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| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 5E8UA | 200 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 7.25 | 14.239 | BLAminus | -134.62, -172.63 | 56.13, 81.95 | -101.29, 16.47 | 292.48, 105.22 | -57.91, -29.22 | in-in | in | 7.887 | Saltbr-in | 2.946 | HRD-in | -72.05, -48.87 | 69.51, 7.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.969 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -102.25, 153.37 | APE9-dihe-na | 113.03, -170.78 | APE8-dihe-in | -89.61, 116.01 | APE8-rot-in | 305.95 | APE67-dihe-in | -56.91, -33.28 | -47.65, -46.01 | APE12-dist-in | 13.141 | APE11-dist-in | 12.522 | APE10-dist-in | 6.48 | APE9-dist-in | 3.958 | T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F | None | None | XRAY | 2.03 | 0.181 | 0.223 | A | 307 | 303 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8u | TKL_TGFBR1_HUMAN | TKL | 2.3e-85 | 292.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 4X2NA | 200 | 501 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.15 | 13.2 | BLAminus | -127.58, -171.48 | 51.56, 55.64 | -81.72, 7.99 | 306.47, 9.87 | -57.69, -30.68 | in-in | in | 7.746 | Saltbr-in | 3.137 | HRD-in | -73.45, -50.82 | 74.64, -6.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.988 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.64, 175.91 | APE9-dihe-na | 96.93, 176.28 | APE8-dihe-in | -81.13, 124.7 | APE8-rot-in | 305.67 | APE67-dihe-in | -55.99, -35.77 | -56.51, -42.26 | APE12-dist-in | 11.788 | APE11-dist-in | 11.876 | APE10-dist-in | 6.194 | APE9-dist-in | 3.712 | None | None | None | XRAY | 1.8 | 0.163 | 0.201 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2n | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5E8SA | 200 | 498 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.227 | 13.345 | BLAminus | -130.71, -170.38 | 50.26, 56.29 | -81.51, 7.19 | 302.58, 10.42 | -59.69, -25.71 | in-in | in | 7.75 | Saltbr-in | 3.098 | HRD-in | -75.18, -50.46 | 75.3, -6.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.942 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.12, 158.63 | APE9-dihe-na | 109.47, 177.89 | APE8-dihe-in | -83.28, 125.6 | APE8-rot-in | 301.61 | APE67-dihe-in | -57.6, -32.67 | -59.04, -39.92 | APE12-dist-in | 13.384 | APE11-dist-in | 12.417 | APE10-dist-in | 6.303 | APE9-dist-in | 3.677 | None | None | None | XRAY | 1.45 | 0.172 | 0.188 | A | 306 | 299 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8s | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| AF-P36897-K1A | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.097 | 12.697 | BLAminus | -127.47, -177.39 | 59.98, 50.67 | -75.64, 9.99 | 303.25, 0.83 | -67.03, -14.65 | in-in | in | 7.75 | Saltbr-in | 2.631 | HRD-in | -79.18, -43.89 | 66.79, -8.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.015 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.74, 159.13 | APE9-dihe-na | 99.19, -175.01 | APE8-dihe-in | -81.52, 117.2 | APE8-rot-in | 304.32 | APE67-dihe-in | -58.11, -28.29 | -49.21, -42.7 | APE12-dist-in | 13.034 | APE11-dist-in | 12.476 | APE10-dist-in | 6.348 | APE9-dist-in | 3.781 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306 | 306 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | AF-P36897-K1 | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| AF-P36897-K3A | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.388 | 12.882 | BLAminus | -127.89, -179.35 | 58.97, 55.86 | -76.18, 6.96 | 301.47, 0.09 | -63.41, -19.74 | in-in | in | 8.095 | Saltbr-in | 2.675 | HRD-in | -77.05, -40.27 | 65.4, -16.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.85 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -117.36, 158.96 | APE9-dihe-na | 107.71, -175.1 | APE8-dihe-in | -94.3, 114.61 | APE8-rot-in | 303.53 | APE67-dihe-in | -61.67, -24.01 | -41.02, -46.98 | APE12-dist-in | 11.212 | APE11-dist-in | 11.814 | APE10-dist-in | 5.925 | APE9-dist-in | 3.7 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306 | 306 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | AF-P36897-K3 | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5E8TA | 200 | 499 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.13 | 13.117 | BLAminus | -129.7, -170.36 | 54.3, 58.56 | -85.47, 9.03 | 309.14, 5.15 | -56.74, -27.28 | in-in | in | 7.84 | Saltbr-in | 2.94 | HRD-in | -72.25, -51.54 | 76.95, -4.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.969 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -78.56, -31.05 | APE9-dihe-na | -81.1, -159.38 | APE8-dihe-in | -84.33, 122.67 | APE8-rot-in | 299.0 | APE67-dihe-in | -55.04, -35.69 | -53.58, -44.7 | APE12-dist-in | 13.067 | APE11-dist-in | 12.282 | APE10-dist-in | 6.237 | APE9-dist-in | 3.791 | T204D | None | None | XRAY | 1.7 | 0.17 | 0.19 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8t | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1IASA | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.721 | 12.723 | BLAminus | -151.41, 164.95 | 71.98, 88.97 | -106.86, 22.49 | 311.89, 1.41 | -60.78, -26.26 | in-in | in | 8.24 | Saltbr-in | 2.79 | HRD-in | -63.37, -49.76 | 71.64, 8.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.974 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.42, 172.85 | APE9-dihe-na | 97.41, 166.83 | APE8-dihe-in | -62.29, 121.18 | APE8-rot-in | 307.67 | APE67-dihe-in | -45.67, -30.78 | -49.33, -54.47 | APE12-dist-in | 11.452 | APE11-dist-in | 11.629 | APE10-dist-in | 6.172 | APE9-dist-in | 4.131 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | A | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1IASB | 171 | 501 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.652 | 12.707 | BLAminus | -150.79, 165.66 | 71.53, 88.91 | -106.55, 22.01 | 312.14, 1.23 | -60.97, -25.51 | in-in | in | 8.241 | Saltbr-in | 2.799 | HRD-in | -64.38, -48.85 | 71.21, 7.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.005 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.79, 173.68 | APE9-dihe-na | 99.72, 167.49 | APE8-dihe-in | -63.26, 121.22 | APE8-rot-in | 308.35 | APE67-dihe-in | -44.49, -32.42 | -49.46, -55.33 | APE12-dist-in | 10.321 | APE11-dist-in | 11.628 | APE10-dist-in | 6.241 | APE9-dist-in | 4.05 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 1ias | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1IASC | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.59 | 12.711 | BLAminus | -150.31, 164.7 | 71.4, 89.07 | -106.94, 23.22 | 312.6, 1.77 | -61.3, -25.67 | in-in | in | 8.197 | Saltbr-in | 2.799 | HRD-in | -63.0, -50.37 | 71.83, 9.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.013 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.75, 170.21 | APE9-dihe-na | 100.55, 167.25 | APE8-dihe-in | -63.65, 121.53 | APE8-rot-in | 308.64 | APE67-dihe-in | -44.33, -30.7 | -49.24, -56.44 | APE12-dist-in | 11.349 | APE11-dist-in | 11.759 | APE10-dist-in | 6.222 | APE9-dist-in | 4.15 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1IASD | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.594 | 12.743 | BLAminus | -152.15, 165.79 | 70.83, 87.83 | -105.27, 21.55 | 312.92, 0.98 | -60.27, -25.54 | in-in | in | 8.189 | Saltbr-in | 2.775 | HRD-in | -64.51, -48.18 | 71.39, 8.63 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.993 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.69, 169.96 | APE9-dihe-na | 98.27, 166.26 | APE8-dihe-in | -61.5, 120.34 | APE8-rot-in | 308.37 | APE67-dihe-in | -44.16, -31.51 | -48.36, -56.13 | APE12-dist-in | 10.732 | APE11-dist-in | 11.784 | APE10-dist-in | 6.18 | APE9-dist-in | 4.04 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1IASE | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.685 | 12.738 | BLAminus | -151.39, 165.15 | 70.82, 89.42 | -106.94, 21.97 | 311.98, 2.05 | -61.66, -24.41 | in-in | in | 8.226 | Saltbr-in | 2.803 | HRD-in | -61.95, -50.33 | 72.19, 7.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.008 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.31, 173.9 | APE9-dihe-na | 98.05, 167.39 | APE8-dihe-in | -64.1, 121.3 | APE8-rot-in | 308.19 | APE67-dihe-in | -45.93, -31.42 | -49.14, -54.62 | APE12-dist-in | 11.636 | APE11-dist-in | 11.505 | APE10-dist-in | 6.149 | APE9-dist-in | 4.002 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5E8XA | 200 | 503 | 503.0 | STU:601 | Type1 | Active | DFGin | 7.401 | 13.771 | BLAminus | -132.02, 177.79 | 68.95, 84.86 | -101.89, 20.89 | 298.69, 99.78 | -60.9, -22.78 | in-in | in | 7.646 | Saltbr-in | 3.316 | HRD-in | -78.83, -50.32 | 78.23, -2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.2, 171.93 | APE9-dihe-na | 104.3, 177.57 | APE8-dihe-in | -80.96, 119.4 | APE8-rot-in | 304.53 | APE67-dihe-in | -55.33, -34.35 | -53.44, -41.29 | APE12-dist-in | 11.709 | APE11-dist-in | 11.927 | APE10-dist-in | 6.258 | APE9-dist-in | 3.946 | T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F | None | None | XRAY | 1.45 | 0.191 | 0.21 | A | 307 | 304 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8x | TKL_TGFBR1_HUMAN | TKL | 2.3e-85 | 292.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5E90A | 200 | 499 | 503.0 | 5L4:60601 | Type1 | Active | DFGin | 7.033 | 13.968 | BLAminus | -132.44, -170.95 | 59.07, 73.91 | -100.08, 11.67 | 293.12, 109.78 | -58.9, -27.5 | in-in | in | 7.732 | Saltbr-in | 2.865 | HRD-in | -62.69, -55.46 | 77.29, -2.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.872 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.74, -31.43 | APE9-dihe-na | -82.55, -164.68 | APE8-dihe-in | -74.68, 122.19 | APE8-rot-in | 303.81 | APE67-dihe-in | -54.67, -36.7 | -55.17, -42.7 | APE12-dist-in | 12.594 | APE11-dist-in | 11.9 | APE10-dist-in | 5.887 | APE9-dist-in | 3.841 | T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F | None | None | XRAY | 2.05 | 0.178 | 0.218 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e90 | TKL_TGFBR1_HUMAN | TKL | 2.3e-85 | 292.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5USQA | 200 | 498 | 503.0 | 8LY:500 | Type1 | Active | DFGin | 6.294 | 13.451 | BLAminus | -128.65, -178.48 | 58.74, 56.74 | -84.73, 2.3 | 308.58, 3.38 | -59.48, -22.95 | in-in | in | 7.752 | Saltbr-in | 3.191 | HRD-in | -74.99, -53.41 | 77.78, -10.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.92 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.34, -32.16 | APE9-dihe-na | -75.45, -164.79 | APE8-dihe-in | -80.15, 126.14 | APE8-rot-in | 305.26 | APE67-dihe-in | -52.52, -34.72 | -59.83, -43.81 | APE12-dist-in | 13.024 | APE11-dist-in | 12.008 | APE10-dist-in | 6.158 | APE9-dist-in | 3.557 | None | None | None | XRAY | 2.55 | 0.182 | 0.231 | A | 299 | 299 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5usq | TKL_TGFBR1_HUMAN | TKL | 3e-85 | 291.9 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5FRIA | 200 | 498 | 503.0 | ZUQ:61501 | Type1 | Active | DFGin | 5.986 | 12.349 | BLAminus | -129.47, -173.22 | 60.99, 71.38 | -101.21, 12.39 | 307.22, 5.28 | -67.89, -22.52 | in-in | in | 7.758 | Saltbr-in | 2.857 | HRD-in | -78.14, -52.35 | 77.86, -1.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.926 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.89, -25.51 | APE9-dihe-na | -92.81, -153.48 | APE8-dihe-in | -86.34, 123.11 | APE8-rot-in | 303.21 | APE67-dihe-in | -53.0, -34.54 | -57.92, -43.35 | APE12-dist-in | 12.836 | APE11-dist-in | 11.987 | APE10-dist-in | 6.05 | APE9-dist-in | 3.945 | None | None | None | XRAY | 2.0 | 0.164 | 0.193 | A | 301 | 299 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5fri | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 9F6XA | 200 | 500 | 503.0 | A1IAZ:60401 | Type1 | Active | DFGin | 6.135 | 13.376 | BLAminus | -110.91, -175.59 | 63.64, 55.87 | -85.09, 3.96 | 315.03, 1.12 | -62.09, -27.8 | in-in | in | 8.172 | Saltbr-in | 2.73 | HRD-in | -72.7, -49.45 | 76.37, -0.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.008 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -96.61, -34.29 | APE9-dihe-na | -78.73, -165.12 | APE8-dihe-in | -74.89, 126.22 | APE8-rot-in | 295.38 | APE67-dihe-in | -52.17, -40.21 | -62.21, -41.17 | APE12-dist-in | 13.477 | APE11-dist-in | 12.232 | APE10-dist-in | 6.103 | APE9-dist-in | 3.604 | None | None | None | XRAY | 2.68 | 0.214 | 0.248 | A | 303 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 9f6x | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 4X0MA | 200 | 501 | 503.0 | 3WA:60601 | Type1 | Active | DFGin | 6.253 | 12.884 | BLAminus | -128.27, -179.8 | 55.38, 57.51 | -85.94, 12.49 | 298.0, 10.23 | -63.66, -28.1 | in-in | in | 7.343 | Saltbr-in | 3.153 | HRD-in | -62.49, -53.22 | 74.03, -11.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.008 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.83, 167.91 | APE9-dihe-na | 99.86, -179.25 | APE8-dihe-in | -77.31, 123.46 | APE8-rot-in | 305.82 | APE67-dihe-in | -54.73, -39.98 | -54.51, -42.68 | APE12-dist-in | 11.689 | APE11-dist-in | 11.872 | APE10-dist-in | 6.21 | APE9-dist-in | 3.823 | None | None | None | XRAY | 1.68 | 0.21 | 0.239 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x0m | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 4X2FA | 200 | 501 | 503.0 | 3WJ:60601 | Type1 | Active | DFGin | 6.198 | 12.989 | BLAminus | -129.57, -169.63 | 49.35, 56.72 | -81.87, 7.01 | 303.23, 9.49 | -60.29, -24.32 | in-in | in | 7.557 | Saltbr-in | 2.939 | HRD-in | -74.24, -48.95 | 76.58, -5.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.03, 171.99 | APE9-dihe-na | 101.85, 179.14 | APE8-dihe-in | -82.12, 123.51 | APE8-rot-in | 300.96 | APE67-dihe-in | -58.79, -32.2 | -58.45, -40.31 | APE12-dist-in | 11.805 | APE11-dist-in | 11.906 | APE10-dist-in | 6.197 | APE9-dist-in | 3.807 | None | None | None | XRAY | 1.49 | 0.165 | 0.191 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2f | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 4X2GA | 200 | 501 | 503.0 | 3WK:60601 | Type1 | Active | DFGin | 6.161 | 12.995 | BLAminus | -126.43, -164.75 | 48.26, 54.97 | -83.24, 5.58 | 306.41, 9.37 | -59.31, -23.57 | in-in | in | 7.56 | Saltbr-in | 3.063 | HRD-in | -73.4, -50.72 | 76.5, -5.82 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.905 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.4, 173.04 | APE9-dihe-na | 101.04, 176.44 | APE8-dihe-in | -79.69, 125.01 | APE8-rot-in | 303.47 | APE67-dihe-in | -59.43, -31.39 | -61.05, -38.4 | APE12-dist-in | 11.852 | APE11-dist-in | 11.925 | APE10-dist-in | 6.221 | APE9-dist-in | 3.793 | None | None | None | XRAY | 1.51 | 0.166 | 0.185 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2g | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2WOTA | 200 | 500 | 503.0 | ZZG:61500 | Type1 | Active | DFGin | 6.1 | 13.031 | BLAminus | -130.27, -169.46 | 60.16, 61.47 | -92.46, 8.2 | 303.12, 6.85 | -64.56, -24.36 | in-in | in | 7.663 | Saltbr-in | 3.074 | HRD-in | -80.51, -53.82 | 76.92, 0.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.95 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -90.42, -22.62 | APE9-dihe-na | -94.01, -157.41 | APE8-dihe-in | -80.51, 121.5 | APE8-rot-in | 307.33 | APE67-dihe-in | -52.87, -38.64 | -55.17, -43.39 | APE12-dist-in | 13.131 | APE11-dist-in | 12.287 | APE10-dist-in | 6.338 | APE9-dist-in | 3.77 | None | None | None | XRAY | 1.85 | 0.181 | 0.221 | A | 306 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2wot | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2WOUA | 200 | 496 | 503.0 | ZZF:61500 | Type1 | Active | DFGin | 6.124 | 13.039 | BLAminus | -133.49, -169.53 | 51.05, 62.4 | -92.04, 13.34 | 298.31, 178.69 | -62.77, -27.98 | in-in | in | 7.586 | Saltbr-in | 2.752 | HRD-in | -65.52, -56.03 | 81.95, -3.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.039 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.77, -22.31 | APE9-dihe-na | -79.77, -172.15 | APE8-dihe-in | -73.94, 125.36 | APE8-rot-in | 306.35 | APE67-dihe-in | -52.11, -29.79 | -56.64, -45.19 | APE12-dist-in | 13.078 | APE11-dist-in | 11.935 | APE10-dist-in | 6.041 | APE9-dist-in | 3.629 | None | None | None | XRAY | 2.3 | 0.229 | 0.302 | A | 306 | 297 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2wou | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 8YHLA | 200 | 501 | 503.0 | A1D6I:60601 | Type1 | Active | DFGin | 6.021 | 13.048 | BLAminus | -124.89, -169.46 | 42.91, 75.25 | -91.67, 10.82 | 300.67, 10.41 | -67.27, -22.16 | in-in | in | 7.699 | Saltbr-in | 2.965 | HRD-in | -79.41, -52.59 | 75.07, -1.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.932 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -72.3, 155.92 | APE9-dihe-na | 107.61, -172.07 | APE8-dihe-in | -88.21, 123.34 | APE8-rot-in | 304.18 | APE67-dihe-in | -56.11, -38.82 | -61.94, -38.97 | APE12-dist-in | 13.343 | APE11-dist-in | 12.518 | APE10-dist-in | 6.314 | APE9-dist-in | 3.816 | None | None | None | XRAY | 1.47 | 0.165 | 0.193 | A | 306 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 8yhl | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5E8WA | 200 | 501 | 503.0 | STU:60601 | Type1 | Active | DFGin | 6.216 | 12.991 | BLAminus | -115.91, -168.56 | 48.03, 66.8 | -87.81, 6.99 | 303.66, 6.47 | -53.89, -34.67 | in-in | in | 7.561 | Saltbr-in | 2.815 | HRD-in | -71.33, -51.46 | 73.08, -1.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.992 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -81.36, -32.83 | APE9-dihe-na | -81.66, -157.24 | APE8-dihe-in | -82.54, 122.58 | APE8-rot-in | 299.35 | APE67-dihe-in | -53.78, -37.25 | -53.32, -45.52 | APE12-dist-in | 13.054 | APE11-dist-in | 12.418 | APE10-dist-in | 6.3 | APE9-dist-in | 3.738 | T204D | None | None | XRAY | 1.86 | 0.168 | 0.186 | A | 307 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8w | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5E8ZA | 200 | 499 | 503.0 | 5L4:60601 | Type1 | Active | DFGin | 5.938 | 12.742 | BLAminus | -131.72, -172.47 | 57.21, 65.07 | -93.0, 9.47 | 305.33, 7.41 | -62.65, -21.83 | in-in | in | 7.87 | Saltbr-in | 2.94 | HRD-in | -73.84, -51.69 | 76.4, -3.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.915 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -86.19, -27.35 | APE9-dihe-na | -88.81, -157.37 | APE8-dihe-in | -81.17, 121.36 | APE8-rot-in | 303.09 | APE67-dihe-in | -55.51, -33.19 | -54.0, -44.23 | APE12-dist-in | 13.117 | APE11-dist-in | 12.181 | APE10-dist-in | 6.139 | APE9-dist-in | 3.775 | T204D | None | None | XRAY | 1.51 | 0.183 | 0.207 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8z | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5QIKA | 200 | 499 | 503.0 | J2M:60601 | Type1 | Active | DFGin | 6.134 | 12.822 | BLAminus | -129.19, -176.86 | 54.93, 67.17 | -89.45, 12.6 | 307.08, 5.45 | -57.51, -28.59 | in-in | in | 8.037 | Saltbr-in | 2.853 | HRD-in | -74.13, -49.19 | 76.47, -1.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -82.77, -28.33 | APE9-dihe-na | -83.38, -158.15 | APE8-dihe-in | -83.03, 121.9 | APE8-rot-in | 297.41 | APE67-dihe-in | -57.88, -31.82 | -55.17, -43.49 | APE12-dist-in | 13.224 | APE11-dist-in | 12.41 | APE10-dist-in | 6.393 | APE9-dist-in | 3.835 | T204D | None | None | XRAY | 1.58 | 0.166 | 0.19 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qik | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5QILA | 200 | 499 | 503.0 | J2V:60601 | Type1 | Active | DFGin | 6.123 | 12.893 | BLAminus | -133.55, -173.28 | 54.13, 68.92 | -94.29, 10.19 | 306.15, 4.81 | -59.56, -26.12 | in-in | in | 7.782 | Saltbr-in | 3.012 | HRD-in | -72.26, -48.55 | 71.72, 0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.977 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.42, -32.81 | APE9-dihe-na | -79.5, -152.05 | APE8-dihe-in | -86.88, 119.67 | APE8-rot-in | 305.45 | APE67-dihe-in | -55.45, -33.57 | -52.15, -44.93 | APE12-dist-in | 12.839 | APE11-dist-in | 12.277 | APE10-dist-in | 6.153 | APE9-dist-in | 3.792 | T204D | None | None | XRAY | 1.98 | 0.171 | 0.21 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qil | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5QTZA | 200 | 499 | 503.0 | QMY:60601 | Type1 | Active | DFGin | 6.173 | 13.35 | BLAminus | -138.39, -173.58 | 55.38, 56.92 | -82.72, 7.96 | 301.94, 5.0 | -56.41, -28.87 | in-in | in | 8.148 | Saltbr-in | 2.898 | HRD-in | -70.33, -51.13 | 74.03, -4.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.025 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -86.52, -26.25 | APE9-dihe-na | -81.63, -163.74 | APE8-dihe-in | -76.85, 122.93 | APE8-rot-in | 300.9 | APE67-dihe-in | -53.47, -35.21 | -52.57, -45.07 | APE12-dist-in | 12.983 | APE11-dist-in | 12.176 | APE10-dist-in | 6.168 | APE9-dist-in | 3.658 | T204D | None | None | XRAY | 1.83 | 0.171 | 0.2 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qtz | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5QU0A | 200 | 502 | 503.0 | QMV:60601 | Type1 | Active | DFGin | 6.226 | 13.493 | BLAminus | -131.41, -169.26 | 50.76, 57.03 | -82.09, 5.13 | 306.24, 2.05 | -53.78, -29.06 | in-in | in | 7.858 | Saltbr-in | 2.924 | HRD-in | -72.09, -52.96 | 76.9, -5.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.961 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -85.59, 161.83 | APE9-dihe-na | 106.22, 171.28 | APE8-dihe-in | -76.79, 124.94 | APE8-rot-in | 300.79 | APE67-dihe-in | -53.51, -36.09 | -55.88, -43.03 | APE12-dist-in | 13.281 | APE11-dist-in | 12.425 | APE10-dist-in | 6.254 | APE9-dist-in | 3.655 | T204D | None | None | XRAY | 1.67 | 0.178 | 0.206 | A | 307 | 303 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qu0 | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2X7OA | 171 | 500 | 503.0 | ZOP:600 | Type1 | Active | DFGin | 6.832 | 13.774 | BLAminus | -128.16, 169.92 | 59.52, 88.44 | -108.37, 28.14 | 289.28, 149.08 | -69.29, -30.37 | in-in | in | 8.088 | Saltbr-in | 3.532 | HRD-in | -65.4, -40.58 | 69.2, -25.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.057 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.88, 149.39 | APE9-dihe-na | 96.51, -171.18 | APE8-dihe-in | -74.29, 131.0 | APE8-rot-in | 315.1 | APE67-dihe-in | -64.94, -34.48 | -61.98, -32.57 | APE12-dist-in | 11.82 | APE11-dist-in | 11.797 | APE10-dist-in | 5.973 | APE9-dist-in | 4.739 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | A | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3FAAA | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 5.904 | 13.047 | BLAminus | -165.74, 163.41 | 74.29, 54.12 | -79.67, 24.05 | 317.06, 176.62 | -56.68, -51.28 | in-in | in | 8.001 | Saltbr-in | 2.936 | HRD-in | -45.11, -27.8 | 52.25, 11.