OTHER_GAK (Cyclin-G-associated kinase)

Total number of chains: 13
Active chains: 2
Uniprot: GAK_HUMAN
Kinase Domain Residues: 40 - 315
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 9 69.2% 4C57A
DFGin BLAminus 4 30.8% AF-O14976-K1A

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PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
AF-O14976-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 32 - 323 0 None None Cyclin-G-associated kinase
AF-O14976-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 32 - 323 0 None None Cyclin-G-associated kinase
4O38A 2.097 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn No_ligand No_ligand 25 - 334 0 None None Cyclin-G-associated kinase
4O38B 2.097 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn No_ligand No_ligand 26 - 337 0 None None Cyclin-G-associated kinase
5Y7ZA 2.804 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii IRE Type1 25 - 335 0 None None Cyclin-G-associated kinase
5Y7ZB 2.804 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii IRE Type1 25 - 335 0 None None Cyclin-G-associated kinase
4C57A 2.55 Inactive DFGin‑ABAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii FEF Type1 25 - 334 0 None None Cyclin-G-associated kinase
4C57B 2.55 Inactive DFGin‑ABAminus out-out in-in nonTYR APEdihe_aaiii APEdist_iiii FEF Type1 27 - 334 0 None None Cyclin-G-associated kinase
4C59A 2.8 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn FEF Type1 27 - 333 0 None None Cyclin-G-associated kinase
5Y80A 2.5 Inactive DFGin‑ABAminus in-in in-out nonTYR APEdihe_aaiii APEdist_oioo IRE, IRE Type1, Allosteric 25 - 332 0 None None Cyclin-G-associated kinase
4C58A 2.16 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn 824 Type1.5_Back 27 - 333 0 None None Cyclin-G-associated kinase
4Y8DA 2.1 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn 49J Type1 27 - 333 0 None None Cyclin-G-associated kinase
4Y8DB 2.1 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn 49J Type1 27 - 333 0 None None Cyclin-G-associated kinase

OTHER_GAK (Cyclin-G-associated kinase)

Total number of chains: 13
Active chains: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 9 69.2% 4C57A
DFGin BLAminus 4 30.8% AF-O14976-K1A

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
GAK_HUMAN AF-O14976-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 32 - 323 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN AF-O14976-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 32 - 323 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4O38A 2.097 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn No_ligand No_ligand 25 - 334 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4O38B 2.097 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn No_ligand No_ligand 26 - 337 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 5Y7ZA 2.804 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii IRE Type1 25 - 335 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 5Y7ZB 2.804 Inactive DFGin‑ABAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii IRE Type1 25 - 335 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4C57A 2.55 Inactive DFGin‑ABAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii FEF Type1 25 - 334 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4C57B 2.55 Inactive DFGin‑ABAminus out-out in-in nonTYR APEdihe_aaiii APEdist_iiii FEF Type1 27 - 334 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4C59A 2.8 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn FEF Type1 27 - 333 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 5Y80A 2.5 Inactive DFGin‑ABAminus in-in in-out nonTYR APEdihe_aaiii APEdist_oioo IRE, IRE Type1, Allosteric 25 - 332 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4C58A 2.16 Inactive DFGin‑ABAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn 824 Type1.5_Back 27 - 333 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4Y8DA 2.1 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn 49J Type1 27 - 333 0 None None Cyclin-G-associated kinase Homo sapiens
GAK_HUMAN 4Y8DB 2.1 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aannn APEdist_nnnn 49J Type1 27 - 333 0 None None Cyclin-G-associated kinase Homo sapiens

OTHER_GAK (Cyclin-G-associated kinase)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism