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| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1U54B | 117 | 388 | 1038.0 | ACP:400 | ATPlike | Active | DFGin | 6.615 | 13.378 | BLAminus | -120.4, -155.16 | 27.84, 85.75 | -104.36, 38.7 | 310.01, 93.15 | -67.71, -28.73 | in-in | in | 7.966 | Saltbr-in | 3.021 | HRD-in | -109.84, -42.56 | 64.6, 13.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.014 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -150.8, 133.1 | APE9-dihe-in | -126.86, 129.0 | APE8-dihe-in | -43.1, 130.27 | APE8-rot-na | 329.12 | APE67-dihe-in | -70.13, -6.6 | -62.78, -39.45 | APE12-dist-na | 12.662 | APE11-dist-na | 7.646 | APE10-dist-na | 11.0 | APE9-dist-in | 5.878 | None | None | None | XRAY | 2.8 | 0.226 | 0.322 | B | 291 | 261 | 11 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 1u54 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| AF-Q07912-K1A | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.402 | 13.809 | BLAminus | -127.81, -172.26 | 52.98, 78.87 | -92.01, 15.18 | 300.66, 98.99 | -61.2, -28.6 | in-in | in | 9.068 | Saltbr-in | 2.884 | HRD-in | -71.74, -46.77 | 66.75, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.883 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.08, 137.58 | APE9-dihe-in | -124.59, 150.42 | APE8-dihe-in | -74.79, 77.42 | APE8-rot-na | 33.67 | APE67-dihe-in | -72.2, -16.05 | -54.65, -32.93 | APE12-dist-na | 14.225 | APE11-dist-na | 8.173 | APE10-dist-na | 10.488 | APE9-dist-in | 6.215 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278 | 278 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K1 | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| AF-Q07912-K3A | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.282 | 13.816 | BLAminus | -132.02, -165.66 | 49.79, 76.66 | -89.46, 13.86 | 302.75, 106.95 | -62.78, -25.76 | in-in | in | 9.153 | Saltbr-in | 2.829 | HRD-in | -75.54, -47.15 | 65.26, -2.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.894 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.1, 134.59 | APE9-dihe-in | -125.28, 155.36 | APE8-dihe-in | -74.53, 75.69 | APE8-rot-na | 36.27 | APE67-dihe-in | -72.66, -16.99 | -53.38, -31.64 | APE12-dist-na | 13.715 | APE11-dist-na | 7.749 | APE10-dist-na | 10.02 | APE9-dist-in | 5.715 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278 | 278 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K3 | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 1U46B | 117 | 390 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.893 | 13.327 | BLAminus | -106.75, -162.4 | 39.69, 86.16 | -96.94, 26.22 | 299.15, 109.43 | -73.67, -16.41 | in-in | in | 8.181 | Saltbr-in | 2.589 | HRD-in | -73.19, -48.75 | 76.75, -0.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.921 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -148.81, 131.4 | APE9-dihe-in | -119.81, 131.46 | APE8-dihe-in | -52.5, 137.43 | APE8-rot-na | 348.53 | APE67-dihe-in | -65.13, -16.63 | -61.62, -36.89 | APE12-dist-na | 12.238 | APE11-dist-na | 7.191 | APE10-dist-na | 10.215 | APE9-dist-in | 5.643 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | B | 291 | 257 | 17 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 1u46 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 6VQMB | 117 | 392 | 1038.0 | R7P:401 | Type1 | Active | DFGin | 6.587 | 13.594 | BLAminus | -126.29, -176.9 | 60.12, 78.79 | -101.99, 43.61 | 309.18, 96.93 | -70.48, -42.01 | in-in | in | 8.354 | Saltbr-in | 2.79 | HRD-in | -70.81, -44.97 | 67.08, 13.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.034 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.03, 107.88 | APE9-dihe-in | -69.66, 138.93 | APE8-dihe-in | -77.17, 95.23 | APE8-rot-na | 27.59 | APE67-dihe-in | -70.22, -21.82 | -51.53, -42.79 | APE12-dist-na | 12.263 | APE11-dist-na | 8.421 | APE10-dist-na | 12.201 | APE9-dist-in | 7.191 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | B | 289 | 267 | 9 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 6vqm | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 1U4DB | 117 | 390 | 1038.0 | DBQ:401 | Type1 | Active | DFGin | 6.743 | 13.286 | BLAminus | -120.44, -165.36 | 55.02, 77.38 | -96.18, 18.83 | 299.22, 128.21 | -61.51, -28.63 | in-in | in | 8.506 | Saltbr-in | 3.09 | HRD-in | -78.19, -51.48 | 79.02, -2.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.79, 137.8 | APE9-dihe-in | -124.54, 129.71 | APE8-dihe-in | -55.28, 140.91 | APE8-rot-na | 333.19 | APE67-dihe-in | -67.74, -15.49 | -65.28, -34.43 | APE12-dist-na | 12.306 | APE11-dist-na | 7.19 | APE10-dist-na | 10.394 | APE9-dist-in | 5.748 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | B | 291 | 262 | 12 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 1u4d | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 1U54A | 115 | 390 | 1038.0 | ACP:101 | ATPlike | Inactive | DFGin | 6.381 | 13.426 | ABAminus | -129.39, -12.11 | -146.47, 102.96 | -102.84, 23.33 | 304.65, 105.91 | -57.05, -37.37 | in-in | in | 7.864 | Saltbr-in | 2.624 | HRD-in | -77.15, -49.8 | 83.51, -10.59 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.835 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 126.54 | APE8-dihe-in | -75.47, 123.76 | APE8-rot-na | 349.96 | APE67-dihe-in | -43.9, -19.78 | -62.08, -52.54 | APE12-dist-na | 11.808 | APE11-dist-na | 8.141 | APE10-dist-na | 999.0 | APE9-dist-in | 6.063 | None | PTR284 | PTR284 | XRAY | 2.8 | 0.226 | 0.322 | A | 291 | 263 | 13 | 0 | 0 | 1 | [[126, 387]] | 1.0 | 1u54 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4HZRA | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.941 | 13.337 | ABAminus | -116.61, 0.1 | -140.48, 143.47 | -137.83, 29.0 | 303.1, 95.78 | -63.74, -22.82 | in-in | in | 8.671 | Saltbr-in | 3.014 | HRD-in | -78.97, -45.99 | 73.0, 0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.852 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -137.45, 121.81 | APE9-dihe-in | -117.27, 126.54 | APE8-dihe-in | -48.18, 134.62 | APE8-rot-na | 331.8 | APE67-dihe-in | -67.06, -18.13 | -62.19, -35.06 | APE12-dist-na | 12.221 | APE11-dist-na | 7.476 | APE10-dist-na | 10.368 | APE9-dist-in | 5.64 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | A | 277 | 261 | 12 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4hzr | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4HZRB | 118 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.926 | 13.203 | ABAminus | -114.0, -2.21 | -142.3, 141.19 | -136.9, 28.97 | 303.67, 94.73 | -65.41, -14.9 | in-in | in | 8.32 | Saltbr-in | 2.784 | HRD-in | -81.57, -44.88 | 71.99, 1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.878 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.7, 123.01 | APE9-dihe-in | -130.03, 154.84 | APE8-dihe-in | -57.54, 124.6 | APE8-rot-na | 334.8 | APE67-dihe-in | -72.23, -12.85 | -67.01, -33.63 | APE12-dist-na | 13.405 | APE11-dist-na | 8.572 | APE10-dist-na | 12.141 | APE9-dist-in | 6.958 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | B | 277 | 258 | 14 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4hzr | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 1U46A | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.677 | 13.606 | ABAminus | -105.04, -15.76 | -135.27, 148.5 | -140.73, 24.35 | 300.72, 95.61 | -66.87, -16.87 | in-in | in | 8.88 | Saltbr-in | 3.042 | HRD-in | -74.47, -45.94 | 65.29, 8.06 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.08 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.6 | APE8-dihe-in | -40.6, 125.73 | APE8-rot-na | 326.91 | APE67-dihe-in | -63.61, -22.03 | -68.77, -33.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.487 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | A | 291 | 255 | 18 | 0 | 0 | 6 | [[126, 387]] | 1.0 | 1u46 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4EWHA | 117 | 391 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.897 | 13.758 | ABAminus | -112.33, -10.32 | -127.98, 158.61 | -163.96, 19.15 | 297.07, 109.95 | -51.93, -22.07 | in-in | in | 8.363 | Saltbr-in | 2.841 | HRD-in | -80.55, -48.4 | 69.82, -0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.784 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.82, 134.34 | APE9-dihe-in | -105.63, 146.75 | APE8-dihe-in | -58.9, 128.31 | APE8-rot-na | 332.95 | APE67-dihe-in | -67.17, -17.01 | -59.23, -34.05 | APE12-dist-na | 12.371 | APE11-dist-na | 7.33 | APE10-dist-na | 11.496 | APE9-dist-in | 5.965 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | A | 275 | 275 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4ewh | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4EWHB | 117 | 390 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.814 | 13.781 | ABAminus | -113.99, 0.05 | -132.38, 146.39 | -142.78, 20.76 | 303.22, 103.13 | -48.09, -26.49 | in-in | in | 8.335 | Saltbr-in | 2.677 | HRD-in | -88.91, -43.41 | 72.85, -2.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -105.83, 138.68 | APE9-dihe-in | -104.08, 148.64 | APE8-dihe-in | -58.72, 120.66 | APE8-rot-na | 340.66 | APE67-dihe-in | -66.41, -17.16 | -49.99, -36.4 | APE12-dist-na | 12.424 | APE11-dist-na | 7.355 | APE10-dist-na | 11.541 | APE9-dist-in | 5.922 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | B | 275 | 274 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4ewh | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 7KP6A | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.987 | 13.074 | ABAminus | -120.5, 2.81 | -142.4, 134.01 | -133.76, 28.84 | 306.02, 91.7 | -68.06, -13.37 | in-out | in | 8.711 | Saltbr-out | 4.439 | HRD-in | -78.88, -45.58 | 72.69, 3.73 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.814 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -141.02, 134.34 | APE9-dihe-in | -120.0, 134.77 | APE8-dihe-in | -57.68, 136.22 | APE8-rot-na | 336.49 | APE67-dihe-in | -65.99, -13.55 | -58.92, -37.48 | APE12-dist-na | 12.273 | APE11-dist-na | 7.282 | APE10-dist-na | 10.479 | APE9-dist-in | 5.598 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | A | 287 | 268 | 7 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 7kp6 | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 7KP6B | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.971 | 13.41 | ABAminus | -118.46, 0.28 | -140.74, 140.65 | -134.73, 29.67 | 302.28, 95.76 | -64.4, -24.8 | in-in | in | 8.466 | Saltbr-in | 2.483 | HRD-in | -80.63, -45.48 | 68.06, 5.55 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.891 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 149.74 | APE9-dihe-in | -131.88, 157.91 | APE8-dihe-in | -71.95, 81.45 | APE8-rot-na | 27.93 | APE67-dihe-in | -74.26, -9.58 | -63.95, -29.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.433 | APE9-dist-in | 6.546 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | B | 287 | 265 | 10 | 0 | 0 | 4 | [[126, 387]] | 1.0 | 7kp6 | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 6VQMA | 117 | 390 | 1038.0 | R7P:401 | Type1 | Inactive | DFGin | 6.168 | 13.464 | ABAminus | -107.72, -37.34 | -107.23, 139.71 | -135.32, 26.09 | 306.21, 97.86 | -71.9, -43.92 | in-in | in | 8.577 | Saltbr-in | 2.571 | HRD-in | -71.98, -51.6 | 65.1, 16.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.996 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.12, 107.17 | APE9-dihe-in | -75.55, 154.5 | APE8-dihe-in | -75.48, 79.2 | APE8-rot-na | 33.66 | APE67-dihe-in | -66.81, -24.97 | -59.46, -37.23 | APE12-dist-na | 13.543 | APE11-dist-na | 8.287 | APE10-dist-na | 10.844 | APE9-dist-in | 6.573 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | A | 289 | 267 | 7 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 6vqm | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 8FE9A | 117 | 390 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 7.37 | 13.018 | ABAminus | -105.28, -25.45 | -117.67, 141.58 | -139.74, 24.77 | 304.61, 88.92 | -62.34, -21.69 | in-in | in | 9.179 | Saltbr-in | 3.598 | HRD-in | -80.64, -42.58 | 70.6, 2.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.919 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.63, 116.01 | APE9-dihe-in | -111.81, 145.17 | APE8-dihe-in | -57.08, 126.3 | APE8-rot-na | 336.42 | APE67-dihe-in | -51.19, -45.24 | -69.67, -25.96 | APE12-dist-na | 13.251 | APE11-dist-na | 7.955 | APE10-dist-na | 11.971 | APE9-dist-in | 6.328 | K161Q | None | None | XRAY | 3.2 | 0.192 | 0.228 | A | 287 | 274 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8fe9 | TYR_TNK2_HUMAN | TYR | 1.7e-85 | 292.4 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4ID7A | 117 | 389 | 1038.0 | 1G0:401 | Type1.5_Back | Inactive | DFGin | 7.3 | 14.149 | ABAminus | -100.89, -41.99 | -119.98, 142.93 | -136.82, 28.94 | 304.41, 92.31 | -64.16, -28.63 | out-out | out | 10.594 | Saltbr-out | 5.173 | HRD-in | -73.52, -37.85 | 67.07, 1.92 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.78 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.45, 115.86 | APE9-dihe-in | -72.04, 137.46 | APE8-dihe-in | -82.5, 104.34 | APE8-rot-na | 27.83 | APE67-dihe-in | -58.7, -32.88 | -52.23, -52.86 | APE12-dist-na | 13.371 | APE11-dist-na | 8.528 | APE10-dist-na | 10.996 | APE9-dist-in | 6.893 | None | None | None | XRAY | 3.0 | 0.213 | 0.259 | A | 273 | 268 | 5 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4id7 | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 8HMTA | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.473 | 13.951 | ABAminus | -118.49, 19.83 | -162.39, 140.84 | -133.87, 20.8 | 306.3, 104.45 | -62.09, -37.78 | in-out | in | 9.042 | Saltbr-out | 3.701 | HRD-in | -83.9, -47.14 | 69.67, 4.35 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.198 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.87, 119.25 | APE9-dihe-in | -119.04, 129.31 | APE8-dihe-in | -48.41, 121.71 | APE8-rot-na | 329.76 | APE67-dihe-in | -54.06, -45.26 | -70.98, -26.96 | APE12-dist-na | 11.892 | APE11-dist-na | 7.024 | APE10-dist-na | 10.328 | APE9-dist-in | 6.224 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | A | 273 | 270 | 3 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 8HMTB | 117 | 388 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.529 | 13.483 | ABAminus | -91.46, -72.88 | -101.02, 153.06 | -135.07, 25.09 | 315.45, 85.41 | -54.87, -35.23 | in-in | in | 8.883 | Saltbr-in | 3.6 | HRD-in | -84.2, -43.48 | 69.63, 0.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.063 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -126.21, 93.78 | APE9-dihe-in | -110.75, 147.04 | APE8-dihe-in | -62.13, 122.57 | APE8-rot-na | 330.26 | APE67-dihe-in | -58.09, -48.9 | -67.75, -29.14 | APE12-dist-na | 12.287 | APE11-dist-na | 7.699 | APE10-dist-na | 10.144 | APE9-dist-in | 6.752 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | B | 273 | 269 | 3 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 8HMTC | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.691 | 13.313 | ABAminus | -131.24, 29.48 | -133.92, 126.7 | -139.44, 20.75 | 308.54, 95.78 | -72.46, -43.8 | in-out | in | 8.879 | Saltbr-out | 6.202 | HRD-in | -85.66, -46.96 | 68.19, 1.14 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.071 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.97, 132.16 | APE9-dihe-in | -105.55, 149.15 | APE8-dihe-in | -44.92, 133.48 | APE8-rot-na | 327.23 | APE67-dihe-in | -37.27, -59.27 | -63.72, -43.44 | APE12-dist-na | 12.373 | APE11-dist-na | 7.113 | APE10-dist-na | 10.731 | APE9-dist-in | 5.956 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | C | 273 | 262 | 11 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 3EQRA | 117 | 392 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.867 | 13.382 | ABAminus | -128.87, 39.52 | -159.68, 137.58 | -136.82, 17.85 | 302.67, 104.42 | -47.59, -35.87 | in-in | in | 8.431 | Saltbr-in | 2.693 | HRD-in | -84.2, -49.01 | 74.75, 3.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.863 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -146.69, 130.79 | APE9-dihe-in | -116.23, 133.53 | APE8-dihe-in | -52.18, 127.34 | APE8-rot-na | 331.23 | APE67-dihe-in | -63.51, -16.76 | -51.88, -37.16 | APE12-dist-na | 12.21 | APE11-dist-na | 7.171 | APE10-dist-na | 10.355 | APE9-dist-in | 5.493 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | A | 276 | 270 | 6 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 3eqr | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 3EQRB | 117 | 390 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.795 | 13.431 | ABAminus | -120.3, 36.38 | -155.51, 142.4 | -140.09, 20.29 | 304.07, 98.58 | -61.13, -29.69 | in-in | in | 8.515 | Saltbr-in | 2.733 | HRD-in | -83.74, -48.84 | 74.17, 1.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.901 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.77, 150.09 | APE9-dihe-in | -122.65, 150.11 | APE8-dihe-in | -70.86, 79.63 | APE8-rot-na | 24.49 | APE67-dihe-in | -77.33, -9.73 | -59.15, -33.0 | APE12-dist-na | 999.0 | APE11-dist-na | 9.236 | APE10-dist-na | 11.329 | APE9-dist-in | 6.67 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | B | 276 | 271 | 3 | 0 | 0 | 3 | [[126, 387]] | 1.0 | 3eqr | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 3EQPA | 117 | 390 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.713 | 14.004 | BLAminus | -122.28, -169.39 | 49.91, 85.82 | -103.52, 29.12 | 298.07, 93.89 | -65.88, -22.57 | in-in | in | 8.558 | Saltbr-in | 2.557 | HRD-in | -67.58, -47.8 | 79.03, -3.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.937 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 41.47, 68.24 | APE9-dihe-in | -80.12, 152.64 | APE8-dihe-in | -67.7, 101.83 | APE8-rot-na | 335.05 | APE67-dihe-in | -66.98, -8.09 | -37.76, -57.12 | APE12-dist-na | 12.432 | APE11-dist-na | 7.613 | APE10-dist-na | 11.69 | APE9-dist-in | 6.301 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | A | 276 | 268 | 6 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 3eqp | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 3EQPB | 117 | 392 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.747 | 13.941 | BLAminus | -134.99, 176.53 | 61.95, 90.21 | -110.2, 23.83 | 297.71, 92.68 | -58.95, -17.74 | in-in | in | 8.422 | Saltbr-in | 2.579 | HRD-in | -73.01, -48.54 | 76.03, -4.13 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.816 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 48.1, 56.77 | APE9-dihe-in | -72.7, 143.2 | APE8-dihe-in | -64.45, 112.29 | APE8-rot-na | 344.7 | APE67-dihe-in | -74.41, -9.69 | -53.7, -41.09 | APE12-dist-na | 12.373 | APE11-dist-na | 7.514 | APE10-dist-na | 11.732 | APE9-dist-in | 6.173 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | B | 276 | 270 | 6 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 3eqp | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4HZSA | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.397 | 13.731 | BLBplus | -128.49, 177.6 | 75.97, 0.07 | -64.52, 114.85 | 48.75, 95.91 | 91.75, 5.84 | out-out | out | 13.902 | Saltbr-out | 13.592 | HRD-in | -83.45, -44.79 | 72.11, -12.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.008 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.92 | APE8-dihe-in | -80.17, 58.22 | APE8-rot-na | 31.2 | APE67-dihe-in | -83.82, 0.51 | -43.12, -45.6 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.561 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | A | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4HZSB | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.402 | 13.697 | BLBplus | -127.73, 176.98 | 75.42, 0.58 | -63.8, 113.76 | 49.58, 96.39 | 93.88, 5.2 | out-out | out | 13.895 | Saltbr-out | 13.564 | HRD-in | -82.56, -44.07 | 71.76, -13.74 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.016 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.49 | APE8-dihe-in | -80.43, 57.86 | APE8-rot-na | 30.79 | APE67-dihe-in | -82.93, -0.7 | -42.53, -45.05 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.552 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | B | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4HZSC | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.42 | 13.728 | BLBplus | -131.14, 178.08 | 74.14, -0.16 | -64.4, 114.39 | 48.24, 95.76 | 92.64, 7.14 | out-out | out | 13.88 | Saltbr-out | 13.56 | HRD-in | -80.94, -46.54 | 73.93, -15.02 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.992 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.59 | APE8-dihe-in | -80.99, 59.29 | APE8-rot-na | 31.45 | APE67-dihe-in | -82.91, 0.04 | -43.57, -45.3 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.568 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | C | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 4HZSD | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.403 | 13.707 | BLBplus | -127.5, 176.15 | 76.3, -0.17 | -64.31, 115.24 | 47.66, 95.75 | 91.47, 5.35 | out-out | out | 13.876 | Saltbr-out | 13.564 | HRD-in | -81.93, -43.89 | 71.65, -14.69 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.016 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 150.39 | APE8-dihe-in | -81.82, 58.59 | APE8-rot-na | 31.39 | APE67-dihe-in | -80.9, -1.27 | -43.09, -46.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.589 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | D | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 8HMTD | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.306 | 13.333 | None | -101.89, -122.34 | -52.57, 148.88 | -124.51, 20.24 | 302.36, 99.89 | -60.05, -38.85 | in-out | in | 8.563 | Saltbr-out | 3.702 | HRD-in | -85.57, -47.32 | 68.53, 3.51 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.061 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.15, 128.97 | APE9-dihe-in | -122.52, 150.9 | APE8-dihe-in | -68.07, 94.15 | APE8-rot-na | 328.13 | APE67-dihe-in | -58.59, -46.12 | -66.12, -27.69 | APE12-dist-na | 12.502 | APE11-dist-na | 7.808 | APE10-dist-na | 10.854 | APE9-dist-in | 5.856 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | D | 273 | 262 | 11 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 5ZXBA | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.852 | 11.264 | None | -126.71, -163.29 | -159.07, 87.59 | -102.57, 999.0 | 328.97, 133.0 | 999.0, 999.0 | in-in | in | 8.666 | Saltbr-in | 2.564 | HRD-in | -73.25, -51.97 | 78.84, -2.72 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.29 | APE8-rot-na | 28.55 | APE67-dihe-in | -73.12, -10.47 | -54.59, -43.66 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | A | 275 | 240 | 33 | 0 | 0 | 21 | [[126, 387]] | 1.0 | 5zxb | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 5ZXBB | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.904 | 10.951 | None | -127.77, -163.1 | -162.7, 90.46 | -101.67, 999.0 | 328.28, 133.86 | 999.0, 999.0 | in-in | in | 8.729 | Saltbr-in | 2.716 | HRD-in | -72.25, -50.4 | 79.44, -3.02 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.74 | APE8-rot-na | 29.71 | APE67-dihe-in | -76.43, -11.56 | -55.87, -46.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | B | 275 | 241 | 32 | 0 | 0 | 21 | [[126, 387]] | 1.0 | 5zxb | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| 1U4DA | 117 | 389 | 1038.0 | DBQ:398 | Type1 | None | DFGin | 6.5 | 13.536 | BLAminus | -127.17, -169.67 | 54.12, 72.77 | -87.16, 24.56 | 310.51, 109.17 | -62.52, -20.25 | in-in | in | 8.735 | Saltbr-in | 3.176 | HRD-in | -80.08, -48.95 | 65.72, 7.9 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.172 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -41.24 | APE8-dihe-in | -76.48, 82.61 | APE8-rot-na | 31.13 | APE67-dihe-in | -69.93, -17.0 | -48.99, -48.23 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.562 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | A | 291 | 258 | 15 | 0 | 0 | 7 | [[126, 387]] | 1.0 | 1u4d | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| ACK1_HUMAN | 1U54B | Q07912 | 117 | 388 | 1038.0 | ACP:400 | ATPlike | Active | DFGin | 6.615 | 13.378 | BLAminus | -120.4, -155.16 | 27.84, 85.75 | -104.36, 38.7 | 310.01, 93.15 | -67.71, -28.73 | in-in | in | 7.966 | Saltbr-in | 3.021 | HRD-in | -109.84, -42.56 | 64.6, 13.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.014 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -150.8, 133.1 | APE9-dihe-in | -126.86, 129.0 | APE8-dihe-in | -43.1, 130.27 | APE8-rot-na | 329.12 | APE67-dihe-in | -70.13, -6.6 | -62.78, -39.45 | APE12-dist-na | 12.662 | APE11-dist-na | 7.646 | APE10-dist-na | 11.0 | APE9-dist-in | 5.878 | None | None | None | XRAY | 2.8 | 0.226 | 0.322 | B | 291 | 261 | 11 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 1u54 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | AF-Q07912-K1A | Q07912 | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.402 | 13.809 | BLAminus | -127.81, -172.26 | 52.98, 78.87 | -92.01, 15.18 | 300.66, 98.99 | -61.2, -28.6 | in-in | in | 9.068 | Saltbr-in | 2.884 | HRD-in | -71.74, -46.77 | 66.75, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.883 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.08, 137.58 | APE9-dihe-in | -124.59, 150.42 | APE8-dihe-in | -74.79, 77.42 | APE8-rot-na | 33.67 | APE67-dihe-in | -72.2, -16.05 | -54.65, -32.93 | APE12-dist-na | 14.225 | APE11-dist-na | 8.173 | APE10-dist-na | 10.488 | APE9-dist-in | 6.215 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278 | 278 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K1 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | AF-Q07912-K3A | Q07912 | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.282 | 13.816 | BLAminus | -132.02, -165.66 | 49.79, 76.66 | -89.46, 13.86 | 302.75, 106.95 | -62.78, -25.76 | in-in | in | 9.153 | Saltbr-in | 2.829 | HRD-in | -75.54, -47.15 | 65.26, -2.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.894 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.1, 134.59 | APE9-dihe-in | -125.28, 155.36 | APE8-dihe-in | -74.53, 75.69 | APE8-rot-na | 36.27 | APE67-dihe-in | -72.66, -16.99 | -53.38, -31.64 | APE12-dist-na | 13.715 | APE11-dist-na | 7.749 | APE10-dist-na | 10.02 | APE9-dist-in | 5.715 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278 | 278 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K3 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 1U46B | Q07912 | 117 | 390 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.893 | 13.327 | BLAminus | -106.75, -162.4 | 39.69, 86.16 | -96.94, 26.22 | 299.15, 109.43 | -73.67, -16.41 | in-in | in | 8.181 | Saltbr-in | 2.589 | HRD-in | -73.19, -48.75 | 76.75, -0.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.921 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -148.81, 131.4 | APE9-dihe-in | -119.81, 131.46 | APE8-dihe-in | -52.5, 137.43 | APE8-rot-na | 348.53 | APE67-dihe-in | -65.13, -16.63 | -61.62, -36.89 | APE12-dist-na | 12.238 | APE11-dist-na | 7.191 | APE10-dist-na | 10.215 | APE9-dist-in | 5.643 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | B | 291 | 257 | 17 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 1u46 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 6VQMB | Q07912 | 117 | 392 | 1038.0 | R7P:401 | Type1 | Active | DFGin | 6.587 | 13.594 | BLAminus | -126.29, -176.9 | 60.12, 78.79 | -101.99, 43.61 | 309.18, 96.93 | -70.48, -42.01 | in-in | in | 8.354 | Saltbr-in | 2.79 | HRD-in | -70.81, -44.97 | 67.08, 13.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.034 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.03, 107.88 | APE9-dihe-in | -69.66, 138.93 | APE8-dihe-in | -77.17, 95.23 | APE8-rot-na | 27.59 | APE67-dihe-in | -70.22, -21.82 | -51.53, -42.79 | APE12-dist-na | 12.263 | APE11-dist-na | 8.421 | APE10-dist-na | 12.201 | APE9-dist-in | 7.191 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | B | 289 | 267 | 9 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 6vqm | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 1U4DB | Q07912 | 117 | 390 | 1038.0 | DBQ:401 | Type1 | Active | DFGin | 6.743 | 13.286 | BLAminus | -120.44, -165.36 | 55.02, 77.38 | -96.18, 18.83 | 299.22, 128.21 | -61.51, -28.63 | in-in | in | 8.506 | Saltbr-in | 3.09 | HRD-in | -78.19, -51.48 | 79.02, -2.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.79, 137.8 | APE9-dihe-in | -124.54, 129.71 | APE8-dihe-in | -55.28, 140.91 | APE8-rot-na | 333.19 | APE67-dihe-in | -67.74, -15.49 | -65.28, -34.43 | APE12-dist-na | 12.306 | APE11-dist-na | 7.19 | APE10-dist-na | 10.394 | APE9-dist-in | 5.748 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | B | 291 | 262 | 12 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 1u4d | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 1U54A | Q07912 | 115 | 390 | 1038.0 | ACP:101 | ATPlike | Inactive | DFGin | 6.381 | 13.426 | ABAminus | -129.39, -12.11 | -146.47, 102.96 | -102.84, 23.33 | 304.65, 105.91 | -57.05, -37.37 | in-in | in | 7.864 | Saltbr-in | 2.624 | HRD-in | -77.15, -49.8 | 83.51, -10.59 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.835 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 126.54 | APE8-dihe-in | -75.47, 123.76 | APE8-rot-na | 349.96 | APE67-dihe-in | -43.9, -19.78 | -62.08, -52.54 | APE12-dist-na | 11.808 | APE11-dist-na | 8.141 | APE10-dist-na | 999.0 | APE9-dist-in | 6.063 | None | PTR284 | PTR284 | XRAY | 2.8 | 0.226 | 0.322 | A | 291 | 263 | 13 | 0 | 0 | 1 | [[126, 387]] | 1.0 | 1u54 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4HZRA | Q07912 | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.941 | 13.337 | ABAminus | -116.61, 0.1 | -140.48, 143.47 | -137.83, 29.0 | 303.1, 95.78 | -63.74, -22.82 | in-in | in | 8.671 | Saltbr-in | 3.014 | HRD-in | -78.97, -45.99 | 73.0, 0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.852 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -137.45, 121.81 | APE9-dihe-in | -117.27, 126.54 | APE8-dihe-in | -48.18, 134.62 | APE8-rot-na | 331.8 | APE67-dihe-in | -67.06, -18.13 | -62.19, -35.06 | APE12-dist-na | 12.221 | APE11-dist-na | 7.476 | APE10-dist-na | 10.368 | APE9-dist-in | 5.64 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | A | 277 | 261 | 12 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4hzr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4HZRB | Q07912 | 118 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.926 | 13.203 | ABAminus | -114.0, -2.21 | -142.3, 141.19 | -136.9, 28.97 | 303.67, 94.73 | -65.41, -14.9 | in-in | in | 8.32 | Saltbr-in | 2.784 | HRD-in | -81.57, -44.88 | 71.99, 1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.878 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.7, 123.01 | APE9-dihe-in | -130.03, 154.84 | APE8-dihe-in | -57.54, 124.6 | APE8-rot-na | 334.8 | APE67-dihe-in | -72.23, -12.85 | -67.01, -33.63 | APE12-dist-na | 13.405 | APE11-dist-na | 8.572 | APE10-dist-na | 12.141 | APE9-dist-in | 6.958 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | B | 277 | 258 | 14 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4hzr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 1U46A | Q07912 | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.677 | 13.606 | ABAminus | -105.04, -15.76 | -135.27, 148.5 | -140.73, 24.35 | 300.72, 95.61 | -66.87, -16.87 | in-in | in | 8.88 | Saltbr-in | 3.042 | HRD-in | -74.47, -45.94 | 65.29, 8.06 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.08 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.6 | APE8-dihe-in | -40.6, 125.73 | APE8-rot-na | 326.91 | APE67-dihe-in | -63.61, -22.03 | -68.77, -33.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.487 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | A | 291 | 255 | 18 | 0 | 0 | 6 | [[126, 387]] | 1.0 | 1u46 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4EWHA | Q07912 | 117 | 391 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.897 | 13.758 | ABAminus | -112.33, -10.32 | -127.98, 158.61 | -163.96, 19.15 | 297.07, 109.95 | -51.93, -22.07 | in-in | in | 8.363 | Saltbr-in | 2.841 | HRD-in | -80.55, -48.4 | 69.82, -0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.784 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.82, 134.34 | APE9-dihe-in | -105.63, 146.75 | APE8-dihe-in | -58.9, 128.31 | APE8-rot-na | 332.95 | APE67-dihe-in | -67.17, -17.01 | -59.23, -34.05 | APE12-dist-na | 12.371 | APE11-dist-na | 7.33 | APE10-dist-na | 11.496 | APE9-dist-in | 5.965 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | A | 275 | 275 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4ewh | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4EWHB | Q07912 | 117 | 390 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.814 | 13.781 | ABAminus | -113.99, 0.05 | -132.38, 146.39 | -142.78, 20.76 | 303.22, 103.13 | -48.09, -26.49 | in-in | in | 8.335 | Saltbr-in | 2.677 | HRD-in | -88.91, -43.41 | 72.85, -2.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -105.83, 138.68 | APE9-dihe-in | -104.08, 148.64 | APE8-dihe-in | -58.72, 120.66 | APE8-rot-na | 340.66 | APE67-dihe-in | -66.41, -17.16 | -49.99, -36.4 | APE12-dist-na | 12.424 | APE11-dist-na | 7.355 | APE10-dist-na | 11.541 | APE9-dist-in | 5.922 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | B | 275 | 274 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4ewh | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 7KP6A | Q07912 | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.987 | 13.074 | ABAminus | -120.5, 2.81 | -142.4, 134.01 | -133.76, 28.84 | 306.02, 91.7 | -68.06, -13.37 | in-out | in | 8.711 | Saltbr-out | 4.439 | HRD-in | -78.88, -45.58 | 72.69, 3.73 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.814 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -141.02, 134.34 | APE9-dihe-in | -120.0, 134.77 | APE8-dihe-in | -57.68, 136.22 | APE8-rot-na | 336.49 | APE67-dihe-in | -65.99, -13.55 | -58.92, -37.48 | APE12-dist-na | 12.273 | APE11-dist-na | 7.282 | APE10-dist-na | 10.479 | APE9-dist-in | 5.598 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | A | 287 | 268 | 7 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 7kp6 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 7KP6B | Q07912 | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.971 | 13.41 | ABAminus | -118.46, 0.28 | -140.74, 140.65 | -134.73, 29.67 | 302.28, 95.76 | -64.4, -24.8 | in-in | in | 8.466 | Saltbr-in | 2.483 | HRD-in | -80.63, -45.48 | 68.06, 5.55 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.891 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 149.74 | APE9-dihe-in | -131.88, 157.91 | APE8-dihe-in | -71.95, 81.45 | APE8-rot-na | 27.93 | APE67-dihe-in | -74.26, -9.58 | -63.95, -29.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.433 | APE9-dist-in | 6.546 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | B | 287 | 265 | 10 | 0 | 0 | 4 | [[126, 387]] | 1.0 | 7kp6 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 6VQMA | Q07912 | 117 | 390 | 1038.0 | R7P:401 | Type1 | Inactive | DFGin | 6.168 | 13.464 | ABAminus | -107.72, -37.34 | -107.23, 139.71 | -135.32, 26.09 | 306.21, 97.86 | -71.9, -43.92 | in-in | in | 8.577 | Saltbr-in | 2.571 | HRD-in | -71.98, -51.6 | 65.1, 16.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.996 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.12, 107.17 | APE9-dihe-in | -75.55, 154.5 | APE8-dihe-in | -75.48, 79.2 | APE8-rot-na | 33.66 | APE67-dihe-in | -66.81, -24.97 | -59.46, -37.23 | APE12-dist-na | 13.543 | APE11-dist-na | 8.287 | APE10-dist-na | 10.844 | APE9-dist-in | 6.573 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | A | 289 | 267 | 7 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 6vqm | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 8FE9A | Q07912 | 117 | 390 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 7.37 | 13.018 | ABAminus | -105.28, -25.45 | -117.67, 141.58 | -139.74, 24.77 | 304.61, 88.92 | -62.34, -21.69 | in-in | in | 9.179 | Saltbr-in | 3.598 | HRD-in | -80.64, -42.58 | 70.6, 2.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.919 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.63, 116.01 | APE9-dihe-in | -111.81, 145.17 | APE8-dihe-in | -57.08, 126.3 | APE8-rot-na | 336.42 | APE67-dihe-in | -51.19, -45.24 | -69.67, -25.96 | APE12-dist-na | 13.251 | APE11-dist-na | 7.955 | APE10-dist-na | 11.971 | APE9-dist-in | 6.328 | K161Q | None | None | XRAY | 3.2 | 0.192 | 0.228 | A | 287 | 274 | 0 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8fe9 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.7e-85 | 292.4 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4ID7A | Q07912 | 117 | 389 | 1038.0 | 1G0:401 | Type1.5_Back | Inactive | DFGin | 7.3 | 14.149 | ABAminus | -100.89, -41.99 | -119.98, 142.93 | -136.82, 28.94 | 304.41, 92.31 | -64.16, -28.63 | out-out | out | 10.594 | Saltbr-out | 5.173 | HRD-in | -73.52, -37.85 | 67.07, 1.92 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.78 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.45, 115.86 | APE9-dihe-in | -72.04, 137.46 | APE8-dihe-in | -82.5, 104.34 | APE8-rot-na | 27.83 | APE67-dihe-in | -58.7, -32.88 | -52.23, -52.86 | APE12-dist-na | 13.371 | APE11-dist-na | 8.528 | APE10-dist-na | 10.996 | APE9-dist-in | 6.893 | None | None | None | XRAY | 3.0 | 0.213 | 0.259 | A | 273 | 268 | 5 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 4id7 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 8HMTA | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.473 | 13.951 | ABAminus | -118.49, 19.83 | -162.39, 140.84 | -133.87, 20.8 | 306.3, 104.45 | -62.09, -37.78 | in-out | in | 9.042 | Saltbr-out | 3.701 | HRD-in | -83.9, -47.14 | 69.67, 4.35 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.198 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.87, 119.25 | APE9-dihe-in | -119.04, 129.31 | APE8-dihe-in | -48.41, 121.71 | APE8-rot-na | 329.76 | APE67-dihe-in | -54.06, -45.26 | -70.98, -26.96 | APE12-dist-na | 11.892 | APE11-dist-na | 7.024 | APE10-dist-na | 10.328 | APE9-dist-in | 6.224 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | A | 273 | 270 | 3 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 8HMTB | Q07912 | 117 | 388 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.529 | 13.483 | ABAminus | -91.46, -72.88 | -101.02, 153.06 | -135.07, 25.09 | 315.45, 85.41 | -54.87, -35.23 | in-in | in | 8.883 | Saltbr-in | 3.6 | HRD-in | -84.2, -43.48 | 69.63, 0.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.063 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -126.21, 93.78 | APE9-dihe-in | -110.75, 147.04 | APE8-dihe-in | -62.13, 122.57 | APE8-rot-na | 330.26 | APE67-dihe-in | -58.09, -48.9 | -67.75, -29.14 | APE12-dist-na | 12.287 | APE11-dist-na | 7.699 | APE10-dist-na | 10.144 | APE9-dist-in | 6.752 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | B | 273 | 269 | 3 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 8HMTC | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.691 | 13.313 | ABAminus | -131.24, 29.48 | -133.92, 126.7 | -139.44, 20.75 | 308.54, 95.78 | -72.46, -43.8 | in-out | in | 8.879 | Saltbr-out | 6.202 | HRD-in | -85.66, -46.96 | 68.19, 1.14 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.071 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.97, 132.16 | APE9-dihe-in | -105.55, 149.15 | APE8-dihe-in | -44.92, 133.48 | APE8-rot-na | 327.23 | APE67-dihe-in | -37.27, -59.27 | -63.72, -43.44 | APE12-dist-na | 12.373 | APE11-dist-na | 7.113 | APE10-dist-na | 10.731 | APE9-dist-in | 5.956 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | C | 273 | 262 | 11 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 3EQRA | Q07912 | 117 | 392 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.867 | 13.382 | ABAminus | -128.87, 39.52 | -159.68, 137.58 | -136.82, 17.85 | 302.67, 104.42 | -47.59, -35.87 | in-in | in | 8.431 | Saltbr-in | 2.693 | HRD-in | -84.2, -49.01 | 74.75, 3.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.863 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -146.69, 130.79 | APE9-dihe-in | -116.23, 133.53 | APE8-dihe-in | -52.18, 127.34 | APE8-rot-na | 331.23 | APE67-dihe-in | -63.51, -16.76 | -51.88, -37.16 | APE12-dist-na | 12.21 | APE11-dist-na | 7.171 | APE10-dist-na | 10.355 | APE9-dist-in | 5.493 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | A | 276 | 270 | 6 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 3eqr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 3EQRB | Q07912 | 117 | 390 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.795 | 13.431 | ABAminus | -120.3, 36.38 | -155.51, 142.4 | -140.09, 20.29 | 304.07, 98.58 | -61.13, -29.69 | in-in | in | 8.515 | Saltbr-in | 2.733 | HRD-in | -83.74, -48.84 | 74.17, 1.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.901 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.77, 150.09 | APE9-dihe-in | -122.65, 150.11 | APE8-dihe-in | -70.86, 79.63 | APE8-rot-na | 24.49 | APE67-dihe-in | -77.33, -9.73 | -59.15, -33.0 | APE12-dist-na | 999.0 | APE11-dist-na | 9.236 | APE10-dist-na | 11.329 | APE9-dist-in | 6.67 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | B | 276 | 271 | 3 | 0 | 0 | 3 | [[126, 387]] | 1.0 | 3eqr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 3EQPA | Q07912 | 117 | 390 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.713 | 14.004 | BLAminus | -122.28, -169.39 | 49.91, 85.82 | -103.52, 29.12 | 298.07, 93.89 | -65.88, -22.57 | in-in | in | 8.558 | Saltbr-in | 2.557 | HRD-in | -67.58, -47.8 | 79.03, -3.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.937 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 41.47, 68.24 | APE9-dihe-in | -80.12, 152.64 | APE8-dihe-in | -67.7, 101.83 | APE8-rot-na | 335.05 | APE67-dihe-in | -66.98, -8.09 | -37.76, -57.12 | APE12-dist-na | 12.432 | APE11-dist-na | 7.613 | APE10-dist-na | 11.69 | APE9-dist-in | 6.301 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | A | 276 | 268 | 6 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 3eqp | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 3EQPB | Q07912 | 117 | 392 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.747 | 13.941 | BLAminus | -134.99, 176.53 | 61.95, 90.21 | -110.2, 23.83 | 297.71, 92.68 | -58.95, -17.74 | in-in | in | 8.422 | Saltbr-in | 2.579 | HRD-in | -73.01, -48.54 | 76.03, -4.13 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.816 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 48.1, 56.77 | APE9-dihe-in | -72.7, 143.2 | APE8-dihe-in | -64.45, 112.29 | APE8-rot-na | 344.7 | APE67-dihe-in | -74.41, -9.69 | -53.7, -41.09 | APE12-dist-na | 12.373 | APE11-dist-na | 7.514 | APE10-dist-na | 11.732 | APE9-dist-in | 6.173 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | B | 276 | 270 | 6 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 3eqp | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4HZSA | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.397 | 13.731 | BLBplus | -128.49, 177.6 | 75.97, 0.07 | -64.52, 114.85 | 48.75, 95.91 | 91.75, 5.84 | out-out | out | 13.902 | Saltbr-out | 13.592 | HRD-in | -83.45, -44.79 | 72.11, -12.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.008 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.92 | APE8-dihe-in | -80.17, 58.22 | APE8-rot-na | 31.2 | APE67-dihe-in | -83.82, 0.51 | -43.12, -45.6 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.561 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | A | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4HZSB | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.402 | 13.697 | BLBplus | -127.73, 176.98 | 75.42, 0.58 | -63.8, 113.76 | 49.58, 96.39 | 93.88, 5.2 | out-out | out | 13.895 | Saltbr-out | 13.564 | HRD-in | -82.56, -44.07 | 71.76, -13.74 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.016 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.49 | APE8-dihe-in | -80.43, 57.86 | APE8-rot-na | 30.79 | APE67-dihe-in | -82.93, -0.7 | -42.53, -45.05 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.552 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | B | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4HZSC | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.42 | 13.728 | BLBplus | -131.14, 178.08 | 74.14, -0.16 | -64.4, 114.39 | 48.24, 95.76 | 92.64, 7.14 | out-out | out | 13.88 | Saltbr-out | 13.56 | HRD-in | -80.94, -46.54 | 73.93, -15.02 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.992 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.59 | APE8-dihe-in | -80.99, 59.29 | APE8-rot-na | 31.45 | APE67-dihe-in | -82.91, 0.04 | -43.57, -45.3 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.568 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | C | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 4HZSD | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.403 | 13.707 | BLBplus | -127.5, 176.15 | 76.3, -0.17 | -64.31, 115.24 | 47.66, 95.75 | 91.47, 5.35 | out-out | out | 13.876 | Saltbr-out | 13.564 | HRD-in | -81.93, -43.89 | 71.65, -14.69 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.016 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 150.39 | APE8-dihe-in | -81.82, 58.59 | APE8-rot-na | 31.39 | APE67-dihe-in | -80.9, -1.27 | -43.09, -46.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.589 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | D | 341 | 319 | 13 | 0 | 0 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 8HMTD | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.306 | 13.333 | None | -101.89, -122.34 | -52.57, 148.88 | -124.51, 20.24 | 302.36, 99.89 | -60.05, -38.85 | in-out | in | 8.563 | Saltbr-out | 3.702 | HRD-in | -85.57, -47.32 | 68.53, 3.51 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.061 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.15, 128.97 | APE9-dihe-in | -122.52, 150.9 | APE8-dihe-in | -68.07, 94.15 | APE8-rot-na | 328.13 | APE67-dihe-in | -58.59, -46.12 | -66.12, -27.69 | APE12-dist-na | 12.502 | APE11-dist-na | 7.808 | APE10-dist-na | 10.854 | APE9-dist-in | 5.856 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | D | 273 | 262 | 11 | 0 | 0 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 5ZXBA | Q07912 | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.852 | 11.264 | None | -126.71, -163.29 | -159.07, 87.59 | -102.57, 999.0 | 328.97, 133.0 | 999.0, 999.0 | in-in | in | 8.666 | Saltbr-in | 2.564 | HRD-in | -73.25, -51.97 | 78.84, -2.72 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.29 | APE8-rot-na | 28.55 | APE67-dihe-in | -73.12, -10.47 | -54.59, -43.66 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | A | 275 | 240 | 33 | 0 | 0 | 21 | [[126, 387]] | 1.0 | 5zxb | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 5ZXBB | Q07912 | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.904 | 10.951 | None | -127.77, -163.1 | -162.7, 90.46 | -101.67, 999.0 | 328.28, 133.86 | 999.0, 999.0 | in-in | in | 8.729 | Saltbr-in | 2.716 | HRD-in | -72.25, -50.4 | 79.44, -3.02 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.74 | APE8-rot-na | 29.71 | APE67-dihe-in | -76.43, -11.56 | -55.87, -46.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | B | 275 | 241 | 32 | 0 | 0 | 21 | [[126, 387]] | 1.0 | 5zxb | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| ACK1_HUMAN | 1U4DA | Q07912 | 117 | 389 | 1038.0 | DBQ:398 | Type1 | None | DFGin | 6.5 | 13.536 | BLAminus | -127.17, -169.67 | 54.12, 72.77 | -87.16, 24.56 | 310.51, 109.17 | -62.52, -20.25 | in-in | in | 8.735 | Saltbr-in | 3.176 | HRD-in | -80.08, -48.95 | 65.72, 7.9 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.172 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -41.24 | APE8-dihe-in | -76.48, 82.61 | APE8-rot-na | 31.13 | APE67-dihe-in | -69.93, -17.0 | -48.99, -48.23 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.562 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | A | 291 | 258 | 15 | 0 | 0 | 7 | [[126, 387]] | 1.0 | 1u4d | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1 | 259 | 259 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|