TKL_TGFBR1 (TGF-beta receptor type-1)

Total number of chains: 59
Active chains: 46
Uniprot: TGFR1_HUMAN
Kinase Domain Residues: 205 - 494
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 59 100.0% AF-P36897-K1A

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PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
5E8UA 2.03 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 502 0 None T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F TGF-beta receptor type-1
4X2NA 1.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 501 0 None None TGF-beta receptor type-1
5E8SA 1.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 498 0 None None TGF-beta receptor type-1
AF-P36897-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 197 - 502 0 None None TGF-beta receptor type-1
AF-P36897-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 197 - 502 0 None None TGF-beta receptor type-1
5E8TA 1.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 499 0 None T204D TGF-beta receptor type-1
1IASA 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1
1IASB 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 501 0 None None TGF-beta receptor type-1
1IASC 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1
1IASD 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1
1IASE 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1
5E8XA 1.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii STU Type1 200 - 503 0 None T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F TGF-beta receptor type-1
5E90A 2.05 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5L4 Type1 200 - 499 0 None T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F TGF-beta receptor type-1
5USQA 2.55 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 8LY Type1 200 - 498 0 None None TGF-beta receptor type-1
5FRIA 2.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZUQ Type1 200 - 498 0 None None TGF-beta receptor type-1
9F6XA 2.68 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii A1IAZ Type1 200 - 500 0 None None TGF-beta receptor type-1
4X0MA 1.68 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WA Type1 200 - 501 0 None None TGF-beta receptor type-1
4X2FA 1.49 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WJ Type1 200 - 501 0 None None TGF-beta receptor type-1
4X2GA 1.51 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WK Type1 200 - 501 0 None None TGF-beta receptor type-1
2WOTA 1.85 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZZG Type1 200 - 500 0 None None TGF-beta receptor type-1
2WOUA 2.3 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZZF Type1 200 - 496 0 None None TGF-beta receptor type-1
8YHLA 1.47 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii A1D6I Type1 200 - 501 0 None None TGF-beta receptor type-1
5E8WA 1.86 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii STU Type1 200 - 501 0 None T204D TGF-beta receptor type-1
5E8ZA 1.51 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5L4 Type1 200 - 499 0 None T204D TGF-beta receptor type-1
5QIKA 1.58 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii J2M Type1 200 - 499 0 None T204D TGF-beta receptor type-1
5QILA 1.98 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii J2V Type1 200 - 499 0 None T204D TGF-beta receptor type-1
5QTZA 1.83 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii QMY Type1 200 - 499 0 None T204D TGF-beta receptor type-1
5QU0A 1.67 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii QMV Type1 200 - 502 0 None T204D TGF-beta receptor type-1
2X7OA 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1 171 - 500 0 None None TGF-beta receptor type-1
3FAAA 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1
3FAAB 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 501 0 None None TGF-beta receptor type-1
3FAAD 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1
3FAAE 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1
8YHFA 1.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii A1D6I Type1 201 - 498 0 None None TGF-beta receptor type-1
4X2JA 1.69 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WN Type1.5_Back 200 - 501 0 None None TGF-beta receptor type-1
4X2KA 1.69 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WO Type1.5_Back 200 - 501 0 None None TGF-beta receptor type-1
5QIMA 1.75 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii J2Y Type1.5_Back 200 - 501 0 None None TGF-beta receptor type-1
6B8YA 1.65 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii D0A Type1.5_Back 200 - 502 0 None T204D TGF-beta receptor type-1
2X7OC 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
2X7OD 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
2X7OE 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
3KCFA 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
3KCFB 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 501 0 None None TGF-beta receptor type-1
3KCFC 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
3KCFD 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
3KCFE 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1
1B6CB 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1
1B6CD 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1
1B6CF 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1
1B6CH 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1
1RW8A 2.4 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_iioi 580 Type1 200 - 500 0 None None TGF-beta receptor type-1
1PY5A 2.3 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_iioi PY1 Type1 200 - 500 0 None None TGF-beta receptor type-1
2X7OB 3.7 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1 171 - 500 0 None None TGF-beta receptor type-1
3FAAC 3.35 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiio APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1
1VJYA 2.0 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii 460 Type1 201 - 503 0 None None TGF-beta receptor type-1
3GXLA 1.8 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii QIG Type1 201 - 498 0 None None TGF-beta receptor type-1
3HMMA 1.7 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_nnni 855 Type1 201 - 498 0 None None TGF-beta receptor type-1
9J9DA 1.337 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii A1L30 Type1 202 - 502 0 None None TGF-beta receptor type-1
3TZMA 1.7 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii 085 Type1 200 - 496 0 None None TGF-beta receptor type-1

TKL_TGFBR1 (TGF-beta receptor type-1)

Total number of chains: 59
Active chains: 46
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 59 100.0% AF-P36897-K1A

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TGFR1_HUMAN 5E8UA 2.03 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 502 0 None T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 4X2NA 1.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5E8SA 1.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 498 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN AF-P36897-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 197 - 502 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN AF-P36897-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 197 - 502 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5E8TA 1.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 200 - 499 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1IASA 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1IASB 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1IASC 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1IASD 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1IASE 2.9 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5E8XA 1.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii STU Type1 200 - 503 0 None T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5E90A 2.05 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5L4 Type1 200 - 499 0 None T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5USQA 2.55 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 8LY Type1 200 - 498 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5FRIA 2.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZUQ Type1 200 - 498 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 9F6XA 2.68 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii A1IAZ Type1 200 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 4X0MA 1.68 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WA Type1 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 4X2FA 1.49 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WJ Type1 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 4X2GA 1.51 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WK Type1 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2WOTA 1.85 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZZG Type1 200 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2WOUA 2.3 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZZF Type1 200 - 496 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 8YHLA 1.47 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii A1D6I Type1 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5E8WA 1.86 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii STU Type1 200 - 501 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5E8ZA 1.51 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 5L4 Type1 200 - 499 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5QIKA 1.58 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii J2M Type1 200 - 499 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5QILA 1.98 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii J2V Type1 200 - 499 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5QTZA 1.83 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii QMY Type1 200 - 499 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5QU0A 1.67 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii QMV Type1 200 - 502 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2X7OA 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3FAAA 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3FAAB 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3FAAD 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3FAAE 3.35 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 8YHFA 1.4 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii A1D6I Type1 201 - 498 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 4X2JA 1.69 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WN Type1.5_Back 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 4X2KA 1.69 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 3WO Type1.5_Back 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 5QIMA 1.75 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii J2Y Type1.5_Back 200 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 6B8YA 1.65 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii D0A Type1.5_Back 200 - 502 0 None T204D TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2X7OC 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2X7OD 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2X7OE 3.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3KCFA 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3KCFB 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 501 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3KCFC 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3KCFD 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3KCFE 2.8 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii JZO Type1.5_Back 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1B6CB 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1B6CD 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1B6CF 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1B6CH 2.6 Inactive DFGin‑BLAminus in-out in-out nonTYR APEdihe_aaiii APEdist_iooi No_ligand No_ligand 175 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1RW8A 2.4 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_iioi 580 Type1 200 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1PY5A 2.3 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiii APEdist_iioi PY1 Type1 200 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 2X7OB 3.7 Inactive DFGin‑BLAminus in-out in-in nonTYR APEdihe_aaiii APEdist_iiii ZOP Type1 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3FAAC 3.35 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaiio APEdist_iiii 55F Type1 171 - 500 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 1VJYA 2.0 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii 460 Type1 201 - 503 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3GXLA 1.8 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii QIG Type1 201 - 498 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3HMMA 1.7 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_nnni 855 Type1 201 - 498 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 9J9DA 1.337 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii A1L30 Type1 202 - 502 0 None None TGF-beta receptor type-1 Homo sapiens
TGFR1_HUMAN 3TZMA 1.7 None DFGin‑BLAminus in-in in-none nonTYR APEdihe_aaiii APEdist_niii 085 Type1 200 - 496 0 None None TGF-beta receptor type-1 Homo sapiens

TKL_TGFBR1 (TGF-beta receptor type-1)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism