 999.0 | HRD-in | -71.73, -48.54 | 69.99, 0.7 | none-in-out | SNCnio | in-out | ActLoopNT-in | 2.8942 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioi | APE10-dihe-na | -128.07, 13.13 | APE9-dihe-na | -91.19, -175.11 | APE8-dihe-in | -69.87, 137.88 | APE8-rot-in | 300.15 | APE67-dihe-in | -63.77, -25.92 | -71.38, -32.74 | APE12-dist-in | 12.5452 | APE11-dist-in | 9.8883 | APE10-dist-out | 8.8439 | APE9-dist-in | 5.9778 | Y340D,Y341D | None | None | XRAY | 2.59 | 0.214 | 0.257 | A | 280.0 | 267.0 | 6 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9aya | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AYAC | P04049 | 341 | 613 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5551 | 14.821 | BLAminus | -133.94, -166.68 | 54.0, 73.37 | -92.76, 23.95 | 288.97, 82.99 | -61.86, -28.32 | in-in | in | 8.7648 | Saltbr-in | 2.8037 | HRD-in | -69.13, -44.61 | 68.35, -7.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8119 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 53.27, 27.21 | APE9-dihe-na | -96.24, -140.6 | APE8-dihe-in | -94.61, 133.74 | APE8-rot-out | 177.74 | APE67-dihe-in | -62.64, -31.47 | -74.96, -14.97 | APE12-dist-in | 12.0325 | APE11-dist-in | 8.2808 | APE10-dist-out | 10.5493 | APE9-dist-out | 7.7979 | Y340D,Y341D | None | None | XRAY | 2.59 | 0.214 | 0.257 | C | 280.0 | 263.0 | 10 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9aya | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AXAA | P04049 | 342 | 625 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.2548 | 13.9989 | BLAminus | -139.05, -163.7 | 58.24, 64.96 | -89.4, 29.46 | 290.36, 82.23 | -69.56, -16.76 | in-out | in | 9.18 | Saltbr-out | 8.4188 | HRD-in | -78.78, -32.03 | 70.97, -14.05 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.116 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioo | APE10-dihe-na | -130.3, -20.74 | APE9-dihe-na | -70.73, -178.58 | APE8-dihe-in | -67.69, 139.48 | APE8-rot-in | 293.88 | APE67-dihe-in | -69.75, -43.45 | -74.78, -4.77 | APE12-dist-in | 12.0486 | APE11-dist-in | 9.617 | APE10-dist-out | 9.0441 | APE9-dist-out | 7.5911 | Y340D,Y341D | SEP621 | SEP621 | EM | 4.36 | 999.0 | 999.0 | A | 563.0 | 273.0 | 11 | 30 | 25 | 5 | [[349, 608]] | 1.0 | 9axa | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AXAC | P04049 | 341 | 625 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.3924 | 14.9903 | BLAminus | -146.66, -157.9 | 56.49, 63.39 | -91.79, 31.37 | 293.16, 80.76 | -67.87, -25.57 | in-out | in | 8.9755 | Saltbr-out | 10.0011 | HRD-in | -78.03, -41.77 | 71.76, -11.87 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.7588 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 54.52, 48.67 | APE9-dihe-na | -119.18, -141.08 | APE8-dihe-in | -96.15, 129.35 | APE8-rot-out | 174.93 | APE67-dihe-in | -72.88, -14.72 | -74.49, -3.91 | APE12-dist-in | 11.8542 | APE11-dist-in | 9.1816 | APE10-dist-out | 11.2816 | APE9-dist-out | 9.0508 | Y340D,Y341D | SEP621 | SEP621 | EM | 4.36 | 999.0 | 999.0 | C | 563.0 | 275.0 | 10 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9axa | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AXCA | P04049 | 342 | 614 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.1921 | 14.4156 | BLAminus | -138.33, -166.81 | 57.53, 66.49 | -89.8, 33.05 | 291.57, 76.32 | -64.02, -29.91 | in-out | in | 9.5136 | Saltbr-out | 7.6297 | HRD-in | -72.6, -42.02 | 72.95, -10.85 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.1646 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioo | APE10-dihe-na | -134.52, -16.63 | APE9-dihe-na | -73.85, -175.48 | APE8-dihe-in | -71.62, 149.24 | APE8-rot-in | 297.36 | APE67-dihe-in | -71.32, -46.0 | -82.78, -6.02 | APE12-dist-in | 12.2652 | APE11-dist-in | 10.7655 | APE10-dist-out | 9.0117 | APE9-dist-out | 7.1409 | Y340D,Y341D | None | None | EM | 4.16 | 999.0 | 999.0 | A | 563.0 | 262.0 | 11 | 30 | 25 | 5 | [[349, 608]] | 1.0 | 9axc | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AXCC | P04049 | 341 | 614 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.0993 | 14.2941 | BLAminus | -140.87, -159.63 | 58.35, 65.16 | -89.93, 32.3 | 288.78, 78.02 | -61.68, -35.06 | in-out | in | 8.1468 | Saltbr-out | 3.9477 | HRD-in | -77.54, -28.87 | 66.49, -1.91 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.6755 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 42.59, 31.87 | APE9-dihe-na | -96.68, -133.02 | APE8-dihe-in | -109.92, 127.09 | APE8-rot-out | 177.26 | APE67-dihe-in | -75.55, -23.65 | -73.76, -3.99 | APE12-dist-in | 11.8637 | APE11-dist-in | 8.5952 | APE10-dist-out | 11.1083 | APE9-dist-out | 8.7613 | Y340D,Y341D | None | None | EM | 4.16 | 999.0 | 999.0 | C | 563.0 | 264.0 | 10 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9axc | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0UG | P04049 | 341 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.6427 | 14.5362 | BLAminus | -137.03, -164.72 | 64.05, 59.07 | -91.31, 23.03 | 298.27, 111.42 | -70.02, -22.85 | in-in | in | 8.466 | Saltbr-in | 2.7929 | HRD-in | -67.69, -46.18 | 73.87, -6.26 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.4083 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -147.61, -172.9 | APE9-dihe-na | 96.11, -111.47 | APE8-dihe-in | -121.52, 159.07 | APE8-rot-out | 179.33 | APE67-dihe-in | -61.77, -27.13 | -108.62, -7.48 | APE12-dist-in | 9.3284 | APE11-dist-in | 9.0351 | APE10-dist-out | 10.4777 | APE9-dist-out | 9.744 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | G | 280.0 | 265.0 | 9 | 30 | 21 | 9 | [[349, 608]] | 1.0 | 9o0u | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0VG | P04049 | 341 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.6518 | 14.5256 | BLAminus | -136.91, -164.75 | 63.88, 58.79 | -91.51, 23.22 | 298.64, 111.76 | -69.75, -22.63 | in-in | in | 8.5288 | Saltbr-in | 2.8267 | HRD-in | -68.13, -46.19 | 73.7, -5.