Ligand: A1AV2

Total number of chains: 5
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAplus 5 100.0% 9CD5B

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
TYR FGFR1 FGFR1_HUMAN 9CD5A 2.939 Inactive DFGin‑BLAplus in-in none-out TYR APEdihe_iioai APEdist_aaao A1AV2 Type1 465 - 764 0 None C488A,C584S Fibroblast growth factor receptor 1
TYR FGFR1 FGFR1_HUMAN 9CD5B 2.939 Inactive DFGin‑BLAplus in-in out-out TYR APEdihe_iioai APEdist_aaao A1AV2 Type1 460 - 764 0 None C488A,C584S Fibroblast growth factor receptor 1
TYR FGFR3 FGFR3_HUMAN 9CD7A 2.53 Inactive DFGin‑BLAplus in-in none-out TYR APEdihe_nnoai APEdist_aaao A1AV2 Type1 451 - 755 0 None C482A,C582S,K650E Fibroblast growth factor receptor 3
TYR FGFR3 FGFR3_HUMAN 9CD7B 2.53 Inactive DFGin‑BLAplus in-in out-out TYR APEdihe_nnoai APEdist_aaao A1AV2 Type1 458 - 755 0 None C482A,C582S,K650E Fibroblast growth factor receptor 3
TYR FGFR3 FGFR3_HUMAN 9CD7C 2.53 Inactive DFGin‑BLAplus in-in out-out TYR APEdihe_nnoai APEdist_aaao A1AV2 Type1 458 - 755 0 None C482A,C582S,K650E Fibroblast growth factor receptor 3

Ligand: A1AV2

Total number of chains: 5
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAplus 5 100.0% 9CD5B

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TYR FGFR1 FGFR1_HUMAN 9CD5A 2.939 Inactive DFGin‑BLAplus in-in none-out TYR APEdihe_iioai APEdist_aaao A1AV2 Type1 465 - 764 0 None C488A,C584S Fibroblast growth factor receptor 1 Homo sapiens
TYR FGFR1 FGFR1_HUMAN 9CD5B 2.939 Inactive DFGin‑BLAplus in-in out-out TYR APEdihe_iioai APEdist_aaao A1AV2 Type1 460 - 764 0 None C488A,C584S Fibroblast growth factor receptor 1 Homo sapiens
TYR FGFR3 FGFR3_HUMAN 9CD7A 2.53 Inactive DFGin‑BLAplus in-in none-out TYR APEdihe_nnoai APEdist_aaao A1AV2 Type1 451 - 755 0 None C482A,C582S,K650E Fibroblast growth factor receptor 3 Homo sapiens
TYR FGFR3 FGFR3_HUMAN 9CD7B 2.53 Inactive DFGin‑BLAplus in-in out-out TYR APEdihe_nnoai APEdist_aaao A1AV2 Type1 458 - 755 0 None C482A,C582S,K650E Fibroblast growth factor receptor 3 Homo sapiens
TYR FGFR3 FGFR3_HUMAN 9CD7C 2.53 Inactive DFGin‑BLAplus in-in out-out TYR APEdihe_nnoai APEdist_aaao A1AV2 Type1 458 - 755 0 None C482A,C582S,K650E Fibroblast growth factor receptor 3 Homo sapiens

Ligand: A1AV2

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism