| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TNK2 | 1U54B | Q07912 | 117 | 388 | 1038.0 | ACP:400 | ATPlike | Active | DFGin | 6.6155 | 13.3776 | BLAminus | -120.4, -155.16 | 27.84, 85.75 | -104.36, 38.7 | 310.01, 93.15 | -67.71, -28.73 | in-in | in | 7.966 | Saltbr-in | 3.0206 | HRD-in | -109.84, -42.56 | 64.6, 13.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0144 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -150.8, 133.1 | APE9-dihe-in | -126.86, 129.0 | APE8-dihe-in | -43.1, 130.27 | APE8-rot-na | 329.12 | APE67-dihe-in | -70.13, -6.6 | -62.78, -39.45 | APE12-dist-na | 12.6617 | APE11-dist-na | 7.6459 | APE10-dist-na | 10.9998 | APE9-dist-in | 5.8775 | None | None | None | XRAY | 2.8 | 0.226 | 0.322 | B | 291.0 | 261.0 | 11 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 1u54 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | AF-Q07912-K1A | Q07912 | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.4024 | 13.8085 | BLAminus | -127.81, -172.26 | 52.98, 78.87 | -92.01, 15.18 | 300.66, 98.99 | -61.2, -28.6 | in-in | in | 9.0677 | Saltbr-in | 2.8838 | HRD-in | -71.74, -46.77 | 66.75, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8834 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.08, 137.58 | APE9-dihe-in | -124.59, 150.42 | APE8-dihe-in | -74.79, 77.42 | APE8-rot-na | 33.67 | APE67-dihe-in | -72.2, -16.05 | -54.65, -32.93 | APE12-dist-na | 14.2254 | APE11-dist-na | 8.1727 | APE10-dist-na | 10.4882 | APE9-dist-in | 6.2148 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278.0 | 278.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K1 | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | AF-Q07912-K3A | Q07912 | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.2816 | 13.8163 | BLAminus | -132.02, -165.66 | 49.79, 76.66 | -89.46, 13.86 | 302.75, 106.95 | -62.78, -25.76 | in-in | in | 9.1531 | Saltbr-in | 2.8291 | HRD-in | -75.54, -47.15 | 65.26, -2.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8945 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.1, 134.59 | APE9-dihe-in | -125.28, 155.36 | APE8-dihe-in | -74.53, 75.69 | APE8-rot-na | 36.27 | APE67-dihe-in | -72.66, -16.99 | -53.38, -31.64 | APE12-dist-na | 13.715 | APE11-dist-na | 7.7486 | APE10-dist-na | 10.0198 | APE9-dist-in | 5.7149 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278.0 | 278.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K3 | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 1U46B | Q07912 | 117 | 390 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.8929 | 13.3269 | BLAminus | -106.75, -162.4 | 39.69, 86.16 | -96.94, 26.22 | 299.15, 109.43 | -73.67, -16.41 | in-in | in | 8.1814 | Saltbr-in | 2.5893 | HRD-in | -73.19, -48.75 | 76.75, -0.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9211 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -148.81, 131.4 | APE9-dihe-in | -119.81, 131.46 | APE8-dihe-in | -52.5, 137.43 | APE8-rot-na | 348.53 | APE67-dihe-in | -65.13, -16.63 | -61.62, -36.89 | APE12-dist-na | 12.2376 | APE11-dist-na | 7.1908 | APE10-dist-na | 10.2147 | APE9-dist-in | 5.6432 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | B | 291.0 | 257.0 | 17 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 1u46 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 6VQMB | Q07912 | 117 | 392 | 1038.0 | R7P:401 | Type1 | Active | DFGin | 6.5869 | 13.5939 | BLAminus | -126.29, -176.9 | 60.12, 78.79 | -101.99, 43.61 | 309.18, 96.93 | -70.48, -42.01 | in-in | in | 8.3539 | Saltbr-in | 2.7897 | HRD-in | -70.81, -44.97 | 67.08, 13.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0338 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.03, 107.88 | APE9-dihe-in | -69.66, 138.93 | APE8-dihe-in | -77.17, 95.23 | APE8-rot-na | 27.59 | APE67-dihe-in | -70.22, -21.82 | -51.53, -42.79 | APE12-dist-na | 12.2631 | APE11-dist-na | 8.4205 | APE10-dist-na | 12.2009 | APE9-dist-in | 7.1911 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | B | 289.0 | 267.0 | 9 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 6vqm | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 1U4DB | Q07912 | 117 | 390 | 1038.0 | DBQ:401 | Type1 | Active | DFGin | 6.7434 | 13.2857 | BLAminus | -120.44, -165.36 | 55.02, 77.38 | -96.18, 18.83 | 299.22, 128.21 | -61.51, -28.63 | in-in | in | 8.506 | Saltbr-in | 3.09 | HRD-in | -78.19, -51.48 | 79.02, -2.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.79, 137.8 | APE9-dihe-in | -124.54, 129.71 | APE8-dihe-in | -55.28, 140.91 | APE8-rot-na | 333.19 | APE67-dihe-in | -67.74, -15.49 | -65.28, -34.43 | APE12-dist-na | 12.3065 | APE11-dist-na | 7.1903 | APE10-dist-na | 10.3941 | APE9-dist-in | 5.7477 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | B | 291.0 | 262.0 | 12 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 1u4d | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 1U54A | Q07912 | 115 | 390 | 1038.0 | ACP:101 | ATPlike | Inactive | DFGin | 6.3812 | 13.4263 | ABAminus | -129.39, -12.11 | -146.47, 102.96 | -102.84, 23.33 | 304.65, 105.91 | -57.05, -37.37 | in-in | in | 7.8643 | Saltbr-in | 2.6244 | HRD-in | -77.15, -49.8 | 83.51, -10.59 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8347 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 126.54 | APE8-dihe-in | -75.47, 123.76 | APE8-rot-na | 349.96 | APE67-dihe-in | -43.9, -19.78 | -62.08, -52.54 | APE12-dist-na | 11.8082 | APE11-dist-na | 8.1412 | APE10-dist-na | 999.0 | APE9-dist-in | 6.0632 | None | PTR284 | PTR284 | XRAY | 2.8 | 0.226 | 0.322 | A | 291.0 | 263.0 | 13 | 31 | 30 | 1 | [[126, 387]] | 1.0 | 1u54 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4HZRA | Q07912 | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9405 | 13.3374 | ABAminus | -116.61, 0.1 | -140.48, 143.47 | -137.83, 29.0 | 303.1, 95.78 | -63.74, -22.82 | in-in | in | 8.6705 | Saltbr-in | 3.0135 | HRD-in | -78.97, -45.99 | 73.0, 0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8523 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -137.45, 121.81 | APE9-dihe-in | -117.27, 126.54 | APE8-dihe-in | -48.18, 134.62 | APE8-rot-na | 331.8 | APE67-dihe-in | -67.06, -18.13 | -62.19, -35.06 | APE12-dist-na | 12.2207 | APE11-dist-na | 7.4764 | APE10-dist-na | 10.3681 | APE9-dist-in | 5.6397 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | A | 277.0 | 261.0 | 12 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4hzr | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4HZRB | Q07912 | 118 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9261 | 13.2029 | ABAminus | -114.0, -2.21 | -142.3, 141.19 | -136.9, 28.97 | 303.67, 94.73 | -65.41, -14.9 | in-in | in | 8.3198 | Saltbr-in | 2.7836 | HRD-in | -81.57, -44.88 | 71.99, 1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8785 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.7, 123.01 | APE9-dihe-in | -130.03, 154.84 | APE8-dihe-in | -57.54, 124.6 | APE8-rot-na | 334.8 | APE67-dihe-in | -72.23, -12.85 | -67.01, -33.63 | APE12-dist-na | 13.4048 | APE11-dist-na | 8.5721 | APE10-dist-na | 12.141 | APE9-dist-in | 6.9585 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | B | 277.0 | 258.0 | 14 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4hzr | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 1U46A | Q07912 | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.6774 | 13.6062 | ABAminus | -105.04, -15.76 | -135.27, 148.5 | -140.73, 24.35 | 300.72, 95.61 | -66.87, -16.87 | in-in | in | 8.88 | Saltbr-in | 3.0421 | HRD-in | -74.47, -45.94 | 65.29, 8.06 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.0797 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.6 | APE8-dihe-in | -40.6, 125.73 | APE8-rot-na | 326.91 | APE67-dihe-in | -63.61, -22.03 | -68.77, -33.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.4874 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | A | 291.0 | 255.0 | 18 | 31 | 25 | 6 | [[126, 387]] | 1.0 | 1u46 | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4EWHA | Q07912 | 117 | 391 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.8969 | 13.7575 | ABAminus | -112.33, -10.32 | -127.98, 158.61 | -163.96, 19.15 | 297.07, 109.95 | -51.93, -22.07 | in-in | in | 8.3631 | Saltbr-in | 2.8413 | HRD-in | -80.55, -48.4 | 69.82, -0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7842 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.82, 134.34 | APE9-dihe-in | -105.63, 146.75 | APE8-dihe-in | -58.9, 128.31 | APE8-rot-na | 332.95 | APE67-dihe-in | -67.17, -17.01 | -59.23, -34.05 | APE12-dist-na | 12.3707 | APE11-dist-na | 7.3299 | APE10-dist-na | 11.496 | APE9-dist-in | 5.9649 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | A | 275.0 | 275.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4ewh | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4EWHB | Q07912 | 117 | 390 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.8136 | 13.7809 | ABAminus | -113.99, 0.05 | -132.38, 146.39 | -142.78, 20.76 | 303.22, 103.13 | -48.09, -26.49 | in-in | in | 8.3351 | Saltbr-in | 2.6774 | HRD-in | -88.91, -43.41 | 72.85, -2.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -105.83, 138.68 | APE9-dihe-in | -104.08, 148.64 | APE8-dihe-in | -58.72, 120.66 | APE8-rot-na | 340.66 | APE67-dihe-in | -66.41, -17.16 | -49.99, -36.4 | APE12-dist-na | 12.4243 | APE11-dist-na | 7.3547 | APE10-dist-na | 11.5408 | APE9-dist-in | 5.9219 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | B | 275.0 | 274.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4ewh | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 7KP6A | Q07912 | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.9868 | 13.0736 | ABAminus | -120.5, 2.81 | -142.4, 134.01 | -133.76, 28.84 | 306.02, 91.7 | -68.06, -13.37 | in-out | in | 8.7113 | Saltbr-out | 4.4386 | HRD-in | -78.88, -45.58 | 72.69, 3.73 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8144 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -141.02, 134.34 | APE9-dihe-in | -120.0, 134.77 | APE8-dihe-in | -57.68, 136.22 | APE8-rot-na | 336.49 | APE67-dihe-in | -65.99, -13.55 | -58.92, -37.48 | APE12-dist-na | 12.2732 | APE11-dist-na | 7.2822 | APE10-dist-na | 10.4793 | APE9-dist-in | 5.5979 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | A | 287.0 | 268.0 | 7 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 7kp6 | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 7KP6B | Q07912 | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.9711 | 13.4096 | ABAminus | -118.46, 0.28 | -140.74, 140.65 | -134.73, 29.67 | 302.28, 95.76 | -64.4, -24.8 | in-in | in | 8.4656 | Saltbr-in | 2.4826 | HRD-in | -80.63, -45.48 | 68.06, 5.55 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.891 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 149.74 | APE9-dihe-in | -131.88, 157.91 | APE8-dihe-in | -71.95, 81.45 | APE8-rot-na | 27.93 | APE67-dihe-in | -74.26, -9.58 | -63.95, -29.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.433 | APE9-dist-in | 6.5464 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | B | 287.0 | 265.0 | 10 | 31 | 27 | 4 | [[126, 387]] | 1.0 | 7kp6 | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 6VQMA | Q07912 | 117 | 390 | 1038.0 | R7P:401 | Type1 | Inactive | DFGin | 6.1676 | 13.4636 | ABAminus | -107.72, -37.34 | -107.23, 139.71 | -135.32, 26.09 | 306.21, 97.86 | -71.9, -43.92 | in-in | in | 8.5769 | Saltbr-in | 2.571 | HRD-in | -71.98, -51.6 | 65.1, 16.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.996 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.12, 107.17 | APE9-dihe-in | -75.55, 154.5 | APE8-dihe-in | -75.48, 79.2 | APE8-rot-na | 33.66 | APE67-dihe-in | -66.81, -24.97 | -59.46, -37.23 | APE12-dist-na | 13.5428 | APE11-dist-na | 8.2872 | APE10-dist-na | 10.8443 | APE9-dist-in | 6.5729 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | A | 289.0 | 267.0 | 7 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 6vqm | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 8FE9A | Q07912 | 117 | 390 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 7.3704 | 13.0176 | ABAminus | -105.28, -25.45 | -117.67, 141.58 | -139.74, 24.77 | 304.61, 88.92 | -62.34, -21.69 | in-in | in | 9.1793 | Saltbr-in | 3.598 | HRD-in | -80.64, -42.58 | 70.6, 2.