Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 169 | AF-O14757-K1A |
PDB | Resolution | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type | Residues in structure | Mutation | Phosphorylation | Unresolved residues in A-loop |
---|---|---|---|---|---|---|---|---|---|---|---|---|
3JVRA | 1.76 | Active | DFGin | BLAminus | in-in | in-in | AGX | Allosteric | 2 - 272 | None | None | 0 |
3JVSA | 1.9 | Inactive | DFGin | BLAminus | in-out | in-in | AGY | Allosteric | 2 - 272 | None | None | 0 |
3F9NA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 38M | Allosteric | 7 - 270 | None | None | 0 |
AF-O14757-K1A | -1.0 | Active | DFGin | BLAminus | in-in | in-in | No_ligand | No_ligand | 1 - 273 | None | None | 0 |
1IA8A | 1.7 | Active | DFGin | BLAminus | in-in | in-in | No_ligand | No_ligand | 2 - 276 | None | None | 0 |
7AKMB | 1.93 | Active | DFGin | BLAminus | in-in | in-in | No_ligand | No_ligand | 2 - 269 | D10R | None | 0 |
1ZYSA | 1.7 | Active | DFGin | BLAminus | in-in | in-in | 199 | Type1 | 3 - 273 | None | None | 0 |
2E9VA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 85A | Type1 | 2 - 269 | None | None | 0 |
2E9VB | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 85A | Type1 | 2 - 269 | None | None | 0 |
2E9OA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A58 | Type1 | 2 - 270 | None | None | 0 |
2E9PA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | 77A | Type1 | 2 - 270 | None | None | 0 |
2E9UA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A25 | Type1 | 2 - 270 | None | None | 0 |
2GHGA | 3.5 | Active | DFGin | BLAminus | in-in | in-in | A53 | Type1 | 2 - 270 | None | None | 0 |
2YWPA | 2.9 | Active | DFGin | BLAminus | in-in | in-in | A42 | Type1 | 2 - 270 | None | None | 0 |
3OT3A | 1.44 | Active | DFGin | BLAminus | in-in | in-in | 22K | Type1 | 4 - 272 | None | None | 0 |
3OT8A | 1.645 | Active | DFGin | BLAminus | in-in | in-in | MI5 | Type1 | 4 - 272 | None | None | 0 |
3PA3A | 1.4 | Active | DFGin | BLAminus | in-in | in-in | C70 | Type1 | 4 - 272 | None | None | 0 |
3PA4A | 1.59 | Active | DFGin | BLAminus | in-in | in-in | C72 | Type1 | 6 - 272 | None | None | 0 |
3PA5A | 1.7 | Active | DFGin | BLAminus | in-in | in-in | C73 | Type1 | 3 - 272 | None | None | 0 |
3U9NA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | 09H | Type1 | 7 - 272 | None | None | 0 |
4JIKA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 1KO | Type1 | 4 - 272 | None | None | 0 |
2X8EA | 2.5 | Active | DFGin | BLAminus | in-in | in-in | X8E | Type1 | 9 - 270 | None | None | 0 |
2YDJA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | YDJ | Type1 | 8 - 269 | None | None | 0 |
2YDJB | 1.85 | Active | DFGin | BLAminus | in-in | in-in | YDJ | Type1 | 9 - 269 | None | None | 0 |
2YDKA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | YDK | Type1 | 3 - 270 | None | None | 0 |
2YERA | 1.83 | Active | DFGin | BLAminus | in-in | in-in | TQ1 | Type1 | 2 - 269 | None | None | 0 |
2YEXA | 1.3 | Active | DFGin | BLAminus | in-in | in-in | YEX | Type1 | 2 - 270 | None | None | 0 |
6FC8A | 1.61 | Active | DFGin | BLAminus | in-in | in-in | D4Q | Type1 | 2 - 270 | None | None | 0 |
6FCFA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | D58 | Type1 | 9 - 269 | None | None | 0 |
6FCKA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | D4Z | Type1 | 2 - 270 | None | None | 0 |
4FSNA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A58 | Type1 | 3 - 280 | None | None | 0 |
4FSMA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK1 | Type1 | 3 - 280 | None | None | 0 |
4FSRA | 2.5 | Active | DFGin | BLAminus | in-in | in-in | HKC | Type1 | 3 - 280 | None | None | 0 |
4FSWA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK6 | Type1 | 3 - 280 | None | None | 0 |
4FSYA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK7 | Type1 | 3 - 280 | None | None | 0 |
4FSZA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK8 | Type1 | 3 - 280 | None | None | 0 |
4FT0A | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK9 | Type1 | 3 - 280 | None | None | 0 |
4FT3A | 2.5 | Active | DFGin | BLAminus | in-in | in-in | H1K | Type1 | 2 - 280 | None | None | 0 |
4FT5A | 2.4 | Active | DFGin | BLAminus | in-in | in-in | H2K | Type1 | 3 - 280 | None | None | 0 |
4FT7A | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H3K | Type1 | 3 - 280 | None | None | 0 |
4FT9A | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H4K | Type1 | 2 - 280 | None | None | 0 |
4FTAA | 2.4 | Active | DFGin | BLAminus | in-in | in-in | H5K | Type1 | 3 - 280 | None | None | 0 |
4FTCA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | H6K | Type1 | 2 - 280 | None | None | 0 |
4FTIA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H7K | Type1 | 3 - 279 | None | None | 0 |
4FTJA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H8K | Type1 | 3 - 279 | None | None | 0 |
4FTOA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | 3HK | Type1 | 3 - 271 | None | None | 0 |
4FTQA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 4HK | Type1 | 3 - 270 | None | None | 0 |
4FTRA | 2.25 | Active | DFGin | BLAminus | in-in | in-in | 5HK | Type1 | 3 - 271 | None | None | 0 |
4FTTA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | 6HK | Type1 | 3 - 280 | None | None | 0 |
4FTUA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | 7HK | Type1 | 3 - 280 | None | None | 0 |
4GH2A | 2.03 | Active | DFGin | BLAminus | in-in | in-in | HK0 | Type1 | 3 - 280 | None | None | 0 |
1NVQA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | UCN | Type1 | 3 - 273 | None | None | 0 |
1NVRA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | STU | Type1 | 3 - 273 | None | None | 0 |
1NVSA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | UCM | Type1 | 3 - 273 | None | None | 0 |
2WMQA | 2.48 | Active | DFGin | BLAminus | in-in | in-in | ZYQ | Type1 | 7 - 269 | None | None | 0 |
2WMRA | 2.43 | Active | DFGin | BLAminus | in-in | in-in | ZYR | Type1 | 7 - 270 | None | None | 0 |
2WMSA | 2.7 | Active | DFGin | BLAminus | in-in | in-in | ZYS | Type1 | 7 - 270 | None | None | 0 |
2WMTA | 2.55 | Active | DFGin | BLAminus | in-in | in-in | ZYT | Type1 | 8 - 270 | None | None | 0 |
2WMUA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | ZYU | Type1 | 9 - 270 | None | None | 0 |
2WMVA | 2.009 | Active | DFGin | BLAminus | in-in | in-in | ZYV | Type1 | 7 - 270 | None | None | 0 |
2WMWA | 2.43 | Active | DFGin | BLAminus | in-in | in-in | ZYW | Type1 | 7 - 269 | None | None | 0 |
2WMXA | 2.45 | Active | DFGin | BLAminus | in-in | in-in | ZY6 | Type1 | 7 - 269 | None | None | 0 |
2X8DA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | X8D | Type1 | 2 - 281 | None | None | 0 |
2X8IA | 1.92 | Active | DFGin | BLAminus | in-in | in-in | X8I | Type1 | 2 - 269 | None | None | 0 |
2XEYA | 2.7 | Active | DFGin | BLAminus | in-in | in-in | YVQ | Type1 | 6 - 269 | None | None | 0 |
2XEZA | 2.25 | Active | DFGin | BLAminus | in-in | in-in | XEZ | Type1 | 7 - 270 | None | None | 0 |
2XF0A | 2.4 | Active | DFGin | BLAminus | in-in | in-in | 4UB | Type1 | 4 - 270 | None | None | 0 |
2YDIA | 1.6 | Active | DFGin | BLAminus | in-in | in-in | YDI | Type1 | 2 - 281 | None | None | 0 |
2YM3A | 2.007 | Active | DFGin | BLAminus | in-in | in-in | YM3 | Type1 | 8 - 270 | None | None | 0 |
2YM4A | 2.35 | Active | DFGin | BLAminus | in-in | in-in | 4YM | Type1 | 4 - 270 | None | None | 0 |
2YM5A | 2.03 | Inactive | DFGin | BLAminus | in-out | in-in | YM5 | Type1 | 8 - 270 | None | None | 0 |
2YM6A | 2.01 | Inactive | DFGin | BLAminus | in-out | in-in | YM6 | Type1 | 7 - 270 | None | None | 0 |
2YM8A | 2.07 | Active | DFGin | BLAminus | in-in | in-in | YM8 | Type1 | 8 - 270 | None | None | 0 |
4HYHA | 1.7 | Active | DFGin | BLAminus | in-in | in-in | 1AM | Type1 | 4 - 272 | None | None | 0 |
4HYIA | 1.399 | Active | DFGin | BLAminus | in-in | in-in | 1AO | Type1 | 3 - 274 | None | None | 0 |
1ZLTA | 1.74 | Active | DFGin | BLAminus | in-in | in-in | HYM | Type1 | 2 - 276 | None | None | 0 |
2GDOA | 3.0 | Active | DFGin | BLAminus | in-in | in-in | 12C | Type1 | 1 - 273 | None | None | 0 |
2BR1A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | PFP | Type1 | 2 - 276 | None | None | 0 |
2BRBA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | PFQ | Type1 | 2 - 276 | None | None | 0 |
2BRGA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | DFY | Type1 | 7 - 269 | None | None | 0 |
2BRHA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | DFW | Type1 | 6 - 271 | None | None | 0 |
2BRMA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | DFZ | Type1 | 7 - 274 | None | None | 0 |
2BRNA | 2.8 | Active | DFGin | BLAminus | in-in | in-in | DF1 | Type1 | 6 - 276 | None | None | 0 |
2BROA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | DF2 | Type1 | 2 - 276 | None | None | 0 |
2C3JA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | DBQ | Type1 | 6 - 270 | None | None | 0 |
2C3LA | 2.35 | Active | DFGin | BLAminus | in-in | in-in | IDZ | Type1 | 2 - 273 | None | None | 0 |
2CGUA | 2.5 | Active | DFGin | BLAminus | in-in | in-in | 3A3 | Type1 | 6 - 271 | None | None | 0 |
2CGVA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | 3B3 | Type1 | 6 - 272 | None | None | 0 |
2CGWA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | 3C3 | Type1 | 6 - 271 | None | None | 0 |
2CGXA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | 3D3 | Type1 | 6 - 273 | None | None | 0 |
3NLBA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 5BE | Type1 | 6 - 271 | None | None | 0 |
5DLSA | 2.15 | Active | DFGin | BLAminus | in-in | in-in | 5CV | Type1 | 6 - 270 | None | None | 0 |
7BKNA | 2.74 | Active | DFGin | BLAminus | in-in | in-in | ADE | Type1 | 7 - 271 | None | None | 0 |
7BKOA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | TVW | Type1 | 7 - 271 | None | None | 0 |
4QYEA | 2.05 | Active | DFGin | BLAminus | in-in | in-in | 3DL | Type1 | 3 - 280 | None | None | 0 |
4QYFA | 2.15 | Active | DFGin | BLAminus | in-in | in-in | 3DV | Type1 | 3 - 280 | None | None | 0 |
4QYGA | 1.75 | Active | DFGin | BLAminus | in-in | in-in | 3DW | Type1 | 3 - 273 | None | None | 0 |
4QYGB | 1.75 | Active | DFGin | BLAminus | in-in | in-in | 3DW | Type1 | 3 - 273 | None | None | 0 |
4QYHA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 3DX | Type1 | 3 - 273 | None | None | 0 |
4QYHB | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 3DX | Type1 | 3 - 273 | None | None | 0 |
4RVKA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | 3XK | Type1 | 3 - 273 | None | None | 0 |
4RVLA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | 3XL | Type1 | 3 - 273 | None | None | 0 |
4RVMA | 1.86 | Active | DFGin | BLAminus | in-in | in-in | 3X7 | Type1 | 3 - 273 | None | None | 0 |
7AKMA | 1.93 | Active | DFGin | BLAminus | in-in | in-in | AGS | Type1 | 2 - 271 | D10R | None | 0 |
7AKOA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | STU | Type1 | 2 - 271 | D10R | None | 0 |
7AKOB | 1.8 | Active | DFGin | BLAminus | in-in | in-in | STU | Type1 | 2 - 271 | D10R | None | 0 |
2HOGA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 710 | Type1 | 2 - 280 | None | None | 0 |
2HXLA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | 422 | Type1 | 2 - 276 | None | None | 0 |
2HXQA | 2.0 | Inactive | DFGin | BLAminus | in-out | in-in | 373 | Type1 | 2 - 276 | None | None | 0 |
2HY0A | 1.7 | Inactive | DFGin | BLAminus | in-out | in-in | 306 | Type1 | 2 - 280 | None | None | 0 |
2QHMA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 7CS | Type1 | 2 - 280 | None | None | 0 |
2QHNA | 1.7 | Active | DFGin | BLAminus | in-in | in-in | 582 | Type1 | 2 - 280 | None | None | 0 |
2R0UA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | M54 | Type1 | 2 - 280 | None | None | 0 |
3TKHA | 1.79 | Active | DFGin | BLAminus | in-in | in-in | 07S | Type1 | 2 - 280 | None | None | 0 |
3TKIA | 1.6 | Active | DFGin | BLAminus | in-in | in-in | S25 | Type1 | 2 - 280 | None | None | 0 |
5OQ5A | 1.4 | Active | DFGin | BLAminus | in-in | in-in | 4K4 | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A | None | 0 |
5OQ7A | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A | None | 0 |
5OQ7B | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 8 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A | None | 0 |
4FSUA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | HK5 | Type1 | 4 - 271 | None | None | 0 |
5OQ6A | 1.95 | Active | DFGin | BLAminus | in-in | in-in | 4K4 | Type1 | 5 - 270 | A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OQ8A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 4 - 270 | A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OOPA | 1.7 | Inactive | DFGin | BLAminus | in-out | in-in | ANP | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OORA | 1.9 | Inactive | DFGin | BLAminus | in-out | in-in | STU | Type1 | 3 - 283 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OOTA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | 4K4 | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OP2A | 1.9 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OP4A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A0T | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OP5A | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 3FE | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OP7A | 1.8 | Active | DFGin | BLAminus | in-in | in-in | A1K | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OPBA | 1.55 | Active | DFGin | BLAminus | in-in | in-in | A1N | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OPRA | 1.95 | Active | DFGin | BLAminus | in-in | in-in | A3E | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OPSA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A3Q | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OPUA | 1.55 | Active | DFGin | BLAminus | in-in | in-in | A3K | Type1 | 3 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5OPVA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | A3H | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJDA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | TVT | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJEA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | ADE | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJHA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | 42C | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJJA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | TVW | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJMA | 2.3 | Inactive | DFGin | BLAminus | in-out | in-in | TW2 | Type1 | 5 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJOA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | TWK | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJRA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | TWH | Type1 | 5 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJXA | 2.4 | Active | DFGin | BLAminus | in-in | in-in | U0Q | Type1 | 8 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BJXB | 2.4 | Active | DFGin | BLAminus | in-in | in-in | U0Q | Type1 | 8 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BK1A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | U0N | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BK2A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | U0K | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7BK3A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | U0T | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7MCKA | 1.65 | Active | DFGin | BLAminus | in-in | in-in | YXD | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7SUFA | 1.48 | Active | DFGin | BLAminus | in-in | in-in | BVI | Type1 | 3 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7SUGA | 1.48 | Active | DFGin | BLAminus | in-in | in-in | BWI | Type1 | 3 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7SUHA | 2.46 | Active | DFGin | BLAminus | in-in | in-in | BXI | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7SUIA | 2.119 | Active | DFGin | BLAminus | in-in | in-in | L80 | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7SUJA | 2.299 | Inactive | DFGin | BLAminus | in-out | in-in | BYL | Type1 | 9 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
7SUJB | 2.299 | Active | DFGin | BLAminus | in-in | in-in | BYL | Type1 | 9 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
8E80A | 1.49 | Active | DFGin | BLAminus | in-in | in-in | UUF | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
8E81A | 1.62 | Active | DFGin | BLAminus | in-in | in-in | UU6 | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
8SIVA | 1.759 | Active | DFGin | BLAminus | in-in | in-in | ZXH | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
8SIWA | 1.877 | Active | DFGin | BLAminus | in-in | in-in | ZXL | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
8SIWB | 1.877 | Active | DFGin | BLAminus | in-in | in-in | ZXL | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
8SIXA | 1.55 | Active | DFGin | BLAminus | in-in | in-in | ZXP | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
5F4NA | 1.91 | Active | DFGin | BLAminus | in-in | in-in | 5UY 5UY | Type1 Allosteric | 5 - 271 | None | None | 0 |
2YM7A | 1.81 | Active | DFGin | BLAminus | in-in | in-in | YM7 YM7 | Type1 Type1 | 7 - 271 | None | None | 0 |
2E9NA | 2.5 | Inactive | DFGin | BLAminus | in-out | in-in | 76A | Type1.5_Back | 2 - 270 | None | None | 0 |
4FSTA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | HK4 | Type1.5_Back | 3 - 270 | None | None | 0 |
2AYPA | 2.9 | Active | DFGin | BLAminus | in-in | in-in | 43A | Type1.5_Back | 2 - 269 | None | None | 0 |
4FSQA | 2.4 | Active | DFGin | BLAminus | in-in | in-in | HK3 | Type1.5_Back | 3 - 280 | None | None | 0 |
4FTKA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | H9K | Type1.5_Back | 3 - 280 | None | None | 0 |
4FTLA | 2.5 | Inactive | DFGin | BLAminus | in-out | in-in | H0K | Type1.5_Back | 3 - 280 | None | None | 0 |
4FTMA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 1HK | Type1.5_Back | 3 - 280 | None | None | 0 |
4FTNA | 2.02 | Active | DFGin | BLAminus | in-in | in-in | 2HK | Type1.5_Back | 3 - 271 | None | None | 0 |
2C3KA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | ABO | Type1.5_Back | 6 - 270 | None | None | 0 |
Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 169 | AF-O14757-K1A |
Organism | UniprotID | PDB | Resolution | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type | Residues in structure | Mutation | Phosphorylation | Unresolved residues in A-loop |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Homo sapiens | CHK1_HUMAN | 3JVRA | 1.76 | Active | DFGin | BLAminus | in-in | in-in | AGX | Allosteric | 2 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3JVSA | 1.9 | Inactive | DFGin | BLAminus | in-out | in-in | AGY | Allosteric | 2 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3F9NA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 38M | Allosteric | 7 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | AF-O14757-K1A | -1.0 | Active | DFGin | BLAminus | in-in | in-in | No_ligand | No_ligand | 1 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 1IA8A | 1.7 | Active | DFGin | BLAminus | in-in | in-in | No_ligand | No_ligand | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 7AKMB | 1.93 | Active | DFGin | BLAminus | in-in | in-in | No_ligand | No_ligand | 2 - 269 | D10R | None | 0 |
Homo sapiens | CHK1_HUMAN | 1ZYSA | 1.7 | Active | DFGin | BLAminus | in-in | in-in | 199 | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2E9VA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 85A | Type1 | 2 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2E9VB | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 85A | Type1 | 2 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2E9OA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A58 | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2E9PA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | 77A | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2E9UA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A25 | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2GHGA | 3.5 | Active | DFGin | BLAminus | in-in | in-in | A53 | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YWPA | 2.9 | Active | DFGin | BLAminus | in-in | in-in | A42 | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3OT3A | 1.44 | Active | DFGin | BLAminus | in-in | in-in | 22K | Type1 | 4 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3OT8A | 1.645 | Active | DFGin | BLAminus | in-in | in-in | MI5 | Type1 | 4 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3PA3A | 1.4 | Active | DFGin | BLAminus | in-in | in-in | C70 | Type1 | 4 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3PA4A | 1.59 | Active | DFGin | BLAminus | in-in | in-in | C72 | Type1 | 6 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3PA5A | 1.7 | Active | DFGin | BLAminus | in-in | in-in | C73 | Type1 | 3 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3U9NA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | 09H | Type1 | 7 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4JIKA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 1KO | Type1 | 4 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2X8EA | 2.5 | Active | DFGin | BLAminus | in-in | in-in | X8E | Type1 | 9 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YDJA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | YDJ | Type1 | 8 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YDJB | 1.85 | Active | DFGin | BLAminus | in-in | in-in | YDJ | Type1 | 9 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YDKA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | YDK | Type1 | 3 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YERA | 1.83 | Active | DFGin | BLAminus | in-in | in-in | TQ1 | Type1 | 2 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YEXA | 1.3 | Active | DFGin | BLAminus | in-in | in-in | YEX | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 6FC8A | 1.61 | Active | DFGin | BLAminus | in-in | in-in | D4Q | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 6FCFA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | D58 | Type1 | 9 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 6FCKA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | D4Z | Type1 | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSNA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A58 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSMA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK1 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSRA | 2.5 | Active | DFGin | BLAminus | in-in | in-in | HKC | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSWA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK6 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSYA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK7 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSZA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK8 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FT0A | 2.3 | Active | DFGin | BLAminus | in-in | in-in | HK9 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FT3A | 2.5 | Active | DFGin | BLAminus | in-in | in-in | H1K | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FT5A | 2.4 | Active | DFGin | BLAminus | in-in | in-in | H2K | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FT7A | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H3K | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FT9A | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H4K | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTAA | 2.4 | Active | DFGin | BLAminus | in-in | in-in | H5K | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTCA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | H6K | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTIA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H7K | Type1 | 3 - 279 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTJA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | H8K | Type1 | 3 - 279 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTOA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | 3HK | Type1 | 3 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTQA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 4HK | Type1 | 3 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTRA | 2.25 | Active | DFGin | BLAminus | in-in | in-in | 5HK | Type1 | 3 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTTA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | 6HK | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTUA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | 7HK | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4GH2A | 2.03 | Active | DFGin | BLAminus | in-in | in-in | HK0 | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 1NVQA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | UCN | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 1NVRA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | STU | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 1NVSA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | UCM | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMQA | 2.48 | Active | DFGin | BLAminus | in-in | in-in | ZYQ | Type1 | 7 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMRA | 2.43 | Active | DFGin | BLAminus | in-in | in-in | ZYR | Type1 | 7 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMSA | 2.7 | Active | DFGin | BLAminus | in-in | in-in | ZYS | Type1 | 7 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMTA | 2.55 | Active | DFGin | BLAminus | in-in | in-in | ZYT | Type1 | 8 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMUA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | ZYU | Type1 | 9 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMVA | 2.009 | Active | DFGin | BLAminus | in-in | in-in | ZYV | Type1 | 7 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMWA | 2.43 | Active | DFGin | BLAminus | in-in | in-in | ZYW | Type1 | 7 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2WMXA | 2.45 | Active | DFGin | BLAminus | in-in | in-in | ZY6 | Type1 | 7 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2X8DA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | X8D | Type1 | 2 - 281 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2X8IA | 1.92 | Active | DFGin | BLAminus | in-in | in-in | X8I | Type1 | 2 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2XEYA | 2.7 | Active | DFGin | BLAminus | in-in | in-in | YVQ | Type1 | 6 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2XEZA | 2.25 | Active | DFGin | BLAminus | in-in | in-in | XEZ | Type1 | 7 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2XF0A | 2.4 | Active | DFGin | BLAminus | in-in | in-in | 4UB | Type1 | 4 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YDIA | 1.6 | Active | DFGin | BLAminus | in-in | in-in | YDI | Type1 | 2 - 281 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YM3A | 2.007 | Active | DFGin | BLAminus | in-in | in-in | YM3 | Type1 | 8 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YM4A | 2.35 | Active | DFGin | BLAminus | in-in | in-in | 4YM | Type1 | 4 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YM5A | 2.03 | Inactive | DFGin | BLAminus | in-out | in-in | YM5 | Type1 | 8 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YM6A | 2.01 | Inactive | DFGin | BLAminus | in-out | in-in | YM6 | Type1 | 7 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YM8A | 2.07 | Active | DFGin | BLAminus | in-in | in-in | YM8 | Type1 | 8 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4HYHA | 1.7 | Active | DFGin | BLAminus | in-in | in-in | 1AM | Type1 | 4 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4HYIA | 1.399 | Active | DFGin | BLAminus | in-in | in-in | 1AO | Type1 | 3 - 274 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 1ZLTA | 1.74 | Active | DFGin | BLAminus | in-in | in-in | HYM | Type1 | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2GDOA | 3.0 | Active | DFGin | BLAminus | in-in | in-in | 12C | Type1 | 1 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BR1A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | PFP | Type1 | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BRBA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | PFQ | Type1 | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BRGA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | DFY | Type1 | 7 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BRHA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | DFW | Type1 | 6 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BRMA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | DFZ | Type1 | 7 - 274 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BRNA | 2.8 | Active | DFGin | BLAminus | in-in | in-in | DF1 | Type1 | 6 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2BROA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | DF2 | Type1 | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2C3JA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | DBQ | Type1 | 6 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2C3LA | 2.35 | Active | DFGin | BLAminus | in-in | in-in | IDZ | Type1 | 2 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2CGUA | 2.5 | Active | DFGin | BLAminus | in-in | in-in | 3A3 | Type1 | 6 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2CGVA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | 3B3 | Type1 | 6 - 272 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2CGWA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | 3C3 | Type1 | 6 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2CGXA | 2.2 | Active | DFGin | BLAminus | in-in | in-in | 3D3 | Type1 | 6 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3NLBA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 5BE | Type1 | 6 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 5DLSA | 2.15 | Active | DFGin | BLAminus | in-in | in-in | 5CV | Type1 | 6 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BKNA | 2.74 | Active | DFGin | BLAminus | in-in | in-in | ADE | Type1 | 7 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BKOA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | TVW | Type1 | 7 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4QYEA | 2.05 | Active | DFGin | BLAminus | in-in | in-in | 3DL | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4QYFA | 2.15 | Active | DFGin | BLAminus | in-in | in-in | 3DV | Type1 | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4QYGA | 1.75 | Active | DFGin | BLAminus | in-in | in-in | 3DW | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4QYGB | 1.75 | Active | DFGin | BLAminus | in-in | in-in | 3DW | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4QYHA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 3DX | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4QYHB | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 3DX | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4RVKA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | 3XK | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4RVLA | 1.85 | Active | DFGin | BLAminus | in-in | in-in | 3XL | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4RVMA | 1.86 | Active | DFGin | BLAminus | in-in | in-in | 3X7 | Type1 | 3 - 273 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 7AKMA | 1.93 | Active | DFGin | BLAminus | in-in | in-in | AGS | Type1 | 2 - 271 | D10R | None | 0 |
Homo sapiens | CHK1_HUMAN | 7AKOA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | STU | Type1 | 2 - 271 | D10R | None | 0 |
Homo sapiens | CHK1_HUMAN | 7AKOB | 1.8 | Active | DFGin | BLAminus | in-in | in-in | STU | Type1 | 2 - 271 | D10R | None | 0 |
Homo sapiens | CHK1_HUMAN | 2HOGA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 710 | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2HXLA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | 422 | Type1 | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2HXQA | 2.0 | Inactive | DFGin | BLAminus | in-out | in-in | 373 | Type1 | 2 - 276 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2HY0A | 1.7 | Inactive | DFGin | BLAminus | in-out | in-in | 306 | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2QHMA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | 7CS | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2QHNA | 1.7 | Active | DFGin | BLAminus | in-in | in-in | 582 | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2R0UA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | M54 | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3TKHA | 1.79 | Active | DFGin | BLAminus | in-in | in-in | 07S | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 3TKIA | 1.6 | Active | DFGin | BLAminus | in-in | in-in | S25 | Type1 | 2 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OQ5A | 1.4 | Active | DFGin | BLAminus | in-in | in-in | 4K4 | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OQ7A | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OQ7B | 2.1 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 8 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSUA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | HK5 | Type1 | 4 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OQ6A | 1.95 | Active | DFGin | BLAminus | in-in | in-in | 4K4 | Type1 | 5 - 270 | A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OQ8A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 4 - 270 | A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OOPA | 1.7 | Inactive | DFGin | BLAminus | in-out | in-in | ANP | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OORA | 1.9 | Inactive | DFGin | BLAminus | in-out | in-in | STU | Type1 | 3 - 283 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OOTA | 2.1 | Active | DFGin | BLAminus | in-in | in-in | 4K4 | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OP2A | 1.9 | Active | DFGin | BLAminus | in-in | in-in | A0Q | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OP4A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A0T | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OP5A | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 3FE | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OP7A | 1.8 | Active | DFGin | BLAminus | in-in | in-in | A1K | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OPBA | 1.55 | Active | DFGin | BLAminus | in-in | in-in | A1N | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OPRA | 1.95 | Active | DFGin | BLAminus | in-in | in-in | A3E | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OPSA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | A3Q | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OPUA | 1.55 | Active | DFGin | BLAminus | in-in | in-in | A3K | Type1 | 3 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5OPVA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | A3H | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJDA | 2.0 | Active | DFGin | BLAminus | in-in | in-in | TVT | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJEA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | ADE | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJHA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | 42C | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJJA | 1.8 | Active | DFGin | BLAminus | in-in | in-in | TVW | Type1 | 3 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJMA | 2.3 | Inactive | DFGin | BLAminus | in-out | in-in | TW2 | Type1 | 5 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJOA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | TWK | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJRA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | TWH | Type1 | 5 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJXA | 2.4 | Active | DFGin | BLAminus | in-in | in-in | U0Q | Type1 | 8 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BJXB | 2.4 | Active | DFGin | BLAminus | in-in | in-in | U0Q | Type1 | 8 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BK1A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | U0N | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BK2A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | U0K | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7BK3A | 2.0 | Active | DFGin | BLAminus | in-in | in-in | U0T | Type1 | 5 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7MCKA | 1.65 | Active | DFGin | BLAminus | in-in | in-in | YXD | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7SUFA | 1.48 | Active | DFGin | BLAminus | in-in | in-in | BVI | Type1 | 3 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7SUGA | 1.48 | Active | DFGin | BLAminus | in-in | in-in | BWI | Type1 | 3 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7SUHA | 2.46 | Active | DFGin | BLAminus | in-in | in-in | BXI | Type1 | 4 - 270 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7SUIA | 2.119 | Active | DFGin | BLAminus | in-in | in-in | L80 | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7SUJA | 2.299 | Inactive | DFGin | BLAminus | in-out | in-in | BYL | Type1 | 9 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 7SUJB | 2.299 | Active | DFGin | BLAminus | in-in | in-in | BYL | Type1 | 9 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 8E80A | 1.49 | Active | DFGin | BLAminus | in-in | in-in | UUF | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 8E81A | 1.62 | Active | DFGin | BLAminus | in-in | in-in | UU6 | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 8SIVA | 1.759 | Active | DFGin | BLAminus | in-in | in-in | ZXH | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 8SIWA | 1.877 | Active | DFGin | BLAminus | in-in | in-in | ZXL | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 8SIWB | 1.877 | Active | DFGin | BLAminus | in-in | in-in | ZXL | Type1 | 4 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 8SIXA | 1.55 | Active | DFGin | BLAminus | in-in | in-in | ZXP | Type1 | 8 - 271 | N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S | None | 0 |
Homo sapiens | CHK1_HUMAN | 5F4NA | 1.91 | Active | DFGin | BLAminus | in-in | in-in | 5UY 5UY | Type1 Allosteric | 5 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2YM7A | 1.81 | Active | DFGin | BLAminus | in-in | in-in | YM7 YM7 | Type1 Type1 | 7 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2E9NA | 2.5 | Inactive | DFGin | BLAminus | in-out | in-in | 76A | Type1.5_Back | 2 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSTA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | HK4 | Type1.5_Back | 3 - 270 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2AYPA | 2.9 | Active | DFGin | BLAminus | in-in | in-in | 43A | Type1.5_Back | 2 - 269 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FSQA | 2.4 | Active | DFGin | BLAminus | in-in | in-in | HK3 | Type1.5_Back | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTKA | 2.3 | Active | DFGin | BLAminus | in-in | in-in | H9K | Type1.5_Back | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTLA | 2.5 | Inactive | DFGin | BLAminus | in-out | in-in | H0K | Type1.5_Back | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTMA | 1.9 | Active | DFGin | BLAminus | in-in | in-in | 1HK | Type1.5_Back | 3 - 280 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 4FTNA | 2.02 | Active | DFGin | BLAminus | in-in | in-in | 2HK | Type1.5_Back | 3 - 271 | None | None | 0 |
Homo sapiens | CHK1_HUMAN | 2C3KA | 2.6 | Active | DFGin | BLAminus | in-in | in-in | ABO | Type1.5_Back | 6 - 270 | None | None | 0 |