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.3624 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -144.93, -171.41 | APE9-dihe-na | 95.72, -110.34 | APE8-dihe-in | -121.89, 159.4 | APE8-rot-out | 179.42 | APE67-dihe-in | -62.17, -27.08 | -108.22, -7.65 | APE12-dist-in | 9.3788 | APE11-dist-in | 8.988 | APE10-dist-out | 10.4038 | APE9-dist-out | 9.6609 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | G | 280.0 | 265.0 | 9 | 30 | 21 | 9 | [[349, 608]] | 1.0 | 9o0v | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 3OMVB | P04049 | 340 | 615 | 648.0 | SM5:2 | Type1 | Inactive | DFGin | 6.2314 | 14.1198 | BLAminus | -128.39, -171.12 | 47.91, 84.95 | -94.99, 35.62 | 285.33, 59.46 | -60.18, -20.41 | in-in | in | 8.4734 | Saltbr-in | 2.9066 | HRD-in | -95.5, -25.99 | 55.76, -81.98 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.4203 | ActLoopCT-out | nonTYR | APEdihe_aaioo | APEdist_nooo | APE10-dihe-na | -64.38, 160.65 | APE9-dihe-na | -138.85, -166.53 | APE8-dihe-in | -147.75, 73.1 | APE8-rot-out | 58.68 | APE67-dihe-out | 164.31, -56.84 | -70.36, 119.54 | APE12-dist-none | 999.0 | APE11-dist-out | 14.3402 | APE10-dist-out | 13.4894 | APE9-dist-out | 10.3958 | None | None | None | XRAY | 4.0 | 0.283 | 0.364 | B | 307.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 3omv | TKL_RAF1_HUMAN | TKL | 3.7e-81 | 278.6 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0UE | P04049 | 339 | 613 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.9555 | 13.4189 | BLAplus | -138.96, -169.14 | 62.02, 34.27 | -105.27, 31.97 | 55.75, 93.21 | -64.59, -47.5 | out-none | out | 11.6319 | Saltbr-none | 999.0 | HRD-in | -66.55, -46.99 | 72.02, -8.83 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -79.43 | APE8-dihe-in | -132.83, 160.57 | APE8-rot-out | 180.68 | APE67-dihe-in | -62.16, -27.71 | -107.14, -6.5 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.74 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | E | 280.0 | 258.0 | 17 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 9o0u | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0VE | P04049 | 339 | 613 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.8024 | 13.3404 | BLAplus | -138.88, -169.03 | 61.87, 34.79 | -104.64, 32.35 | 56.09, 93.36 | -64.43, -47.67 | out-none | out | 11.5845 | Saltbr-none | 999.0 | HRD-in | -66.6, -47.0 | 72.05, -8.97 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 56.8, 24.32 | APE9-dihe-na | -101.33, -80.31 | APE8-dihe-in | -132.61, 160.7 | APE8-rot-out | 180.75 | APE67-dihe-in | -62.26, -27.57 | -106.96, -6.66 | APE12-dist-in | 11.2624 | APE11-dist-in | 9.0411 | APE10-dist-out | 12.024 | APE9-dist-out | 9.4519 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | E | 280.0 | 261.0 | 14 | 30 | 16 | 14 | [[349, 608]] | 1.0 | 9o0v | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0UC | P04049 | 339 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.4118 | 14.92 | BLBminus | -135.2, -162.93 | 65.39, 47.79 | -89.17, 153.49 | 305.13, 119.24 | 148.83, -36.3 | in-in | in | 8.1119 | Saltbr-in | 3.1081 | HRD-in | -65.51, -42.52 | 74.23, -8.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.2736 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -140.95 | APE9-dihe-na | 87.04, -108.57 | APE8-dihe-in | -126.35, 163.82 | APE8-rot-out | 179.91 | APE67-dihe-in | -66.05, -28.24 | -108.28, -15.46 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 9.537 | APE9-dist-out | 7.8436 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | C | 280.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 9o0u | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0VC | P04049 | 339 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.507 | 14.8484 | BLBminus | -135.62, -163.14 | 65.12, 48.02 | -88.94, 153.23 | 304.77, 118.58 | 148.73, -35.99 | in-in | in | 8.1644 | Saltbr-in | 3.3442 | HRD-in | -65.49, -42.82 | 73.84, -8.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.3433 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -150.01 | APE9-dihe-na | 93.34, -107.4 | APE8-dihe-in | -126.38, 163.35 | APE8-rot-out | 180.01 | APE67-dihe-in | -65.89, -28.16 | -108.44, -15.01 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 9.4019 | APE9-dist-out | 7.9115 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | C | 280.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 9o0v | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9AY7A | P04049 | 343 | 612 | 648.0 | ANP:701 | ATPlike | Inactive | DFGin | 5.8053 | 13.462 | BLBplus | -133.55, 174.37 | 58.47, 38.44 | -90.49, 142.18 | 44.05, 90.72 | 78.29, -134.9 | out-out | out | 14.0699 | Saltbr-out | 12.7376 | HRD-in | -73.02, -44.7 | 76.86, -25.12 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.1822 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -145.48, 130.61 | APE9-dihe-na | 129.03, -169.57 | APE8-dihe-in | -79.63, 137.79 | APE8-rot-in | 302.79 | APE67-dihe-in | -63.4, -34.24 | -69.33, -38.68 | APE12-dist-out | 15.2361 | APE11-dist-out | 15.0562 | APE10-dist-out | 10.6236 | APE9-dist-out | 6.3059 | Y340D,Y341D | None | None | XRAY | 2.41 | 0.203 | 0.236 | A | 280.0 | 260.0 | 10 | 30 | 24 | 6 | [[349, 608]] | 1.0 | 9ay7 | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9MMRA | P04049 | 343 | 625 | 648.0 | AGS:60701 | ATPlike | Inactive | DFGin | 5.4464 | 13.6261 | BLBplus | -135.09, 172.16 | 58.87, 36.16 | -92.53, 159.81 | 52.16, 102.21 | 63.65, -134.37 | out-out | out | 13.8632 | Saltbr-out | 12.3622 | HRD-out | -74.45, 80.03 | -68.85, 163.44 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.7183 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -153.07, 160.07 | APE9-dihe-na | 91.95, -174.93 | APE8-dihe-in | -63.61, 140.51 | APE8-rot-in | 299.95 | APE67-dihe-in | -59.35, -38.77 | -86.72, -25.37 | APE12-dist-out | 15.0543 | APE11-dist-out | 14.7515 | APE10-dist-out | 11.0339 | APE9-dist-out | 8.4046 | Q156R,Y340D,Y341D,D587E | SEP621 | SEP621 | EM | 3.9 | 999.0 | 999.0 | A | 681.0 | 283.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mmr | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9MMSA | P04049 | 343 | 610 | 648.0 | AGS:701 | ATPlike | Inactive | DFGin | 6.0432 | 13.4123 | BLBplus | -130.72, 176.22 | 57.09, 37.64 | -95.88, 150.42 | 38.9, 90.55 | 70.15, -138.14 | out-out | out | 13.239 | Saltbr-out | 11.9633 | HRD-out | -75.89, 77.72 | -68.75, 167.65 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.0132 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -153.3, 137.93 | APE9-dihe-na | 117.05, 178.36 | APE8-dihe-in | -66.7, 143.78 | APE8-rot-in | 289.18 | APE67-dihe-in | -66.49, -26.11 | -89.17, -21.29 | APE12-dist-out | 15.1652 | APE11-dist-out | 14.8651 | APE10-dist-out | 10.7824 | APE9-dist-out | 8.09 | Q156R,Y340D,Y341D,D587E | None | None | EM | 3.3 | 999.0 | 999.0 | A | 681.0 | 268.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mms | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9MMQA | P04049 | 341 | 612 | 648.0 | AGS:701 | ATPlike | Inactive | DFGin | 6.0418 | 13.4878 | BLBplus | -128.47, 173.58 | 60.41, 41.33 | -95.4, 154.76 | 40.5, 88.25 | 68.22, -137.22 | out-out | out | 13.7306 | Saltbr-out | 12.7147 | HRD-out | -73.84, 78.36 | -65.55, 163.21 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.1331 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -154.13, 160.3 | APE9-dihe-na | 98.38, -176.64 | APE8-dihe-in | -67.06, 138.58 | APE8-rot-in | 288.86 | APE67-dihe-in | -64.64, -31.65 | -87.38, -18.69 | APE12-dist-out | 15.1677 | APE11-dist-out | 14.4229 | APE10-dist-out | 10.8266 | APE9-dist-out | 8.1068 | Q156R,D587E | None | None | EM | 2.9 | 999.0 | 999.0 | A | 681.0 | 272.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mmq | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9MMPA | P04049 | 138 | 630 | 648.0 | AGS:60701 | ATPlike | Inactive | DFGin | 6.1073 | 13.2684 | BLBplus | -130.39, 177.17 | 56.68, 47.87 | -99.84, 149.88 | 40.92, 87.91 | 73.17, -140.77 | out-out | out | 14.3612 | Saltbr-out | 12.3822 | HRD-out | -74.8, 81.36 | -67.74, 154.91 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.1666 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -156.54, 146.13 | APE9-dihe-na | 117.78, -173.39 | APE8-dihe-in | -67.5, 146.42 | APE8-rot-in | 282.71 | APE67-dihe-in | -62.97, -41.04 | -80.62, -35.94 | APE12-dist-out | 14.2949 | APE11-dist-out | 14.3656 | APE10-dist-out | 10.6756 | APE9-dist-out | 7.9092 | Q156R,D587E | SEP259,SEP621 | SEP259,SEP621 | EM | 3.4 | 999.0 | 999.0 | A | 683.0 | 348.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mmp | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0UA | P04049 | 339 | 612 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.49 | 13.4253 | BLBplus | -137.77, -168.21 | 60.54, 23.67 | -97.39, 164.85 | 62.85, 94.03 | 74.33, 173.3 | out-none | out | 11.6361 | Saltbr-none | 999.0 | HRD-in | -67.32, -47.26 | 72.53, -10.19 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 8.5215 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -79.91, 164.26 | APE9-dihe-na | 133.94, -179.25 | APE8-dihe-in | -151.13, 161.47 | APE8-rot-out | 181.14 | APE67-dihe-in | -63.28, -28.75 | -107.76, -7.41 | APE12-dist-out | 21.2876 | APE11-dist-out | 15.3594 | APE10-dist-out | 15.2178 | APE9-dist-out | 10.0158 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | A | 280.0 | 267.0 | 7 | 30 | 23 | 7 | [[349, 608]] | 1.0 | 9o0u | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 9O0VA | P04049 | 339 | 612 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.6121 | 13.5412 | BLBplus | -137.53, -168.14 | 60.68, 23.81 | -97.37, 165.11 | 62.5, 93.91 | 74.63, 173.9 | out-none | out | 11.5178 | Saltbr-none | 999.0 | HRD-in | -67.23, -47.12 | 72.36, -10.39 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 8.5821 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oioo | APE10-dihe-na | -121.31, 23.23 | APE9-dihe-na | -94.2, -61.86 | APE8-dihe-in | -150.39, 162.26 | APE8-rot-out | 181.1 | APE67-dihe-in | -63.35, -28.52 | -106.79, -7.22 | APE12-dist-out | 14.0563 | APE11-dist-in | 11.3326 | APE10-dist-out | 13.0181 | APE9-dist-out | 9.5213 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | A | 280.0 | 266.0 | 8 | 30 | 22 | 8 | [[349, 608]] | 1.0 | 9o0v | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8CPDA | P04049 | 341 | 626 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.2527 | 14.8427 | None | -88.44, -129.65 | -68.47, 153.64 | -115.46, 32.54 | 280.62, 22.29 | -59.2, -38.85 | in-in | in | 8.9962 | Saltbr-in | 3.2393 | HRD-out | -71.21, -9.87 | 61.06, -133.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.3344 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, -31.3 | APE9-dihe-na | -64.2, -40.67 | APE8-dihe-in | -125.25, 125.51 | APE8-rot-in | 293.24 | APE67-dihe-in | -70.13, -31.13 | -109.07, 11.27 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 13.0605 | APE9-dist-out | 15.3926 | Y341D | SEP621 | SEP621 | EM | 3.46 | 999.0 | 999.0 | A | 648.0 | 269.0 | 17 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 8cpd | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8CPDB | P04049 | 341 | 626 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.3243 | 14.7834 | None | -88.37, -130.06 | -68.25, 153.07 | -115.22, 33.93 | 283.48, 10.19 | -59.44, -38.94 | in-in | in | 8.9968 | Saltbr-in | 3.2413 | HRD-out | -70.18, -11.24 | 60.41, -132.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.2815 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, -32.01 | APE9-dihe-na | -64.34, -40.91 | APE8-dihe-in | -123.99, 124.82 | APE8-rot-in | 292.66 | APE67-dihe-in | -70.59, -30.16 | -110.37, 10.88 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 13.0602 | APE9-dist-out | 15.4329 | Y341D | SEP621 | SEP621 | EM | 3.46 | 999.0 | 999.0 | B | 648.0 | 269.0 | 17 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 8cpd | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 3OMVA | P04049 | 340 | 615 | 648.0 | SM5:1 | Type1 | Inactive | DFGin | 6.0105 | 14.0395 | None | -72.19, -157.95 | -69.65, 158.45 | -112.95, 18.14 | 298.92, 73.64 | -38.54, -34.68 | in-in | in | 8.8405 | Saltbr-in | 2.8181 | HRD-in | -81.59, -27.52 | 64.4, -79.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.128 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nioo | APE10-dihe-na | -67.59, 120.25 | APE9-dihe-na | -106.5, 137.12 | APE8-dihe-in | -106.61, 64.59 | APE8-rot-out | 44.73 | APE67-dihe-inflip | 112.91, -48.44 | -57.65, 161.85 | APE12-dist-none | 999.0 | APE11-dist-in | 13.3289 | APE10-dist-out | 12.1479 | APE9-dist-out | 10.4545 | None | None | None | XRAY | 4.0 | 0.283 | 0.364 | A | 307.