3NYN

GRK6 (G protein-coupled receptor kinase 6)
Group: AGC
Uniprot: GRK6_HUMAN
Organism: Homo sapiens
Domain boundary: 186 - 448
Resolu: 2.72

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in SGV Type1 2 - 557 0
B Active DFGin BLAminus in-in in-in SGV Type1 2 - 557 0
Representative sequence - Chain B
10 20 30 40
XELENIVANT VLLKAREGGG GNRKGKSKKW RQMLQFPHIS
50 60 70 80
QCEELRLSLE RDYHSLCERQ PIGRLLFREF CATRPELSRC
90 100 110 120
VAFLDGVAEY EVTPDDKRKA CGRQLTQNFL SHTGPDLIPE
130 140 150 160
VPRQLVTNCT QRLEQGPCKD LFQELTRLTH EYLSVAPFAD
170 180 190 200
YLDSIYFNRF LQWKWLERQP VTKNTFRQYR VLGKGGFGEV
210 220 230 240
CACQVRATGK MYACKKLEKK RIKKRKGEAM ALNEKQILEK
250 260 270 280
VNSRFVVSLA YAYETKDALC LVLTLMNGGD LKFHIYHMGQ
290 300 310 320
AGFPEARAVF YAAEICCGLE DLHRERIVYR DLKPENILLD
330 340 350 360
DHGHIRISDL GLAVHVPEGQ TIKGRVGTVG YMAPEVVKNE
370 380 390 400
RYTFSPDWWA LGCLLYEMIA GQSPFQqrkK KIKREEVERL
410 420 430 440
VKEVPEEYSE RFSPQARSLC SQLLCKDPAE RLGCRGGSAR
450 460 470 480
EVKEHPLFKK LNFKRLGAGM LEPPFKPDPQ AIYCKDVLDI
490 500 510 520
EQFSTVKGVE LEPTDQDFYQ KFATGSVPIP WQNEMVETEC
530 540 550 560
FQELNVFGLD GSVPPDLDWK GQPPAPPKKG LLQRLFSrqd
570
ccgncsdsee elptrl
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: None