AGC_PKN1 (Serine/threonine-protein kinase N1)

Total number of chains: 6
Active chains: 2
Uniprot: PKN1_HUMAN
Kinase Domain Residues: 615 - 874
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 2 33.3% 4OTDA
DFGin BLAminus 2 33.3% AF-Q16512-K1A
DFGin BLAplus 2 33.3% 4OTHA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PKN1 AF-Q16512-K1A Q16512 607 882 942.0 No_ligand No_ligand Active DFGin 6.125 12.8034 BLAminus -104.04, -164.64 32.68, 89.18 -91.79, 14.64 301.92, 91.88 -63.04, -27.24 in-in in 9.0668 Saltbr-in 2.6714 HRD-in -84.1, -49.81 66.41, 1.28 in-in-in SNCiii in-in ActLoopNT-in 2.8908 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.08, 154.4 APE9-dihe-na 137.89, 173.8 APE8-dihe-in -75.84, 131.35 APE8-rot-in 298.99 APE67-dihe-in -68.2, -19.42 -47.26, -48.97 APE12-dist-in 8.4844 APE11-dist-in 11.5084 APE10-dist-in 5.8485 APE9-dist-in 3.5612 None None None AF2 -1.0 1.0 1.0 A 276.0 276.0 0 28 28 0 [[615, 874]] 1.0 AF-Q16512-K1 AGC_PKN1_HUMAN AGC 9e-91 309.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 AF-Q16512-K3A Q16512 607 882 942.0 No_ligand No_ligand Active DFGin 5.8695 13.0226 BLAminus -110.25, -171.62 42.06, 78.21 -81.03, 13.32 306.32, 97.97 -64.16, -27.17 in-in in 8.964 Saltbr-in 2.6998 HRD-in -80.36, -49.64 68.98, 3.43 in-in-in SNCiii in-in ActLoopNT-in 2.8514 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.89, 155.38 APE9-dihe-na 131.55, -178.6 APE8-dihe-in -90.87, 131.72 APE8-rot-in 298.43 APE67-dihe-in -65.82, -21.14 -44.47, -52.21 APE12-dist-in 8.5748 APE11-dist-in 11.4832 APE10-dist-in 5.8406 APE9-dist-in 3.3687 None None None AF2 -1.0 1.0 1.0 A 276.0 276.0 0 28 28 0 [[615, 874]] 1.0 AF-Q16512-K3 AGC_PKN1_HUMAN AGC 9e-91 309.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 4OTDA Q16512 605 940 942.0 No_ligand No_ligand Inactive DFGin 7.3597 12.6959 ABAminus -114.19, -18.5 -138.56, 150.95 -133.34, 23.62 298.57, 89.18 -66.17, -19.07 in-in in 9.7616 Saltbr-in 2.5507 HRD-in -83.06, -49.66 76.99, -22.78 in-in-in SNCiii in-in ActLoopNT-in 2.9384 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.27, 161.28 APE9-dihe-na 106.58, 166.23 APE8-dihe-in -86.12, 113.11 APE8-rot-in 305.18 APE67-dihe-in -71.87, -13.23 -45.86, -32.67 APE12-dist-in 8.3456 APE11-dist-in 11.7332 APE10-dist-in 6.1085 APE9-dist-in 4.8065 None TPO774,SEP916 TPO774,SEP916 XRAY 2.0 0.177 0.221 A 341.0 336.0 0 28 28 0 [[615, 874]] 1.0 4otd AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 4OTGA Q16512 605 940 942.0 2V9:61001 Type1 Inactive DFGin 6.7387 12.4491 ABAminus -116.77, -25.12 -127.23, 113.95 -111.64, 25.58 303.73, 88.71 -62.85, -32.83 in-in in 9.3806 Saltbr-in 3.1333 HRD-in -89.2, -47.92 78.18, -34.6 in-in-in SNCiii in-in ActLoopNT-in 3.0927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.02, 157.82 APE9-dihe-na 102.38, 173.73 APE8-dihe-in -80.23, 111.75 APE8-rot-in 307.07 APE67-dihe-in -68.66, -15.76 -46.78, -35.82 APE12-dist-in 8.3339 APE11-dist-in 11.6687 APE10-dist-in 6.0556 APE9-dist-in 5.4231 None TPO774,SEP916 TPO774,SEP916 XRAY 2.6 0.212 0.268 A 341.0 324.0 0 28 28 0 [[615, 874]] 1.0 4otg AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 4OTHA Q16512 606 940 942.0 DRN:61001 Type1 Inactive DFGin 5.3268 13.288 BLAplus -95.02, 155.9 62.95, 34.93 -89.79, -14.47 67.06, 79.11 -76.51, -15.56 in-in in 9.7901 Saltbr-in 2.9971 HRD-in -77.84, -54.58 76.79, -52.02 in-out-none SNCion out-none ActLoopNT-out 6.2776 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None TPO774,SEP916 TPO774,SEP916 XRAY 1.8 0.204 0.266 A 341.0 306.0 29 28 6 22 [[615, 874]] 1.0 4oth AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 4OTIA Q16512 606 940 942.0 MI1:61001 Type1 Inactive DFGin 4.7795 13.6113 BLAplus -100.89, 152.42 49.3, 49.67 -84.2, -8.42 65.57, 87.61 -86.86, -16.27 in-in in 9.5969 Saltbr-in 2.577 HRD-in -94.1, -68.68 77.6, -28.44 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None TPO774,SEP916 TPO774,SEP916 XRAY 1.93 0.187 0.226 A 341.0 304.0 31 28 4 24 [[615, 874]] 1.0 4oti AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1