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 3omv | TKL_RAF1_HUMAN | TKL | 3.7e-81 | 278.6 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8CHFA | P04049 | 341 | 626 | 648.0 | 29L:60701 | Type1 | Inactive | DFGin | 6.9193 | 13.7979 | None | -77.69, -137.87 | -62.1, 150.83 | -123.34, 43.11 | 304.09, 90.48 | -53.76, -47.63 | in-out | in | 8.5922 | Saltbr-out | 6.6899 | HRD-in | -62.51, -43.32 | 69.96, -9.45 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8262 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiio | APE10-dihe-na | 55.74, 2.9 | APE9-dihe-na | 55.92, 40.68 | APE8-dihe-in | -131.33, 94.1 | APE8-rot-out | 59.25 | APE67-dihe-inflip | 81.42, -0.92 | -97.97, 165.62 | APE12-dist-in | 7.3494 | APE11-dist-in | 11.6311 | APE10-dist-in | 6.9434 | APE9-dist-out | 10.1571 | Y341D | SEP621 | SEP621 | EM | 4.25 | 0.445 | 999.0 | A | 648.0 | 280.0 | 6 | 30 | 24 | 6 | [[349, 608]] | 1.0 | 8chf | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8CHFB | P04049 | 341 | 626 | 648.0 | 29L:60701 | Type1 | Inactive | DFGin | 6.9191 | 13.7979 | None | -77.67, -137.85 | -62.16, 150.83 | -123.29, 43.03 | 304.08, 90.5 | -53.73, -47.64 | in-out | in | 8.5922 | Saltbr-out | 6.6905 | HRD-in | -62.53, -43.31 | 69.92, -9.4 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8268 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiio | APE10-dihe-na | 55.74, 2.9 | APE9-dihe-na | 55.89, 40.65 | APE8-dihe-in | -131.28, 94.15 | APE8-rot-out | 59.25 | APE67-dihe-inflip | 81.39, -0.89 | -98.01, 165.61 | APE12-dist-in | 7.3494 | APE11-dist-in | 11.631 | APE10-dist-in | 6.9423 | APE9-dist-out | 10.1569 | Y341D | SEP621 | SEP621 | EM | 4.25 | 0.445 | 999.0 | B | 648.0 | 280.0 | 6 | 30 | 24 | 6 | [[349, 608]] | 1.0 | 8chf | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8GFTD | P04049 | 404 | 611 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -164.39, -179.79 | -89.82, 12.52 | -72.24, -18.95 | 181.77, 70.31 | -73.4, 999.0 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -68.87, -46.27 | 64.82, -56.23 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, -56.49 | APE9-dihe-na | 100.69, -17.61 | APE8-dihe-out | -72.27, -36.0 | APE8-rot-out | 67.45 | APE67-dihe-in | -49.85, -47.25 | -97.25, -47.78 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.5368 | None | None | None | EM | 3.8 | 999.0 | 999.0 | D | 304.0 | 191.0 | 72 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 8gft | TKL_RAF1_HUMAN | TKL | 3.6e-81 | 278.6 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8U1LC | P04049 | 418 | 615 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | 87.15, 3.03 | -74.84, 77.99 | -74.97, 76.67 | 289.42, 93.79 | 116.56, -171.97 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-out | -100.67, 144.24 | -121.66, -8.0 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nooo | APE10-dihe-na | 51.33, 57.43 | APE9-dihe-na | 61.35, -123.96 | APE8-dihe-out | 55.11, 35.51 | APE8-rot-in | 302.03 | APE67-dihe-in | -59.19, -23.13 | -70.4, -10.97 | APE12-dist-none | 999.0 | APE11-dist-out | 19.2568 | APE10-dist-out | 16.2609 | APE9-dist-out | 9.904 | None | None | None | EM | 3.7 | 999.0 | 999.0 | C | 656.0 | 184.0 | 83 | 30 | 16 | 14 | [[349, 608]] | 1.0 | 8u1l | TKL_RAF1_HUMAN | TKL | 3.1e-80 | 275.7 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 7Z37CP1 | P04049 | 406 | 615 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -51.69, 113.04 | -59.31, 132.91 | -63.39, -37.52 | 182.06, 73.21 | 115.94, -41.02 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -94.28, -51.52 | 64.79, -72.58 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -172.19 | APE8-rot-out | 162.56 | APE67-dihe-inflip | 70.01, -5.7 | -83.36, 166.62 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | EM | 3.67 | 999.0 | 999.0 | CP1 | 659.0 | 193.0 | 74 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 7z37 | TKL_RAF1_HUMAN | TKL | 1e-79 | 274.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 7Z38C | P04049 | 406 | 615 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -54.5, 132.93 | -69.32, 104.66 | -85.43, 53.34 | 267.31, 92.72 | 60.74, -125.52 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -113.4, -61.21 | 60.49, -2.03 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -92.5 | APE8-rot-out | 164.68 | APE67-dihe-inflip | 72.83, -7.22 | -110.4, 137.31 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | EM | 3.16 | 999.0 | 999.0 | C | 659.0 | 193.0 | 74 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 7z38 | TKL_RAF1_HUMAN | TKL | 1e-79 | 274.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | 8GAED | P04049 | 404 | 610 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -126.25, -170.67 | -128.75, -9.64 | -62.05, -51.04 | 170.23, 78.51 | 57.98, 999.0 | none-na | none | 999.0 | Saltbr-na | 999.0 | HRD-out | -112.46, 123.69 | -73.96, 156.28 | na-none-out | SNCano | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioo | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -175.21 | APE8-dihe-in | -78.72, 159.13 | APE8-rot-out | 52.86 | APE67-dihe-out | -91.67, 147.13 | -88.13, 88.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 16.09 | None | None | None | EM | 3.3 | 999.0 | 999.0 | D | 207.0 | 189.0 | 18 | 30 | 12 | 18 | [[349, 608]] | 1.0 | 8gae | TKL_RAF1_HUMAN | TKL | 4e-62 | 216.0 | 57.0 | 266.0 | 210.0 | 485 | 486 | 487 | 489 | 491 | 0 | 0 | 0 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| RAF1 | RAF1_HUMAN | AF-P04049-K1A | P04049 | 341 | 616 | 648.0 | No_ligand | No_ligand | Active | DFGin | 6.5203 | 13.7817 | BLAminus | -132.07, -167.34 | 50.52, 81.79 | -93.0, 17.5 | 287.63, 84.75 | -60.82, -26.68 | in-in | in | 8.771 | Saltbr-in | 2.7908 | HRD-in | -75.2, -41.77 | 65.71, -17.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.891 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -82.32, 124.86 | APE9-dihe-na | 150.0, -177.65 | APE8-dihe-in | -88.86, 110.11 | APE8-rot-in | 297.22 | APE67-dihe-in | -59.64, -29.86 | -48.29, -38.25 | APE12-dist-in | 13.3725 | APE11-dist-in | 11.5758 | APE10-dist-in | 7.2465 | APE9-dist-in | 5.6357 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | AF-P04049-K1 | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.5e-81 | 279.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | AF-P04049-K3A | P04049 | 341 | 616 | 648.0 | No_ligand | No_ligand | Active | DFGin | 6.6956 | 13.8203 | BLAminus | -127.79, -164.94 | 51.29, 73.3 | -87.25, 15.65 | 292.37, 90.99 | -61.36, -23.57 | in-in | in | 9.3042 | Saltbr-in | 2.9127 | HRD-in | -75.32, -37.72 | 66.17, -19.03 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9047 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.73, 136.21 | APE9-dihe-na | 118.54, -171.69 | APE8-dihe-in | -96.47, 111.5 | APE8-rot-in | 306.19 | APE67-dihe-in | -65.71, -24.96 | -56.51, -31.57 | APE12-dist-in | 12.8315 | APE11-dist-in | 12.1084 | APE10-dist-in | 6.6368 | APE9-dist-in | 4.1332 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | AF-P04049-K3 | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.5e-81 | 279.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AYAA | P04049 | 342 | 614 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.3662 | 14.2668 | BLAminus | -136.12, -165.85 | 49.32, 86.99 | -103.48, 21.74 | 291.83, 76.13 | -59.74, -18.47 | in-none | in | 9.0808 | Saltbr-none | 999.0 | HRD-in | -71.73, -48.54 | 69.99, 0.7 | none-in-out | SNCnio | in-out | ActLoopNT-in | 2.8942 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioi | APE10-dihe-na | -128.07, 13.13 | APE9-dihe-na | -91.19, -175.11 | APE8-dihe-in | -69.87, 137.88 | APE8-rot-in | 300.15 | APE67-dihe-in | -63.77, -25.92 | -71.38, -32.74 | APE12-dist-in | 12.5452 | APE11-dist-in | 9.8883 | APE10-dist-out | 8.8439 | APE9-dist-in | 5.9778 | Y340D,Y341D | None | None | XRAY | 2.59 | 0.214 | 0.257 | A | 280.0 | 267.0 | 6 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9aya | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AYAC | P04049 | 341 | 613 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5551 | 14.821 | BLAminus | -133.94, -166.68 | 54.0, 73.37 | -92.76, 23.95 | 288.97, 82.99 | -61.86, -28.32 | in-in | in | 8.7648 | Saltbr-in | 2.8037 | HRD-in | -69.13, -44.61 | 68.35, -7.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8119 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 53.27, 27.21 | APE9-dihe-na | -96.24, -140.6 | APE8-dihe-in | -94.61, 133.74 | APE8-rot-out | 177.74 | APE67-dihe-in | -62.64, -31.47 | -74.96, -14.97 | APE12-dist-in | 12.0325 | APE11-dist-in | 8.2808 | APE10-dist-out | 10.5493 | APE9-dist-out | 7.7979 | Y340D,Y341D | None | None | XRAY | 2.59 | 0.214 | 0.257 | C | 280.0 | 263.0 | 10 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9aya | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AXAA | P04049 | 342 | 625 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.2548 | 13.9989 | BLAminus | -139.05, -163.7 | 58.24, 64.96 | -89.4, 29.46 | 290.36, 82.23 | -69.56, -16.76 | in-out | in | 9.18 | Saltbr-out | 8.4188 | HRD-in | -78.78, -32.03 | 70.97, -14.05 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.116 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioo | APE10-dihe-na | -130.3, -20.74 | APE9-dihe-na | -70.73, -178.58 | APE8-dihe-in | -67.69, 139.48 | APE8-rot-in | 293.88 | APE67-dihe-in | -69.75, -43.45 | -74.78, -4.77 | APE12-dist-in | 12.0486 | APE11-dist-in | 9.617 | APE10-dist-out | 9.0441 | APE9-dist-out | 7.5911 | Y340D,Y341D | SEP621 | SEP621 | EM | 4.36 | 999.0 | 999.0 | A | 563.0 | 273.0 | 11 | 30 | 25 | 5 | [[349, 608]] | 1.0 | 9axa | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AXAC | P04049 | 341 | 625 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.3924 | 14.9903 | BLAminus | -146.66, -157.9 | 56.49, 63.39 | -91.79, 31.37 | 293.16, 80.76 | -67.87, -25.57 | in-out | in | 8.9755 | Saltbr-out | 10.0011 | HRD-in | -78.03, -41.77 | 71.76, -11.87 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.7588 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 54.52, 48.67 | APE9-dihe-na | -119.18, -141.08 | APE8-dihe-in | -96.15, 129.35 | APE8-rot-out | 174.93 | APE67-dihe-in | -72.88, -14.72 | -74.49, -3.91 | APE12-dist-in | 11.8542 | APE11-dist-in | 9.1816 | APE10-dist-out | 11.2816 | APE9-dist-out | 9.0508 | Y340D,Y341D | SEP621 | SEP621 | EM | 4.36 | 999.0 | 999.0 | C | 563.0 | 275.0 | 10 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9axa | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AXCA | P04049 | 342 | 614 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.1921 | 14.4156 | BLAminus | -138.33, -166.81 | 57.53, 66.49 | -89.8, 33.05 | 291.57, 76.32 | -64.02, -29.91 | in-out | in | 9.5136 | Saltbr-out | 7.6297 | HRD-in | -72.6, -42.02 | 72.95, -10.85 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.1646 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioo | APE10-dihe-na | -134.52, -16.63 | APE9-dihe-na | -73.85, -175.48 | APE8-dihe-in | -71.62, 149.24 | APE8-rot-in | 297.36 | APE67-dihe-in | -71.32, -46.0 | -82.78, -6.02 | APE12-dist-in | 12.2652 | APE11-dist-in | 10.7655 | APE10-dist-out | 9.0117 | APE9-dist-out | 7.1409 | Y340D,Y341D | None | None | EM | 4.16 | 999.0 | 999.0 | A | 563.0 | 262.0 | 11 | 30 | 25 | 5 | [[349, 608]] | 1.0 | 9axc | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AXCC | P04049 | 341 | 614 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 7.0993 | 14.2941 | BLAminus | -140.87, -159.63 | 58.35, 65.16 | -89.93, 32.3 | 288.78, 78.02 | -61.68, -35.06 | in-out | in | 8.1468 | Saltbr-out | 3.9477 | HRD-in | -77.54, -28.87 | 66.49, -1.91 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.6755 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 42.59, 31.87 | APE9-dihe-na | -96.68, -133.02 | APE8-dihe-in | -109.92, 127.09 | APE8-rot-out | 177.26 | APE67-dihe-in | -75.55, -23.65 | -73.76, -3.99 | APE12-dist-in | 11.8637 | APE11-dist-in | 8.5952 | APE10-dist-out | 11.1083 | APE9-dist-out | 8.7613 | Y340D,Y341D | None | None | EM | 4.16 | 999.0 | 999.0 | C | 563.0 | 264.0 | 10 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9axc | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.2e-80 | 276.1 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0UG | P04049 | 341 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.6427 | 14.5362 | BLAminus | -137.03, -164.72 | 64.05, 59.07 | -91.31, 23.03 | 298.27, 111.42 | -70.02, -22.85 | in-in | in | 8.466 | Saltbr-in | 2.7929 | HRD-in | -67.69, -46.18 | 73.87, -6.26 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.4083 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -147.61, -172.9 | APE9-dihe-na | 96.11, -111.47 | APE8-dihe-in | -121.52, 159.07 | APE8-rot-out | 179.33 | APE67-dihe-in | -61.77, -27.13 | -108.62, -7.48 | APE12-dist-in | 9.3284 | APE11-dist-in | 9.0351 | APE10-dist-out | 10.4777 | APE9-dist-out | 9.744 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | G | 280.0 | 265.0 | 9 | 30 | 21 | 9 | [[349, 608]] | 1.0 | 9o0u | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0VG | P04049 | 341 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.6518 | 14.5256 | BLAminus | -136.91, -164.75 | 63.88, 58.79 | -91.51, 23.22 | 298.64, 111.76 | -69.75, -22.63 | in-in | in | 8.5288 | Saltbr-in | 2.8267 | HRD-in | -68.13, -46.19 | 73.7, -5.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.3624 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -144.93, -171.41 | APE9-dihe-na | 95.72, -110.34 | APE8-dihe-in | -121.89, 159.4 | APE8-rot-out | 179.42 | APE67-dihe-in | -62.17, -27.08 | -108.22, -7.65 | APE12-dist-in | 9.3788 | APE11-dist-in | 8.988 | APE10-dist-out | 10.4038 | APE9-dist-out | 9.6609 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | G | 280.0 | 265.0 | 9 | 30 | 21 | 9 | [[349, 608]] | 1.0 | 9o0v | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 3OMVB | P04049 | 340 | 615 | 648.0 | SM5:2 | Type1 | Inactive | DFGin | 6.2314 | 14.1198 | BLAminus | -128.39, -171.12 | 47.91, 84.95 | -94.99, 35.62 | 285.33, 59.46 | -60.18, -20.41 | in-in | in | 8.4734 | Saltbr-in | 2.9066 | HRD-in | -95.5, -25.99 | 55.76, -81.98 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.4203 | ActLoopCT-out | nonTYR | APEdihe_aaioo | APEdist_nooo | APE10-dihe-na | -64.38, 160.65 | APE9-dihe-na | -138.85, -166.53 | APE8-dihe-in | -147.75, 73.1 | APE8-rot-out | 58.68 | APE67-dihe-out | 164.31, -56.84 | -70.36, 119.54 | APE12-dist-none | 999.0 | APE11-dist-out | 14.3402 | APE10-dist-out | 13.4894 | APE9-dist-out | 10.3958 | None | None | None | XRAY | 4.0 | 0.283 | 0.364 | B | 307.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 3omv | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3.7e-81 | 278.6 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0UE | P04049 | 339 | 613 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.9555 | 13.4189 | BLAplus | -138.96, -169.14 | 62.02, 34.27 | -105.27, 31.97 | 55.75, 93.21 | -64.59, -47.5 | out-none | out | 11.6319 | Saltbr-none | 999.0 | HRD-in | -66.55, -46.99 | 72.02, -8.83 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -79.43 | APE8-dihe-in | -132.83, 160.57 | APE8-rot-out | 180.68 | APE67-dihe-in | -62.16, -27.71 | -107.14, -6.5 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 9.74 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | E | 280.0 | 258.0 | 17 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 9o0u | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0VE | P04049 | 339 | 613 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.8024 | 13.3404 | BLAplus | -138.88, -169.03 | 61.87, 34.79 | -104.64, 32.35 | 56.09, 93.36 | -64.43, -47.67 | out-none | out | 11.5845 | Saltbr-none | 999.0 | HRD-in | -66.6, -47.0 | 72.05, -8.97 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | 56.8, 24.32 | APE9-dihe-na | -101.33, -80.31 | APE8-dihe-in | -132.61, 160.7 | APE8-rot-out | 180.75 | APE67-dihe-in | -62.26, -27.57 | -106.96, -6.66 | APE12-dist-in | 11.2624 | APE11-dist-in | 9.0411 | APE10-dist-out | 12.024 | APE9-dist-out | 9.4519 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | E | 280.0 | 261.0 | 14 | 30 | 16 | 14 | [[349, 608]] | 1.0 | 9o0v | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0UC | P04049 | 339 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.4118 | 14.92 | BLBminus | -135.2, -162.93 | 65.39, 47.79 | -89.17, 153.49 | 305.13, 119.24 | 148.83, -36.3 | in-in | in | 8.1119 | Saltbr-in | 3.1081 | HRD-in | -65.51, -42.52 | 74.23, -8.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.2736 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -140.95 | APE9-dihe-na | 87.04, -108.57 | APE8-dihe-in | -126.35, 163.82 | APE8-rot-out | 179.91 | APE67-dihe-in | -66.05, -28.24 | -108.28, -15.46 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 9.537 | APE9-dist-out | 7.8436 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | C | 280.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 9o0u | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0VC | P04049 | 339 | 614 | 648.0 | 324:701 | Type1 | Inactive | DFGin | 6.507 | 14.8484 | BLBminus | -135.62, -163.14 | 65.12, 48.02 | -88.94, 153.23 | 304.77, 118.58 | 148.73, -35.99 | in-in | in | 8.1644 | Saltbr-in | 3.3442 | HRD-in | -65.49, -42.82 | 73.84, -8.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.3433 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -150.01 | APE9-dihe-na | 93.34, -107.4 | APE8-dihe-in | -126.38, 163.35 | APE8-rot-out | 180.01 | APE67-dihe-in | -65.89, -28.16 | -108.44, -15.01 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 9.4019 | APE9-dist-out | 7.9115 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | C | 280.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 9o0v | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9AY7A | P04049 | 343 | 612 | 648.0 | ANP:701 | ATPlike | Inactive | DFGin | 5.8053 | 13.462 | BLBplus | -133.55, 174.37 | 58.47, 38.44 | -90.49, 142.18 | 44.05, 90.72 | 78.29, -134.9 | out-out | out | 14.0699 | Saltbr-out | 12.7376 | HRD-in | -73.02, -44.7 | 76.86, -25.12 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.1822 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -145.48, 130.61 | APE9-dihe-na | 129.03, -169.57 | APE8-dihe-in | -79.63, 137.79 | APE8-rot-in | 302.79 | APE67-dihe-in | -63.4, -34.24 | -69.33, -38.68 | APE12-dist-out | 15.2361 | APE11-dist-out | 15.0562 | APE10-dist-out | 10.6236 | APE9-dist-out | 6.3059 | Y340D,Y341D | None | None | XRAY | 2.41 | 0.203 | 0.236 | A | 280.0 | 260.0 | 10 | 30 | 24 | 6 | [[349, 608]] | 1.0 | 9ay7 | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9MMRA | P04049 | 343 | 625 | 648.0 | AGS:60701 | ATPlike | Inactive | DFGin | 5.4464 | 13.6261 | BLBplus | -135.09, 172.16 | 58.87, 36.16 | -92.53, 159.81 | 52.16, 102.21 | 63.65, -134.37 | out-out | out | 13.8632 | Saltbr-out | 12.3622 | HRD-out | -74.45, 80.03 | -68.85, 163.44 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.7183 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -153.07, 160.07 | APE9-dihe-na | 91.95, -174.93 | APE8-dihe-in | -63.61, 140.51 | APE8-rot-in | 299.95 | APE67-dihe-in | -59.35, -38.77 | -86.72, -25.37 | APE12-dist-out | 15.0543 | APE11-dist-out | 14.7515 | APE10-dist-out | 11.0339 | APE9-dist-out | 8.4046 | Q156R,Y340D,Y341D,D587E | SEP621 | SEP621 | EM | 3.9 | 999.0 | 999.0 | A | 681.0 | 283.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mmr | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9MMSA | P04049 | 343 | 610 | 648.0 | AGS:701 | ATPlike | Inactive | DFGin | 6.0432 | 13.4123 | BLBplus | -130.72, 176.22 | 57.09, 37.64 | -95.88, 150.42 | 38.9, 90.55 | 70.15, -138.14 | out-out | out | 13.239 | Saltbr-out | 11.9633 | HRD-out | -75.89, 77.72 | -68.75, 167.65 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.0132 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -153.3, 137.93 | APE9-dihe-na | 117.05, 178.36 | APE8-dihe-in | -66.7, 143.78 | APE8-rot-in | 289.18 | APE67-dihe-in | -66.49, -26.11 | -89.17, -21.29 | APE12-dist-out | 15.1652 | APE11-dist-out | 14.8651 | APE10-dist-out | 10.7824 | APE9-dist-out | 8.09 | Q156R,Y340D,Y341D,D587E | None | None | EM | 3.3 | 999.0 | 999.0 | A | 681.0 | 268.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mms | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9MMQA | P04049 | 341 | 612 | 648.0 | AGS:701 | ATPlike | Inactive | DFGin | 6.0418 | 13.4878 | BLBplus | -128.47, 173.58 | 60.41, 41.33 | -95.4, 154.76 | 40.5, 88.25 | 68.22, -137.22 | out-out | out | 13.7306 | Saltbr-out | 12.7147 | HRD-out | -73.84, 78.36 | -65.55, 163.21 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.1331 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -154.13, 160.3 | APE9-dihe-na | 98.38, -176.64 | APE8-dihe-in | -67.06, 138.58 | APE8-rot-in | 288.86 | APE67-dihe-in | -64.64, -31.65 | -87.38, -18.69 | APE12-dist-out | 15.1677 | APE11-dist-out | 14.4229 | APE10-dist-out | 10.8266 | APE9-dist-out | 8.1068 | Q156R,D587E | None | None | EM | 2.9 | 999.0 | 999.0 | A | 681.0 | 272.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mmq | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9MMPA | P04049 | 138 | 630 | 648.0 | AGS:60701 | ATPlike | Inactive | DFGin | 6.1073 | 13.2684 | BLBplus | -130.39, 177.17 | 56.68, 47.87 | -99.84, 149.88 | 40.92, 87.91 | 73.17, -140.77 | out-out | out | 14.3612 | Saltbr-out | 12.3822 | HRD-out | -74.8, 81.36 | -67.74, 154.91 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.1666 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -156.54, 146.13 | APE9-dihe-na | 117.78, -173.39 | APE8-dihe-in | -67.5, 146.42 | APE8-rot-in | 282.71 | APE67-dihe-in | -62.97, -41.04 | -80.62, -35.94 | APE12-dist-out | 14.2949 | APE11-dist-out | 14.3656 | APE10-dist-out | 10.6756 | APE9-dist-out | 7.9092 | Q156R,D587E | SEP259,SEP621 | SEP259,SEP621 | EM | 3.4 | 999.0 | 999.0 | A | 683.0 | 348.0 | 0 | 30 | 30 | 0 | [[349, 608]] | 1.0 | 9mmp | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2e-80 | 276.3 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0UA | P04049 | 339 | 612 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.49 | 13.4253 | BLBplus | -137.77, -168.21 | 60.54, 23.67 | -97.39, 164.85 | 62.85, 94.03 | 74.33, 173.3 | out-none | out | 11.6361 | Saltbr-none | 999.0 | HRD-in | -67.32, -47.26 | 72.53, -10.19 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 8.5215 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -79.91, 164.26 | APE9-dihe-na | 133.94, -179.25 | APE8-dihe-in | -151.13, 161.47 | APE8-rot-out | 181.14 | APE67-dihe-in | -63.28, -28.75 | -107.76, -7.41 | APE12-dist-out | 21.2876 | APE11-dist-out | 15.3594 | APE10-dist-out | 15.2178 | APE9-dist-out | 10.0158 | Y340D,Y341D | None | None | XRAY | 2.91 | 0.232 | 0.264 | A | 280.0 | 267.0 | 7 | 30 | 23 | 7 | [[349, 608]] | 1.0 | 9o0u | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 9O0VA | P04049 | 339 | 612 | 648.0 | 324:701 | Type1.5_Back | Inactive | DFGin | 5.6121 | 13.5412 | BLBplus | -137.53, -168.14 | 60.68, 23.81 | -97.37, 165.11 | 62.5, 93.91 | 74.63, 173.9 | out-none | out | 11.5178 | Saltbr-none | 999.0 | HRD-in | -67.23, -47.12 | 72.36, -10.39 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 8.5821 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oioo | APE10-dihe-na | -121.31, 23.23 | APE9-dihe-na | -94.2, -61.86 | APE8-dihe-in | -150.39, 162.26 | APE8-rot-out | 181.1 | APE67-dihe-in | -63.35, -28.52 | -106.79, -7.22 | APE12-dist-out | 14.0563 | APE11-dist-in | 11.3326 | APE10-dist-out | 13.0181 | APE9-dist-out | 9.5213 | Y340D,Y341D | None | None | XRAY | 3.5 | 0.208 | 0.254 | A | 280.0 | 266.0 | 8 | 30 | 22 | 8 | [[349, 608]] | 1.0 | 9o0v | Homo sapiens | TKL_RAF1_HUMAN | TKL | 2.6e-81 | 279.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8CPDA | P04049 | 341 | 626 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.2527 | 14.8427 | None | -88.44, -129.65 | -68.47, 153.64 | -115.46, 32.54 | 280.62, 22.29 | -59.2, -38.85 | in-in | in | 8.9962 | Saltbr-in | 3.2393 | HRD-out | -71.21, -9.87 | 61.06, -133.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.3344 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, -31.3 | APE9-dihe-na | -64.2, -40.67 | APE8-dihe-in | -125.25, 125.51 | APE8-rot-in | 293.24 | APE67-dihe-in | -70.13, -31.13 | -109.07, 11.27 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 13.0605 | APE9-dist-out | 15.3926 | Y341D | SEP621 | SEP621 | EM | 3.46 | 999.0 | 999.0 | A | 648.0 | 269.0 | 17 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 8cpd | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8CPDB | P04049 | 341 | 626 | 648.0 | No_ligand | No_ligand | Inactive | DFGin | 6.3243 | 14.7834 | None | -88.37, -130.06 | -68.25, 153.07 | -115.22, 33.93 | 283.48, 10.19 | -59.44, -38.94 | in-in | in | 8.9968 | Saltbr-in | 3.2413 | HRD-out | -70.18, -11.24 | 60.41, -132.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.2815 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, -32.01 | APE9-dihe-na | -64.34, -40.91 | APE8-dihe-in | -123.99, 124.82 | APE8-rot-in | 292.66 | APE67-dihe-in | -70.59, -30.16 | -110.37, 10.88 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 13.0602 | APE9-dist-out | 15.4329 | Y341D | SEP621 | SEP621 | EM | 3.46 | 999.0 | 999.0 | B | 648.0 | 269.0 | 17 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 8cpd | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 3OMVA | P04049 | 340 | 615 | 648.0 | SM5:1 | Type1 | Inactive | DFGin | 6.0105 | 14.0395 | None | -72.19, -157.95 | -69.65, 158.45 | -112.95, 18.14 | 298.92, 73.64 | -38.54, -34.68 | in-in | in | 8.8405 | Saltbr-in | 2.8181 | HRD-in | -81.59, -27.52 | 64.4, -79.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.128 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nioo | APE10-dihe-na | -67.59, 120.25 | APE9-dihe-na | -106.5, 137.12 | APE8-dihe-in | -106.61, 64.59 | APE8-rot-out | 44.73 | APE67-dihe-inflip | 112.91, -48.44 | -57.65, 161.85 | APE12-dist-none | 999.0 | APE11-dist-in | 13.3289 | APE10-dist-out | 12.1479 | APE9-dist-out | 10.4545 | None | None | None | XRAY | 4.0 | 0.283 | 0.364 | A | 307.0 | 264.0 | 12 | 30 | 18 | 12 | [[349, 608]] | 1.0 | 3omv | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3.7e-81 | 278.6 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8CHFA | P04049 | 341 | 626 | 648.0 | 29L:60701 | Type1 | Inactive | DFGin | 6.9193 | 13.7979 | None | -77.69, -137.87 | -62.1, 150.83 | -123.34, 43.11 | 304.09, 90.48 | -53.76, -47.63 | in-out | in | 8.5922 | Saltbr-out | 6.6899 | HRD-in | -62.51, -43.32 | 69.96, -9.45 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8262 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiio | APE10-dihe-na | 55.74, 2.9 | APE9-dihe-na | 55.92, 40.68 | APE8-dihe-in | -131.33, 94.1 | APE8-rot-out | 59.25 | APE67-dihe-inflip | 81.42, -0.92 | -97.97, 165.62 | APE12-dist-in | 7.3494 | APE11-dist-in | 11.6311 | APE10-dist-in | 6.9434 | APE9-dist-out | 10.1571 | Y341D | SEP621 | SEP621 | EM | 4.25 | 0.445 | 999.0 | A | 648.0 | 280.0 | 6 | 30 | 24 | 6 | [[349, 608]] | 1.0 | 8chf | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8CHFB | P04049 | 341 | 626 | 648.0 | 29L:60701 | Type1 | Inactive | DFGin | 6.9191 | 13.7979 | None | -77.67, -137.85 | -62.16, 150.83 | -123.29, 43.03 | 304.08, 90.5 | -53.73, -47.64 | in-out | in | 8.5922 | Saltbr-out | 6.6905 | HRD-in | -62.53, -43.31 | 69.92, -9.4 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8268 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiio | APE10-dihe-na | 55.74, 2.9 | APE9-dihe-na | 55.89, 40.65 | APE8-dihe-in | -131.28, 94.15 | APE8-rot-out | 59.25 | APE67-dihe-inflip | 81.39, -0.89 | -98.01, 165.61 | APE12-dist-in | 7.3494 | APE11-dist-in | 11.631 | APE10-dist-in | 6.9423 | APE9-dist-out | 10.1569 | Y341D | SEP621 | SEP621 | EM | 4.25 | 0.445 | 999.0 | B | 648.0 | 280.0 | 6 | 30 | 24 | 6 | [[349, 608]] | 1.0 | 8chf | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3e-80 | 275.8 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8GFTD | P04049 | 404 | 611 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -164.39, -179.79 | -89.82, 12.52 | -72.24, -18.95 | 181.77, 70.31 | -73.4, 999.0 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -68.87, -46.27 | 64.82, -56.23 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, -56.49 | APE9-dihe-na | 100.69, -17.61 | APE8-dihe-out | -72.27, -36.0 | APE8-rot-out | 67.45 | APE67-dihe-in | -49.85, -47.25 | -97.25, -47.78 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.5368 | None | None | None | EM | 3.8 | 999.0 | 999.0 | D | 304.0 | 191.0 | 72 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 8gft | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3.6e-81 | 278.6 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8U1LC | P04049 | 418 | 615 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | 87.15, 3.03 | -74.84, 77.99 | -74.97, 76.67 | 289.42, 93.79 | 116.56, -171.97 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-out | -100.67, 144.24 | -121.66, -8.0 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nooo | APE10-dihe-na | 51.33, 57.43 | APE9-dihe-na | 61.35, -123.96 | APE8-dihe-out | 55.11, 35.51 | APE8-rot-in | 302.03 | APE67-dihe-in | -59.19, -23.13 | -70.4, -10.97 | APE12-dist-none | 999.0 | APE11-dist-out | 19.2568 | APE10-dist-out | 16.2609 | APE9-dist-out | 9.904 | None | None | None | EM | 3.7 | 999.0 | 999.0 | C | 656.0 | 184.0 | 83 | 30 | 16 | 14 | [[349, 608]] | 1.0 | 8u1l | Homo sapiens | TKL_RAF1_HUMAN | TKL | 3.1e-80 | 275.7 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 7Z37CP1 | P04049 | 406 | 615 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -51.69, 113.04 | -59.31, 132.91 | -63.39, -37.52 | 182.06, 73.21 | 115.94, -41.02 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -94.28, -51.52 | 64.79, -72.58 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -172.19 | APE8-rot-out | 162.56 | APE67-dihe-inflip | 70.01, -5.7 | -83.36, 166.62 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | EM | 3.67 | 999.0 | 999.0 | CP1 | 659.0 | 193.0 | 74 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 7z37 | Homo sapiens | TKL_RAF1_HUMAN | TKL | 1e-79 | 274.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 7Z38C | P04049 | 406 | 615 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -54.5, 132.93 | -69.32, 104.66 | -85.43, 53.34 | 267.31, 92.72 | 60.74, -125.52 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -113.4, -61.21 | 60.49, -2.03 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, -92.5 | APE8-rot-out | 164.68 | APE67-dihe-inflip | 72.83, -7.22 | -110.4, 137.31 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | EM | 3.16 | 999.0 | 999.0 | C | 659.0 | 193.0 | 74 | 30 | 13 | 17 | [[349, 608]] | 1.0 | 7z38 | Homo sapiens | TKL_RAF1_HUMAN | TKL | 1e-79 | 274.0 | 3.0 | 266.0 | 264.0 | 485 | 486 | 487 | 489 | 491 | 375 | 393 | 397 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| RAF1 | RAF1_HUMAN | 8GAED | P04049 | 404 | 610 | 648.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -126.25, -170.67 | -128.75, -9.64 | -62.05, -51.04 | 170.23, 78.51 | 57.98, 999.0 | none-na | none | 999.0 | Saltbr-na | 999.0 | HRD-out | -112.46, 123.69 | -73.96, 156.28 | na-none-out | SNCano | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioo | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -175.21 | APE8-dihe-in | -78.72, 159.13 | APE8-rot-out | 52.86 | APE67-dihe-out | -91.67, 147.13 | -88.13, 88.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 16.09 | None | None | None | EM | 3.3 | 999.0 | 999.0 | D | 207.0 | 189.0 | 18 | 30 | 12 | 18 | [[349, 608]] | 1.0 | 8gae | Homo sapiens | TKL_RAF1_HUMAN | TKL | 4e-62 | 216.0 | 57.0 | 266.0 | 210.0 | 485 | 486 | 487 | 489 | 491 | 0 | 0 | 0 | 465 | 467 | 466 | 468.0 | 530 | 515 | 510 | 509 | 508 | 507 | 506 | 505 | 504 | 422 | RAF proto-oncogene serine/threonine-protein kinase |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|