Ligand: BMU

Total number of chains: 6
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGout None 3 50.0% 3O8TA
DFGout BBAminus 2 33.3% 3O8UA
DFGin None 1 16.7% 3O8PA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC MAPK14 MK14_HUMAN 3O8PA Q16539 5 351 360.0 BMU:361 Type1 Inactive DFGin 10.863 12.014 None -115.52, 162.58 -99.08, -26.53 -122.71, 117.21 291.85, 138.97 -42.63, -102.67 in-out in 9.092 Saltbr-out 5.085 HRD-in -69.17, -52.21 73.92, -4.49 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 3.16 APE9-dihe-na -166.83, -167.55 APE8-dihe-out -116.39, -25.53 APE8-rot-in 271.29 APE67-dihe-in -61.81, -26.71 -69.76, -21.19 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 12.159 APE9-dist-out 10.453 D168G None None XRAY 2.1 0.218 0.276 A 360 336 11 0 0 11 [[24, 308]] 1.0 3o8p CMGC_MAPK14_HUMAN CMGC 2.7e-83 285.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3O8UA Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 13.796 9.306 BBAminus -146.29, -170.4 -144.05, 102.12 -67.29, -15.97 286.91, 115.68 99.79, 999.0 in-in in 9.331 Saltbr-in 3.364 HRD-in -63.28, -51.7 74.53, -20.43 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 144.38 APE8-dihe-out -70.85, -30.66 APE8-rot-in 258.69 APE67-dihe-in -65.11, -25.9 -59.1, -20.9 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 12.104 F169Y None None XRAY 2.1 0.224 0.285 A 360 332 16 0 0 13 [[24, 308]] 1.0 3o8u CMGC_MAPK14_HUMAN CMGC 3.3e-84 288.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3OBJA Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 14.513 11.366 BBAminus -154.08, -178.49 -133.48, 111.98 -61.66, -36.04 255.28, 56.42 -103.05, -92.49 in-out in 9.304 Saltbr-out 5.802 HRD-in -72.07, -52.81 76.05, -16.45 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 143.04 APE8-dihe-out -70.24, -30.65 APE8-rot-out 197.91 APE67-dihe-in -70.14, -17.15 -63.21, -16.69 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.973 F169R None None XRAY 2.4 0.22 0.287 A 360 332 16 0 0 12 [[24, 308]] 1.0 3obj CMGC_MAPK14_HUMAN CMGC 2e-83 286.1 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 1KV1A Q16539 5 352 360.0 BMU:391 Type3 Inactive DFGout 13.635 9.556 None -159.24, -177.02 -146.07, 100.83 -75.42, -134.45 282.12, 117.71 154.13, 999.0 in-in in 9.163 Saltbr-in 3.578 HRD-in -68.61, -47.67 58.19, -2.62 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -172.94 APE8-dihe-out -125.34, -40.47 APE8-rot-in 276.42 APE67-dihe-in -57.32, -20.72 -62.12, -27.76 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.271 None None None XRAY 2.5 0.24 0.284 A 360 331 17 0 0 13 [[24, 308]] 1.0 1kv1 CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3O8TA Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 13.263 10.326 None -137.91, -177.55 -138.77, 94.77 -70.74, -1.41 999.0, 999.0 121.86, 999.0 in-out in 9.427 Saltbr-out 4.27 HRD-in -65.83, -55.54 74.19, -14.68 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 158.65 APE8-dihe-out -42.15, -37.49 APE8-rot-out 44.7 APE67-dihe-in -68.78, -13.14 -104.02, 1.06 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 12.491 F169A None None XRAY 2.0 0.229 0.282 A 360 332 16 0 0 13 [[24, 308]] 1.0 3o8t CMGC_MAPK14_HUMAN CMGC 1.1e-83 287.0 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3OC1A Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 12.729 11.102 None -150.55, -172.96 -134.29, 139.02 -118.77, 999.0 999.0, 999.0 999.0, 999.0 in-in in 9.418 Saltbr-in 3.337 HRD-in -75.41, -45.78 70.08, -9.86 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 106.76 APE8-dihe-out -49.39, -49.27 APE8-rot-in 287.36 APE67-dihe-in -53.47, -28.65 -54.1, -35.8 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.094 F169G None None XRAY 2.59 0.229 0.303 A 360 330 18 0 0 14 [[24, 308]] 1.0 3oc1 CMGC_MAPK14_HUMAN CMGC 3e-83 285.5 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14

