CAMK_PIM1 (Serine/threonine-protein kinase pim-1)

Total number of chains: 198
Active chains: 188
Uniprot: PIM1_HUMAN
Kinase Domain Residues: 38 - 290
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 190 96.0% AF-P11309-K1A
DFGin ABAminus 5 2.5% 4RC2A
DFGin None 2 1.0% 4XH6A
DFGin BLBminus 1 0.5% 6KZIA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PIM1 1YXTA P11309 33 306 313.0 ANP:322 ATPlike Active DFGin 6.0285 14.2451 BLAminus -131.81, 176.98 66.39, 83.69 -99.64, 19.64 287.53, 80.25 -65.72, -15.35 in-in in 8.3094 Saltbr-in 2.8936 HRD-naA -67.95, -50.18 66.45, 4.68 in-in-in SNCiii in-in ActLoopNT-in 2.8088 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.69, 12.99 APE9-dihe-na -80.03, -158.46 APE8-dihe-in -83.46, 121.7 APE8-rot-in 308.53 APE67-dihe-in -70.36, -3.81 -49.69, -52.76 APE12-dist-in 9.7291 APE11-dist-in 8.6653 APE10-dist-in 5.2788 APE9-dist-in 3.8051 None None None XRAY 2.0 0.183 0.216 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxt CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXUA P11309 33 305 313.0 AMP:550 ATPlike Active DFGin 6.0455 14.5804 BLAminus -128.48, 170.01 62.85, 77.77 -90.35, 20.24 287.6, 77.99 -74.7, 1.63 in-in in 8.5131 Saltbr-in 2.4861 HRD-naA -60.24, -50.74 67.33, 4.52 in-in-in SNCiii in-in ActLoopNT-in 2.8925 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.18, 25.46 APE9-dihe-na -90.91, -158.18 APE8-dihe-in -86.5, 120.86 APE8-rot-in 310.09 APE67-dihe-in -63.06, -9.2 -60.21, -45.83 APE12-dist-in 9.9588 APE11-dist-in 8.8348 APE10-dist-in 5.6887 APE9-dist-in 3.8693 None None None XRAY 2.24 0.231 0.276 A 293.0 273.0 0 26 26 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXUB P11309 33 305 313.0 AMP:650 ATPlike Active DFGin 6.1203 14.6734 BLAminus -120.37, 167.93 65.74, 85.44 -95.36, 14.03 285.37, 78.45 -64.71, -9.22 in-in in 8.6002 Saltbr-in 2.814 HRD-naA -59.51, -51.25 68.06, 6.92 in-in-in SNCiii in-in ActLoopNT-in 2.9988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.12, 36.18 APE9-dihe-na -84.74, -152.35 APE8-dihe-in -93.27, 122.65 APE8-rot-in 302.12 APE67-dihe-in -68.21, -7.03 -55.31, -45.11 APE12-dist-in 9.8003 APE11-dist-in 8.5338 APE10-dist-in 5.4571 APE9-dist-in 3.8415 None None None XRAY 2.24 0.231 0.276 B 293.0 273.0 0 26 26 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXUC P11309 34 305 313.0 AMP:750 ATPlike Active DFGin 6.1096 14.7409 BLAminus -134.94, 167.86 62.59, 83.1 -95.62, 21.45 280.06, 80.63 -81.83, 7.92 in-in in 8.7162 Saltbr-in 2.6122 HRD-naA -67.31, -48.53 67.93, 5.85 in-in-in SNCiii in-in ActLoopNT-in 2.8989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.01, 44.98 APE9-dihe-na -103.92, -155.25 APE8-dihe-in -86.11, 117.99 APE8-rot-in 310.09 APE67-dihe-in -68.22, -9.23 -52.45, -45.39 APE12-dist-in 9.6966 APE11-dist-in 8.6541 APE10-dist-in 5.6036 APE9-dist-in 3.8474 None None None XRAY 2.24 0.231 0.276 C 293.0 272.0 0 26 26 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXUD P11309 33 305 313.0 AMP:850 ATPlike Active DFGin 6.2355 14.5561 BLAminus -126.04, 169.08 67.7, 73.28 -88.52, 13.94 289.01, 78.99 -70.28, -2.85 in-in in 8.7886 Saltbr-in 2.4658 HRD-naA -64.06, -51.29 66.47, 10.4 in-in-in SNCiii in-in ActLoopNT-in 2.9168 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.8, 31.82 APE9-dihe-na -93.66, -159.09 APE8-dihe-in -85.99, 118.35 APE8-rot-in 303.12 APE67-dihe-in -71.66, -13.36 -52.91, -39.75 APE12-dist-in 9.8955 APE11-dist-in 8.6446 APE10-dist-in 5.4567 APE9-dist-in 3.827 None None None XRAY 2.24 0.231 0.276 D 293.0 273.0 0 26 26 0 [[38, 290]] 1.0 1yxu CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1XR1A P11309 32 308 313.0 ANP:501 ATPlike Active DFGin 5.8877 14.2143 BLAminus -138.05, 176.98 59.78, 85.31 -96.55, 16.88 287.93, 82.19 -61.38, -7.19 in-in in 8.717 Saltbr-in 2.833 HRD-naA -59.95, -51.82 71.23, 5.72 in-in-in SNCiii in-in ActLoopNT-in 2.7525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.05, 45.66 APE9-dihe-na -114.17, -171.15 APE8-dihe-in -64.11, 112.97 APE8-rot-in 299.41 APE67-dihe-in -49.28, -12.21 -42.84, -67.53 APE12-dist-in 9.6083 APE11-dist-in 8.6947 APE10-dist-in 5.5225 APE9-dist-in 4.0703 None None None XRAY 2.1 0.267 0.301 A 300.0 277.0 0 26 26 0 [[38, 290]] 1.0 1xr1 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3A99A P11309 33 305 313.0 ANP:501 ATPlike Active DFGin 5.9337 14.254 BLAminus -128.38, 171.59 60.85, 87.29 -96.61, 22.08 288.57, 75.78 -65.84, -9.23 in-in in 8.7536 Saltbr-in 2.6044 HRD-naA -66.86, -47.45 66.12, 8.26 in-in-in SNCiii in-in ActLoopNT-in 2.8889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.19, 26.41 APE9-dihe-na -87.51, -159.07 APE8-dihe-in -85.64, 119.66 APE8-rot-in 305.41 APE67-dihe-in -70.7, -5.81 -56.65, -39.81 APE12-dist-in 9.6122 APE11-dist-in 8.4607 APE10-dist-in 5.2903 APE9-dist-in 3.7779 None None None XRAY 1.6 0.187 0.206 A 320.0 273.0 0 26 26 0 [[38, 290]] 1.0 3a99 CAMK_PIM1_HUMAN CAMK 4.3e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2BZKB P11309 33 305 313.0 ANP:1306 ATPlike Active DFGin 6.1262 14.4434 BLAminus -123.86, 174.78 64.57, 79.13 -87.5, 17.23 286.98, 86.61 -67.5, -17.62 in-in in 8.7809 Saltbr-in 2.7266 HRD-naA -70.49, -48.81 68.36, 6.4 in-in-in SNCiii in-in ActLoopNT-in 2.8129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.63, 10.91 APE9-dihe-na -77.79, -156.22 APE8-dihe-in -90.85, 124.06 APE8-rot-in 315.85 APE67-dihe-in -68.94, -10.63 -60.69, -42.64 APE12-dist-in 9.4641 APE11-dist-in 8.4783 APE10-dist-in 4.8507 APE9-dist-in 3.7821 R250G None None XRAY 2.45 0.191 0.225 B 313.0 268.0 5 26 26 0 [[38, 290]] 1.0 2bzk CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXSA P11309 33 306 313.0 No_ligand No_ligand Active DFGin 6.0435 14.6911 BLAminus -127.76, 171.69 59.08, 88.63 -95.69, 24.45 285.74, 79.92 -71.89, -12.05 in-in in 8.8359 Saltbr-in 2.5148 HRD-naA -69.25, -46.6 65.7, 9.18 in-in-in SNCiii in-in ActLoopNT-in 2.8874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.7, 28.09 APE9-dihe-na -94.38, -153.78 APE8-dihe-in -89.3, 121.74 APE8-rot-in 312.97 APE67-dihe-in -69.81, -9.24 -57.4, -43.57 APE12-dist-in 9.6115 APE11-dist-in 8.495 APE10-dist-in 5.3233 APE9-dist-in 3.8299 P123M None None XRAY 2.2 0.197 0.237 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxs CAMK_PIM1_HUMAN CAMK 5.7e-66 228.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 AF-P11309-K1A P11309 30 298 313.0 No_ligand No_ligand Active DFGin 5.9244 14.426 BLAminus -123.59, 173.12 59.42, 75.84 -84.42, 19.94 286.93, 72.18 -59.74, -40.02 in-in in 8.502 Saltbr-in 2.6923 HRD-naA -69.93, -42.11 63.25, -11.96 in-in-in SNCiii in-in ActLoopNT-in 2.8371 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.01, 20.91 APE9-dihe-na -84.17, 176.91 APE8-dihe-in -67.72, 122.1 APE8-rot-in 305.72 APE67-dihe-in -69.25, -16.84 -56.89, -41.09 APE12-dist-in 9.5789 APE11-dist-in 8.723 APE10-dist-in 4.8295 APE9-dist-in 3.8227 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 26 26 0 [[38, 290]] 1.0 AF-P11309-K1 CAMK_PIM1_HUMAN CAMK 2.3e-65 226.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 AF-P11309-K3A P11309 30 298 313.0 No_ligand No_ligand Active DFGin 5.794 14.2839 BLAminus -126.38, 175.52 54.92, 81.68 -85.76, 15.39 286.52, 75.42 -58.44, -43.23 in-in in 8.4804 Saltbr-in 2.6753 HRD-naA -72.55, -35.61 62.65, -28.81 in-in-in SNCiii in-in ActLoopNT-in 2.818 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.76, 133.51 APE9-dihe-na 135.29, -179.73 APE8-dihe-in -78.77, 123.98 APE8-rot-in 299.06 APE67-dihe-in -67.9, -19.52 -59.41, -42.11 APE12-dist-in 10.2793 APE11-dist-in 9.2154 APE10-dist-in 4.16 APE9-dist-in 4.4335 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 26 26 0 [[38, 290]] 1.0 AF-P11309-K3 CAMK_PIM1_HUMAN CAMK 2.3e-65 226.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YWVA P11309 33 306 313.0 No_ligand No_ligand Active DFGin 6.1075 14.6848 BLAminus -128.69, 170.23 59.45, 82.37 -93.38, 16.91 284.75, 80.98 -65.5, -15.92 in-in in 8.8752 Saltbr-in 2.4035 HRD-naA -68.35, -45.31 66.91, 0.56 in-in-in SNCiii in-in ActLoopNT-in 2.9161 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.63, 18.4 APE9-dihe-na -83.53, -173.89 APE8-dihe-in -74.3, 128.16 APE8-rot-in 308.34 APE67-dihe-in -66.79, -7.76 -58.38, -49.12 APE12-dist-in 9.4097 APE11-dist-in 8.6884 APE10-dist-in 5.159 APE9-dist-in 3.9453 None None None XRAY 2.0 0.213 0.239 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1ywv CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1XQZA P11309 32 308 313.0 No_ligand No_ligand Active DFGin 6.113 14.3232 BLAminus -132.59, 173.59 55.58, 88.87 -95.24, 18.48 288.46, 74.92 -59.23, -7.62 in-in in 8.4544 Saltbr-in 2.8339 HRD-naA -64.93, -53.25 74.7, 0.79 in-in-in SNCiii in-in ActLoopNT-in 2.8964 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.51, 32.32 APE9-dihe-na -92.62, -159.59 APE8-dihe-in -84.16, 115.96 APE8-rot-in 305.78 APE67-dihe-in -51.85, -11.5 -41.07, -65.14 APE12-dist-in 9.6322 APE11-dist-in 8.7408 APE10-dist-in 5.5845 APE9-dist-in 3.8829 None None None XRAY 2.1 0.249 0.297 A 300.0 277.0 0 26 26 0 [[38, 290]] 1.0 1xqz CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7VSYA P11309 33 305 313.0 No_ligand No_ligand Active DFGin 6.1466 14.8353 BLAminus -134.49, 172.31 56.25, 85.19 -90.8, 13.5 283.59, 75.74 -71.18, -5.96 in-in in 8.9886 Saltbr-in 2.572 HRD-naA -72.16, -48.61 72.01, 2.74 in-in-in SNCiii in-in ActLoopNT-in 2.8186 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.2, 35.54 APE9-dihe-na -94.69, -147.72 APE8-dihe-in -96.93, 120.22 APE8-rot-in 307.41 APE67-dihe-in -68.94, -11.56 -54.86, -45.03 APE12-dist-in 10.1896 APE11-dist-in 8.7411 APE10-dist-in 5.5966 APE9-dist-in 3.8972 N82K None None XRAY 2.141 0.198 0.22 A 326.0 273.0 0 26 26 0 [[38, 290]] 1.0 7vsy CAMK_PIM1_HUMAN CAMK 4.5e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4JX3A P11309 33 306 313.0 No_ligand No_ligand Active DFGin 6.2546 14.8623 BLAminus -127.82, 159.43 82.11, 81.67 -96.33, 22.05 278.91, 78.81 -66.22, -18.54 in-in in 9.0351 Saltbr-in 2.8635 HRD-naA -65.27, -47.76 69.76, -1.05 in-in-in SNCiii in-in ActLoopNT-in 2.647 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.67, 50.36 APE9-dihe-na -106.43, -151.13 APE8-dihe-in -91.89, 110.71 APE8-rot-in 312.27 APE67-dihe-in -55.41, -25.98 -43.33, -53.94 APE12-dist-in 9.6927 APE11-dist-in 8.5235 APE10-dist-in 5.6535 APE9-dist-in 4.0695 None None None XRAY 2.5 0.222 0.249 A 326.0 274.0 0 26 26 0 [[38, 290]] 1.0 4jx3 CAMK_PIM1_HUMAN CAMK 4.6e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7OOVA P11309 33 305 313.0 No_ligand No_ligand Active DFGin 6.203 14.5695 BLAminus -122.84, 171.74 65.68, 80.45 -90.31, 16.43 288.09, 76.06 -72.31, -11.34 in-in in 8.7995 Saltbr-in 2.608 HRD-naA -67.33, -47.42 68.65, 9.26 in-in-in SNCiii in-in ActLoopNT-in 2.8419 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.94, 17.29 APE9-dihe-na -81.04, -164.98 APE8-dihe-in -82.61, 126.44 APE8-rot-in 309.83 APE67-dihe-in -78.03, -5.17 -57.01, -47.48 APE12-dist-in 9.5122 APE11-dist-in 8.789 APE10-dist-in 5.4863 APE9-dist-in 3.8884 None None None XRAY 1.96 0.163 0.195 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 7oov CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7OOWA P11309 33 305 313.0 No_ligand No_ligand Active DFGin 6.3063 14.7477 BLAminus -122.68, 175.54 62.53, 73.89 -87.93, 12.78 283.68, 73.03 -76.55, -12.97 in-in in 8.7425 Saltbr-in 2.6023 HRD-naA -68.81, -49.98 73.35, 5.62 in-in-in SNCiii in-in ActLoopNT-in 2.9105 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.14, 32.43 APE9-dihe-na -87.5, -147.91 APE8-dihe-in -98.97, 121.57 APE8-rot-in 305.26 APE67-dihe-in -77.55, -5.21 -53.13, -44.92 APE12-dist-in 9.5933 APE11-dist-in 8.9762 APE10-dist-in 5.5753 APE9-dist-in 3.7722 None None None XRAY 1.95 0.161 0.184 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 7oow CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5TOEA P11309 34 306 313.0 7GK:401 Type1 Active DFGin 6.0724 14.6604 BLAminus -139.61, 170.18 66.65, 79.11 -92.13, 15.86 288.09, 73.32 -71.9, -3.59 in-in in 8.9752 Saltbr-in 2.649 HRD-naA -71.41, -51.31 74.77, 4.24 in-in-in SNCiii in-in ActLoopNT-in 2.7859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.61, 20.8 APE9-dihe-na -92.31, -158.45 APE8-dihe-in -81.21, 122.35 APE8-rot-in 309.79 APE67-dihe-in -65.59, -11.22 -66.85, -44.0 APE12-dist-in 9.6842 APE11-dist-in 8.6635 APE10-dist-in 5.3884 APE9-dist-in 3.9063 None None None XRAY 2.301 0.194 0.233 A 273.0 272.0 1 26 26 0 [[38, 290]] 1.0 5toe CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YHSA P11309 33 305 313.0 STU:306 Type1 Active DFGin 6.3607 14.5116 BLAminus -129.35, 165.16 65.09, 87.92 -99.2, 21.71 283.47, 69.45 -67.38, -11.76 in-in in 8.5242 Saltbr-in 2.8992 HRD-naA -65.05, -49.56 68.79, 3.6 in-in-in SNCiii in-in ActLoopNT-in 2.9031 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.4, 26.1 APE9-dihe-na -84.03, -156.82 APE8-dihe-in -85.78, 122.63 APE8-rot-in 304.34 APE67-dihe-in -62.69, -6.01 -56.85, -49.38 APE12-dist-in 9.327 APE11-dist-in 8.5203 APE10-dist-in 5.5084 APE9-dist-in 3.8321 None SEP261 CME161,SEP261 XRAY 2.15 0.233 0.233 A 273.0 269.0 4 26 26 0 [[38, 290]] 1.0 1yhs CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YI3A P11309 33 305 313.0 LY2:306 Type1 Active DFGin 6.2916 14.7641 BLAminus -128.81, 164.98 60.01, 85.31 -95.12, 30.71 287.86, 62.33 -66.19, -20.32 in-in in 7.7949 Saltbr-in 2.7333 HRD-naA -63.25, -48.22 66.78, 7.96 in-in-in SNCiii in-in ActLoopNT-in 2.8372 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.69, 36.2 APE9-dihe-na -99.79, -161.83 APE8-dihe-in -81.08, 117.39 APE8-rot-in 309.96 APE67-dihe-in -55.73, -11.01 -50.65, -56.8 APE12-dist-in 9.4522 APE11-dist-in 8.685 APE10-dist-in 5.2315 APE9-dist-in 4.0187 None SEP261 CME161,SEP261 XRAY 2.5 0.208 0.259 A 273.0 269.0 4 26 26 0 [[38, 290]] 1.0 1yi3 CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YI4A P11309 33 305 313.0 ADN:306 Type1 Active DFGin 6.0722 14.6981 BLAminus -134.71, 164.97 59.13, 80.78 -89.82, 21.93 287.09, 72.06 -64.68, -12.33 in-in in 8.788 Saltbr-in 2.7168 HRD-naA -68.53, -44.87 69.57, -1.62 in-in-in SNCiii in-in ActLoopNT-in 2.9339 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.9, 36.65 APE9-dihe-na -82.94, -132.28 APE8-dihe-in -114.84, 117.13 APE8-rot-in 309.09 APE67-dihe-in -54.56, -19.23 -51.71, -52.26 APE12-dist-in 9.605 APE11-dist-in 8.6743 APE10-dist-in 5.878 APE9-dist-in 4.1822 None SEP261 CME161,SEP261 XRAY 2.4 0.21 0.246 A 273.0 269.0 4 26 26 0 [[38, 290]] 1.0 1yi4 CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3C4EA P11309 33 305 313.0 C4E:306 Type1 Active DFGin 6.0215 14.7761 BLAminus -128.35, 166.0 69.48, 82.58 -93.7, 21.6 286.61, 78.83 -72.51, -9.22 in-in in 8.8865 Saltbr-in 2.7325 HRD-naA -67.91, -51.23 70.69, 5.52 in-in-in SNCiii in-in ActLoopNT-in 2.8123 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.94, 10.44 APE9-dihe-na -76.24, -163.31 APE8-dihe-in -81.86, 120.75 APE8-rot-in 311.66 APE67-dihe-in -66.61, -7.38 -59.14, -42.78 APE12-dist-in 9.659 APE11-dist-in 8.5496 APE10-dist-in 5.1757 APE9-dist-in 3.7908 None None None XRAY 1.98 0.216 0.245 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3c4e CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3C4EB P11309 33 305 313.0 C4E:306 Type1 Active DFGin 6.0749 14.7907 BLAminus -125.63, 166.99 68.65, 82.63 -92.11, 15.76 285.08, 79.16 -64.7, -9.12 in-in in 8.8733 Saltbr-in 2.9369 HRD-naA -73.69, -46.03 62.22, 13.94 in-in-in SNCiii in-in ActLoopNT-in 2.8715 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.74, 17.74 APE9-dihe-na -78.68, -151.78 APE8-dihe-in -92.25, 117.75 APE8-rot-in 301.9 APE67-dihe-in -69.85, -9.71 -53.08, -43.68 APE12-dist-in 9.7383 APE11-dist-in 8.5606 APE10-dist-in 5.43 APE9-dist-in 3.6989 None None None XRAY 1.98 0.216 0.245 B 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3c4e CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3C4EC P11309 34 305 313.0 C4E:306 Type1 Active DFGin 6.0604 14.7651 BLAminus -128.73, 171.78 61.45, 83.06 -93.51, 22.09 285.2, 77.36 -74.45, -9.29 in-in in 9.0241 Saltbr-in 2.46 HRD-naA -74.89, -48.06 74.46, 0.4 in-in-in SNCiii in-in ActLoopNT-in 2.9066 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.43, 22.53 APE9-dihe-na -88.97, -156.05 APE8-dihe-in -88.82, 119.66 APE8-rot-in 306.87 APE67-dihe-in -73.65, -3.54 -57.42, -41.13 APE12-dist-in 9.7009 APE11-dist-in 8.436 APE10-dist-in 5.1657 APE9-dist-in 3.9214 None None None XRAY 1.98 0.216 0.245 C 273.0 272.0 0 26 26 0 [[38, 290]] 1.0 3c4e CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3C4ED P11309 33 305 313.0 C4E:306 Type1 Active DFGin 6.3092 14.7094 BLAminus -130.13, 172.88 59.98, 79.45 -88.47, 15.36 281.95, 81.3 -75.02, -5.99 in-in in 8.7901 Saltbr-in 2.4435 HRD-naA -70.24, -47.69 69.35, 4.35 in-in-in SNCiii in-in ActLoopNT-in 2.8326 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.82, 22.76 APE9-dihe-na -80.15, -163.14 APE8-dihe-in -81.97, 115.05 APE8-rot-in 309.18 APE67-dihe-in -70.46, -13.8 -51.69, -41.7 APE12-dist-in 9.7262 APE11-dist-in 8.5833 APE10-dist-in 5.5064 APE9-dist-in 3.7583 None None None XRAY 1.98 0.216 0.245 D 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3c4e CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4K1BA P11309 33 305 313.0 1OC:402 Type1 Active DFGin 6.0427 14.6126 BLAminus -132.6, 164.86 70.11, 79.62 -92.82, 21.53 288.39, 81.35 -65.25, -17.96 in-in in 8.8563 Saltbr-in 2.6319 HRD-naA -70.69, -51.38 75.39, 5.68 in-in-in SNCiii in-in ActLoopNT-in 2.8194 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.17, 19.78 APE9-dihe-na -83.3, -161.37 APE8-dihe-in -81.98, 126.09 APE8-rot-in 308.93 APE67-dihe-in -65.14, -9.59 -61.45, -45.63 APE12-dist-in 9.5986 APE11-dist-in 8.6775 APE10-dist-in 5.2847 APE9-dist-in 3.8229 None None None XRAY 2.082 0.172 0.199 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 4k1b CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6NO8A P11309 33 305 313.0 KUY:401 Type1 Active DFGin 6.245 14.4648 BLAminus -136.93, 161.07 71.64, 80.45 -96.46, 11.0 281.89, 88.38 -60.27, -17.64 in-in in 8.6572 Saltbr-in 2.6047 HRD-naA -78.06, -49.34 70.05, 6.39 in-in-in SNCiii in-in ActLoopNT-in 2.8128 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.3, 11.35 APE9-dihe-na -78.95, -162.34 APE8-dihe-in -79.37, 127.44 APE8-rot-in 316.96 APE67-dihe-in -61.79, -7.22 -64.64, -48.15 APE12-dist-in 9.6679 APE11-dist-in 8.7765 APE10-dist-in 5.2156 APE9-dist-in 3.7941 None None None XRAY 2.377 0.187 0.232 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 6no8 CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6NO9A P11309 33 305 313.0 KUV:504 Type1 Active DFGin 6.1556 14.4327 BLAminus -126.34, 166.87 60.03, 83.92 -89.43, 21.76 289.02, 78.21 -70.19, -16.22 in-in in 8.6109 Saltbr-in 2.4384 HRD-naA -72.3, -46.64 69.8, 3.74 in-in-in SNCiii in-in ActLoopNT-in 2.8144 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.26, 10.84 APE9-dihe-na -76.6, -153.49 APE8-dihe-in -92.15, 125.02 APE8-rot-in 306.25 APE67-dihe-in -69.76, -6.68 -64.44, -39.96 APE12-dist-in 9.6794 APE11-dist-in 8.7289 APE10-dist-in 5.0813 APE9-dist-in 3.6717 None None None XRAY 1.712 0.17 0.205 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 6no9 CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4K0YA P11309 33 306 313.0 1OA:401 Type1 Active DFGin 6.292 14.3895 BLAminus -121.94, 171.4 62.4, 86.58 -95.92, 17.62 287.73, 79.01 -70.57, -9.06 in-in in 8.9044 Saltbr-in 2.5085 HRD-naA -73.78, -47.42 68.19, 7.19 in-in-in SNCiii in-in ActLoopNT-in 2.7966 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.37, 25.39 APE9-dihe-na -84.39, -155.13 APE8-dihe-in -90.58, 120.54 APE8-rot-in 303.27 APE67-dihe-in -71.06, -6.6 -61.16, -38.44 APE12-dist-in 9.6715 APE11-dist-in 8.6212 APE10-dist-in 5.5489 APE9-dist-in 3.6456 None None None XRAY 1.954 0.177 0.214 A 274.0 274.0 0 26 26 0 [[38, 290]] 1.0 4k0y CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5TELA P11309 33 306 313.0 7AJ:402 Type1 Active DFGin 6.1394 14.6282 BLAminus -138.92, 170.35 61.02, 78.29 -89.18, 17.43 286.77, 73.8 -69.83, -8.87 in-in in 8.9252 Saltbr-in 2.5481 HRD-naA -74.49, -48.42 69.85, 6.32 in-in-in SNCiii in-in ActLoopNT-in 2.8228 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.37, 35.58 APE9-dihe-na -94.48, -159.56 APE8-dihe-in -83.62, 124.38 APE8-rot-in 309.44 APE67-dihe-in -63.92, -12.31 -66.13, -42.06 APE12-dist-in 9.6957 APE11-dist-in 8.6914 APE10-dist-in 5.4702 APE9-dist-in 3.9726 None None None XRAY 2.214 0.182 0.207 A 274.0 273.0 1 26 26 0 [[38, 290]] 1.0 5tel CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5TEXA P11309 33 306 313.0 7AU:402 Type1 Active DFGin 6.0104 14.8294 