| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| STE | MAP3K2 | M3K2_HUMAN | 9P6AA | Q9Y2U5 | 351 | 617 | 619.0 | 0LI:701 | Type2 | Inactive | DFGout | 14.1431 | 9.8906 | BBAminus | -146.02, -172.59 | -157.95, 116.33 | -87.88, -36.33 | 294.81, 102.45 | -88.54, 36.79 | in-in | in | 8.4578 | Saltbr-in | 2.5939 | HRD-in | -76.59, -52.31 | 80.62, -19.75 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -98.17, -51.62 | APE9-dihe-na | -96.01, 162.48 | APE8-dihe-in | -81.48, 131.06 | APE8-rot-out | 69.69 | APE67-dihe-in | -67.88, -22.22 | -92.28, 3.15 | APE12-dist-out | 20.6817 | APE11-dist-out | 19.1439 | APE10-dist-out | 14.3088 | APE9-dist-out | 10.4562 | None | None | None | XRAY | 2.4 | 0.228 | 0.246 | A | 299.0 | 253.0 | 14 | 31 | 17 | 14 | [[356, 616]] | 1.0 | 9p6a | STE_MAP3K2_HUMAN | STE | 1.9e-81 | 279.1 | 1.0 | 257.0 | 257.0 | 500 | 501 | 502 | 504 | 506 | 385 | 406 | 410 | 480 | 482 | 481 | 483.0 | 543 | 531 | 526 | 525 | 524 | 523 | 522 | 521 | 520 | 438 | Mitogen-activated protein kinase kinase kinase 2 |
| STE | MAP3K2 | M3K2_HUMAN | 9P6AB | Q9Y2U5 | 347 | 618 | 619.0 | 0LI:701 | Type2 | Inactive | DFGout | 13.8018 | 9.7559 | None | -145.97, -173.02 | -157.2, 114.58 | -90.61, 158.12 | 297.06, 102.49 | 67.12, -99.7 | in-in | in | 8.6308 | Saltbr-in | 2.7273 | HRD-in | -74.0, -48.74 | 85.04, -22.17 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -168.99 | APE9-dihe-na | -96.92, -27.66 | APE8-dihe-in | -82.09, 127.1 | APE8-rot-out | 70.19 | APE67-dihe-in | -70.58, -23.59 | -96.42, -0.55 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 8.6373 | APE9-dist-out | 10.7871 | None | None | None | XRAY | 2.4 | 0.228 | 0.246 | B | 299.0 | 247.0 | 25 | 31 | 15 | 16 | [[356, 616]] | 1.0 | 9p6a | STE_MAP3K2_HUMAN | STE | 1.9e-81 | 279.1 | 1.0 | 257.0 | 257.0 | 500 | 501 | 502 | 504 | 506 | 385 | 406 | 410 | 480 | 482 | 481 | 483.0 | 543 | 531 | 526 | 525 | 524 | 523 | 522 | 521 | 520 | 438 | Mitogen-activated protein kinase kinase kinase 2 |
| TKL | BRAF | BRAF_HUMAN | 6P3DA | P15056 | 448 | 721 | 766.0 | 0LI:61001 | Type2 | Inactive | DFGout | 12.35 | 10.9052 | BBAminus | -138.54, -166.92 | -135.05, 80.45 | -80.66, -37.84 | 293.17, 97.28 | 81.0, 10.25 | in-in | in | 8.6648 | Saltbr-in | 2.9974 | HRD-in | -65.6, -55.77 | 77.59, -19.55 | in-out-out | SNCioo | out-out | ActLoopNT-out | 19.9448 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnoo | APE10-dihe-na | 999.0, -19.82 | APE9-dihe-na | 76.62, -63.3 | APE8-dihe-out | -51.89, -23.77 | APE8-rot-out | 78.9 | APE67-dihe-in | -55.73, -23.59 | -56.01, -24.35 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 12.7002 | APE9-dist-out | 11.8707 | None | None | None | XRAY | 2.11 | 0.188 | 0.245 | A | 297.0 | 261.0 | 13 | 30 | 17 | 13 | [[457, 716]] | 1.0 | 6p3d | TKL_BRAF_HUMAN | TKL | 5.8e-84 | 287.7 | 4.0 | 267.0 | 264.0 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576.0 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | IRAK4 | IRAK4_HUMAN | 6EG9A | Q9NWZ3 | 164 | 459 | 460.0 | 0LI:501 | Type2 | Inactive | DFGout | 14.0712 | 10.7156 | None | -127.45, 167.3 | -138.69, 101.47 | -85.85, 140.23 | 309.7, 100.41 | -43.19, 999.0 | in-out | in | 9.0273 | Saltbr-out | 6.6465 | HRD-in | -71.51, -48.43 | 70.86, -5.67 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 6.91 | APE9-dihe-na | 158.59, -165.8 | APE8-dihe-in | -114.99, 116.82 | APE8-rot-in | 299.55 | APE67-dihe-in | -67.65, -20.43 | -63.19, -29.42 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.972 | None | None | None | XRAY | 2.414 | 0.224 | 0.249 | A | 312.0 | 276.0 | 20 | 30 | 13 | 17 | [[183, 456]] | 1.0 | 6eg9 | TKL_IRAK4_HUMAN | TKL | 4.6e-84 | 288.0 | 5.0 | 266.0 | 262.0 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311.0 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6EG9B | Q9NWZ3 | 165 | 459 | 460.0 | 0LI:501 | Type2 | Inactive | DFGout | 14.2443 | 9.3953 | None | -135.81, 174.82 | -152.29, 126.78 | -163.75, 999.0 | 33.58, 60.29 | 999.0, 999.0 | in-in | in | 8.9787 | Saltbr-in | 3.0904 | HRD-in | -69.81, -51.27 | 77.39, -7.02 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 146.5 | APE9-dihe-na | 95.5, 175.38 | APE8-dihe-in | -117.78, 118.94 | APE8-rot-in | 307.93 | APE67-dihe-in | -67.02, -18.64 | -61.22, -30.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.6297 | None | None | None | XRAY | 2.414 | 0.224 | 0.249 | B | 312.0 | 274.0 | 21 | 30 | 12 | 18 | [[183, 456]] | 1.0 | 6eg9 | TKL_IRAK4_HUMAN | TKL | 4.6e-84 | 288.0 | 5.0 | 266.0 | 262.0 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311.0 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | LRRK2 | LRRK2_HUMAN | 8U8AB | Q5S007 | 558 | 2526 | 2527.0 | 0LI:2601 | Type2 | Inactive | DFGout | 14.859 | 10.8454 | BBAminus | -150.37, 144.32 | -124.19, 97.68 | -69.79, -11.11 | 321.73, 111.63 | 66.57, 27.33 | in-out | in | 8.8739 | Saltbr-out | 3.6727 | HRD-out | -76.07, 95.41 | -48.17, -63.17 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 177.03 | APE8-dihe-in | -61.6, 136.03 | APE8-rot-in | 305.18 | APE67-dihe-in | -74.33, -25.33 | -56.72, -44.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 6.2972 | None | None | None | EM | 3.4 | 999.0 | 999.0 | B | 2527.0 | 1705.0 | 29 | 26 | 13 | 13 | [[1875, 2134]] | 1.0 | 8u8a | TKL_LRRK2_HUMAN | TKL | 3.8e-57 | 200.3 | 5.0 | 266.0 | 262.0 | 2016 | 2017 | 2018 | 2020 | 2022 | 1906 | 1920 | 1924 | 1991 | 1993 | 1992 | 1994.0 | 2055 | 2042 | 2037 | 2036 | 2035 | 2034 | 2033 | 2032 | 2031 | 1948 | Leucine-rich repeat serine/threonine-protein kinase 2 |
| TKL | LRRK2 | LRRK2_HUMAN | 8U8AC | Q5S007 | 558 | 2526 | 2527.0 | 0LI:2601 | Type2 | Inactive | DFGout | 14.8696 | 10.8459 | BBAminus | -150.46, 144.31 | -124.23, 97.69 | -69.77, -11.06 | 321.78, 111.5 | 66.48, 27.35 | in-out | in | 8.8719 | Saltbr-out | 3.6608 | HRD-out | -76.02, 95.48 | -48.33, -63.13 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 177.01 | APE8-dihe-in | -61.57, 135.98 | APE8-rot-in | 305.14 | APE67-dihe-in | -74.37, -25.35 | -56.73, -44.17 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 6.3006 | None | None | None | EM | 3.4 | 999.0 | 999.0 | C | 2527.0 | 1705.0 | 29 | 26 | 13 | 13 | [[1875, 2134]] | 1.0 | 8u8a | TKL_LRRK2_HUMAN | TKL | 3.8e-57 | 200.3 | 5.0 | 266.0 | 262.0 | 2016 | 2017 | 2018 | 2020 | 2022 | 1906 | 1920 | 1924 | 1991 | 1993 | 1992 | 1994.0 | 2055 | 2042 | 2037 | 2036 | 2035 | 2034 | 2033 | 2032 | 2031 | 1948 | Leucine-rich repeat serine/threonine-protein kinase 2 |
| TKL | RIPK2 | RIPK2_HUMAN | 4C8BA | O43353 | 8 | 316 | 540.0 | 0LI:1000 | Type2 | Inactive | DFGout | 12.7285 | 8.5841 | None | -142.99, -175.55 | -154.35, 140.4 | -129.56, 999.0 | 290.55, 114.67 | 999.0, 999.0 | in-in | in | 8.2431 | Saltbr-in | 2.8173 | HRD-in | -79.84, -58.2 | 64.89, 19.36 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -36.9 | APE8-dihe-out | -84.71, -55.98 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.98, -25.64 | -68.13, -16.01 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.2944 | None | None | None | XRAY | 2.75 | 0.203 | 0.244 | A | 334.0 | 279.0 | 30 | 33 | 11 | 22 | [[18, 292]] | 1.0 | 4c8b | TKL_RIPK2_HUMAN | TKL | 3.4e-73 | 252.4 | 4.0 | 266.0 | 263.0 | 163 | 164 | 165 | 167 | 169 | 47 | 66 | 70 | 143 | 145 | 144 | 146.0 | 211 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 96 | Receptor-interacting serine/threonine-protein kinase 2 |
| TKL | RIPK2 | RIPK2_HUMAN | 4C8BB | O43353 | 9 | 316 | 540.0 | 0LI:1000 | Type2 | Inactive | DFGout | 12.8402 | 8.8595 | None | -140.63, -176.63 | -153.18, 138.54 | -119.75, 999.0 | 285.35, 113.34 | 999.0, 999.0 | in-in | in | 8.2645 | Saltbr-in | 2.8058 | HRD-in | -79.98, -59.74 | 66.42, 17.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -39.27 | APE8-dihe-out | -68.6, -38.75 | APE8-rot-out | 169.06 | APE67-dihe-in | -64.78, -24.38 | -61.46, -15.15 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.4449 | None | None | None | XRAY | 2.75 | 0.203 | 0.244 | B | 334.0 | 281.0 | 27 | 33 | 11 | 22 | [[18, 292]] | 1.0 | 4c8b | TKL_RIPK2_HUMAN | TKL | 3.4e-73 | 252.4 | 4.0 | 266.0 | 263.0 | 163 | 164 | 165 | 167 | 169 | 47 | 66 | 70 | 143 | 145 | 144 | 146.0 | 211 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 96 | Receptor-interacting serine/threonine-protein kinase 2 |
| TYR | DDR1 | DDR1_HUMAN | 3ZOSB | Q08345 | 601 | 913 | 913.0 | 0LI:61000 | Type2 | Inactive | DFGout | 13.6455 | 9.6295 | BBAminus | -143.84, 178.94 | -153.3, 114.42 | -82.71, -15.18 | 287.49, 108.73 | 52.14, -127.46 | in-in | in | 7.9604 | Saltbr-in | 2.8828 | HRD-in | -60.43, -59.89 | 83.25, -8.8 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.4003 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.91, 133.24 | APE9-dihe-in | -130.81, 142.32 | APE8-dihe-in | -80.63, 68.61 | APE8-rot-na | 30.08 | APE67-dihe-in | -67.12, -16.99 | -59.3, -31.33 | APE12-dist-na | 11.7194 | APE11-dist-na | 12.9393 | APE10-dist-na | 10.2231 | APE9-dist-in | 7.9237 | None | None | None | XRAY | 1.92 | 0.208 | 0.234 | B | 315.0 | 301.0 | 12 | 30 | 30 | 0 | [[610, 907]] | 1.0 | 3zos | TYR_DDR1_HUMAN | TYR | 1.5e-92 | 315.5 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 3ZOSA | Q08345 | 602 | 913 | 913.0 | 0LI:61000,0LI:61004 | Type2,Allosteric | Inactive | DFGout | 13.6836 | 9.7654 | BBAminus | -140.01, 179.9 | -153.22, 112.84 | -85.26, -13.51 | 285.68, 107.96 | 48.92, -126.09 | in-in | in | 7.9981 | Saltbr-in | 2.8815 | HRD-in | -61.25, -58.95 | 80.5, -7.41 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.4763 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.17, 140.69 | APE9-dihe-in | -129.43, 143.43 | APE8-dihe-in | -82.4, 69.11 | APE8-rot-na | 29.15 | APE67-dihe-in | -67.51, -15.14 | -58.33, -33.07 | APE12-dist-na | 11.7075 | APE11-dist-na | 12.3847 | APE10-dist-na | 10.1712 | APE9-dist-in | 7.9197 | None | None | None | XRAY | 1.92 | 0.208 | 0.234 | A | 315.0 | 301.0 | 11 | 30 | 30 | 0 | [[610, 907]] | 1.0 | 3zos | TYR_DDR1_HUMAN | TYR | 1.5e-92 | 315.5 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V04B | P11362 | 458 | 765 | 822.0 | 0LI:1771 | Type2 | Inactive | DFGout | 13.974 | 9.8725 | BBAminus | -127.4, -173.98 | -164.99, 120.92 | -104.35, 44.71 | 306.97, 107.67 | 29.41, -12.23 | in-in | in | 7.692 | Saltbr-in | 3.0147 | HRD-in | -72.1, -51.88 | 81.11, -15.75 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.55, 155.16 | APE9-dihe-in | -98.03, 109.95 | APE8-dihe-out | -52.12, -21.56 | APE8-rot-na | 329.22 | APE67-dihe-in | -70.06, -7.36 | -58.08, -24.0 | APE12-dist-na | 19.5141 | APE11-dist-na | 20.9701 | APE10-dist-na | 19.2978 | APE9-dist-out | 11.5913 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | B | 309.0 | 289.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V01A | P11362 | 465 | 765 | 822.0 | 0LI:1776 | Type2 | Inactive | DFGout | 13.6478 | 9.6834 | None | -136.22, -176.63 | -157.46, 111.62 | -99.01, 999.0 | 301.26, 98.54 | 999.0, 999.0 | in-in | in | 7.8519 | Saltbr-in | 2.8239 | HRD-in | -71.33, -57.3 | 83.26, -24.31 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.02, 147.14 | APE9-dihe-in | -94.17, 112.67 | APE8-dihe-out | -54.82, -21.48 | APE8-rot-na | 334.27 | APE67-dihe-in | -70.4, -11.17 | -58.27, -24.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.7272 | C488A,C584S | None | None | XRAY | 2.33 | 0.191 | 0.238 | A | 309.0 | 273.0 | 28 | 30 | 22 | 8 | [[478, 756]] | 1.0 | 4v01 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V01B | P11362 | 461 | 763 | 822.0 | 0LI:1770 | Type2 | Inactive | DFGout | 13.4764 | 9.083 | None | -140.66, -178.05 | -156.06, 123.42 | -117.89, 999.0 | 302.59, 94.37 | 999.0, 999.0 | in-in | in | 7.9159 | Saltbr-in | 2.8067 | HRD-in | -63.92, -54.57 | 77.31, -15.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -101.11, 164.12 | APE9-dihe-in | -107.61, 109.54 | APE8-dihe-out | -56.39, -11.31 | APE8-rot-na | 332.13 | APE67-dihe-in | -66.82, -7.77 | -66.39, -26.4 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.8136 | C488A,C584S | None | None | XRAY | 2.33 | 0.191 | 0.238 | B | 309.0 | 275.0 | 28 | 30 | 22 | 8 | [[478, 756]] | 1.0 | 4v01 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V04A | P11362 | 463 | 765 | 822.0 | 0LI:1772 | Type2 | Inactive | DFGout | 14.0506 | 10.3941 | None | -127.25, -179.24 | -145.47, 116.11 | -167.94, 35.9 | 26.55, 54.39 | 23.93, -5.2 | in-in | in | 7.8637 | Saltbr-in | 3.2056 | HRD-in | -65.2, -58.04 | 83.28, -16.