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| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 4EKKA | 144 | 477 | 480.0 | ANP:60501 | ATPlike | Active | DFGin | 6.048 | 13.113 | BLAminus | -112.5, -177.27 | 66.46, 90.66 | -111.95, 23.34 | 296.26, 86.16 | -69.26, -23.9 | in-in | in | 8.651 | Saltbr-in | 2.978 | HRD-in | -63.51, -40.13 | 66.5, -18.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.05 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -155.71, 172.01 | APE9-dihe-na | 121.09, -152.4 | APE8-dihe-in | -119.32, 125.09 | APE8-rot-in | 285.38 | APE67-dihe-in | -63.61, -25.53 | -44.69, -42.52 | APE12-dist-in | 8.814 | APE11-dist-in | 11.718 | APE10-dist-in | 6.07 | APE9-dist-in | 4.069 | S473D | TPO308 | TPO308 | XRAY | 2.8 | 0.22 | 0.28 | A | 341 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekk | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 4EKKB | 144 | 477 | 480.0 | ANP:60501 | ATPlike | Active | DFGin | 6.075 | 13.046 | BLAminus | -112.98, 175.61 | 60.18, 117.01 | -127.72, 18.67 | 304.81, 92.19 | -54.85, -36.32 | in-in | in | 8.766 | Saltbr-in | 2.665 | HRD-in | -65.56, -47.0 | 73.75, -27.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.819 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -156.2, 164.76 | APE9-dihe-na | 136.6, -155.35 | APE8-dihe-in | -114.57, 129.15 | APE8-rot-in | 273.31 | APE67-dihe-in | -63.86, -22.96 | -45.74, -46.48 | APE12-dist-in | 8.77 | APE11-dist-in | 11.686 | APE10-dist-in | 6.125 | APE9-dist-in | 4.285 | S473D | TPO308 | TPO308 | XRAY | 2.8 | 0.22 | 0.28 | B | 341 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekk | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AF-P31749-K1A | 142 | 416 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.263 | 13.145 | BLAminus | -114.62, -167.38 | 40.57, 67.78 | -78.23, 20.61 | 301.26, 84.0 | -56.98, -40.88 | in-in | in | 8.68 | Saltbr-in | 2.68 | HRD-in | -78.93, -42.17 | 64.1, 0.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.868 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.25, 159.39 | APE9-dihe-na | 136.34, -176.15 | APE8-dihe-in | -90.74, 129.43 | APE8-rot-in | 299.37 | APE67-dihe-in | -70.7, -14.81 | -47.91, -45.56 | APE12-dist-in | 8.322 | APE11-dist-in | 11.748 | APE10-dist-in | 6.046 | APE9-dist-in | 3.779 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275 | 275 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | AF-P31749-K1 | AGC_AKT1_HUMAN | AGC | 1.1e-99 | 338.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AF-P31749-K3A | 142 | 416 | 480.0 | No_ligand | No_ligand | Active | DFGin | 5.861 | 13.331 | BLAminus | -119.71, -175.9 | 43.31, 87.62 | -90.32, 18.66 | 297.34, 81.96 | -61.74, -29.8 | in-in | in | 8.79 | Saltbr-in | 2.698 | HRD-in | -81.85, -49.76 | 69.24, 0.24 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.887 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.64, 153.01 | APE9-dihe-na | 135.73, 179.27 | APE8-dihe-in | -81.81, 130.02 | APE8-rot-in | 289.58 | APE67-dihe-in | -69.79, -14.8 | -47.58, -43.93 | APE12-dist-in | 8.487 | APE11-dist-in | 11.473 | APE10-dist-in | 5.866 | APE9-dist-in | 4.262 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275 | 275 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | AF-P31749-K3 | AGC_AKT1_HUMAN | AGC | 1.1e-99 | 338.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6BUUA | 144 | 478 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.46 | 13.561 | BLAminus | -129.81, 166.71 | 63.43, 103.36 | -112.37, 8.26 | 300.4, 87.1 | -62.82, -21.63 | in-in | in | 8.565 | Saltbr-in | 3.321 | HRD-in | -78.21, -43.42 | 65.34, -10.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.785 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -162.8, 159.61 | APE9-dihe-na | 139.87, -147.27 | APE8-dihe-in | -120.07, 129.86 | APE8-rot-in | 299.9 | APE67-dihe-in | -65.46, -21.29 | -53.54, -42.3 | APE12-dist-in | 8.72 | APE11-dist-in | 11.732 | APE10-dist-in | 6.238 | APE9-dist-in | 4.085 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.4 | 0.185 | 0.23 | A | 337 | 323 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6buu | AGC_AKT1_HUMAN | AGC | 2.2e-99 | 337.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6BUUB | 144 | 477 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.422 | 13.475 | BLAminus | -128.87, 158.63 | 82.78, 97.45 | -111.26, 12.46 | 302.86, 92.31 | -62.01, -29.27 | in-in | in | 8.622 | Saltbr-in | 2.612 | HRD-in | -74.01, -46.33 | 68.16, -15.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.946 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -158.84, 167.54 | APE9-dihe-na | 132.85, -158.22 | APE8-dihe-in | -118.97, 130.29 | APE8-rot-in | 299.43 | APE67-dihe-in | -70.47, -18.64 | -52.17, -43.37 | APE12-dist-in | 8.8 | APE11-dist-in | 11.759 | APE10-dist-in | 6.078 | APE9-dist-in | 3.935 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.4 | 0.185 | 0.23 | B | 337 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6buu | AGC_AKT1_HUMAN | AGC | 2.2e-99 | 337.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6NPZA | 142 | 478 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.243 | 13.517 | BLAminus | -119.48, 178.99 | 63.44, 89.04 | -107.85, 9.08 | 296.64, 94.01 | -63.0, -21.88 | in-in | in | 8.904 | Saltbr-in | 3.005 | HRD-in | -76.14, -48.91 | 69.19, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.995 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -163.99, 160.01 | APE9-dihe-na | 134.89, -153.13 | APE8-dihe-in | -119.22, 128.69 | APE8-rot-in | 299.44 | APE67-dihe-in | -61.81, -21.05 | -49.68, -44.36 | APE12-dist-in | 8.283 | APE11-dist-in | 11.557 | APE10-dist-in | 5.957 | APE9-dist-in | 3.903 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.12 | 0.188 | 0.241 | A | 358 | 322 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6npz | AGC_AKT1_HUMAN | AGC | 2.7e-99 | 337.5 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6NPZB | 141 | 477 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.492 | 13.71 | BLAminus | -117.03, 171.77 | 71.96, 91.9 | -107.91, 11.41 | 295.22, 94.23 | -65.12, -23.31 | in-in | in | 8.806 | Saltbr-in | 3.089 | HRD-in | -77.35, -47.58 | 69.03, -7.27 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.868 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.06, 158.85 | APE9-dihe-na | 134.94, -150.01 | APE8-dihe-in | -122.61, 125.21 | APE8-rot-in | 296.0 | APE67-dihe-in | -68.07, -17.45 | -48.75, -43.62 | APE12-dist-in | 8.484 | APE11-dist-in | 11.691 | APE10-dist-in | 6.044 | APE9-dist-in | 3.856 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.12 | 0.188 | 0.241 | B | 358 | 323 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6npz | AGC_AKT1_HUMAN | AGC | 2.7e-99 | 337.5 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 4GV1A | 144 | 477 | 480.0 | 0XZ:60501 | Type1 | Active | DFGin | 6.488 | 13.562 | BLAminus | -122.36, 161.99 | 68.48, 91.61 | -104.89, 11.22 | 297.02, 96.69 | -63.45, -24.57 | in-in | in | 8.817 | Saltbr-in | 2.472 | HRD-in | -73.6, -46.3 | 69.86, -10.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -158.52, 165.79 | APE9-dihe-na | 129.18, -173.05 | APE8-dihe-in | -103.26, 131.39 | APE8-rot-in | 301.03 | APE67-dihe-in | -66.34, -18.55 | -46.14, -49.45 | APE12-dist-in | 8.481 | APE11-dist-in | 11.553 | APE10-dist-in | 5.998 | APE9-dist-in | 4.098 | None | TPO308 | TPO308 | XRAY | 1.49 | 0.182 | 0.21 | A | 340 | 329 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4gv1 | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3OCBA | 144 | 478 | 480.0 | XM1:1 | Type1 | Active | DFGin | 6.638 | 13.803 | BLAminus | -116.95, 176.33 | 66.85, 80.21 | -101.71, 15.06 | 291.18, 80.12 | -62.95, -27.15 | in-in | in | 8.771 | Saltbr-in | 2.77 | HRD-in | -68.69, -47.69 | 74.78, -17.