AGC_PKN1 (Serine/threonine-protein kinase N1)

Total number of chains: 6
Active chains: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 2 33.3% 4OTDA
DFGin BLAminus 2 33.3% AF-Q16512-K1A
DFGin BLAplus 2 33.3% 4OTHA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PKN1 PKN1_HUMAN AF-Q16512-K1A Q16512 607 882 942.0 No_ligand No_ligand Active DFGin 6.125 12.8034 BLAminus -104.04, -164.64 32.68, 89.18 -91.79, 14.64 301.92, 91.88 -63.04, -27.24 in-in in 9.0668 Saltbr-in 2.6714 HRD-in -84.1, -49.81 66.41, 1.28 in-in-in SNCiii in-in ActLoopNT-in 2.8908 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.08, 154.4 APE9-dihe-na 137.89, 173.8 APE8-dihe-in -75.84, 131.35 APE8-rot-in 298.99 APE67-dihe-in -68.2, -19.42 -47.26, -48.97 APE12-dist-in 8.4844 APE11-dist-in 11.5084 APE10-dist-in 5.8485 APE9-dist-in 3.5612 None None None AF2 -1.0 1.0 1.0 A 276.0 276.0 0 28 28 0 [[615, 874]] 1.0 AF-Q16512-K1 Homo sapiens AGC_PKN1_HUMAN AGC 9e-91 309.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 PKN1_HUMAN AF-Q16512-K3A Q16512 607 882 942.0 No_ligand No_ligand Active DFGin 5.8695 13.0226 BLAminus -110.25, -171.62 42.06, 78.21 -81.03, 13.32 306.32, 97.97 -64.16, -27.17 in-in in 8.964 Saltbr-in 2.6998 HRD-in -80.36, -49.64 68.98, 3.43 in-in-in SNCiii in-in ActLoopNT-in 2.8514 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.89, 155.38 APE9-dihe-na 131.55, -178.6 APE8-dihe-in -90.87, 131.72 APE8-rot-in 298.43 APE67-dihe-in -65.82, -21.14 -44.47, -52.21 APE12-dist-in 8.5748 APE11-dist-in 11.4832 APE10-dist-in 5.8406 APE9-dist-in 3.3687 None None None AF2 -1.0 1.0 1.0 A 276.0 276.0 0 28 28 0 [[615, 874]] 1.0 AF-Q16512-K3 Homo sapiens AGC_PKN1_HUMAN AGC 9e-91 309.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 PKN1_HUMAN 4OTDA Q16512 605 940 942.0 No_ligand No_ligand Inactive DFGin 7.3597 12.6959 ABAminus -114.19, -18.5 -138.56, 150.95 -133.34, 23.62 298.57, 89.18 -66.17, -19.07 in-in in 9.7616 Saltbr-in 2.5507 HRD-in -83.06, -49.66 76.99, -22.78 in-in-in SNCiii in-in ActLoopNT-in 2.9384 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.27, 161.28 APE9-dihe-na 106.58, 166.23 APE8-dihe-in -86.12, 113.11 APE8-rot-in 305.18 APE67-dihe-in -71.87, -13.23 -45.86, -32.67 