| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CDK8 | AF-P49336-K1A | P49336 | 12 | 343 | 464.0 | No_ligand | No_ligand | Active | DFGin | 6.9313 | 15.6629 | BLAminus | -128.17, 177.28 | 55.68, 59.43 | -72.54, 15.56 | 300.04, 114.68 | -62.04, -32.39 | in-in | in | 9.1654 | Saltbr-in | 2.8975 | HRD-in | -73.5, -51.19 | 62.86, 10.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8327 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.05, 164.39 | APE9-dihe-na | 83.32, 124.4 | APE8-dihe-in | -52.27, 134.37 | APE8-rot-in | 287.61 | APE67-dihe-in | -65.17, -26.48 | -44.23, -41.35 | APE12-dist-in | 12.0588 | APE11-dist-in | 11.607 | APE10-dist-in | 5.8083 | APE9-dist-in | 3.4091 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 332.0 | 332.0 | 0 | 31 | 31 | 0 | [[22, 335]] | 1.0 | AF-P49336-K1 | CMGC_CDK8_HUMAN | CMGC | 2.9e-82 | 282.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | AF-P49336-K3A | P49336 | 12 | 343 | 464.0 | No_ligand | No_ligand | Active | DFGin | 7.0585 | 14.4146 | BLAminus | -125.11, 179.05 | 58.06, 66.16 | -75.42, 13.63 | 298.43, 116.53 | -58.59, -38.0 | in-in | in | 9.222 | Saltbr-in | 2.7201 | HRD-in | -77.81, -49.38 | 63.32, 9.66 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8729 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.07, 166.88 | APE9-dihe-na | 60.71, 128.33 | APE8-dihe-in | -54.75, 135.42 | APE8-rot-in | 297.36 | APE67-dihe-in | -67.37, -15.46 | -44.59, -50.0 | APE12-dist-in | 12.5614 | APE11-dist-in | 10.811 | APE10-dist-in | 6.5807 | APE9-dist-in | 3.286 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 332.0 | 332.0 | 0 | 31 | 31 | 0 | [[22, 335]] | 1.0 | AF-P49336-K3 | CMGC_CDK8_HUMAN | CMGC | 2.9e-82 | 282.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5HBJA | P49336 | 1 | 361 | 464.0 | 5Y8:60401 | Type1 | Inactive | DFGin | 7.5418 | 14.7786 | BLAminus | -106.87, 176.98 | 71.07, 89.31 | -114.96, 61.9 | 305.41, 118.79 | -100.84, -170.16 | in-in | in | 9.7609 | Saltbr-in | 2.6824 | HRD-in | -77.67, -52.92 | 73.2, 5.3 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -16.09 | APE8-dihe-in | -117.57, 98.85 | APE8-rot-in | 304.83 | APE67-dihe-in | -72.47, -22.93 | -102.77, 29.67 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.3779 | None | None | None | XRAY | 3.0 | 999.0 | 0.288 | A | 364.0 | 340.0 | 21 | 31 | 19 | 12 | [[22, 335]] | 1.0 | 5hbj | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5ICPA | P49336 | 1 | 362 | 464.0 | 69Z:60401 | Type1 | Inactive | DFGin | 6.1473 | 13.6394 | BLAminus | -129.39, 179.13 | 50.41, 56.76 | -66.42, 4.81 | 256.2, 78.89 | 56.91, 53.37 | in-in | in | 9.1898 | Saltbr-in | 2.5875 | HRD-in | -78.65, -54.95 | 77.97, -2.02 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7892 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, 83.07 | APE9-dihe-na | -127.02, 140.47 | APE8-dihe-in | -112.3, 142.07 | APE8-rot-out | 57.72 | APE67-dihe-in | -65.52, -25.52 | -110.98, 18.82 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.6843 | APE9-dist-out | 12.5091 | None | None | None | XRAY | 2.18 | 0.185 | 0.216 | A | 364.0 | 343.0 | 19 | 31 | 23 | 8 | [[22, 335]] | 1.0 | 5icp | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5IDNA | P49336 | 1 | 363 | 464.0 | 6A7:60401 | Type1 | Inactive | DFGin | 7.3226 | 16.0877 | BLAminus | -124.47, 174.0 | 67.51, 75.48 | -91.55, 21.99 | 294.62, 123.1 | -96.7, 0.53 | in-in | in | 8.9702 | Saltbr-in | 2.647 | HRD-in | -71.0, -49.83 | 80.54, -0.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.4045 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 147.78 | APE8-dihe-in | -125.68, 150.04 | APE8-rot-out | 46.55 | APE67-dihe-in | -67.71, -25.83 | -125.87, 33.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.7732 | None | None | None | XRAY | 2.26 | 0.221 | 0.253 | A | 370.0 | 336.0 | 27 | 31 | 15 | 16 | [[22, 335]] | 1.0 | 5idn | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5XQXA | P49336 | 1 | 362 | 464.0 | 8CC:60402 | Type1 | Inactive | DFGin | 7.1009 | 13.3766 | BLAminus | -124.76, 173.54 | 67.85, 87.06 | -93.65, 13.06 | 285.44, 142.36 | -53.92, -30.2 | in-in | in | 8.5993 | Saltbr-in | 2.6458 | HRD-in | -76.07, -52.85 | 74.84, 2.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.797 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -162.45 | APE8-dihe-in | -121.89, 118.59 | APE8-rot-in | 276.05 | APE67-dihe-in | -59.33, -23.95 | -109.46, 21.35 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.0086 | None | None | None | XRAY | 2.3 | 0.19 | 0.222 | A | 380.0 | 337.0 | 25 | 31 | 18 | 13 | [[22, 335]] | 1.0 | 5xqx | CMGC_CDK8_HUMAN | CMGC | 4.7e-82 | 281.6 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5XS2A | P49336 | 1 | 363 | 464.0 | 8D6:60402 | Type1 | Inactive | DFGin | 7.1 | 13.2185 | BLAminus | -125.86, 168.92 | 68.44, 89.08 | -85.59, 13.7 | 295.46, 132.91 | -57.29, -23.08 | in-in | in | 8.5472 | Saltbr-in | 2.6849 | HRD-in | -77.09, -53.4 | 74.45, 0.97 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7249 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -119.34, 129.98 | APE9-dihe-na | -115.73, -15.25 | APE8-dihe-in | -128.4, 144.08 | APE8-rot-out | 53.94 | APE67-dihe-in | -59.75, -24.05 | -125.87, 25.67 | APE12-dist-in | 7.1385 | APE11-dist-in | 11.8021 | APE10-dist-out | 9.8465 | APE9-dist-out | 12.3679 | None | None | None | XRAY | 2.04 | 0.197 | 0.225 | A | 380.0 | 363.0 | 0 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 5xs2 | CMGC_CDK8_HUMAN | CMGC | 4.7e-82 | 281.6 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 6QTJA | P49336 | 1 | 359 | 464.0 | JHK:60501 | Type1 | Inactive | DFGin | 7.5864 | 14.0745 | BLAminus | -112.22, -179.25 | 62.71, 86.71 | -102.98, 13.61 | 301.92, 111.63 | -83.54, 3.25 | in-in | in | 8.4612 | Saltbr-in | 2.9368 | HRD-in | -68.14, -49.62 | 76.51, -6.19 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -45.96 | APE8-dihe-in | -121.23, 128.93 | APE8-rot-in | 272.12 | APE67-dihe-in | -58.17, -25.47 | -117.92, 17.96 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.2357 | None | None | None | XRAY | 2.48 | 0.187 | 0.22 | A | 405.0 | 329.0 | 30 | 31 | 13 | 18 | [[22, 335]] | 1.0 | 6qtj | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 9H8CA | P49336 | 1 | 361 | 464.0 | A1IS8:60503 | Type1 | Inactive | DFGin | 7.5455 | 14.2354 | BLAminus | -123.76, 163.44 | 68.83, 82.68 | -94.14, 12.47 | 302.05, 120.29 | -95.45, 18.7 | in-in | in | 8.8322 | Saltbr-in | 2.6869 | HRD-in | -71.9, -45.8 | 76.46, -12.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8362 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 1.06 | APE8-dihe-in | -111.33, 130.78 | APE8-rot-in | 270.85 | APE67-dihe-in | -58.13, -22.76 | -124.23, 26.3 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.0634 | None | None | None | XRAY | 2.573 | 0.192 | 0.262 | A | 414.0 | 336.0 | 25 | 31 | 16 | 15 | [[22, 335]] | 1.0 | 9h8c | CMGC_CDK8_HUMAN | CMGC | 6.3e-82 | 281.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 9H8SA | P49336 | 1 | 362 | 464.0 | A1ITF:60509 | Type1 | Inactive | DFGin | 7.3437 | 13.9243 | BLAminus | -119.28, 163.44 | 74.84, 82.25 | -92.61, 11.91 | 298.93, 132.0 | -87.41, 10.8 | in-in | in | 8.6117 | Saltbr-in | 2.6241 | HRD-in | -75.25, -51.5 | 79.06, -6.52 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6589 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 160.05 | APE8-rot-out | 75.96 | APE67-dihe-in | -54.19, -23.95 | -111.96, 19.45 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.157 | 0.197 | 0.248 | A | 414.0 | 335.0 | 27 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 9h8s | CMGC_CDK8_HUMAN | CMGC | 6.3e-82 | 281.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 8TQ2A | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 5.9534 | 13.4093 | BLAplus | -149.38, -174.61 | 57.66, 42.3 | -94.56, 56.63 | 80.28, 25.13 | -65.65, -33.03 | in-out | in | 9.074 | Saltbr-out | 5.0175 | HRD-in | -71.17, -43.38 | 62.04, 12.67 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.9073 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -111.63, -27.07 | APE9-dihe-na | -152.97, 160.77 | APE8-dihe-in | -61.74, 149.93 | APE8-rot-out | 187.22 | APE67-dihe-in | -65.55, -27.76 | -65.32, -15.56 | APE12-dist-in | 13.0056 | APE11-dist-in | 10.6044 | APE10-dist-in | 7.3395 | APE9-dist-in | 4.2314 | None | None | None | EM | 3.8 | 999.0 | 999.0 | A | 464.0 | 313.0 | 46 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 8tq2 | CMGC_CDK8_HUMAN | CMGC | 9.1e-82 | 280.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 8TQCA | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 5.954 | 13.4098 | BLAplus | -149.38, -174.65 | 57.7, 42.3 | -94.58, 56.63 | 80.22, 25.15 | -65.67, -33.03 | in-out | in | 9.0736 | Saltbr-out | 5.0166 | HRD-in | -71.16, -43.39 | 62.07, 12.66 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.9071 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -111.64, -27.07 | APE9-dihe-na | -152.99, 160.74 | APE8-dihe-in | -61.68, 149.91 | APE8-rot-out | 187.24 | APE67-dihe-in | -65.64, -27.68 | -65.36, -15.51 | APE12-dist-in | 13.006 | APE11-dist-in | 10.6041 | APE10-dist-in | 7.3394 | APE9-dist-in | 4.2313 | None | None | None | EM | 3.8 | 999.0 | 999.0 | A | 464.0 | 313.0 | 46 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 8tqc | CMGC_CDK8_HUMAN | CMGC | 9.1e-82 | 280.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 8TQWA | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9194 | 11.7033 | BLAplus | -136.58, -174.19 | 58.52, 55.8 | -94.53, 48.46 | 79.76, 124.7 | -72.57, -22.17 | in-out | in | 9.013 | Saltbr-out | 4.2612 | HRD-in | -69.7, -41.94 | 60.18, 16.8 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.2241 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -107.3, -18.61 | APE9-dihe-na | -153.74, 161.23 | APE8-dihe-in | -65.82, 153.77 | APE8-rot-out | 180.15 | APE67-dihe-in | -67.85, -29.18 | -70.07, -16.17 | APE12-dist-in | 12.7643 | APE11-dist-in | 10.6621 | APE10-dist-in | 7.0853 | APE9-dist-in | 4.3173 | None | None | None | EM | 8.2 | 999.0 | 999.0 | a | 464.0 | 313.0 | 46 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 8tqw | CMGC_CDK8_HUMAN | CMGC | 9.1e-82 | 280.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4G6LA | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 7.7821 | 13.1649 | BLBminus | -140.33, 170.43 | 60.07, 39.76 | -65.01, 139.84 | 287.11, 130.96 | -72.68, 84.6 | in-in | in | 9.41 | Saltbr-in | 2.7316 | HRD-in | -90.39, -58.08 | 80.12, -10.69 | in-out-none | SNCion | out-none | ActLoopNT-out | 8.7909 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.75, -20.61 | 999.0, 14.23 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.214 | 0.266 | A | 406.0 | 333.0 | 26 | 31 | 19 | 12 | [[22, 335]] | 1.0 | 4g6l | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5FGKA | P49336 | 1 | 362 | 464.0 | 5XG:60401 | Type1 | Inactive | DFGin | 8.4978 | 15.5831 | BLBminus | -133.54, 169.31 | 57.53, 42.29 | -55.85, 144.8 | 295.15, 85.37 | -70.31, 91.66 | in-in | in | 9.829 | Saltbr-in | 2.8534 | HRD-in | -79.53, -56.66 | 86.65, -4.01 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 157.88 | APE8-dihe-in | -124.66, 135.5 | APE8-rot-in | 267.49 | APE67-dihe-in | -66.95, -24.09 | -119.64, 24.09 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.9461 | None | None | None | XRAY | 2.36 | 999.0 | 0.237 | A | 364.0 | 331.0 | 31 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 5fgk | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5HBEA | P49336 | 1 | 361 | 464.0 | 5Y6:60401 | Type1 | Inactive | DFGin | 6.3817 | 13.4796 | BLBminus | -150.55, 174.93 | 54.88, 46.99 | -64.39, 138.78 | 282.35, 68.64 | -73.7, 83.07 | in-in | in | 9.4752 | Saltbr-in | 2.6635 | HRD-in | -80.78, -53.55 | 75.81, 1.36 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.0331 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 124.46 | APE8-dihe-in | -128.69, 136.48 | APE8-rot-out | 167.77 | APE67-dihe-in | -66.35, -22.41 | -120.15, 22.04 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.377 | None | None | None | XRAY | 2.38 | 0.23 | 0.256 | A | 364.0 | 343.0 | 18 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 5hbe | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5HNBA | P49336 | 1 | 359 | 464.0 | 62M:60401 | Type1 | Inactive | DFGin | 6.6498 | 13.1706 | BLBminus | -138.74, 167.16 | 57.27, 44.77 | -53.04, 139.99 | 284.36, 64.87 | -77.11, 80.76 | in-in | in | 9.3522 | Saltbr-in | 2.6998 | HRD-in | -81.89, -52.43 | 75.49, 2.56 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8745 | ActLoopCT-out | nonTYR | APEdihe_aanio | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 22.41 | APE8-rot-in | 326.4 | APE67-dihe-out | -68.33, -25.9 | 68.06, 1.32 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.35 | 0.218 | 0.252 | A | 370.0 | 339.0 | 20 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 5hnb | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5I5ZA | P49336 | 1 | 362 | 464.0 | 68U:60401 | Type1 | Inactive | DFGin | 6.4155 | 13.0643 | BLBminus | -146.19, 175.23 | 51.04, 37.29 | -51.44, 128.07 | 281.53, 66.91 | -69.5, 65.99 | in-in | in | 9.1148 | Saltbr-in | 2.9017 | HRD-in | -79.94, -54.75 | 78.35, 1.56 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7902 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 116.55 | APE8-rot-out | 180.69 | APE67-dihe-in | -62.72, -27.98 | -92.64, 5.94 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.6 | 0.239 | 0.274 | A | 370.0 | 342.0 | 20 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 5i5z | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5IDPA | P49336 | 1 | 359 | 464.0 | 6A6:60401 | Type1 | Inactive | DFGin | 6.659 | 13.1177 | BLBminus | -136.27, 172.07 | 59.2, 45.18 | -61.59, 132.52 | 281.19, 68.65 | -74.88, 80.04 | in-in | in | 9.3926 | Saltbr-in | 2.8965 | HRD-in | -79.39, -54.81 | 77.61, 1.02 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6935 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 164.27 | APE8-rot-out | 60.39 | APE67-dihe-in | -68.82, -22.92 | -114.95, 18.44 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.65 | 0.232 | 0.272 | A | 370.0 | 341.0 | 18 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 5idp | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F7SA | P49336 | 1 | 359 | 464.0 | 0SW:60501 | Type1 | Inactive | DFGin | 6.495 | 13.0688 | BLBminus | -136.61, 176.12 | 53.35, 42.37 | -54.98, 136.0 | 280.12, 74.29 | -77.21, 78.52 | in-in | in | 9.2294 | Saltbr-in | 2.7473 | HRD-in | -79.34, -55.77 | 76.41, 2.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7597 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 131.9 | APE8-rot-out | 180.5 | APE67-dihe-in | -68.08, -24.25 | -110.68, 14.48 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.2 | 0.194 | 0.222 | A | 405.0 | 339.0 | 20 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 4f7s | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5BNJA | P49336 | 1 | 362 | 464.0 | 4TV:60501 | Type1 | Inactive | DFGin | 6.1998 | 14.6125 | BLBminus | -127.23, 163.17 | 60.48, 55.04 | -65.81, 148.47 | 290.88, 72.47 | -70.37, 93.4 | in-in | in | 9.8117 | Saltbr-in | 2.7276 | HRD-in | -79.48, -50.1 | 76.1, -2.58 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.736 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 162.07 | APE8-rot-out | 56.78 | APE67-dihe-in | -68.21, -22.51 | -112.22, 14.37 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.64 | 0.228 | 0.273 | A | 405.0 | 341.0 | 21 | 31 | 20 | 11 | [[22, 335]] | 1.0 | 5bnj | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 6QTGA | P49336 | 1 | 359 | 464.0 | JH8:60501 | Type1 | Inactive | DFGin | 6.8548 | 13.5978 | BLBminus | -115.69, 168.8 | 67.93, 119.69 | -128.98, 119.87 | 314.23, 115.38 | -156.88, 999.0 | in-in | in | 8.458 | Saltbr-in | 2.9444 | HRD-in | -69.43, -47.54 | 81.38, -19.97 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -47.73 | APE8-dihe-in | -122.24, 124.81 | APE8-rot-in | 266.36 | APE67-dihe-in | -67.96, -18.93 | -113.56, 25.73 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.0679 | None | None | None | XRAY | 2.7 | 0.202 | 0.231 | A | 405.0 | 328.0 | 31 | 31 | 12 | 19 | [[22, 335]] | 1.0 | 6qtg | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4CRLA | P49336 | 1 | 359 | 464.0 | C1I:61360 | Type1 | Inactive | DFGin | 6.2635 | 12.9653 | BLBminus | -130.84, 167.17 | 41.28, 61.34 | -57.58, 143.29 | 285.19, 53.46 | -56.15, 77.43 | in-in | in | 9.2784 | Saltbr-in | 2.7647 | HRD-in | -77.87, -48.76 | 70.82, 12.4 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8293 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -12.95 | APE8-dihe-in | -65.77, 114.52 | APE8-rot-out | 186.25 | APE67-dihe-in | -70.31, -18.88 | -108.2, 7.99 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.3551 | None | None | None | XRAY | 2.4 | 0.201 | 0.256 | A | 406.0 | 336.0 | 23 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 4crl | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5CEIA | P49336 | 1 | 362 | 464.0 | 50R:60508 | Type1 | Inactive | DFGin | 6.4332 | 13.0148 | BLBminus | -132.66, 174.92 | 55.78, 44.71 | -56.21, 137.6 | 280.16, 70.73 | -77.01, 72.68 | in-in | in | 9.2797 | Saltbr-in | 2.5792 | HRD-in | -79.82, -54.28 | 77.75, 0.99 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6632 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 169.41 | APE8-rot-out | 67.16 | APE67-dihe-in | -60.87, -22.55 | -115.47, 18.61 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.24 | 0.175 | 0.227 | A | 406.0 | 344.0 | 18 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 5cei | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 6R3SA | P49336 | 1 | 362 | 464.0 | JRE:60501 | Type1 | Inactive | DFGin | 6.4489 | 13.1166 | BLBminus | -136.26, 169.85 | 57.34, 42.45 | -52.43, 144.8 | 287.58, 63.16 | -78.12, 79.2 | in-in | in | 9.3756 | Saltbr-in | 2.8296 | HRD-in | -80.26, -51.73 | 75.92, 4.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6882 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 130.83 | APE8-rot-out | 181.78 | APE67-dihe-in | -67.95, -25.35 | -103.82, 11.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.19 | 0.202 | 0.227 | A | 406.0 | 343.0 | 19 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 6r3s | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 6Y0AA | P49336 | 1 | 362 | 464.0 | JRE:60501 | Type1 | Inactive | DFGin | 6.4489 | 13.1166 | BLBminus | -136.26, 169.85 | 57.34, 42.45 | -52.43, 144.8 | 287.58, 63.16 | -78.12, 79.2 | in-in | in | 9.3756 | Saltbr-in | 2.8296 | HRD-in | -80.26, -51.73 | 75.92, 4.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6882 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 130.83 | APE8-rot-out | 181.78 | APE67-dihe-in | -67.95, -25.35 | -103.82, 11.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.19 | 0.202 | 0.227 | A | 406.0 | 343.0 | 19 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 6y0a | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 6T41A | P49336 | 1 | 359 | 464.0 | MFE:60501 | Type1 | Inactive | DFGin | 8.6301 | 13.5154 | BLBminus | -130.72, 167.87 | 65.4, 35.77 | -47.77, 142.68 | 290.97, 94.77 | -79.52, 87.36 | in-in | in | 9.2255 | Saltbr-in | 2.9666 | HRD-in | -82.44, -61.41 | 81.57, -4.44 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8749 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 161.03 | APE8-rot-out | 58.35 | APE67-dihe-in | -69.81, -18.57 | -101.28, 19.75 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.45 | 0.185 | 0.256 | A | 407.0 | 343.0 | 16 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 6t41 | CMGC_CDK8_HUMAN | CMGC | 6e-82 | 281.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5HBHA | P49336 | 1 | 361 | 464.0 | 5Y7:60401 | Type1 | Inactive | DFGin | 5.4841 | 13.3356 | BLBplus | -129.14, 169.91 | 65.09, 34.73 | -89.33, 139.59 | 54.15, 87.69 | 88.57, 16.73 | in-in | in | 9.1442 | Saltbr-in | 2.8415 | HRD-in | -73.61, -55.97 | 88.78, -11.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.6525 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, 146.42 | APE9-dihe-na | -93.82, 144.5 | APE8-dihe-in | -120.03, 143.32 | APE8-rot-out | 75.1 | APE67-dihe-in | -65.56, -22.05 | -107.02, 22.5 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.8418 | APE9-dist-out | 12.1846 | None | None | None | XRAY | 2.5 | 0.235 | 0.268 | A | 364.0 | 334.0 | 27 | 31 | 17 | 14 | [[22, 335]] | 1.0 | 5hbh | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 3RGFA | P49336 | 1 | 353 | 464.0 | BAX:60465 | Type2 | Inactive | DFGout | 15.0897 | 10.8645 | BBAminus | -128.79, 167.92 | -135.88, 84.21 | -83.29, -7.22 | 304.7, 18.84 | -121.06, 44.25 | in-out | in | 9.3695 | Saltbr-out | 4.8518 | HRD-in | -76.1, -55.23 | 78.73, 2.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 12.2242 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 133.12 | APE8-dihe-in | -111.84, 132.17 | APE8-rot-out | 185.32 | APE67-dihe-in | -67.42, -19.98 | -109.35, 18.38 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.6368 | None | None | None | XRAY | 2.2 | 0.183 | 0.221 | A | 405.0 | 319.0 | 34 | 31 | 15 | 16 | [[22, 335]] | 1.0 | 3rgf | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F6UA | P49336 | 1 | 359 | 464.0 | 0SR:60501 | Type2 | Inactive | DFGout | 14.5288 | 8.1472 | BBAminus | -137.04, 173.39 | -132.48, 97.94 | -82.11, -23.16 | 303.07, 124.54 | 89.51, -145.66 | in-in | in | 8.5274 | Saltbr-in | 2.6265 | HRD-in | -75.69, -54.68 | 80.97, 0.65 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnio | APE10-dihe-na | 999.0, -48.5 | APE9-dihe-na | -168.88, 136.11 | APE8-dihe-in | -116.43, 154.29 | APE8-rot-out | 81.86 | APE67-dihe-in | -65.37, -20.81 | -106.87, 16.32 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 7.2334 | APE9-dist-out | 10.9418 | None | None | None | XRAY | 2.1 | 0.177 | 0.198 | A | 405.0 | 332.0 | 27 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 4f6u | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F6WA | P49336 | 1 | 359 | 464.0 | 0SS:60501 | Type2 | Inactive | DFGout | 17.0447 | 13.9468 | BBAminus | -134.04, 175.74 | -149.99, 134.58 | -80.54, -17.82 | 302.37, 168.31 | 89.71, 32.24 | in-in | in | 8.5227 | Saltbr-in | 2.6647 | HRD-in | -81.35, -56.06 | 84.43, -4.37 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 94.48 | APE8-rot-in | 298.45 | APE67-dihe-in | -64.37, -22.4 | -100.8, 19.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.39 | 0.193 | 0.234 | A | 405.0 | 330.0 | 29 | 31 | 13 | 18 | [[22, 335]] | 1.0 | 4f6w | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F7LA | P49336 | 1 | 359 | 464.0 | 0SO:60501 | Type2 | Inactive | DFGout | 13.5433 | 10.487 | BBAminus | -144.39, 166.94 | -130.48, 125.05 | -101.12, -66.88 | 314.21, 89.91 | 174.94, 999.0 | in-in | in | 9.0525 | Saltbr-in | 2.7304 | HRD-in | -72.87, -46.64 | 81.38, -4.09 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 155.76 | APE8-rot-out | 66.51 | APE67-dihe-in | -72.52, -24.41 | -123.27, 25.01 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.9 | 0.226 | 0.27 | A | 405.0 | 326.0 | 33 | 31 | 11 | 20 | [[22, 335]] | 1.0 | 4f7l | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F7NA | P49336 | 1 | 361 | 464.0 | 0SV:60501 | Type2 | Inactive | DFGout | 14.194 | 8.2102 | BBAminus | -139.77, 176.54 | -136.01, 97.7 | -86.48, -26.06 | 306.23, 126.32 | 100.15, -136.94 | in-in | in | 8.7798 | Saltbr-in | 2.7862 | HRD-in | -78.13, -54.62 | 75.98, 5.37 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnio | APE10-dihe-na | 999.0, 43.71 | APE9-dihe-na | -114.3, 132.58 | APE8-dihe-in | -127.74, 146.12 | APE8-rot-out | 68.03 | APE67-dihe-in | -66.61, -22.51 | -99.38, 17.25 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 5.8201 | APE9-dist-out | 11.2715 | None | None | None | XRAY | 2.65 | 0.2 | 0.228 | A | 405.0 | 333.0 | 28 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 4f7n | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 5HVYA | P49336 | 1 | 359 | 464.0 | 66X:60501 | Type2 | Inactive | DFGout | 15.175 | 9.3117 | BBAminus | -147.75, 175.04 | -130.64, 103.81 | -80.2, 9.83 | 305.77, 118.03 | 84.07, 29.62 | out-out | out | 11.2669 | Saltbr-out | 6.1116 | HRD-in | -85.57, -56.75 | 82.18, -2.99 | out-out-out | SNCooo | out-out | ActLoopNT-out | 12.8606 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oioo | APE10-dihe-na | -86.7, 132.16 | APE9-dihe-na | -171.76, 167.74 | APE8-dihe-in | -116.95, 139.23 | APE8-rot-out | 61.83 | APE67-dihe-in | -58.0, -28.58 | -98.28, 0.53 | APE12-dist-out | 14.3713 | APE11-dist-in | 9.0319 | APE10-dist-out | 8.2992 | APE9-dist-out | 10.3787 | None | None | None | XRAY | 2.39 | 0.181 | 0.22 | A | 406.0 | 333.0 | 26 | 31 | 19 | 12 | [[22, 335]] | 1.0 | 5hvy | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 6TPAA | P49336 | 1 | 359 | 464.0 | NZ8:60501,NZ5:60505,NZ5:60506,NZ5:60507 | Type2,Allosteric,Allosteric,Allosteric | Inactive | DFGout | 13.8318 | 11.8175 | BBAminus | -130.48, -178.36 | -144.36, 91.14 | -84.2, -4.16 | 322.15, 13.04 | -124.91, 44.75 | out-out | out | 10.1823 | Saltbr-out | 4.9546 | HRD-in | -82.95, -50.83 | 78.95, 15.78 | out-out-out | SNCooo | out-out | ActLoopNT-out | 11.9075 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 123.19 | APE8-rot-out | 87.86 | APE67-dihe-in | -63.33, -23.46 | -113.41, 27.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.8 | 0.228 | 0.264 | A | 405.0 | 334.0 | 25 | 31 | 15 | 16 | [[22, 335]] | 1.0 | 6tpa | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F6SA | P49336 | 1 | 359 | 464.0 | 0SQ:60501 | Type3 | Inactive | DFGout | 13.8778 | 7.5572 | BBAminus | -143.37, 174.31 | -133.59, 95.54 | -89.33, -12.55 | 298.0, 127.79 | 85.97, -154.1 | in-in | in | 8.6698 | Saltbr-in | 2.8135 | HRD-in | -74.89, -55.83 | 78.59, -0.68 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 151.84 | APE8-dihe-in | -132.11, 155.15 | APE8-rot-out | 82.42 | APE67-dihe-in | -62.47, -25.65 | -106.71, 17.74 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.8701 | None | None | None | XRAY | 2.6 | 0.205 | 0.26 | A | 405.0 | 327.0 | 32 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 4f6s | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F7JA | P49336 | 1 | 359 | 464.0 | 0SU:60501 | Type3 | Inactive | DFGout | 14.4229 | 8.5945 | BBAminus | -131.55, -173.38 | -148.17, 95.28 | -72.43, -38.8 | 311.88, 131.51 | 104.34, -133.92 | in-in | in | 8.7236 | Saltbr-in | 2.6641 | HRD-in | -75.51, -51.42 | 85.3, -13.72 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -31.87 | APE8-dihe-in | -70.46, 100.26 | APE8-rot-in | 296.32 | APE67-dihe-in | -60.95, -26.84 | -87.97, 10.5 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.055 | None | None | None | XRAY | 2.6 | 0.229 | 0.276 | A | 405.0 | 326.0 | 33 | 31 | 13 | 18 | [[22, 335]] | 1.0 | 4f7j | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | 4F70A | P49336 | 1 | 359 | 464.0 | 0ST:60501 | Type3 | Inactive | None | 18.6473 | 14.4213 | None | -123.12, -177.92 | -154.05, 113.27 | -90.85, 999.0 | 75.63, 12.09 | 999.0, 999.0 | in-in | in | 8.9927 | Saltbr-in | 3.0079 | HRD-in | -82.85, -48.58 | 74.91, -2.44 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 73.37 | APE8-dihe-in | -133.51, 141.85 | APE8-rot-out | 58.33 | APE67-dihe-in | -73.19, -29.13 | -108.0, 28.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.5615 | None | None | None | XRAY | 3.0 | 0.204 | 0.239 | A | 405.0 | 326.0 | 33 | 31 | 11 | 20 | [[22, 335]] | 1.0 | 4f70 | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CDK8 | CDK8_HUMAN | AF-P49336-K1A | P49336 | 12 | 343 | 464.0 | No_ligand | No_ligand | Active | DFGin | 6.9313 | 15.6629 | BLAminus | -128.17, 177.28 | 55.68, 59.43 | -72.54, 15.56 | 300.04, 114.68 | -62.04, -32.39 | in-in | in | 9.1654 | Saltbr-in | 2.8975 | HRD-in | -73.5, -51.19 | 62.86, 10.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8327 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.05, 164.39 | APE9-dihe-na | 83.32, 124.4 | APE8-dihe-in | -52.27, 134.37 | APE8-rot-in | 287.61 | APE67-dihe-in | -65.17, -26.48 | -44.23, -41.35 | APE12-dist-in | 12.0588 | APE11-dist-in | 11.607 | APE10-dist-in | 5.8083 | APE9-dist-in | 3.4091 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 332.0 | 332.0 | 0 | 31 | 31 | 0 | [[22, 335]] | 1.0 | AF-P49336-K1 | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 2.9e-82 | 282.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | AF-P49336-K3A | P49336 | 12 | 343 | 464.0 | No_ligand | No_ligand | Active | DFGin | 7.0585 | 14.4146 | BLAminus | -125.11, 179.05 | 58.06, 66.16 | -75.42, 13.63 | 298.43, 116.53 | -58.59, -38.0 | in-in | in | 9.222 | Saltbr-in | 2.7201 | HRD-in | -77.81, -49.38 | 63.32, 9.66 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8729 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.07, 166.88 | APE9-dihe-na | 60.71, 128.33 | APE8-dihe-in | -54.75, 135.42 | APE8-rot-in | 297.36 | APE67-dihe-in | -67.37, -15.46 | -44.59, -50.0 | APE12-dist-in | 12.5614 | APE11-dist-in | 10.811 | APE10-dist-in | 6.5807 | APE9-dist-in | 3.286 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 332.0 | 332.0 | 0 | 31 | 31 | 0 | [[22, 335]] | 1.0 | AF-P49336-K3 | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 2.9e-82 | 282.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5HBJA | P49336 | 1 | 361 | 464.0 | 5Y8:60401 | Type1 | Inactive | DFGin | 7.5418 | 14.7786 | BLAminus | -106.87, 176.98 | 71.07, 89.31 | -114.96, 61.9 | 305.41, 118.79 | -100.84, -170.16 | in-in | in | 9.7609 | Saltbr-in | 2.6824 | HRD-in | -77.67, -52.92 | 73.2, 5.3 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -16.09 | APE8-dihe-in | -117.57, 98.85 | APE8-rot-in | 304.83 | APE67-dihe-in | -72.47, -22.93 | -102.77, 29.67 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.3779 | None | None | None | XRAY | 3.0 | 999.0 | 0.288 | A | 364.0 | 340.0 | 21 | 31 | 19 | 12 | [[22, 335]] | 1.0 | 5hbj | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5ICPA | P49336 | 1 | 362 | 464.0 | 69Z:60401 | Type1 | Inactive | DFGin | 6.1473 | 13.6394 | BLAminus | -129.39, 179.13 | 50.41, 56.76 | -66.42, 4.81 | 256.2, 78.89 | 56.91, 53.37 | in-in | in | 9.1898 | Saltbr-in | 2.5875 | HRD-in | -78.65, -54.95 | 77.97, -2.02 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7892 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, 83.07 | APE9-dihe-na | -127.02, 140.47 | APE8-dihe-in | -112.3, 142.07 | APE8-rot-out | 57.72 | APE67-dihe-in | -65.52, -25.52 | -110.98, 18.82 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.6843 | APE9-dist-out | 12.5091 | None | None | None | XRAY | 2.18 | 0.185 | 0.216 | A | 364.0 | 343.0 | 19 | 31 | 23 | 8 | [[22, 335]] | 1.0 | 5icp | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5IDNA | P49336 | 1 | 363 | 464.0 | 6A7:60401 | Type1 | Inactive | DFGin | 7.3226 | 16.0877 | BLAminus | -124.47, 174.0 | 67.51, 75.48 | -91.55, 21.99 | 294.62, 123.1 | -96.7, 0.53 | in-in | in | 8.9702 | Saltbr-in | 2.647 | HRD-in | -71.0, -49.83 | 80.54, -0.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.4045 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 147.78 | APE8-dihe-in | -125.68, 150.04 | APE8-rot-out | 46.55 | APE67-dihe-in | -67.71, -25.83 | -125.87, 33.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.7732 | None | None | None | XRAY | 2.26 | 0.221 | 0.253 | A | 370.0 | 336.0 | 27 | 31 | 15 | 16 | [[22, 335]] | 1.0 | 5idn | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5XQXA | P49336 | 1 | 362 | 464.0 | 8CC:60402 | Type1 | Inactive | DFGin | 7.1009 | 13.3766 | BLAminus | -124.76, 173.54 | 67.85, 87.06 | -93.65, 13.06 | 285.44, 142.36 | -53.92, -30.2 | in-in | in | 8.5993 | Saltbr-in | 2.6458 | HRD-in | -76.07, -52.85 | 74.84, 2.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.797 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -162.45 | APE8-dihe-in | -121.89, 118.59 | APE8-rot-in | 276.05 | APE67-dihe-in | -59.33, -23.95 | -109.46, 21.35 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.0086 | None | None | None | XRAY | 2.3 | 0.19 | 0.222 | A | 380.0 | 337.0 | 25 | 31 | 18 | 13 | [[22, 335]] | 1.0 | 5xqx | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.7e-82 | 281.6 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5XS2A | P49336 | 1 | 363 | 464.0 | 8D6:60402 | Type1 | Inactive | DFGin | 7.1 | 13.2185 | BLAminus | -125.86, 168.92 | 68.44, 89.08 | -85.59, 13.7 | 295.46, 132.91 | -57.29, -23.08 | in-in | in | 8.5472 | Saltbr-in | 2.6849 | HRD-in | -77.09, -53.4 | 74.45, 0.97 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7249 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -119.34, 129.98 | APE9-dihe-na | -115.73, -15.25 | APE8-dihe-in | -128.4, 144.08 | APE8-rot-out | 53.94 | APE67-dihe-in | -59.75, -24.05 | -125.87, 25.67 | APE12-dist-in | 7.1385 | APE11-dist-in | 11.8021 | APE10-dist-out | 9.8465 | APE9-dist-out | 12.3679 | None | None | None | XRAY | 2.04 | 0.197 | 0.225 | A | 380.0 | 363.0 | 0 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 5xs2 | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.7e-82 | 281.6 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 6QTJA | P49336 | 1 | 359 | 464.0 | JHK:60501 | Type1 | Inactive | DFGin | 7.5864 | 14.0745 | BLAminus | -112.22, -179.25 | 62.71, 86.71 | -102.98, 13.61 | 301.92, 111.63 | -83.54, 3.25 | in-in | in | 8.4612 | Saltbr-in | 2.9368 | HRD-in | -68.14, -49.62 | 76.51, -6.19 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -45.96 | APE8-dihe-in | -121.23, 128.93 | APE8-rot-in | 272.12 | APE67-dihe-in | -58.17, -25.47 | -117.92, 17.96 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.2357 | None | None | None | XRAY | 2.48 | 0.187 | 0.22 | A | 405.0 | 329.0 | 30 | 31 | 13 | 18 | [[22, 335]] | 1.0 | 6qtj | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 9H8CA | P49336 | 1 | 361 | 464.0 | A1IS8:60503 | Type1 | Inactive | DFGin | 7.5455 | 14.2354 | BLAminus | -123.76, 163.44 | 68.83, 82.68 | -94.14, 12.47 | 302.05, 120.29 | -95.45, 18.7 | in-in | in | 8.8322 | Saltbr-in | 2.6869 | HRD-in | -71.9, -45.8 | 76.46, -12.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8362 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 1.06 | APE8-dihe-in | -111.33, 130.78 | APE8-rot-in | 270.85 | APE67-dihe-in | -58.13, -22.76 | -124.23, 26.3 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.0634 | None | None | None | XRAY | 2.573 | 0.192 | 0.262 | A | 414.0 | 336.0 | 25 | 31 | 16 | 15 | [[22, 335]] | 1.0 | 9h8c | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 6.3e-82 | 281.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 9H8SA | P49336 | 1 | 362 | 464.0 | A1ITF:60509 | Type1 | Inactive | DFGin | 7.3437 | 13.9243 | BLAminus | -119.28, 163.44 | 74.84, 82.25 | -92.61, 11.91 | 298.93, 132.0 | -87.41, 10.8 | in-in | in | 8.6117 | Saltbr-in | 2.6241 | HRD-in | -75.25, -51.5 | 79.06, -6.52 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6589 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 160.05 | APE8-rot-out | 75.96 | APE67-dihe-in | -54.19, -23.95 | -111.96, 19.45 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.157 | 0.197 | 0.248 | A | 414.0 | 335.0 | 27 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 9h8s | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 6.3e-82 | 281.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 8TQ2A | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 5.9534 | 13.4093 | BLAplus | -149.38, -174.61 | 57.66, 42.3 | -94.56, 56.63 | 80.28, 25.13 | -65.65, -33.03 | in-out | in | 9.074 | Saltbr-out | 5.0175 | HRD-in | -71.17, -43.38 | 62.04, 12.67 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.9073 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -111.63, -27.07 | APE9-dihe-na | -152.97, 160.77 | APE8-dihe-in | -61.74, 149.93 | APE8-rot-out | 187.22 | APE67-dihe-in | -65.55, -27.76 | -65.32, -15.56 | APE12-dist-in | 13.0056 | APE11-dist-in | 10.6044 | APE10-dist-in | 7.3395 | APE9-dist-in | 4.2314 | None | None | None | EM | 3.8 | 999.0 | 999.0 | A | 464.0 | 313.0 | 46 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 8tq2 | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 9.1e-82 | 280.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 8TQCA | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 5.954 | 13.4098 | BLAplus | -149.38, -174.65 | 57.7, 42.3 | -94.58, 56.63 | 80.22, 25.15 | -65.67, -33.03 | in-out | in | 9.0736 | Saltbr-out | 5.0166 | HRD-in | -71.16, -43.39 | 62.07, 12.66 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.9071 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -111.64, -27.07 | APE9-dihe-na | -152.99, 160.74 | APE8-dihe-in | -61.68, 149.91 | APE8-rot-out | 187.24 | APE67-dihe-in | -65.64, -27.68 | -65.36, -15.51 | APE12-dist-in | 13.006 | APE11-dist-in | 10.6041 | APE10-dist-in | 7.3394 | APE9-dist-in | 4.2313 | None | None | None | EM | 3.8 | 999.0 | 999.0 | A | 464.0 | 313.0 | 46 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 8tqc | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 9.1e-82 | 280.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 8TQWA | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9194 | 11.7033 | BLAplus | -136.58, -174.19 | 58.52, 55.8 | -94.53, 48.46 | 79.76, 124.7 | -72.57, -22.17 | in-out | in | 9.013 | Saltbr-out | 4.2612 | HRD-in | -69.7, -41.94 | 60.18, 16.8 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.2241 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -107.3, -18.61 | APE9-dihe-na | -153.74, 161.23 | APE8-dihe-in | -65.82, 153.77 | APE8-rot-out | 180.15 | APE67-dihe-in | -67.85, -29.18 | -70.07, -16.17 | APE12-dist-in | 12.7643 | APE11-dist-in | 10.6621 | APE10-dist-in | 7.0853 | APE9-dist-in | 4.3173 | None | None | None | EM | 8.2 | 999.0 | 999.0 | a | 464.0 | 313.0 | 46 | 31 | 31 | 0 | [[22, 335]] | 1.0 | 8tqw | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 9.1e-82 | 280.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4G6LA | P49336 | 1 | 359 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 7.7821 | 13.1649 | BLBminus | -140.33, 170.43 | 60.07, 39.76 | -65.01, 139.84 | 287.11, 130.96 | -72.68, 84.6 | in-in | in | 9.41 | Saltbr-in | 2.7316 | HRD-in | -90.39, -58.08 | 80.12, -10.69 | in-out-none | SNCion | out-none | ActLoopNT-out | 8.7909 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.75, -20.61 | 999.0, 14.23 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.214 | 0.266 | A | 406.0 | 333.0 | 26 | 31 | 19 | 12 | [[22, 335]] | 1.0 | 4g6l | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5FGKA | P49336 | 1 | 362 | 464.0 | 5XG:60401 | Type1 | Inactive | DFGin | 8.4978 | 15.5831 | BLBminus | -133.54, 169.31 | 57.53, 42.29 | -55.85, 144.8 | 295.15, 85.37 | -70.31, 91.66 | in-in | in | 9.829 | Saltbr-in | 2.8534 | HRD-in | -79.53, -56.66 | 86.65, -4.01 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 157.88 | APE8-dihe-in | -124.66, 135.5 | APE8-rot-in | 267.49 | APE67-dihe-in | -66.95, -24.09 | -119.64, 24.09 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.9461 | None | None | None | XRAY | 2.36 | 999.0 | 0.237 | A | 364.0 | 331.0 | 31 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 5fgk | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5HBEA | P49336 | 1 | 361 | 464.0 | 5Y6:60401 | Type1 | Inactive | DFGin | 6.3817 | 13.4796 | BLBminus | -150.55, 174.93 | 54.88, 46.99 | -64.39, 138.78 | 282.35, 68.64 | -73.7, 83.07 | in-in | in | 9.4752 | Saltbr-in | 2.6635 | HRD-in | -80.78, -53.55 | 75.81, 1.36 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.0331 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 124.46 | APE8-dihe-in | -128.69, 136.48 | APE8-rot-out | 167.77 | APE67-dihe-in | -66.35, -22.41 | -120.15, 22.04 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.377 | None | None | None | XRAY | 2.38 | 0.23 | 0.256 | A | 364.0 | 343.0 | 18 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 5hbe | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5HNBA | P49336 | 1 | 359 | 464.0 | 62M:60401 | Type1 | Inactive | DFGin | 6.6498 | 13.1706 | BLBminus | -138.74, 167.16 | 57.27, 44.77 | -53.04, 139.99 | 284.36, 64.87 | -77.11, 80.76 | in-in | in | 9.3522 | Saltbr-in | 2.6998 | HRD-in | -81.89, -52.43 | 75.49, 2.56 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8745 | ActLoopCT-out | nonTYR | APEdihe_aanio | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 22.41 | APE8-rot-in | 326.4 | APE67-dihe-out | -68.33, -25.9 | 68.06, 1.32 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.35 | 0.218 | 0.252 | A | 370.0 | 339.0 | 20 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 5hnb | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5I5ZA | P49336 | 1 | 362 | 464.0 | 68U:60401 | Type1 | Inactive | DFGin | 6.4155 | 13.0643 | BLBminus | -146.19, 175.23 | 51.04, 37.29 | -51.44, 128.07 | 281.53, 66.91 | -69.5, 65.99 | in-in | in | 9.1148 | Saltbr-in | 2.9017 | HRD-in | -79.94, -54.75 | 78.35, 1.56 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7902 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 116.55 | APE8-rot-out | 180.69 | APE67-dihe-in | -62.72, -27.98 | -92.64, 5.94 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.6 | 0.239 | 0.274 | A | 370.0 | 342.0 | 20 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 5i5z | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5IDPA | P49336 | 1 | 359 | 464.0 | 6A6:60401 | Type1 | Inactive | DFGin | 6.659 | 13.1177 | BLBminus | -136.27, 172.07 | 59.2, 45.18 | -61.59, 132.52 | 281.19, 68.65 | -74.88, 80.04 | in-in | in | 9.3926 | Saltbr-in | 2.8965 | HRD-in | -79.39, -54.81 | 77.61, 1.02 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6935 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 164.27 | APE8-rot-out | 60.39 | APE67-dihe-in | -68.82, -22.92 | -114.95, 18.44 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.65 | 0.232 | 0.272 | A | 370.0 | 341.0 | 18 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 5idp | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.3e-82 | 281.7 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F7SA | P49336 | 1 | 359 | 464.0 | 0SW:60501 | Type1 | Inactive | DFGin | 6.495 | 13.0688 | BLBminus | -136.61, 176.12 | 53.35, 42.37 | -54.98, 136.0 | 280.12, 74.29 | -77.21, 78.52 | in-in | in | 9.2294 | Saltbr-in | 2.7473 | HRD-in | -79.34, -55.77 | 76.41, 2.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7597 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 131.9 | APE8-rot-out | 180.5 | APE67-dihe-in | -68.08, -24.25 | -110.68, 14.48 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.2 | 0.194 | 0.222 | A | 405.0 | 339.0 | 20 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 4f7s | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5BNJA | P49336 | 1 | 362 | 464.0 | 4TV:60501 | Type1 | Inactive | DFGin | 6.1998 | 14.6125 | BLBminus | -127.23, 163.17 | 60.48, 55.04 | -65.81, 148.47 | 290.88, 72.47 | -70.37, 93.4 | in-in | in | 9.8117 | Saltbr-in | 2.7276 | HRD-in | -79.48, -50.1 | 76.1, -2.58 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.736 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 162.07 | APE8-rot-out | 56.78 | APE67-dihe-in | -68.21, -22.51 | -112.22, 14.37 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.64 | 0.228 | 0.273 | A | 405.0 | 341.0 | 21 | 31 | 20 | 11 | [[22, 335]] | 1.0 | 5bnj | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 6QTGA | P49336 | 1 | 359 | 464.0 | JH8:60501 | Type1 | Inactive | DFGin | 6.8548 | 13.5978 | BLBminus | -115.69, 168.8 | 67.93, 119.69 | -128.98, 119.87 | 314.23, 115.38 | -156.88, 999.0 | in-in | in | 8.458 | Saltbr-in | 2.9444 | HRD-in | -69.43, -47.54 | 81.38, -19.97 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -47.73 | APE8-dihe-in | -122.24, 124.81 | APE8-rot-in | 266.36 | APE67-dihe-in | -67.96, -18.93 | -113.56, 25.73 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.0679 | None | None | None | XRAY | 2.7 | 0.202 | 0.231 | A | 405.0 | 328.0 | 31 | 31 | 12 | 19 | [[22, 335]] | 1.0 | 6qtg | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4CRLA | P49336 | 1 | 359 | 464.0 | C1I:61360 | Type1 | Inactive | DFGin | 6.2635 | 12.9653 | BLBminus | -130.84, 167.17 | 41.28, 61.34 | -57.58, 143.29 | 285.19, 53.46 | -56.15, 77.43 | in-in | in | 9.2784 | Saltbr-in | 2.7647 | HRD-in | -77.87, -48.76 | 70.82, 12.4 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8293 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -12.95 | APE8-dihe-in | -65.77, 114.52 | APE8-rot-out | 186.25 | APE67-dihe-in | -70.31, -18.88 | -108.2, 7.99 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.3551 | None | None | None | XRAY | 2.4 | 0.201 | 0.256 | A | 406.0 | 336.0 | 23 | 31 | 21 | 10 | [[22, 335]] | 1.0 | 4crl | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5CEIA | P49336 | 1 | 362 | 464.0 | 50R:60508 | Type1 | Inactive | DFGin | 6.4332 | 13.0148 | BLBminus | -132.66, 174.92 | 55.78, 44.71 | -56.21, 137.6 | 280.16, 70.73 | -77.01, 72.68 | in-in | in | 9.2797 | Saltbr-in | 2.5792 | HRD-in | -79.82, -54.28 | 77.75, 0.99 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6632 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 169.41 | APE8-rot-out | 67.16 | APE67-dihe-in | -60.87, -22.55 | -115.47, 18.61 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.24 | 0.175 | 0.227 | A | 406.0 | 344.0 | 18 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 5cei | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 6R3SA | P49336 | 1 | 362 | 464.0 | JRE:60501 | Type1 | Inactive | DFGin | 6.4489 | 13.1166 | BLBminus | -136.26, 169.85 | 57.34, 42.45 | -52.43, 144.8 | 287.58, 63.16 | -78.12, 79.2 | in-in | in | 9.3756 | Saltbr-in | 2.8296 | HRD-in | -80.26, -51.73 | 75.92, 4.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6882 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 130.83 | APE8-rot-out | 181.78 | APE67-dihe-in | -67.95, -25.35 | -103.82, 11.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.19 | 0.202 | 0.227 | A | 406.0 | 343.0 | 19 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 6r3s | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 6Y0AA | P49336 | 1 | 362 | 464.0 | JRE:60501 | Type1 | Inactive | DFGin | 6.4489 | 13.1166 | BLBminus | -136.26, 169.85 | 57.34, 42.45 | -52.43, 144.8 | 287.58, 63.16 | -78.12, 79.2 | in-in | in | 9.3756 | Saltbr-in | 2.8296 | HRD-in | -80.26, -51.73 | 75.92, 4.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6882 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 130.83 | APE8-rot-out | 181.78 | APE67-dihe-in | -67.95, -25.35 | -103.82, 11.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.19 | 0.202 | 0.227 | A | 406.0 | 343.0 | 19 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 6y0a | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 6T41A | P49336 | 1 | 359 | 464.0 | MFE:60501 | Type1 | Inactive | DFGin | 8.6301 | 13.5154 | BLBminus | -130.72, 167.87 | 65.4, 35.77 | -47.77, 142.68 | 290.97, 94.77 | -79.52, 87.36 | in-in | in | 9.2255 | Saltbr-in | 2.9666 | HRD-in | -82.44, -61.41 | 81.57, -4.44 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8749 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 161.03 | APE8-rot-out | 58.35 | APE67-dihe-in | -69.81, -18.57 | -101.28, 19.75 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.45 | 0.185 | 0.256 | A | 407.0 | 343.0 | 16 | 31 | 22 | 9 | [[22, 335]] | 1.0 | 6t41 | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 6e-82 | 281.3 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5HBHA | P49336 | 1 | 361 | 464.0 | 5Y7:60401 | Type1 | Inactive | DFGin | 5.4841 | 13.3356 | BLBplus | -129.14, 169.91 | 65.09, 34.73 | -89.33, 139.59 | 54.15, 87.69 | 88.57, 16.73 | in-in | in | 9.1442 | Saltbr-in | 2.8415 | HRD-in | -73.61, -55.97 | 88.78, -11.96 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.6525 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, 146.42 | APE9-dihe-na | -93.82, 144.5 | APE8-dihe-in | -120.03, 143.32 | APE8-rot-out | 75.1 | APE67-dihe-in | -65.56, -22.05 | -107.02, 22.5 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 20.8418 | APE9-dist-out | 12.1846 | None | None | None | XRAY | 2.5 | 0.235 | 0.268 | A | 364.0 | 334.0 | 27 | 31 | 17 | 14 | [[22, 335]] | 1.0 | 5hbh | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 4.1e-82 | 281.8 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 3RGFA | P49336 | 1 | 353 | 464.0 | BAX:60465 | Type2 | Inactive | DFGout | 15.0897 | 10.8645 | BBAminus | -128.79, 167.92 | -135.88, 84.21 | -83.29, -7.22 | 304.7, 18.84 | -121.06, 44.25 | in-out | in | 9.3695 | Saltbr-out | 4.8518 | HRD-in | -76.1, -55.23 | 78.73, 2.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 12.2242 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 133.12 | APE8-dihe-in | -111.84, 132.17 | APE8-rot-out | 185.32 | APE67-dihe-in | -67.42, -19.98 | -109.35, 18.38 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.6368 | None | None | None | XRAY | 2.2 | 0.183 | 0.221 | A | 405.0 | 319.0 | 34 | 31 | 15 | 16 | [[22, 335]] | 1.0 | 3rgf | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F6UA | P49336 | 1 | 359 | 464.0 | 0SR:60501 | Type2 | Inactive | DFGout | 14.5288 | 8.1472 | BBAminus | -137.04, 173.39 | -132.48, 97.94 | -82.11, -23.16 | 303.07, 124.54 | 89.51, -145.66 | in-in | in | 8.5274 | Saltbr-in | 2.6265 | HRD-in | -75.69, -54.68 | 80.97, 0.65 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnio | APE10-dihe-na | 999.0, -48.5 | APE9-dihe-na | -168.88, 136.11 | APE8-dihe-in | -116.43, 154.29 | APE8-rot-out | 81.86 | APE67-dihe-in | -65.37, -20.81 | -106.87, 16.32 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 7.2334 | APE9-dist-out | 10.9418 | None | None | None | XRAY | 2.1 | 0.177 | 0.198 | A | 405.0 | 332.0 | 27 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 4f6u | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F6WA | P49336 | 1 | 359 | 464.0 | 0SS:60501 | Type2 | Inactive | DFGout | 17.0447 | 13.9468 | BBAminus | -134.04, 175.74 | -149.99, 134.58 | -80.54, -17.82 | 302.37, 168.31 | 89.71, 32.24 | in-in | in | 8.5227 | Saltbr-in | 2.6647 | HRD-in | -81.35, -56.06 | 84.43, -4.37 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 94.48 | APE8-rot-in | 298.45 | APE67-dihe-in | -64.37, -22.4 | -100.8, 19.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.39 | 0.193 | 0.234 | A | 405.0 | 330.0 | 29 | 31 | 13 | 18 | [[22, 335]] | 1.0 | 4f6w | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F7LA | P49336 | 1 | 359 | 464.0 | 0SO:60501 | Type2 | Inactive | DFGout | 13.5433 | 10.487 | BBAminus | -144.39, 166.94 | -130.48, 125.05 | -101.12, -66.88 | 314.21, 89.91 | 174.94, 999.0 | in-in | in | 9.0525 | Saltbr-in | 2.7304 | HRD-in | -72.87, -46.64 | 81.38, -4.09 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 155.76 | APE8-rot-out | 66.51 | APE67-dihe-in | -72.52, -24.41 | -123.27, 25.01 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.9 | 0.226 | 0.27 | A | 405.0 | 326.0 | 33 | 31 | 11 | 20 | [[22, 335]] | 1.0 | 4f7l | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F7NA | P49336 | 1 | 361 | 464.0 | 0SV:60501 | Type2 | Inactive | DFGout | 14.194 | 8.2102 | BBAminus | -139.77, 176.54 | -136.01, 97.7 | -86.48, -26.06 | 306.23, 126.32 | 100.15, -136.94 | in-in | in | 8.7798 | Saltbr-in | 2.7862 | HRD-in | -78.13, -54.62 | 75.98, 5.37 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnio | APE10-dihe-na | 999.0, 43.71 | APE9-dihe-na | -114.3, 132.58 | APE8-dihe-in | -127.74, 146.12 | APE8-rot-out | 68.03 | APE67-dihe-in | -66.61, -22.51 | -99.38, 17.25 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 5.8201 | APE9-dist-out | 11.2715 | None | None | None | XRAY | 2.65 | 0.2 | 0.228 | A | 405.0 | 333.0 | 28 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 4f7n | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 5HVYA | P49336 | 1 | 359 | 464.0 | 66X:60501 | Type2 | Inactive | DFGout | 15.175 | 9.3117 | BBAminus | -147.75, 175.04 | -130.64, 103.81 | -80.2, 9.83 | 305.77, 118.03 | 84.07, 29.62 | out-out | out | 11.2669 | Saltbr-out | 6.1116 | HRD-in | -85.57, -56.75 | 82.18, -2.99 | out-out-out | SNCooo | out-out | ActLoopNT-out | 12.8606 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oioo | APE10-dihe-na | -86.7, 132.16 | APE9-dihe-na | -171.76, 167.74 | APE8-dihe-in | -116.95, 139.23 | APE8-rot-out | 61.83 | APE67-dihe-in | -58.0, -28.58 | -98.28, 0.53 | APE12-dist-out | 14.3713 | APE11-dist-in | 9.0319 | APE10-dist-out | 8.2992 | APE9-dist-out | 10.3787 | None | None | None | XRAY | 2.39 | 0.181 | 0.22 | A | 406.0 | 333.0 | 26 | 31 | 19 | 12 | [[22, 335]] | 1.0 | 5hvy | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 6TPAA | P49336 | 1 | 359 | 464.0 | NZ8:60501,NZ5:60505,NZ5:60506,NZ5:60507 | Type2,Allosteric,Allosteric,Allosteric | Inactive | DFGout | 13.8318 | 11.8175 | BBAminus | -130.48, -178.36 | -144.36, 91.14 | -84.2, -4.16 | 322.15, 13.04 | -124.91, 44.75 | out-out | out | 10.1823 | Saltbr-out | 4.9546 | HRD-in | -82.95, -50.83 | 78.95, 15.78 | out-out-out | SNCooo | out-out | ActLoopNT-out | 11.9075 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 123.19 | APE8-rot-out | 87.86 | APE67-dihe-in | -63.33, -23.46 | -113.41, 27.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.8 | 0.228 | 0.264 | A | 405.0 | 334.0 | 25 | 31 | 15 | 16 | [[22, 335]] | 1.0 | 6tpa | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F6SA | P49336 | 1 | 359 | 464.0 | 0SQ:60501 | Type3 | Inactive | DFGout | 13.8778 | 7.5572 | BBAminus | -143.37, 174.31 | -133.59, 95.54 | -89.33, -12.55 | 298.0, 127.79 | 85.97, -154.1 | in-in | in | 8.6698 | Saltbr-in | 2.8135 | HRD-in | -74.89, -55.83 | 78.59, -0.68 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 151.84 | APE8-dihe-in | -132.11, 155.15 | APE8-rot-out | 82.42 | APE67-dihe-in | -62.47, -25.65 | -106.71, 17.74 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 10.8701 | None | None | None | XRAY | 2.6 | 0.205 | 0.26 | A | 405.0 | 327.0 | 32 | 31 | 14 | 17 | [[22, 335]] | 1.0 | 4f6s | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F7JA | P49336 | 1 | 359 | 464.0 | 0SU:60501 | Type3 | Inactive | DFGout | 14.4229 | 8.5945 | BBAminus | -131.55, -173.38 | -148.17, 95.28 | -72.43, -38.8 | 311.88, 131.51 | 104.34, -133.92 | in-in | in | 8.7236 | Saltbr-in | 2.6641 | HRD-in | -75.51, -51.42 | 85.3, -13.72 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -31.87 | APE8-dihe-in | -70.46, 100.26 | APE8-rot-in | 296.32 | APE67-dihe-in | -60.95, -26.84 | -87.97, 10.5 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.055 | None | None | None | XRAY | 2.6 | 0.229 | 0.276 | A | 405.0 | 326.0 | 33 | 31 | 13 | 18 | [[22, 335]] | 1.0 | 4f7j | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| CDK8 | CDK8_HUMAN | 4F70A | P49336 | 1 | 359 | 464.0 | 0ST:60501 | Type3 | Inactive | None | 18.6473 | 14.4213 | None | -123.12, -177.92 | -154.05, 113.27 | -90.85, 999.0 | 75.63, 12.09 | 999.0, 999.0 | in-in | in | 8.9927 | Saltbr-in | 3.0079 | HRD-in | -82.85, -48.58 | 74.91, -2.44 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 73.37 | APE8-dihe-in | -133.51, 141.85 | APE8-rot-out | 58.33 | APE67-dihe-in | -73.19, -29.13 | -108.0, 28.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.5615 | None | None | None | XRAY | 3.0 | 0.204 | 0.239 | A | 405.0 | 326.0 | 33 | 31 | 11 | 20 | [[22, 335]] | 1.0 | 4f70 | Homo sapiens | CMGC_CDK8_HUMAN | CMGC | 5.9e-82 | 281.4 | 5.0 | 301.0 | 297.0 | 172 | 173 | 174 | 176 | 178 | 52 | 66 | 70 | 148 | 150 | 149 | 151.0 | 216 | 203 | 198 | 197 | 196 | 195 | 194 | 193 | 192 | 98 | Cyclin-dependent kinase 8 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|