Protein kinases in complex with 7DZ

Total number of genes: 3
Total number of chains: 6
Spatial Dihedral Chains Representative
DFGin BLAminus 4 5UVFA
DFGin ABAminus 1 5UU1A
DFGin None 1 5UT1A

Database table as tsv
Group Gene UniprotID Protein PDB Resolu Activity Label Spatial Label Dihedral Label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type
CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFA 2.0 None DFGin BLAminus in-none in-in 7DZ Type1
CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFB 2.0 Inactive DFGin BLAminus in-out in-in 7DZ Type1
CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFC 2.0 Active DFGin BLAminus in-in in-in 7DZ Type1.5_Back
CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFD 2.0 Active DFGin BLAminus in-in in-in 7DZ Type1.5_Back
CK1 VRK2 VRK2_HUMAN Serine/threonine-protein kinase VRK2 5UU1A 2.0 Inactive DFGin ABAminus in-in in-in 7DZ Type1.5_Back
TYR JAK2 JAK2_HUMAN Tyrosine-protein kinase JAK2 5UT1A 1.95 Inactive DFGin None in-none out-out 7DZ Type1

Protein kinases in complex with 7DZ

Total number of genes: 3
Total number of chains: 6
Spatial Dihedral Chains Representative
DFGin BLAminus 4 5UVFA
DFGin ABAminus 1 5UU1A
DFGin None 1 5UT1A

Database table as tsv
Organism Group Gene UniprotID Protein PDB Resolu Activity Label Spatial Label Dihedral Label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type
Homo sapiens CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFA 2.0 None DFGin BLAminus in-none in-in 7DZ Type1
Homo sapiens CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFB 2.0 Inactive DFGin BLAminus in-out in-in 7DZ Type1
Homo sapiens CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFC 2.0 Active DFGin BLAminus in-in in-in 7DZ Type1.5_Back
Homo sapiens CK1 VRK1 VRK1_HUMAN Serine/threonine-protein kinase VRK1 5UVFD 2.0 Active DFGin BLAminus in-in in-in 7DZ Type1.5_Back
Homo sapiens CK1 VRK2 VRK2_HUMAN Serine/threonine-protein kinase VRK2 5UU1A 2.0 Inactive DFGin ABAminus in-in in-in 7DZ Type1.5_Back
Homo sapiens TYR JAK2 JAK2_HUMAN Tyrosine-protein kinase JAK2 5UT1A 1.95 Inactive DFGin None in-none out-out 7DZ Type1

Protein kinases in complex with 7DZ

Total number of genes: 0
Total number of chains: 0
Spatial Dihedral Chains Representative

Database table as tsv

Organism Group Gene UniprotID Protein PDB Resolu Activity Label Spatial Label Dihedral Label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type