APE12-dist-in 8.3456 APE11-dist-in 11.7332 APE10-dist-in 6.1085 APE9-dist-in 4.8065 None TPO774,SEP916 TPO774,SEP916 XRAY 2.0 0.177 0.221 A 341.0 336.0 0 28 28 0 [[615, 874]] 1.0 4otd Homo sapiens AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 PKN1_HUMAN 4OTGA Q16512 605 940 942.0 2V9:61001 Type1 Inactive DFGin 6.7387 12.4491 ABAminus -116.77, -25.12 -127.23, 113.95 -111.64, 25.58 303.73, 88.71 -62.85, -32.83 in-in in 9.3806 Saltbr-in 3.1333 HRD-in -89.2, -47.92 78.18, -34.6 in-in-in SNCiii in-in ActLoopNT-in 3.0927 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.02, 157.82 APE9-dihe-na 102.38, 173.73 APE8-dihe-in -80.23, 111.75 APE8-rot-in 307.07 APE67-dihe-in -68.66, -15.76 -46.78, -35.82 APE12-dist-in 8.3339 APE11-dist-in 11.6687 APE10-dist-in 6.0556 APE9-dist-in 5.4231 None TPO774,SEP916 TPO774,SEP916 XRAY 2.6 0.212 0.268 A 341.0 324.0 0 28 28 0 [[615, 874]] 1.0 4otg Homo sapiens AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 PKN1_HUMAN 4OTHA Q16512 606 940 942.0 DRN:61001 Type1 Inactive DFGin 5.3268 13.288 BLAplus -95.02, 155.9 62.95, 34.93 -89.79, -14.47 67.06, 79.11 -76.51, -15.56 in-in in 9.7901 Saltbr-in 2.9971 HRD-in -77.84, -54.58 76.79, -52.02 in-out-none SNCion out-none ActLoopNT-out 6.2776 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None TPO774,SEP916 TPO774,SEP916 XRAY 1.8 0.204 0.266 A 341.0 306.0 29 28 6 22 [[615, 874]] 1.0 4oth Homo sapiens AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1
PKN1 PKN1_HUMAN 4OTIA Q16512 606 940 942.0 MI1:61001 Type1 Inactive DFGin 4.7795 13.6113 BLAplus -100.89, 152.42 49.3, 49.67 -84.2, -8.42 65.57, 87.61 -86.86, -16.27 in-in in 9.5969 Saltbr-in 2.577 HRD-in -94.1, -68.68 77.6, -28.44 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None TPO774,SEP916 TPO774,SEP916 XRAY 1.93 0.187 0.226 A 341.0 304.0 31 28 4 24 [[615, 874]] 1.0 4oti Homo sapiens AGC_PKN1_HUMAN AGC 1.9e-90 308.4 1.0 260.0 260.0 757 758 759 761 763 644 663 667 737 739 738 740.0 797 785 780 779 778 777 776 775 774 696 Serine/threonine-protein kinase N1

AGC_PKN1 (Serine/threonine-protein kinase N1)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help.

Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name