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.41, 155.12 | APE9-dihe-in | -98.09, 110.26 | APE8-dihe-out | -52.77, -21.99 | APE8-rot-na | 329.65 | APE67-dihe-in | -70.41, -8.08 | -56.89, -24.83 | APE12-dist-na | 19.6385 | APE11-dist-na | 21.0205 | APE10-dist-na | 19.3218 | APE9-dist-out | 11.7003 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | A | 309.0 | 293.0 | 10 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR4 | FGFR4_HUMAN | 4UXQA | P22455 | 452 | 750 | 802.0 | 0LI:1752 | Type2 | Inactive | DFGout | 13.2886 | 9.6881 | BBAminus | -132.52, -175.6 | -154.98, 108.32 | -101.68, -37.05 | 301.67, 99.59 | -82.32, -172.58 | in-in | in | 7.8131 | Saltbr-in | 2.7274 | HRD-in | -74.83, -56.93 | 88.13, -22.48 | in-out-out | SNCioo | out-out | ActLoopNT-out | 15.96 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -78.09, 139.64 | APE9-dihe-in | -109.24, 95.28 | APE8-dihe-out | -52.11, -28.25 | APE8-rot-na | 327.58 | APE67-dihe-in | -73.35, -9.88 | -60.02, -19.19 | APE12-dist-na | 12.2275 | APE11-dist-na | 12.9237 | APE10-dist-na | 10.1127 | APE9-dist-out | 11.6116 | C477A | None | None | XRAY | 1.85 | 0.205 | 0.268 | A | 309.0 | 286.0 | 13 | 30 | 30 | 0 | [[467, 745]] | 1.0 | 4uxq | TYR_FGFR4_HUMAN | TYR | 8.2e-101 | 342.6 | 1.0 | 261.0 | 261.0 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612.0 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 4TYJA | P22455 | 447 | 753 | 802.0 | 0LI:60801 | Type2 | Inactive | DFGout | 13.629 | 9.6017 | BBAminus | -136.8, -177.28 | -149.4, 114.79 | -98.18, 9.17 | 298.44, 103.78 | 79.91, -171.4 | in-in | in | 7.8197 | Saltbr-in | 2.7569 | HRD-in | -71.95, -55.51 | 84.74, -19.01 | in-out-out | SNCioo | out-out | ActLoopNT-out | 19.1078 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 130.68 | APE8-dihe-in | -83.91, 64.17 | APE8-rot-na | 36.55 | APE67-dihe-in | -73.09, -8.81 | -53.35, -41.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.8188 | None | None | None | XRAY | 2.45 | 0.217 | 0.247 | A | 311.0 | 275.0 | 32 | 30 | 15 | 15 | [[467, 745]] | 1.0 | 4tyj | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.0 | 1.0 | 261.0 | 261.0 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612.0 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 4QRCA | P22455 | 454 | 750 | 802.0 | 0LI:802 | Type2 | Inactive | DFGout | 13.8479 | 9.4478 | None | -128.93, 176.89 | -168.87, 140.49 | 58.84, 41.6 | 314.29, 151.03 | 128.95, 161.76 | in-in | in | 7.2685 | Saltbr-in | 2.5447 | HRD-in | -73.23, -52.1 | 79.8, -10.52 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6625 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -79.02, 138.09 | APE9-dihe-in | -108.95, 92.74 | APE8-dihe-out | -61.85, -18.49 | APE8-rot-na | 333.49 | APE67-dihe-in | -72.31, -7.32 | -59.05, -24.57 | APE12-dist-na | 19.5374 | APE11-dist-na | 21.0468 | APE10-dist-na | 16.8729 | APE9-dist-out | 12.0169 | C477A,R664E | None | None | XRAY | 1.901 | 0.173 | 0.207 | A | 323.0 | 297.0 | 0 | 30 | 30 | 0 | [[467, 745]] | 1.0 | 4qrc | TYR_FGFR4_HUMAN | TYR | 1.5e-100 | 341.7 | 1.0 | 261.0 | 261.0 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612.0 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | KIT | KIT_HUMAN | 8S17A | P10721 | 567 | 931 | 976.0 | 0LI:61001 | Type2 | Inactive | DFGout | 15.4253 | 9.9509 | BBAminus | -145.25, 179.39 | -143.98, 106.64 | -67.34, -40.16 | 274.67, 96.68 | 58.73, -115.03 | in-in | in | 7.749 | Saltbr-in | 2.6955 | HRD-in | -73.68, -54.05 | 81.88, -13.47 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.3106 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -118.0, 112.95 | APE9-dihe-in | -124.02, 150.83 | APE8-dihe-in | -80.03, 74.01 | APE8-rot-na | 32.18 | APE67-dihe-in | -67.91, -14.83 | -61.86, -40.28 | APE12-dist-na | 16.635 | APE11-dist-na | 13.2018 | APE10-dist-na | 11.5146 | APE9-dist-in | 7.7012 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.2 | 0.203 | 0.228 | A | 327.0 | 287.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s17 | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S17B | P10721 | 578 | 931 | 976.0 | 0LI:61001 | Type2 | Inactive | DFGout | 15.2272 | 9.8787 | BBAminus | -145.11, 172.96 | -138.62, 103.76 | -65.65, -38.27 | 276.93, 92.02 | 61.53, -118.4 | in-in | in | 7.6517 | Saltbr-in | 2.7434 | HRD-in | -69.78, -55.3 | 82.77, -9.47 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4084 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.26, 116.47 | APE9-dihe-in | -128.18, 149.58 | APE8-dihe-in | -80.46, 72.63 | APE8-rot-na | 32.73 | APE67-dihe-in | -67.64, -17.39 | -58.96, -38.89 | APE12-dist-na | 16.5047 | APE11-dist-na | 13.3085 | APE10-dist-na | 11.7177 | APE9-dist-in | 7.9746 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.2 | 0.203 | 0.228 | B | 327.0 | 276.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s17 | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 4U0IA | P10721 | 565 | 933 | 976.0 | 0LI:1001 | Type2 | Inactive | DFGout | 15.1525 | 9.7578 | BBAminus | -145.62, -174.19 | -155.03, 115.98 | -76.91, -26.31 | 285.47, 90.73 | 51.17, -116.44 | in-in | in | 7.6858 | Saltbr-in | 2.6193 | HRD-in | -74.87, -53.81 | 79.28, -20.01 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4462 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.86, 120.83 | APE9-dihe-in | -126.16, 149.12 | APE8-dihe-in | -78.54, 70.26 | APE8-rot-na | 32.2 | APE67-dihe-in | -61.59, -16.21 | -59.65, -43.09 | APE12-dist-na | 17.1926 | APE11-dist-na | 14.015 | APE10-dist-na | 12.1639 | APE9-dist-in | 7.6808 | None | None | None | XRAY | 2.0 | 0.204 | 0.239 | A | 315.0 | 297.0 | 12 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 4u0i | TYR_KIT_HUMAN | TYR | 3.8e-102 | 347.0 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | ROR1 | ROR1_HUMAN | 6TU9A | Q01973 | 460 | 749 | 937.0 | 0LI:801 | Type1 | Pseudo | None | 999.0 | 999.0 | None | -143.45, 175.76 | -148.29, 81.04 | -104.43, 119.64 | 999.0, 999.0 | -53.65, -7.79 | in-in | in | 8.2268 | Saltbr-in | 2.7255 | HRD-in | -69.35, -57.72 | 81.6, -11.35 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.3953 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -88.59, 129.49 | APE9-dihe-in | -125.15, 133.19 | APE8-dihe-in | -78.4, 68.8 | APE8-rot-na | 36.93 | APE67-dihe-in | -68.17, -18.18 | -55.42, -35.07 | APE12-dist-na | 999.0 | APE11-dist-na | 15.6904 | APE10-dist-na | 11.605 | APE9-dist-in | 6.9924 | None | None | None | XRAY | 1.94 | 0.21 | 0.241 | A | 306.0 | 268.0 | 22 | 30 | 26 | 4 | [[473, 748]] | 1.0 | 6tu9 | TYR_ROR1_HUMAN | TYR | 1.2e-94 | 322.4 | 2.0 | 260.0 | 259.0 | 632 | 633 | 634 | 636 | 638 | 506 | 523 | 527 | 612 | 614 | 613 | 615.0 | 674 | 662 | 657 | 656 | 655 | 654 | 653 | 652 | 651 | 553 | Inactive tyrosine-protein kinase transmembrane receptor ROR1 |
| TYR | ROR1 | ROR1_HUMAN | 6TU9B | Q01973 | 465 | 750 | 937.0 | 0LI:801 | Type1 | Pseudo | None | 999.0 | 999.0 | None | -143.03, 176.7 | -144.7, 81.77 | -85.65, -31.03 | 999.0, 999.0 | 92.49, -44.82 | in-in | in | 8.2829 | Saltbr-in | 2.9737 | HRD-in | -64.86, -61.91 | 82.91, -9.99 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -100.96, 129.63 | APE9-dihe-in | -119.15, 127.45 | APE8-dihe-in | -76.72, 68.52 | APE8-rot-na | 33.66 | APE67-dihe-in | -67.05, -20.69 | -57.04, -32.64 | APE12-dist-na | 17.0248 | APE11-dist-na | 15.144 | APE10-dist-na | 11.1966 | APE9-dist-in | 6.9698 | None | None | None | XRAY | 1.94 | 0.21 | 0.241 | B | 306.0 | 261.0 | 25 | 30 | 28 | 2 | [[473, 748]] | 1.0 | 6tu9 | TYR_ROR1_HUMAN | TYR | 1.2e-94 | 322.4 | 2.0 | 260.0 | 259.0 | 632 | 633 | 634 | 636 | 638 | 506 | 523 | 527 | 612 | 614 | 613 | 615.0 | 674 | 662 | 657 | 656 | 655 | 654 | 653 | 652 | 651 | 553 | Inactive tyrosine-protein kinase transmembrane receptor ROR1 |
| TYR | SRC | SRC_HUMAN | 7OTEA | P12931 | 261 | 536 | 536.0 | 0LI:601 | Type2 | Inactive | DFGout | 13.678 | 9.0255 | BBAminus | -119.79, 176.26 | -136.22, 145.66 | -117.56, 59.41 | 289.7, 90.17 | 173.51, 999.0 | in-in | in | 7.8789 | Saltbr-in | 2.5317 | HRD-in | -78.56, -49.16 | 85.49, -24.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 150.65 | APE8-dihe-in | -61.46, 92.79 | APE8-rot-na | 30.48 | APE67-dihe-in | -70.25, -17.48 | -54.65, -43.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.6182 | None | None | None | XRAY | 2.49 | 0.179 | 0.252 | A | 293.0 | 259.0 | 17 | 29 | 12 | 17 | [[270, 521]] | 1.0 | 7ote | TYR_SRC_HUMAN | TYR | 1.8e-94 | 321.9 | 1.0 | 260.0 | 260.0 | 406 | 407 | 408 | 410 | 412 | 298 | 313 | 317 | 386 | 388 | 387 | 389.0 | 447 | 435 | 430 | 429 | 428 | 427 | 426 | 425 | 424 | 342 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_HUMAN | 7OTEB | P12931 | 261 | 536 | 536.0 | 0LI:601 | Type2 | Inactive | DFGout | 14.5076 | 9.1805 | BBAminus | -149.51, 179.45 | -147.71, 103.83 | -80.1, -7.38 | 295.65, 135.68 | 68.38, 999.0 | in-out | in | 8.9117 | Saltbr-out | 4.1347 | HRD-in | -81.29, -57.98 | 98.12, -42.77 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.79 | APE8-dihe-in | -102.78, 62.88 | APE8-rot-na | 39.14 | APE67-dihe-in | -65.77, -18.22 | -41.35, -46.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.2979 | None | None | None | XRAY | 2.49 | 0.179 | 0.252 | B | 293.0 | 259.0 | 17 | 29 | 12 | 17 | [[270, 521]] | 1.0 | 7ote | TYR_SRC_HUMAN | TYR | 1.8e-94 | 321.9 | 1.0 | 260.0 | 260.0 | 406 | 407 | 408 | 410 | 412 | 298 | 313 | 317 | 386 | 388 | 387 | 389.0 | 447 | 435 | 430 | 429 | 428 | 427 | 426 | 425 | 424 | 342 | Proto-oncogene tyrosine-protein kinase Src |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SRC | SRC_CHICK | 7WF5A | P00523 | 257 | 533 | 533.0 | 0LI:601 | Type2 | Inactive | DFGout | 13.2929 | 8.8534 | BBAminus | -138.86, 178.47 | -148.72, 117.06 | -103.55, 7.74 | 290.87, 100.32 | 61.55, 53.93 | in-in | in | 7.6711 | Saltbr-in | 2.6168 | HRD-in | -81.35, -59.57 | 92.68, -15.97 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.23 | APE8-dihe-in | -80.1, 61.84 | APE8-rot-na | 34.61 | APE67-dihe-in | -62.67, -20.24 | -53.79, -38.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.0033 | None | None | None | XRAY | 1.798 | 0.163 | 0.183 | A | 286.0 | 261.0 | 16 | 29 | 13 | 16 | [[267, 518]] | 1.0 | 7wf5 | Gallus gallus | TYR_SRC_CHICK | TYR | 3.4e-94 | 320.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 7WF5B | P00523 | 254 | 533 | 533.0 | 0LI:601 | Type2 | Inactive | DFGout | 13.3369 | 8.808 | BBAminus | -139.72, 178.97 | -149.88, 114.3 | -104.08, 8.92 | 292.96, 104.73 | 64.81, 53.74 | in-in | in | 7.856 | Saltbr-in | 2.7923 | HRD-in | -81.76, -58.24 | 93.94, -19.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 96.23 | APE8-dihe-in | -81.79, 58.44 | APE8-rot-na | 33.89 | APE67-dihe-in | -61.6, -25.83 | -54.2, -35.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.5617 | None | None | None | XRAY | 1.798 | 0.163 | 0.183 | B | 286.0 | 265.0 | 15 | 29 | 14 | 15 | [[267, 518]] | 1.0 | 7wf5 | Gallus gallus | TYR_SRC_CHICK | TYR | 3.4e-94 | 320.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| STE | MAP3K2 | M3K2_HUMAN | 9P6AA | Q9Y2U5 | 351 | 617 | 619.0 | 0LI:701 | Type2 | Inactive | DFGout | 14.1431 | 9.8906 | BBAminus | -146.02, -172.59 | -157.95, 116.33 | -87.88, -36.33 | 294.81, 102.45 | -88.54, 36.79 | in-in | in | 8.4578 | Saltbr-in | 2.5939 | HRD-in | -76.59, -52.31 | 80.62, -19.75 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_oooo | APE10-dihe-na | -98.17, -51.62 | APE9-dihe-na | -96.01, 162.48 | APE8-dihe-in | -81.48, 131.06 | APE8-rot-out | 69.69 | APE67-dihe-in | -67.88, -22.22 | -92.28, 3.15 | APE12-dist-out | 20.6817 | APE11-dist-out | 19.1439 | APE10-dist-out | 14.3088 | APE9-dist-out | 10.4562 | None | None | None | XRAY | 2.4 | 0.228 | 0.246 | A | 299.0 | 253.0 | 14 | 31 | 17 | 14 | [[356, 616]] | 1.0 | 9p6a | Homo sapiens | STE_MAP3K2_HUMAN | STE | 1.9e-81 | 279.1 | 1.0 | 257.0 | 257.0 | 500 | 501 | 502 | 504 | 506 | 385 | 406 | 410 | 480 | 482 | 481 | 483.0 | 543 | 531 | 526 | 525 | 524 | 523 | 522 | 521 | 520 | 438 | Mitogen-activated protein kinase kinase kinase 2 |
| STE | MAP3K2 | M3K2_HUMAN | 9P6AB | Q9Y2U5 | 347 | 618 | 619.0 | 0LI:701 | Type2 | Inactive | DFGout | 13.8018 | 9.7559 | None | -145.97, -173.02 | -157.2, 114.58 | -90.61, 158.12 | 297.06, 102.49 | 67.12, -99.7 | in-in | in | 8.6308 | Saltbr-in | 2.7273 | HRD-in | -74.0, -48.74 | 85.04, -22.17 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -168.99 | APE9-dihe-na | -96.92, -27.66 | APE8-dihe-in | -82.09, 127.1 | APE8-rot-out | 70.19 | APE67-dihe-in | -70.58, -23.59 | -96.42, -0.55 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 8.6373 | APE9-dist-out | 10.7871 | None | None | None | XRAY | 2.4 | 0.228 | 0.246 | B | 299.0 | 247.0 | 25 | 31 | 15 | 16 | [[356, 616]] | 1.0 | 9p6a | Homo sapiens | STE_MAP3K2_HUMAN | STE | 1.9e-81 | 279.1 | 1.0 | 257.0 | 257.0 | 500 | 501 | 502 | 504 | 506 | 385 | 406 | 410 | 480 | 482 | 481 | 483.0 | 543 | 531 | 526 | 525 | 524 | 523 | 522 | 521 | 520 | 438 | Mitogen-activated protein kinase kinase kinase 2 |
| TKL | BRAF | BRAF_HUMAN | 6P3DA | P15056 | 448 | 721 | 766.0 | 0LI:61001 | Type2 | Inactive | DFGout | 12.35 | 10.9052 | BBAminus | -138.54, -166.92 | -135.05, 80.45 | -80.66, -37.84 | 293.17, 97.28 | 81.0, 10.25 | in-in | in | 8.6648 | Saltbr-in | 2.9974 | HRD-in | -65.6, -55.77 | 77.59, -19.55 | in-out-out | SNCioo | out-out | ActLoopNT-out | 19.9448 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnoo | APE10-dihe-na | 999.0, -19.82 | APE9-dihe-na | 76.62, -63.3 | APE8-dihe-out | -51.89, -23.77 | APE8-rot-out | 78.9 | APE67-dihe-in | -55.73, -23.59 | -56.01, -24.35 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 12.7002 | APE9-dist-out | 11.8707 | None | None | None | XRAY | 2.11 | 0.188 | 0.245 | A | 297.0 | 261.0 | 13 | 30 | 17 | 13 | [[457, 716]] | 1.0 | 6p3d | Homo sapiens | TKL_BRAF_HUMAN | TKL | 5.8e-84 | 287.7 | 4.0 | 267.0 | 264.0 | 593 | 594 | 595 | 597 | 599 | 483 | 501 | 505 | 573 | 575 | 574 | 576.0 | 638 | 623 | 618 | 617 | 616 | 615 | 614 | 613 | 612 | 530 | Serine/threonine-protein kinase B-raf |
| TKL | IRAK4 | IRAK4_HUMAN | 6EG9A | Q9NWZ3 | 164 | 459 | 460.0 | 0LI:501 | Type2 | Inactive | DFGout | 14.0712 | 10.7156 | None | -127.45, 167.3 | -138.69, 101.47 | -85.85, 140.23 | 309.7, 100.41 | -43.19, 999.0 | in-out | in | 9.0273 | Saltbr-out | 6.6465 | HRD-in | -71.51, -48.43 | 70.86, -5.67 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 6.91 | APE9-dihe-na | 158.59, -165.8 | APE8-dihe-in | -114.99, 116.82 | APE8-rot-in | 299.55 | APE67-dihe-in | -67.65, -20.43 | -63.19, -29.42 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.972 | None | None | None | XRAY | 2.414 | 0.224 | 0.249 | A | 312.0 | 276.0 | 20 | 30 | 13 | 17 | [[183, 456]] | 1.0 | 6eg9 | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.6e-84 | 288.0 | 5.0 | 266.0 | 262.0 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311.0 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | IRAK4 | IRAK4_HUMAN | 6EG9B | Q9NWZ3 | 165 | 459 | 460.0 | 0LI:501 | Type2 | Inactive | DFGout | 14.2443 | 9.3953 | None | -135.81, 174.82 | -152.29, 126.78 | -163.75, 999.0 | 33.58, 60.29 | 999.0, 999.0 | in-in | in | 8.9787 | Saltbr-in | 3.0904 | HRD-in | -69.81, -51.27 | 77.39, -7.02 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 146.5 | APE9-dihe-na | 95.5, 175.38 | APE8-dihe-in | -117.78, 118.94 | APE8-rot-in | 307.93 | APE67-dihe-in | -67.02, -18.64 | -61.22, -30.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 3.6297 | None | None | None | XRAY | 2.414 | 0.224 | 0.249 | B | 312.0 | 274.0 | 21 | 30 | 12 | 18 | [[183, 456]] | 1.0 | 6eg9 | Homo sapiens | TKL_IRAK4_HUMAN | TKL | 4.6e-84 | 288.0 | 5.0 | 266.0 | 262.0 | 328 | 329 | 330 | 332 | 334 | 213 | 233 | 237 | 308 | 310 | 309 | 311.0 | 369 | 358 | 353 | 352 | 351 | 350 | 349 | 348 | 347 | 263 | Interleukin-1 receptor-associated kinase 4 |
| TKL | LRRK2 | LRRK2_HUMAN | 8U8AB | Q5S007 | 558 | 2526 | 2527.0 | 0LI:2601 | Type2 | Inactive | DFGout | 14.859 | 10.8454 | BBAminus | -150.37, 144.32 | -124.19, 97.68 | -69.79, -11.11 | 321.73, 111.63 | 66.57, 27.33 | in-out | in | 8.8739 | Saltbr-out | 3.6727 | HRD-out | -76.07, 95.41 | -48.17, -63.17 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 177.03 | APE8-dihe-in | -61.6, 136.03 | APE8-rot-in | 305.18 | APE67-dihe-in | -74.33, -25.33 | -56.72, -44.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 6.2972 | None | None | None | EM | 3.4 | 999.0 | 999.0 | B | 2527.0 | 1705.0 | 29 | 26 | 13 | 13 | [[1875, 2134]] | 1.0 | 8u8a | Homo sapiens | TKL_LRRK2_HUMAN | TKL | 3.8e-57 | 200.3 | 5.0 | 266.0 | 262.0 | 2016 | 2017 | 2018 | 2020 | 2022 | 1906 | 1920 | 1924 | 1991 | 1993 | 1992 | 1994.0 | 2055 | 2042 | 2037 | 2036 | 2035 | 2034 | 2033 | 2032 | 2031 | 1948 | Leucine-rich repeat serine/threonine-protein kinase 2 |
| TKL | LRRK2 | LRRK2_HUMAN | 8U8AC | Q5S007 | 558 | 2526 | 2527.0 | 0LI:2601 | Type2 | Inactive | DFGout | 14.8696 | 10.8459 | BBAminus | -150.46, 144.31 | -124.23, 97.69 | -69.77, -11.06 | 321.78, 111.5 | 66.48, 27.35 | in-out | in | 8.8719 | Saltbr-out | 3.6608 | HRD-out | -76.02, 95.48 | -48.33, -63.13 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 177.01 | APE8-dihe-in | -61.57, 135.98 | APE8-rot-in | 305.14 | APE67-dihe-in | -74.37, -25.35 | -56.73, -44.17 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 6.3006 | None | None | None | EM | 3.4 | 999.0 | 999.0 | C | 2527.0 | 1705.0 | 29 | 26 | 13 | 13 | [[1875, 2134]] | 1.0 | 8u8a | Homo sapiens | TKL_LRRK2_HUMAN | TKL | 3.8e-57 | 200.3 | 5.0 | 266.0 | 262.0 | 2016 | 2017 | 2018 | 2020 | 2022 | 1906 | 1920 | 1924 | 1991 | 1993 | 1992 | 1994.0 | 2055 | 2042 | 2037 | 2036 | 2035 | 2034 | 2033 | 2032 | 2031 | 1948 | Leucine-rich repeat serine/threonine-protein kinase 2 |
| TKL | RIPK2 | RIPK2_HUMAN | 4C8BA | O43353 | 8 | 316 | 540.0 | 0LI:1000 | Type2 | Inactive | DFGout | 12.7285 | 8.5841 | None | -142.99, -175.55 | -154.35, 140.4 | -129.56, 999.0 | 290.55, 114.67 | 999.0, 999.0 | in-in | in | 8.2431 | Saltbr-in | 2.8173 | HRD-in | -79.84, -58.2 | 64.89, 19.36 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -36.9 | APE8-dihe-out | -84.71, -55.98 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.98, -25.64 | -68.13, -16.01 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.2944 | None | None | None | XRAY | 2.75 | 0.203 | 0.244 | A | 334.0 | 279.0 | 30 | 33 | 11 | 22 | [[18, 292]] | 1.0 | 4c8b | Homo sapiens | TKL_RIPK2_HUMAN | TKL | 3.4e-73 | 252.4 | 4.0 | 266.0 | 263.0 | 163 | 164 | 165 | 167 | 169 | 47 | 66 | 70 | 143 | 145 | 144 | 146.0 | 211 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 96 | Receptor-interacting serine/threonine-protein kinase 2 |
| TKL | RIPK2 | RIPK2_HUMAN | 4C8BB | O43353 | 9 | 316 | 540.0 | 0LI:1000 | Type2 | Inactive | DFGout | 12.8402 | 8.8595 | None | -140.63, -176.63 | -153.18, 138.54 | -119.75, 999.0 | 285.35, 113.34 | 999.0, 999.0 | in-in | in | 8.2645 | Saltbr-in | 2.8058 | HRD-in | -79.98, -59.74 | 66.42, 17.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -39.27 | APE8-dihe-out | -68.6, -38.75 | APE8-rot-out | 169.06 | APE67-dihe-in | -64.78, -24.38 | -61.46, -15.15 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 13.4449 | None | None | None | XRAY | 2.75 | 0.203 | 0.244 | B | 334.0 | 281.0 | 27 | 33 | 11 | 22 | [[18, 292]] | 1.0 | 4c8b | Homo sapiens | TKL_RIPK2_HUMAN | TKL | 3.4e-73 | 252.4 | 4.0 | 266.0 | 263.0 | 163 | 164 | 165 | 167 | 169 | 47 | 66 | 70 | 143 | 145 | 144 | 146.0 | 211 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 96 | Receptor-interacting serine/threonine-protein kinase 2 |