BLAminus -138.39, 174.01 63.47, 82.62 -93.78, 16.92 290.32, 76.89 -70.47, -10.69 in-in in 9.269 Saltbr-in 2.8453 HRD-naA -75.68, -50.36 69.23, 7.58 in-in-in SNCiii in-in ActLoopNT-in 2.8374 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.29, 24.17 APE9-dihe-na -86.25, -152.07 APE8-dihe-in -90.77, 121.09 APE8-rot-in 307.82 APE67-dihe-in -67.29, -11.31 -64.01, -39.58 APE12-dist-in 9.6917 APE11-dist-in 8.5519 APE10-dist-in 5.4035 APE9-dist-in 3.8882 None None None XRAY 2.149 0.184 0.217 A 274.0 274.0 0 26 26 0 [[38, 290]] 1.0 5tex CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6VRUA P11309 34 306 313.0 ROY:402 Type1 Active DFGin 6.2493 14.7341 BLAminus -126.97, 167.03 70.01, 79.24 -93.65, 20.02 287.24, 69.33 -68.9, -13.34 in-in in 8.636 Saltbr-in 2.498 HRD-naA -74.69, -47.82 68.45, 8.0 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.88, 21.88 APE9-dihe-na -81.69, -157.22 APE8-dihe-in -91.46, 126.79 APE8-rot-in 307.71 APE67-dihe-in -66.96, -7.81 -67.63, -41.62 APE12-dist-in 9.5785 APE11-dist-in 8.5741 APE10-dist-in 5.2117 APE9-dist-in 3.7056 None None None XRAY 2.07 0.179 0.202 A 274.0 273.0 0 26 26 0 [[38, 290]] 1.0 6vru CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6VRVA P11309 35 305 313.0 WFY:401 Type1 Active DFGin 6.31 14.7748 BLAminus -128.18, 168.1 70.4, 82.6 -93.17, 16.82 287.59, 75.85 -67.39, -13.62 in-in in 8.7763 Saltbr-in 2.5274 HRD-naA -73.57, -42.57 66.05, 10.02 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.71, 32.21 APE9-dihe-na -87.53, -152.73 APE8-dihe-in -95.97, 120.66 APE8-rot-in 293.39 APE67-dihe-in -72.79, -2.49 -61.51, -35.74 APE12-dist-in 9.5715 APE11-dist-in 8.5796 APE10-dist-in 5.6753 APE9-dist-in 3.7577 None None None XRAY 1.74 0.173 0.197 A 274.0 271.0 0 26 26 0 [[38, 290]] 1.0 6vrv CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4DTKA P11309 33 305 313.0 7LI:408 Type1 Active DFGin 6.1421 14.6613 BLAminus -128.39, 173.69 63.23, 87.87 -95.85, 17.29 285.67, 80.15 -64.1, -18.22 in-in in 8.8606 Saltbr-in 2.5881 HRD-naA -66.25, -50.01 70.2, 5.45 in-in-in SNCiii in-in ActLoopNT-in 2.8698 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.52, 26.77 APE9-dihe-na -86.23, -154.0 APE8-dihe-in -89.22, 120.59 APE8-rot-in 306.1 APE67-dihe-in -65.85, -11.4 -53.32, -45.84 APE12-dist-in 9.7014 APE11-dist-in 8.5854 APE10-dist-in 5.4744 APE9-dist-in 3.6925 None None None XRAY 1.86 0.166 0.182 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 4dtk CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KGDA P11309 33 305 313.0 6SL:420 Type1 Active DFGin 6.1941 14.5978 BLAminus -129.0, 173.16 59.49, 81.21 -91.39, 15.51 283.61, 78.67 -67.75, -14.27 in-in in 8.8183 Saltbr-in 2.7249 HRD-naA -68.62, -47.74 69.23, 3.07 in-in-in SNCiii in-in ActLoopNT-in 2.8548 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.77, 31.72 APE9-dihe-na -89.5, -153.75 APE8-dihe-in -91.96, 121.37 APE8-rot-in 309.6 APE67-dihe-in -67.17, -11.15 -55.07, -44.24 APE12-dist-in 9.602 APE11-dist-in 8.6734 APE10-dist-in 5.6063 APE9-dist-in 3.7255 None None None XRAY 1.98 0.163 0.184 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgd CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KGEA P11309 33 305 313.0 6SN:416 Type1 Active DFGin 6.1855 14.6068 BLAminus -127.16, 171.98 58.94, 83.36 -93.06, 16.77 283.0, 80.17 -66.19, -15.51 in-in in 8.8007 Saltbr-in 2.6657 HRD-naA -68.2, -48.81 68.27, 3.74 in-in-in SNCiii in-in ActLoopNT-in 2.8389 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.87, 31.34 APE9-dihe-na -88.89, -156.61 APE8-dihe-in -88.29, 120.88 APE8-rot-in 311.55 APE67-dihe-in -66.51, -12.56 -54.59, -43.9 APE12-dist-in 9.6589 APE11-dist-in 8.6942 APE10-dist-in 5.6243 APE9-dist-in 3.7446 None None None XRAY 2.23 0.196 0.208 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kge CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KGGA P11309 33 305 313.0 6SO:423 Type1 Active DFGin 6.0952 14.601 BLAminus -129.17, 178.0 55.81, 74.89 -86.97, 13.61 281.87, 79.94 -67.04, -14.98 in-in in 8.9363 Saltbr-in 2.6656 HRD-naA -69.61, -46.82 68.9, 2.47 in-in-in SNCiii in-in ActLoopNT-in 2.883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.69, 27.94 APE9-dihe-na -86.85, -153.1 APE8-dihe-in -91.39, 121.35 APE8-rot-in 307.73 APE67-dihe-in -68.33, -11.23 -55.33, -42.82 APE12-dist-in 9.8085 APE11-dist-in 8.7335 APE10-dist-in 5.6043 APE9-dist-in 3.6841 None None None XRAY 1.95 0.159 0.17 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgg CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KGIA P11309 33 305 313.0 6SF:414 Type1 Active DFGin 6.1959 14.6781 BLAminus -128.85, 173.72 58.37, 80.83 -91.15, 15.65 283.15, 78.86 -67.29, -15.19 in-in in 8.8975 Saltbr-in 2.6991 HRD-naA -66.85, -48.52 69.49, 3.32 in-in-in SNCiii in-in ActLoopNT-in 2.8537 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.48, 30.3 APE9-dihe-na -88.67, -155.26 APE8-dihe-in -89.24, 121.14 APE8-rot-in 310.96 APE67-dihe-in -66.24, -12.88 -55.29, -44.34 APE12-dist-in 9.7233 APE11-dist-in 8.7346 APE10-dist-in 5.6424 APE9-dist-in 3.7397 None None None XRAY 2.13 0.173 0.186 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgi CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KGKA P11309 33 305 313.0 6SD:407 Type1 Active DFGin 6.3082 14.8602 BLAminus -128.4, 171.34 59.1, 83.1 -92.34, 16.26 283.46, 79.02 -66.84, -16.78 in-in in 8.9281 Saltbr-in 2.7226 HRD-naA -66.62, -48.72 69.73, 2.6 in-in-in SNCiii in-in ActLoopNT-in 2.8541 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.74, 32.55 APE9-dihe-na -90.23, -157.96 APE8-dihe-in -86.86, 120.62 APE8-rot-in 311.8 APE67-dihe-in -66.57, -13.56 -54.03, -44.15 APE12-dist-in 9.7032 APE11-dist-in 8.8498 APE10-dist-in 5.6821 APE9-dist-in 3.7634 None None None XRAY 2.66 0.188 0.206 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgk CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6BSKA P11309 33 305 313.0 MVG:405 Type1 Active DFGin 6.1061 14.5261 BLAminus -127.81, 171.26 61.28, 88.13 -94.14, 14.55 285.4, 81.12 -65.15, -15.23 in-in in 8.7334 Saltbr-in 2.6534 HRD-naA -65.0, -51.26 70.65, 3.06 in-in-in SNCiii in-in ActLoopNT-in 2.8175 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.1, 36.25 APE9-dihe-na -95.43, -156.67 APE8-dihe-in -85.65, 120.06 APE8-rot-in 311.62 APE67-dihe-in -68.39, -14.22 -55.35, -43.45 APE12-dist-in 9.8022 APE11-dist-in 8.5486 APE10-dist-in 5.6356 APE9-dist-in 3.7924 None None None XRAY 2.573 0.171 0.196 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 6bsk CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4K18A P11309 32 308 313.0 1OB:402 Type1 Active DFGin 6.0917 14.4411 BLAminus -127.16, 170.25 67.68, 77.49 -90.65, 24.19 290.3, 84.83 -68.81, -16.15 in-in in 8.7657 Saltbr-in 2.6128 HRD-naA -73.4, -51.44 75.59, 3.74 in-in-in SNCiii in-in ActLoopNT-in 2.8538 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.67, 18.39 APE9-dihe-na -83.8, -157.76 APE8-dihe-in -87.59, 123.77 APE8-rot-in 308.05 APE67-dihe-in -70.86, -5.11 -63.89, -39.96 APE12-dist-in 9.7914 APE11-dist-in 8.8029 APE10-dist-in 5.401 APE9-dist-in 3.9252 None None None XRAY 2.051 0.186 0.22 A 277.0 277.0 0 26 26 0 [[38, 290]] 1.0 4k18 CAMK_PIM1_HUMAN CAMK 2.6e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5IISA P11309 32 305 313.0 6CB:402 Type1 Active DFGin 6.3878 14.7567 BLAminus -128.84, 173.3 61.28, 84.09 -98.54, 16.15 284.91, 73.79 -69.44, -13.21 in-in in 8.2803 Saltbr-in 2.7008 HRD-naA -69.32, -50.23 68.69, 7.8 in-in-in SNCiii in-in ActLoopNT-in 2.9101 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.03, 27.99 APE9-dihe-na -88.44, -153.73 APE8-dihe-in -93.14, 121.31 APE8-rot-in 307.37 APE67-dihe-in -67.36, -12.92 -53.81, -44.97 APE12-dist-in 9.4712 APE11-dist-in 8.5316 APE10-dist-in 5.2689 APE9-dist-in 3.6397 None SEP261 SEP261 XRAY 2.1 0.172 0.193 A 277.0 274.0 0 26 26 0 [[38, 290]] 1.0 5iis CAMK_PIM1_HUMAN CAMK 2.6e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4TY1A P11309 33 305 313.0 38W:401 Type1 Active DFGin 6.387 14.5113 BLAminus -133.05, 165.34 66.19, 78.61 -90.98, 18.04 289.04, 69.92 -66.35, -17.07 in-in in 8.0757 Saltbr-in 2.8545 HRD-naA -75.5, -52.3 76.47, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.8796 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.39, -3.83 APE9-dihe-na -80.99, -152.88 APE8-dihe-in -92.77, 125.02 APE8-rot-in 308.7 APE67-dihe-in -59.27, -21.7 -50.58, -57.32 APE12-dist-in 9.5504 APE11-dist-in 8.7416 APE10-dist-in 4.3675 APE9-dist-in 3.6288 None None None XRAY 2.7 0.183 0.237 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4ty1 CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4WRSA P11309 33 305 313.0 3U1:403 Type1 Active DFGin 6.1624 14.6882 BLAminus -131.19, 168.19 62.17, 84.39 -94.94, 19.3 284.32, 75.21 -73.2, -12.05 in-in in 8.9033 Saltbr-in 2.6155 HRD-naA -70.39, -48.07 69.42, 8.56 in-in-in SNCiii in-in ActLoopNT-in 2.9235 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.6, 16.03 APE9-dihe-na -86.28, -152.26 APE8-dihe-in -92.85, 128.8 APE8-rot-in 308.26 APE67-dihe-in -65.67, -10.81 -62.91, -47.38 APE12-dist-in 9.4769 APE11-dist-in 8.6179 APE10-dist-in 4.9364 APE9-dist-in 3.7627 None None None XRAY 2.2 0.18 0.208 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4wrs CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4WSYA P11309 33 305 313.0 3U5:401 Type1 Active DFGin 6.1044 14.6207 BLAminus -127.31, -178.18 57.57, 65.12 -84.25, 18.54 286.02, 73.35 -69.75, -14.58 in-in in 8.9086 Saltbr-in 2.7849 HRD-naA -70.92, -47.77 70.77, 0.48 in-in-in SNCiii in-in ActLoopNT-in 2.9139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.56, 17.45 APE9-dihe-na -80.04, -158.16 APE8-dihe-in -87.23, 129.67 APE8-rot-in 306.6 APE67-dihe-in -63.98, -11.76 -66.05, -47.25 APE12-dist-in 9.5 APE11-dist-in 8.5775 APE10-dist-in 5.3469 APE9-dist-in 3.7953 None None None XRAY 2.3 0.184 0.224 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4wsy CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4WT6A P11309 33 305 313.0 3U6:401 Type1 Active DFGin 6.2247 14.7413 BLAminus -129.31, 179.15 54.14, 72.7 -88.4, 20.56 284.51, 71.19 -73.36, -15.22 in-in in 8.4691 Saltbr-in 2.6562 HRD-naA -72.36, -44.25 65.88, 2.27 in-in-in SNCiii in-in ActLoopNT-in 2.9723 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.26, 22.96 APE9-dihe-na -91.6, -154.03 APE8-dihe-in -92.19, 