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9194 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.63, 116.01 | APE9-dihe-in | -111.81, 145.17 | APE8-dihe-in | -57.08, 126.3 | APE8-rot-na | 336.42 | APE67-dihe-in | -51.19, -45.24 | -69.67, -25.96 | APE12-dist-na | 13.2508 | APE11-dist-na | 7.9549 | APE10-dist-na | 11.9713 | APE9-dist-in | 6.328 | K161Q | None | None | XRAY | 3.2 | 0.192 | 0.228 | A | 287.0 | 274.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8fe9 | TYR_TNK2_HUMAN | TYR | 1.7e-85 | 292.4 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4ID7A | Q07912 | 117 | 389 | 1038.0 | 1G0:401 | Type1.5_Back | Inactive | DFGin | 7.3004 | 14.1492 | ABAminus | -100.89, -41.99 | -119.98, 142.93 | -136.82, 28.94 | 304.41, 92.31 | -64.16, -28.63 | out-out | out | 10.5943 | Saltbr-out | 5.1735 | HRD-in | -73.52, -37.85 | 67.07, 1.92 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7798 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.45, 115.86 | APE9-dihe-in | -72.04, 137.46 | APE8-dihe-in | -82.5, 104.34 | APE8-rot-na | 27.83 | APE67-dihe-in | -58.7, -32.88 | -52.23, -52.86 | APE12-dist-na | 13.3714 | APE11-dist-na | 8.5283 | APE10-dist-na | 10.9965 | APE9-dist-in | 6.8929 | None | None | None | XRAY | 3.0 | 0.213 | 0.259 | A | 273.0 | 268.0 | 5 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4id7 | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 8HMTA | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.4729 | 13.951 | ABAminus | -118.49, 19.83 | -162.39, 140.84 | -133.87, 20.8 | 306.3, 104.45 | -62.09, -37.78 | in-out | in | 9.0421 | Saltbr-out | 3.7008 | HRD-in | -83.9, -47.14 | 69.67, 4.35 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.1982 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.87, 119.25 | APE9-dihe-in | -119.04, 129.31 | APE8-dihe-in | -48.41, 121.71 | APE8-rot-na | 329.76 | APE67-dihe-in | -54.06, -45.26 | -70.98, -26.96 | APE12-dist-na | 11.8922 | APE11-dist-na | 7.0236 | APE10-dist-na | 10.3283 | APE9-dist-in | 6.2242 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | A | 273.0 | 270.0 | 3 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 8HMTB | Q07912 | 117 | 388 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.5293 | 13.483 | ABAminus | -91.46, -72.88 | -101.02, 153.06 | -135.07, 25.09 | 315.45, 85.41 | -54.87, -35.23 | in-in | in | 8.8835 | Saltbr-in | 3.5996 | HRD-in | -84.2, -43.48 | 69.63, 0.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0633 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -126.21, 93.78 | APE9-dihe-in | -110.75, 147.04 | APE8-dihe-in | -62.13, 122.57 | APE8-rot-na | 330.26 | APE67-dihe-in | -58.09, -48.9 | -67.75, -29.14 | APE12-dist-na | 12.2872 | APE11-dist-na | 7.6989 | APE10-dist-na | 10.1436 | APE9-dist-in | 6.7515 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | B | 273.0 | 269.0 | 3 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 8HMTC | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.6912 | 13.3132 | ABAminus | -131.24, 29.48 | -133.92, 126.7 | -139.44, 20.75 | 308.54, 95.78 | -72.46, -43.8 | in-out | in | 8.8786 | Saltbr-out | 6.2022 | HRD-in | -85.66, -46.96 | 68.19, 1.14 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.0707 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.97, 132.16 | APE9-dihe-in | -105.55, 149.15 | APE8-dihe-in | -44.92, 133.48 | APE8-rot-na | 327.23 | APE67-dihe-in | -37.27, -59.27 | -63.72, -43.44 | APE12-dist-na | 12.373 | APE11-dist-na | 7.1129 | APE10-dist-na | 10.7313 | APE9-dist-in | 5.9562 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | C | 273.0 | 262.0 | 11 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 3EQRA | Q07912 | 117 | 392 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.8667 | 13.3824 | ABAminus | -128.87, 39.52 | -159.68, 137.58 | -136.82, 17.85 | 302.67, 104.42 | -47.59, -35.87 | in-in | in | 8.4309 | Saltbr-in | 2.6926 | HRD-in | -84.2, -49.01 | 74.75, 3.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8626 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -146.69, 130.79 | APE9-dihe-in | -116.23, 133.53 | APE8-dihe-in | -52.18, 127.34 | APE8-rot-na | 331.23 | APE67-dihe-in | -63.51, -16.76 | -51.88, -37.16 | APE12-dist-na | 12.2102 | APE11-dist-na | 7.1706 | APE10-dist-na | 10.3549 | APE9-dist-in | 5.493 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | A | 276.0 | 270.0 | 6 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 3eqr | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 3EQRB | Q07912 | 117 | 390 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.7947 | 13.431 | ABAminus | -120.3, 36.38 | -155.51, 142.4 | -140.09, 20.29 | 304.07, 98.58 | -61.13, -29.69 | in-in | in | 8.5153 | Saltbr-in | 2.733 | HRD-in | -83.74, -48.84 | 74.17, 1.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9014 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.77, 150.09 | APE9-dihe-in | -122.65, 150.11 | APE8-dihe-in | -70.86, 79.63 | APE8-rot-na | 24.49 | APE67-dihe-in | -77.33, -9.73 | -59.15, -33.0 | APE12-dist-na | 999.0 | APE11-dist-na | 9.2365 | APE10-dist-na | 11.3291 | APE9-dist-in | 6.6703 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | B | 276.0 | 271.0 | 3 | 31 | 28 | 3 | [[126, 387]] | 1.0 | 3eqr | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 3EQPA | Q07912 | 117 | 390 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.7129 | 14.0036 | BLAminus | -122.28, -169.39 | 49.91, 85.82 | -103.52, 29.12 | 298.07, 93.89 | -65.88, -22.57 | in-in | in | 8.5579 | Saltbr-in | 2.5574 | HRD-in | -67.58, -47.8 | 79.03, -3.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9373 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 41.47, 68.24 | APE9-dihe-in | -80.12, 152.64 | APE8-dihe-in | -67.7, 101.83 | APE8-rot-na | 335.05 | APE67-dihe-in | -66.98, -8.09 | -37.76, -57.12 | APE12-dist-na | 12.432 | APE11-dist-na | 7.613 | APE10-dist-na | 11.6899 | APE9-dist-in | 6.3009 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | A | 276.0 | 268.0 | 6 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 3eqp | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 3EQPB | Q07912 | 117 | 392 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.7469 | 13.9414 | BLAminus | -134.99, 176.53 | 61.95, 90.21 | -110.2, 23.83 | 297.71, 92.68 | -58.95, -17.74 | in-in | in | 8.4225 | Saltbr-in | 2.5793 | HRD-in | -73.01, -48.54 | 76.03, -4.13 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.816 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 48.1, 56.77 | APE9-dihe-in | -72.7, 143.2 | APE8-dihe-in | -64.45, 112.29 | APE8-rot-na | 344.7 | APE67-dihe-in | -74.41, -9.69 | -53.7, -41.09 | APE12-dist-na | 12.3732 | APE11-dist-na | 7.5143 | APE10-dist-na | 11.7317 | APE9-dist-in | 6.1729 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | B | 276.0 | 270.0 | 6 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 3eqp | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4HZSA | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.3975 | 13.7313 | BLBplus | -128.49, 177.6 | 75.97, 0.07 | -64.52, 114.85 | 48.75, 95.91 | 91.75, 5.84 | out-out | out | 13.902 | Saltbr-out | 13.592 | HRD-in | -83.45, -44.79 | 72.11, -12.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0079 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.92 | APE8-dihe-in | -80.17, 58.22 | APE8-rot-na | 31.2 | APE67-dihe-in | -83.82, 0.51 | -43.12, -45.6 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5609 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | A | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4HZSB | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4015 | 13.6973 | BLBplus | -127.73, 176.98 | 75.42, 0.58 | -63.8, 113.76 | 49.58, 96.39 | 93.88, 5.2 | out-out | out | 13.8949 | Saltbr-out | 13.5644 | HRD-in | -82.56, -44.07 | 71.76, -13.74 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0156 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.49 | APE8-dihe-in | -80.43, 57.86 | APE8-rot-na | 30.79 | APE67-dihe-in | -82.93, -0.7 | -42.53, -45.05 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5517 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | B | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4HZSC | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4202 | 13.7278 | BLBplus | -131.14, 178.08 | 74.14, -0.16 | -64.4, 114.39 | 48.24, 95.76 | 92.64, 7.14 | out-out | out | 13.8795 | Saltbr-out | 13.5598 | HRD-in | -80.94, -46.54 | 73.93, -15.02 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.9918 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.59 | APE8-dihe-in | -80.99, 59.29 | APE8-rot-na | 31.45 | APE67-dihe-in | -82.91, 0.04 | -43.57, -45.3 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5678 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | C | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 4HZSD | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4031 | 13.7071 | BLBplus | -127.5, 176.15 | 76.3, -0.17 | -64.31, 115.24 | 47.66, 95.75 | 91.47, 5.35 | out-out | out | 13.8763 | Saltbr-out | 13.5638 | HRD-in | -81.93, -43.89 | 71.65, -14.69 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0158 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 150.39 | APE8-dihe-in | -81.82, 58.59 | APE8-rot-na | 31.39 | APE67-dihe-in | -80.9, -1.27 | -43.09, -46.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5893 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | D | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 8HMTD | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.3063 | 13.3328 | None | -101.89, -122.34 | -52.57, 148.88 | -124.51, 20.24 | 302.36, 99.89 | -60.05, -38.85 | in-out | in | 8.5635 | Saltbr-out | 3.702 | HRD-in | -85.57, -47.32 | 68.53, 3.51 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.0608 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.15, 128.97 | APE9-dihe-in | -122.52, 150.9 | APE8-dihe-in | -68.07, 94.15 | APE8-rot-na | 328.13 | APE67-dihe-in | -58.59, -46.12 | -66.12, -27.69 | APE12-dist-na | 12.502 | APE11-dist-na | 7.8076 | APE10-dist-na | 10.8535 | APE9-dist-in | 5.8558 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | D | 273.0 | 262.0 | 11 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 5ZXBA | Q07912 | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.852 | 11.2639 | None | -126.71, -163.29 | -159.07, 87.59 | -102.57, 999.0 | 328.97, 133.0 | 999.0, 999.0 | in-in | in | 8.6657 | Saltbr-in | 2.5638 | HRD-in | -73.25, -51.97 | 78.84, -2.72 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.29 | APE8-rot-na | 28.55 | APE67-dihe-in | -73.12, -10.47 | -54.59, -43.66 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | A | 275.0 | 240.0 | 33 | 31 | 10 | 21 | [[126, 387]] | 1.0 | 5zxb | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 5ZXBB | Q07912 | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.9037 | 10.9514 | None | -127.77, -163.1 | -162.7, 90.46 | -101.67, 999.0 | 328.28, 133.86 | 999.0, 999.0 | in-in | in | 8.7292 | Saltbr-in | 2.7157 | HRD-in | -72.25, -50.4 | 79.44, -3.02 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.74 | APE8-rot-na | 29.71 | APE67-dihe-in | -76.43, -11.56 | -55.87, -46.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | B | 275.0 | 241.0 | 32 | 31 | 10 | 21 | [[126, 387]] | 1.0 | 5zxb | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | 1U4DA | Q07912 | 117 | 389 | 1038.0 | DBQ:398 | Type1 | None | DFGin | 6.4998 | 13.5355 | BLAminus | -127.17, -169.67 | 54.12, 72.77 | -87.16, 24.56 | 310.51, 109.17 | -62.52, -20.25 | in-in | in | 8.7352 | Saltbr-in | 3.176 | HRD-in | -80.08, -48.95 | 65.72, 7.9 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.1723 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -41.24 | APE8-dihe-in | -76.48, 82.61 | APE8-rot-na | 31.13 | APE67-dihe-in | -69.93, -17.0 | -48.99, -48.23 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.5623 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | A | 291.0 | 258.0 | 15 | 31 | 24 | 7 | [[126, 387]] | 1.0 | 1u4d | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TNK2 | ACK1_HUMAN | 1U54B | Q07912 | 117 | 388 | 1038.0 | ACP:400 | ATPlike | Active | DFGin | 6.6155 | 13.3776 | BLAminus | -120.4, -155.16 | 27.84, 85.75 | -104.36, 38.7 | 310.01, 93.15 | -67.71, -28.73 | in-in | in | 7.966 | Saltbr-in | 3.0206 | HRD-in | -109.84, -42.56 | 64.6, 13.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0144 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -150.8, 133.1 | APE9-dihe-in | -126.86, 129.0 | APE8-dihe-in | -43.1, 130.27 | APE8-rot-na | 329.12 | APE67-dihe-in | -70.13, -6.6 | -62.78, -39.45 | APE12-dist-na | 12.6617 | APE11-dist-na | 7.6459 | APE10-dist-na | 10.9998 | APE9-dist-in | 5.8775 | None | None | None | XRAY | 2.8 | 0.226 | 0.322 | B | 291.0 | 261.0 | 11 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 1u54 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | AF-Q07912-K1A | Q07912 | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.4024 | 13.8085 | BLAminus | -127.81, -172.26 | 52.98, 78.87 | -92.01, 15.18 | 300.66, 98.99 | -61.2, -28.6 | in-in | in | 9.0677 | Saltbr-in | 2.8838 | HRD-in | -71.74, -46.77 | 66.75, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8834 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.08, 137.58 | APE9-dihe-in | -124.59, 150.42 | APE8-dihe-in | -74.79, 77.42 | APE8-rot-na | 33.67 | APE67-dihe-in | -72.2, -16.05 | -54.65, -32.93 | APE12-dist-na | 14.2254 | APE11-dist-na | 8.1727 | APE10-dist-na | 10.4882 | APE9-dist-in | 6.2148 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278.0 | 278.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K1 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | AF-Q07912-K3A | Q07912 | 118 | 395 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.2816 | 13.8163 | BLAminus | -132.02, -165.66 | 49.79, 76.66 | -89.46, 13.86 | 302.75, 106.95 | -62.78, -25.76 | in-in | in | 9.1531 | Saltbr-in | 2.8291 | HRD-in | -75.54, -47.15 | 65.26, -2.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8945 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.1, 134.59 | APE9-dihe-in | -125.28, 155.36 | APE8-dihe-in | -74.53, 75.69 | APE8-rot-na | 36.27 | APE67-dihe-in | -72.66, -16.99 | -53.38, -31.64 | APE12-dist-na | 13.715 | APE11-dist-na | 7.7486 | APE10-dist-na | 10.0198 | APE9-dist-in | 5.7149 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 278.0 | 278.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | AF-Q07912-K3 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.6e-86 | 293.5 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 1U46B | Q07912 | 117 | 390 | 1038.0 | No_ligand | No_ligand | Active | DFGin | 6.8929 | 13.3269 | BLAminus | -106.75, -162.4 | 39.69, 86.16 | -96.94, 26.22 | 299.15, 109.43 | -73.67, -16.41 | in-in | in | 8.1814 | Saltbr-in | 2.5893 | HRD-in | -73.19, -48.75 | 76.75, -0.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9211 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -148.81, 131.4 | APE9-dihe-in | -119.81, 131.46 | APE8-dihe-in | -52.5, 137.43 | APE8-rot-na | 348.53 | APE67-dihe-in | -65.13, -16.63 | -61.62, -36.89 | APE12-dist-na | 12.2376 | APE11-dist-na | 7.1908 | APE10-dist-na | 10.2147 | APE9-dist-in | 5.6432 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | B | 291.0 | 257.0 | 17 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 1u46 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 6VQMB | Q07912 | 117 | 392 | 1038.0 | R7P:401 | Type1 | Active | DFGin | 6.5869 | 13.5939 | BLAminus | -126.29, -176.9 | 60.12, 78.79 | -101.99, 43.61 | 309.18, 96.93 | -70.48, -42.01 | in-in | in | 8.3539 | Saltbr-in | 2.7897 | HRD-in | -70.81, -44.97 | 67.08, 13.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0338 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.03, 107.88 | APE9-dihe-in | -69.66, 138.93 | APE8-dihe-in | -77.17, 95.23 | APE8-rot-na | 27.59 | APE67-dihe-in | -70.22, -21.82 | -51.53, -42.79 | APE12-dist-na | 12.2631 | APE11-dist-na | 8.4205 | APE10-dist-na | 12.2009 | APE9-dist-in | 7.1911 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | B | 289.0 | 267.0 | 9 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 6vqm | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 1U4DB | Q07912 | 117 | 390 | 1038.0 | DBQ:401 | Type1 | Active | DFGin | 6.7434 | 13.2857 | BLAminus | -120.44, -165.36 | 55.02, 77.38 | -96.18, 18.83 | 299.22, 128.21 | -61.51, -28.63 | in-in | in | 8.506 | Saltbr-in | 3.09 | HRD-in | -78.19, -51.48 | 79.02, -2.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.79, 137.8 | APE9-dihe-in | -124.54, 129.71 | APE8-dihe-in | -55.28, 140.91 | APE8-rot-na | 333.19 | APE67-dihe-in | -67.74, -15.49 | -65.28, -34.43 | APE12-dist-na | 12.3065 | APE11-dist-na | 7.1903 | APE10-dist-na | 10.3941 | APE9-dist-in | 5.7477 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | B | 291.0 | 262.0 | 12 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 1u4d | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 1U54A | Q07912 | 115 | 390 | 1038.0 | ACP:101 | ATPlike | Inactive | DFGin | 6.3812 | 13.4263 | ABAminus | -129.39, -12.11 | -146.47, 102.96 | -102.84, 23.33 | 304.65, 105.91 | -57.05, -37.37 | in-in | in | 7.8643 | Saltbr-in | 2.6244 | HRD-in | -77.15, -49.8 | 83.51, -10.59 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8347 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 126.54 | APE8-dihe-in | -75.47, 123.76 | APE8-rot-na | 349.96 | APE67-dihe-in | -43.9, -19.78 | -62.08, -52.54 | APE12-dist-na | 11.8082 | APE11-dist-na | 8.1412 | APE10-dist-na | 999.0 | APE9-dist-in | 6.0632 | None | PTR284 | PTR284 | XRAY | 2.8 | 0.226 | 0.322 | A | 291.0 | 263.0 | 13 | 31 | 30 | 1 | [[126, 387]] | 1.0 | 1u54 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4HZRA | Q07912 | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9405 | 13.3374 | ABAminus | -116.61, 0.1 | -140.48, 143.47 | -137.83, 29.0 | 303.1, 95.78 | -63.74, -22.82 | in-in | in | 8.6705 | Saltbr-in | 3.0135 | HRD-in | -78.97, -45.99 | 73.0, 0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8523 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -137.45, 121.81 | APE9-dihe-in | -117.27, 126.54 | APE8-dihe-in | -48.18, 134.62 | APE8-rot-na | 331.8 | APE67-dihe-in | -67.06, -18.13 | -62.19, -35.06 | APE12-dist-na | 12.2207 | APE11-dist-na | 7.4764 | APE10-dist-na | 10.3681 | APE9-dist-in | 5.6397 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | A | 277.0 | 261.0 | 12 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4hzr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4HZRB | Q07912 | 118 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9261 | 13.2029 | ABAminus | -114.0, -2.21 | -142.3, 141.19 | -136.9, 28.97 | 303.67, 94.73 | -65.41, -14.9 | in-in | in | 8.3198 | Saltbr-in | 2.7836 | HRD-in | -81.57, -44.88 | 71.99, 1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8785 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -115.7, 123.01 | APE9-dihe-in | -130.03, 154.84 | APE8-dihe-in | -57.54, 124.6 | APE8-rot-na | 334.8 | APE67-dihe-in | -72.23, -12.85 | -67.01, -33.63 | APE12-dist-na | 13.4048 | APE11-dist-na | 8.5721 | APE10-dist-na | 12.141 | APE9-dist-in | 6.9585 | None | None | None | XRAY | 1.31 | 0.197 | 0.209 | B | 277.0 | 258.0 | 14 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4hzr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.5e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 1U46A | Q07912 | 117 | 389 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 6.6774 | 13.6062 | ABAminus | -105.04, -15.76 | -135.27, 148.5 | -140.73, 24.35 | 300.72, 95.61 | -66.87, -16.87 | in-in | in | 8.88 | Saltbr-in | 3.0421 | HRD-in | -74.47, -45.94 | 65.29, 8.06 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.0797 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 148.6 | APE8-dihe-in | -40.6, 125.73 | APE8-rot-na | 326.91 | APE67-dihe-in | -63.61, -22.03 | -68.77, -33.68 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.4874 | None | None | None | XRAY | 2.0 | 0.202 | 0.249 | A | 291.0 | 255.0 | 18 | 31 | 25 | 6 | [[126, 387]] | 1.0 | 1u46 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4EWHA | Q07912 | 117 | 391 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.8969 | 13.7575 | ABAminus | -112.33, -10.32 | -127.98, 158.61 | -163.96, 19.15 | 297.07, 109.95 | -51.93, -22.07 | in-in | in | 8.3631 | Saltbr-in | 2.8413 | HRD-in | -80.55, -48.4 | 69.82, -0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7842 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.82, 134.34 | APE9-dihe-in | -105.63, 146.75 | APE8-dihe-in | -58.9, 128.31 | APE8-rot-na | 332.95 | APE67-dihe-in | -67.17, -17.01 | -59.23, -34.05 | APE12-dist-na | 12.3707 | APE11-dist-na | 7.3299 | APE10-dist-na | 11.496 | APE9-dist-in | 5.9649 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | A | 275.0 | 275.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4ewh | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4EWHB | Q07912 | 117 | 390 | 1038.0 | T77:401 | Type1 | Inactive | DFGin | 6.8136 | 13.7809 | ABAminus | -113.99, 0.05 | -132.38, 146.39 | -142.78, 20.76 | 303.22, 103.13 | -48.09, -26.49 | in-in | in | 8.3351 | Saltbr-in | 2.6774 | HRD-in | -88.91, -43.41 | 72.85, -2.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -105.83, 138.68 | APE9-dihe-in | -104.08, 148.64 | APE8-dihe-in | -58.72, 120.66 | APE8-rot-na | 340.66 | APE67-dihe-in | -66.41, -17.16 | -49.99, -36.4 | APE12-dist-na | 12.4243 | APE11-dist-na | 7.3547 | APE10-dist-na | 11.5408 | APE9-dist-in | 5.9219 | None | PTR284 | PTR284 | XRAY | 2.5 | 0.259 | 0.313 | B | 275.0 | 274.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4ewh | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 7KP6A | Q07912 | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.9868 | 13.0736 | ABAminus | -120.5, 2.81 | -142.4, 134.01 | -133.76, 28.84 | 306.02, 91.7 | -68.06, -13.37 | in-out | in | 8.7113 | Saltbr-out | 4.4386 | HRD-in | -78.88, -45.58 | 72.69, 3.73 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8144 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -141.02, 134.34 | APE9-dihe-in | -120.0, 134.77 | APE8-dihe-in | -57.68, 136.22 | APE8-rot-na | 336.49 | APE67-dihe-in | -65.99, -13.55 | -58.92, -37.48 | APE12-dist-na | 12.2732 | APE11-dist-na | 7.2822 | APE10-dist-na | 10.4793 | APE9-dist-in | 5.5979 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | A | 287.0 | 268.0 | 7 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 7kp6 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 7KP6B | Q07912 | 117 | 391 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 6.9711 | 13.4096 | ABAminus | -118.46, 0.28 | -140.74, 140.65 | -134.73, 29.67 | 302.28, 95.76 | -64.4, -24.8 | in-in | in | 8.4656 | Saltbr-in | 2.4826 | HRD-in | -80.63, -45.48 | 68.06, 5.55 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.891 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 149.74 | APE9-dihe-in | -131.88, 157.91 | APE8-dihe-in | -71.95, 81.45 | APE8-rot-na | 27.93 | APE67-dihe-in | -74.26, -9.58 | -63.95, -29.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.433 | APE9-dist-in | 6.5464 | None | None | None | XRAY | 1.79 | 0.179 | 0.203 | B | 287.0 | 265.0 | 10 | 31 | 27 | 4 | [[126, 387]] | 1.0 | 7kp6 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.6e-86 | 293.4 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 6VQMA | Q07912 | 117 | 390 | 1038.0 | R7P:401 | Type1 | Inactive | DFGin | 6.1676 | 13.4636 | ABAminus | -107.72, -37.34 | -107.23, 139.71 | -135.32, 26.09 | 306.21, 97.86 | -71.9, -43.92 | in-in | in | 8.5769 | Saltbr-in | 2.571 | HRD-in | -71.98, -51.6 | 65.1, 16.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.996 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.12, 107.17 | APE9-dihe-in | -75.55, 154.5 | APE8-dihe-in | -75.48, 79.2 | APE8-rot-na | 33.66 | APE67-dihe-in | -66.81, -24.97 | -59.46, -37.23 | APE12-dist-na | 13.5428 | APE11-dist-na | 8.2872 | APE10-dist-na | 10.8443 | APE9-dist-in | 6.5729 | None | None | None | XRAY | 2.87 | 0.273 | 0.33 | A | 289.0 | 267.0 | 7 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 6vqm | Homo sapiens | TYR_TNK2_HUMAN | TYR | 8.8e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 8FE9A | Q07912 | 117 | 390 | 1038.0 | WTP:401 | Type1 | Inactive | DFGin | 7.3704 | 13.0176 | ABAminus | -105.28, -25.45 | -117.67, 141.58 | -139.74, 24.77 | 304.61, 88.92 | -62.34, -21.69 | in-in | in | 9.1793 | Saltbr-in | 3.598 | HRD-in | -80.64, -42.58 | 70.6, 2.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9194 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.63, 116.01 | APE9-dihe-in | -111.81, 145.17 | APE8-dihe-in | -57.08, 126.3 | APE8-rot-na | 336.42 | APE67-dihe-in | -51.19, -45.24 | -69.67, -25.96 | APE12-dist-na | 13.2508 | APE11-dist-na | 7.9549 | APE10-dist-na | 11.9713 | APE9-dist-in | 6.328 | K161Q | None | None | XRAY | 3.2 | 0.192 | 0.228 | A | 287.0 | 274.0 | 0 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8fe9 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.7e-85 | 292.4 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4ID7A | Q07912 | 117 | 389 | 1038.0 | 1G0:401 | Type1.5_Back | Inactive | DFGin | 7.3004 | 14.1492 | ABAminus | -100.89, -41.99 | -119.98, 142.93 | -136.82, 28.94 | 304.41, 92.31 | -64.16, -28.63 | out-out | out | 10.5943 | Saltbr-out | 5.1735 | HRD-in | -73.52, -37.85 | 67.07, 1.92 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7798 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.45, 115.86 | APE9-dihe-in | -72.04, 137.46 | APE8-dihe-in | -82.5, 104.34 | APE8-rot-na | 27.83 | APE67-dihe-in | -58.7, -32.88 | -52.23, -52.86 | APE12-dist-na | 13.3714 | APE11-dist-na | 8.5283 | APE10-dist-na | 10.9965 | APE9-dist-in | 6.8929 | None | None | None | XRAY | 3.0 | 0.213 | 0.259 | A | 273.0 | 268.0 | 5 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 4id7 | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 8HMTA | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.4729 | 13.951 | ABAminus | -118.49, 19.83 | -162.39, 140.84 | -133.87, 20.8 | 306.3, 104.45 | -62.09, -37.78 | in-out | in | 9.0421 | Saltbr-out | 3.7008 | HRD-in | -83.9, -47.14 | 69.67, 4.35 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.1982 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.87, 119.25 | APE9-dihe-in | -119.04, 129.31 | APE8-dihe-in | -48.41, 121.71 | APE8-rot-na | 329.76 | APE67-dihe-in | -54.06, -45.26 | -70.98, -26.96 | APE12-dist-na | 11.8922 | APE11-dist-na | 7.0236 | APE10-dist-na | 10.3283 | APE9-dist-in | 6.2242 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | A | 273.0 | 270.0 | 3 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 8HMTB | Q07912 | 117 | 388 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.5293 | 13.483 | ABAminus | -91.46, -72.88 | -101.02, 153.06 | -135.07, 25.09 | 315.45, 85.41 | -54.87, -35.23 | in-in | in | 8.8835 | Saltbr-in | 3.5996 | HRD-in | -84.2, -43.48 | 69.63, 0.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0633 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -126.21, 93.78 | APE9-dihe-in | -110.75, 147.04 | APE8-dihe-in | -62.13, 122.57 | APE8-rot-na | 330.26 | APE67-dihe-in | -58.09, -48.9 | -67.75, -29.14 | APE12-dist-na | 12.2872 | APE11-dist-na | 7.6989 | APE10-dist-na | 10.1436 | APE9-dist-in | 6.7515 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | B | 273.0 | 269.0 | 3 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 8HMTC | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.6912 | 13.3132 | ABAminus | -131.24, 29.48 | -133.92, 126.7 | -139.44, 20.75 | 308.54, 95.78 | -72.46, -43.8 | in-out | in | 8.8786 | Saltbr-out | 6.2022 | HRD-in | -85.66, -46.96 | 68.19, 1.14 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.0707 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -138.97, 132.16 | APE9-dihe-in | -105.55, 149.15 | APE8-dihe-in | -44.92, 133.48 | APE8-rot-na | 327.23 | APE67-dihe-in | -37.27, -59.27 | -63.72, -43.44 | APE12-dist-na | 12.373 | APE11-dist-na | 7.1129 | APE10-dist-na | 10.7313 | APE9-dist-in | 5.9562 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | C | 273.0 | 262.0 | 11 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 3EQRA | Q07912 | 117 | 392 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.8667 | 13.3824 | ABAminus | -128.87, 39.52 | -159.68, 137.58 | -136.82, 17.85 | 302.67, 104.42 | -47.59, -35.87 | in-in | in | 8.4309 | Saltbr-in | 2.6926 | HRD-in | -84.2, -49.01 | 74.75, 3.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8626 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -146.69, 130.79 | APE9-dihe-in | -116.23, 133.53 | APE8-dihe-in | -52.18, 127.34 | APE8-rot-na | 331.23 | APE67-dihe-in | -63.51, -16.76 | -51.88, -37.16 | APE12-dist-na | 12.2102 | APE11-dist-na | 7.1706 | APE10-dist-na | 10.3549 | APE9-dist-in | 5.493 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | A | 276.0 | 270.0 | 6 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 3eqr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 3EQRB | Q07912 | 117 | 390 | 1038.0 | T74:1 | Type1.5_Back | Inactive | DFGin | 6.7947 | 13.431 | ABAminus | -120.3, 36.38 | -155.51, 142.4 | -140.09, 20.29 | 304.07, 98.58 | -61.13, -29.69 | in-in | in | 8.5153 | Saltbr-in | 2.733 | HRD-in | -83.74, -48.84 | 74.17, 1.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9014 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.77, 150.09 | APE9-dihe-in | -122.65, 150.11 | APE8-dihe-in | -70.86, 79.63 | APE8-rot-na | 24.49 | APE67-dihe-in | -77.33, -9.73 | -59.15, -33.0 | APE12-dist-na | 999.0 | APE11-dist-na | 9.2365 | APE10-dist-na | 11.3291 | APE9-dist-in | 6.6703 | None | None | None | XRAY | 2.0 | 0.212 | 0.256 | B | 276.0 | 271.0 | 3 | 31 | 28 | 3 | [[126, 387]] | 1.0 | 3eqr | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 3EQPA | Q07912 | 117 | 390 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.7129 | 14.0036 | BLAminus | -122.28, -169.39 | 49.91, 85.82 | -103.52, 29.12 | 298.07, 93.89 | -65.88, -22.57 | in-in | in | 8.5579 | Saltbr-in | 2.5574 | HRD-in | -67.58, -47.8 | 79.03, -3.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9373 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 41.47, 68.24 | APE9-dihe-in | -80.12, 152.64 | APE8-dihe-in | -67.7, 101.83 | APE8-rot-na | 335.05 | APE67-dihe-in | -66.98, -8.09 | -37.76, -57.12 | APE12-dist-na | 12.432 | APE11-dist-na | 7.613 | APE10-dist-na | 11.6899 | APE9-dist-in | 6.3009 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | A | 276.0 | 268.0 | 6 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 3eqp | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 3EQPB | Q07912 | 117 | 392 | 1038.0 | T95:1 | Type1 | Inactive | DFGin | 6.7469 | 13.9414 | BLAminus | -134.99, 176.53 | 61.95, 90.21 | -110.2, 23.83 | 297.71, 92.68 | -58.95, -17.74 | in-in | in | 8.4225 | Saltbr-in | 2.5793 | HRD-in | -73.01, -48.54 | 76.03, -4.13 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.816 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 48.1, 56.77 | APE9-dihe-in | -72.7, 143.2 | APE8-dihe-in | -64.45, 112.29 | APE8-rot-na | 344.7 | APE67-dihe-in | -74.41, -9.69 | -53.7, -41.09 | APE12-dist-na | 12.3732 | APE11-dist-na | 7.5143 | APE10-dist-na | 11.7317 | APE9-dist-in | 6.1729 | None | None | None | XRAY | 2.3 | 0.224 | 0.284 | B | 276.0 | 270.0 | 6 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 3eqp | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.4e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4HZSA | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.3975 | 13.7313 | BLBplus | -128.49, 177.6 | 75.97, 0.07 | -64.52, 114.85 | 48.75, 95.91 | 91.75, 5.84 | out-out | out | 13.902 | Saltbr-out | 13.592 | HRD-in | -83.45, -44.79 | 72.11, -12.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0079 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.92 | APE8-dihe-in | -80.17, 58.22 | APE8-rot-na | 31.2 | APE67-dihe-in | -83.82, 0.51 | -43.12, -45.6 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5609 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | A | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4HZSB | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4015 | 13.6973 | BLBplus | -127.73, 176.98 | 75.42, 0.58 | -63.8, 113.76 | 49.58, 96.39 | 93.88, 5.2 | out-out | out | 13.8949 | Saltbr-out | 13.5644 | HRD-in | -82.56, -44.07 | 71.76, -13.74 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0156 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.49 | APE8-dihe-in | -80.43, 57.86 | APE8-rot-na | 30.79 | APE67-dihe-in | -82.93, -0.7 | -42.53, -45.05 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5517 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | B | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4HZSC | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4202 | 13.7278 | BLBplus | -131.14, 178.08 | 74.14, -0.16 | -64.4, 114.39 | 48.24, 95.76 | 92.64, 7.14 | out-out | out | 13.8795 | Saltbr-out | 13.5598 | HRD-in | -80.94, -46.54 | 73.93, -15.02 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.9918 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.59 | APE8-dihe-in | -80.99, 59.29 | APE8-rot-na | 31.45 | APE67-dihe-in | -82.91, 0.04 | -43.57, -45.3 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5678 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | C | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 4HZSD | Q07912 | 115 | 446 | 1038.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4031 | 13.7071 | BLBplus | -127.5, 176.15 | 76.3, -0.17 | -64.31, 115.24 | 47.66, 95.75 | 91.47, 5.35 | out-out | out | 13.8763 | Saltbr-out | 13.5638 | HRD-in | -81.93, -43.89 | 71.65, -14.69 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0158 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 150.39 | APE8-dihe-in | -81.82, 58.59 | APE8-rot-na | 31.39 | APE67-dihe-in | -80.9, -1.27 | -43.09, -46.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.5893 | None | None | None | XRAY | 3.23 | 0.247 | 0.27 | D | 341.0 | 319.0 | 13 | 31 | 18 | 13 | [[126, 387]] | 1.0 | 4hzs | Homo sapiens | TYR_TNK2_HUMAN | TYR | 1.6e-85 | 292.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 8HMTD | Q07912 | 117 | 389 | 1038.0 | LWX:401 | Type1.5_Back | Inactive | DFGin | 6.3063 | 13.3328 | None | -101.89, -122.34 | -52.57, 148.88 | -124.51, 20.24 | 302.36, 99.89 | -60.05, -38.85 | in-out | in | 8.5635 | Saltbr-out | 3.702 | HRD-in | -85.57, -47.32 | 68.53, 3.51 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.0608 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.15, 128.97 | APE9-dihe-in | -122.52, 150.9 | APE8-dihe-in | -68.07, 94.15 | APE8-rot-na | 328.13 | APE67-dihe-in | -58.59, -46.12 | -66.12, -27.69 | APE12-dist-na | 12.502 | APE11-dist-na | 7.8076 | APE10-dist-na | 10.8535 | APE9-dist-in | 5.8558 | None | None | None | XRAY | 3.17 | 0.209 | 0.264 | D | 273.0 | 262.0 | 11 | 31 | 31 | 0 | [[126, 387]] | 1.0 | 8hmt | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.1e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 5ZXBA | Q07912 | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.852 | 11.2639 | None | -126.71, -163.29 | -159.07, 87.59 | -102.57, 999.0 | 328.97, 133.0 | 999.0, 999.0 | in-in | in | 8.6657 | Saltbr-in | 2.5638 | HRD-in | -73.25, -51.97 | 78.84, -2.72 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.29 | APE8-rot-na | 28.55 | APE67-dihe-in | -73.12, -10.47 | -54.59, -43.66 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | A | 275.0 | 240.0 | 33 | 31 | 10 | 21 | [[126, 387]] | 1.0 | 5zxb | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 5ZXBB | Q07912 | 117 | 389 | 1038.0 | 9KO:401 | Type2 | Inactive | DFGout | 12.9037 | 10.9514 | None | -127.77, -163.1 | -162.7, 90.46 | -101.67, 999.0 | 328.28, 133.86 | 999.0, 999.0 | in-in | in | 8.7292 | Saltbr-in | 2.7157 | HRD-in | -72.25, -50.4 | 79.44, -3.02 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.74 | APE8-rot-na | 29.71 | APE67-dihe-in | -76.43, -11.56 | -55.87, -46.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.198 | 0.209 | 0.257 | B | 275.0 | 241.0 | 32 | 31 | 10 | 21 | [[126, 387]] | 1.0 | 5zxb | Homo sapiens | TYR_TNK2_HUMAN | TYR | 7.3e-86 | 293.6 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| TNK2 | ACK1_HUMAN | 1U4DA | Q07912 | 117 | 389 | 1038.0 | DBQ:398 | Type1 | None | DFGin | 6.4998 | 13.5355 | BLAminus | -127.17, -169.67 | 54.12, 72.77 | -87.16, 24.56 | 310.51, 109.17 | -62.52, -20.25 | in-in | in | 8.7352 | Saltbr-in | 3.176 | HRD-in | -80.08, -48.95 | 65.72, 7.9 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.1723 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -41.24 | APE8-dihe-in | -76.48, 82.61 | APE8-rot-na | 31.13 | APE67-dihe-in | -69.93, -17.0 | -48.99, -48.23 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.5623 | None | None | None | XRAY | 2.1 | 0.205 | 0.248 | A | 291.0 | 258.0 | 15 | 31 | 24 | 7 | [[126, 387]] | 1.0 | 1u4d | Homo sapiens | TYR_TNK2_HUMAN | TYR | 9e-86 | 293.3 | 1.0 | 259.0 | 259.0 | 269 | 270 | 271 | 273 | 275 | 158 | 177 | 181 | 249 | 251 | 250 | 252.0 | 312 | 300 | 295 | 294 | 293 | 292 | 291 | 290 | 289 | 206 | Activated CDC42 kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|