| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK14 | MK14_HUMAN | 3HL7A | Q16539 | 6 | 352 | 360.0 | I47:60401,I46:60402 | Type1,Allosteric | Inactive | DFGin | 5.2347 | 13.6446 | BLBplus | -124.2, 170.0 | 68.57, 19.0 | -68.49, 146.41 | 46.64, 88.83 | 77.19, -0.15 | in-in | in | 9.0409 | Saltbr-in | 2.4506 | HRD-in | -63.1, -58.98 | 80.27, -17.67 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 155.78 | APE8-dihe-out | -66.44, -27.56 | APE8-rot-none | 999.0 | APE67-dihe-in | -57.86, -27.57 | -47.26, -39.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.5313 | None | None | None | XRAY | 1.88 | 0.2 | 0.228 | A | 360.0 | 336.0 | 11 | 25 | 14 | 11 | [[24, 308]] | 1.0 | 3hl7 | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3HLLA | Q16539 | 5 | 352 | 360.0 | I45:60401,I46:60402,PO2:60501 | Type1,Allosteric,Allosteric | Inactive | DFGin | 5.053 | 13.5716 | BLBplus | -104.99, 158.54 | 67.03, 24.11 | -71.37, 152.95 | 45.58, 87.31 | 67.6, 1.84 | in-out | in | 9.1864 | Saltbr-out | 3.9688 | HRD-in | -64.7, -58.11 | 82.94, -23.06 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnoo | APE10-dihe-na | 999.0, -18.34 | APE9-dihe-na | -77.72, 94.48 | APE8-dihe-out | -49.19, -31.53 | APE8-rot-none | 999.0 | APE67-dihe-in | -66.1, -25.14 | -64.45, -21.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 16.8147 | APE9-dist-out | 11.6667 | None | None | None | XRAY | 1.95 | 0.219 | 0.254 | A | 360.0 | 337.0 | 11 | 25 | 14 | 11 | [[24, 308]] | 1.0 | 3hll | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3HP2A | Q16539 | 4 | 355 | 360.0 | P36:401,I46:402,I46:403 | Type1,Allosteric,Allosteric | Inactive | DFGin | 10.3229 | 12.0791 | None | -88.89, 117.93 | 0.95, -90.69 | -132.19, 144.91 | 307.84, 89.53 | -100.53, 179.64 | in-in | in | 8.9859 | Saltbr-in | 3.0157 | HRD-in | -62.69, -56.28 | 83.82, -16.84 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, -83.28 | APE9-dihe-na | -69.46, 121.84 | APE8-dihe-out | -57.79, -33.94 | APE8-rot-in | 290.47 | APE67-dihe-in | -56.52, -29.08 | -65.16, -23.99 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 11.8086 | APE9-dist-out | 11.9697 | None | None | None | XRAY | 2.15 | 0.208 | 0.252 | A | 360.0 | 341.0 | 11 | 25 | 14 | 11 | [[24, 308]] | 1.0 | 3hp2 | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3HP5A | Q16539 | 6 | 352 | 360.0 | 52P:401,I46:402,I46:403 | Type1,Allosteric,Allosteric | Inactive | DFGin | 6.4998 | 14.3567 | None | -122.62, 154.65 | 81.43, 43.95 | -64.35, -69.27 | 340.23, 142.83 | -47.68, 999.0 | in-in | in | 8.692 | Saltbr-in | 3.0371 | HRD-in | -62.14, -57.25 | 84.4, -19.04 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnno | APE10-dihe-na | 999.0, -175.23 | APE9-dihe-na | -178.51, 127.74 | APE8-dihe-out | -56.55, -39.12 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.7, -27.21 | -46.07, -42.48 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.3903 | None | None | None | XRAY | 2.3 | 0.217 | 0.262 | A | 360.0 | 330.0 | 17 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 3hp5 | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 6QDZA | Q16539 | 5 | 352 | 360.0 | I46:401,HYK:402 | Allosteric,Type2 | Inactive | DFGout | 14.9123 | 9.0812 | BBAminus | -134.77, -179.97 | -142.81, 109.12 | -72.73, -21.08 | 264.45, 91.98 | 63.26, 999.0 | in-in | in | 8.4999 | Saltbr-in | 2.7579 | HRD-in | -75.35, -56.13 | 84.01, -14.16 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 120.14 | APE8-dihe-out | -58.44, -38.6 | APE8-rot-in | 261.35 | APE67-dihe-in | -64.54, -27.76 | -61.68, -25.18 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.4049 | None | None | None | XRAY | 1.73 | 0.206 | 0.246 | A | 362.0 | 327.0 | 21 | 25 | 12 | 13 | [[24, 308]] | 1.0 | 6qdz | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 6QE1A | Q16539 | 5 | 352 | 360.0 | I46:401,HYW:402 | Allosteric,Type2 | Inactive | DFGout | 14.5033 | 9.1773 | BBAminus | -141.03, -172.04 | -146.99, 109.37 | -71.94, -17.35 | 270.92, 90.33 | 65.73, 999.0 | in-in | in | 8.7612 | Saltbr-in | 2.6233 | HRD-in | -65.85, -55.55 | 81.72, -12.94 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 126.37 | APE8-dihe-out | -53.58, -40.3 | APE8-rot-in | 269.79 | APE67-dihe-in | -62.76, -30.98 | -60.8, -26.41 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.3191 | None | None | None | XRAY | 1.85 | 0.181 | 0.222 | A | 362.0 | 328.0 | 20 | 25 | 12 | 13 | [[24, 308]] | 1.0 | 6qe1 | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3K3IA | Q16539 | 5 | 352 | 360.0 | JZJ:1,I46:353,I46:2 | Type3,Allosteric,Allosteric | Inactive | DFGout | 13.8744 | 9.8725 | BBAminus | -143.79, -170.14 | -141.75, 114.95 | -78.16, -16.52 | 274.05, 114.76 | 49.78, 999.0 | in-in | in | 9.3253 | Saltbr-in | 2.6305 | HRD-in | -66.69, -52.65 | 76.63, -11.32 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 118.08 | APE9-dihe-na | -84.9, 132.08 | APE8-dihe-out | -50.88, -42.58 | APE8-rot-in | 276.73 | APE67-dihe-in | -63.3, -21.91 | -56.89, -25.41 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.1293 | None | None | None | XRAY | 1.7 | 0.196 | 0.242 | A | 350.0 | 332.0 | 16 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 3k3i | CMGC_MAPK14_HUMAN | CMGC | 5.3e-85 | 291.3 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 2YISA | Q16539 | 5 | 353 | 360.0 | YIS:1353,I46:1354 | Type2,Allosteric | Inactive | DFGout | 15.833 | 8.5763 | None | -138.39, -175.22 | -139.39, 106.04 | -86.53, 999.0 | 192.46, 60.65 | 999.0, 999.0 | in-in | in | 8.5948 | Saltbr-in | 2.6488 | HRD-in | -65.43, -49.96 | 74.88, -12.76 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | -110.86, 112.45 | APE9-dihe-na | -50.05, 127.69 | APE8-dihe-out | -57.83, -43.06 | APE8-rot-in | 274.36 | APE67-dihe-in | -59.28, -29.93 | -54.84, -31.58 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.1314 | None | None | None | XRAY | 2.0 | 0.216 | 0.255 | A | 359.0 | 326.0 | 23 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 2yis | CMGC_MAPK14_HUMAN | CMGC | 5.8e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 2YIWA | Q16539 | 5 | 353 | 360.0 | YIW:1353,I46:1354 | Type2,Allosteric | Inactive | DFGout | 15.1257 | 8.2719 | None | -141.89, -172.05 | -138.89, 100.26 | -82.98, 999.0 | 217.28, 137.57 | 999.0, 999.0 | in-in | in | 8.5919 | Saltbr-in | 2.7683 | HRD-in | -71.94, -52.53 | 77.45, -13.14 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | -110.91, 126.0 | APE9-dihe-na | -61.22, 128.26 | APE8-dihe-out | -61.06, -42.06 | APE8-rot-in | 267.54 | APE67-dihe-in | -58.91, -30.27 | -58.86, -25.2 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.076 | None | None | None | XRAY | 2.0 | 0.223 | 0.259 | A | 359.0 | 326.0 | 23 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 2yiw | CMGC_MAPK14_HUMAN | CMGC | 5.8e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3K3JA | Q16539 | 5 | 352 | 360.0 | F4C:361,I46:362 | Type2,Allosteric | Inactive | DFGout | 14.065 | 10.2016 | None | -131.58, -161.61 | -147.02, 101.88 | -61.41, 999.0 | 271.38, 120.65 | 999.0, 999.0 | in-in | in | 9.5761 | Saltbr-in | 3.4443 | HRD-in | -69.65, -53.93 | 78.02, -14.39 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 102.6 | APE9-dihe-na | -77.21, 127.93 | APE8-dihe-out | -43.12, -42.69 | APE8-rot-in | 284.51 | APE67-dihe-in | -68.28, -22.44 | -62.73, -22.61 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.0063 | None | None | None | XRAY | 1.995 | 0.196 | 0.245 | A | 362.0 | 329.0 | 19 | 25 | 12 | 13 | [[24, 308]] | 1.0 | 3k3j | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK14 | MK14_HUMAN | 3HL7A | Q16539 | 6 | 352 | 360.0 | I47:60401,I46:60402 | Type1,Allosteric | Inactive | DFGin | 5.2347 | 13.6446 | BLBplus | -124.2, 170.0 | 68.57, 19.0 | -68.49, 146.41 | 46.64, 88.83 | 77.19, -0.15 | in-in | in | 9.0409 | Saltbr-in | 2.4506 | HRD-in | -63.1, -58.98 | 80.27, -17.67 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 155.78 | APE8-dihe-out | -66.44, -27.56 | APE8-rot-none | 999.0 | APE67-dihe-in | -57.86, -27.57 | -47.26, -39.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.5313 | None | None | None | XRAY | 1.88 | 0.2 | 0.228 | A | 360.0 | 336.0 | 11 | 25 | 14 | 11 | [[24, 308]] | 1.0 | 3hl7 | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3HLLA | Q16539 | 5 | 352 | 360.0 | I45:60401,I46:60402,PO2:60501 | Type1,Allosteric,Allosteric | Inactive | DFGin | 5.053 | 13.5716 | BLBplus | -104.99, 158.54 | 67.03, 24.11 | -71.37, 152.95 | 45.58, 87.31 | 67.6, 1.84 | in-out | in | 9.1864 | Saltbr-out | 3.9688 | HRD-in | -64.7, -58.11 | 82.94, -23.06 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnoo | APE10-dihe-na | 999.0, -18.34 | APE9-dihe-na | -77.72, 94.48 | APE8-dihe-out | -49.19, -31.53 | APE8-rot-none | 999.0 | APE67-dihe-in | -66.1, -25.14 | -64.45, -21.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 16.8147 | APE9-dist-out | 11.6667 | None | None | None | XRAY | 1.95 | 0.219 | 0.254 | A | 360.0 | 337.0 | 11 | 25 | 14 | 11 | [[24, 308]] | 1.0 | 3hll | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3HP2A | Q16539 | 4 | 355 | 360.0 | P36:401,I46:402,I46:403 | Type1,Allosteric,Allosteric | Inactive | DFGin | 10.3229 | 12.0791 | None | -88.89, 117.93 | 0.95, -90.69 | -132.19, 144.91 | 307.84, 89.53 | -100.53, 179.64 | in-in | in | 8.9859 | Saltbr-in | 3.0157 | HRD-in | -62.69, -56.28 | 83.82, -16.84 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, -83.28 | APE9-dihe-na | -69.46, 121.84 | APE8-dihe-out | -57.79, -33.94 | APE8-rot-in | 290.47 | APE67-dihe-in | -56.52, -29.08 | -65.16, -23.99 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 11.8086 | APE9-dist-out | 11.9697 | None | None | None | XRAY | 2.15 | 0.208 | 0.252 | A | 360.0 | 341.0 | 11 | 25 | 14 | 11 | [[24, 308]] | 1.0 | 3hp2 | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3HP5A | Q16539 | 6 | 352 | 360.0 | 52P:401,I46:402,I46:403 | Type1,Allosteric,Allosteric | Inactive | DFGin | 6.4998 | 14.3567 | None | -122.62, 154.65 | 81.43, 43.95 | -64.35, -69.27 | 340.23, 142.83 | -47.68, 999.0 | in-in | in | 8.692 | Saltbr-in | 3.0371 | HRD-in | -62.14, -57.25 | 84.4, -19.04 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnno | APE10-dihe-na | 999.0, -175.23 | APE9-dihe-na | -178.51, 127.74 | APE8-dihe-out | -56.55, -39.12 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.7, -27.21 | -46.07, -42.48 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.3903 | None | None | None | XRAY | 2.3 | 0.217 | 0.262 | A | 360.0 | 330.0 | 17 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 3hp5 | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.9e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 6QDZA | Q16539 | 5 | 352 | 360.0 | I46:401,HYK:402 | Allosteric,Type2 | Inactive | DFGout | 14.9123 | 9.0812 | BBAminus | -134.77, -179.97 | -142.81, 109.12 | -72.73, -21.08 | 264.45, 91.98 | 63.26, 999.0 | in-in | in | 8.4999 | Saltbr-in | 2.7579 | HRD-in | -75.35, -56.13 | 84.01, -14.16 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 120.14 | APE8-dihe-out | -58.44, -38.6 | APE8-rot-in | 261.35 | APE67-dihe-in | -64.54, -27.76 | -61.68, -25.18 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.4049 | None | None | None | XRAY | 1.73 | 0.206 | 0.246 | A | 362.0 | 327.0 | 21 | 25 | 12 | 13 | [[24, 308]] | 1.0 | 6qdz | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 6QE1A | Q16539 | 5 | 352 | 360.0 | I46:401,HYW:402 | Allosteric,Type2 | Inactive | DFGout | 14.5033 | 9.1773 | BBAminus | -141.03, -172.04 | -146.99, 109.37 | -71.94, -17.35 | 270.92, 90.33 | 65.73, 999.0 | in-in | in | 8.7612 | Saltbr-in | 2.6233 | HRD-in | -65.85, -55.55 | 81.72, -12.94 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 126.37 | APE8-dihe-out | -53.58, -40.3 | APE8-rot-in | 269.79 | APE67-dihe-in | -62.76, -30.98 | -60.8, -26.41 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.3191 | None | None | None | XRAY | 1.85 | 0.181 | 0.222 | A | 362.0 | 328.0 | 20 | 25 | 12 | 13 | [[24, 308]] | 1.0 | 6qe1 | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3K3IA | Q16539 | 5 | 352 | 360.0 | JZJ:1,I46:353,I46:2 | Type3,Allosteric,Allosteric | Inactive | DFGout | 13.8744 | 9.8725 | BBAminus | -143.79, -170.14 | -141.75, 114.95 | -78.16, -16.52 | 274.05, 114.76 | 49.78, 999.0 | in-in | in | 9.3253 | Saltbr-in | 2.6305 | HRD-in | -66.69, -52.65 | 76.63, -11.32 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 118.08 | APE9-dihe-na | -84.9, 132.08 | APE8-dihe-out | -50.88, -42.58 | APE8-rot-in | 276.73 | APE67-dihe-in | -63.3, -21.91 | -56.89, -25.41 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.1293 | None | None | None | XRAY | 1.7 | 0.196 | 0.242 | A | 350.0 | 332.0 | 16 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 3k3i | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.3e-85 | 291.3 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 2YISA | Q16539 | 5 | 353 | 360.0 | YIS:1353,I46:1354 | Type2,Allosteric | Inactive | DFGout | 15.833 | 8.5763 | None | -138.39, -175.22 | -139.39, 106.04 | -86.53, 999.0 | 192.46, 60.65 | 999.0, 999.0 | in-in | in | 8.5948 | Saltbr-in | 2.6488 | HRD-in | -65.43, -49.96 | 74.88, -12.76 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | -110.86, 112.45 | APE9-dihe-na | -50.05, 127.69 | APE8-dihe-out | -57.83, -43.06 | APE8-rot-in | 274.36 | APE67-dihe-in | -59.28, -29.93 | -54.84, -31.58 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.1314 | None | None | None | XRAY | 2.0 | 0.216 | 0.255 | A | 359.0 | 326.0 | 23 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 2yis | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.8e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 2YIWA | Q16539 | 5 | 353 | 360.0 | YIW:1353,I46:1354 | Type2,Allosteric | Inactive | DFGout | 15.1257 | 8.2719 | None | -141.89, -172.05 | -138.89, 100.26 | -82.98, 999.0 | 217.28, 137.57 | 999.0, 999.0 | in-in | in | 8.5919 | Saltbr-in | 2.7683 | HRD-in | -71.94, -52.53 | 77.45, -13.14 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | -110.91, 126.0 | APE9-dihe-na | -61.22, 128.26 | APE8-dihe-out | -61.06, -42.06 | APE8-rot-in | 267.54 | APE67-dihe-in | -58.91, -30.27 | -58.86, -25.2 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.076 | None | None | None | XRAY | 2.0 | 0.223 | 0.259 | A | 359.0 | 326.0 | 23 | 25 | 13 | 12 | [[24, 308]] | 1.0 | 2yiw | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 5.8e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| CMGC | MAPK14 | MK14_HUMAN | 3K3JA | Q16539 | 5 | 352 | 360.0 | F4C:361,I46:362 | Type2,Allosteric | Inactive | DFGout | 14.065 | 10.2016 | None | -131.58, -161.61 | -147.02, 101.88 | -61.41, 999.0 | 271.38, 120.65 | 999.0, 999.0 | in-in | in | 9.5761 | Saltbr-in | 3.4443 | HRD-in | -69.65, -53.93 | 78.02, -14.39 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 102.6 | APE9-dihe-na | -77.21, 127.93 | APE8-dihe-out | -43.12, -42.69 | APE8-rot-in | 284.51 | APE67-dihe-in | -68.28, -22.44 | -62.73, -22.61 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.0063 | None | None | None | XRAY | 1.995 | 0.196 | 0.245 | A | 362.0 | 329.0 | 19 | 25 | 12 | 13 | [[24, 308]] | 1.0 | 3k3j | Homo sapiens | CMGC_MAPK14_HUMAN | CMGC | 6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 167 | 168 | 169 | 171 | 173 | 53 | 71 | 75 | 147 | 149 | 148 | 150.0 | 205 | 192 | 187 | 186 | 185 | 184 | 183 | 182 | 181 | 107 | Mitogen-activated protein kinase 14 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|