127.1 APE8-rot-in 312.31 APE67-dihe-in -65.83, -13.24 -60.93, -48.29 APE12-dist-in 9.496 APE11-dist-in 8.6131 APE10-dist-in 5.0588 APE9-dist-in 3.9979 None None None XRAY 2.3 0.178 0.211 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4wt6 CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5EOLA P11309 33 305 313.0 5QO:401 Type1 Active DFGin 6.2561 14.6307 BLAminus -125.24, 171.83 59.51, 79.96 -92.44, 22.49 285.02, 73.25 -70.93, -14.06 in-in in 8.7627 Saltbr-in 2.5732 HRD-naA -73.1, -47.95 68.92, 3.14 in-in-in SNCiii in-in ActLoopNT-in 2.8417 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.99, 8.97 APE9-dihe-na -79.78, -148.56 APE8-dihe-in -97.04, 122.04 APE8-rot-in 309.05 APE67-dihe-in -66.69, -11.1 -58.67, -42.55 APE12-dist-in 9.5827 APE11-dist-in 8.513 APE10-dist-in 4.9128 APE9-dist-in 3.6325 None None None XRAY 2.2 0.196 0.223 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 5eol CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5IPJA P11309 33 305 313.0 6CD:401 Type1 Active DFGin 6.1587 14.6449 BLAminus -129.06, 166.2 63.4, 89.79 -98.28, 24.16 286.53, 74.98 -69.52, -15.68 in-in in 8.8615 Saltbr-in 2.6437 HRD-naA -72.25, -47.9 67.86, 13.58 in-in-in SNCiii in-in ActLoopNT-in 2.8528 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.03, 18.83 APE9-dihe-na -86.4, -154.92 APE8-dihe-in -92.64, 123.62 APE8-rot-in 306.86 APE67-dihe-in -66.21, -11.28 -62.03, -43.15 APE12-dist-in 9.5154 APE11-dist-in 8.5252 APE10-dist-in 4.9669 APE9-dist-in 3.5939 None None None XRAY 2.1 0.181 0.221 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 5ipj CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KZIA P11309 33 305 313.0 6YN:401 Type1 Active DFGin 6.2318 14.4593 BLAminus -125.28, 171.61 59.7, 76.37 -89.66, 23.41 287.5, 74.51 -76.32, -14.48 in-in in 8.5633 Saltbr-in 2.6219 HRD-naA -74.51, -47.69 70.34, 4.33 in-in-in SNCiii in-in ActLoopNT-in 2.7817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.16, 14.87 APE9-dihe-na -85.38, -150.81 APE8-dihe-in -98.45, 122.78 APE8-rot-in 307.97 APE67-dihe-in -69.43, -12.03 -61.1, -42.73 APE12-dist-in 9.6227 APE11-dist-in 8.7118 APE10-dist-in 4.9438 APE9-dist-in 3.8102 None None None XRAY 2.1 0.179 0.205 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kzi CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6MT0A P11309 33 305 313.0 JYG:401 Type1 Active DFGin 6.1797 14.6437 BLAminus -129.1, 162.88 69.48, 92.17 -101.8, 22.17 287.32, 75.1 -69.24, -17.14 in-in in 8.6669 Saltbr-in 2.7291 HRD-naA -70.67, -47.42 66.78, 12.82 in-in-in SNCiii in-in ActLoopNT-in 2.8517 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -118.16, 8.39 APE9-dihe-na -79.87, -163.75 APE8-dihe-in -86.85, 127.4 APE8-rot-in 308.59 APE67-dihe-in -66.88, -11.27 -60.5, -47.04 APE12-dist-in 9.3772 APE11-dist-in 8.5534 APE10-dist-in 4.6116 APE9-dist-in 3.5443 None None None XRAY 2.2 0.18 0.208 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 6mt0 CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4MTAA P11309 33 305 313.0 2D2:401 Type1 Active DFGin 6.2759 14.3366 BLAminus -121.41, 177.86 55.53, 82.62 -93.46, 16.76 281.52, 74.78 -72.09, -10.86 in-in in 8.719 Saltbr-in 2.6113 HRD-naA -62.2, -48.48 67.49, 3.7 in-in-in SNCiii in-in ActLoopNT-in 2.7947 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.11, 24.3 APE9-dihe-na -85.34, -152.54 APE8-dihe-in -92.96, 123.11 APE8-rot-in 306.26 APE67-dihe-in -67.9, -13.27 -54.99, -44.77 APE12-dist-in 9.5277 APE11-dist-in 8.5158 APE10-dist-in 5.416 APE9-dist-in 3.5754 None None None XRAY 2.2 0.16 0.192 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4mta CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5C1QB P11309 33 305 313.0 4YK:401 Type1 Active DFGin 5.891 13.333 BLAminus -134.33, 156.38 72.1, 106.74 -112.64, 17.25 301.94, 90.76 -59.71, -41.8 in-in in 8.6215 Saltbr-in 2.5933 HRD-naA -64.46, -50.63 69.52, -24.55 in-in-in SNCiii in-in ActLoopNT-in 2.8007 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.39, 56.57 APE9-dihe-na -121.47, -173.24 APE8-dihe-in -77.48, 148.97 APE8-rot-in 348.38 APE67-dihe-in -42.36, -34.75 -61.79, -66.84 APE12-dist-in 9.4062 APE11-dist-in 8.2515 APE10-dist-in 5.3773 APE9-dist-in 4.9262 None None None XRAY 3.0 0.178 0.246 B 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 5c1q CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L11A P11309 33 305 313.0 E2C:401 Type1 Active DFGin 6.1626 14.9671 BLAminus -125.67, 168.03 67.88, 78.16 -84.6, 16.39 285.76, 87.64 -71.05, -19.61 in-in in 8.9964 Saltbr-in 2.7022 HRD-naA -66.89, -52.69 70.36, 8.44 in-in-in SNCiii in-in ActLoopNT-in 2.767 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.89, 29.6 APE9-dihe-na -84.12, -156.34 APE8-dihe-in -92.4, 128.66 APE8-rot-in 306.74 APE67-dihe-in -67.11, -6.47 -60.7, -48.56 APE12-dist-in 9.3558 APE11-dist-in 8.3863 APE10-dist-in 5.4313 APE9-dist-in 3.7089 None SEP261 SEP261 XRAY 2.05 0.214 0.24 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l11 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L12A P11309 33 305 313.0 E2R:401 Type1 Active DFGin 6.2158 14.7026 BLAminus -127.05, 170.42 68.23, 81.09 -92.51, 16.44 287.76, 81.55 -64.97, -20.04 in-in in 8.983 Saltbr-in 2.7221 HRD-naA -72.18, -48.09 70.82, 3.37 in-in-in SNCiii in-in ActLoopNT-in 2.8382 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.36, 18.6 APE9-dihe-na -85.64, -160.05 APE8-dihe-in -87.61, 125.01 APE8-rot-in 307.11 APE67-dihe-in -68.37, -12.11 -58.28, -46.28 APE12-dist-in 9.3781 APE11-dist-in 8.5814 APE10-dist-in 5.0596 APE9-dist-in 3.8326 None SEP261 SEP261 XRAY 1.87 0.197 0.21 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l12 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L13A P11309 33 305 313.0 E2F:401 Type1 Active DFGin 6.1902 14.7858 BLAminus -130.24, 168.2 68.46, 80.68 -89.17, 16.05 288.1, 80.31 -69.01, -19.61 in-in in 9.1055 Saltbr-in 2.9362 HRD-naA -68.46, -51.8 71.9, 8.52 in-in-in SNCiii in-in ActLoopNT-in 2.7778 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.76, 29.56 APE9-dihe-na -92.34, -153.25 APE8-dihe-in -98.43, 124.2 APE8-rot-in 303.55 APE67-dihe-in -68.48, -12.49 -58.68, -45.06 APE12-dist-in 9.5 APE11-dist-in 8.5109 APE10-dist-in 5.0987 APE9-dist-in 3.6586 None SEP261 SEP261 XRAY 2.24 0.18 0.214 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l13 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L14A P11309 33 305 313.0 E2L:401 Type1 Active DFGin 6.2009 14.8938 BLAminus -126.69, 169.11 67.27, 79.53 -86.62, 19.33 288.75, 82.28 -66.99, -22.84 in-in in 9.0448 Saltbr-in 2.8364 HRD-naA -67.72, -50.1 68.21, 9.79 in-in-in SNCiii in-in ActLoopNT-in 2.8055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.83, 24.46 APE9-dihe-na -89.25, -158.62 APE8-dihe-in -92.28, 125.41 APE8-rot-in 306.06 APE67-dihe-in -68.05, -12.07 -60.25, -45.14 APE12-dist-in 9.5091 APE11-dist-in 8.5175 APE10-dist-in 5.0735 APE9-dist-in 3.7712 None SEP261 SEP261 XRAY 1.95 0.193 0.209 A 289.0 271.0 2 26 26 0 [[38, 290]] 1.0 6l14 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L15A P11309 33 305 313.0 E2O:401 Type1 Active DFGin 6.3499 14.598 BLAminus -131.83, 163.47 71.59, 79.35 -89.78, 14.2 284.41, 77.37 -65.48, -21.82 in-in in 8.235 Saltbr-in 2.5656 HRD-naA -64.16, -54.27 75.51, 4.04 in-in-in SNCiii in-in ActLoopNT-in 2.7413 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.69, 27.17 APE9-dihe-na -98.51, -154.05 APE8-dihe-in -93.58, 128.93 APE8-rot-in 316.57 APE67-dihe-in -60.96, -21.44 -58.79, -53.8 APE12-dist-in 9.4071 APE11-dist-in 8.6356 APE10-dist-in 4.9291 APE9-dist-in 3.916 None SEP261 SEP261 XRAY 2.6 0.184 0.221 A 289.0 270.0 3 26 26 0 [[38, 290]] 1.0 6l15 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L16A P11309 33 305 313.0 E2U:401 Type1 Active DFGin 6.3278 14.74 BLAminus -130.86, 166.29 65.26, 82.88 -91.87, 18.01 283.01, 76.97 -72.19, -13.53 in-in in 8.7021 Saltbr-in 2.4147 HRD-naA -67.28, -47.47 67.45, 11.65 in-in-in SNCiii in-in ActLoopNT-in 2.8263 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.92, 16.39 APE9-dihe-na -84.74, -155.75 APE8-dihe-in -95.92, 129.43 APE8-rot-in 310.51 APE67-dihe-in -64.98, -15.76 -62.83, -46.58 APE12-dist-in 9.3102 APE11-dist-in 8.5215 APE10-dist-in 4.7385 APE9-dist-in 3.7782 None SEP261 SEP261 XRAY 2.1 0.199 0.218 A 289.0 270.0 3 26 26 0 [[38, 290]] 1.0 6l16 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6L17A P11309 33 305 313.0 E2X:401 Type1 Active DFGin 6.3235 14.6531 BLAminus -129.55, 165.34 65.87, 81.97 -92.53, 17.46 286.99, 73.6 -66.81, -14.75 in-in in 8.3978 Saltbr-in 2.601 HRD-naA -68.49, -49.87 68.95, 13.18 in-in-in SNCiii in-in ActLoopNT-in 2.8216 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.96, 18.29 APE9-dihe-na -82.73, -153.32 APE8-dihe-in -94.04, 120.15 APE8-rot-in 303.42 APE67-dihe-in -68.29, -9.26 -56.68, -41.93 APE12-dist-in 9.5105 APE11-dist-in 8.5589 APE10-dist-in 5.2242 APE9-dist-in 3.7004 None SEP261 SEP261 XRAY 1.75 0.185 0.205 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l17 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7XSVA P11309 32 305 313.0 I4M:401 Type1 Active DFGin 6.058 14.3167 BLAminus -136.35, 175.71 54.46, 80.4 -90.61, 15.51 289.45, 76.26 -61.12, -29.45 in-in in 8.1673 Saltbr-in 2.4868 HRD-naA -80.1, -41.91 69.45, -9.52 in-in-in SNCiii in-in ActLoopNT-in 2.7914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.82, 18.64 APE9-dihe-na -91.64, 171.14 APE8-dihe-in -71.59, 144.23 APE8-rot-in 295.24 APE67-dihe-in -74.83, -31.12 -57.05, -23.4 APE12-dist-in 8.859 APE11-dist-in 8.4261 APE10-dist-in 4.6305 APE9-dist-in 4.8183 None SEP261 SEP261 XRAY 2.66 0.197 0.233 A 289.0 274.0 0 26 26 0 [[38, 290]] 1.0 7xsv CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5KCXA P11309 34 305 313.0 6S3:403 Type1 Active DFGin 6.2209 14.9168 BLAminus -132.88, 167.48 63.01, 80.22 -91.16, 17.8 283.48, 68.85 -71.72, -7.39 in-in in 8.8485 Saltbr-in 2.5228 HRD-naA -73.28, -48.22 75.07, 1.67 in-in-in SNCiii in-in ActLoopNT-in 2.8307 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.64, 15.26 APE9-dihe-na -83.36, -157.62 APE8-dihe-in -86.75, 121.87 APE8-rot-in 307.36 APE67-dihe-in -65.54, -9.34 -59.93, -45.42 APE12-dist-in 9.6483 APE11-dist-in 8.6086 APE10-dist-in 5.2518 APE9-dist-in 3.8637 None None None XRAY 2.2 0.19 0.211 A 291.0 272.0 0 26 26 0 [[38, 290]] 1.0 5kcx CAMK_PIM1_HUMAN CAMK 3.1e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4MBIA P11309 33 306 313.0 26K:401 Type1 Active DFGin 6.1239 14.4723 BLAminus -131.89, 168.18 61.53, 68.36 -79.59, 15.15 287.22, 79.02 -64.78, -12.91 in-in in 8.6887 Saltbr-in 2.7726 HRD-naA -75.96, -48.7 66.71, 16.19 in-in-in SNCiii in-in ActLoopNT-in 2.7522 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.73, 31.55 APE9-dihe-na -87.7, -149.18 APE8-dihe-in -95.91, 132.2 APE8-rot-in 306.67 APE67-dihe-in -76.77, -11.58 -65.7, -39.07 APE12-dist-in 9.5635 APE11-dist-in 8.4731 APE10-dist-in 5.1024 APE9-dist-in 3.6425 None None None XRAY 2.3 0.215 0.246 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 4mbi CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4MBLA P11309 33 306 313.0 26L:401 Type1 Active DFGin 6.3571 14.6471 BLAminus -140.97, 162.32 61.82, 87.23 -100.32, 23.61 288.64, 85.04 -75.88, -10.71 in-in in 8.4627 Saltbr-in 2.705 HRD-naA -66.61, -53.32 68.87, 14.83 in-in-in SNCiii in-in ActLoopNT-in 2.7923 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.99, 40.01 APE9-dihe-na -114.3, -171.32 APE8-dihe-in -75.76, 118.27 APE8-rot-in 314.72 APE67-dihe-in -58.14, -19.65 -55.56, -49.63 APE12-dist-in 9.0327 APE11-dist-in 8.6582 APE10-dist-in 4.8819 APE9-dist-in 4.1912 None None None XRAY 2.6 0.202 0.242 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 4mbl CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXVA P11309 33 306 313.0 LI6:323 Type1 Active DFGin 6.1534 14.6197 BLAminus -131.19, 171.32 56.28, 85.76 -94.29, 14.73 284.91, 75.06 -64.34, -11.63 in-in in 8.8928 Saltbr-in 2.5423 HRD-naA -66.61, -47.26 65.08, 9.89 in-in-in SNCiii in-in ActLoopNT-in 2.9207 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.55, 31.12 APE9-dihe-na -89.85, -157.25 APE8-dihe-in -87.05, 122.1 APE8-rot-in 305.25 APE67-dihe-in -67.3, -11.88 -57.54, -43.12 APE12-dist-in 9.6965 APE11-dist-in 8.4898 APE10-dist-in 5.4378 APE9-dist-in 3.7355 None None None XRAY 2.0 0.189 0.211 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxv CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1YXXA P11309 33 306 313.0 LI7:323 Type1 Active DFGin 6.1644 14.4349 BLAminus -118.82, 172.49 62.96, 83.76 -93.84, 24.35 282.94, 80.67 -77.24, -2.76 in-in in 8.8737 Saltbr-in 2.4462 HRD-naA -72.3, -43.39 62.78, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.9232 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.23, 43.27 APE9-dihe-na -100.31, -154.93 APE8-dihe-in -89.78, 124.47 APE8-rot-in 309.92 APE67-dihe-in -69.42, -9.61 -60.64, -40.01 APE12-dist-in 9.7437 APE11-dist-in 8.4051 APE10-dist-in 5.643 APE9-dist-in 3.8007 None None None XRAY 2.0 0.219 0.251 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxx CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2O3PA P11309 33 306 313.0 QUE:501 Type1 Active DFGin 6.2383 14.5362 BLAminus -130.88, 170.78 53.54, 90.02 -97.28, 20.48 282.33, 78.83 -71.95, -12.75 in-in in 8.6674 Saltbr-in 2.2959 HRD-naA -68.04, -46.2 63.08, 8.81 in-in-in SNCiii in-in ActLoopNT-in 2.8581 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.42, 29.49 APE9-dihe-na -90.86, -153.23 APE8-dihe-in -86.96, 125.45 APE8-rot-in 306.17 APE67-dihe-in -64.91, -8.64 -61.09, -46.67 APE12-dist-in 9.6614 APE11-dist-in 8.5306 APE10-dist-in 5.4294 APE9-dist-in 3.8478 None None None XRAY 2.24 0.189 0.22 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o3p CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2O63A P11309 33 306 313.0 MYC:501 Type1 Active DFGin 6.0925 14.4288 BLAminus -133.37, 172.38 63.28, 75.17 -88.32, 15.11 286.1, 77.55 -67.51, -7.66 in-in in 8.5833 Saltbr-in 2.552 HRD-naA -71.09, -45.59 61.3, 13.27 in-in-in SNCiii in-in ActLoopNT-in 2.9029 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.73, 31.74 APE9-dihe-na -90.0, -152.24 APE8-dihe-in -91.1, 122.3 APE8-rot-in 305.54 APE67-dihe-in -66.75, -10.3 -56.16, -45.71 APE12-dist-in 9.8969 APE11-dist-in 8.6251 APE10-dist-in 5.6381 APE9-dist-in 3.7828 None None None XRAY 2.0 0.194 0.218 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o63 CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2O64A P11309 33 306 313.0 MYU:501 Type1 Active DFGin 6.2715 14.6755 BLAminus -128.75, 172.17 61.57, 79.87 -92.44, 15.52 285.23, 76.88 -62.99, -16.57 in-in in 8.4121 Saltbr-in 2.672 HRD-naA -65.21, -51.23 71.84, 4.17 in-in-in SNCiii in-in ActLoopNT-in 2.9535 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.67, 34.14 APE9-dihe-na -99.78, -147.67 APE8-dihe-in -92.72, 124.85 APE8-rot-in 309.85 APE67-dihe-in -64.3, -15.3 -61.26, -48.06 APE12-dist-in 9.6056 APE11-dist-in 8.584 APE10-dist-in 5.4192 APE9-dist-in 3.9479 None None None XRAY 2.44 0.191 0.23 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o64 CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2O65A P11309 33 306 313.0 MYF:501 Type1 Active DFGin 5.7731 14.2228 BLAminus -134.9, 170.04 60.08, 89.22 -101.35, 10.62 287.34, 92.73 -63.96, -9.9 in-in in 8.7039 Saltbr-in 2.4715 HRD-naA -65.14, -47.59 70.03, -4.07 in-in-in SNCiii in-in ActLoopNT-in 2.9803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.66, 34.64 APE9-dihe-na -104.35, -148.26 APE8-dihe-in -83.11, 121.1 APE8-rot-in 316.59 APE67-dihe-in -62.15, -16.44 -57.04, -47.52 APE12-dist-in 9.9881 APE11-dist-in 8.6279 APE10-dist-in 5.2887 APE9-dist-in 4.1355 None None None XRAY 2.85 0.21 0.262 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o65 CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3JXWA P11309 33 306 313.0 LXG:1000 Type1 Active DFGin 6.2103 14.5966 BLAminus -134.41, 162.67 73.18, 86.78 -94.42, 16.28 283.72, 78.67 -67.2, -7.05 in-in in 8.9431 Saltbr-in 2.7638 HRD-naA -66.64, -45.65 67.32, 6.42 in-in-in SNCiii in-in ActLoopNT-in 2.7858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.1, 39.58 APE9-dihe-na -109.74, -153.05 APE8-dihe-in -85.54, 118.8 APE8-rot-in 317.48 APE67-dihe-in -60.88, -20.58 -50.76, -58.31 APE12-dist-in 9.5275 APE11-dist-in 8.5452 APE10-dist-in 5.4917 APE9-dist-in 4.2563 None None None XRAY 2.8 0.219 0.266 A 294.0 274.0 0 26 26 0 [[38, 290]] 1.0 3jxw CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3JY0A P11309 33 307 313.0 LYG:1000 Type1 Active DFGin 5.9655 14.4592 BLAminus -136.0, 169.05 67.14, 86.13 -88.57, 12.42 285.25, 84.28 -62.59, -9.01 in-in in 8.897 Saltbr-in 2.5785 HRD-naA -73.59, -52.32 72.38, 9.82 in-in-in SNCiii in-in ActLoopNT-in 2.7783 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.33, 17.31 APE9-dihe-na -90.28, -146.77 APE8-dihe-in -93.89, 122.92 APE8-rot-in 318.19 APE67-dihe-in -68.56, -0.09 -56.36, -49.84 APE12-dist-in 9.7621 APE11-dist-in 8.4913 APE10-dist-in 4.9707 APE9-dist-in 3.8014 None None None XRAY 2.4 0.226 0.257 A 294.0 275.0 0 26 26 0 [[38, 290]] 1.0 3jy0 CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3JYAA P11309 33 306 313.0 LWG:1000 Type1 Active DFGin 6.2096 14.5113 BLAminus -132.92, 173.52 45.25, 85.32 -90.21, 14.37 285.74, 75.57 -67.67, -13.84 in-in in 9.0619 Saltbr-in 2.4726 HRD-naA -71.42, -47.46 64.92, 10.13 in-in-in SNCiii in-in ActLoopNT-in 2.7063 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.34, 26.83 APE9-dihe-na -88.37, -156.09 APE8-dihe-in -89.17, 119.95 APE8-rot-in 305.54 APE67-dihe-in -68.16, -12.31 -55.92, -42.85 APE12-dist-in 9.5401 APE11-dist-in 8.4965 APE10-dist-in 5.3913 APE9-dist-in 3.7507 None None None XRAY 2.1 0.234 0.257 A 294.0 274.0 0 26 26 0 [[38, 290]] 1.0 3jya CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5O11A P11309 34 305 313.0 3NG:401 Type1 Active DFGin 6.1285 14.6109 BLAminus -127.88, 174.91 62.14, 80.5 -88.8, 17.09 290.86, 80.03 -61.06, -19.7 in-in in 8.8564 Saltbr-in 2.6066 HRD-naA -68.12, -50.16 69.42, 1.48 in-in-in SNCiii in-in ActLoopNT-in 2.8771 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.35, 8.9 APE9-dihe-na -86.78, -150.83 APE8-dihe-in -93.81, 133.37 APE8-rot-in 308.93 APE67-dihe-in -69.86, -10.11 -67.48, -44.09 APE12-dist-in 9.7422 APE11-dist-in 8.7304 APE10-dist-in 4.8611 APE9-dist-in 3.817 None SEP261 CME161,SEP261 XRAY 2.4 0.167 0.212 A 298.0 270.0 2 26 26 0 [[38, 290]] 1.0 5o11 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5O12A P11309 34 305 313.0 1RO:401 Type1 Active DFGin 6.2318 14.4999 BLAminus -126.26, 172.57 61.88, 84.82 -89.13, 24.53 288.01, 80.82 -77.95, -15.0 in-in in 8.881 Saltbr-in 2.7 HRD-naA -70.16, -50.1 71.34, 2.69 in-in-in SNCiii in-in ActLoopNT-in 2.8956 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.86, 30.76 APE9-dihe-na -86.98, -148.45 APE8-dihe-in -99.72, 127.71 APE8-rot-in 312.69 APE67-dihe-in -67.78, -9.89 -65.97, -45.8 APE12-dist-in 9.5158 APE11-dist-in 8.4456 APE10-dist-in 5.6506 APE9-dist-in 3.7177 None SEP261 CME161,SEP261 XRAY 2.4 0.179 0.223 A 298.0 266.0 6 26 26 0 [[38, 290]] 1.0 5o12 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5O13A P11309 34 305 313.0 9G5:401 Type1 Active DFGin 6.232 14.5703 BLAminus -126.22, 173.43 61.18, 82.34 -90.65, 15.63 288.81, 77.08 -66.25, -16.88 in-in in 8.8079 Saltbr-in 2.6206 HRD-naA -66.53, -48.7 66.86, 2.99 in-in-in SNCiii in-in ActLoopNT-in 2.8173 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.42, 11.87 APE9-dihe-na -70.23, -134.62 APE8-dihe-in -110.38, 131.64 APE8-rot-in 317.06 APE67-dihe-in -70.9, -10.23 -68.47, -45.42 APE12-dist-in 9.6816 APE11-dist-in 8.5431 APE10-dist-in 5.4383 APE9-dist-in 4.0623 None SEP261 CSX161,SEP261 XRAY 2.44 0.162 0.214 A 298.0 272.0 0 26 26 0 [[38, 290]] 1.0 5o13 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5DGZA P11309 33 305 313.0 L20:401 Type1 Active DFGin 6.3283 14.8412 BLAminus -128.71, 169.75 60.97, 88.72 -102.55, 22.85 284.63, 77.63 -73.84, -14.69 in-in in 8.5704 Saltbr-in 2.5393 HRD-naA -79.61, -44.74 68.32, 8.97 in-in-in SNCiii in-in ActLoopNT-in 2.9586 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.12, 19.6 APE9-dihe-na -84.49, -168.79 APE8-dihe-in -78.12, 137.4 APE8-rot-in 353.29 APE67-dihe-in -67.56, -8.39 -54.96, -54.27 APE12-dist-in 9.4821 APE11-dist-in 8.7924 APE10-dist-in 5.0905 APE9-dist-in 3.8694 None None None XRAY 2.502 0.182 0.213 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5dgz CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5DHJA P11309 33 305 313.0 5E5:401 Type1 Active DFGin 6.2772 14.6413 BLAminus -132.48, 165.98 68.77, 75.26 -89.6, 23.34 285.29, 75.18 -66.63, -15.53 in-in in 8.6776 Saltbr-in 