6PJX

GRK5 (G protein-coupled receptor kinase 5)
Group: AGC
Uniprot: GRK5_HUMAN
Organism: Homo sapiens
Domain boundary: 186 - 448
Resolu: 1.96

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Inactive DFGin None in-in in-in SGV Type1 1 - 542 0
Representative sequence - Chain A
9 19 29 39
XMELENIVAN TVLLKAREGG GGKRKGKSKK WKEILKFPHI
49 59 69 79
SQCEDLRRTI DRDYCSLCDK QPIGRLLFRQ FCETRPGLEC
89 99 109 119
YIQFLDSVAE YEVTPDEKLG EKGKKIMTKY LTPKSPVFIA
129 139 149 159
QVGQDLVSQT EEKLLQKPCK ELFSACAQSV HEYLRGEPFH
169 179 189 199
EYLDSMFFDR FLQWKWLERQ PVTKNTFRQY RVLGKGGFGE
209 219 229 239
VCACQVRATG KMYACKRLEK KRIKKRKGES MALNEKQILE
249 259 269 279
KVNSQFVVNL AYAYETKDAL CLVLTIMNGG DLKFHIYNMG
289 299 309 319
NPGFEEERAL FYAAEILCGL EDLHHENTVY RDLKPENILL
329 339 349 359
DDYGHIRISD LGLAVKIPEG DLIRGRVGTV GYMAPEVLNN
369 379 389 399
QRYGLSPDYW GLGCLIYEMI EGQSPFRGRK EKVKREEVDR
409 419 429 439
RVLETEEVYS HKFSEEAKSI CKMLLTKDAK QRLGCQEEEA
449 459 469 479
AEVKRHPFFR NMNFKRLEAG MLDPPFVPDP RAVYCKDVLD
489 499 509 519
IEQFSTVKGV NLDHTDDDFY SKFSTGSVSI PWQNEMIETE
529 539 549 559
CFKELNVFGP NGTLPPDLNR NHPpeppkkg llqrlfkrqh
569 579 589
qnnsksspss ktsfnhhins nhvssnstgs s
Lower-case residues are disordered in structure.
Mutations: E104K,R304H,G438E
Phosphorylation: None