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| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| STE | MAP2K1 | MP2K1_HUMAN | 9AXMC | Q02750 | 43 | 376 | 393.0 | A1AHE:60401 | Type1 | Inactive | DFGin | 6.668 | 14.132 | BLBplus | -150.29, 169.67 | 59.1, 61.29 | -116.51, 166.39 | 40.92, 86.38 | -72.68, 94.97 | out-none | out | 15.379 | Saltbr-none | 999.0 | HRD-in | -102.21, -42.14 | 67.4, -10.68 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 9.75 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -64.72, 121.05 | APE9-dihe-na | -67.96, 179.71 | APE8-dihe-out | -110.15, -27.15 | APE8-rot-out | 56.89 | APE67-dihe-out | -127.4, 134.54 | -138.28, 164.48 | APE12-dist-out | 17.162 | APE11-dist-out | 22.178 | APE10-dist-out | 24.239 | APE9-dist-out | 13.24 | S218A,S222A | None | None | XRAY | 2.42 | 0.263 | 0.301 | C | 310 | 290 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axm | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXHA | Q02750 | 39 | 381 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.113 | 14.205 | BLBplus | -138.52, 176.84 | 56.32, 45.26 | -98.43, 166.79 | 48.45, 76.71 | -79.29, 73.17 | out-out | out | 15.389 | Saltbr-out | 15.461 | HRD-in | -79.27, -55.22 | 75.38, 2.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.391 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -141.27, 126.74 | APE9-dihe-na | -91.23, -150.48 | APE8-dihe-out | -108.84, -16.83 | APE8-rot-out | 178.7 | APE67-dihe-out | -130.79, 128.8 | -115.86, 151.78 | APE12-dist-out | 17.417 | APE11-dist-out | 17.624 | APE10-dist-out | 20.898 | APE9-dist-out | 13.154 | None | None | None | XRAY | 2.81 | 0.206 | 0.253 | A | 310 | 299 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axh | STE_MAP2K1_HUMAN | STE | 1.5e-98 | 335.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXHB | Q02750 | 38 | 381 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.028 | 13.959 | BLBplus | -143.4, 172.79 | 59.61, 49.11 | -104.03, 163.1 | 47.48, 79.51 | -74.37, 70.81 | out-out | out | 15.415 | Saltbr-out | 14.817 | HRD-in | -76.49, -58.47 | 81.39, -4.23 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.322 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -140.95, 129.53 | APE9-dihe-na | -95.7, -172.17 | APE8-dihe-out | -83.87, -23.26 | APE8-rot-out | 67.32 | APE67-dihe-out | -134.03, 129.22 | -119.03, 156.34 | APE12-dist-out | 17.307 | APE11-dist-out | 17.575 | APE10-dist-out | 20.9 | APE9-dist-out | 12.718 | None | None | None | XRAY | 2.81 | 0.206 | 0.253 | B | 310 | 300 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axh | STE_MAP2K1_HUMAN | STE | 1.5e-98 | 335.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXMA | Q02750 | 38 | 382 | 393.0 | A1AHE:60401,ANP:60403 | Type1,ATPlike | Inactive | DFGin | 6.204 | 13.999 | BLBplus | -146.84, 170.95 | 57.84, 58.3 | -113.46, 158.4 | 47.1, 81.42 | -71.93, 78.64 | out-out | out | 15.426 | Saltbr-out | 15.513 | HRD-in | -80.25, -54.29 | 71.05, 3.5 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.11 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -58.81, 135.38 | APE9-dihe-na | -86.44, -174.93 | APE8-dihe-out | -114.7, -19.48 | APE8-rot-out | 61.33 | APE67-dihe-out | -156.42, 133.96 | -137.25, 175.14 | APE12-dist-out | 17.347 | APE11-dist-out | 22.123 | APE10-dist-out | 24.223 | APE9-dist-out | 13.241 | S218A,S222A | None | None | XRAY | 2.42 | 0.263 | 0.301 | A | 310 | 301 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axm | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXXA | Q02750 | 41 | 382 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.157 | 14.473 | BLBplus | -142.21, 167.57 | 61.94, 40.19 | -92.82, 170.58 | 38.95, 89.02 | -82.21, 74.48 | out-out | out | 15.925 | Saltbr-out | 15.661 | HRD-in | -77.34, -56.94 | 85.02, -11.71 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.623 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -70.01, 140.02 | APE9-dihe-na | -107.63, 178.58 | APE8-dihe-out | -103.64, -13.88 | APE8-rot-out | 56.98 | APE67-dihe-out | -152.18, 145.48 | -132.34, 175.09 | APE12-dist-out | 18.633 | APE11-dist-out | 16.086 | APE10-dist-out | 21.091 | APE9-dist-out | 12.771 | S218A,S222A | None | None | XRAY | 2.07 | 0.215 | 0.248 | A | 310 | 298 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axx | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXXC | Q02750 | 37 | 378 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.066 | 14.251 | BLBplus | -153.34, 165.37 | 62.85, 41.08 | -93.54, 164.6 | 44.67, 86.41 | -75.31, 71.49 | out-out | out | 15.517 | Saltbr-out | 15.022 | HRD-in | -80.68, -38.87 | 53.15, 7.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.691 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -68.91, 127.09 | APE9-dihe-na | -100.27, 169.31 | APE8-dihe-out | -98.12, -23.61 | APE8-rot-out | 61.42 | APE67-dihe-out | -153.77, 146.66 | -125.41, 178.29 | APE12-dist-out | 18.45 | APE11-dist-out | 16.119 | APE10-dist-out | 21.581 | APE9-dist-out | 12.749 | S218A,S222A | None | None | XRAY | 2.07 | 0.215 | 0.248 | C | 310 | 297 | 1 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axx | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AYAB | Q02750 | 42 | 382 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.209 | 14.117 | BLBplus | -156.4, 169.03 | 57.59, 47.08 | -100.39, 159.82 | 46.95, 83.0 | -73.48, 80.99 | out-out | out | 15.444 | Saltbr-out | 14.957 | HRD-in | -72.22, -50.64 | 78.5, -7.92 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.725 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -67.32, 133.53 | APE9-dihe-na | -94.07, -169.54 | APE8-dihe-out | -110.54, -56.8 | APE8-rot-out | 71.18 | APE67-dihe-out | -155.6, 139.89 | -98.61, 175.74 | APE12-dist-out | 17.221 | APE11-dist-out | 22.149 | APE10-dist-out | 24.195 | APE9-dist-out | 13.766 | S218A,S222A | None | None | XRAY | 2.59 | 0.214 | 0.257 | B | 310 | 297 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9aya | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AYAD | Q02750 | 39 | 382 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.236 | 14.114 | BLBplus | -150.42, 169.48 | 62.14, 35.37 | -84.74, 166.85 | 39.42, 88.37 | -83.08, 73.44 | out-out | out | 15.382 | Saltbr-out | 15.287 | HRD-in | -84.82, -56.5 | 86.5, -11.08 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.653 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 132.69 | APE8-dihe-out | -103.38, -24.48 | APE8-rot-out | 47.89 | APE67-dihe-out | -161.23, 135.82 | -100.94, -174.52 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.749 | S218A,S222A | None | None | XRAY | 2.59 | 0.214 | 0.257 | D | 310 | 293 | 7 | 0 | 0 | 3 | [[68, 361]] | 1.0 | 9aya | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AY7B | Q02750 | 33 | 383 | 393.0 | A1AHE:401,ANP:402 | Type1,ATPlike | Inactive | DFGin | 6.131 | 14.268 | BLBplus | -154.96, 169.08 | 61.0, 36.72 | -91.6, 162.02 | 49.73, 81.71 | -77.61, 77.19 | out-out | out | 15.513 | Saltbr-out | 15.402 | HRD-in | -75.89, -55.94 | 83.29, -11.88 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.576 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -66.62, 136.57 | APE9-dihe-na | -89.93, -175.43 | APE8-dihe-out | -113.57, -10.62 | APE8-rot-out | 51.26 | APE67-dihe-out | -146.5, 144.85 | -157.42, 170.13 | APE12-dist-out | 17.344 | APE11-dist-out | 22.114 | APE10-dist-out | 24.207 | APE9-dist-out | 13.729 | S218A,S222A | None | None | XRAY | 2.41 | 0.203 | 0.236 | B | 394 | 322 | 29 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9ay7 | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXAB | Q02750 | 52 | 380 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 6.813 | 13.768 | BLBplus | -157.46, 170.37 | 59.28, 64.98 | -117.48, 165.11 | 40.29, 81.19 | -81.1, 74.19 | out-out | out | 15.431 | Saltbr-out | 17.41 | HRD-in | -75.24, -42.64 | 72.38, -11.77 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.208 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -68.37, -62.71 | APE9-dihe-na | 103.09, 102.94 | APE8-dihe-out | -88.38, -48.33 | APE8-rot-out | 62.02 | APE67-dihe-out | -122.1, 131.17 | -98.78, 143.35 | APE12-dist-out | 16.696 | APE11-dist-out | 18.126 | APE10-dist-out | 22.852 | APE9-dist-out | 12.424 | S218A,S222A | None | None | EM | 4.36 | 999.0 | 999.0 | B | 394 | 278 | 51 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axa | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXAD | Q02750 | 59 | 383 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 6.188 | 15.038 | BLBplus | -161.59, 167.64 | 63.71, 27.36 | -77.56, 162.55 | 63.45, 90.49 | -80.72, 76.54 | out-out | out | 17.613 | Saltbr-out | 18.798 | HRD-in | -103.62, -49.66 | 71.76, -9.27 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.797 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | 56.39, -81.94 | APE9-dihe-na | 48.87, 69.85 | APE8-dihe-out | -71.23, -18.7 | APE8-rot-out | 181.91 | APE67-dihe-out | -127.48, 156.86 | -129.99, 139.21 | APE12-dist-out | 19.162 | APE11-dist-out | 16.676 | APE10-dist-out | 21.374 | APE9-dist-out | 12.272 | S218A,S222A | None | None | EM | 4.36 | 999.0 | 999.0 | D | 394 | 275 | 50 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axa | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXCB | Q02750 | 52 | 380 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 5.979 | 13.857 | BLBplus | -156.34, 159.86 | 58.05, 51.28 | -90.68, 168.57 | 45.43, 79.18 | -80.79, 77.37 | out-out | out | 15.525 | Saltbr-out | 16.483 | HRD-in | -82.47, -42.11 | 70.94, -10.4 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.445 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -71.13, -44.57 | APE9-dihe-na | 100.23, 100.79 | APE8-dihe-out | -96.55, -49.37 | APE8-rot-out | 61.77 | APE67-dihe-out | -125.36, 134.49 | -112.13, 139.3 | APE12-dist-out | 16.732 | APE11-dist-out | 18.062 | APE10-dist-out | 22.927 | APE9-dist-out | 12.623 | S218A,S222A | None | None | EM | 4.16 | 999.0 | 999.0 | B | 394 | 278 | 51 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axc | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXCD | Q02750 | 59 | 383 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 5.944 | 14.943 | BLBplus | -155.71, -173.77 | 60.85, 40.35 | -100.84, 165.38 | 63.0, 90.55 | -83.19, 80.54 | out-out | out | 17.464 | Saltbr-out | 19.882 | HRD-in | -94.68, -47.55 | 72.62, -11.59 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.375 | ActLoopCT-out | nonTYR | APEdihe_aaoio | APEdist_oooo | APE10-dihe-na | 51.94, -88.31 | APE9-dihe-na | 51.11, 70.23 | APE8-dihe-out | -66.0, -35.69 | APE8-rot-in | 292.49 | APE67-dihe-out | -158.48, 126.03 | -105.47, -179.54 | APE12-dist-out | 18.774 | APE11-dist-out | 17.062 | APE10-dist-out | 21.141 | APE9-dist-out | 12.44 | S218A,S222A | None | None | EM | 4.16 | 999.0 | 999.0 | D | 394 | 275 | 50 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axc | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXYB | Q02750 | 40 | 383 | 393.0 | A1AHE:401,ANP:402 | Type3,ATPlike | Inactive | DFGin | 5.938 | 14.134 | BLBplus | -149.11, 165.49 | 51.9, 40.29 | -92.3, 159.5 | 54.58, 76.32 | -75.9, 70.87 | out-out | out | 15.399 | Saltbr-out | 14.988 | HRD-in | -57.0, -47.47 | 79.88, -10.87 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.337 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -115.09, 128.49 | APE9-dihe-na | -79.18, 173.05 | APE8-dihe-out | -111.11, -19.81 | APE8-rot-out | 47.95 | APE67-dihe-out | -148.5, 141.81 | -130.51, 175.5 | APE12-dist-out | 18.176 | APE11-dist-out | 19.731 | APE10-dist-out | 22.785 | APE9-dist-out | 13.229 | S218A,S222A | None | None | XRAY | 3.6 | 0.19 | 0.237 | B | 394 | 312 | 32 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axy | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| STE | MAP2K1 | MP2K1_HUMAN | 9AXMC | Q02750 | 43 | 376 | 393.0 | A1AHE:60401 | Type1 | Inactive | DFGin | 6.668 | 14.132 | BLBplus | -150.29, 169.67 | 59.1, 61.29 | -116.51, 166.39 | 40.92, 86.38 | -72.68, 94.97 | out-none | out | 15.379 | Saltbr-none | 999.0 | HRD-in | -102.21, -42.14 | 67.4, -10.68 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 9.75 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -64.72, 121.05 | APE9-dihe-na | -67.96, 179.71 | APE8-dihe-out | -110.15, -27.15 | APE8-rot-out | 56.89 | APE67-dihe-out | -127.4, 134.54 | -138.28, 164.48 | APE12-dist-out | 17.162 | APE11-dist-out | 22.178 | APE10-dist-out | 24.239 | APE9-dist-out | 13.24 | S218A,S222A | None | None | XRAY | 2.42 | 0.263 | 0.301 | C | 310 | 290 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axm | Homo sapiens | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXHA | Q02750 | 39 | 381 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.113 | 14.205 | BLBplus | -138.52, 176.84 | 56.32, 45.26 | -98.43, 166.79 | 48.45, 76.71 | -79.29, 73.17 | out-out | out | 15.389 | Saltbr-out | 15.461 | HRD-in | -79.27, -55.22 | 75.38, 2.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.391 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -141.27, 126.74 | APE9-dihe-na | -91.23, -150.48 | APE8-dihe-out | -108.84, -16.83 | APE8-rot-out | 178.7 | APE67-dihe-out | -130.79, 128.8 | -115.86, 151.78 | APE12-dist-out | 17.417 | APE11-dist-out | 17.624 | APE10-dist-out | 20.898 | APE9-dist-out | 13.154 | None | None | None | XRAY | 2.81 | 0.206 | 0.253 | A | 310 | 299 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axh | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.5e-98 | 335.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXHB | Q02750 | 38 | 381 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.028 | 13.959 | BLBplus | -143.4, 172.79 | 59.61, 49.11 | -104.03, 163.1 | 47.48, 79.51 | -74.37, 70.81 | out-out | out | 15.415 | Saltbr-out | 14.817 | HRD-in | -76.49, -58.47 | 81.39, -4.23 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.322 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -140.95, 129.53 | APE9-dihe-na | -95.7, -172.17 | APE8-dihe-out | -83.87, -23.26 | APE8-rot-out | 67.32 | APE67-dihe-out | -134.03, 129.22 | -119.03, 156.34 | APE12-dist-out | 17.307 | APE11-dist-out | 17.575 | APE10-dist-out | 20.9 | APE9-dist-out | 12.718 | None | None | None | XRAY | 2.81 | 0.206 | 0.253 | B | 310 | 300 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axh | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.5e-98 | 335.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXMA | Q02750 | 38 | 382 | 393.0 | A1AHE:60401,ANP:60403 | Type1,ATPlike | Inactive | DFGin | 6.204 | 13.999 | BLBplus | -146.84, 170.95 | 57.84, 58.3 | -113.46, 158.4 | 47.1, 81.42 | -71.93, 78.64 | out-out | out | 15.426 | Saltbr-out | 15.513 | HRD-in | -80.25, -54.29 | 71.05, 3.5 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.11 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -58.81, 135.38 | APE9-dihe-na | -86.44, -174.93 | APE8-dihe-out | -114.7, -19.48 | APE8-rot-out | 61.33 | APE67-dihe-out | -156.42, 133.96 | -137.25, 175.14 | APE12-dist-out | 17.347 | APE11-dist-out | 22.123 | APE10-dist-out | 24.223 | APE9-dist-out | 13.241 | S218A,S222A | None | None | XRAY | 2.42 | 0.263 | 0.301 | A | 310 | 301 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axm | Homo sapiens | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXXA | Q02750 | 41 | 382 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.157 | 14.473 | BLBplus | -142.21, 167.57 | 61.94, 40.19 | -92.82, 170.58 | 38.95, 89.02 | -82.21, 74.48 | out-out | out | 15.925 | Saltbr-out | 15.661 | HRD-in | -77.34, -56.94 | 85.02, -11.71 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.623 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -70.01, 140.02 | APE9-dihe-na | -107.63, 178.58 | APE8-dihe-out | -103.64, -13.88 | APE8-rot-out | 56.98 | APE67-dihe-out | -152.18, 145.48 | -132.34, 175.09 | APE12-dist-out | 18.633 | APE11-dist-out | 16.086 | APE10-dist-out | 21.091 | APE9-dist-out | 12.771 | S218A,S222A | None | None | XRAY | 2.07 | 0.215 | 0.248 | A | 310 | 298 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axx | Homo sapiens | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXXC | Q02750 | 37 | 378 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.066 | 14.251 | BLBplus | -153.34, 165.37 | 62.85, 41.08 | -93.54, 164.6 | 44.67, 86.41 | -75.31, 71.49 | out-out | out | 15.517 | Saltbr-out | 15.022 | HRD-in | -80.68, -38.87 | 53.15, 7.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.691 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -68.91, 127.09 | APE9-dihe-na | -100.27, 169.31 | APE8-dihe-out | -98.12, -23.61 | APE8-rot-out | 61.42 | APE67-dihe-out | -153.77, 146.66 | -125.41, 178.29 | APE12-dist-out | 18.45 | APE11-dist-out | 16.119 | APE10-dist-out | 21.581 | APE9-dist-out | 12.749 | S218A,S222A | None | None | XRAY | 2.07 | 0.215 | 0.248 | C | 310 | 297 | 1 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axx | Homo sapiens | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AYAB | Q02750 | 42 | 382 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.209 | 14.117 | BLBplus | -156.4, 169.03 | 57.59, 47.08 | -100.39, 159.82 | 46.95, 83.0 | -73.48, 80.99 | out-out | out | 15.444 | Saltbr-out | 14.957 | HRD-in | -72.22, -50.64 | 78.5, -7.92 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.725 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -67.32, 133.53 | APE9-dihe-na | -94.07, -169.54 | APE8-dihe-out | -110.54, -56.8 | APE8-rot-out | 71.18 | APE67-dihe-out | -155.6, 139.89 | -98.61, 175.74 | APE12-dist-out | 17.221 | APE11-dist-out | 22.149 | APE10-dist-out | 24.195 | APE9-dist-out | 13.766 | S218A,S222A | None | None | XRAY | 2.59 | 0.214 | 0.257 | B | 310 | 297 | 0 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9aya | Homo sapiens | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AYAD | Q02750 | 39 | 382 | 393.0 | A1AHE:60401,ANP:60402 | Type1,ATPlike | Inactive | DFGin | 6.236 | 14.114 | BLBplus | -150.42, 169.48 | 62.14, 35.37 | -84.74, 166.85 | 39.42, 88.37 | -83.08, 73.44 | out-out | out | 15.382 | Saltbr-out | 15.287 | HRD-in | -84.82, -56.5 | 86.5, -11.08 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.653 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 132.69 | APE8-dihe-out | -103.38, -24.48 | APE8-rot-out | 47.89 | APE67-dihe-out | -161.23, 135.82 | -100.94, -174.52 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.749 | S218A,S222A | None | None | XRAY | 2.59 | 0.214 | 0.257 | D | 310 | 293 | 7 | 0 | 0 | 3 | [[68, 361]] | 1.0 | 9aya | Homo sapiens | STE_MAP2K1_HUMAN | STE | 6.5e-98 | 333.1 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AY7B | Q02750 | 33 | 383 | 393.0 | A1AHE:401,ANP:402 | Type1,ATPlike | Inactive | DFGin | 6.131 | 14.268 | BLBplus | -154.96, 169.08 | 61.0, 36.72 | -91.6, 162.02 | 49.73, 81.71 | -77.61, 77.19 | out-out | out | 15.513 | Saltbr-out | 15.402 | HRD-in | -75.89, -55.94 | 83.29, -11.88 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.576 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -66.62, 136.57 | APE9-dihe-na | -89.93, -175.43 | APE8-dihe-out | -113.57, -10.62 | APE8-rot-out | 51.26 | APE67-dihe-out | -146.5, 144.85 | -157.42, 170.13 | APE12-dist-out | 17.344 | APE11-dist-out | 22.114 | APE10-dist-out | 24.207 | APE9-dist-out | 13.729 | S218A,S222A | None | None | XRAY | 2.41 | 0.203 | 0.236 | B | 394 | 322 | 29 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9ay7 | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXAB | Q02750 | 52 | 380 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 6.813 | 13.768 | BLBplus | -157.46, 170.37 | 59.28, 64.98 | -117.48, 165.11 | 40.29, 81.19 | -81.1, 74.19 | out-out | out | 15.431 | Saltbr-out | 17.41 | HRD-in | -75.24, -42.64 | 72.38, -11.77 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.208 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -68.37, -62.71 | APE9-dihe-na | 103.09, 102.94 | APE8-dihe-out | -88.38, -48.33 | APE8-rot-out | 62.02 | APE67-dihe-out | -122.1, 131.17 | -98.78, 143.35 | APE12-dist-out | 16.696 | APE11-dist-out | 18.126 | APE10-dist-out | 22.852 | APE9-dist-out | 12.424 | S218A,S222A | None | None | EM | 4.36 | 999.0 | 999.0 | B | 394 | 278 | 51 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axa | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXAD | Q02750 | 59 | 383 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 6.188 | 15.038 | BLBplus | -161.59, 167.64 | 63.71, 27.36 | -77.56, 162.55 | 63.45, 90.49 | -80.72, 76.54 | out-out | out | 17.613 | Saltbr-out | 18.798 | HRD-in | -103.62, -49.66 | 71.76, -9.27 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.797 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | 56.39, -81.94 | APE9-dihe-na | 48.87, 69.85 | APE8-dihe-out | -71.23, -18.7 | APE8-rot-out | 181.91 | APE67-dihe-out | -127.48, 156.86 | -129.99, 139.21 | APE12-dist-out | 19.162 | APE11-dist-out | 16.676 | APE10-dist-out | 21.374 | APE9-dist-out | 12.272 | S218A,S222A | None | None | EM | 4.36 | 999.0 | 999.0 | D | 394 | 275 | 50 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axa | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXCB | Q02750 | 52 | 380 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 5.979 | 13.857 | BLBplus | -156.34, 159.86 | 58.05, 51.28 | -90.68, 168.57 | 45.43, 79.18 | -80.79, 77.37 | out-out | out | 15.525 | Saltbr-out | 16.483 | HRD-in | -82.47, -42.11 | 70.94, -10.4 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.445 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -71.13, -44.57 | APE9-dihe-na | 100.23, 100.79 | APE8-dihe-out | -96.55, -49.37 | APE8-rot-out | 61.77 | APE67-dihe-out | -125.36, 134.49 | -112.13, 139.3 | APE12-dist-out | 16.732 | APE11-dist-out | 18.062 | APE10-dist-out | 22.927 | APE9-dist-out | 12.623 | S218A,S222A | None | None | EM | 4.16 | 999.0 | 999.0 | B | 394 | 278 | 51 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axc | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXCD | Q02750 | 59 | 383 | 393.0 | A1AHE:401 | Type3 | Inactive | DFGin | 5.944 | 14.943 | BLBplus | -155.71, -173.77 | 60.85, 40.35 | -100.84, 165.38 | 63.0, 90.55 | -83.19, 80.54 | out-out | out | 17.464 | Saltbr-out | 19.882 | HRD-in | -94.68, -47.55 | 72.62, -11.59 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.375 | ActLoopCT-out | nonTYR | APEdihe_aaoio | APEdist_oooo | APE10-dihe-na | 51.94, -88.31 | APE9-dihe-na | 51.11, 70.23 | APE8-dihe-out | -66.0, -35.69 | APE8-rot-in | 292.49 | APE67-dihe-out | -158.48, 126.03 | -105.47, -179.54 | APE12-dist-out | 18.774 | APE11-dist-out | 17.062 | APE10-dist-out | 21.141 | APE9-dist-out | 12.44 | S218A,S222A | None | None | EM | 4.16 | 999.0 | 999.0 | D | 394 | 275 | 50 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axc | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| STE | MAP2K1 | MP2K1_HUMAN | 9AXYB | Q02750 | 40 | 383 | 393.0 | A1AHE:401,ANP:402 | Type3,ATPlike | Inactive | DFGin | 5.938 | 14.134 | BLBplus | -149.11, 165.49 | 51.9, 40.29 | -92.3, 159.5 | 54.58, 76.32 | -75.9, 70.87 | out-out | out | 15.399 | Saltbr-out | 14.988 | HRD-in | -57.0, -47.47 | 79.88, -10.87 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.337 | ActLoopCT-out | nonTYR | APEdihe_aaooo | APEdist_oooo | APE10-dihe-na | -115.09, 128.49 | APE9-dihe-na | -79.18, 173.05 | APE8-dihe-out | -111.11, -19.81 | APE8-rot-out | 47.95 | APE67-dihe-out | -148.5, 141.81 | -130.51, 175.5 | APE12-dist-out | 18.176 | APE11-dist-out | 19.731 | APE10-dist-out | 22.785 | APE9-dist-out | 13.229 | S218A,S222A | None | None | XRAY | 3.6 | 0.19 | 0.237 | B | 394 | 312 | 32 | 0 | 0 | 0 | [[68, 361]] | 1.0 | 9axy | Homo sapiens | STE_MAP2K1_HUMAN | STE | 1.1e-96 | 329.3 | 1 | 257 | 257 | 207 | 208 | 209 | 211 | 213 | 97 | 114 | 118 | 187 | 189 | 188 | 190 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 144 | Dual specificity mitogen-activated protein kinase kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
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Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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