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.111 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.43, -171.19 | APE9-dihe-na | 80.03, 171.79 | APE8-dihe-in | -67.98, 121.11 | APE8-rot-in | 302.91 | APE67-dihe-in | -99.71, -73.49 | -46.09, -5.99 | APE12-dist-in | 11.624 | APE11-dist-in | 11.967 | APE10-dist-in | 6.015 | APE9-dist-in | 4.061 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | A | 342 | 328 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3FAAB | 171 | 501 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.017 | 13.306 | BLAminus | -136.45, -176.24 | 60.04, 54.86 | -81.47, 12.98 | 307.95, 5.19 | -52.57, -45.29 | in-in | in | 8.1 | Saltbr-in | 3.037 | HRD-in | -75.89, -39.75 | 60.74, 14.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.115 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.32, 175.24 | APE9-dihe-na | 101.52, 166.7 | APE8-dihe-in | -70.87, 127.35 | APE8-rot-in | 315.28 | APE67-dihe-in | -36.34, -44.33 | -43.95, -69.54 | APE12-dist-in | 11.94 | APE11-dist-in | 12.0 | APE10-dist-in | 6.373 | APE9-dist-in | 4.084 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3FAAD | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.26 | 13.168 | BLAminus | -151.5, 176.63 | 62.94, 64.2 | -90.99, 26.98 | 302.19, 4.38 | -66.56, -19.34 | in-in | in | 7.809 | Saltbr-in | 2.745 | HRD-in | -63.44, -55.82 | 78.14, 1.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.86, 174.28 | APE9-dihe-na | 87.09, 173.14 | APE8-dihe-in | -66.87, 116.28 | APE8-rot-in | 325.42 | APE67-dihe-in | -60.47, -38.15 | -48.63, -36.35 | APE12-dist-in | 11.714 | APE11-dist-in | 11.894 | APE10-dist-in | 6.37 | APE9-dist-in | 4.229 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3FAAE | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.355 | 13.366 | BLAminus | -131.48, -168.05 | 37.37, 86.28 | -107.7, 26.02 | 296.92, 176.17 | -65.92, -19.56 | in-in | in | 7.781 | Saltbr-in | 3.095 | HRD-in | -66.77, -57.93 | 79.95, 12.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.85 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.13, 169.87 | APE9-dihe-na | 90.72, 172.5 | APE8-dihe-in | -64.72, 129.04 | APE8-rot-in | 310.98 | APE67-dihe-in | -56.46, -40.64 | -59.57, -42.14 | APE12-dist-in | 11.99 | APE11-dist-in | 12.056 | APE10-dist-in | 6.57 | APE9-dist-in | 3.982 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 8YHFA | 201 | 498 | 503.0 | A1D6I:601 | Type1 | Active | DFGin | 6.037 | 13.152 | BLAminus | -127.63, -168.18 | 39.33, 73.78 | -89.91, 13.29 | 302.44, 7.93 | -62.86, -27.56 | in-in | in | 7.799 | Saltbr-in | 3.029 | HRD-in | -79.9, -54.99 | 79.42, -3.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.954 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.79, -23.11 | APE9-dihe-na | -96.35, -152.57 | APE8-dihe-in | -84.18, 124.71 | APE8-rot-in | 302.64 | APE67-dihe-in | -56.72, -32.39 | -61.45, -41.11 | APE12-dist-in | 13.178 | APE11-dist-in | 12.22 | APE10-dist-in | 6.218 | APE9-dist-in | 3.834 | None | None | None | XRAY | 1.4 | 0.167 | 0.192 | A | 343 | 298 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 8yhf | TKL_TGFBR1_HUMAN | TKL | 5e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 4X2JA | 200 | 501 | 503.0 | 3WN:60601 | Type1.5_Back | Active | DFGin | 6.245 | 13.082 | BLAminus | -129.47, -176.48 | 54.06, 62.42 | -89.1, 7.12 | 300.54, 6.95 | -58.75, -23.34 | in-in | in | 7.595 | Saltbr-in | 2.782 | HRD-in | -70.93, -49.34 | 73.15, -2.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.918 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.13, 172.46 | APE9-dihe-na | 95.45, -178.89 | APE8-dihe-in | -79.7, 121.22 | APE8-rot-in | 304.99 | APE67-dihe-in | -57.38, -35.27 | -55.84, -42.14 | APE12-dist-in | 11.79 | APE11-dist-in | 11.898 | APE10-dist-in | 6.199 | APE9-dist-in | 3.764 | None | None | None | XRAY | 1.69 | 0.167 | 0.184 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2j | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 4X2KA | 200 | 501 | 503.0 | 3WO:60601 | Type1.5_Back | Active | DFGin | 6.245 | 13.082 | BLAminus | -129.47, -176.48 | 54.06, 62.42 | -89.1, 7.12 | 300.54, 6.95 | -58.75, -23.34 | in-in | in | 7.595 | Saltbr-in | 2.782 | HRD-in | -70.93, -49.34 | 73.15, -2.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.918 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.13, 172.46 | APE9-dihe-na | 95.45, -178.89 | APE8-dihe-in | -79.7, 121.22 | APE8-rot-in | 304.99 | APE67-dihe-in | -57.38, -35.27 | -55.84, -42.14 | APE12-dist-in | 11.79 | APE11-dist-in | 11.898 | APE10-dist-in | 6.199 | APE9-dist-in | 3.764 | None | None | None | XRAY | 1.69 | 0.167 | 0.184 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2k | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 5QIMA | 200 | 501 | 503.0 | J2Y:60601 | Type1.5_Back | Active | DFGin | 6.324 | 13.322 | BLAminus | -128.33, -166.59 | 51.25, 57.82 | -86.79, 6.35 | 301.95, 6.09 | -60.92, -25.47 | in-in | in | 7.847 | Saltbr-in | 2.81 | HRD-in | -73.31, -54.57 | 78.67, -3.84 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.931 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.1, -24.0 | APE9-dihe-na | -84.65, -159.21 | APE8-dihe-in | -83.03, 124.26 | APE8-rot-in | 298.64 | APE67-dihe-in | -57.08, -33.68 | -53.72, -43.01 | APE12-dist-in | 13.141 | APE11-dist-in | 12.324 | APE10-dist-in | 6.259 | APE9-dist-in | 3.636 | None | None | None | XRAY | 1.75 | 0.169 | 0.188 | A | 306 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qim | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 6B8YA | 200 | 502 | 503.0 | D0A:60601 | Type1.5_Back | Active | DFGin | 6.054 | 13.076 | BLAminus | -131.41, -174.19 | 61.19, 66.23 | -95.1, 10.56 | 300.15, 7.66 | -60.38, -25.6 | in-in | in | 7.771 | Saltbr-in | 2.908 | HRD-in | -74.58, -53.37 | 74.48, -1.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.69, -30.19 | APE9-dihe-na | -79.71, -163.36 | APE8-dihe-in | -78.33, 124.12 | APE8-rot-in | 302.16 | APE67-dihe-in | -55.15, -33.95 | -56.38, -43.01 | APE12-dist-in | 12.896 | APE11-dist-in | 12.272 | APE10-dist-in | 6.192 | APE9-dist-in | 3.665 | T204D | None | None | XRAY | 1.65 | 0.18 | 0.208 | A | 307 | 303 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 6b8y | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2X7OC | 171 | 500 | 503.0 | ZOP:600 | Type1.5_Back | Active | DFGin | 6.853 | 13.741 | BLAminus | -128.05, 170.08 | 59.35, 88.53 | -108.53, 28.35 | 289.5, 149.12 | -69.05, -31.39 | in-in | in | 8.073 | Saltbr-in | 3.511 | HRD-in | -65.39, -40.6 | 69.36, -25.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.06 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.94, 148.96 | APE9-dihe-na | 97.31, -171.76 | APE8-dihe-in | -74.42, 131.23 | APE8-rot-in | 314.85 | APE67-dihe-in | -65.62, -33.63 | -61.56, -33.26 | APE12-dist-in | 11.785 | APE11-dist-in | 11.793 | APE10-dist-in | 5.967 | APE9-dist-in | 4.732 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2X7OD | 171 | 500 | 503.0 | ZOP:600 | Type1.5_Back | Active | DFGin | 6.851 | 13.771 | BLAminus | -128.04, 169.94 | 59.4, 88.47 | -108.43, 28.21 | 289.11, 149.16 | -69.32, -30.88 | in-in | in | 8.091 | Saltbr-in | 3.535 | HRD-in | -65.64, -40.65 | 69.2, -26.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.057 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.87, 149.08 | APE9-dihe-na | 96.88, -171.59 | APE8-dihe-in | -74.3, 131.16 | APE8-rot-in | 314.89 | APE67-dihe-in | -64.63, -35.86 | -61.66, -32.82 | APE12-dist-in | 11.796 | APE11-dist-in | 11.801 | APE10-dist-in | 5.972 | APE9-dist-in | 4.735 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2X7OE | 171 | 500 | 503.0 | ZOP:600 | Type1.5_Back | Active | DFGin | 6.856 | 13.729 | BLAminus | -128.08, 169.89 | 59.79, 88.24 | -108.3, 28.24 | 289.35, 149.2 | -69.25, -30.86 | in-in | in | 8.09 | Saltbr-in | 3.552 | HRD-in | -65.48, -40.48 | 69.3, -25.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.059 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.31, 151.21 | APE9-dihe-na | 97.11, -171.6 | APE8-dihe-in | -74.4, 131.12 | APE8-rot-in | 315.09 | APE67-dihe-in | -65.13, -34.5 | -61.63, -32.52 | APE12-dist-in | 11.779 | APE11-dist-in | 11.735 | APE10-dist-in | 5.956 | APE9-dist-in | 4.731 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3KCFA | 171 | 500 | 503.0 | JZO:1 | Type1.5_Back | Active | DFGin | 6.193 | 12.905 | BLAminus | -150.7, 165.18 | 67.92, 79.43 | -90.06, 14.08 | 309.25, 11.69 | -44.14, -39.87 | in-in | in | 8.196 | Saltbr-in | 2.837 | HRD-in | -56.75, -49.06 | 70.7, 0.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -96.99, 164.53 | APE9-dihe-na | 104.66, 167.11 | APE8-dihe-in | -69.97, 124.0 | APE8-rot-in | 297.54 | APE67-dihe-in | -37.23, -57.4 | -40.07, -69.34 | APE12-dist-in | 11.463 | APE11-dist-in | 12.171 | APE10-dist-in | 6.162 | APE9-dist-in | 3.762 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | A | 342 | 328 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3KCFB | 171 | 501 | 503.0 | JZO:2 | Type1.5_Back | Active | DFGin | 6.025 | 12.627 | BLAminus | -135.28, -176.57 | 58.41, 88.07 | -103.95, 28.48 | 315.03, 7.91 | -62.87, -35.81 | in-in | in | 8.145 | Saltbr-in | 2.601 | HRD-in | -81.18, -54.27 | 77.68, -8.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.97 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.7, -176.11 | APE9-dihe-na | 95.21, 172.61 | APE8-dihe-in | -76.23, 133.32 | APE8-rot-in | 308.48 | APE67-dihe-in | -45.62, -25.89 | -46.72, -68.47 | APE12-dist-in | 11.519 | APE11-dist-in | 11.413 | APE10-dist-in | 5.954 | APE9-dist-in | 3.732 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3KCFC | 171 | 500 | 503.0 | JZO:3 | Type1.5_Back | Active | DFGin | 6.692 | 12.959 | BLAminus | -135.28, 165.04 | 69.33, 88.35 | -106.61, 31.51 | 302.0, 1.76 | -58.82, -55.68 | in-in | in | 8.036 | Saltbr-in | 2.379 | HRD-in | -81.96, -30.19 | 61.27, -12.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.897 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -114.43, -160.74 | APE9-dihe-na | 83.32, -178.05 | APE8-dihe-in | -94.01, 131.52 | APE8-rot-in | 317.12 | APE67-dihe-in | -41.44, -18.99 | -53.51, -67.7 | APE12-dist-in | 10.742 | APE11-dist-in | 11.842 | APE10-dist-in | 6.224 | APE9-dist-in | 3.856 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3KCFD | 171 | 500 | 503.0 | JZO:4 | Type1.5_Back | Active | DFGin | 6.889 | 12.999 | BLAminus | -135.85, -173.78 | 57.12, 75.33 | -93.52, 22.15 | 298.91, 178.96 | -63.23, -14.31 | in-in | in | 8.264 | Saltbr-in | 2.894 | HRD-in | -62.47, -52.01 | 74.47, -2.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.771 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.66, 172.34 | APE9-dihe-na | 99.39, 173.59 | APE8-dihe-in | -80.33, 105.05 | APE8-rot-in | 316.25 | APE67-dihe-in | -46.61, -41.72 | -34.28, -49.6 | APE12-dist-in | 12.043 | APE11-dist-in | 12.05 | APE10-dist-in | 6.327 | APE9-dist-in | 4.044 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3KCFE | 171 | 500 | 503.0 | JZO:5 | Type1.5_Back | Active | DFGin | 6.468 | 12.982 | BLAminus | -143.17, -179.95 | 57.87, 88.27 | -108.02, 21.93 | 307.67, 3.89 | -69.37, -7.25 | in-in | in | 8.028 | Saltbr-in | 2.856 | HRD-in | -68.17, -50.18 | 73.66, 3.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.902 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.74, 177.4 | APE9-dihe-na | 104.24, -175.74 | APE8-dihe-in | -89.11, 123.84 | APE8-rot-in | 292.33 | APE67-dihe-in | -50.81, -36.21 | -50.11, -48.46 | APE12-dist-in | 9.931 | APE11-dist-in | 12.001 | APE10-dist-in | 6.217 | APE9-dist-in | 3.796 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1B6CB | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.851 | 13.394 | BLAminus | -130.85, -177.18 | 52.69, 80.31 | -95.42, 25.6 | 300.29, 176.12 | -64.72, -15.76 | in-out | in | 8.603 | Saltbr-out | 4.114 | HRD-in | -69.56, -62.44 | 85.43, -5.19 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.956 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.23, 170.19 | APE9-dihe-na | -45.35, 160.71 | APE8-dihe-in | -68.99, 127.88 | APE8-rot-in | 301.39 | APE67-dihe-in | -71.24, -15.17 | -60.4, -35.84 | APE12-dist-in | 11.453 | APE11-dist-out | 7.315 | APE10-dist-out | 8.448 | APE9-dist-in | 3.73 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | B | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1B6CD | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.963 | 13.317 | BLAminus | -130.99, -177.26 | 52.75, 80.27 | -95.41, 25.6 | 300.53, 176.04 | -64.6, -15.85 | in-out | in | 8.6 | Saltbr-out | 4.115 | HRD-in | -69.77, -62.44 | 85.53, -5.06 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.958 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.35, 170.01 | APE9-dihe-na | -45.12, 160.61 | APE8-dihe-in | -69.1, 128.03 | APE8-rot-in | 301.09 | APE67-dihe-in | -71.13, -15.35 | -60.35, -36.04 | APE12-dist-in | 11.453 | APE11-dist-out | 7.314 | APE10-dist-out | 8.445 | APE9-dist-in | 3.725 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | D | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1B6CF | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.998 | 13.814 | BLAminus | -130.93, -177.22 | 52.78, 80.13 | -95.35, 25.63 | 300.41, 176.19 | -64.73, -15.73 | in-out | in | 8.602 | Saltbr-out | 4.114 | HRD-in | -69.45, -62.52 | 85.59, -5.04 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.957 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.38, 170.18 | APE9-dihe-na | -45.27, 160.69 | APE8-dihe-in | -69.12, 128.05 | APE8-rot-in | 301.08 | APE67-dihe-in | -71.24, -15.27 | -60.51, -35.82 | APE12-dist-in | 11.454 | APE11-dist-out | 7.314 | APE10-dist-out | 8.445 | APE9-dist-in | 3.727 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | F | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1B6CH | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.933 | 13.373 | BLAminus | -131.03, -177.2 | 52.83, 80.24 | -95.22, 25.39 | 300.35, 176.04 | -64.71, -15.81 | in-out | in | 8.601 | Saltbr-out | 4.113 | HRD-in | -69.67, -62.6 | 85.56, -5.13 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.956 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.24, 170.15 | APE9-dihe-na | -45.32, 160.68 | APE8-dihe-in | -69.01, 127.87 | APE8-rot-in | 301.38 | APE67-dihe-in | -71.25, -15.25 | -60.38, -35.9 | APE12-dist-in | 11.451 | APE11-dist-out | 7.311 | APE10-dist-out | 8.446 | APE9-dist-in | 3.729 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | H | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1RW8A | 200 | 500 | 503.0 | 580:501 | Type1 | Inactive | DFGin | 6.023 | 12.845 | BLAminus | -123.87, -176.48 | 52.01, 78.57 | -101.69, 16.55 | 307.13, 6.03 | -62.1, -24.92 | in-in | in | 7.841 | Saltbr-in | 3.467 | HRD-in | -69.23, -61.02 | 80.12, 4.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.902 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioi | APE10-dihe-na | -83.25, -151.65 | APE9-dihe-na | -88.81, -163.17 | APE8-dihe-in | -80.66, 118.18 | APE8-rot-in | 309.35 | APE67-dihe-in | -55.07, -38.39 | -52.69, -43.2 | APE12-dist-in | 11.486 | APE11-dist-in | 8.854 | APE10-dist-out | 8.62 | APE9-dist-in | 4.107 | None | None | None | XRAY | 2.4 | 0.26 | 0.291 | A | 301 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1rw8 | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1PY5A | 200 | 500 | 503.0 | PY1:700 | Type1 | Inactive | DFGin | 6.325 | 13.096 | BLAminus | -139.22, -176.23 | 51.49, 62.68 | -91.32, 17.81 | 306.9, 168.43 | -57.65, -31.73 | in-in | in | 7.831 | Saltbr-in | 2.897 | HRD-in | -74.07, -48.58 | 75.5, -7.56 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.862 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioi | APE10-dihe-na | -82.55, -147.04 | APE9-dihe-na | -97.21, -166.02 | APE8-dihe-in | -77.65, 124.21 | APE8-rot-in | 307.07 | APE67-dihe-in | -64.31, -27.94 | -63.63, -30.26 | APE12-dist-in | 11.444 | APE11-dist-in | 8.66 | APE10-dist-out | 8.572 | APE9-dist-in | 4.119 | None | None | None | XRAY | 2.3 | 0.26 | 0.292 | A | 326 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1py5 | TKL_TGFBR1_HUMAN | TKL | 4.1e-85 | 291.4 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 2X7OB | 171 | 500 | 503.0 | ZOP:600 | Type1 | Inactive | DFGin | 6.858 | 13.746 | BLAminus | -128.22, 169.83 | 59.7, 88.26 | -108.23, 28.26 | 289.27, 149.16 | -69.33, -30.83 | in-out | in | 8.118 | Saltbr-out | 3.833 | HRD-in | -65.55, -40.47 | 69.31, -25.99 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.059 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.06, 149.04 | APE9-dihe-na | 97.27, -171.94 | APE8-dihe-in | -74.39, 131.11 | APE8-rot-in | 314.97 | APE67-dihe-in | -65.1, -35.09 | -61.66, -32.49 | APE12-dist-in | 11.793 | APE11-dist-in | 11.793 | APE10-dist-in | 5.967 | APE9-dist-in | 4.727 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | B | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3FAAC | 171 | 500 | 503.0 | 55F:601 | Type1 | Inactive | DFGin | 6.142 | 13.141 | BLAminus | -126.27, 176.42 | 50.71, 78.49 | -102.58, 30.06 | 320.3, 19.34 | -66.31, -17.95 | in-in | in | 7.99 | Saltbr-in | 2.662 | HRD-in | -67.56, -21.99 | 46.1, 19.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.947 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -120.66, 131.05 | APE9-dihe-na | 148.7, 175.0 | APE8-dihe-in | -102.93, 87.73 | APE8-rot-in | 305.5 | APE67-dihe-out | -28.83, -55.82 | 5.18, -84.04 | APE12-dist-in | 11.481 | APE11-dist-in | 12.149 | APE10-dist-in | 6.247 | APE9-dist-in | 4.208 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 1VJYA | 201 | 503 | 503.0 | 460:999 | Type1 | None | DFGin | 6.095 | 12.796 | BLAminus | -131.96, -168.3 | 46.73, 72.17 | -95.27, 7.02 | 307.89, 4.49 | -49.86, -32.3 | in-in | in | 7.726 | Saltbr-in | 2.753 | HRD-in | -71.95, -49.94 | 73.94, 4.16 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.848 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -108.72, 178.34 | APE9-dihe-na | 100.08, -177.16 | APE8-dihe-in | -88.48, 114.15 | APE8-rot-in | 304.07 | APE67-dihe-in | -56.76, -36.75 | -44.55, -45.61 | APE12-dist-none | 999.0 | APE11-dist-in | 11.557 | APE10-dist-in | 6.513 | APE9-dist-in | 3.865 | None | None | None | XRAY | 2.0 | 0.223 | 0.275 | A | 303 | 299 | 4 | 0 | 0 | 4 | [[205, 494]] | 1.0 | 1vjy | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3GXLA | 201 | 498 | 503.0 | QIG:60999 | Type1 | None | DFGin | 5.986 | 13.162 | BLAminus | -117.01, -170.6 | 33.6, 86.88 | -102.63, 15.85 | 311.96, 176.51 | -62.1, -23.52 | in-in | in | 8.223 | Saltbr-in | 2.93 | HRD-in | -71.35, -53.37 | 77.01, 1.76 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.958 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -62.74, 167.86 | APE9-dihe-na | 117.67, 172.21 | APE8-dihe-in | -83.62, 118.05 | APE8-rot-in | 304.44 | APE67-dihe-in | -50.23, -35.35 | -45.35, -55.49 | APE12-dist-none | 999.0 | APE11-dist-in | 12.158 | APE10-dist-in | 6.739 | APE9-dist-in | 4.173 | None | None | None | XRAY | 1.8 | 0.228 | 0.263 | A | 303 | 285 | 13 | 0 | 0 | 5 | [[205, 494]] | 1.0 | 3gxl | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3HMMA | 201 | 498 | 503.0 | 855:60857 | Type1 | None | DFGin | 6.119 | 13.049 | BLAminus | -127.07, -168.91 | 53.99, 65.82 | -94.96, 13.15 | 305.68, 3.69 | -60.53, -23.27 | in-in | in | 8.024 | Saltbr-in | 2.812 | HRD-in | -74.05, -51.32 | 76.01, -1.97 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.934 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -160.63 | APE8-dihe-in | -79.78, 120.6 | APE8-rot-in | 300.84 | APE67-dihe-in | -55.11, -37.41 | -48.22, -47.79 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.917 | None | None | None | XRAY | 1.7 | 0.223 | 0.241 | A | 303 | 293 | 5 | 0 | 0 | 5 | [[205, 494]] | 1.0 | 3hmm | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 9J9DA | 202 | 502 | 503.0 | A1L30:701 | Type1 | None | DFGin | 5.967 | 12.455 | BLAminus | -128.65, -173.5 | 51.95, 67.83 | -91.44, 10.62 | 307.73, 2.77 | -64.11, -26.42 | in-in | in | 8.02 | Saltbr-in | 2.807 | HRD-in | -76.64, -51.57 | 79.18, -0.61 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.92 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -92.35, -34.47 | APE9-dihe-na | -89.02, -159.15 | APE8-dihe-in | -77.18, 122.97 | APE8-rot-in | 307.18 | APE67-dihe-in | -57.12, -34.57 | -60.97, -41.48 | APE12-dist-none | 999.0 | APE11-dist-in | 12.145 | APE10-dist-in | 6.163 | APE9-dist-in | 4.067 | None | None | None | XRAY | 1.337 | 0.191 | 0.209 | A | 306 | 296 | 5 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 9j9d | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| 3TZMA | 200 | 496 | 503.0 | 085:1 | Type1 | None | DFGin | 6.065 | 13.106 | BLAminus | -122.58, -169.81 | 59.22, 59.29 | -91.38, 11.48 | 304.6, 5.41 | -64.05, -23.93 | in-in | in | 7.963 | Saltbr-in | 2.833 | HRD-in | -81.31, -50.79 | 80.1, -5.96 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.968 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -87.36, 160.54 | APE9-dihe-na | 102.22, -177.2 | APE8-dihe-in | -87.37, 126.2 | APE8-rot-in | 298.62 | APE67-dihe-in | -59.36, -31.96 | -58.47, -41.28 | APE12-dist-none | 999.0 | APE11-dist-in | 12.238 | APE10-dist-in | 6.184 | APE9-dist-in | 3.825 | None | None | None | XRAY | 1.7 | 0.172 | 0.205 | A | 309 | 295 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3tzm | TKL_TGFBR1_HUMAN | TKL | 3.4e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TGFR1_HUMAN | 5E8UA | P36897 | 200 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 7.25 | 14.239 | BLAminus | -134.62, -172.63 | 56.13, 81.95 | -101.29, 16.47 | 292.48, 105.22 | -57.91, -29.22 | in-in | in | 7.887 | Saltbr-in | 2.946 | HRD-in | -72.05, -48.87 | 69.51, 7.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.969 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -102.25, 153.37 | APE9-dihe-na | 113.03, -170.78 | APE8-dihe-in | -89.61, 116.01 | APE8-rot-in | 305.95 | APE67-dihe-in | -56.91, -33.28 | -47.65, -46.01 | APE12-dist-in | 13.141 | APE11-dist-in | 12.522 | APE10-dist-in | 6.48 | APE9-dist-in | 3.958 | T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F | None | None | XRAY | 2.03 | 0.181 | 0.223 | A | 307 | 303 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8u | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 2.3e-85 | 292.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 4X2NA | P36897 | 200 | 501 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.15 | 13.2 | BLAminus | -127.58, -171.48 | 51.56, 55.64 | -81.72, 7.99 | 306.47, 9.87 | -57.69, -30.68 | in-in | in | 7.746 | Saltbr-in | 3.137 | HRD-in | -73.45, -50.82 | 74.64, -6.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.988 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.64, 175.91 | APE9-dihe-na | 96.93, 176.28 | APE8-dihe-in | -81.13, 124.7 | APE8-rot-in | 305.67 | APE67-dihe-in | -55.99, -35.77 | -56.51, -42.26 | APE12-dist-in | 11.788 | APE11-dist-in | 11.876 | APE10-dist-in | 6.194 | APE9-dist-in | 3.712 | None | None | None | XRAY | 1.8 | 0.163 | 0.201 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2n | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5E8SA | P36897 | 200 | 498 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.227 | 13.345 | BLAminus | -130.71, -170.38 | 50.26, 56.29 | -81.51, 7.19 | 302.58, 10.42 | -59.69, -25.71 | in-in | in | 7.75 | Saltbr-in | 3.098 | HRD-in | -75.18, -50.46 | 75.3, -6.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.942 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.12, 158.63 | APE9-dihe-na | 109.47, 177.89 | APE8-dihe-in | -83.28, 125.6 | APE8-rot-in | 301.61 | APE67-dihe-in | -57.6, -32.67 | -59.04, -39.92 | APE12-dist-in | 13.384 | APE11-dist-in | 12.417 | APE10-dist-in | 6.303 | APE9-dist-in | 3.677 | None | None | None | XRAY | 1.45 | 0.172 | 0.188 | A | 306 | 299 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8s | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | AF-P36897-K1A | P36897 | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.097 | 12.697 | BLAminus | -127.47, -177.39 | 59.98, 50.67 | -75.64, 9.99 | 303.25, 0.83 | -67.03, -14.65 | in-in | in | 7.75 | Saltbr-in | 2.631 | HRD-in | -79.18, -43.89 | 66.79, -8.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.015 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.74, 159.13 | APE9-dihe-na | 99.19, -175.01 | APE8-dihe-in | -81.52, 117.2 | APE8-rot-in | 304.32 | APE67-dihe-in | -58.11, -28.29 | -49.21, -42.7 | APE12-dist-in | 13.034 | APE11-dist-in | 12.476 | APE10-dist-in | 6.348 | APE9-dist-in | 3.781 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306 | 306 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | AF-P36897-K1 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | AF-P36897-K3A | P36897 | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.388 | 12.882 | BLAminus | -127.89, -179.35 | 58.97, 55.86 | -76.18, 6.96 | 301.47, 0.09 | -63.41, -19.74 | in-in | in | 8.095 | Saltbr-in | 2.675 | HRD-in | -77.05, -40.27 | 65.4, -16.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.85 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -117.36, 158.96 | APE9-dihe-na | 107.71, -175.1 | APE8-dihe-in | -94.3, 114.61 | APE8-rot-in | 303.53 | APE67-dihe-in | -61.67, -24.01 | -41.02, -46.98 | APE12-dist-in | 11.212 | APE11-dist-in | 11.814 | APE10-dist-in | 5.925 | APE9-dist-in | 3.7 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306 | 306 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | AF-P36897-K3 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5E8TA | P36897 | 200 | 499 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.13 | 13.117 | BLAminus | -129.7, -170.36 | 54.3, 58.56 | -85.47, 9.03 | 309.14, 5.15 | -56.74, -27.28 | in-in | in | 7.84 | Saltbr-in | 2.94 | HRD-in | -72.25, -51.54 | 76.95, -4.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.969 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -78.56, -31.05 | APE9-dihe-na | -81.1, -159.38 | APE8-dihe-in | -84.33, 122.67 | APE8-rot-in | 299.0 | APE67-dihe-in | -55.04, -35.69 | -53.58, -44.7 | APE12-dist-in | 13.067 | APE11-dist-in | 12.282 | APE10-dist-in | 6.237 | APE9-dist-in | 3.791 | T204D | None | None | XRAY | 1.7 | 0.17 | 0.19 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8t | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1IASA | P36897 | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.721 | 12.723 | BLAminus | -151.41, 164.95 | 71.98, 88.97 | -106.86, 22.49 | 311.89, 1.41 | -60.78, -26.26 | in-in | in | 8.24 | Saltbr-in | 2.79 | HRD-in | -63.37, -49.76 | 71.64, 8.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.974 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.42, 172.85 | APE9-dihe-na | 97.41, 166.83 | APE8-dihe-in | -62.29, 121.18 | APE8-rot-in | 307.67 | APE67-dihe-in | -45.67, -30.78 | -49.33, -54.47 | APE12-dist-in | 11.452 | APE11-dist-in | 11.629 | APE10-dist-in | 6.172 | APE9-dist-in | 4.131 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | A | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1IASB | P36897 | 171 | 501 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.652 | 12.707 | BLAminus | -150.79, 165.66 | 71.53, 88.91 | -106.55, 22.01 | 312.14, 1.23 | -60.97, -25.51 | in-in | in | 8.241 | Saltbr-in | 2.799 | HRD-in | -64.38, -48.85 | 71.21, 7.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.005 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.79, 173.68 | APE9-dihe-na | 99.72, 167.49 | APE8-dihe-in | -63.26, 121.22 | APE8-rot-in | 308.35 | APE67-dihe-in | -44.49, -32.42 | -49.46, -55.33 | APE12-dist-in | 10.321 | APE11-dist-in | 11.628 | APE10-dist-in | 6.241 | APE9-dist-in | 4.05 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 1ias | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1IASC | P36897 | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.59 | 12.711 | BLAminus | -150.31, 164.7 | 71.4, 89.07 | -106.94, 23.22 | 312.6, 1.77 | -61.3, -25.67 | in-in | in | 8.197 | Saltbr-in | 2.799 | HRD-in | -63.0, -50.37 | 71.83, 9.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.013 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.75, 170.21 | APE9-dihe-na | 100.55, 167.25 | APE8-dihe-in | -63.65, 121.53 | APE8-rot-in | 308.64 | APE67-dihe-in | -44.33, -30.7 | -49.24, -56.44 | APE12-dist-in | 11.349 | APE11-dist-in | 11.759 | APE10-dist-in | 6.222 | APE9-dist-in | 4.15 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1IASD | P36897 | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.594 | 12.743 | BLAminus | -152.15, 165.79 | 70.83, 87.83 | -105.27, 21.55 | 312.92, 0.98 | -60.27, -25.54 | in-in | in | 8.189 | Saltbr-in | 2.775 | HRD-in | -64.51, -48.18 | 71.39, 8.63 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.993 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.69, 169.96 | APE9-dihe-na | 98.27, 166.26 | APE8-dihe-in | -61.5, 120.34 | APE8-rot-in | 308.37 | APE67-dihe-in | -44.16, -31.51 | -48.36, -56.13 | APE12-dist-in | 10.732 | APE11-dist-in | 11.784 | APE10-dist-in | 6.18 | APE9-dist-in | 4.04 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1IASE | P36897 | 171 | 500 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.685 | 12.738 | BLAminus | -151.39, 165.15 | 70.82, 89.42 | -106.94, 21.97 | 311.98, 2.05 | -61.66, -24.41 | in-in | in | 8.226 | Saltbr-in | 2.803 | HRD-in | -61.95, -50.33 | 72.19, 7.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.008 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.31, 173.9 | APE9-dihe-na | 98.05, 167.39 | APE8-dihe-in | -64.1, 121.3 | APE8-rot-in | 308.19 | APE67-dihe-in | -45.93, -31.42 | -49.14, -54.62 | APE12-dist-in | 11.636 | APE11-dist-in | 11.505 | APE10-dist-in | 6.149 | APE9-dist-in | 4.002 | None | None | None | XRAY | 2.9 | 0.255 | 0.284 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1ias | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5E8XA | P36897 | 200 | 503 | 503.0 | STU:601 | Type1 | Active | DFGin | 7.401 | 13.771 | BLAminus | -132.02, 177.79 | 68.95, 84.86 | -101.89, 20.89 | 298.69, 99.78 | -60.9, -22.78 | in-in | in | 7.646 | Saltbr-in | 3.316 | HRD-in | -78.83, -50.32 | 78.23, -2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.2, 171.93 | APE9-dihe-na | 104.3, 177.57 | APE8-dihe-in | -80.96, 119.4 | APE8-rot-in | 304.53 | APE67-dihe-in | -55.33, -34.35 | -53.44, -41.29 | APE12-dist-in | 11.709 | APE11-dist-in | 11.927 | APE10-dist-in | 6.258 | APE9-dist-in | 3.946 | T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F | None | None | XRAY | 1.45 | 0.191 | 0.21 | A | 307 | 304 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8x | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 2.3e-85 | 292.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5E90A | P36897 | 200 | 499 | 503.0 | 5L4:60601 | Type1 | Active | DFGin | 7.033 | 13.968 | BLAminus | -132.44, -170.95 | 59.07, 73.91 | -100.08, 11.67 | 293.12, 109.78 | -58.9, -27.5 | in-in | in | 7.732 | Saltbr-in | 2.865 | HRD-in | -62.69, -55.46 | 77.29, -2.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.872 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.74, -31.43 | APE9-dihe-na | -82.55, -164.68 | APE8-dihe-in | -74.68, 122.19 | APE8-rot-in | 303.81 | APE67-dihe-in | -54.67, -36.7 | -55.17, -42.7 | APE12-dist-in | 12.594 | APE11-dist-in | 11.9 | APE10-dist-in | 5.887 | APE9-dist-in | 3.841 | T204D,I211V,Y249F,S280T,Y282F,S287N,A350C,L352F | None | None | XRAY | 2.05 | 0.178 | 0.218 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e90 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 2.3e-85 | 292.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5USQA | P36897 | 200 | 498 | 503.0 | 8LY:500 | Type1 | Active | DFGin | 6.294 | 13.451 | BLAminus | -128.65, -178.48 | 58.74, 56.74 | -84.73, 2.3 | 308.58, 3.38 | -59.48, -22.95 | in-in | in | 7.752 | Saltbr-in | 3.191 | HRD-in | -74.99, -53.41 | 77.78, -10.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.92 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.34, -32.16 | APE9-dihe-na | -75.45, -164.79 | APE8-dihe-in | -80.15, 126.14 | APE8-rot-in | 305.26 | APE67-dihe-in | -52.52, -34.72 | -59.83, -43.81 | APE12-dist-in | 13.024 | APE11-dist-in | 12.008 | APE10-dist-in | 6.158 | APE9-dist-in | 3.557 | None | None | None | XRAY | 2.55 | 0.182 | 0.231 | A | 299 | 299 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5usq | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3e-85 | 291.9 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5FRIA | P36897 | 200 | 498 | 503.0 | ZUQ:61501 | Type1 | Active | DFGin | 5.986 | 12.349 | BLAminus | -129.47, -173.22 | 60.99, 71.38 | -101.21, 12.39 | 307.22, 5.28 | -67.89, -22.52 | in-in | in | 7.758 | Saltbr-in | 2.857 | HRD-in | -78.14, -52.35 | 77.86, -1.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.926 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.89, -25.51 | APE9-dihe-na | -92.81, -153.48 | APE8-dihe-in | -86.34, 123.11 | APE8-rot-in | 303.21 | APE67-dihe-in | -53.0, -34.54 | -57.92, -43.35 | APE12-dist-in | 12.836 | APE11-dist-in | 11.987 | APE10-dist-in | 6.05 | APE9-dist-in | 3.945 | None | None | None | XRAY | 2.0 | 0.164 | 0.193 | A | 301 | 299 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5fri | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 9F6XA | P36897 | 200 | 500 | 503.0 | A1IAZ:60401 | Type1 | Active | DFGin | 6.135 | 13.376 | BLAminus | -110.91, -175.59 | 63.64, 55.87 | -85.09, 3.96 | 315.03, 1.12 | -62.09, -27.8 | in-in | in | 8.172 | Saltbr-in | 2.73 | HRD-in | -72.7, -49.45 | 76.37, -0.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.008 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -96.61, -34.29 | APE9-dihe-na | -78.73, -165.12 | APE8-dihe-in | -74.89, 126.22 | APE8-rot-in | 295.38 | APE67-dihe-in | -52.17, -40.21 | -62.21, -41.17 | APE12-dist-in | 13.477 | APE11-dist-in | 12.232 | APE10-dist-in | 6.103 | APE9-dist-in | 3.604 | None | None | None | XRAY | 2.68 | 0.214 | 0.248 | A | 303 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 9f6x | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 4X0MA | P36897 | 200 | 501 | 503.0 | 3WA:60601 | Type1 | Active | DFGin | 6.253 | 12.884 | BLAminus | -128.27, -179.8 | 55.38, 57.51 | -85.94, 12.49 | 298.0, 10.23 | -63.66, -28.1 | in-in | in | 7.343 | Saltbr-in | 3.153 | HRD-in | -62.49, -53.22 | 74.03, -11.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.008 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.83, 167.91 | APE9-dihe-na | 99.86, -179.25 | APE8-dihe-in | -77.31, 123.46 | APE8-rot-in | 305.82 | APE67-dihe-in | -54.73, -39.98 | -54.51, -42.68 | APE12-dist-in | 11.689 | APE11-dist-in | 11.872 | APE10-dist-in | 6.21 | APE9-dist-in | 3.823 | None | None | None | XRAY | 1.68 | 0.21 | 0.239 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x0m | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 4X2FA | P36897 | 200 | 501 | 503.0 | 3WJ:60601 | Type1 | Active | DFGin | 6.198 | 12.989 | BLAminus | -129.57, -169.63 | 49.35, 56.72 | -81.87, 7.01 | 303.23, 9.49 | -60.29, -24.32 | in-in | in | 7.557 | Saltbr-in | 2.939 | HRD-in | -74.24, -48.95 | 76.58, -5.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.03, 171.99 | APE9-dihe-na | 101.85, 179.14 | APE8-dihe-in | -82.12, 123.51 | APE8-rot-in | 300.96 | APE67-dihe-in | -58.79, -32.2 | -58.45, -40.31 | APE12-dist-in | 11.805 | APE11-dist-in | 11.906 | APE10-dist-in | 6.197 | APE9-dist-in | 3.807 | None | None | None | XRAY | 1.49 | 0.165 | 0.191 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2f | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 4X2GA | P36897 | 200 | 501 | 503.0 | 3WK:60601 | Type1 | Active | DFGin | 6.161 | 12.995 | BLAminus | -126.43, -164.75 | 48.26, 54.97 | -83.24, 5.58 | 306.41, 9.37 | -59.31, -23.57 | in-in | in | 7.56 | Saltbr-in | 3.063 | HRD-in | -73.4, -50.72 | 76.5, -5.82 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.905 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.4, 173.04 | APE9-dihe-na | 101.04, 176.44 | APE8-dihe-in | -79.69, 125.01 | APE8-rot-in | 303.47 | APE67-dihe-in | -59.43, -31.39 | -61.05, -38.4 | APE12-dist-in | 11.852 | APE11-dist-in | 11.925 | APE10-dist-in | 6.221 | APE9-dist-in | 3.793 | None | None | None | XRAY | 1.51 | 0.166 | 0.185 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2g | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2WOTA | P36897 | 200 | 500 | 503.0 | ZZG:61500 | Type1 | Active | DFGin | 6.1 | 13.031 | BLAminus | -130.27, -169.46 | 60.16, 61.47 | -92.46, 8.2 | 303.12, 6.85 | -64.56, -24.36 | in-in | in | 7.663 | Saltbr-in | 3.074 | HRD-in | -80.51, -53.82 | 76.92, 0.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.95 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -90.42, -22.62 | APE9-dihe-na | -94.01, -157.41 | APE8-dihe-in | -80.51, 121.5 | APE8-rot-in | 307.33 | APE67-dihe-in | -52.87, -38.64 | -55.17, -43.39 | APE12-dist-in | 13.131 | APE11-dist-in | 12.287 | APE10-dist-in | 6.338 | APE9-dist-in | 3.77 | None | None | None | XRAY | 1.85 | 0.181 | 0.221 | A | 306 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2wot | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2WOUA | P36897 | 200 | 496 | 503.0 | ZZF:61500 | Type1 | Active | DFGin | 6.124 | 13.039 | BLAminus | -133.49, -169.53 | 51.05, 62.4 | -92.04, 13.34 | 298.31, 178.69 | -62.77, -27.98 | in-in | in | 7.586 | Saltbr-in | 2.752 | HRD-in | -65.52, -56.03 | 81.95, -3.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.039 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.77, -22.31 | APE9-dihe-na | -79.77, -172.15 | APE8-dihe-in | -73.94, 125.36 | APE8-rot-in | 306.35 | APE67-dihe-in | -52.11, -29.79 | -56.64, -45.19 | APE12-dist-in | 13.078 | APE11-dist-in | 11.935 | APE10-dist-in | 6.041 | APE9-dist-in | 3.629 | None | None | None | XRAY | 2.3 | 0.229 | 0.302 | A | 306 | 297 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2wou | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 8YHLA | P36897 | 200 | 501 | 503.0 | A1D6I:60601 | Type1 | Active | DFGin | 6.021 | 13.048 | BLAminus | -124.89, -169.46 | 42.91, 75.25 | -91.67, 10.82 | 300.67, 10.41 | -67.27, -22.16 | in-in | in | 7.699 | Saltbr-in | 2.965 | HRD-in | -79.41, -52.59 | 75.07, -1.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.932 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -72.3, 155.92 | APE9-dihe-na | 107.61, -172.07 | APE8-dihe-in | -88.21, 123.34 | APE8-rot-in | 304.18 | APE67-dihe-in | -56.11, -38.82 | -61.94, -38.97 | APE12-dist-in | 13.343 | APE11-dist-in | 12.518 | APE10-dist-in | 6.314 | APE9-dist-in | 3.816 | None | None | None | XRAY | 1.47 | 0.165 | 0.193 | A | 306 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 8yhl | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5E8WA | P36897 | 200 | 501 | 503.0 | STU:60601 | Type1 | Active | DFGin | 6.216 | 12.991 | BLAminus | -115.91, -168.56 | 48.03, 66.8 | -87.81, 6.99 | 303.66, 6.47 | -53.89, -34.67 | in-in | in | 7.561 | Saltbr-in | 2.815 | HRD-in | -71.33, -51.46 | 73.08, -1.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.992 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -81.36, -32.83 | APE9-dihe-na | -81.66, -157.24 | APE8-dihe-in | -82.54, 122.58 | APE8-rot-in | 299.35 | APE67-dihe-in | -53.78, -37.25 | -53.32, -45.52 | APE12-dist-in | 13.054 | APE11-dist-in | 12.418 | APE10-dist-in | 6.3 | APE9-dist-in | 3.738 | T204D | None | None | XRAY | 1.86 | 0.168 | 0.186 | A | 307 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8w | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5E8ZA | P36897 | 200 | 499 | 503.0 | 5L4:60601 | Type1 | Active | DFGin | 5.938 | 12.742 | BLAminus | -131.72, -172.47 | 57.21, 65.07 | -93.0, 9.47 | 305.33, 7.41 | -62.65, -21.83 | in-in | in | 7.87 | Saltbr-in | 2.94 | HRD-in | -73.84, -51.69 | 76.4, -3.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.915 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -86.19, -27.35 | APE9-dihe-na | -88.81, -157.37 | APE8-dihe-in | -81.17, 121.36 | APE8-rot-in | 303.09 | APE67-dihe-in | -55.51, -33.19 | -54.0, -44.23 | APE12-dist-in | 13.117 | APE11-dist-in | 12.181 | APE10-dist-in | 6.139 | APE9-dist-in | 3.775 | T204D | None | None | XRAY | 1.51 | 0.183 | 0.207 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5e8z | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5QIKA | P36897 | 200 | 499 | 503.0 | J2M:60601 | Type1 | Active | DFGin | 6.134 | 12.822 | BLAminus | -129.19, -176.86 | 54.93, 67.17 | -89.45, 12.6 | 307.08, 5.45 | -57.51, -28.59 | in-in | in | 8.037 | Saltbr-in | 2.853 | HRD-in | -74.13, -49.19 | 76.47, -1.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -82.77, -28.33 | APE9-dihe-na | -83.38, -158.15 | APE8-dihe-in | -83.03, 121.9 | APE8-rot-in | 297.41 | APE67-dihe-in | -57.88, -31.82 | -55.17, -43.49 | APE12-dist-in | 13.224 | APE11-dist-in | 12.41 | APE10-dist-in | 6.393 | APE9-dist-in | 3.835 | T204D | None | None | XRAY | 1.58 | 0.166 | 0.19 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qik | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5QILA | P36897 | 200 | 499 | 503.0 | J2V:60601 | Type1 | Active | DFGin | 6.123 | 12.893 | BLAminus | -133.55, -173.28 | 54.13, 68.92 | -94.29, 10.19 | 306.15, 4.81 | -59.56, -26.12 | in-in | in | 7.782 | Saltbr-in | 3.012 | HRD-in | -72.26, -48.55 | 71.72, 0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.977 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.42, -32.81 | APE9-dihe-na | -79.5, -152.05 | APE8-dihe-in | -86.88, 119.67 | APE8-rot-in | 305.45 | APE67-dihe-in | -55.45, -33.57 | -52.15, -44.93 | APE12-dist-in | 12.839 | APE11-dist-in | 12.277 | APE10-dist-in | 6.153 | APE9-dist-in | 3.792 | T204D | None | None | XRAY | 1.98 | 0.171 | 0.21 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qil | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5QTZA | P36897 | 200 | 499 | 503.0 | QMY:60601 | Type1 | Active | DFGin | 6.173 | 13.35 | BLAminus | -138.39, -173.58 | 55.38, 56.92 | -82.72, 7.96 | 301.94, 5.0 | -56.41, -28.87 | in-in | in | 8.148 | Saltbr-in | 2.898 | HRD-in | -70.33, -51.13 | 74.03, -4.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.025 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -86.52, -26.25 | APE9-dihe-na | -81.63, -163.74 | APE8-dihe-in | -76.85, 122.93 | APE8-rot-in | 300.9 | APE67-dihe-in | -53.47, -35.21 | -52.57, -45.07 | APE12-dist-in | 12.983 | APE11-dist-in | 12.176 | APE10-dist-in | 6.168 | APE9-dist-in | 3.658 | T204D | None | None | XRAY | 1.83 | 0.171 | 0.2 | A | 307 | 300 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qtz | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5QU0A | P36897 | 200 | 502 | 503.0 | QMV:60601 | Type1 | Active | DFGin | 6.226 | 13.493 | BLAminus | -131.41, -169.26 | 50.76, 57.03 | -82.09, 5.13 | 306.24, 2.05 | -53.78, -29.06 | in-in | in | 7.858 | Saltbr-in | 2.924 | HRD-in | -72.09, -52.96 | 76.9, -5.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.961 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -85.59, 161.83 | APE9-dihe-na | 106.22, 171.28 | APE8-dihe-in | -76.79, 124.94 | APE8-rot-in | 300.79 | APE67-dihe-in | -53.51, -36.09 | -55.88, -43.03 | APE12-dist-in | 13.281 | APE11-dist-in | 12.425 | APE10-dist-in | 6.254 | APE9-dist-in | 3.655 | T204D | None | None | XRAY | 1.67 | 0.178 | 0.206 | A | 307 | 303 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qu0 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2X7OA | P36897 | 171 | 500 | 503.0 | ZOP:600 | Type1 | Active | DFGin | 6.832 | 13.774 | BLAminus | -128.16, 169.92 | 59.52, 88.44 | -108.37, 28.14 | 289.28, 149.08 | -69.29, -30.37 | in-in | in | 8.088 | Saltbr-in | 3.532 | HRD-in | -65.4, -40.58 | 69.2, -25.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.057 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.88, 149.39 | APE9-dihe-na | 96.51, -171.18 | APE8-dihe-in | -74.29, 131.0 | APE8-rot-in | 315.1 | APE67-dihe-in | -64.94, -34.48 | -61.98, -32.57 | APE12-dist-in | 11.82 | APE11-dist-in | 11.797 | APE10-dist-in | 5.973 | APE9-dist-in | 4.739 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | A | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3FAAA | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 5.904 | 13.047 | BLAminus | -165.74, 163.41 | 74.29, 54.12 | -79.67, 24.05 | 317.06, 176.62 | -56.68, -51.28 | in-in | in | 8.001 | Saltbr-in | 2.936 | HRD-in | -45.11, -27.8 | 52.25, 11.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.111 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.43, -171.19 | APE9-dihe-na | 80.03, 171.79 | APE8-dihe-in | -67.98, 121.11 | APE8-rot-in | 302.91 | APE67-dihe-in | -99.71, -73.49 | -46.09, -5.99 | APE12-dist-in | 11.624 | APE11-dist-in | 11.967 | APE10-dist-in | 6.015 | APE9-dist-in | 4.061 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | A | 342 | 328 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3FAAB | P36897 | 171 | 501 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.017 | 13.306 | BLAminus | -136.45, -176.24 | 60.04, 54.86 | -81.47, 12.98 | 307.95, 5.19 | -52.57, -45.29 | in-in | in | 8.1 | Saltbr-in | 3.037 | HRD-in | -75.89, -39.75 | 60.74, 14.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.115 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.32, 175.24 | APE9-dihe-na | 101.52, 166.7 | APE8-dihe-in | -70.87, 127.35 | APE8-rot-in | 315.28 | APE67-dihe-in | -36.34, -44.33 | -43.95, -69.54 | APE12-dist-in | 11.94 | APE11-dist-in | 12.0 | APE10-dist-in | 6.373 | APE9-dist-in | 4.084 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3FAAD | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.26 | 13.168 | BLAminus | -151.5, 176.63 | 62.94, 64.2 | -90.99, 26.98 | 302.19, 4.38 | -66.56, -19.34 | in-in | in | 7.809 | Saltbr-in | 2.745 | HRD-in | -63.44, -55.82 | 78.14, 1.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.86, 174.28 | APE9-dihe-na | 87.09, 173.14 | APE8-dihe-in | -66.87, 116.28 | APE8-rot-in | 325.42 | APE67-dihe-in | -60.47, -38.15 | -48.63, -36.35 | APE12-dist-in | 11.714 | APE11-dist-in | 11.894 | APE10-dist-in | 6.37 | APE9-dist-in | 4.229 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3FAAE | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Active | DFGin | 6.355 | 13.366 | BLAminus | -131.48, -168.05 | 37.37, 86.28 | -107.7, 26.02 | 296.92, 176.17 | -65.92, -19.56 | in-in | in | 7.781 | Saltbr-in | 3.095 | HRD-in | -66.77, -57.93 | 79.95, 12.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.85 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.13, 169.87 | APE9-dihe-na | 90.72, 172.5 | APE8-dihe-in | -64.72, 129.04 | APE8-rot-in | 310.98 | APE67-dihe-in | -56.46, -40.64 | -59.57, -42.14 | APE12-dist-in | 11.99 | APE11-dist-in | 12.056 | APE10-dist-in | 6.57 | APE9-dist-in | 3.982 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 8YHFA | P36897 | 201 | 498 | 503.0 | A1D6I:601 | Type1 | Active | DFGin | 6.037 | 13.152 | BLAminus | -127.63, -168.18 | 39.33, 73.78 | -89.91, 13.29 | 302.44, 7.93 | -62.86, -27.56 | in-in | in | 7.799 | Saltbr-in | 3.029 | HRD-in | -79.9, -54.99 | 79.42, -3.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.954 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.79, -23.11 | APE9-dihe-na | -96.35, -152.57 | APE8-dihe-in | -84.18, 124.71 | APE8-rot-in | 302.64 | APE67-dihe-in | -56.72, -32.39 | -61.45, -41.11 | APE12-dist-in | 13.178 | APE11-dist-in | 12.22 | APE10-dist-in | 6.218 | APE9-dist-in | 3.834 | None | None | None | XRAY | 1.4 | 0.167 | 0.192 | A | 343 | 298 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 8yhf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 5e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 4X2JA | P36897 | 200 | 501 | 503.0 | 3WN:60601 | Type1.5_Back | Active | DFGin | 6.245 | 13.082 | BLAminus | -129.47, -176.48 | 54.06, 62.42 | -89.1, 7.12 | 300.54, 6.95 | -58.75, -23.34 | in-in | in | 7.595 | Saltbr-in | 2.782 | HRD-in | -70.93, -49.34 | 73.15, -2.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.918 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.13, 172.46 | APE9-dihe-na | 95.45, -178.89 | APE8-dihe-in | -79.7, 121.22 | APE8-rot-in | 304.99 | APE67-dihe-in | -57.38, -35.27 | -55.84, -42.14 | APE12-dist-in | 11.79 | APE11-dist-in | 11.898 | APE10-dist-in | 6.199 | APE9-dist-in | 3.764 | None | None | None | XRAY | 1.69 | 0.167 | 0.184 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2j | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 4X2KA | P36897 | 200 | 501 | 503.0 | 3WO:60601 | Type1.5_Back | Active | DFGin | 6.245 | 13.082 | BLAminus | -129.47, -176.48 | 54.06, 62.42 | -89.1, 7.12 | 300.54, 6.95 | -58.75, -23.34 | in-in | in | 7.595 | Saltbr-in | 2.782 | HRD-in | -70.93, -49.34 | 73.15, -2.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.918 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.13, 172.46 | APE9-dihe-na | 95.45, -178.89 | APE8-dihe-in | -79.7, 121.22 | APE8-rot-in | 304.99 | APE67-dihe-in | -57.38, -35.27 | -55.84, -42.14 | APE12-dist-in | 11.79 | APE11-dist-in | 11.898 | APE10-dist-in | 6.199 | APE9-dist-in | 3.764 | None | None | None | XRAY | 1.69 | 0.167 | 0.184 | A | 305 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 4x2k | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.2e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 5QIMA | P36897 | 200 | 501 | 503.0 | J2Y:60601 | Type1.5_Back | Active | DFGin | 6.324 | 13.322 | BLAminus | -128.33, -166.59 | 51.25, 57.82 | -86.79, 6.35 | 301.95, 6.09 | -60.92, -25.47 | in-in | in | 7.847 | Saltbr-in | 2.81 | HRD-in | -73.31, -54.57 | 78.67, -3.84 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.931 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.1, -24.0 | APE9-dihe-na | -84.65, -159.21 | APE8-dihe-in | -83.03, 124.26 | APE8-rot-in | 298.64 | APE67-dihe-in | -57.08, -33.68 | -53.72, -43.01 | APE12-dist-in | 13.141 | APE11-dist-in | 12.324 | APE10-dist-in | 6.259 | APE9-dist-in | 3.636 | None | None | None | XRAY | 1.75 | 0.169 | 0.188 | A | 306 | 302 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 5qim | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 6B8YA | P36897 | 200 | 502 | 503.0 | D0A:60601 | Type1.5_Back | Active | DFGin | 6.054 | 13.076 | BLAminus | -131.41, -174.19 | 61.19, 66.23 | -95.1, 10.56 | 300.15, 7.66 | -60.38, -25.6 | in-in | in | 7.771 | Saltbr-in | 2.908 | HRD-in | -74.58, -53.37 | 74.48, -1.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.69, -30.19 | APE9-dihe-na | -79.71, -163.36 | APE8-dihe-in | -78.33, 124.12 | APE8-rot-in | 302.16 | APE67-dihe-in | -55.15, -33.95 | -56.38, -43.01 | APE12-dist-in | 12.896 | APE11-dist-in | 12.272 | APE10-dist-in | 6.192 | APE9-dist-in | 3.665 | T204D | None | None | XRAY | 1.65 | 0.18 | 0.208 | A | 307 | 303 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 6b8y | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2X7OC | P36897 | 171 | 500 | 503.0 | ZOP:600 | Type1.5_Back | Active | DFGin | 6.853 | 13.741 | BLAminus | -128.05, 170.08 | 59.35, 88.53 | -108.53, 28.35 | 289.5, 149.12 | -69.05, -31.39 | in-in | in | 8.073 | Saltbr-in | 3.511 | HRD-in | -65.39, -40.6 | 69.36, -25.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.06 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.94, 148.96 | APE9-dihe-na | 97.31, -171.76 | APE8-dihe-in | -74.42, 131.23 | APE8-rot-in | 314.85 | APE67-dihe-in | -65.62, -33.63 | -61.56, -33.26 | APE12-dist-in | 11.785 | APE11-dist-in | 11.793 | APE10-dist-in | 5.967 | APE9-dist-in | 4.732 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2X7OD | P36897 | 171 | 500 | 503.0 | ZOP:600 | Type1.5_Back | Active | DFGin | 6.851 | 13.771 | BLAminus | -128.04, 169.94 | 59.4, 88.47 | -108.43, 28.21 | 289.11, 149.16 | -69.32, -30.88 | in-in | in | 8.091 | Saltbr-in | 3.535 | HRD-in | -65.64, -40.65 | 69.2, -26.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.057 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.87, 149.08 | APE9-dihe-na | 96.88, -171.59 | APE8-dihe-in | -74.3, 131.16 | APE8-rot-in | 314.89 | APE67-dihe-in | -64.63, -35.86 | -61.66, -32.82 | APE12-dist-in | 11.796 | APE11-dist-in | 11.801 | APE10-dist-in | 5.972 | APE9-dist-in | 4.735 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2X7OE | P36897 | 171 | 500 | 503.0 | ZOP:600 | Type1.5_Back | Active | DFGin | 6.856 | 13.729 | BLAminus | -128.08, 169.89 | 59.79, 88.24 | -108.3, 28.24 | 289.35, 149.2 | -69.25, -30.86 | in-in | in | 8.09 | Saltbr-in | 3.552 | HRD-in | -65.48, -40.48 | 69.3, -25.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.059 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.31, 151.21 | APE9-dihe-na | 97.11, -171.6 | APE8-dihe-in | -74.4, 131.12 | APE8-rot-in | 315.09 | APE67-dihe-in | -65.13, -34.5 | -61.63, -32.52 | APE12-dist-in | 11.779 | APE11-dist-in | 11.735 | APE10-dist-in | 5.956 | APE9-dist-in | 4.731 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3KCFA | P36897 | 171 | 500 | 503.0 | JZO:1 | Type1.5_Back | Active | DFGin | 6.193 | 12.905 | BLAminus | -150.7, 165.18 | 67.92, 79.43 | -90.06, 14.08 | 309.25, 11.69 | -44.14, -39.87 | in-in | in | 8.196 | Saltbr-in | 2.837 | HRD-in | -56.75, -49.06 | 70.7, 0.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -96.99, 164.53 | APE9-dihe-na | 104.66, 167.11 | APE8-dihe-in | -69.97, 124.0 | APE8-rot-in | 297.54 | APE67-dihe-in | -37.23, -57.4 | -40.07, -69.34 | APE12-dist-in | 11.463 | APE11-dist-in | 12.171 | APE10-dist-in | 6.162 | APE9-dist-in | 3.762 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | A | 342 | 328 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3KCFB | P36897 | 171 | 501 | 503.0 | JZO:2 | Type1.5_Back | Active | DFGin | 6.025 | 12.627 | BLAminus | -135.28, -176.57 | 58.41, 88.07 | -103.95, 28.48 | 315.03, 7.91 | -62.87, -35.81 | in-in | in | 8.145 | Saltbr-in | 2.601 | HRD-in | -81.18, -54.27 | 77.68, -8.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.97 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.7, -176.11 | APE9-dihe-na | 95.21, 172.61 | APE8-dihe-in | -76.23, 133.32 | APE8-rot-in | 308.48 | APE67-dihe-in | -45.62, -25.89 | -46.72, -68.47 | APE12-dist-in | 11.519 | APE11-dist-in | 11.413 | APE10-dist-in | 5.954 | APE9-dist-in | 3.732 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | B | 342 | 324 | 7 | 0 | 0 | 3 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3KCFC | P36897 | 171 | 500 | 503.0 | JZO:3 | Type1.5_Back | Active | DFGin | 6.692 | 12.959 | BLAminus | -135.28, 165.04 | 69.33, 88.35 | -106.61, 31.51 | 302.0, 1.76 | -58.82, -55.68 | in-in | in | 8.036 | Saltbr-in | 2.379 | HRD-in | -81.96, -30.19 | 61.27, -12.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.897 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -114.43, -160.74 | APE9-dihe-na | 83.32, -178.05 | APE8-dihe-in | -94.01, 131.52 | APE8-rot-in | 317.12 | APE67-dihe-in | -41.44, -18.99 | -53.51, -67.7 | APE12-dist-in | 10.742 | APE11-dist-in | 11.842 | APE10-dist-in | 6.224 | APE9-dist-in | 3.856 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3KCFD | P36897 | 171 | 500 | 503.0 | JZO:4 | Type1.5_Back | Active | DFGin | 6.889 | 12.999 | BLAminus | -135.85, -173.78 | 57.12, 75.33 | -93.52, 22.15 | 298.91, 178.96 | -63.23, -14.31 | in-in | in | 8.264 | Saltbr-in | 2.894 | HRD-in | -62.47, -52.01 | 74.47, -2.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.771 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.66, 172.34 | APE9-dihe-na | 99.39, 173.59 | APE8-dihe-in | -80.33, 105.05 | APE8-rot-in | 316.25 | APE67-dihe-in | -46.61, -41.72 | -34.28, -49.6 | APE12-dist-in | 12.043 | APE11-dist-in | 12.05 | APE10-dist-in | 6.327 | APE9-dist-in | 4.044 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | D | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3KCFE | P36897 | 171 | 500 | 503.0 | JZO:5 | Type1.5_Back | Active | DFGin | 6.468 | 12.982 | BLAminus | -143.17, -179.95 | 57.87, 88.27 | -108.02, 21.93 | 307.67, 3.89 | -69.37, -7.25 | in-in | in | 8.028 | Saltbr-in | 2.856 | HRD-in | -68.17, -50.18 | 73.66, 3.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.902 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.74, 177.4 | APE9-dihe-na | 104.24, -175.74 | APE8-dihe-in | -89.11, 123.84 | APE8-rot-in | 292.33 | APE67-dihe-in | -50.81, -36.21 | -50.11, -48.46 | APE12-dist-in | 9.931 | APE11-dist-in | 12.001 | APE10-dist-in | 6.217 | APE9-dist-in | 3.796 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | E | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1B6CB | P36897 | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.851 | 13.394 | BLAminus | -130.85, -177.18 | 52.69, 80.31 | -95.42, 25.6 | 300.29, 176.12 | -64.72, -15.76 | in-out | in | 8.603 | Saltbr-out | 4.114 | HRD-in | -69.56, -62.44 | 85.43, -5.19 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.956 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.23, 170.19 | APE9-dihe-na | -45.35, 160.71 | APE8-dihe-in | -68.99, 127.88 | APE8-rot-in | 301.39 | APE67-dihe-in | -71.24, -15.17 | -60.4, -35.84 | APE12-dist-in | 11.453 | APE11-dist-out | 7.315 | APE10-dist-out | 8.448 | APE9-dist-in | 3.73 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | B | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1B6CD | P36897 | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.963 | 13.317 | BLAminus | -130.99, -177.26 | 52.75, 80.27 | -95.41, 25.6 | 300.53, 176.04 | -64.6, -15.85 | in-out | in | 8.6 | Saltbr-out | 4.115 | HRD-in | -69.77, -62.44 | 85.53, -5.06 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.958 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.35, 170.01 | APE9-dihe-na | -45.12, 160.61 | APE8-dihe-in | -69.1, 128.03 | APE8-rot-in | 301.09 | APE67-dihe-in | -71.13, -15.35 | -60.35, -36.04 | APE12-dist-in | 11.453 | APE11-dist-out | 7.314 | APE10-dist-out | 8.445 | APE9-dist-in | 3.725 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | D | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1B6CF | P36897 | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.998 | 13.814 | BLAminus | -130.93, -177.22 | 52.78, 80.13 | -95.35, 25.63 | 300.41, 176.19 | -64.73, -15.73 | in-out | in | 8.602 | Saltbr-out | 4.114 | HRD-in | -69.45, -62.52 | 85.59, -5.04 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.957 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.38, 170.18 | APE9-dihe-na | -45.27, 160.69 | APE8-dihe-in | -69.12, 128.05 | APE8-rot-in | 301.08 | APE67-dihe-in | -71.24, -15.27 | -60.51, -35.82 | APE12-dist-in | 11.454 | APE11-dist-out | 7.314 | APE10-dist-out | 8.445 | APE9-dist-in | 3.727 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | F | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1B6CH | P36897 | 175 | 500 | 503.0 | No_ligand | No_ligand | Inactive | DFGin | 6.933 | 13.373 | BLAminus | -131.03, -177.2 | 52.83, 80.24 | -95.22, 25.39 | 300.35, 176.04 | -64.71, -15.81 | in-out | in | 8.601 | Saltbr-out | 4.113 | HRD-in | -69.67, -62.6 | 85.56, -5.13 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.956 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -139.24, 170.15 | APE9-dihe-na | -45.32, 160.68 | APE8-dihe-in | -69.01, 127.87 | APE8-rot-in | 301.38 | APE67-dihe-in | -71.25, -15.25 | -60.38, -35.9 | APE12-dist-in | 11.451 | APE11-dist-out | 7.311 | APE10-dist-out | 8.446 | APE9-dist-in | 3.729 | None | None | None | XRAY | 2.6 | 0.249 | 0.269 | H | 342 | 326 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1b6c | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1RW8A | P36897 | 200 | 500 | 503.0 | 580:501 | Type1 | Inactive | DFGin | 6.023 | 12.845 | BLAminus | -123.87, -176.48 | 52.01, 78.57 | -101.69, 16.55 | 307.13, 6.03 | -62.1, -24.92 | in-in | in | 7.841 | Saltbr-in | 3.467 | HRD-in | -69.23, -61.02 | 80.12, 4.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.902 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioi | APE10-dihe-na | -83.25, -151.65 | APE9-dihe-na | -88.81, -163.17 | APE8-dihe-in | -80.66, 118.18 | APE8-rot-in | 309.35 | APE67-dihe-in | -55.07, -38.39 | -52.69, -43.2 | APE12-dist-in | 11.486 | APE11-dist-in | 8.854 | APE10-dist-out | 8.62 | APE9-dist-in | 4.107 | None | None | None | XRAY | 2.4 | 0.26 | 0.291 | A | 301 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1rw8 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1PY5A | P36897 | 200 | 500 | 503.0 | PY1:700 | Type1 | Inactive | DFGin | 6.325 | 13.096 | BLAminus | -139.22, -176.23 | 51.49, 62.68 | -91.32, 17.81 | 306.9, 168.43 | -57.65, -31.73 | in-in | in | 7.831 | Saltbr-in | 2.897 | HRD-in | -74.07, -48.58 | 75.5, -7.56 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.862 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iioi | APE10-dihe-na | -82.55, -147.04 | APE9-dihe-na | -97.21, -166.02 | APE8-dihe-in | -77.65, 124.21 | APE8-rot-in | 307.07 | APE67-dihe-in | -64.31, -27.94 | -63.63, -30.26 | APE12-dist-in | 11.444 | APE11-dist-in | 8.66 | APE10-dist-out | 8.572 | APE9-dist-in | 4.119 | None | None | None | XRAY | 2.3 | 0.26 | 0.292 | A | 326 | 301 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 1py5 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.1e-85 | 291.4 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 2X7OB | P36897 | 171 | 500 | 503.0 | ZOP:600 | Type1 | Inactive | DFGin | 6.858 | 13.746 | BLAminus | -128.22, 169.83 | 59.7, 88.26 | -108.23, 28.26 | 289.27, 149.16 | -69.33, -30.83 | in-out | in | 8.118 | Saltbr-out | 3.833 | HRD-in | -65.55, -40.47 | 69.31, -25.99 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.059 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.06, 149.04 | APE9-dihe-na | 97.27, -171.94 | APE8-dihe-in | -74.39, 131.11 | APE8-rot-in | 314.97 | APE67-dihe-in | -65.1, -35.09 | -61.66, -32.49 | APE12-dist-in | 11.793 | APE11-dist-in | 11.793 | APE10-dist-in | 5.967 | APE9-dist-in | 4.727 | None | None | None | XRAY | 3.7 | 0.267 | 0.273 | B | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 2x7o | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3FAAC | P36897 | 171 | 500 | 503.0 | 55F:601 | Type1 | Inactive | DFGin | 6.142 | 13.141 | BLAminus | -126.27, 176.42 | 50.71, 78.49 | -102.58, 30.06 | 320.3, 19.34 | -66.31, -17.95 | in-in | in | 7.99 | Saltbr-in | 2.662 | HRD-in | -67.56, -21.99 | 46.1, 19.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.947 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -120.66, 131.05 | APE9-dihe-na | 148.7, 175.0 | APE8-dihe-in | -102.93, 87.73 | APE8-rot-in | 305.5 | APE67-dihe-out | -28.83, -55.82 | 5.18, -84.04 | APE12-dist-in | 11.481 | APE11-dist-in | 12.149 | APE10-dist-in | 6.247 | APE9-dist-in | 4.208 | None | None | None | XRAY | 3.35 | 0.228 | 0.271 | C | 342 | 330 | 0 | 0 | 0 | 0 | [[205, 494]] | 1.0 | 3faa | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 1VJYA | P36897 | 201 | 503 | 503.0 | 460:999 | Type1 | None | DFGin | 6.095 | 12.796 | BLAminus | -131.96, -168.3 | 46.73, 72.17 | -95.27, 7.02 | 307.89, 4.49 | -49.86, -32.3 | in-in | in | 7.726 | Saltbr-in | 2.753 | HRD-in | -71.95, -49.94 | 73.94, 4.16 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.848 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -108.72, 178.34 | APE9-dihe-na | 100.08, -177.16 | APE8-dihe-in | -88.48, 114.15 | APE8-rot-in | 304.07 | APE67-dihe-in | -56.76, -36.75 | -44.55, -45.61 | APE12-dist-none | 999.0 | APE11-dist-in | 11.557 | APE10-dist-in | 6.513 | APE9-dist-in | 3.865 | None | None | None | XRAY | 2.0 | 0.223 | 0.275 | A | 303 | 299 | 4 | 0 | 0 | 4 | [[205, 494]] | 1.0 | 1vjy | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3GXLA | P36897 | 201 | 498 | 503.0 | QIG:60999 | Type1 | None | DFGin | 5.986 | 13.162 | BLAminus | -117.01, -170.6 | 33.6, 86.88 | -102.63, 15.85 | 311.96, 176.51 | -62.1, -23.52 | in-in | in | 8.223 | Saltbr-in | 2.93 | HRD-in | -71.35, -53.37 | 77.01, 1.76 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.958 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -62.74, 167.86 | APE9-dihe-na | 117.67, 172.21 | APE8-dihe-in | -83.62, 118.05 | APE8-rot-in | 304.44 | APE67-dihe-in | -50.23, -35.35 | -45.35, -55.49 | APE12-dist-none | 999.0 | APE11-dist-in | 12.158 | APE10-dist-in | 6.739 | APE9-dist-in | 4.173 | None | None | None | XRAY | 1.8 | 0.228 | 0.263 | A | 303 | 285 | 13 | 0 | 0 | 5 | [[205, 494]] | 1.0 | 3gxl | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3HMMA | P36897 | 201 | 498 | 503.0 | 855:60857 | Type1 | None | DFGin | 6.119 | 13.049 | BLAminus | -127.07, -168.91 | 53.99, 65.82 | -94.96, 13.15 | 305.68, 3.69 | -60.53, -23.27 | in-in | in | 8.024 | Saltbr-in | 2.812 | HRD-in | -74.05, -51.32 | 76.01, -1.97 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.934 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -160.63 | APE8-dihe-in | -79.78, 120.6 | APE8-rot-in | 300.84 | APE67-dihe-in | -55.11, -37.41 | -48.22, -47.79 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.917 | None | None | None | XRAY | 1.7 | 0.223 | 0.241 | A | 303 | 293 | 5 | 0 | 0 | 5 | [[205, 494]] | 1.0 | 3hmm | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.1e-85 | 291.8 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 9J9DA | P36897 | 202 | 502 | 503.0 | A1L30:701 | Type1 | None | DFGin | 5.967 | 12.455 | BLAminus | -128.65, -173.5 | 51.95, 67.83 | -91.44, 10.62 | 307.73, 2.77 | -64.11, -26.42 | in-in | in | 8.02 | Saltbr-in | 2.807 | HRD-in | -76.64, -51.57 | 79.18, -0.61 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.92 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -92.35, -34.47 | APE9-dihe-na | -89.02, -159.15 | APE8-dihe-in | -77.18, 122.97 | APE8-rot-in | 307.18 | APE67-dihe-in | -57.12, -34.57 | -60.97, -41.48 | APE12-dist-none | 999.0 | APE11-dist-in | 12.145 | APE10-dist-in | 6.163 | APE9-dist-in | 4.067 | None | None | None | XRAY | 1.337 | 0.191 | 0.209 | A | 306 | 296 | 5 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 9j9d | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TGFR1_HUMAN | 3TZMA | P36897 | 200 | 496 | 503.0 | 085:1 | Type1 | None | DFGin | 6.065 | 13.106 | BLAminus | -122.58, -169.81 | 59.22, 59.29 | -91.38, 11.48 | 304.6, 5.41 | -64.05, -23.93 | in-in | in | 7.963 | Saltbr-in | 2.833 | HRD-in | -81.31, -50.79 | 80.1, -5.96 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.968 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -87.36, 160.54 | APE9-dihe-na | 102.22, -177.2 | APE8-dihe-in | -87.37, 126.2 | APE8-rot-in | 298.62 | APE67-dihe-in | -59.36, -31.96 | -58.47, -41.28 | APE12-dist-none | 999.0 | APE11-dist-in | 12.238 | APE10-dist-in | 6.184 | APE9-dist-in | 3.825 | None | None | None | XRAY | 1.7 | 0.172 | 0.205 | A | 309 | 295 | 2 | 0 | 0 | 2 | [[205, 494]] | 1.0 | 3tzm | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.4e-85 | 291.7 | 3 | 266 | 264 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|