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.986 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -155.18, 163.1 | APE9-dihe-na | 135.15, -135.96 | APE8-dihe-in | -136.2, 122.51 | APE8-rot-in | 298.45 | APE67-dihe-in | -66.42, -19.48 | -44.24, -42.98 | APE12-dist-in | 8.435 | APE11-dist-in | 11.489 | APE10-dist-in | 5.888 | APE9-dist-in | 4.058 | S473D | TPO308 | TPO308 | XRAY | 2.7 | 0.217 | 0.282 | A | 341 | 316 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ocb | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3OCBB | 144 | 478 | 480.0 | XM1:2 | Type1 | Active | DFGin | 6.332 | 13.399 | BLAminus | -134.12, 162.45 | 65.57, 102.27 | -117.67, 11.66 | 296.51, 86.34 | -58.99, -28.22 | in-in | in | 8.815 | Saltbr-in | 2.871 | HRD-in | -68.9, -44.89 | 75.11, -22.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.078 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.43, 165.77 | APE9-dihe-na | 133.07, -137.47 | APE8-dihe-in | -130.52, 128.21 | APE8-rot-in | 301.82 | APE67-dihe-in | -61.46, -22.02 | -42.63, -52.7 | APE12-dist-in | 8.732 | APE11-dist-in | 11.603 | APE10-dist-in | 6.079 | APE9-dist-in | 4.134 | S473D | TPO308 | TPO308 | XRAY | 2.7 | 0.217 | 0.282 | B | 341 | 320 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ocb | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3OW4A | 144 | 478 | 480.0 | SMY:60001 | Type1 | Active | DFGin | 6.386 | 13.523 | BLAminus | -119.32, 159.71 | 79.63, 82.83 | -104.78, 4.01 | 298.86, 82.1 | -54.94, -24.29 | in-in | in | 8.955 | Saltbr-in | 2.902 | HRD-in | -70.99, -49.36 | 69.67, -8.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.936 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -157.63, 156.89 | APE9-dihe-na | 142.86, -142.49 | APE8-dihe-in | -124.25, 130.13 | APE8-rot-in | 298.03 | APE67-dihe-in | -63.26, -12.53 | -44.97, -47.55 | APE12-dist-in | 8.407 | APE11-dist-in | 11.499 | APE10-dist-in | 5.943 | APE9-dist-in | 4.122 | S473D | TPO308 | TPO308 | XRAY | 2.6 | 0.197 | 0.268 | A | 341 | 318 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ow4 | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3OW4B | 144 | 478 | 480.0 | SMY:60002 | Type1 | Active | DFGin | 6.468 | 13.471 | BLAminus | -110.6, 166.76 | 74.64, 94.72 | -107.78, 10.54 | 297.92, 88.21 | -53.21, -30.59 | in-in | in | 9.014 | Saltbr-in | 2.873 | HRD-in | -68.95, -46.49 | 77.32, -19.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.905 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.84, 158.48 | APE9-dihe-na | 136.94, -160.6 | APE8-dihe-in | -112.04, 132.88 | APE8-rot-in | 279.55 | APE67-dihe-in | -64.15, -17.53 | -43.71, -49.28 | APE12-dist-in | 8.567 | APE11-dist-in | 11.482 | APE10-dist-in | 6.0 | APE9-dist-in | 4.209 | S473D | TPO308 | TPO308 | XRAY | 2.6 | 0.197 | 0.268 | B | 341 | 318 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ow4 | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3QKLA | 144 | 478 | 480.0 | SMR:60001 | Type1 | Active | DFGin | 6.338 | 13.63 | BLAminus | -120.73, 173.12 | 65.05, 75.71 | -95.61, 13.62 | 302.87, 90.58 | -65.29, -24.68 | in-in | in | 9.025 | Saltbr-in | 2.669 | HRD-in | -79.32, -50.18 | 77.61, -12.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.808 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.72, 167.27 | APE9-dihe-na | 129.72, -141.45 | APE8-dihe-in | -129.9, 128.86 | APE8-rot-in | 291.61 | APE67-dihe-in | -64.11, -23.78 | -46.08, -46.14 | APE12-dist-in | 8.149 | APE11-dist-in | 11.608 | APE10-dist-in | 5.994 | APE9-dist-in | 3.707 | S473D | TPO308 | TPO308 | XRAY | 1.9 | 0.196 | 0.243 | A | 341 | 318 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3qkl | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3QKMA | 144 | 478 | 480.0 | SM9:1 | Type1 | Active | DFGin | 6.551 | 13.483 | BLAminus | -120.8, 163.74 | 70.66, 92.07 | -106.66, 15.27 | 300.92, 94.29 | -62.34, -28.26 | in-in | in | 9.201 | Saltbr-in | 2.666 | HRD-in | -70.68, -45.98 | 71.02, -16.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.824 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -153.62, 157.36 | APE9-dihe-na | 116.69, 169.89 | APE8-dihe-in | -83.27, 128.83 | APE8-rot-in | 296.3 | APE67-dihe-in | -66.75, -19.54 | -36.8, -50.73 | APE12-dist-in | 8.46 | APE11-dist-in | 11.525 | APE10-dist-in | 5.915 | APE9-dist-in | 4.629 | S473D | TPO308 | TPO308 | XRAY | 2.2 | 0.191 | 0.252 | A | 341 | 330 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3qkm | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 4EKLA | 144 | 478 | 480.0 | 0RF:501 | Type1 | Active | DFGin | 6.496 | 13.423 | BLAminus | -130.08, 156.46 | 77.16, 99.77 | -112.66, 14.16 | 298.65, 90.33 | -61.32, -30.96 | in-in | in | 8.958 | Saltbr-in | 2.452 | HRD-in | -78.38, -44.96 | 68.93, -13.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.757 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.83, 160.76 | APE9-dihe-na | 116.71, 166.32 | APE8-dihe-in | -83.66, 133.51 | APE8-rot-in | 293.53 | APE67-dihe-in | -68.09, -18.95 | -43.13, -46.31 | APE12-dist-in | 8.36 | APE11-dist-in | 11.512 | APE10-dist-in | 6.011 | APE9-dist-in | 4.443 | S473D | TPO308 | TPO308 | XRAY | 2.0 | 0.175 | 0.235 | A | 341 | 330 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekl | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3CQWA | 144 | 478 | 480.0 | CQW:60999 | Type1 | Active | DFGin | 6.338 | 13.09 | BLAminus | -122.41, 167.11 | 74.19, 82.7 | -100.79, 9.25 | 295.72, 101.99 | -67.19, -25.09 | in-in | in | 8.608 | Saltbr-in | 3.437 | HRD-in | -79.68, -40.11 | 70.25, -18.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -154.61, 166.29 | APE9-dihe-na | 132.98, -141.71 | APE8-dihe-in | -134.77, 132.14 | APE8-rot-in | 286.58 | APE67-dihe-in | -67.95, -20.8 | -49.28, -45.72 | APE12-dist-in | 8.374 | APE11-dist-in | 11.536 | APE10-dist-in | 5.934 | APE9-dist-in | 3.951 | S473D | TPO308 | TPO308 | XRAY | 2.0 | 0.203 | 0.257 | A | 342 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3cqw | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3MV5A | 144 | 477 | 480.0 | XFE:60999 | Type1 | Active | DFGin | 6.512 | 13.107 | BLAminus | -110.68, 173.87 | 55.61, 106.15 | -116.13, 8.16 | 292.02, 88.05 | -68.88, -21.78 | in-in | in | 8.573 | Saltbr-in | 2.645 | HRD-in | -81.07, -37.62 | 75.3, -21.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -163.23, 167.83 | APE9-dihe-na | 126.38, -137.1 | APE8-dihe-in | -133.69, 127.23 | APE8-rot-in | 287.39 | APE67-dihe-in | -69.19, -14.76 | -48.38, -39.25 | APE12-dist-in | 8.467 | APE11-dist-in | 11.692 | APE10-dist-in | 6.145 | APE9-dist-in | 4.185 | S473D | TPO308 | TPO308 | XRAY | 2.47 | 0.205 | 0.282 | A | 342 | 316 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3mv5 | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3MVHA | 145 | 476 | 480.0 | WFE:999 | Type1 | Active | DFGin | 6.609 | 13.205 | BLAminus | -120.33, 157.64 | 77.18, 89.81 | -109.14, 14.39 | 295.05, 87.49 | -62.89, -24.97 | in-in | in | 8.782 | Saltbr-in | 2.62 | HRD-in | -82.77, -44.94 | 75.58, -15.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.836 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.65, 167.39 | APE9-dihe-na | 135.14, -139.29 | APE8-dihe-in | -137.11, 131.02 | APE8-rot-in | 291.39 | APE67-dihe-in | -63.24, -17.86 | -53.88, -42.66 | APE12-dist-in | 8.149 | APE11-dist-in | 11.591 | APE10-dist-in | 5.855 | APE9-dist-in | 3.756 | S473D | TPO308 | TPO308 | XRAY | 2.01 | 0.181 | 0.23 | A | 342 | 312 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3mvh | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6CCYA | 144 | 983 | 480.0 | EX4:60501 | Type1 | Active | DFGin | 6.833 | 14.216 | BLAminus | -118.22, 172.28 | 65.22, 87.23 | -99.08, 6.12 | 296.87, 97.72 | -61.52, -36.28 | in-in | in | 9.387 | Saltbr-in | 2.725 | HRD-in | -70.12, -46.7 | 65.1, -15.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.814 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.15, 164.77 | APE9-dihe-na | 117.98, 177.81 | APE8-dihe-in | -89.16, 122.56 | APE8-rot-in | 287.17 | APE67-dihe-in | -60.32, -21.6 | -32.19, -51.09 | APE12-dist-in | 8.32 | APE11-dist-in | 11.49 | APE10-dist-in | 5.811 | APE9-dist-in | 4.408 | N199S,S396P,E397S,T433V | TPO308 | TPO308 | XRAY | 2.18 | 0.237 | 0.276 | A | 343 | 307 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6ccy | AGC_AKT1_HUMAN | AGC | 4.1e-99 | 336.9 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3QKKA | 144 | 478 | 480.0 | SMH:60001 | Type1.5_Front | Active | DFGin | 6.383 | 13.598 | BLAminus | -116.54, -179.44 | 52.7, 85.0 | -102.02, 14.36 | 303.33, 93.01 | -66.45, -23.02 | in-in | in | 8.916 | Saltbr-in | 2.342 | HRD-in | -78.65, -51.68 | 79.72, -12.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.763 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.57, 164.52 | APE9-dihe-na | 135.56, -139.12 | APE8-dihe-in | -127.86, 127.7 | APE8-rot-in | 299.02 | APE67-dihe-in | -62.38, -25.83 | -44.42, -46.66 | APE12-dist-in | 8.22 | APE11-dist-in | 11.566 | APE10-dist-in | 6.028 | APE9-dist-in | 3.779 | S473D | TPO308 | TPO308 | XRAY | 2.3 | 0.202 | 0.25 | A | 341 | 327 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3qkk | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3CQUA | 144 | 478 | 480.0 | CQU:60999 | Type1 | Inactive | DFGin | 6.162 | 12.752 | BLAminus | -125.29, 173.04 | 74.77, 101.51 | -111.55, 14.45 | 309.48, 77.95 | -55.91, -32.71 | in-out | in | 9.246 | Saltbr-out | 4.113 | HRD-in | -63.98, -47.97 | 77.74, -15.86 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.003 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.44, 176.23 | APE9-dihe-na | 125.93, -142.07 | APE8-dihe-in | -126.34, 131.3 | APE8-rot-in | 289.37 | APE67-dihe-in | -62.32, -24.17 | -48.41, -45.96 | APE12-dist-in | 8.309 | APE11-dist-in | 11.455 | APE10-dist-in | 6.059 | APE9-dist-in | 3.993 | S473D | TPO308 | TPO308 | XRAY | 2.2 | 0.207 | 0.283 | A | 342 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3cqu | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 8UVYA | 3 | 439 | 480.0 | XOO:60502 | Allosteric | Inactive | DFGout | 19.147 | 9.117 | BBAminus | -87.71, 159.46 | -125.79, 51.81 | -104.71, 8.89 | 306.76, 157.9 | -76.01, 144.81 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -80.44, -49.7 | 65.22, 18.47 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.329 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -75.27, -63.55 | APE9-dihe-na | -84.1, -150.14 | APE8-dihe-in | -112.51, 118.73 | APE8-rot-in | 303.11 | APE67-dihe-in | -70.02, -8.73 | -61.09, -34.89 | APE12-dist-in | 11.509 | APE11-dist-in | 11.913 | APE10-dist-in | 7.703 | APE9-dist-out | 6.561 | E17K | None | None | XRAY | 2.11 | 0.209 | 0.255 | A | 438 | 396 | 21 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 8uvy | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 8UW2A | 4 | 437 | 480.0 | XOO:60502 | Allosteric | Inactive | DFGout | 19.594 | 9.174 | BBAminus | -85.5, 157.67 | -121.72, 55.74 | -105.08, 2.24 | 304.7, 161.96 | -67.3, 146.74 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -75.89, -48.3 | 59.85, 6.57 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 13.673 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -78.7, 9.37 | APE9-dihe-na | -151.7, -145.87 | APE8-dihe-in | -109.15, 106.27 | APE8-rot-out | 18.96 | APE67-dihe-in | -70.15, -8.9 | -92.15, -6.4 | APE12-dist-out | 18.057 | APE11-dist-out | 14.765 | APE10-dist-out | 10.604 | APE9-dist-out | 11.153 | None | None | None | XRAY | 2.2 | 0.223 | 0.279 | A | 438 | 392 | 19 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 8uw2 | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 8UW9A | 3 | 428 | 480.0 | XQ2:60501 | Allosteric | Inactive | DFGout | 18.976 | 9.3 | BBAminus | -90.79, 158.27 | -126.08, 50.43 | -104.96, 7.49 | 302.98, 161.85 | -82.17, 151.97 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -80.58, -46.97 | 73.31, -13.02 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.346 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -78.06, -70.69 | APE9-dihe-na | -63.13, 144.96 | APE8-dihe-in | -69.73, 119.44 | APE8-rot-in | 308.33 | APE67-dihe-in | -66.64, -12.63 | -58.13, -37.16 | APE12-dist-in | 12.561 | APE11-dist-in | 12.026 | APE10-dist-in | 7.549 | APE9-dist-out | 6.208 | None | None | None | XRAY | 1.9 | 0.207 | 0.245 | A | 438 | 388 | 19 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 8uw9 | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 8UW7A | 3 | 439 | 480.0 | XOO:60502 | Allosteric | Inactive | DFGout | 19.268 | 9.131 | BBAminus | -88.27, 162.56 | -129.0, 47.08 | -101.62, 6.17 | 304.62, 157.46 | -65.02, 141.6 | out-out | out | 14.185 | Saltbr-out | 16.163 | HRD-in | -77.74, -48.14 | 69.36, -7.13 | out-out-out | SNCooo | out-out | ActLoopNT-out | 15.133 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 168.57 | APE8-dihe-in | -110.93, 76.79 | APE8-rot-out | 38.95 | APE67-dihe-in | -76.05, -14.39 | -64.32, -17.63 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.831 | None | None | YCM77,YCM296 | XRAY | 1.972 | 0.22 | 0.265 | A | 438 | 399 | 17 | 0 | 0 | 12 | [[150, 408]] | 1.0 | 8uw7 | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 3O96A | 2 | 429 | 480.0 | IQO:444 | Allosteric | Inactive | DFGout | 16.13 | 7.768 | BBAminus | -84.04, 164.11 | -138.96, 67.69 | -114.58, 18.46 | 294.17, 141.85 | -57.09, 121.09 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -85.54, -46.27 | 73.79, -8.96 | none-out-none | SNCnon | out-none | ActLoopNT-out | 14.705 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -63.73, -20.88 | 999.0, -53.98 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.249 | 0.308 | A | 446 | 367 | 24 | 0 | 0 | 14 | [[150, 408]] | 1.0 | 3o96 | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6HHHA | 2 | 439 | 480.0 | G4Q:501 | Allosteric | Inactive | DFGout | 19.432 | 8.904 | BBAminus | -82.84, 168.78 | -138.99, 51.81 | -104.05, 22.45 | 309.63, 151.96 | -74.89, 142.62 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -70.92, -45.22 | 71.01, -6.93 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.659 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -141.4 | APE8-dihe-out | -68.07, -39.94 | APE8-rot-out | 43.05 | APE67-dihe-in | -61.63, -40.25 | -82.49, 7.03 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 14.39 | E114A,E115A,E116A | None | None | XRAY | 2.7 | 0.217 | 0.266 | A | 446 | 379 | 25 | 0 | 0 | 11 | [[150, 408]] | 1.0 | 6hhh | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6HHJA | 3 | 444 | 480.0 | G4H:501 | Allosteric | Inactive | DFGout | 18.637 | 9.927 | BBAminus | -85.85, 154.25 | -131.76, 65.33 | -114.43, 2.7 | 306.85, 152.03 | -81.33, 157.37 | out-out | out | 16.597 | Saltbr-out | 20.784 | HRD-in | -70.38, -43.13 | 62.3, -0.73 | out-out-out | SNCooo | out-out | ActLoopNT-out | 15.398 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -96.59, 105.04 | APE9-dihe-na | 69.68, -150.96 | APE8-dihe-in | -112.16, 140.11 | APE8-rot-out | 58.43 | APE67-dihe-in | -58.84, -27.51 | -94.58, 2.39 | APE12-dist-out | 16.493 | APE11-dist-out | 16.034 | APE10-dist-out | 10.684 | APE9-dist-out | 11.298 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.223 | 0.243 | A | 446 | 410 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6hhj | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6S9WA | 3 | 444 | 480.0 | L1Z:501 | Allosteric | Inactive | DFGout | 18.014 | 9.778 | BBAminus | -88.23, 159.68 | -135.32, 63.28 | -108.07, 5.2 | 307.51, 150.05 | -79.62, 159.51 | out-out | out | 16.719 | Saltbr-out | 21.04 | HRD-in | -77.04, -47.59 | 74.55, -19.15 | out-out-out | SNCooo | out-out | ActLoopNT-out | 15.677 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -115.76, 103.74 | APE9-dihe-na | 82.07, -166.58 | APE8-dihe-in | -98.52, 141.96 | APE8-rot-out | 173.15 | APE67-dihe-in | -62.82, -22.8 | -94.37, -0.32 | APE12-dist-out | 16.616 | APE11-dist-out | 16.139 | APE10-dist-out | 10.913 | APE9-dist-out | 11.124 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.21 | 0.263 | A | 446 | 411 | 2 | 0 | 0 | 2 | [[150, 408]] | 1.0 | 6s9w | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 4EJNA | 4 | 438 | 480.0 | 0R4:501 | Type1 | Inactive | DFGout | 18.374 | 8.329 | BBAminus | -86.73, 154.01 | -129.51, 54.97 | -106.79, 23.78 | 305.4, 154.78 | -69.14, 128.42 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -74.68, -58.46 | 77.98, 6.43 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 16.065 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioo | APE10-dihe-na | -97.72, 139.0 | APE9-dihe-na | 109.04, 163.38 | APE8-dihe-in | -97.01, 108.52 | APE8-rot-in | 315.65 | APE67-dihe-in | -57.15, -23.24 | -58.45, -30.75 | APE12-dist-out | 14.955 | APE11-dist-in | 13.395 | APE10-dist-out | 8.158 | APE9-dist-out | 6.501 | E114A,E115A,E116A | None | None | XRAY | 2.19 | 0.239 | 0.276 | A | 446 | 376 | 18 | 0 | 0 | 5 | [[150, 408]] | 1.0 | 4ejn | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 5KCVA | 6 | 438 | 480.0 | 6S1:501 | Allosteric | Inactive | DFGout | 18.399 | 8.593 | None | -66.09, 150.37 | -131.74, 48.39 | -109.26, 34.53 | 301.12, 163.72 | -73.63, 124.84 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -80.28, -36.69 | 71.61, -16.44 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.9, -11.63 | 999.0, -43.42 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | E114A,E115A,E116A | None | None | XRAY | 2.7 | 0.213 | 0.269 | A | 460 | 353 | 33 | 0 | 0 | 16 | [[150, 408]] | 1.0 | 5kcv | AGC_AKT1_HUMAN | AGC | 5.6e-99 | 336.5 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 7APJA | 3 | 439 | 480.0 | No_ligand | No_ligand | Inactive | DFGout | 15.36 | 7.847 | None | -119.51, 172.58 | -151.35, 78.25 | -78.82, 999.0 | 276.7, 1.08 | 999.0, 999.0 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -72.58, -35.61 | 73.77, -41.9 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 73.92 | APE8-rot-out | 58.45 | APE67-dihe-in | -70.85, -7.62 | -68.6, -17.11 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | S2N | None | None | XRAY | 2.05 | 0.213 | 0.252 | A | 440 | 376 | 39 | 0 | 0 | 18 | [[150, 408]] | 1.0 | 7apj | AGC_AKT1_HUMAN | AGC | 5e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6HHFA | 3 | 439 | 480.0 | G4K:501 | Allosteric | Inactive | None | 999.0 | 8.943 | None | -81.4, 157.14 | -136.1, 63.0 | -116.97, 21.98 | 304.54, 147.84 | -76.24, 135.42 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -67.92, -42.11 | 68.98, -10.23 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 16.026 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 110.64 | APE8-rot-out | 65.96 | APE67-dihe-in | -73.6, -35.94 | -67.69, -4.64 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | E114A,E115A,E116A | None | None | XRAY | 2.9 | 0.233 | 0.274 | A | 446 | 366 | 32 | 0 | 0 | 14 | [[150, 408]] | 1.0 | 6hhf | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6HHGA | 3 | 444 | 480.0 | G4T:501 | Allosteric | Inactive | None | 999.0 | 9.861 | None | -89.51, 153.73 | -128.41, 67.53 | -114.64, 10.8 | 307.59, 150.55 | -85.41, 154.74 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -68.28, -46.2 | 67.11, -14.18 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.289 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -107.85, 97.08 | APE9-dihe-na | 87.64, -165.9 | APE8-dihe-in | -105.98, 137.43 | APE8-rot-out | 58.9 | APE67-dihe-in | -57.38, -21.16 | -89.5, -4.41 | APE12-dist-out | 17.366 | APE11-dist-out | 16.179 | APE10-dist-out | 10.888 | APE9-dist-out | 11.447 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.212 | 0.246 | A | 446 | 386 | 21 | 0 | 0 | 3 | [[150, 408]] | 1.0 | 6hhg | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6HHIA | 3 | 444 | 480.0 | G4N:501 | Allosteric | Inactive | None | 999.0 | 9.394 | None | -89.1, 165.97 | -135.32, 55.99 | -110.01, 13.3 | 309.82, 146.72 | -70.54, 150.25 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -69.6, -44.24 | 72.4, -22.65 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.413 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -105.21, 101.21 | APE9-dihe-na | 81.98, -162.79 | APE8-dihe-in | -113.39, 139.7 | APE8-rot-out | 66.27 | APE67-dihe-in | -49.46, -24.76 | -86.47, -13.4 | APE12-dist-out | 17.097 | APE11-dist-out | 15.773 | APE10-dist-out | 10.853 | APE9-dist-out | 11.014 | E114A,E115A,E116A | None | None | XRAY | 2.7 | 0.229 | 0.258 | A | 446 | 389 | 19 | 0 | 0 | 3 | [[150, 408]] | 1.0 | 6hhi | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 6S9XA | 3 | 443 | 480.0 | L1W:501 | Allosteric | Inactive | None | 999.0 | 9.471 | None | -83.65, 171.5 | -148.58, 59.04 | -110.35, 19.84 | 309.98, 147.1 | -81.71, 151.08 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -70.64, -44.34 | 67.14, 2.45 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.655 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nooo | APE10-dihe-na | -128.24, 142.43 | APE9-dihe-na | 73.42, -170.52 | APE8-dihe-in | -106.82, 110.63 | APE8-rot-out | 60.31 | APE67-dihe-in | -66.32, -9.87 | -76.1, -5.54 | APE12-dist-none | 999.0 | APE11-dist-out | 16.242 | APE10-dist-out | 10.715 | APE9-dist-out | 10.287 | E114A,E115A,E116A | None | None | XRAY | 2.6 | 0.214 | 0.234 | A | 446 | 382 | 23 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 6s9x | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 7NH4A | 4 | 444 | 480.0 | UCE:501 | Allosteric | Inactive | None | 999.0 | 9.714 | None | -89.66, 161.99 | -134.99, 53.83 | -102.41, 15.77 | 307.61, 150.23 | -85.21, 156.95 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -71.71, -43.96 | 65.0, -1.87 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.71 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -91.29, 122.41 | APE9-dihe-na | 62.81, -158.06 | APE8-dihe-in | -116.84, 141.55 | APE8-rot-out | 65.03 | APE67-dihe-in | -52.37, -30.57 | -89.05, -2.1 | APE12-dist-out | 16.82 | APE11-dist-out | 16.123 | APE10-dist-out | 10.705 | APE9-dist-out | 11.149 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.224 | 0.246 | A | 446 | 383 | 24 | 0 | 0 | 6 | [[150, 408]] | 1.0 | 7nh4 | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| 7NH5A | 3 | 444 | 480.0 | UC8:502 | Allosteric | Inactive | None | 999.0 | 9.683 | None | -94.24, 161.49 | -131.31, 59.8 | -111.8, 8.17 | 304.51, 156.46 | -83.9, 163.26 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -72.19, -47.43 | 76.17, -13.35 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.616 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nooo | APE10-dihe-na | -89.96, 112.26 | APE9-dihe-na | 68.59, -149.12 | APE8-dihe-in | -121.33, 137.31 | APE8-rot-in | 284.5 | APE67-dihe-in | -57.38, -14.67 | -81.19, -19.07 | APE12-dist-none | 999.0 | APE11-dist-out | 15.973 | APE10-dist-out | 10.445 | APE9-dist-out | 11.434 | E114A,E115A,E116A | None | None | XRAY | 1.9 | 0.201 | 0.228 | A | 446 | 383 | 24 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 7nh5 | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AKT1_HUMAN | 4EKKA | P31749 | 144 | 477 | 480.0 | ANP:60501 | ATPlike | Active | DFGin | 6.048 | 13.113 | BLAminus | -112.5, -177.27 | 66.46, 90.66 | -111.95, 23.34 | 296.26, 86.16 | -69.26, -23.9 | in-in | in | 8.651 | Saltbr-in | 2.978 | HRD-in | -63.51, -40.13 | 66.5, -18.