Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 6 | 4QMUA |
DFGin | ABAminus | 3 | 5DT0A |
DFGin | None | 3 | 8B99A |
None | None | 1 | 5OBRA |
Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|
AGC | PRKACA | KAPCA_HUMAN | cAMP-dependent protein kinase catalytic subunit alpha | 3AMAA | 1.75 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DPVA | 2.285 | Inactive | DFGin | ABAminus | out-in | in-out | 5DN SKE | Allosteric Type1 |
CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DR6A | 2.534 | Inactive | DFGin | ABAminus | out-in | in-out | 5E1 SKE | Allosteric Type1 |
CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DT0A | 2.15 | Inactive | DFGin | ABAminus | in-in | in-out | SKE | Type1 |
CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DR9A | 2.47 | Inactive | DFGin | BLAminus | out-out | out-out | SKE 5E2 | Type1 Allosteric |
CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5OBRA | 2.62 | Inactive | None | None | out-out | out-out | 9QT SKE | Allosteric Type1 |
STE | STK24 | STK24_HUMAN | Serine/threonine-protein kinase 24 | 4QMUA | 1.546 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5USYA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5USYB | 2.0 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 6DRWA | 2.303 | Inactive | DFGin | BLAminus | in-out | in-in | SKE | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 8B99A | 1.6 | Inactive | DFGin | None | out-none | out-out | SKE | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5WINA | 2.38 | Inactive | DFGin | None | out-none | out-out | SKE | Type1 |
TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5USZA | 2.103 | Inactive | DFGin | None | in-none | out-out | SKE | Type1 |
Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 6 | 4QMUA |
DFGin | ABAminus | 3 | 5DT0A |
DFGin | None | 3 | 8B99A |
None | None | 1 | 5OBRA |
Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Homo sapiens | AGC | PRKACA | KAPCA_HUMAN | cAMP-dependent protein kinase catalytic subunit alpha | 3AMAA | 1.75 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
Homo sapiens | CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DPVA | 2.285 | Inactive | DFGin | ABAminus | out-in | in-out | 5DN SKE | Allosteric Type1 |
Homo sapiens | CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DR6A | 2.534 | Inactive | DFGin | ABAminus | out-in | in-out | 5E1 SKE | Allosteric Type1 |
Homo sapiens | CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DT0A | 2.15 | Inactive | DFGin | ABAminus | in-in | in-out | SKE | Type1 |
Homo sapiens | CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5DR9A | 2.47 | Inactive | DFGin | BLAminus | out-out | out-out | SKE 5E2 | Type1 Allosteric |
Homo sapiens | CAMK | AURKA | AURKA_HUMAN | Aurora kinase A | 5OBRA | 2.62 | Inactive | None | None | out-out | out-out | 9QT SKE | Allosteric Type1 |
Homo sapiens | STE | STK24 | STK24_HUMAN | Serine/threonine-protein kinase 24 | 4QMUA | 1.546 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5USYA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5USYB | 2.0 | Active | DFGin | BLAminus | in-in | in-in | SKE | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 6DRWA | 2.303 | Inactive | DFGin | BLAminus | in-out | in-in | SKE | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 8B99A | 1.6 | Inactive | DFGin | None | out-none | out-out | SKE | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5WINA | 2.38 | Inactive | DFGin | None | out-none | out-out | SKE | Type1 |
Homo sapiens | TYR | JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 | 5USZA | 2.103 | Inactive | DFGin | None | in-none | out-out | SKE | Type1 |
Spatial | Dihedral | Chains | Representative |
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Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
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