Ligand: BMU

Total number of chains: 6
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGout None 3 50.0% 3O8TA
DFGout BBAminus 2 33.3% 3O8UA
DFGin None 1 16.7% 3O8PA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC MAPK14 MK14_HUMAN 3O8PA Q16539 5 351 360.0 BMU:361 Type1 Inactive DFGin 10.863 12.014 None -115.52, 162.58 -99.08, -26.53 -122.71, 117.21 291.85, 138.97 -42.63, -102.67 in-out in 9.092 Saltbr-out 5.085 HRD-in -69.17, -52.21 73.92, -4.49 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnoo APE10-dihe-na 999.0, 3.16 APE9-dihe-na -166.83, -167.55 APE8-dihe-out -116.39, -25.53 APE8-rot-in 271.29 APE67-dihe-in -61.81, -26.71 -69.76, -21.19 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 12.159 APE9-dist-out 10.453 D168G None None XRAY 2.1 0.218 0.276 A 360 336 11 0 0 11 [[24, 308]] 1.0 3o8p Homo sapiens CMGC_MAPK14_HUMAN CMGC 2.7e-83 285.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3O8UA Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 13.796 9.306 BBAminus -146.29, -170.4 -144.05, 102.12 -67.29, -15.97 286.91, 115.68 99.79, 999.0 in-in in 9.331 Saltbr-in 3.364 HRD-in -63.28, -51.7 74.53, -20.43 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 144.38 APE8-dihe-out -70.85, -30.66 APE8-rot-in 258.69 APE67-dihe-in -65.11, -25.9 -59.1, -20.9 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 12.104 F169Y None None XRAY 2.1 0.224 0.285 A 360 332 16 0 0 13 [[24, 308]] 1.0 3o8u Homo sapiens CMGC_MAPK14_HUMAN CMGC 3.3e-84 288.7 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3OBJA Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 14.513 11.366 BBAminus -154.08, -178.49 -133.48, 111.98 -61.66, -36.04 255.28, 56.42 -103.05, -92.49 in-out in 9.304 Saltbr-out 5.802 HRD-in -72.07, -52.81 76.05, -16.45 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 143.04 APE8-dihe-out -70.24, -30.65 APE8-rot-out 197.91 APE67-dihe-in -70.14, -17.15 -63.21, -16.69 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.973 F169R None None XRAY 2.4 0.22 0.287 A 360 332 16 0 0 12 [[24, 308]] 1.0 3obj Homo sapiens CMGC_MAPK14_HUMAN CMGC 2e-83 286.1 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 1KV1A Q16539 5 352 360.0 BMU:391 Type3 Inactive DFGout 13.635 9.556 None -159.24, -177.02 -146.07, 100.83 -75.42, -134.45 282.12, 117.71 154.13, 999.0 in-in in 9.163 Saltbr-in 3.578 HRD-in -68.61, -47.67 58.19, -2.62 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -172.94 APE8-dihe-out -125.34, -40.47 APE8-rot-in 276.42 APE67-dihe-in -57.32, -20.72 -62.12, -27.76 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.271 None None None XRAY 2.5 0.24 0.284 A 360 331 17 0 0 13 [[24, 308]] 1.0 1kv1 Homo sapiens CMGC_MAPK14_HUMAN CMGC 5.9e-85 291.1 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3O8TA Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 13.263 10.326 None -137.91, -177.55 -138.77, 94.77 -70.74, -1.41 999.0, 999.0 121.86, 999.0 in-out in 9.427 Saltbr-out 4.27 HRD-in -65.83, -55.54 74.19, -14.68 out-none-out SNCono none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 158.65 APE8-dihe-out -42.15, -37.49 APE8-rot-out 44.7 APE67-dihe-in -68.78, -13.14 -104.02, 1.06 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 12.491 F169A None None XRAY 2.0 0.229 0.282 A 360 332 16 0 0 13 [[24, 308]] 1.0 3o8t Homo sapiens CMGC_MAPK14_HUMAN CMGC 1.1e-83 287.0 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14
CMGC MAPK14 MK14_HUMAN 3OC1A Q16539 5 352 360.0 BMU:361 Type3 Inactive DFGout 12.729 11.102 None -150.55, -172.96 -134.29, 139.02 -118.77, 999.0 999.0, 999.0 999.0, 999.0 in-in in 9.418 Saltbr-in 3.337 HRD-in -75.41, -45.78 70.08, -9.86 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 106.76 APE8-dihe-out -49.39, -49.27 APE8-rot-in 287.36 APE67-dihe-in -53.47, -28.65 -54.1, -35.8 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.094 F169G None None XRAY 2.59 0.229 0.303 A 360 330 18 0 0 14 [[24, 308]] 1.0 3oc1 Homo sapiens CMGC_MAPK14_HUMAN CMGC 3e-83 285.5 1 301 301 167 168 169 171 173 53 71 75 147 149 148 150 205 192 187 186 185 184 183 182 181 107 Mitogen-activated protein kinase 14

Ligand: BMU

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name