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.05 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -155.71, 172.01 | APE9-dihe-na | 121.09, -152.4 | APE8-dihe-in | -119.32, 125.09 | APE8-rot-in | 285.38 | APE67-dihe-in | -63.61, -25.53 | -44.69, -42.52 | APE12-dist-in | 8.814 | APE11-dist-in | 11.718 | APE10-dist-in | 6.07 | APE9-dist-in | 4.069 | S473D | TPO308 | TPO308 | XRAY | 2.8 | 0.22 | 0.28 | A | 341 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekk | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 4EKKB | P31749 | 144 | 477 | 480.0 | ANP:60501 | ATPlike | Active | DFGin | 6.075 | 13.046 | BLAminus | -112.98, 175.61 | 60.18, 117.01 | -127.72, 18.67 | 304.81, 92.19 | -54.85, -36.32 | in-in | in | 8.766 | Saltbr-in | 2.665 | HRD-in | -65.56, -47.0 | 73.75, -27.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.819 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -156.2, 164.76 | APE9-dihe-na | 136.6, -155.35 | APE8-dihe-in | -114.57, 129.15 | APE8-rot-in | 273.31 | APE67-dihe-in | -63.86, -22.96 | -45.74, -46.48 | APE12-dist-in | 8.77 | APE11-dist-in | 11.686 | APE10-dist-in | 6.125 | APE9-dist-in | 4.285 | S473D | TPO308 | TPO308 | XRAY | 2.8 | 0.22 | 0.28 | B | 341 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekk | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | AF-P31749-K1A | P31749 | 142 | 416 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.263 | 13.145 | BLAminus | -114.62, -167.38 | 40.57, 67.78 | -78.23, 20.61 | 301.26, 84.0 | -56.98, -40.88 | in-in | in | 8.68 | Saltbr-in | 2.68 | HRD-in | -78.93, -42.17 | 64.1, 0.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.868 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.25, 159.39 | APE9-dihe-na | 136.34, -176.15 | APE8-dihe-in | -90.74, 129.43 | APE8-rot-in | 299.37 | APE67-dihe-in | -70.7, -14.81 | -47.91, -45.56 | APE12-dist-in | 8.322 | APE11-dist-in | 11.748 | APE10-dist-in | 6.046 | APE9-dist-in | 3.779 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275 | 275 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | AF-P31749-K1 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 1.1e-99 | 338.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | AF-P31749-K3A | P31749 | 142 | 416 | 480.0 | No_ligand | No_ligand | Active | DFGin | 5.861 | 13.331 | BLAminus | -119.71, -175.9 | 43.31, 87.62 | -90.32, 18.66 | 297.34, 81.96 | -61.74, -29.8 | in-in | in | 8.79 | Saltbr-in | 2.698 | HRD-in | -81.85, -49.76 | 69.24, 0.24 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.887 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.64, 153.01 | APE9-dihe-na | 135.73, 179.27 | APE8-dihe-in | -81.81, 130.02 | APE8-rot-in | 289.58 | APE67-dihe-in | -69.79, -14.8 | -47.58, -43.93 | APE12-dist-in | 8.487 | APE11-dist-in | 11.473 | APE10-dist-in | 5.866 | APE9-dist-in | 4.262 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275 | 275 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | AF-P31749-K3 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 1.1e-99 | 338.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6BUUA | P31749 | 144 | 478 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.46 | 13.561 | BLAminus | -129.81, 166.71 | 63.43, 103.36 | -112.37, 8.26 | 300.4, 87.1 | -62.82, -21.63 | in-in | in | 8.565 | Saltbr-in | 3.321 | HRD-in | -78.21, -43.42 | 65.34, -10.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.785 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -162.8, 159.61 | APE9-dihe-na | 139.87, -147.27 | APE8-dihe-in | -120.07, 129.86 | APE8-rot-in | 299.9 | APE67-dihe-in | -65.46, -21.29 | -53.54, -42.3 | APE12-dist-in | 8.72 | APE11-dist-in | 11.732 | APE10-dist-in | 6.238 | APE9-dist-in | 4.085 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.4 | 0.185 | 0.23 | A | 337 | 323 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6buu | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.2e-99 | 337.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6BUUB | P31749 | 144 | 477 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.422 | 13.475 | BLAminus | -128.87, 158.63 | 82.78, 97.45 | -111.26, 12.46 | 302.86, 92.31 | -62.01, -29.27 | in-in | in | 8.622 | Saltbr-in | 2.612 | HRD-in | -74.01, -46.33 | 68.16, -15.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.946 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -158.84, 167.54 | APE9-dihe-na | 132.85, -158.22 | APE8-dihe-in | -118.97, 130.29 | APE8-rot-in | 299.43 | APE67-dihe-in | -70.47, -18.64 | -52.17, -43.37 | APE12-dist-in | 8.8 | APE11-dist-in | 11.759 | APE10-dist-in | 6.078 | APE9-dist-in | 3.935 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.4 | 0.185 | 0.23 | B | 337 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6buu | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.2e-99 | 337.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6NPZA | P31749 | 142 | 478 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.243 | 13.517 | BLAminus | -119.48, 178.99 | 63.44, 89.04 | -107.85, 9.08 | 296.64, 94.01 | -63.0, -21.88 | in-in | in | 8.904 | Saltbr-in | 3.005 | HRD-in | -76.14, -48.91 | 69.19, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.995 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -163.99, 160.01 | APE9-dihe-na | 134.89, -153.13 | APE8-dihe-in | -119.22, 128.69 | APE8-rot-in | 299.44 | APE67-dihe-in | -61.81, -21.05 | -49.68, -44.36 | APE12-dist-in | 8.283 | APE11-dist-in | 11.557 | APE10-dist-in | 5.957 | APE9-dist-in | 3.903 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.12 | 0.188 | 0.241 | A | 358 | 322 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6npz | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.7e-99 | 337.5 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6NPZB | P31749 | 141 | 477 | 480.0 | No_ligand | No_ligand | Active | DFGin | 6.492 | 13.71 | BLAminus | -117.03, 171.77 | 71.96, 91.9 | -107.91, 11.41 | 295.22, 94.23 | -65.12, -23.31 | in-in | in | 8.806 | Saltbr-in | 3.089 | HRD-in | -77.35, -47.58 | 69.03, -7.27 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.868 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.06, 158.85 | APE9-dihe-na | 134.94, -150.01 | APE8-dihe-in | -122.61, 125.21 | APE8-rot-in | 296.0 | APE67-dihe-in | -68.07, -17.45 | -48.75, -43.62 | APE12-dist-in | 8.484 | APE11-dist-in | 11.691 | APE10-dist-in | 6.044 | APE9-dist-in | 3.856 | None | TPO308,SEP473,SEP477 | TPO308,SEP473,SEP477 | XRAY | 2.12 | 0.188 | 0.241 | B | 358 | 323 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6npz | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.7e-99 | 337.5 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 4GV1A | P31749 | 144 | 477 | 480.0 | 0XZ:60501 | Type1 | Active | DFGin | 6.488 | 13.562 | BLAminus | -122.36, 161.99 | 68.48, 91.61 | -104.89, 11.22 | 297.02, 96.69 | -63.45, -24.57 | in-in | in | 8.817 | Saltbr-in | 2.472 | HRD-in | -73.6, -46.3 | 69.86, -10.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -158.52, 165.79 | APE9-dihe-na | 129.18, -173.05 | APE8-dihe-in | -103.26, 131.39 | APE8-rot-in | 301.03 | APE67-dihe-in | -66.34, -18.55 | -46.14, -49.45 | APE12-dist-in | 8.481 | APE11-dist-in | 11.553 | APE10-dist-in | 5.998 | APE9-dist-in | 4.098 | None | TPO308 | TPO308 | XRAY | 1.49 | 0.182 | 0.21 | A | 340 | 329 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4gv1 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3OCBA | P31749 | 144 | 478 | 480.0 | XM1:1 | Type1 | Active | DFGin | 6.638 | 13.803 | BLAminus | -116.95, 176.33 | 66.85, 80.21 | -101.71, 15.06 | 291.18, 80.12 | -62.95, -27.15 | in-in | in | 8.771 | Saltbr-in | 2.77 | HRD-in | -68.69, -47.69 | 74.78, -17.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.986 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -155.18, 163.1 | APE9-dihe-na | 135.15, -135.96 | APE8-dihe-in | -136.2, 122.51 | APE8-rot-in | 298.45 | APE67-dihe-in | -66.42, -19.48 | -44.24, -42.98 | APE12-dist-in | 8.435 | APE11-dist-in | 11.489 | APE10-dist-in | 5.888 | APE9-dist-in | 4.058 | S473D | TPO308 | TPO308 | XRAY | 2.7 | 0.217 | 0.282 | A | 341 | 316 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ocb | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3OCBB | P31749 | 144 | 478 | 480.0 | XM1:2 | Type1 | Active | DFGin | 6.332 | 13.399 | BLAminus | -134.12, 162.45 | 65.57, 102.27 | -117.67, 11.66 | 296.51, 86.34 | -58.99, -28.22 | in-in | in | 8.815 | Saltbr-in | 2.871 | HRD-in | -68.9, -44.89 | 75.11, -22.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.078 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.43, 165.77 | APE9-dihe-na | 133.07, -137.47 | APE8-dihe-in | -130.52, 128.21 | APE8-rot-in | 301.82 | APE67-dihe-in | -61.46, -22.02 | -42.63, -52.7 | APE12-dist-in | 8.732 | APE11-dist-in | 11.603 | APE10-dist-in | 6.079 | APE9-dist-in | 4.134 | S473D | TPO308 | TPO308 | XRAY | 2.7 | 0.217 | 0.282 | B | 341 | 320 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ocb | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3OW4A | P31749 | 144 | 478 | 480.0 | SMY:60001 | Type1 | Active | DFGin | 6.386 | 13.523 | BLAminus | -119.32, 159.71 | 79.63, 82.83 | -104.78, 4.01 | 298.86, 82.1 | -54.94, -24.29 | in-in | in | 8.955 | Saltbr-in | 2.902 | HRD-in | -70.99, -49.36 | 69.67, -8.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.936 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -157.63, 156.89 | APE9-dihe-na | 142.86, -142.49 | APE8-dihe-in | -124.25, 130.13 | APE8-rot-in | 298.03 | APE67-dihe-in | -63.26, -12.53 | -44.97, -47.55 | APE12-dist-in | 8.407 | APE11-dist-in | 11.499 | APE10-dist-in | 5.943 | APE9-dist-in | 4.122 | S473D | TPO308 | TPO308 | XRAY | 2.6 | 0.197 | 0.268 | A | 341 | 318 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ow4 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3OW4B | P31749 | 144 | 478 | 480.0 | SMY:60002 | Type1 | Active | DFGin | 6.468 | 13.471 | BLAminus | -110.6, 166.76 | 74.64, 94.72 | -107.78, 10.54 | 297.92, 88.21 | -53.21, -30.59 | in-in | in | 9.014 | Saltbr-in | 2.873 | HRD-in | -68.95, -46.49 | 77.32, -19.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.905 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.84, 158.48 | APE9-dihe-na | 136.94, -160.6 | APE8-dihe-in | -112.04, 132.88 | APE8-rot-in | 279.55 | APE67-dihe-in | -64.15, -17.53 | -43.71, -49.28 | APE12-dist-in | 8.567 | APE11-dist-in | 11.482 | APE10-dist-in | 6.0 | APE9-dist-in | 4.209 | S473D | TPO308 | TPO308 | XRAY | 2.6 | 0.197 | 0.268 | B | 341 | 318 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3ow4 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3QKLA | P31749 | 144 | 478 | 480.0 | SMR:60001 | Type1 | Active | DFGin | 6.338 | 13.63 | BLAminus | -120.73, 173.12 | 65.05, 75.71 | -95.61, 13.62 | 302.87, 90.58 | -65.29, -24.68 | in-in | in | 9.025 | Saltbr-in | 2.669 | HRD-in | -79.32, -50.18 | 77.61, -12.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.808 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.72, 167.27 | APE9-dihe-na | 129.72, -141.45 | APE8-dihe-in | -129.9, 128.86 | APE8-rot-in | 291.61 | APE67-dihe-in | -64.11, -23.78 | -46.08, -46.14 | APE12-dist-in | 8.149 | APE11-dist-in | 11.608 | APE10-dist-in | 5.994 | APE9-dist-in | 3.707 | S473D | TPO308 | TPO308 | XRAY | 1.9 | 0.196 | 0.243 | A | 341 | 318 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3qkl | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3QKMA | P31749 | 144 | 478 | 480.0 | SM9:1 | Type1 | Active | DFGin | 6.551 | 13.483 | BLAminus | -120.8, 163.74 | 70.66, 92.07 | -106.66, 15.27 | 300.92, 94.29 | -62.34, -28.26 | in-in | in | 9.201 | Saltbr-in | 2.666 | HRD-in | -70.68, -45.98 | 71.02, -16.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.824 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -153.62, 157.36 | APE9-dihe-na | 116.69, 169.89 | APE8-dihe-in | -83.27, 128.83 | APE8-rot-in | 296.3 | APE67-dihe-in | -66.75, -19.54 | -36.8, -50.73 | APE12-dist-in | 8.46 | APE11-dist-in | 11.525 | APE10-dist-in | 5.915 | APE9-dist-in | 4.629 | S473D | TPO308 | TPO308 | XRAY | 2.2 | 0.191 | 0.252 | A | 341 | 330 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3qkm | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 4EKLA | P31749 | 144 | 478 | 480.0 | 0RF:501 | Type1 | Active | DFGin | 6.496 | 13.423 | BLAminus | -130.08, 156.46 | 77.16, 99.77 | -112.66, 14.16 | 298.65, 90.33 | -61.32, -30.96 | in-in | in | 8.958 | Saltbr-in | 2.452 | HRD-in | -78.38, -44.96 | 68.93, -13.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.757 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.83, 160.76 | APE9-dihe-na | 116.71, 166.32 | APE8-dihe-in | -83.66, 133.51 | APE8-rot-in | 293.53 | APE67-dihe-in | -68.09, -18.95 | -43.13, -46.31 | APE12-dist-in | 8.36 | APE11-dist-in | 11.512 | APE10-dist-in | 6.011 | APE9-dist-in | 4.443 | S473D | TPO308 | TPO308 | XRAY | 2.0 | 0.175 | 0.235 | A | 341 | 330 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 4ekl | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3CQWA | P31749 | 144 | 478 | 480.0 | CQW:60999 | Type1 | Active | DFGin | 6.338 | 13.09 | BLAminus | -122.41, 167.11 | 74.19, 82.7 | -100.79, 9.25 | 295.72, 101.99 | -67.19, -25.09 | in-in | in | 8.608 | Saltbr-in | 3.437 | HRD-in | -79.68, -40.11 | 70.25, -18.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -154.61, 166.29 | APE9-dihe-na | 132.98, -141.71 | APE8-dihe-in | -134.77, 132.14 | APE8-rot-in | 286.58 | APE67-dihe-in | -67.95, -20.8 | -49.28, -45.72 | APE12-dist-in | 8.374 | APE11-dist-in | 11.536 | APE10-dist-in | 5.934 | APE9-dist-in | 3.951 | S473D | TPO308 | TPO308 | XRAY | 2.0 | 0.203 | 0.257 | A | 342 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3cqw | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3MV5A | P31749 | 144 | 477 | 480.0 | XFE:60999 | Type1 | Active | DFGin | 6.512 | 13.107 | BLAminus | -110.68, 173.87 | 55.61, 106.15 | -116.13, 8.16 | 292.02, 88.05 | -68.88, -21.78 | in-in | in | 8.573 | Saltbr-in | 2.645 | HRD-in | -81.07, -37.62 | 75.3, -21.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -163.23, 167.83 | APE9-dihe-na | 126.38, -137.1 | APE8-dihe-in | -133.69, 127.23 | APE8-rot-in | 287.39 | APE67-dihe-in | -69.19, -14.76 | -48.38, -39.25 | APE12-dist-in | 8.467 | APE11-dist-in | 11.692 | APE10-dist-in | 6.145 | APE9-dist-in | 4.185 | S473D | TPO308 | TPO308 | XRAY | 2.47 | 0.205 | 0.282 | A | 342 | 316 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3mv5 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3MVHA | P31749 | 145 | 476 | 480.0 | WFE:999 | Type1 | Active | DFGin | 6.609 | 13.205 | BLAminus | -120.33, 157.64 | 77.18, 89.81 | -109.14, 14.39 | 295.05, 87.49 | -62.89, -24.97 | in-in | in | 8.782 | Saltbr-in | 2.62 | HRD-in | -82.77, -44.94 | 75.58, -15.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.836 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.65, 167.39 | APE9-dihe-na | 135.14, -139.29 | APE8-dihe-in | -137.11, 131.02 | APE8-rot-in | 291.39 | APE67-dihe-in | -63.24, -17.86 | -53.88, -42.66 | APE12-dist-in | 8.149 | APE11-dist-in | 11.591 | APE10-dist-in | 5.855 | APE9-dist-in | 3.756 | S473D | TPO308 | TPO308 | XRAY | 2.01 | 0.181 | 0.23 | A | 342 | 312 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3mvh | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6CCYA | P31749 | 144 | 983 | 480.0 | EX4:60501 | Type1 | Active | DFGin | 6.833 | 14.216 | BLAminus | -118.22, 172.28 | 65.22, 87.23 | -99.08, 6.12 | 296.87, 97.72 | -61.52, -36.28 | in-in | in | 9.387 | Saltbr-in | 2.725 | HRD-in | -70.12, -46.7 | 65.1, -15.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.814 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.15, 164.77 | APE9-dihe-na | 117.98, 177.81 | APE8-dihe-in | -89.16, 122.56 | APE8-rot-in | 287.17 | APE67-dihe-in | -60.32, -21.6 | -32.19, -51.09 | APE12-dist-in | 8.32 | APE11-dist-in | 11.49 | APE10-dist-in | 5.811 | APE9-dist-in | 4.408 | N199S,S396P,E397S,T433V | TPO308 | TPO308 | XRAY | 2.18 | 0.237 | 0.276 | A | 343 | 307 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6ccy | Homo sapiens | AGC_AKT1_HUMAN | AGC | 4.1e-99 | 336.9 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3QKKA | P31749 | 144 | 478 | 480.0 | SMH:60001 | Type1.5_Front | Active | DFGin | 6.383 | 13.598 | BLAminus | -116.54, -179.44 | 52.7, 85.0 | -102.02, 14.36 | 303.33, 93.01 | -66.45, -23.02 | in-in | in | 8.916 | Saltbr-in | 2.342 | HRD-in | -78.65, -51.68 | 79.72, -12.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.763 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.57, 164.52 | APE9-dihe-na | 135.56, -139.12 | APE8-dihe-in | -127.86, 127.7 | APE8-rot-in | 299.02 | APE67-dihe-in | -62.38, -25.83 | -44.42, -46.66 | APE12-dist-in | 8.22 | APE11-dist-in | 11.566 | APE10-dist-in | 6.028 | APE9-dist-in | 3.779 | S473D | TPO308 | TPO308 | XRAY | 2.3 | 0.202 | 0.25 | A | 341 | 327 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3qkk | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3CQUA | P31749 | 144 | 478 | 480.0 | CQU:60999 | Type1 | Inactive | DFGin | 6.162 | 12.752 | BLAminus | -125.29, 173.04 | 74.77, 101.51 | -111.55, 14.45 | 309.48, 77.95 | -55.91, -32.71 | in-out | in | 9.246 | Saltbr-out | 4.113 | HRD-in | -63.98, -47.97 | 77.74, -15.86 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.003 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.44, 176.23 | APE9-dihe-na | 125.93, -142.07 | APE8-dihe-in | -126.34, 131.3 | APE8-rot-in | 289.37 | APE67-dihe-in | -62.32, -24.17 | -48.41, -45.96 | APE12-dist-in | 8.309 | APE11-dist-in | 11.455 | APE10-dist-in | 6.059 | APE9-dist-in | 3.993 | S473D | TPO308 | TPO308 | XRAY | 2.2 | 0.207 | 0.283 | A | 342 | 319 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 3cqu | Homo sapiens | AGC_AKT1_HUMAN | AGC | 2.3e-99 | 337.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 8UVYA | P31749 | 3 | 439 | 480.0 | XOO:60502 | Allosteric | Inactive | DFGout | 19.147 | 9.117 | BBAminus | -87.71, 159.46 | -125.79, 51.81 | -104.71, 8.89 | 306.76, 157.9 | -76.01, 144.81 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -80.44, -49.7 | 65.22, 18.47 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.329 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -75.27, -63.55 | APE9-dihe-na | -84.1, -150.14 | APE8-dihe-in | -112.51, 118.73 | APE8-rot-in | 303.11 | APE67-dihe-in | -70.02, -8.73 | -61.09, -34.89 | APE12-dist-in | 11.509 | APE11-dist-in | 11.913 | APE10-dist-in | 7.703 | APE9-dist-out | 6.561 | E17K | None | None | XRAY | 2.11 | 0.209 | 0.255 | A | 438 | 396 | 21 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 8uvy | Homo sapiens | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 8UW2A | P31749 | 4 | 437 | 480.0 | XOO:60502 | Allosteric | Inactive | DFGout | 19.594 | 9.174 | BBAminus | -85.5, 157.67 | -121.72, 55.74 | -105.08, 2.24 | 304.7, 161.96 | -67.3, 146.74 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -75.89, -48.3 | 59.85, 6.57 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 13.673 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -78.7, 9.37 | APE9-dihe-na | -151.7, -145.87 | APE8-dihe-in | -109.15, 106.27 | APE8-rot-out | 18.96 | APE67-dihe-in | -70.15, -8.9 | -92.15, -6.4 | APE12-dist-out | 18.057 | APE11-dist-out | 14.765 | APE10-dist-out | 10.604 | APE9-dist-out | 11.153 | None | None | None | XRAY | 2.2 | 0.223 | 0.279 | A | 438 | 392 | 19 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 8uw2 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 8UW9A | P31749 | 3 | 428 | 480.0 | XQ2:60501 | Allosteric | Inactive | DFGout | 18.976 | 9.3 | BBAminus | -90.79, 158.27 | -126.08, 50.43 | -104.96, 7.49 | 302.98, 161.85 | -82.17, 151.97 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -80.58, -46.97 | 73.31, -13.02 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.346 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -78.06, -70.69 | APE9-dihe-na | -63.13, 144.96 | APE8-dihe-in | -69.73, 119.44 | APE8-rot-in | 308.33 | APE67-dihe-in | -66.64, -12.63 | -58.13, -37.16 | APE12-dist-in | 12.561 | APE11-dist-in | 12.026 | APE10-dist-in | 7.549 | APE9-dist-out | 6.208 | None | None | None | XRAY | 1.9 | 0.207 | 0.245 | A | 438 | 388 | 19 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 8uw9 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 8UW7A | P31749 | 3 | 439 | 480.0 | XOO:60502 | Allosteric | Inactive | DFGout | 19.268 | 9.131 | BBAminus | -88.27, 162.56 | -129.0, 47.08 | -101.62, 6.17 | 304.62, 157.46 | -65.02, 141.6 | out-out | out | 14.185 | Saltbr-out | 16.163 | HRD-in | -77.74, -48.14 | 69.36, -7.13 | out-out-out | SNCooo | out-out | ActLoopNT-out | 15.133 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 168.57 | APE8-dihe-in | -110.93, 76.79 | APE8-rot-out | 38.95 | APE67-dihe-in | -76.05, -14.39 | -64.32, -17.63 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.831 | None | None | YCM77,YCM296 | XRAY | 1.972 | 0.22 | 0.265 | A | 438 | 399 | 17 | 0 | 0 | 12 | [[150, 408]] | 1.0 | 8uw7 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 4.9e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 3O96A | P31749 | 2 | 429 | 480.0 | IQO:444 | Allosteric | Inactive | DFGout | 16.13 | 7.768 | BBAminus | -84.04, 164.11 | -138.96, 67.69 | -114.58, 18.46 | 294.17, 141.85 | -57.09, 121.09 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -85.54, -46.27 | 73.79, -8.96 | none-out-none | SNCnon | out-none | ActLoopNT-out | 14.705 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -63.73, -20.88 | 999.0, -53.98 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.249 | 0.308 | A | 446 | 367 | 24 | 0 | 0 | 14 | [[150, 408]] | 1.0 | 3o96 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.7 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6HHHA | P31749 | 2 | 439 | 480.0 | G4Q:501 | Allosteric | Inactive | DFGout | 19.432 | 8.904 | BBAminus | -82.84, 168.78 | -138.99, 51.81 | -104.05, 22.45 | 309.63, 151.96 | -74.89, 142.62 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -70.92, -45.22 | 71.01, -6.93 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.659 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -141.4 | APE8-dihe-out | -68.07, -39.94 | APE8-rot-out | 43.05 | APE67-dihe-in | -61.63, -40.25 | -82.49, 7.03 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 14.39 | E114A,E115A,E116A | None | None | XRAY | 2.7 | 0.217 | 0.266 | A | 446 | 379 | 25 | 0 | 0 | 11 | [[150, 408]] | 1.0 | 6hhh | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6HHJA | P31749 | 3 | 444 | 480.0 | G4H:501 | Allosteric | Inactive | DFGout | 18.637 | 9.927 | BBAminus | -85.85, 154.25 | -131.76, 65.33 | -114.43, 2.7 | 306.85, 152.03 | -81.33, 157.37 | out-out | out | 16.597 | Saltbr-out | 20.784 | HRD-in | -70.38, -43.13 | 62.3, -0.73 | out-out-out | SNCooo | out-out | ActLoopNT-out | 15.398 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -96.59, 105.04 | APE9-dihe-na | 69.68, -150.96 | APE8-dihe-in | -112.16, 140.11 | APE8-rot-out | 58.43 | APE67-dihe-in | -58.84, -27.51 | -94.58, 2.39 | APE12-dist-out | 16.493 | APE11-dist-out | 16.034 | APE10-dist-out | 10.684 | APE9-dist-out | 11.298 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.223 | 0.243 | A | 446 | 410 | 0 | 0 | 0 | 0 | [[150, 408]] | 1.0 | 6hhj | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6S9WA | P31749 | 3 | 444 | 480.0 | L1Z:501 | Allosteric | Inactive | DFGout | 18.014 | 9.778 | BBAminus | -88.23, 159.68 | -135.32, 63.28 | -108.07, 5.2 | 307.51, 150.05 | -79.62, 159.51 | out-out | out | 16.719 | Saltbr-out | 21.04 | HRD-in | -77.04, -47.59 | 74.55, -19.15 | out-out-out | SNCooo | out-out | ActLoopNT-out | 15.677 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -115.76, 103.74 | APE9-dihe-na | 82.07, -166.58 | APE8-dihe-in | -98.52, 141.96 | APE8-rot-out | 173.15 | APE67-dihe-in | -62.82, -22.8 | -94.37, -0.32 | APE12-dist-out | 16.616 | APE11-dist-out | 16.139 | APE10-dist-out | 10.913 | APE9-dist-out | 11.124 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.21 | 0.263 | A | 446 | 411 | 2 | 0 | 0 | 2 | [[150, 408]] | 1.0 | 6s9w | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 4EJNA | P31749 | 4 | 438 | 480.0 | 0R4:501 | Type1 | Inactive | DFGout | 18.374 | 8.329 | BBAminus | -86.73, 154.01 | -129.51, 54.97 | -106.79, 23.78 | 305.4, 154.78 | -69.14, 128.42 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -74.68, -58.46 | 77.98, 6.43 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 16.065 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioo | APE10-dihe-na | -97.72, 139.0 | APE9-dihe-na | 109.04, 163.38 | APE8-dihe-in | -97.01, 108.52 | APE8-rot-in | 315.65 | APE67-dihe-in | -57.15, -23.24 | -58.45, -30.75 | APE12-dist-out | 14.955 | APE11-dist-in | 13.395 | APE10-dist-out | 8.158 | APE9-dist-out | 6.501 | E114A,E115A,E116A | None | None | XRAY | 2.19 | 0.239 | 0.276 | A | 446 | 376 | 18 | 0 | 0 | 5 | [[150, 408]] | 1.0 | 4ejn | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 5KCVA | P31749 | 6 | 438 | 480.0 | 6S1:501 | Allosteric | Inactive | DFGout | 18.399 | 8.593 | None | -66.09, 150.37 | -131.74, 48.39 | -109.26, 34.53 | 301.12, 163.72 | -73.63, 124.84 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -80.28, -36.69 | 71.61, -16.44 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.9, -11.63 | 999.0, -43.42 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | E114A,E115A,E116A | None | None | XRAY | 2.7 | 0.213 | 0.269 | A | 460 | 353 | 33 | 0 | 0 | 16 | [[150, 408]] | 1.0 | 5kcv | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.6e-99 | 336.5 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 7APJA | P31749 | 3 | 439 | 480.0 | No_ligand | No_ligand | Inactive | DFGout | 15.36 | 7.847 | None | -119.51, 172.58 | -151.35, 78.25 | -78.82, 999.0 | 276.7, 1.08 | 999.0, 999.0 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -72.58, -35.61 | 73.77, -41.9 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 73.92 | APE8-rot-out | 58.45 | APE67-dihe-in | -70.85, -7.62 | -68.6, -17.11 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | S2N | None | None | XRAY | 2.05 | 0.213 | 0.252 | A | 440 | 376 | 39 | 0 | 0 | 18 | [[150, 408]] | 1.0 | 7apj | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5e-99 | 336.8 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6HHFA | P31749 | 3 | 439 | 480.0 | G4K:501 | Allosteric | Inactive | None | 999.0 | 8.943 | None | -81.4, 157.14 | -136.1, 63.0 | -116.97, 21.98 | 304.54, 147.84 | -76.24, 135.42 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -67.92, -42.11 | 68.98, -10.23 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 16.026 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 110.64 | APE8-rot-out | 65.96 | APE67-dihe-in | -73.6, -35.94 | -67.69, -4.64 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | E114A,E115A,E116A | None | None | XRAY | 2.9 | 0.233 | 0.274 | A | 446 | 366 | 32 | 0 | 0 | 14 | [[150, 408]] | 1.0 | 6hhf | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6HHGA | P31749 | 3 | 444 | 480.0 | G4T:501 | Allosteric | Inactive | None | 999.0 | 9.861 | None | -89.51, 153.73 | -128.41, 67.53 | -114.64, 10.8 | 307.59, 150.55 | -85.41, 154.74 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -68.28, -46.2 | 67.11, -14.18 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.289 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -107.85, 97.08 | APE9-dihe-na | 87.64, -165.9 | APE8-dihe-in | -105.98, 137.43 | APE8-rot-out | 58.9 | APE67-dihe-in | -57.38, -21.16 | -89.5, -4.41 | APE12-dist-out | 17.366 | APE11-dist-out | 16.179 | APE10-dist-out | 10.888 | APE9-dist-out | 11.447 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.212 | 0.246 | A | 446 | 386 | 21 | 0 | 0 | 3 | [[150, 408]] | 1.0 | 6hhg | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6HHIA | P31749 | 3 | 444 | 480.0 | G4N:501 | Allosteric | Inactive | None | 999.0 | 9.394 | None | -89.1, 165.97 | -135.32, 55.99 | -110.01, 13.3 | 309.82, 146.72 | -70.54, 150.25 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -69.6, -44.24 | 72.4, -22.65 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.413 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -105.21, 101.21 | APE9-dihe-na | 81.98, -162.79 | APE8-dihe-in | -113.39, 139.7 | APE8-rot-out | 66.27 | APE67-dihe-in | -49.46, -24.76 | -86.47, -13.4 | APE12-dist-out | 17.097 | APE11-dist-out | 15.773 | APE10-dist-out | 10.853 | APE9-dist-out | 11.014 | E114A,E115A,E116A | None | None | XRAY | 2.7 | 0.229 | 0.258 | A | 446 | 389 | 19 | 0 | 0 | 3 | [[150, 408]] | 1.0 | 6hhi | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 6S9XA | P31749 | 3 | 443 | 480.0 | L1W:501 | Allosteric | Inactive | None | 999.0 | 9.471 | None | -83.65, 171.5 | -148.58, 59.04 | -110.35, 19.84 | 309.98, 147.1 | -81.71, 151.08 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -70.64, -44.34 | 67.14, 2.45 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.655 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nooo | APE10-dihe-na | -128.24, 142.43 | APE9-dihe-na | 73.42, -170.52 | APE8-dihe-in | -106.82, 110.63 | APE8-rot-out | 60.31 | APE67-dihe-in | -66.32, -9.87 | -76.1, -5.54 | APE12-dist-none | 999.0 | APE11-dist-out | 16.242 | APE10-dist-out | 10.715 | APE9-dist-out | 10.287 | E114A,E115A,E116A | None | None | XRAY | 2.6 | 0.214 | 0.234 | A | 446 | 382 | 23 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 6s9x | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 7NH4A | P31749 | 4 | 444 | 480.0 | UCE:501 | Allosteric | Inactive | None | 999.0 | 9.714 | None | -89.66, 161.99 | -134.99, 53.83 | -102.41, 15.77 | 307.61, 150.23 | -85.21, 156.95 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -71.71, -43.96 | 65.0, -1.87 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.71 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -91.29, 122.41 | APE9-dihe-na | 62.81, -158.06 | APE8-dihe-in | -116.84, 141.55 | APE8-rot-out | 65.03 | APE67-dihe-in | -52.37, -30.57 | -89.05, -2.1 | APE12-dist-out | 16.82 | APE11-dist-out | 16.123 | APE10-dist-out | 10.705 | APE9-dist-out | 11.149 | E114A,E115A,E116A | None | None | XRAY | 2.3 | 0.224 | 0.246 | A | 446 | 383 | 24 | 0 | 0 | 6 | [[150, 408]] | 1.0 | 7nh4 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| AKT1_HUMAN | 7NH5A | P31749 | 3 | 444 | 480.0 | UC8:502 | Allosteric | Inactive | None | 999.0 | 9.683 | None | -94.24, 161.49 | -131.31, 59.8 | -111.8, 8.17 | 304.51, 156.46 | -83.9, 163.26 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -72.19, -47.43 | 76.17, -13.35 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 15.616 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nooo | APE10-dihe-na | -89.96, 112.26 | APE9-dihe-na | 68.59, -149.12 | APE8-dihe-in | -121.33, 137.31 | APE8-rot-in | 284.5 | APE67-dihe-in | -57.38, -14.67 | -81.19, -19.07 | APE12-dist-none | 999.0 | APE11-dist-out | 15.973 | APE10-dist-out | 10.445 | APE9-dist-out | 11.434 | E114A,E115A,E116A | None | None | XRAY | 1.9 | 0.201 | 0.228 | A | 446 | 383 | 24 | 0 | 0 | 7 | [[150, 408]] | 1.0 | 7nh5 | Homo sapiens | AGC_AKT1_HUMAN | AGC | 5.2e-99 | 336.6 | 1 | 260 | 260 | 291 | 292 | 293 | 295 | 297 | 179 | 198 | 202 | 271 | 273 | 272 | 274 | 331 | 319 | 314 | 313 | 312 | 311 | 310 | 309 | 308 | 228 | RAC-alpha serine/threonine-protein kinase |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|