| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| OTHER | PKMYT1 | PMYT1_HUMAN | 5VCXA | Q99640 | 75 | 361 | 499.0 | H8H:401 | Type1 | Inactive | DFGin | 5.9448 | 14.566 | BLAminus | -133.1, -159.74 | 56.06, 76.15 | -98.03, 28.4 | 300.17, 108.44 | -60.31, -33.85 | in-in | in | 8.9959 | Saltbr-in | 3.0634 | HRD-in | -70.1, -45.94 | 70.27, -2.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0515 | ActLoopCT-out | nonTYR | APEdihe_aaiai | APEdist_iooi | APE10-dihe-na | -72.13, 165.11 | APE9-dihe-na | -95.53, -151.65 | APE8-dihe-in | -59.58, 124.62 | APE8-rot-na | 194.34 | APE67-dihe-in | -61.23, -27.43 | -59.74, -28.49 | APE12-dist-in | 7.8512 | APE11-dist-out | 6.3134 | APE10-dist-out | 9.3734 | APE9-dist-in | 3.3043 | None | None | None | XRAY | 2.7 | 0.201 | 0.244 | A | 311.0 | 287.0 | 0 | 27 | 27 | 0 | [[110, 359]] | 1.0 | 5vcx | OTHER_PKMYT1_HUMAN | STE | 9.9e-39 | 139.4 | 1.0 | 255.0 | 255.0 | 250 | 251 | 252 | 254 | 256 | 139 | 157 | 161 | 230 | 232 | 231 | 233.0 | 288 | 277 | 272 | 271 | 270 | 269 | 268 | 267 | 266 | 188 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| OTHER | PKMYT1 | PMYT1_HUMAN | 5VD3A | Q99640 | 78 | 360 | 499.0 | H8H:60401 | Type1 | Inactive | DFGin | 5.988 | 14.4248 | BLAminus | -136.31, -163.22 | 68.56, 66.31 | -95.1, 21.81 | 295.33, 125.87 | -68.4, -23.33 | in-in | in | 8.4946 | Saltbr-in | 2.6731 | HRD-in | -69.52, -49.09 | 74.0, 4.67 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9079 | ActLoopCT-out | nonTYR | APEdihe_aaiai | APEdist_iooi | APE10-dihe-na | -97.34, 136.82 | APE9-dihe-na | -76.5, -172.94 | APE8-dihe-in | -60.8, 125.68 | APE8-rot-na | 188.67 | APE67-dihe-in | -61.07, -31.05 | -63.33, -22.08 | APE12-dist-in | 7.6901 | APE11-dist-out | 5.948 | APE10-dist-out | 9.3375 | APE9-dist-in | 3.5904 | None | None | None | XRAY | 1.8 | 0.167 | 0.204 | A | 311.0 | 283.0 | 0 | 27 | 27 | 0 | [[110, 359]] | 1.0 | 5vd3 | OTHER_PKMYT1_HUMAN | STE | 9.9e-39 | 139.4 | 1.0 | 255.0 | 255.0 | 250 | 251 | 252 | 254 | 256 | 139 | 157 | 161 | 230 | 232 | 231 | 233.0 | 288 | 277 | 272 | 271 | 270 | 269 | 268 | 267 | 266 | 188 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| STE | STK24 | STK24_HUMAN | 4QMXA | Q9Y6E0 | 24 | 311 | 443.0 | H8H:60401 | Type1 | Active | DFGin | 6.9146 | 15.2182 | BLAminus | -132.03, 170.35 | 60.05, 85.66 | -98.54, 25.16 | 282.88, 75.66 | -58.11, -25.51 | in-in | in | 8.9595 | Saltbr-in | 2.7307 | HRD-in | -69.57, -50.6 | 71.02, 5.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7507 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.76, 159.44 | APE9-dihe-na | 124.78, -161.46 | APE8-dihe-in | -119.38, 119.23 | APE8-rot-in | 305.8 | APE67-dihe-in | -56.19, -29.84 | -38.71, -52.83 | APE12-dist-in | 8.3116 | APE11-dist-in | 10.9571 | APE10-dist-in | 5.1773 | APE9-dist-in | 3.2554 | None | TPO190 | TPO190 | XRAY | 1.882 | 0.179 | 0.218 | A | 310.0 | 288.0 | 0 | 28 | 28 | 0 | [[36, 286]] | 1.0 | 4qmx | STE_STK24_HUMAN | STE | 3.9e-100 | 340.4 | 1.0 | 257.0 | 257.0 | 173 | 174 | 175 | 177 | 179 | 65 | 82 | 86 | 153 | 155 | 154 | 156.0 | 213 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 112 | Serine/threonine-protein kinase 24 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCA | Q04771 | 205 | 499 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 7.6808 | 12.7079 | ABAminus | -107.89, -60.92 | -94.08, 111.73 | -110.3, 16.97 | 303.67, 166.99 | -67.99, -29.57 | in-out | in | 8.6609 | Saltbr-out | 4.5318 | HRD-in | -76.83, -55.96 | 76.97, 3.64 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9026 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -97.86, 149.98 | APE9-dihe-na | 117.18, 157.89 | APE8-dihe-in | -61.4, 123.56 | APE8-rot-in | 297.81 | APE67-dihe-in | -59.38, -25.03 | -58.82, -36.53 | APE12-dist-in | 12.2539 | APE11-dist-in | 12.3679 | APE10-dist-in | 6.6349 | APE9-dist-in | 4.2434 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | A | 301.0 | 292.0 | 3 | 32 | 29 | 3 | [[207, 497]] | 1.0 | 6zgc | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCB | Q04771 | 203 | 499 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 8.0586 | 13.0758 | ABAminus | -110.37, -58.89 | -92.47, 102.08 | -108.51, 23.12 | 297.16, 160.33 | -68.67, -30.3 | in-out | in | 8.5094 | Saltbr-out | 4.0893 | HRD-in | -75.39, -56.68 | 79.53, 2.12 | out-in-none | SNCoin | in-none | ActLoopNT-in | 3.0574 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -104.09, -8.88 | APE9-dihe-na | -69.88, 178.01 | APE8-dihe-in | -69.34, 130.54 | APE8-rot-in | 309.97 | APE67-dihe-in | -59.99, -26.01 | -62.71, -39.0 | APE12-dist-none | 999.0 | APE11-dist-in | 11.4985 | APE10-dist-in | 6.6932 | APE9-dist-in | 3.9531 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | B | 301.0 | 291.0 | 6 | 32 | 27 | 5 | [[207, 497]] | 1.0 | 6zgc | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCC | Q04771 | 201 | 498 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 7.6488 | 13.123 | ABAminus | -111.55, -59.07 | -96.03, 103.07 | -100.54, 20.17 | 312.53, 170.02 | -62.85, -32.84 | in-none | in | 8.7179 | Saltbr-none | 999.0 | HRD-in | -78.56, -58.95 | 79.27, 6.55 | none-in-out | SNCnio | in-out | ActLoopNT-in | 3.0338 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -126.95, 173.39 | APE9-dihe-na | -60.53, 177.19 | APE8-dihe-in | -72.99, 133.32 | APE8-rot-in | 299.82 | APE67-dihe-in | -70.68, -22.46 | -67.18, -24.36 | APE12-dist-in | 10.3742 | APE11-dist-out | 7.4875 | APE10-dist-out | 8.4624 | APE9-dist-in | 3.9174 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | C | 301.0 | 296.0 | 2 | 32 | 30 | 2 | [[207, 497]] | 1.0 | 6zgc | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCD | Q04771 | 203 | 498 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 8.1291 | 12.9873 | ABAminus | -118.4, -60.05 | -92.31, 105.89 | -107.46, 26.29 | 296.86, 166.24 | -65.26, -28.18 | in-out | in | 8.4011 | Saltbr-out | 3.9875 | HRD-in | -73.86, -57.34 | 80.97, -1.67 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.024 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.47, 108.31 | APE9-dihe-na | 164.09, 161.61 | APE8-dihe-in | -63.97, 128.7 | APE8-rot-in | 301.77 | APE67-dihe-in | -60.64, -22.49 | -67.87, -34.64 | APE12-dist-in | 12.4999 | APE11-dist-in | 11.8523 | APE10-dist-in | 6.4627 | APE9-dist-in | 4.0328 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | D | 301.0 | 291.0 | 5 | 32 | 29 | 3 | [[207, 497]] | 1.0 | 6zgc | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TYR | SRC | SRC_HUMAN | 2H8HA | P12931 | 88 | 532 | 536.0 | H8H:60534 | Type1 | Inactive | DFGin | 6.2056 | 12.9819 | BLBplus | -115.05, 164.5 | 78.38, 19.66 | -80.35, 138.41 | 38.05, 100.6 | 107.76, -33.37 | out-out | out | 13.8527 | Saltbr-out | 13.575 | HRD-in | -77.24, -52.16 | 75.83, -8.86 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.221 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -87.67, -13.19 | APE9-dihe-in | -104.38, 132.48 | APE8-dihe-in | -86.38, 72.02 | APE8-rot-na | 33.02 | APE67-dihe-in | -72.18, -20.32 | -60.54, -27.69 | APE12-dist-na | 17.2384 | APE11-dist-na | 18.2049 | APE10-dist-na | 12.8167 | APE9-dist-out | 8.5094 | None | PTR530 | PTR530 | XRAY | 2.2 | 0.207 | 0.272 | A | 535.0 | 445.0 | 0 | 29 | 29 | 0 | [[270, 521]] | 1.0 | 2h8h | TYR_SRC_HUMAN | TYR | 1e-93 | 319.5 | 1.0 | 260.0 | 260.0 | 406 | 407 | 408 | 410 | 412 | 298 | 313 | 317 | 386 | 388 | 387 | 389.0 | 447 | 435 | 430 | 429 | 428 | 427 | 426 | 425 | 424 | 342 | Proto-oncogene tyrosine-protein kinase Src |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| OTHER | PKMYT1 | PMYT1_HUMAN | 5VCXA | Q99640 | 75 | 361 | 499.0 | H8H:401 | Type1 | Inactive | DFGin | 5.9448 | 14.566 | BLAminus | -133.1, -159.74 | 56.06, 76.15 | -98.03, 28.4 | 300.17, 108.44 | -60.31, -33.85 | in-in | in | 8.9959 | Saltbr-in | 3.0634 | HRD-in | -70.1, -45.94 | 70.27, -2.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0515 | ActLoopCT-out | nonTYR | APEdihe_aaiai | APEdist_iooi | APE10-dihe-na | -72.13, 165.11 | APE9-dihe-na | -95.53, -151.65 | APE8-dihe-in | -59.58, 124.62 | APE8-rot-na | 194.34 | APE67-dihe-in | -61.23, -27.43 | -59.74, -28.49 | APE12-dist-in | 7.8512 | APE11-dist-out | 6.3134 | APE10-dist-out | 9.3734 | APE9-dist-in | 3.3043 | None | None | None | XRAY | 2.7 | 0.201 | 0.244 | A | 311.0 | 287.0 | 0 | 27 | 27 | 0 | [[110, 359]] | 1.0 | 5vcx | Homo sapiens | OTHER_PKMYT1_HUMAN | STE | 9.9e-39 | 139.4 | 1.0 | 255.0 | 255.0 | 250 | 251 | 252 | 254 | 256 | 139 | 157 | 161 | 230 | 232 | 231 | 233.0 | 288 | 277 | 272 | 271 | 270 | 269 | 268 | 267 | 266 | 188 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| OTHER | PKMYT1 | PMYT1_HUMAN | 5VD3A | Q99640 | 78 | 360 | 499.0 | H8H:60401 | Type1 | Inactive | DFGin | 5.988 | 14.4248 | BLAminus | -136.31, -163.22 | 68.56, 66.31 | -95.1, 21.81 | 295.33, 125.87 | -68.4, -23.33 | in-in | in | 8.4946 | Saltbr-in | 2.6731 | HRD-in | -69.52, -49.09 | 74.0, 4.67 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9079 | ActLoopCT-out | nonTYR | APEdihe_aaiai | APEdist_iooi | APE10-dihe-na | -97.34, 136.82 | APE9-dihe-na | -76.5, -172.94 | APE8-dihe-in | -60.8, 125.68 | APE8-rot-na | 188.67 | APE67-dihe-in | -61.07, -31.05 | -63.33, -22.08 | APE12-dist-in | 7.6901 | APE11-dist-out | 5.948 | APE10-dist-out | 9.3375 | APE9-dist-in | 3.5904 | None | None | None | XRAY | 1.8 | 0.167 | 0.204 | A | 311.0 | 283.0 | 0 | 27 | 27 | 0 | [[110, 359]] | 1.0 | 5vd3 | Homo sapiens | OTHER_PKMYT1_HUMAN | STE | 9.9e-39 | 139.4 | 1.0 | 255.0 | 255.0 | 250 | 251 | 252 | 254 | 256 | 139 | 157 | 161 | 230 | 232 | 231 | 233.0 | 288 | 277 | 272 | 271 | 270 | 269 | 268 | 267 | 266 | 188 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| STE | STK24 | STK24_HUMAN | 4QMXA | Q9Y6E0 | 24 | 311 | 443.0 | H8H:60401 | Type1 | Active | DFGin | 6.9146 | 15.2182 | BLAminus | -132.03, 170.35 | 60.05, 85.66 | -98.54, 25.16 | 282.88, 75.66 | -58.11, -25.51 | in-in | in | 8.9595 | Saltbr-in | 2.7307 | HRD-in | -69.57, -50.6 | 71.02, 5.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7507 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.76, 159.44 | APE9-dihe-na | 124.78, -161.46 | APE8-dihe-in | -119.38, 119.23 | APE8-rot-in | 305.8 | APE67-dihe-in | -56.19, -29.84 | -38.71, -52.83 | APE12-dist-in | 8.3116 | APE11-dist-in | 10.9571 | APE10-dist-in | 5.1773 | APE9-dist-in | 3.2554 | None | TPO190 | TPO190 | XRAY | 1.882 | 0.179 | 0.218 | A | 310.0 | 288.0 | 0 | 28 | 28 | 0 | [[36, 286]] | 1.0 | 4qmx | Homo sapiens | STE_STK24_HUMAN | STE | 3.9e-100 | 340.4 | 1.0 | 257.0 | 257.0 | 173 | 174 | 175 | 177 | 179 | 65 | 82 | 86 | 153 | 155 | 154 | 156.0 | 213 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 112 | Serine/threonine-protein kinase 24 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCA | Q04771 | 205 | 499 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 7.6808 | 12.7079 | ABAminus | -107.89, -60.92 | -94.08, 111.73 | -110.3, 16.97 | 303.67, 166.99 | -67.99, -29.57 | in-out | in | 8.6609 | Saltbr-out | 4.5318 | HRD-in | -76.83, -55.96 | 76.97, 3.64 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9026 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -97.86, 149.98 | APE9-dihe-na | 117.18, 157.89 | APE8-dihe-in | -61.4, 123.56 | APE8-rot-in | 297.81 | APE67-dihe-in | -59.38, -25.03 | -58.82, -36.53 | APE12-dist-in | 12.2539 | APE11-dist-in | 12.3679 | APE10-dist-in | 6.6349 | APE9-dist-in | 4.2434 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | A | 301.0 | 292.0 | 3 | 32 | 29 | 3 | [[207, 497]] | 1.0 | 6zgc | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCB | Q04771 | 203 | 499 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 8.0586 | 13.0758 | ABAminus | -110.37, -58.89 | -92.47, 102.08 | -108.51, 23.12 | 297.16, 160.33 | -68.67, -30.3 | in-out | in | 8.5094 | Saltbr-out | 4.0893 | HRD-in | -75.39, -56.68 | 79.53, 2.12 | out-in-none | SNCoin | in-none | ActLoopNT-in | 3.0574 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -104.09, -8.88 | APE9-dihe-na | -69.88, 178.01 | APE8-dihe-in | -69.34, 130.54 | APE8-rot-in | 309.97 | APE67-dihe-in | -59.99, -26.01 | -62.71, -39.0 | APE12-dist-none | 999.0 | APE11-dist-in | 11.4985 | APE10-dist-in | 6.6932 | APE9-dist-in | 3.9531 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | B | 301.0 | 291.0 | 6 | 32 | 27 | 5 | [[207, 497]] | 1.0 | 6zgc | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCC | Q04771 | 201 | 498 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 7.6488 | 13.123 | ABAminus | -111.55, -59.07 | -96.03, 103.07 | -100.54, 20.17 | 312.53, 170.02 | -62.85, -32.84 | in-none | in | 8.7179 | Saltbr-none | 999.0 | HRD-in | -78.56, -58.95 | 79.27, 6.55 | none-in-out | SNCnio | in-out | ActLoopNT-in | 3.0338 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -126.95, 173.39 | APE9-dihe-na | -60.53, 177.19 | APE8-dihe-in | -72.99, 133.32 | APE8-rot-in | 299.82 | APE67-dihe-in | -70.68, -22.46 | -67.18, -24.36 | APE12-dist-in | 10.3742 | APE11-dist-out | 7.4875 | APE10-dist-out | 8.4624 | APE9-dist-in | 3.9174 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | C | 301.0 | 296.0 | 2 | 32 | 30 | 2 | [[207, 497]] | 1.0 | 6zgc | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TKL | ACVR1 | ACVR1_HUMAN | 6ZGCD | Q04771 | 203 | 498 | 509.0 | H8H:501 | Type1 | Inactive | DFGin | 8.1291 | 12.9873 | ABAminus | -118.4, -60.05 | -92.31, 105.89 | -107.46, 26.29 | 296.86, 166.24 | -65.26, -28.18 | in-out | in | 8.4011 | Saltbr-out | 3.9875 | HRD-in | -73.86, -57.34 | 80.97, -1.67 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.024 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.47, 108.31 | APE9-dihe-na | 164.09, 161.61 | APE8-dihe-in | -63.97, 128.7 | APE8-rot-in | 301.77 | APE67-dihe-in | -60.64, -22.49 | -67.87, -34.64 | APE12-dist-in | 12.4999 | APE11-dist-in | 11.8523 | APE10-dist-in | 6.4627 | APE9-dist-in | 4.0328 | Q207D | None | None | XRAY | 2.67 | 0.215 | 0.26 | D | 301.0 | 291.0 | 5 | 32 | 29 | 3 | [[207, 497]] | 1.0 | 6zgc | Homo sapiens | TKL_ACVR1_HUMAN | TKL | 1.9e-85 | 292.5 | 2.0 | 267.0 | 266.0 | 353 | 354 | 355 | 357 | 359 | 235 | 248 | 252 | 333 | 335 | 334 | 336.0 | 403 | 385 | 380 | 379 | 378 | 377 | 376 | 375 | 374 | 284 | Activin receptor type-1 |
| TYR | SRC | SRC_HUMAN | 2H8HA | P12931 | 88 | 532 | 536.0 | H8H:60534 | Type1 | Inactive | DFGin | 6.2056 | 12.9819 | BLBplus | -115.05, 164.5 | 78.38, 19.66 | -80.35, 138.41 | 38.05, 100.6 | 107.76, -33.37 | out-out | out | 13.8527 | Saltbr-out | 13.575 | HRD-in | -77.24, -52.16 | 75.83, -8.86 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.221 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -87.67, -13.19 | APE9-dihe-in | -104.38, 132.48 | APE8-dihe-in | -86.38, 72.02 | APE8-rot-na | 33.02 | APE67-dihe-in | -72.18, -20.32 | -60.54, -27.69 | APE12-dist-na | 17.2384 | APE11-dist-na | 18.2049 | APE10-dist-na | 12.8167 | APE9-dist-out | 8.5094 | None | PTR530 | PTR530 | XRAY | 2.2 | 0.207 | 0.272 | A | 535.0 | 445.0 | 0 | 29 | 29 | 0 | [[270, 521]] | 1.0 | 2h8h | Homo sapiens | TYR_SRC_HUMAN | TYR | 1e-93 | 319.5 | 1.0 | 260.0 | 260.0 | 406 | 407 | 408 | 410 | 412 | 298 | 313 | 317 | 386 | 388 | 387 | 389.0 | 447 | 435 | 430 | 429 | 428 | 427 | 426 | 425 | 424 | 342 | Proto-oncogene tyrosine-protein kinase Src |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|