Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 3 | 4TNBA |
DFGin | None | 1 | 6PJXA |
Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|
AGC | GRK5 | GRK5_HUMAN | G protein-coupled receptor kinase 5 | 4TNBA | 2.113 | Active | DFGin | BLAminus | in-in | in-in | SGV | Type1 |
AGC | GRK5 | GRK5_HUMAN | G protein-coupled receptor kinase 5 | 6PJXA | 1.96 | Inactive | DFGin | None | in-in | in-in | SGV | Type1 |
AGC | GRK6 | GRK6_HUMAN | G protein-coupled receptor kinase 6 | 3NYNA | 2.72 | Active | DFGin | BLAminus | in-in | in-in | SGV | Type1 |
AGC | GRK6 | GRK6_HUMAN | G protein-coupled receptor kinase 6 | 3NYNB | 2.72 | Active | DFGin | BLAminus | in-in | in-in | SGV | Type1 |
Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 7 | 4TNBA |
DFGin | None | 1 | 6PJXA |
Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MT9G | 7.0 | Inactive | DFGin | BLAminus | in-out | in-out | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MT8G | 5.8 | Active | DFGin | BLAminus | in-in | in-in | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MTAG | 4.1 | Inactive | DFGin | BLAminus | in-out | in-in | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MTBG | 4.0 | Active | DFGin | BLAminus | in-in | in-in | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Homo sapiens | AGC | GRK5 | GRK5_HUMAN | G protein-coupled receptor kinase 5 | 4TNBA | 2.113 | Active | DFGin | BLAminus | in-in | in-in | SGV | Type1 |
Homo sapiens | AGC | GRK5 | GRK5_HUMAN | G protein-coupled receptor kinase 5 | 6PJXA | 1.96 | Inactive | DFGin | None | in-in | in-in | SGV | Type1 |
Homo sapiens | AGC | GRK6 | GRK6_HUMAN | G protein-coupled receptor kinase 6 | 3NYNA | 2.72 | Active | DFGin | BLAminus | in-in | in-in | SGV | Type1 |
Homo sapiens | AGC | GRK6 | GRK6_HUMAN | G protein-coupled receptor kinase 6 | 3NYNB | 2.72 | Active | DFGin | BLAminus | in-in | in-in | SGV | Type1 |
Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 4 | 7MTBG |
Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MT9G | 7.0 | Inactive | DFGin | BLAminus | in-out | in-out | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MT8G | 5.8 | Active | DFGin | BLAminus | in-in | in-in | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MTAG | 4.1 | Inactive | DFGin | BLAminus | in-out | in-in | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |
Bos taurus | AGC | GRK1 | GRK1_BOVIN | Rhodopsin kinase GRK1 | 7MTBG | 4.0 | Active | DFGin | BLAminus | in-in | in-in | SGV SGV SGV SGV SGV SGV | Type1 Type1 Type1 Type1 Type1 Type1 |