| TYR | DDR1 | DDR1_HUMAN | 3ZOSB | Q08345 | 601 | 913 | 913.0 | 0LI:61000 | Type2 | Inactive | DFGout | 13.6455 | 9.6295 | BBAminus | -143.84, 178.94 | -153.3, 114.42 | -82.71, -15.18 | 287.49, 108.73 | 52.14, -127.46 | in-in | in | 7.9604 | Saltbr-in | 2.8828 | HRD-in | -60.43, -59.89 | 83.25, -8.8 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.4003 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.91, 133.24 | APE9-dihe-in | -130.81, 142.32 | APE8-dihe-in | -80.63, 68.61 | APE8-rot-na | 30.08 | APE67-dihe-in | -67.12, -16.99 | -59.3, -31.33 | APE12-dist-na | 11.7194 | APE11-dist-na | 12.9393 | APE10-dist-na | 10.2231 | APE9-dist-in | 7.9237 | None | None | None | XRAY | 1.92 | 0.208 | 0.234 | B | 315.0 | 301.0 | 12 | 30 | 30 | 0 | [[610, 907]] | 1.0 | 3zos | Homo sapiens | TYR_DDR1_HUMAN | TYR | 1.5e-92 | 315.5 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 3ZOSA | Q08345 | 602 | 913 | 913.0 | 0LI:61000,0LI:61004 | Type2,Allosteric | Inactive | DFGout | 13.6836 | 9.7654 | BBAminus | -140.01, 179.9 | -153.22, 112.84 | -85.26, -13.51 | 285.68, 107.96 | 48.92, -126.09 | in-in | in | 7.9981 | Saltbr-in | 2.8815 | HRD-in | -61.25, -58.95 | 80.5, -7.41 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.4763 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.17, 140.69 | APE9-dihe-in | -129.43, 143.43 | APE8-dihe-in | -82.4, 69.11 | APE8-rot-na | 29.15 | APE67-dihe-in | -67.51, -15.14 | -58.33, -33.07 | APE12-dist-na | 11.7075 | APE11-dist-na | 12.3847 | APE10-dist-na | 10.1712 | APE9-dist-in | 7.9197 | None | None | None | XRAY | 1.92 | 0.208 | 0.234 | A | 315.0 | 301.0 | 11 | 30 | 30 | 0 | [[610, 907]] | 1.0 | 3zos | Homo sapiens | TYR_DDR1_HUMAN | TYR | 1.5e-92 | 315.5 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V04B | P11362 | 458 | 765 | 822.0 | 0LI:1771 | Type2 | Inactive | DFGout | 13.974 | 9.8725 | BBAminus | -127.4, -173.98 | -164.99, 120.92 | -104.35, 44.71 | 306.97, 107.67 | 29.41, -12.23 | in-in | in | 7.692 | Saltbr-in | 3.0147 | HRD-in | -72.1, -51.88 | 81.11, -15.75 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.55, 155.16 | APE9-dihe-in | -98.03, 109.95 | APE8-dihe-out | -52.12, -21.56 | APE8-rot-na | 329.22 | APE67-dihe-in | -70.06, -7.36 | -58.08, -24.0 | APE12-dist-na | 19.5141 | APE11-dist-na | 20.9701 | APE10-dist-na | 19.2978 | APE9-dist-out | 11.5913 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | B | 309.0 | 289.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V01A | P11362 | 465 | 765 | 822.0 | 0LI:1776 | Type2 | Inactive | DFGout | 13.6478 | 9.6834 | None | -136.22, -176.63 | -157.46, 111.62 | -99.01, 999.0 | 301.26, 98.54 | 999.0, 999.0 | in-in | in | 7.8519 | Saltbr-in | 2.8239 | HRD-in | -71.33, -57.3 | 83.26, -24.31 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.02, 147.14 | APE9-dihe-in | -94.17, 112.67 | APE8-dihe-out | -54.82, -21.48 | APE8-rot-na | 334.27 | APE67-dihe-in | -70.4, -11.17 | -58.27, -24.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.7272 | C488A,C584S | None | None | XRAY | 2.33 | 0.191 | 0.238 | A | 309.0 | 273.0 | 28 | 30 | 22 | 8 | [[478, 756]] | 1.0 | 4v01 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V01B | P11362 | 461 | 763 | 822.0 | 0LI:1770 | Type2 | Inactive | DFGout | 13.4764 | 9.083 | None | -140.66, -178.05 | -156.06, 123.42 | -117.89, 999.0 | 302.59, 94.37 | 999.0, 999.0 | in-in | in | 7.9159 | Saltbr-in | 2.8067 | HRD-in | -63.92, -54.57 | 77.31, -15.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -101.11, 164.12 | APE9-dihe-in | -107.61, 109.54 | APE8-dihe-out | -56.39, -11.31 | APE8-rot-na | 332.13 | APE67-dihe-in | -66.82, -7.77 | -66.39, -26.4 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.8136 | C488A,C584S | None | None | XRAY | 2.33 | 0.191 | 0.238 | B | 309.0 | 275.0 | 28 | 30 | 22 | 8 | [[478, 756]] | 1.0 | 4v01 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V04A | P11362 | 463 | 765 | 822.0 | 0LI:1772 | Type2 | Inactive | DFGout | 14.0506 | 10.3941 | None | -127.25, -179.24 | -145.47, 116.11 | -167.94, 35.9 | 26.55, 54.39 | 23.93, -5.2 | in-in | in | 7.8637 | Saltbr-in | 3.2056 | HRD-in | -65.2, -58.04 | 83.28, -16.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.41, 155.12 | APE9-dihe-in | -98.09, 110.26 | APE8-dihe-out | -52.77, -21.99 | APE8-rot-na | 329.65 | APE67-dihe-in | -70.41, -8.08 | -56.89, -24.83 | APE12-dist-na | 19.6385 | APE11-dist-na | 21.0205 | APE10-dist-na | 19.3218 | APE9-dist-out | 11.7003 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | A | 309.0 | 293.0 | 10 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR4 | FGFR4_HUMAN | 4UXQA | P22455 | 452 | 750 | 802.0 | 0LI:1752 | Type2 | Inactive | DFGout | 13.2886 | 9.6881 | BBAminus | -132.52, -175.6 | -154.98, 108.32 | -101.68, -37.05 | 301.67, 99.59 | -82.32, -172.58 | in-in | in | 7.8131 | Saltbr-in | 2.7274 | HRD-in | -74.83, -56.93 | 88.13, -22.48 | in-out-out | SNCioo | out-out | ActLoopNT-out | 15.96 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -78.09, 139.64 | APE9-dihe-in | -109.24, 95.28 | APE8-dihe-out | -52.11, -28.25 | APE8-rot-na | 327.58 | APE67-dihe-in | -73.35, -9.88 | -60.02, -19.19 | APE12-dist-na | 12.2275 | APE11-dist-na | 12.9237 | APE10-dist-na | 10.1127 | APE9-dist-out | 11.6116 | C477A | None | None | XRAY | 1.85 | 0.205 | 0.268 | A | 309.0 | 286.0 | 13 | 30 | 30 | 0 | [[467, 745]] | 1.0 | 4uxq | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 8.2e-101 | 342.6 | 1.0 | 261.0 | 261.0 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612.0 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 4TYJA | P22455 | 447 | 753 | 802.0 | 0LI:60801 | Type2 | Inactive | DFGout | 13.629 | 9.6017 | BBAminus | -136.8, -177.28 | -149.4, 114.79 | -98.18, 9.17 | 298.44, 103.78 | 79.91, -171.4 | in-in | in | 7.8197 | Saltbr-in | 2.7569 | HRD-in | -71.95, -55.51 | 84.74, -19.01 | in-out-out | SNCioo | out-out | ActLoopNT-out | 19.1078 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 130.68 | APE8-dihe-in | -83.91, 64.17 | APE8-rot-na | 36.55 | APE67-dihe-in | -73.09, -8.81 | -53.35, -41.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.8188 | None | None | None | XRAY | 2.45 | 0.217 | 0.247 | A | 311.0 | 275.0 | 32 | 30 | 15 | 15 | [[467, 745]] | 1.0 | 4tyj | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.2e-100 | 342.0 | 1.0 | 261.0 | 261.0 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612.0 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | FGFR4 | FGFR4_HUMAN | 4QRCA | P22455 | 454 | 750 | 802.0 | 0LI:802 | Type2 | Inactive | DFGout | 13.8479 | 9.4478 | None | -128.93, 176.89 | -168.87, 140.49 | 58.84, 41.6 | 314.29, 151.03 | 128.95, 161.76 | in-in | in | 7.2685 | Saltbr-in | 2.5447 | HRD-in | -73.23, -52.1 | 79.8, -10.52 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6625 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -79.02, 138.09 | APE9-dihe-in | -108.95, 92.74 | APE8-dihe-out | -61.85, -18.49 | APE8-rot-na | 333.49 | APE67-dihe-in | -72.31, -7.32 | -59.05, -24.57 | APE12-dist-na | 19.5374 | APE11-dist-na | 21.0468 | APE10-dist-na | 16.8729 | APE9-dist-out | 12.0169 | C477A,R664E | None | None | XRAY | 1.901 | 0.173 | 0.207 | A | 323.0 | 297.0 | 0 | 30 | 30 | 0 | [[467, 745]] | 1.0 | 4qrc | Homo sapiens | TYR_FGFR4_HUMAN | TYR | 1.5e-100 | 341.7 | 1.0 | 261.0 | 261.0 | 629 | 630 | 631 | 633 | 635 | 503 | 520 | 524 | 609 | 611 | 610 | 612.0 | 671 | 659 | 654 | 653 | 652 | 651 | 650 | 649 | 648 | 551 | Fibroblast growth factor receptor 4 |
| TYR | KIT | KIT_HUMAN | 8S17A | P10721 | 567 | 931 | 976.0 | 0LI:61001 | Type2 | Inactive | DFGout | 15.4253 | 9.9509 | BBAminus | -145.25, 179.39 | -143.98, 106.64 | -67.34, -40.16 | 274.67, 96.68 | 58.73, -115.03 | in-in | in | 7.749 | Saltbr-in | 2.6955 | HRD-in | -73.68, -54.05 | 81.88, -13.47 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.3106 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -118.0, 112.95 | APE9-dihe-in | -124.02, 150.83 | APE8-dihe-in | -80.03, 74.01 | APE8-rot-na | 32.18 | APE67-dihe-in | -67.91, -14.83 | -61.86, -40.28 | APE12-dist-na | 16.635 | APE11-dist-na | 13.2018 | APE10-dist-na | 11.5146 | APE9-dist-in | 7.7012 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.2 | 0.203 | 0.228 | A | 327.0 | 287.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s17 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S17B | P10721 | 578 | 931 | 976.0 | 0LI:61001 | Type2 | Inactive | DFGout | 15.2272 | 9.8787 | BBAminus | -145.11, 172.96 | -138.62, 103.76 | -65.65, -38.27 | 276.93, 92.02 | 61.53, -118.4 | in-in | in | 7.6517 | Saltbr-in | 2.7434 | HRD-in | -69.78, -55.3 | 82.77, -9.47 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4084 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.26, 116.47 | APE9-dihe-in | -128.18, 149.58 | APE8-dihe-in | -80.46, 72.63 | APE8-rot-na | 32.73 | APE67-dihe-in | -67.64, -17.39 | -58.96, -38.89 | APE12-dist-na | 16.5047 | APE11-dist-na | 13.3085 | APE10-dist-na | 11.7177 | APE9-dist-in | 7.9746 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.2 | 0.203 | 0.228 | B | 327.0 | 276.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s17 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 4U0IA | P10721 | 565 | 933 | 976.0 | 0LI:1001 | Type2 | Inactive | DFGout | 15.1525 | 9.7578 | BBAminus | -145.62, -174.19 | -155.03, 115.98 | -76.91, -26.31 | 285.47, 90.73 | 51.17, -116.44 | in-in | in | 7.6858 | Saltbr-in | 2.6193 | HRD-in | -74.87, -53.81 | 79.28, -20.01 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4462 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.86, 120.83 | APE9-dihe-in | -126.16, 149.12 | APE8-dihe-in | -78.54, 70.26 | APE8-rot-na | 32.2 | APE67-dihe-in | -61.59, -16.21 | -59.65, -43.09 | APE12-dist-na | 17.1926 | APE11-dist-na | 14.015 | APE10-dist-na | 12.1639 | APE9-dist-in | 7.6808 | None | None | None | XRAY | 2.0 | 0.204 | 0.239 | A | 315.0 | 297.0 | 12 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 4u0i | Homo sapiens | TYR_KIT_HUMAN | TYR | 3.8e-102 | 347.0 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | ROR1 | ROR1_HUMAN | 6TU9A | Q01973 | 460 | 749 | 937.0 | 0LI:801 | Type1 | Pseudo | None | 999.0 | 999.0 | None | -143.45, 175.76 | -148.29, 81.04 | -104.43, 119.64 | 999.0, 999.0 | -53.65, -7.79 | in-in | in | 8.2268 | Saltbr-in | 2.7255 | HRD-in | -69.35, -57.72 | 81.6, -11.35 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.3953 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -88.59, 129.49 | APE9-dihe-in | -125.15, 133.19 | APE8-dihe-in | -78.4, 68.8 | APE8-rot-na | 36.93 | APE67-dihe-in | -68.17, -18.18 | -55.42, -35.07 | APE12-dist-na | 999.0 | APE11-dist-na | 15.6904 | APE10-dist-na | 11.605 | APE9-dist-in | 6.9924 | None | None | None | XRAY | 1.94 | 0.21 | 0.241 | A | 306.0 | 268.0 | 22 | 30 | 26 | 4 | [[473, 748]] | 1.0 | 6tu9 | Homo sapiens | TYR_ROR1_HUMAN | TYR | 1.2e-94 | 322.4 | 2.0 | 260.0 | 259.0 | 632 | 633 | 634 | 636 | 638 | 506 | 523 | 527 | 612 | 614 | 613 | 615.0 | 674 | 662 | 657 | 656 | 655 | 654 | 653 | 652 | 651 | 553 | Inactive tyrosine-protein kinase transmembrane receptor ROR1 |
| TYR | ROR1 | ROR1_HUMAN | 6TU9B | Q01973 | 465 | 750 | 937.0 | 0LI:801 | Type1 | Pseudo | None | 999.0 | 999.0 | None | -143.03, 176.7 | -144.7, 81.77 | -85.65, -31.03 | 999.0, 999.0 | 92.49, -44.82 | in-in | in | 8.2829 | Saltbr-in | 2.9737 | HRD-in | -64.86, -61.91 | 82.91, -9.99 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -100.96, 129.63 | APE9-dihe-in | -119.15, 127.45 | APE8-dihe-in | -76.72, 68.52 | APE8-rot-na | 33.66 | APE67-dihe-in | -67.05, -20.69 | -57.04, -32.64 | APE12-dist-na | 17.0248 | APE11-dist-na | 15.144 | APE10-dist-na | 11.1966 | APE9-dist-in | 6.9698 | None | None | None | XRAY | 1.94 | 0.21 | 0.241 | B | 306.0 | 261.0 | 25 | 30 | 28 | 2 | [[473, 748]] | 1.0 | 6tu9 | Homo sapiens | TYR_ROR1_HUMAN | TYR | 1.2e-94 | 322.4 | 2.0 | 260.0 | 259.0 | 632 | 633 | 634 | 636 | 638 | 506 | 523 | 527 | 612 | 614 | 613 | 615.0 | 674 | 662 | 657 | 656 | 655 | 654 | 653 | 652 | 651 | 553 | Inactive tyrosine-protein kinase transmembrane receptor ROR1 |
| TYR | SRC | SRC_HUMAN | 7OTEA | P12931 | 261 | 536 | 536.0 | 0LI:601 | Type2 | Inactive | DFGout | 13.678 | 9.0255 | BBAminus | -119.79, 176.26 | -136.22, 145.66 | -117.56, 59.41 | 289.7, 90.17 | 173.51, 999.0 | in-in | in | 7.8789 | Saltbr-in | 2.5317 | HRD-in | -78.56, -49.16 | 85.49, -24.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 150.65 | APE8-dihe-in | -61.46, 92.79 | APE8-rot-na | 30.48 | APE67-dihe-in | -70.25, -17.48 | -54.65, -43.51 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.6182 | None | None | None | XRAY | 2.49 | 0.179 | 0.252 | A | 293.0 | 259.0 | 17 | 29 | 12 | 17 | [[270, 521]] | 1.0 | 7ote | Homo sapiens | TYR_SRC_HUMAN | TYR | 1.8e-94 | 321.9 | 1.0 | 260.0 | 260.0 | 406 | 407 | 408 | 410 | 412 | 298 | 313 | 317 | 386 | 388 | 387 | 389.0 | 447 | 435 | 430 | 429 | 428 | 427 | 426 | 425 | 424 | 342 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_HUMAN | 7OTEB | P12931 | 261 | 536 | 536.0 | 0LI:601 | Type2 | Inactive | DFGout | 14.5076 | 9.1805 | BBAminus | -149.51, 179.45 | -147.71, 103.83 | -80.1, -7.38 | 295.65, 135.68 | 68.38, 999.0 | in-out | in | 8.9117 | Saltbr-out | 4.1347 | HRD-in | -81.29, -57.98 | 98.12, -42.77 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.79 | APE8-dihe-in | -102.78, 62.88 | APE8-rot-na | 39.14 | APE67-dihe-in | -65.77, -18.22 | -41.35, -46.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.2979 | None | None | None | XRAY | 2.49 | 0.179 | 0.252 | B | 293.0 | 259.0 | 17 | 29 | 12 | 17 | [[270, 521]] | 1.0 | 7ote | Homo sapiens | TYR_SRC_HUMAN | TYR | 1.8e-94 | 321.9 | 1.0 | 260.0 | 260.0 | 406 | 407 | 408 | 410 | 412 | 298 | 313 | 317 | 386 | 388 | 387 | 389.0 | 447 | 435 | 430 | 429 | 428 | 427 | 426 | 425 | 424 | 342 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | ABL1 | ABL1_MOUSE | 3IK3A | P00520 | 229 | 513 | 1123.0 | 0LI:60001 | Type2 | Inactive | DFGout | 13.5039 | 9.4383 | BBAminus | -139.29, -179.88 | -153.49, 108.65 | -85.72, -9.94 | 290.6, 95.91 | 72.02, 48.56 | in-in | in | 7.934 | Saltbr-in | 2.5375 | HRD-in | -70.15, -60.9 | 90.87, -12.1 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -111.42, 120.77 | APE9-dihe-in | -114.74, 139.96 | APE8-dihe-in | -82.31, 89.85 | APE8-rot-na | 32.91 | APE67-dihe-in | -77.22, -7.68 | -48.36, -44.8 | APE12-dist-na | 16.0102 | APE11-dist-na | 11.8397 | APE10-dist-na | 8.4563 | APE9-dist-in | 7.993 | T315I | None | None | XRAY | 1.9 | 0.216 | 0.258 | A | 288.0 | 279.0 | 6 | 29 | 23 | 6 | [[242, 495]] | 1.0 | 3ik3 | Mus musculus | TYR_ABL1_MOUSE | TYR | 5.5e-100 | 339.9 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_MOUSE | 3IK3B | P00520 | 229 | 513 | 1123.0 | 0LI:60002 | Type2 | Inactive | DFGout | 13.4975 | 9.1697 | BBAminus | -129.46, 178.53 | -148.47, 114.27 | -91.94, -7.12 | 286.37, 101.01 | 64.82, 50.27 | in-in | in | 7.9919 | Saltbr-in | 2.6552 | HRD-in | -76.51, -54.44 | 85.69, -10.99 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.7027 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -129.88, 123.97 | APE9-dihe-in | -117.43, 141.07 | APE8-dihe-in | -76.99, 85.79 | APE8-rot-na | 29.46 | APE67-dihe-in | -85.08, -5.45 | -41.61, -41.71 | APE12-dist-na | 15.8259 | APE11-dist-na | 11.5962 | APE10-dist-na | 8.603 | APE9-dist-in | 7.8512 | T315I | None | None | XRAY | 1.9 | 0.216 | 0.258 | B | 288.0 | 285.0 | 0 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 3ik3 | Mus musculus | TYR_ABL1_MOUSE | TYR | 5.5e-100 | 339.9 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_MOUSE | 3OXZA | P00520 | 229 | 511 | 1123.0 | 0LI:60001 | Type2 | Inactive | DFGout | 13.3158 | 8.9403 | BBAminus | -130.11, -171.24 | -154.37, 127.79 | -115.42, 5.71 | 286.77, 98.95 | 48.45, 62.42 | in-in | in | 8.0038 | Saltbr-in | 3.005 | HRD-in | -71.2, -52.05 | 81.82, -16.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -90.47, 133.09 | APE9-dihe-in | -119.78, 140.42 | APE8-dihe-in | -76.32, 77.74 | APE8-rot-na | 32.13 | APE67-dihe-in | -76.96, -8.32 | -43.1, -46.11 | APE12-dist-na | 15.3775 | APE11-dist-na | 10.76 | APE10-dist-na | 8.339 | APE9-dist-out | 8.088 | None | None | None | XRAY | 2.2 | 0.218 | 0.261 | A | 284.0 | 267.0 | 16 | 29 | 19 | 10 | [[242, 495]] | 1.0 | 3oxz | Mus musculus | TYR_ABL1_MOUSE | TYR | 2.6e-100 | 341.0 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SRC | SRC_CHICK | 7WF5A | P00523 | 257 | 533 | 533.0 | 0LI:601 | Type2 | Inactive | DFGout | 13.2929 | 8.8534 | BBAminus | -138.86, 178.47 | -148.72, 117.06 | -103.55, 7.74 | 290.87, 100.32 | 61.55, 53.93 | in-in | in | 7.6711 | Saltbr-in | 2.6168 | HRD-in | -81.35, -59.57 | 92.68, -15.97 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.23 | APE8-dihe-in | -80.1, 61.84 | APE8-rot-na | 34.61 | APE67-dihe-in | -62.67, -20.24 | -53.79, -38.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.0033 | None | None | None | XRAY | 1.798 | 0.163 | 0.183 | A | 286.0 | 261.0 | 16 | 29 | 13 | 16 | [[267, 518]] | 1.0 | 7wf5 | Gallus gallus | TYR_SRC_CHICK | TYR | 3.4e-94 | 320.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | SRC | SRC_CHICK | 7WF5B | P00523 | 254 | 533 | 533.0 | 0LI:601 | Type2 | Inactive | DFGout | 13.3369 | 8.808 | BBAminus | -139.72, 178.97 | -149.88, 114.3 | -104.08, 8.92 | 292.96, 104.73 | 64.81, 53.74 | in-in | in | 7.856 | Saltbr-in | 2.7923 | HRD-in | -81.76, -58.24 | 93.94, -19.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 96.23 | APE8-dihe-in | -81.79, 58.44 | APE8-rot-na | 33.89 | APE67-dihe-in | -61.6, -25.83 | -54.2, -35.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.5617 | None | None | None | XRAY | 1.798 | 0.163 | 0.183 | B | 286.0 | 265.0 | 15 | 29 | 14 | 15 | [[267, 518]] | 1.0 | 7wf5 | Gallus gallus | TYR_SRC_CHICK | TYR | 3.4e-94 | 320.9 | 1.0 | 260.0 | 260.0 | 403 | 404 | 405 | 407 | 409 | 295 | 310 | 314 | 383 | 385 | 384 | 386.0 | 444 | 432 | 427 | 426 | 425 | 424 | 423 | 422 | 421 | 339 | Proto-oncogene tyrosine-protein kinase Src |
| TYR | ABL1 | ABL1_MOUSE | 3IK3A | P00520 | 229 | 513 | 1123.0 | 0LI:60001 | Type2 | Inactive | DFGout | 13.5039 | 9.4383 | BBAminus | -139.29, -179.88 | -153.49, 108.65 | -85.72, -9.94 | 290.6, 95.91 | 72.02, 48.56 | in-in | in | 7.934 | Saltbr-in | 2.5375 | HRD-in | -70.15, -60.9 | 90.87, -12.1 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -111.42, 120.77 | APE9-dihe-in | -114.74, 139.96 | APE8-dihe-in | -82.31, 89.85 | APE8-rot-na | 32.91 | APE67-dihe-in | -77.22, -7.68 | -48.36, -44.8 | APE12-dist-na | 16.0102 | APE11-dist-na | 11.8397 | APE10-dist-na | 8.4563 | APE9-dist-in | 7.993 | T315I | None | None | XRAY | 1.9 | 0.216 | 0.258 | A | 288.0 | 279.0 | 6 | 29 | 23 | 6 | [[242, 495]] | 1.0 | 3ik3 | Mus musculus | TYR_ABL1_MOUSE | TYR | 5.5e-100 | 339.9 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_MOUSE | 3IK3B | P00520 | 229 | 513 | 1123.0 | 0LI:60002 | Type2 | Inactive | DFGout | 13.4975 | 9.1697 | BBAminus | -129.46, 178.53 | -148.47, 114.27 | -91.94, -7.12 | 286.37, 101.01 | 64.82, 50.27 | in-in | in | 7.9919 | Saltbr-in | 2.6552 | HRD-in | -76.51, -54.44 | 85.69, -10.99 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.7027 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -129.88, 123.97 | APE9-dihe-in | -117.43, 141.07 | APE8-dihe-in | -76.99, 85.79 | APE8-rot-na | 29.46 | APE67-dihe-in | -85.08, -5.45 | -41.61, -41.71 | APE12-dist-na | 15.8259 | APE11-dist-na | 11.5962 | APE10-dist-na | 8.603 | APE9-dist-in | 7.8512 | T315I | None | None | XRAY | 1.9 | 0.216 | 0.258 | B | 288.0 | 285.0 | 0 | 29 | 29 | 0 | [[242, 495]] | 1.0 | 3ik3 | Mus musculus | TYR_ABL1_MOUSE | TYR | 5.5e-100 | 339.9 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_MOUSE | 3OXZA | P00520 | 229 | 511 | 1123.0 | 0LI:60001 | Type2 | Inactive | DFGout | 13.3158 | 8.9403 | BBAminus | -130.11, -171.24 | -154.37, 127.79 | -115.42, 5.71 | 286.77, 98.95 | 48.45, 62.42 | in-in | in | 8.0038 | Saltbr-in | 3.005 | HRD-in | -71.2, -52.05 | 81.82, -16.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -90.47, 133.09 | APE9-dihe-in | -119.78, 140.42 | APE8-dihe-in | -76.32, 77.74 | APE8-rot-na | 32.13 | APE67-dihe-in | -76.96, -8.32 | -43.1, -46.11 | APE12-dist-na | 15.3775 | APE11-dist-na | 10.76 | APE10-dist-na | 8.339 | APE9-dist-out | 8.088 | None | None | None | XRAY | 2.2 | 0.218 | 0.261 | A | 284.0 | 267.0 | 16 | 29 | 19 | 10 | [[242, 495]] | 1.0 | 3oxz | Mus musculus | TYR_ABL1_MOUSE | TYR | 2.6e-100 | 341.0 | 1.0 | 260.0 | 260.0 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363.0 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |