Ligand: IRG

Total number of chains: 10
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
None None 4 40.0% 4EH3A
DFGin None 2 20.0% 4EH4A
DFGinter None 2 20.0% 4EHVA
DFGin BLBplus 1 10.0% 4EH2A
DFGout None 1 10.0% 4EH8A

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC MAPK14 MK14_HUMAN 4EH2A Q16539 4 354 360.0 IRG:401,0OK:402 Allosteric,Type1 Inactive DFGin 5.0488 13.9493 BLBplus -117.8, 162.51 72.3, 21.2 -57.69, 163.34 31.01, 95.16 92.75, 999.0 in-in in 9.39 Saltbr-in 2.9127 HRD-in -68.61, -52.99 79.87, -17.03 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 104.22 APE9-dihe-na -64.21, 119.38 APE8-dihe-out -37.73, -46.13 APE8-rot-in 267.35 APE67-dihe-in -65.75, -23.42 -54.51, -28.85 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.4245 None None None XRAY 2.0 0.226 0.274 A 360.0 337.0 14 25 13 12 [[24, 308]] 1.0 4eh2 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4DLIA Q16539 5 354 360.0 IRG:401,IRG:402 Allosteric,Allosteric Inactive DFGin 9.8147 11.8562 None -104.36, 150.39 -73.0, -47.15 -137.92, 126.59 314.79, 100.08 -44.68, 999.0 in-in in 9.4387 Saltbr-in 2.8448 HRD-in -68.95, -53.08 77.7, -11.22 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 123.1 APE9-dihe-na -70.95, 129.15 APE8-dihe-out -52.5, -43.49 APE8-rot-in 288.97 APE67-dihe-in -64.32, -23.54 -55.51, -29.37 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.0955 None None None XRAY 1.91 0.216 0.255 A 360.0 334.0 16 25 13 12 [[24, 308]] 1.0 4dli CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH4A Q16539 4 354 360.0 IRG:401,0OL:402 Allosteric,Type1 Inactive DFGin 10.8466 12.1969 None -91.43, 145.17 -57.64, -47.01 -148.78, 133.96 289.87, 102.95 -106.02, 178.5 in-in in 9.3455 Saltbr-in 3.5333 HRD-in -75.34, -49.4 79.8, -22.99 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 89.91 APE9-dihe-na -88.64, 150.01 APE8-dihe-out -60.61, -41.02 APE8-rot-in 254.43 APE67-dihe-in -62.83, -20.65 -63.82, -26.94 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 10.1023 APE9-dist-out 11.2223 None None None XRAY 2.5 0.234 0.317 A 360.0 337.0 14 25 15 10 [[24, 308]] 1.0 4eh4 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH9A Q16539 5 354 360.0 IRG:401,0OQ:402 Allosteric,Type3 Inactive DFGinter 10.8996 6.2057 None -97.42, 159.57 -62.33, -60.46 -150.13, 147.17 64.11, 82.71 -78.55, 25.4 in-out in 9.4044 Saltbr-out 4.5758 HRD-in -71.05, -53.71 82.13, -21.54 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 115.29 APE9-dihe-na -99.26, 134.28 APE8-dihe-out -59.4, -32.47 APE8-rot-in 294.18 APE67-dihe-in -64.19, -25.37 -57.95, -25.13 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 12.356 APE9-dist-out 11.8242 None None None XRAY 2.1 0.232 0.28 A 360.0 334.0 16 25 14 11 [[24, 308]] 1.0 4eh9 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EHVA Q16539 5 352 360.0 0SJ:401,0SJ:402,IRG:403,0SJ:404 Type3,Allosteric,Allosteric,Allosteric Inactive DFGinter 10.9229 6.2755 None -99.66, 162.35 -69.64, -55.96 -152.93, 157.53 62.39, 91.72 -108.25, -179.88 in-none in 9.2374 Saltbr-none 999.0 HRD-in -69.34, -50.13 82.95, -13.29 none-none-out SNCnno none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 107.52 APE9-dihe-na -78.18, 127.1 APE8-dihe-out -52.4, -41.18 APE8-rot-in 282.24 APE67-dihe-in -64.93, -23.91 -55.78, -30.86 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 9.946 APE9-dist-out 11.0047 None None None XRAY 1.6 0.223 0.252 A 360.0 337.0 11 25 14 11 [[24, 308]] 1.0 4ehv CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH8A Q16539 4 354 360.0 IRG:401,0OP:402,0OP:403 Allosteric,Type3,Type1 Inactive DFGout 11.6887 12.5312 None -126.98, -173.26 -129.13, 140.31 68.37, 999.0 306.63, 121.42 999.0, 999.0 in-in in 9.382 Saltbr-in 3.0908 HRD-in -73.46, -51.4 85.92, -19.81 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 158.35 APE9-dihe-na -105.67, 133.81 APE8-dihe-out -60.04, -38.46 APE8-rot-in 291.54 APE67-dihe-in -62.35, -25.05 -51.18, -35.54 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.2127 None None None XRAY 2.2 0.242 0.282 A 360.0 336.0 15 25 12 13 [[24, 308]] 1.0 4eh8 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH5A Q16539 4 354 360.0 IRG:401,0OM:402 Allosteric,Type1 Inactive None 999.0 999.0 None -108.39, 163.33 57.95, 999.0 999.0, 999.0 999.0, 999.0 999.0, 999.0 in-in in 9.3088 Saltbr-in 2.9014 HRD-in -72.32, -49.67 77.23, -19.04 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 134.62 APE8-dihe-out -54.92, -38.6 APE8-rot-in 283.85 APE67-dihe-in -62.06, -24.82 -60.96, -29.32 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.251 None None None XRAY 2.0 0.232 0.285 A 360.0 329.0 22 25 10 15 [[24, 308]] 1.0 4eh5 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH6A Q16539 4 354 360.0 IRG:401,0ON:402 Allosteric,Type1 Inactive None 999.0 999.0 None -123.46, -172.29 -120.99, 34.21 -158.17, 999.0 999.0, 999.0 999.0, 999.0 in-in in 9.1714 Saltbr-in 2.742 HRD-in -69.9, -51.68 78.55, -21.68 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 141.55 APE8-dihe-out -58.14, -38.92 APE8-rot-in 265.12 APE67-dihe-in -64.71, -26.03 -57.04, -28.73 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.2302 None None None XRAY 2.1 0.227 0.277 A 360.0 335.0 16 25 11 14 [[24, 308]] 1.0 4eh6 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH7A Q16539 4 354 360.0 IRG:401,0OO:402 Allosteric,Type1 Inactive None 999.0 999.0 None -98.76, 137.9 -63.12, -45.22 -156.84, 139.66 999.0, 999.0 98.21, 999.0 in-in in 9.2463 Saltbr-in 3.0514 HRD-in -69.27, -51.42 76.94, -19.49 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 98.3 APE9-dihe-na -75.8, 145.15 APE8-dihe-out -61.37, -38.48 APE8-rot-in 268.7 APE67-dihe-in -62.89, -26.04 -57.18, -28.26 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.3386 None None None XRAY 2.1 0.224 0.265 A 360.0 337.0 14 25 13 12 [[24, 308]] 1.0 4eh7 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH3A Q16539 4 354 360.0 NAR:401,IRG:402 Type1,Allosteric Inactive None 999.0 999.0 None -93.8, 152.76 -77.66, -36.64 -150.96, 113.75 999.0, 999.0 -75.95, -166.36 in-out in 9.6206 Saltbr-out 4.0293 HRD-in -80.03, -53.65 83.21, -19.96 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 103.56 APE9-dihe-na -87.37, 152.3 APE8-dihe-out -66.91, -31.74 APE8-rot-in 263.06 APE67-dihe-in -67.51, -22.33 -71.06, -17.46 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 10.9391 APE9-dist-out 11.2796 None None None XRAY 2.4 0.219 0.277 A 360.0 339.0 12 25 15 10 [[24, 308]] 1.0 4eh3 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14

Ligand: IRG

Total number of chains: 10
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
None None 4 40.0% 4EH3A
DFGin None 2 20.0% 4EH4A
DFGinter None 2 20.0% 4EHVA
DFGin BLBplus 1 10.0% 4EH2A
DFGout None 1 10.0% 4EH8A

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC MAPK14 MK14_HUMAN 4EH2A Q16539 4 354 360.0 IRG:401,0OK:402 Allosteric,Type1 Inactive DFGin 5.0488 13.9493 BLBplus -117.8, 162.51 72.3, 21.2 -57.69, 163.34 31.01, 95.16 92.75, 999.0 in-in in 9.39 Saltbr-in 2.9127 HRD-in -68.61, -52.99 79.87, -17.03 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 104.22 APE9-dihe-na -64.21, 119.38 APE8-dihe-out -37.73, -46.13 APE8-rot-in 267.35 APE67-dihe-in -65.75, -23.42 -54.51, -28.85 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.4245 None None None XRAY 2.0 0.226 0.274 A 360.0 337.0 14 25 13 12 [[24, 308]] 1.0 4eh2 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4DLIA Q16539 5 354 360.0 IRG:401,IRG:402 Allosteric,Allosteric Inactive DFGin 9.8147 11.8562 None -104.36, 150.39 -73.0, -47.15 -137.92, 126.59 314.79, 100.08 -44.68, 999.0 in-in in 9.4387 Saltbr-in 2.8448 HRD-in -68.95, -53.08 77.7, -11.22 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 123.1 APE9-dihe-na -70.95, 129.15 APE8-dihe-out -52.5, -43.49 APE8-rot-in 288.97 APE67-dihe-in -64.32, -23.54 -55.51, -29.37 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.0955 None None None XRAY 1.91 0.216 0.255 A 360.0 334.0 16 25 13 12 [[24, 308]] 1.0 4dli Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH4A Q16539 4 354 360.0 IRG:401,0OL:402 Allosteric,Type1 Inactive DFGin 10.8466 12.1969 None -91.43, 145.17 -57.64, -47.01 -148.78, 133.96 289.87, 102.95 -106.02, 178.5 in-in in 9.3455 Saltbr-in 3.5333 HRD-in -75.34, -49.4 79.8, -22.99 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 89.91 APE9-dihe-na -88.64, 150.01 APE8-dihe-out -60.61, -41.02 APE8-rot-in 254.43 APE67-dihe-in -62.83, -20.65 -63.82, -26.94 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 10.1023 APE9-dist-out 11.2223 None None None XRAY 2.5 0.234 0.317 A 360.0 337.0 14 25 15 10 [[24, 308]] 1.0 4eh4 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH9A Q16539 5 354 360.0 IRG:401,0OQ:402 Allosteric,Type3 Inactive DFGinter 10.8996 6.2057 None -97.42, 159.57 -62.33, -60.46 -150.13, 147.17 64.11, 82.71 -78.55, 25.4 in-out in 9.4044 Saltbr-out 4.5758 HRD-in -71.05, -53.71 82.13, -21.54 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 115.29 APE9-dihe-na -99.26, 134.28 APE8-dihe-out -59.4, -32.47 APE8-rot-in 294.18 APE67-dihe-in -64.19, -25.37 -57.95, -25.13 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 12.356 APE9-dist-out 11.8242 None None None XRAY 2.1 0.232 0.28 A 360.0 334.0 16 25 14 11 [[24, 308]] 1.0 4eh9 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EHVA Q16539 5 352 360.0 0SJ:401,0SJ:402,IRG:403,0SJ:404 Type3,Allosteric,Allosteric,Allosteric Inactive DFGinter 10.9229 6.2755 None -99.66, 162.35 -69.64, -55.96 -152.93, 157.53 62.39, 91.72 -108.25, -179.88 in-none in 9.2374 Saltbr-none 999.0 HRD-in -69.34, -50.13 82.95, -13.29 none-none-out SNCnno none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 107.52 APE9-dihe-na -78.18, 127.1 APE8-dihe-out -52.4, -41.18 APE8-rot-in 282.24 APE67-dihe-in -64.93, -23.91 -55.78, -30.86 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 9.946 APE9-dist-out 11.0047 None None None XRAY 1.6 0.223 0.252 A 360.0 337.0 11 25 14 11 [[24, 308]] 1.0 4ehv Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH8A Q16539 4 354 360.0 IRG:401,0OP:402,0OP:403 Allosteric,Type3,Type1 Inactive DFGout 11.6887 12.5312 None -126.98, -173.26 -129.13, 140.31 68.37, 999.0 306.63, 121.42 999.0, 999.0 in-in in 9.382 Saltbr-in 3.0908 HRD-in -73.46, -51.4 85.92, -19.81 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 158.35 APE9-dihe-na -105.67, 133.81 APE8-dihe-out -60.04, -38.46 APE8-rot-in 291.54 APE67-dihe-in -62.35, -25.05 -51.18, -35.54 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.2127 None None None XRAY 2.2 0.242 0.282 A 360.0 336.0 15 25 12 13 [[24, 308]] 1.0 4eh8 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH5A Q16539 4 354 360.0 IRG:401,0OM:402 Allosteric,Type1 Inactive None 999.0 999.0 None -108.39, 163.33 57.95, 999.0 999.0, 999.0 999.0, 999.0 999.0, 999.0 in-in in 9.3088 Saltbr-in 2.9014 HRD-in -72.32, -49.67 77.23, -19.04 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 134.62 APE8-dihe-out -54.92, -38.6 APE8-rot-in 283.85 APE67-dihe-in -62.06, -24.82 -60.96, -29.32 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.251 None None None XRAY 2.0 0.232 0.285 A 360.0 329.0 22 25 10 15 [[24, 308]] 1.0 4eh5 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH6A Q16539 4 354 360.0 IRG:401,0ON:402 Allosteric,Type1 Inactive None 999.0 999.0 None -123.46, -172.29 -120.99, 34.21 -158.17, 999.0 999.0, 999.0 999.0, 999.0 in-in in 9.1714 Saltbr-in 2.742 HRD-in -69.9, -51.68 78.55, -21.68 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 141.55 APE8-dihe-out -58.14, -38.92 APE8-rot-in 265.12 APE67-dihe-in -64.71, -26.03 -57.04, -28.73 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.2302 None None None XRAY 2.1 0.227 0.277 A 360.0 335.0 16 25 11 14 [[24, 308]] 1.0 4eh6 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH7A Q16539 4 354 360.0 IRG:401,0OO:402 Allosteric,Type1 Inactive None 999.0 999.0 None -98.76, 137.9 -63.12, -45.22 -156.84, 139.66 999.0, 999.0 98.21, 999.0 in-in in 9.2463 Saltbr-in 3.0514 HRD-in -69.27, -51.42 76.94, -19.49 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 98.3 APE9-dihe-na -75.8, 145.15 APE8-dihe-out -61.37, -38.48 APE8-rot-in 268.7 APE67-dihe-in -62.89, -26.04 -57.18, -28.26 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.3386 None None None XRAY 2.1 0.224 0.265 A 360.0 337.0 14 25 13 12 [[24, 308]] 1.0 4eh7 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 4EH3A Q16539 4 354 360.0 NAR:401,IRG:402 Type1,Allosteric Inactive None 999.0 999.0 None -93.8, 152.76 -77.66, -36.64 -150.96, 113.75 999.0, 999.0 -75.95, -166.36 in-out in 9.6206 Saltbr-out 4.0293 HRD-in -80.03, -53.65 83.21, -19.96 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 103.56 APE9-dihe-na -87.37, 152.3 APE8-dihe-out -66.91, -31.74 APE8-rot-in 263.06 APE67-dihe-in -67.51, -22.33 -71.06, -17.46 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 10.9391 APE9-dist-out 11.2796 None None None XRAY 2.4 0.219 0.277 A 360.0 339.0 12 25 15 10 [[24, 308]] 1.0 4eh3 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1.0 301.0 301.0 167 168 169 171 173 53 71 75 147 149 148 150.0 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14

Ligand: IRG

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name