2.5997 HRD-naA -74.9, -49.69 73.89, 5.62 in-in-in SNCiii in-in ActLoopNT-in 2.8008 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.14, 28.7 APE9-dihe-na -93.46, -149.0 APE8-dihe-in -88.51, 125.57 APE8-rot-in 319.11 APE67-dihe-in -63.27, -9.53 -60.93, -48.3 APE12-dist-in 9.6899 APE11-dist-in 8.7094 APE10-dist-in 5.5758 APE9-dist-in 3.8895 None None None XRAY 2.457 0.191 0.25 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5dhj CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5DIAA P11309 33 305 313.0 5E6:401 Type1 Active DFGin 6.1094 14.3642 BLAminus -131.51, 162.73 65.64, 95.79 -106.0, 22.43 288.31, 75.68 -70.61, -13.53 in-in in 8.8932 Saltbr-in 2.6632 HRD-naA -70.21, -53.43 79.23, -0.98 in-in-in SNCiii in-in ActLoopNT-in 2.8151 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.54, 25.72 APE9-dihe-na -78.57, -156.72 APE8-dihe-in -91.47, 121.1 APE8-rot-in 309.49 APE67-dihe-in -70.58, -6.62 -58.72, -40.2 APE12-dist-in 9.6002 APE11-dist-in 8.6495 APE10-dist-in 5.4875 APE9-dist-in 3.7674 None None None XRAY 1.964 0.198 0.229 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5dia CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5V80A P11309 33 305 313.0 971:402 Type1 Active DFGin 6.2933 14.711 BLAminus -125.21, 168.1 67.15, 84.62 -97.5, 21.56 283.85, 73.58 -74.5, -9.73 in-in in 8.8229 Saltbr-in 2.4892 HRD-naA -71.2, -48.76 73.46, -4.54 in-in-in SNCiii in-in ActLoopNT-in 2.8494 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 17.28 APE9-dihe-na -81.45, -156.95 APE8-dihe-in -91.64, 124.53 APE8-rot-in 310.44 APE67-dihe-in -65.24, -8.9 -57.42, -46.72 APE12-dist-in 9.6206 APE11-dist-in 8.7016 APE10-dist-in 5.1963 APE9-dist-in 3.9237 None None None XRAY 2.252 0.177 0.212 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5v80 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5V82A P11309 34 306 313.0 96Y:401 Type1 Active DFGin 6.2131 14.4118 BLAminus -125.78, 171.27 64.15, 78.85 -91.71, 19.69 286.42, 77.38 -68.31, -20.73 in-in in 8.8236 Saltbr-in 2.5709 HRD-naA -70.88, -47.55 68.67, 4.77 in-in-in SNCiii in-in ActLoopNT-in 2.7889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.07, 17.68 APE9-dihe-na -81.71, -152.79 APE8-dihe-in -94.55, 121.67 APE8-rot-in 301.55 APE67-dihe-in -68.27, -8.9 -60.36, -41.63 APE12-dist-in 9.7433 APE11-dist-in 8.6739 APE10-dist-in 5.1826 APE9-dist-in 3.5857 None None None XRAY 1.888 0.182 0.199 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5v82 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3UIXA P11309 37 305 313.0 Q17:400 Type1 Active DFGin 6.1591 14.8214 BLAminus -133.2, 170.02 65.66, 77.49 -86.97, 13.03 288.74, 81.94 -68.85, -14.59 in-in in 9.0654 Saltbr-in 2.8853 HRD-naA -68.2, -50.15 66.82, 5.77 in-in-in SNCiii in-in ActLoopNT-in 2.7993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.4, 30.15 APE9-dihe-na -90.24, -149.24 APE8-dihe-in -93.32, 120.98 APE8-rot-in 306.79 APE67-dihe-in -70.28, -11.9 -58.72, -40.96 APE12-dist-in 9.6064 APE11-dist-in 8.5237 APE10-dist-in 5.4885 APE9-dist-in 3.7562 None None None XRAY 2.2 0.168 0.201 A 298.0 266.0 3 26 26 0 [[38, 290]] 1.0 3uix CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3UMWA P11309 37 304 313.0 596:400 Type1 Active DFGin 6.2909 14.5837 BLAminus -128.68, 168.78 67.21, 80.33 -91.49, 18.98 287.81, 74.46 -67.02, -11.8 in-in in 8.4885 Saltbr-in 2.8503 HRD-naA -69.92, -48.57 70.74, 4.13 in-in-in SNCiii in-in ActLoopNT-in 2.8096 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.82, 23.54 APE9-dihe-na -81.68, -155.27 APE8-dihe-in -92.32, 121.26 APE8-rot-in 306.5 APE67-dihe-in -69.25, -11.28 -53.65, -48.44 APE12-dist-in 9.1537 APE11-dist-in 8.5631 APE10-dist-in 5.5517 APE9-dist-in 3.7718 None None None XRAY 2.08 0.175 0.2 A 298.0 264.0 4 26 26 0 [[38, 290]] 1.0 3umw CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3UMXA P11309 37 304 313.0 Q18:400 Type1 Active DFGin 6.3211 14.6927 BLAminus -128.18, 168.05 66.13, 83.77 -95.39, 17.61 280.32, 78.57 -66.8, -16.44 in-in in 8.4362 Saltbr-in 2.9518 HRD-naA -70.86, -46.1 72.14, -3.21 in-in-in SNCiii in-in ActLoopNT-in 2.9654 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.18, 34.19 APE9-dihe-na -90.9, -156.14 APE8-dihe-in -92.65, 120.83 APE8-rot-in 316.33 APE67-dihe-in -56.49, -20.39 -55.25, -56.16 APE12-dist-in 9.0182 APE11-dist-in 8.6132 APE10-dist-in 5.466 APE9-dist-in 3.9429 None None None XRAY 2.55 0.18 0.229 A 298.0 261.0 7 26 26 0 [[38, 290]] 1.0 3umx CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4ENXA P11309 37 305 313.0 Z20:402 Type1 Active DFGin 6.0724 14.2577 BLAminus -124.23, 174.95 56.93, 87.82 -99.36, 21.71 285.95, 80.74 -78.01, -5.47 in-in in 8.7919 Saltbr-in 2.4703 HRD-naA -68.51, -45.47 67.84, 12.31 in-in-in SNCiii in-in ActLoopNT-in 2.803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.34, 41.24 APE9-dihe-na -101.41, -153.2 APE8-dihe-in -90.61, 127.01 APE8-rot-in 310.22 APE67-dihe-in -64.59, -15.43 -67.29, -43.92 APE12-dist-in 9.2342 APE11-dist-in 8.6621 APE10-dist-in 5.4211 APE9-dist-in 3.7373 None None None XRAY 2.8 0.192 0.233 A 298.0 266.0 3 26 26 0 [[38, 290]] 1.0 4enx CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4ENYA P11309 37 305 313.0 J19:404 Type1 Active DFGin 6.1683 14.409 BLAminus -126.77, 176.31 56.15, 81.83 -92.01, 22.92 285.19, 76.91 -75.2, -11.55 in-in in 8.8121 Saltbr-in 2.6741 HRD-naA -67.09, -45.67 67.16, 8.93 in-in-in SNCiii in-in ActLoopNT-in 2.7579 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.12, 33.6 APE9-dihe-na -103.74, -163.7 APE8-dihe-in -76.76, 123.85 APE8-rot-in 309.22 APE67-dihe-in -67.99, -11.42 -63.9, -43.13 APE12-dist-in 9.4542 APE11-dist-in 8.6678 APE10-dist-in 5.2094 APE9-dist-in 3.8101 None None None XRAY 2.801 0.175 0.224 A 298.0 261.0 8 26 26 0 [[38, 290]] 1.0 4eny CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4LL5A P11309 34 305 313.0 SK8:401 Type1 Active DFGin 6.1536 14.9413 BLAminus -130.09, 167.4 64.64, 85.24 -96.78, 19.13 285.46, 79.08 -67.1, -17.77 in-in in 8.9048 Saltbr-in 2.9074 HRD-naA -72.89, -48.94 71.1, 5.66 in-in-in SNCiii in-in ActLoopNT-in 2.8583 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.97, 33.17 APE9-dihe-na -91.19, -159.67 APE8-dihe-in -86.75, 127.22 APE8-rot-in 309.08 APE67-dihe-in -69.44, -9.3 -64.52, -42.1 APE12-dist-in 9.5929 APE11-dist-in 8.6246 APE10-dist-in 5.5027 APE9-dist-in 3.7227 None None None XRAY 2.0 0.169 0.189 A 298.0 268.0 4 26 26 0 [[38, 290]] 1.0 4ll5 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4LM5A P11309 35 305 313.0 Q17:401 Type1 Active DFGin 6.1717 14.8472 BLAminus -129.33, 170.23 65.43, 81.43 -93.64, 15.07 286.04, 82.64 -63.86, -18.24 in-in in 9.1345 Saltbr-in 2.7309 HRD-naA -69.11, -47.25 68.05, 2.81 in-in-in SNCiii in-in ActLoopNT-in 2.8293 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.68, 24.87 APE9-dihe-na -83.15, -151.88 APE8-dihe-in -95.39, 124.37 APE8-rot-in 310.14 APE67-dihe-in -64.57, -11.11 -60.82, -46.98 APE12-dist-in 9.5104 APE11-dist-in 8.5146 APE10-dist-in 5.4234 APE9-dist-in 3.7127 None None CSO161 XRAY 2.25 0.158 0.198 A 298.0 265.0 6 26 26 0 [[38, 290]] 1.0 4lm5 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4LMUA P11309 36 304 313.0 QUE:401 Type1 Active DFGin 6.1615 14.4307 BLAminus -125.85, 174.43 58.26, 85.32 -97.42, 18.39 285.76, 76.14 -68.38, -9.73 in-in in 8.702 Saltbr-in 2.3854 HRD-naA -71.42, -45.75 68.18, 3.07 in-in-in SNCiii in-in ActLoopNT-in 2.8482 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.78, 30.35 APE9-dihe-na -86.53, -151.77 APE8-dihe-in -97.13, 122.66 APE8-rot-in 306.98 APE67-dihe-in -65.32, -7.73 -59.99, -46.55 APE12-dist-in 9.4521 APE11-dist-in 8.6168 APE10-dist-in 5.5144 APE9-dist-in 3.8345 None None None XRAY 2.38 0.172 0.204 A 298.0 265.0 4 26 26 0 [[38, 290]] 1.0 4lmu CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5VUAB P11309 36 305 313.0 8GX:403 Type1 Active DFGin 6.2674 14.6306 BLAminus -131.5, 169.5 65.68, 85.46 -98.43, 24.84 284.2, 75.16 -72.94, -9.76 in-in in 8.4537 Saltbr-in 2.8407 HRD-naA -72.0, -46.73 70.73, 2.09 in-in-in SNCiii in-in ActLoopNT-in 2.8479 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.51, 33.95 APE9-dihe-na -87.15, -156.37 APE8-dihe-in -92.0, 123.34 APE8-rot-in 311.17 APE67-dihe-in -66.19, -11.92 -56.69, -48.02 APE12-dist-in 9.2638 APE11-dist-in 8.5434 APE10-dist-in 5.6059 APE9-dist-in 3.7837 None None None XRAY 2.2 0.167 0.196 B 298.0 270.0 0 26 26 0 [[38, 290]] 1.0 5vua CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5VUBB P11309 36 305 313.0 8GU:402 Type1 Active DFGin 6.2652 14.6046 BLAminus -124.74, 173.14 60.11, 84.16 -95.33, 18.9 286.57, 72.73 -67.18, -11.28 in-in in 8.585 Saltbr-in 2.3633 HRD-naA -74.43, -46.89 71.06, 5.3 in-in-in SNCiii in-in ActLoopNT-in 2.8541 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.25, 31.18 APE9-dihe-na -85.43, -151.45 APE8-dihe-in -96.33, 120.96 APE8-rot-in 305.35 APE67-dihe-in -68.9, -7.9 -56.39, -44.27 APE12-dist-in 9.3708 APE11-dist-in 8.5694 APE10-dist-in 5.5734 APE9-dist-in 3.6525 None None CSO161 XRAY 2.0 0.161 0.184 B 298.0 270.0 0 26 26 0 [[38, 290]] 1.0 5vub CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5VUCB P11309 36 305 313.0 8GR:402 Type1 Active DFGin 6.2599 14.5902 BLAminus -130.18, 165.22 63.78, 87.26 -96.8, 21.67 286.89, 72.33 -70.38, -11.1 in-in in 8.2713 Saltbr-in 2.7802 HRD-naA -75.49, -49.39 71.96, 7.41 in-in-in SNCiii in-in ActLoopNT-in 2.9022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.01, 27.32 APE9-dihe-na -81.89, -157.57 APE8-dihe-in -92.9, 123.77 APE8-rot-in 305.96 APE67-dihe-in -68.92, -9.19 -62.84, -43.07 APE12-dist-in 9.1928 APE11-dist-in 8.5586 APE10-dist-in 5.4339 APE9-dist-in 3.7674 None None CSO161 XRAY 2.0 0.176 0.199 B 298.0 270.0 0 26 26 0 [[38, 290]] 1.0 5vuc CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3R00A P11309 33 306 313.0 UNJ:1 Type1 Active DFGin 6.0775 14.5853 BLAminus -129.23, 179.95 62.78, 78.65 -92.67, 17.69 284.89, 76.92 -65.27, -12.58 in-in in 8.9851 Saltbr-in 2.6149 HRD-naA -69.03, -46.16 61.18, 15.3 in-in-in SNCiii in-in ActLoopNT-in 2.8737 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.83, 36.17 APE9-dihe-na -94.5, -143.14 APE8-dihe-in -99.32, 120.22 APE8-rot-in 298.64 APE67-dihe-in -66.4, -11.74 -58.9, -42.32 APE12-dist-in 9.8111 APE11-dist-in 8.5314 APE10-dist-in 5.6392 APE9-dist-in 3.7189 None None None XRAY 2.1 0.175 0.216 A 299.0 274.0 0 26 26 0 [[38, 290]] 1.0 3r00 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3R01A P11309 33 306 313.0 UNE:1 Type1 Active DFGin 6.1709 14.6386 BLAminus -135.6, 167.7 70.77, 75.77 -84.82, 17.16 285.86, 84.24 -68.67, -10.33 in-in in 8.8032 Saltbr-in 2.8831 HRD-naA -70.35, -49.23 74.71, 2.68 in-in-in SNCiii in-in ActLoopNT-in 2.8788 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.59, 35.76 APE9-dihe-na -87.25, -132.26 APE8-dihe-in -117.56, 118.78 APE8-rot-in 316.73 APE67-dihe-in -73.58, -11.68 -54.47, -42.96 APE12-dist-in 9.7376 APE11-dist-in 8.5085 APE10-dist-in 5.818 APE9-dist-in 3.9243 None None None XRAY 2.6 0.219 0.287 A 299.0 274.0 0 26 26 0 [[38, 290]] 1.0 3r01 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3R02A P11309 35 305 313.0 UNM:555 Type1 Active DFGin 6.1751 14.5657 BLAminus -128.64, 175.57 56.97, 87.35 -90.49, 17.56 285.73, 81.34 -74.51, -7.05 in-in in 9.0281 Saltbr-in 2.6339 HRD-naA -75.58, -44.47 72.61, 3.3 in-in-in SNCiii in-in ActLoopNT-in 2.8106 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.47, 29.58 APE9-dihe-na -87.11, -147.11 APE8-dihe-in -98.53, 121.85 APE8-rot-in 301.03 APE67-dihe-in -70.13, -7.69 -53.51, -42.81 APE12-dist-in 9.8451 APE11-dist-in 8.5843 APE10-dist-in 5.7937 APE9-dist-in 3.7583 None None None XRAY 1.95 0.168 0.189 A 299.0 271.0 0 26 26 0 [[38, 290]] 1.0 3r02 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3R04A P11309 35 305 313.0 UNQ:555 Type1 Active DFGin 6.1113 14.4928 BLAminus -119.88, 174.34 65.61, 74.31 -82.3, 14.36 287.66, 74.37 -62.06, -16.62 in-in in 8.9281 Saltbr-in 2.6342 HRD-naA -74.82, -45.09 62.9, 11.66 in-in-in SNCiii in-in ActLoopNT-in 2.8523 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.54, 31.05 APE9-dihe-na -88.35, -143.56 APE8-dihe-in -101.19, 121.66 APE8-rot-in 294.82 APE67-dihe-in -73.54, -5.15 -62.57, -37.68 APE12-dist-in 9.8484 APE11-dist-in 8.5024 APE10-dist-in 5.6442 APE9-dist-in 3.7219 None None None XRAY 1.7 0.179 0.206 A 299.0 271.0 0 26 26 0 [[38, 290]] 1.0 3r04 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VBQA P11309 35 305 313.0 0F5:555 Type1 Active DFGin 6.1979 14.5767 BLAminus -127.7, 179.22 57.68, 76.69 -85.86, 12.59 286.24, 73.15 -68.96, -5.86 in-in in 8.7676 Saltbr-in 2.64 HRD-naA -70.31, -44.96 66.03, 8.09 in-in-in SNCiii in-in ActLoopNT-in 2.8903 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.65, 27.89 APE9-dihe-na -90.08, -142.39 APE8-dihe-in -98.6, 121.83 APE8-rot-in 304.23 APE67-dihe-in -72.3, -7.09 -58.75, -37.63 APE12-dist-in 9.8116 APE11-dist-in 8.5951 APE10-dist-in 5.6985 APE9-dist-in 3.7029 None None None XRAY 1.85 0.206 0.206 A 299.0 271.0 0 26 26 0 [[38, 290]] 1.0 3vbq CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VBTA P11309 35 305 313.0 0F9:1 Type1 Active DFGin 6.1544 14.4155 BLAminus -130.27, 172.67 63.33, 71.31 -82.69, 17.12 286.5, 71.57 -76.38, -5.32 in-in in 8.7106 Saltbr-in 2.6583 HRD-naA -67.81, -46.73 67.69, 4.14 in-in-in SNCiii in-in ActLoopNT-in 2.8556 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.09, 27.22 APE9-dihe-na -88.86, -143.07 APE8-dihe-in -97.4, 123.61 APE8-rot-in 305.69 APE67-dihe-in -63.29, -9.77 -57.85, -48.3 APE12-dist-in 9.4897 APE11-dist-in 8.3934 APE10-dist-in 5.6037 APE9-dist-in 3.764 None None None XRAY 2.23 0.273 0.273 A 299.0 267.0 4 26 26 0 [[38, 290]] 1.0 3vbt CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VBVA P11309 35 305 313.0 0FK:1 Type1 Active DFGin 6.1684 14.5244 BLAminus -132.06, 170.0 63.81, 81.21 -91.04, 16.51 285.74, 75.33 -71.88, -8.41 in-in in 8.8343 Saltbr-in 2.6332 HRD-naA -65.91, -47.52 66.96, 5.14 in-in-in SNCiii in-in ActLoopNT-in 2.8482 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.35, 27.86 APE9-dihe-na -84.91, -139.46 APE8-dihe-in -108.06, 126.97 APE8-rot-in 303.82 APE67-dihe-in -70.7, -8.74 -60.57, -44.13 APE12-dist-in 9.4986 APE11-dist-in 8.4391 APE10-dist-in 5.6633 APE9-dist-in 3.6721 None None None XRAY 2.08 0.245 0.245 A 299.0 268.0 3 26 26 0 [[38, 290]] 1.0 3vbv CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VBWA P11309 35 305 313.0 0FN:1 Type1 Active DFGin 6.0586 14.28 BLAminus -127.49, 167.57 67.98, 79.4 -86.02, 16.62 293.39, 81.3 -60.91, -19.46 in-in in 8.8607 Saltbr-in 2.8787 HRD-naA -70.94, -49.39 81.06, -4.45 in-in-in SNCiii in-in ActLoopNT-in 2.7981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.47, 33.12 APE9-dihe-na -84.03, -133.93 APE8-dihe-in -105.55, 127.02 APE8-rot-in 315.81 APE67-dihe-in -63.23, -11.02 -61.62, -47.09 APE12-dist-in 9.5414 APE11-dist-in 8.3432 APE10-dist-in 5.6723 APE9-dist-in 3.8503 None None None XRAY 2.48 0.299 0.299 A 299.0 264.0 7 26 26 0 [[38, 290]] 1.0 3vbw CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VBXA P11309 35 305 313.0 0FO:1 Type1 Active DFGin 6.0578 14.5368 BLAminus -132.08, 169.91 71.33, 70.33 -85.72, 14.8 288.27, 79.72 -65.16, -16.66 in-in in 8.9539 Saltbr-in 2.6816 HRD-naA -64.87, -49.91 70.18, 2.86 in-in-in SNCiii in-in ActLoopNT-in 2.7949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.29, 28.64 APE9-dihe-na -87.57, -146.06 APE8-dihe-in -95.38, 125.1 APE8-rot-in 301.97 APE67-dihe-in -65.7, -15.04 -61.83, -41.49 APE12-dist-in 9.426 APE11-dist-in 8.3985 APE10-dist-in 5.5184 APE9-dist-in 3.8074 None None None XRAY 2.03 0.258 0.258 A 299.0 268.0 3 26 26 0 [[38, 290]] 1.0 3vbx CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VBYA P11309 35 305 313.0 0FR:1 Type1 Active DFGin 6.1427 14.6314 BLAminus -131.01, 169.0 66.5, 79.73 -89.48, 18.31 287.57, 72.75 -74.21, -13.52 in-in in 8.9517 Saltbr-in 2.7609 HRD-naA -68.42, -44.76 63.69, 3.49 in-in-in SNCiii in-in ActLoopNT-in 2.7963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.13, 34.14 APE9-dihe-na -92.9, -153.09 APE8-dihe-in -93.99, 123.58 APE8-rot-in 305.15 APE67-dihe-in -72.64, -2.35 -57.97, -45.41 APE12-dist-in 9.3282 APE11-dist-in 8.3473 APE10-dist-in 5.5122 APE9-dist-in 3.8248 None None None XRAY 2.27 0.261 0.261 A 299.0 267.0 4 26 26 0 [[38, 290]] 1.0 3vby CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3VC4A P11309 33 306 313.0 0FS:1 Type1 Active DFGin 6.0756 14.6091 BLAminus -139.74, 164.89 72.09, 84.05 -96.17, 20.14 288.43, 67.45 -72.44, -2.97 in-in in 9.0297 Saltbr-in 2.6612 HRD-naA -61.2, -51.03 71.16, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.7242 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.23, 31.29 APE9-dihe-na -95.97, -149.39 APE8-dihe-in -93.38, 121.01 APE8-rot-in 311.86 APE67-dihe-in -66.44, -6.52 -55.27, -50.39 APE12-dist-in 9.953 APE11-dist-in 8.5606 APE10-dist-in 5.4613 APE9-dist-in 3.8012 None None None XRAY 2.23 0.319 0.319 A 299.0 274.0 0 26 26 0 [[38, 290]] 1.0 3vc4 CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3F2AA P11309 32 308 313.0 985:1 Type1 Active DFGin 6.0885 14.3121 BLAminus -128.57, 176.64 59.08, 83.27 -93.92, 21.71 288.01, 71.24 -68.66, -6.64 in-in in 8.7442 Saltbr-in 2.7888 HRD-naA -68.81, -50.19 71.47, 2.55 in-in-in SNCiii in-in ActLoopNT-in 2.8314 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.81, 27.99 APE9-dihe-na -90.31, -146.93 APE8-dihe-in -92.75, 125.96 APE8-rot-in 310.85 APE67-dihe-in -59.77, -4.55 -52.49, -57.5 APE12-dist-in 9.8822 APE11-dist-in 8.7738 APE10-dist-in 5.5518 APE9-dist-in 3.6432 None SEP261 SEP261 XRAY 1.9 0.256 0.282 A 300.0 277.0 0 26 26 0 [[38, 290]] 1.0 3f2a CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2XIXA P11309 33 306 313.0 XIX:1307 Type1 Active DFGin 6.198 14.4047 BLAminus -127.72, 172.47 53.38, 85.02 -93.57, 22.7 288.78, 75.96 -73.48, -9.49 in-in in 8.7954 Saltbr-in 2.6185 HRD-naA -70.78, -45.87 74.83, 0.99 in-in-in SNCiii in-in ActLoopNT-in 2.79 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.52, 26.26 APE9-dihe-na -83.36, -151.06 APE8-dihe-in -94.01, 119.49 APE8-rot-in 303.81 APE67-dihe-in -72.45, -16.36 -55.92, -38.22 APE12-dist-in 9.7148 APE11-dist-in 8.6346 APE10-dist-in 5.6984 APE9-dist-in 3.6685 None SEP261,SEP276 SEP261,SEP276 XRAY 2.4 0.173 0.214 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xix CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2XIYA P11309 33 306 313.0 XIY:1307 Type1 Active DFGin 6.3046 14.5836 BLAminus -122.45, 177.21 60.39, 73.41 -90.27, 13.91 284.0, 74.82 -69.72, -11.86 in-in in 9.0115 Saltbr-in 2.5935 HRD-naA -65.92, -48.71 70.04, 1.22 in-in-in SNCiii in-in ActLoopNT-in 2.7462 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.76, 20.93 APE9-dihe-na -80.08, -150.81 APE8-dihe-in -97.46, 126.22 APE8-rot-in 306.41 APE67-dihe-in -71.61, -13.32 -59.57, -41.49 APE12-dist-in 9.8366 APE11-dist-in 8.6241 APE10-dist-in 5.5581 APE9-dist-in 3.6392 None SEP261 SEP261 XRAY 2.2 0.172 0.201 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xiy CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2XIZA P11309 33 306 313.0 XIZ:1307 Type1 Active DFGin 6.1763 14.5485 BLAminus -122.54, 175.77 58.35, 84.58 -93.18, 17.46 282.52, 76.08 -67.84, -13.59 in-in in 8.8664 Saltbr-in 2.5793 HRD-naA -67.92, -44.32 48.8, 19.99 in-in-in SNCiii in-in ActLoopNT-in 2.8687 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.12, 25.76 APE9-dihe-na -79.92, -145.43 APE8-dihe-in -101.02, 126.08 APE8-rot-in 309.36 APE67-dihe-in -71.71, -14.75 -59.22, -39.66 APE12-dist-in 9.7528 APE11-dist-in 8.6841 APE10-dist-in 5.6508 APE9-dist-in 3.6837 None SEP261 SEP261 XRAY 2.21 0.258 0.286 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xiz CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2XJ0A P11309 33 307 313.0 XJ0:1307 Type1 Active DFGin 5.9294 13.6758 BLAminus -134.6, 165.43 58.42, 101.5 -112.27, 25.85 290.56, 60.01 -70.79, -14.26 in-in in 8.6795 Saltbr-in 2.9659 HRD-naA -62.77, -42.06 61.42, 5.55 in-in-in SNCiii in-in ActLoopNT-in 2.9811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 10.17 APE9-dihe-na -82.33, -169.45 APE8-dihe-in -68.0, 130.83 APE8-rot-in 305.92 APE67-dihe-in -52.49, -21.01 -63.78, -52.51 APE12-dist-in 9.7715 APE11-dist-in 8.4681 APE10-dist-in 4.9761 APE9-dist-in 3.8973 None None None XRAY 3.1 0.218 0.263 A 301.0 275.0 0 26 26 0 [[38, 290]] 1.0 2xj0 CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2XJ1A P11309 33 306 313.0 XJ1:1307 Type1 Active DFGin 6.2498 14.2958 BLAminus -129.27, 177.63 56.13, 82.39 -92.13, 21.02 283.59, 76.59 -73.33, -11.63 in-in in 8.8725 Saltbr-in 2.7085 HRD-naA -72.25, -47.05 68.39, 1.49 in-in-in SNCiii in-in ActLoopNT-in 2.6939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.13, 25.06 APE9-dihe-na -81.21, -153.15 APE8-dihe-in -95.3, 123.79 APE8-rot-in 303.34 APE67-dihe-in -71.81, -9.27 -59.4, -42.14 APE12-dist-in 9.8771 APE11-dist-in 8.5709 APE10-dist-in 5.6004 APE9-dist-in 3.6104 None SEP261 SEP261 XRAY 2.13 0.178 0.212 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xj1 CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2XJ2A P11309 33 306 313.0 985:1001 Type1 Active DFGin 6.1572 14.3889 BLAminus -121.97, 176.14 56.84, 82.15 -90.5, 18.96 286.44, 74.76 -71.88, -10.32 in-in in 8.8085 Saltbr-in 2.6446 HRD-naA -70.41, -47.45 68.26, 1.41 in-in-in SNCiii in-in ActLoopNT-in 2.7186 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.43, 24.44 APE9-dihe-na -81.03, -149.66 APE8-dihe-in -95.09, 121.86 APE8-rot-in 305.59 APE67-dihe-in -74.97, -11.2 -56.65, -40.34 APE12-dist-in 9.8346 APE11-dist-in 8.6692 APE10-dist-in 5.671 APE9-dist-in 3.522 None SEP261 SEP261 XRAY 2.2 0.169 0.202 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xj2 CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4A7CA P11309 32 305 313.0 E46:1306 Type1 Active DFGin 6.1794 14.789 BLAminus -131.67, 167.73 66.77, 79.73 -90.97, 18.69 290.12, 73.93 -69.69, -11.45 in-in in 8.9034 Saltbr-in 2.5501 HRD-naA -69.9, -49.4 70.62, 3.17 in-in-in SNCiii in-in ActLoopNT-in 2.7677 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.97, 35.42 APE9-dihe-na -90.39, -152.55 APE8-dihe-in -91.86, 121.24 APE8-rot-in 305.64 APE67-dihe-in -69.15, -9.02 -58.09, -44.18 APE12-dist-in 9.5612 APE11-dist-in 8.6243 APE10-dist-in 5.6568 APE9-dist-in 3.8767 None SEP261 SEP261 XRAY 2.3 0.171 0.207 A 308.0 274.0 0 26 26 0 [[38, 290]] 1.0 4a7c CAMK_PIM1_HUMAN CAMK 3.8e-65 225.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 1XWSA P11309 33 305 313.0 BI1:1001 Type1 Active DFGin 6.1159 14.9341 BLAminus -129.52, 166.95 66.18, 81.14 -88.91, 13.45 284.44, 80.6 -63.86, -15.19 in-in in 8.8578 Saltbr-in 2.8112 HRD-naA -69.66, -47.71 69.42, 1.43 in-in-in SNCiii in-in ActLoopNT-in 2.84 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.43, 26.37 APE9-dihe-na -77.62, -162.66 APE8-dihe-in -79.83, 125.2 APE8-rot-in 307.07 APE67-dihe-in -74.93, -11.45 -55.08, -43.34 APE12-dist-in 9.7063 APE11-dist-in 8.7658 APE10-dist-in 5.8681 APE9-dist-in 3.8449 None None None XRAY 1.8 0.182 0.213 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 1xws CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4BZNA P11309 33 305 313.0 UGX:1306 Type1 Active DFGin 6.1991 14.5084 BLAminus -123.83, 168.52 64.99, 88.0 -96.39, 24.65 289.87, 72.27 -71.02, -12.29 in-in in 8.3963 Saltbr-in 2.5786 HRD-naA -70.91, -47.25 68.09, 6.65 in-in-in SNCiii in-in ActLoopNT-in 2.868 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.83, 29.38 APE9-dihe-na -84.39, -152.15 APE8-dihe-in -95.81, 123.59 APE8-rot-in 305.15 APE67-dihe-in -71.92, -8.16 -59.74, -41.18 APE12-dist-in 9.3592 APE11-dist-in 8.4435 APE10-dist-in 5.5192 APE9-dist-in 3.6102 None SEP261 SEP261 XRAY 1.9 0.178 0.199 A 314.0 273.0 0 26 26 0 [[38, 290]] 1.0 4bzn CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4BZOA P11309 33 305 313.0 676:1306 Type1 Active DFGin 6.254 14.7622 BLAminus -127.92, 165.55 68.25, 84.97 -95.87, 20.96 286.29, 72.86 -74.22, -6.71 in-in in 8.4398 Saltbr-in 2.622 HRD-naA -71.06, -49.33 68.13, 9.04 in-in-in SNCiii in-in ActLoopNT-in 2.8672 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.68, 32.17 APE9-dihe-na -87.85, -152.26 APE8-dihe-in -92.39, 123.96 APE8-rot-in 304.04 APE67-dihe-in -67.43, -9.74 -60.54, -43.52 APE12-dist-in 9.6012 APE11-dist-in 8.5854 APE10-dist-in 5.5358 APE9-dist-in 3.6618 None SEP261 SEP261 XRAY 2.1 0.183 0.216 A 314.0 273.0 0 26 26 0 [[38, 290]] 1.0 4bzo CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7ZUNA P11309 33 305 313.0 JYO:401 Type1 Active DFGin 6.2197 14.2081 BLAminus -133.16, 165.47 67.55, 84.83 -98.38, 21.66 289.12, 75.62 -70.0, -22.74 in-in in 8.2062 Saltbr-in 2.792 HRD-naA -67.79, -58.14 75.87, 8.23 in-in-in SNCiii in-in ActLoopNT-in 2.8668 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.98, 24.87 APE9-dihe-na -93.48, -164.33 APE8-dihe-in -86.18, 121.45 APE8-rot-in 312.27 APE67-dihe-in -61.31, -13.56 -57.48, -51.41 APE12-dist-in 9.4299 APE11-dist-in 8.4442 APE10-dist-in 5.0492 APE9-dist-in 3.8725 None SEP261 SEP261 XRAY 2.5 0.177 0.235 A 314.0 270.0 3 26 26 0 [[38, 290]] 1.0 7zun CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4XHKB P11309 32 305 313.0 3YR:401 Type1 Active DFGin 6.2265 14.5249 BLAminus -126.44, 167.48 62.73, 73.24 -76.02, 8.65 289.12, 83.25 -72.3, -9.91 in-in in 8.8608 Saltbr-in 2.6139 HRD-naA -68.85, -46.46 65.48, 11.28 in-in-in SNCiii in-in ActLoopNT-in 2.8772 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.53, 24.82 APE9-dihe-na -81.56, -148.04 APE8-dihe-in -105.73, 126.46 APE8-rot-in 298.97 APE67-dihe-in -77.31, -6.66 -69.47, -34.63 APE12-dist-in 9.5732 APE11-dist-in 8.6835 APE10-dist-in 5.642 APE9-dist-in 3.7202 None SEP261 SEP261 XRAY 1.9 0.158 0.184 B 315.0 270.0 4 26 26 0 [[38, 290]] 1.0 4xhk CAMK_PIM1_HUMAN CAMK 4.1e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4JX7A P11309 33 306 313.0 1N6:401 Type1 Active DFGin 6.2835 14.7533 BLAminus -127.31, 170.34 63.68, 81.99 -92.92, 12.24 283.66, 75.72 -67.48, -14.52 in-in in 8.8428 Saltbr-in 2.7677 HRD-naA -66.3, -47.17 67.1, 1.58 in-in-in SNCiii in-in ActLoopNT-in 2.7336 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.4, 25.92 APE9-dihe-na -85.09, -149.75 APE8-dihe-in -93.53, 123.68 APE8-rot-in 312.23 APE67-dihe-in -66.8, -17.18 -56.19, -45.11 APE12-dist-in 9.7559 APE11-dist-in 8.5902 APE10-dist-in 5.6048 APE9-dist-in 3.9044 None None None XRAY 2.4 0.193 0.228 A 326.0 274.0 0 26 26 0 [[38, 290]] 1.0 4jx7 CAMK_PIM1_HUMAN CAMK 4.6e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4ALVA P11309 33 306 313.0 R9P:1308 Type1 Active DFGin 6.0359 14.4757 BLAminus -137.53, 165.69 68.25, 83.91 -91.38, 16.23 287.59, 75.48 -60.65, -18.54 in-in in 8.6626 Saltbr-in 2.3403 HRD-naA -75.94, -45.06 66.41, 17.82 in-in-in SNCiii in-in ActLoopNT-in 2.9682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.01, 38.02 APE9-dihe-na -89.15, -139.06 APE8-dihe-in -112.86, 124.4 APE8-rot-in 319.08 APE67-dihe-in -51.23, -17.72 -57.73, -58.1 APE12-dist-in 9.4151 APE11-dist-in 8.6868 APE10-dist-in 5.7072 APE9-dist-in 3.6859 None None None XRAY 2.59 0.195 0.256 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 4alv CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4ALWA P11309 34 306 313.0 HY7:1308 Type1 Active DFGin 6.0045 14.5947 BLAminus -122.86, 171.92 71.12, 81.46 -94.23, 18.88 291.83, 80.43 -59.13, -19.56 in-in in 8.8614 Saltbr-in 2.6093 HRD-naA -72.84, -43.49 62.9, 3.06 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.98, 32.2 APE9-dihe-na -91.86, -145.44 APE8-dihe-in -92.13, 124.7 APE8-rot-in 302.73 APE67-dihe-in -76.25, -2.93 -59.68, -41.94 APE12-dist-in 9.6324 APE11-dist-in 8.5086 APE10-dist-in 5.7436 APE9-dist-in 3.771 None None None XRAY 1.92 0.158 0.207 A 328.0 273.0 0 26 26 0 [[38, 290]] 1.0 4alw CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4N6YA P11309 32 305 313.0 2HV:401 Type1 Active DFGin 6.2593 14.8808 BLAminus -123.98, 165.51 60.84, 90.41 -100.85, 18.31 286.86, 79.6 -74.61, -13.5 in-in in 8.7605 Saltbr-in 2.7094 HRD-naA -69.76, -50.01 73.25, 2.39 in-in-in SNCiii in-in ActLoopNT-in 2.9037 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.48, 35.75 APE9-dihe-na -98.87, -155.99 APE8-dihe-in -86.09, 125.72 APE8-rot-in 310.58 APE67-dihe-in -66.86, -9.74 -54.28, -49.47 APE12-dist-in 9.3871 APE11-dist-in 8.4414 APE10-dist-in 5.4013 APE9-dist-in 3.7697 None SEP261 SEP261 XRAY 2.6 0.159 0.212 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 4n6y CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4N6ZA P11309 33 305 313.0 2HW:401 Type1 Active DFGin 6.463 14.6459 BLAminus -126.99, 169.95 59.29, 83.89 -97.92, 18.69 285.67, 67.47 -72.35, -9.24 in-in in 8.2536 Saltbr-in 2.7291 HRD-naA -69.23, -47.57 69.1, 0.1 in-in-in SNCiii in-in ActLoopNT-in 2.9924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.18, 25.75 APE9-dihe-na -86.3, -154.15 APE8-dihe-in -92.66, 118.79 APE8-rot-in 308.24 APE67-dihe-in -66.17, -14.41 -51.57, -45.87 APE12-dist-in 9.4646 APE11-dist-in 8.5132 APE10-dist-in 5.3789 APE9-dist-in 3.6943 None SEP261 SEP261 XRAY 2.2 0.161 0.189 A 328.0 273.0 0 26 26 0 [[38, 290]] 1.0 4n6z CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4N70A P11309 32 306 313.0 2HX:401 Type1 Active DFGin 6.1649 14.5694 BLAminus -137.89, 169.53 64.36, 80.83 -93.88, 21.26 288.11, 67.53 -75.41, -5.31 in-in in 8.6245 Saltbr-in 2.6005 HRD-naA -69.13, -48.86 67.14, 6.63 in-in-in SNCiii in-in ActLoopNT-in 2.8242 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.37, 33.23 APE9-dihe-na -89.84, -146.82 APE8-dihe-in -98.54, 120.46 APE8-rot-in 304.86 APE67-dihe-in -67.47, -8.0 -60.04, -43.4 APE12-dist-in 9.5943 APE11-dist-in 8.6595 APE10-dist-in 5.7234 APE9-dist-in 3.7572 None SEP261 SEP261 XRAY 2.1 0.169 0.208 A 328.0 275.0 0 26 26 0 [[38, 290]] 1.0 4n70 CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5DWRA P11309 33 306 313.0 5H7:401 Type1 Active DFGin 6.2423 14.6643 BLAminus -131.54, 168.2 64.5, 84.97 -98.37, 18.01 285.62, 75.32 -66.32, -15.3 in-in in 8.5476 Saltbr-in 2.6698 HRD-naA -72.01, -47.63 67.32, 6.26 in-in-in SNCiii in-in ActLoopNT-in 2.9583 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.09, 26.57 APE9-dihe-na -84.89, -152.84 APE8-dihe-in -93.58, 121.01 APE8-rot-in 307.85 APE67-dihe-in -68.04, -7.01 -54.84, -45.5 APE12-dist-in 9.522 APE11-dist-in 8.5314 APE10-dist-in 5.4179 APE9-dist-in 3.6508 None SEP261 SEP261 XRAY 2.0 0.175 0.202 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 5dwr CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6YKDA P11309 33 305 313.0 OWB:60400 Type1 Active DFGin 6.1577 14.6899 BLAminus -121.19, 171.99 65.51, 79.7 -90.44, 14.31 281.37, 83.04 -61.46, -20.23 in-in in 8.9313 Saltbr-in 2.6812 HRD-naA -69.86, -48.77 63.9, 14.36 in-in-in SNCiii in-in ActLoopNT-in 2.8682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.12, 24.2 APE9-dihe-na -86.9, -151.63 APE8-dihe-in -93.7, 123.39 APE8-rot-in 303.13 APE67-dihe-in -72.97, -5.5 -60.57, -42.11 APE12-dist-in 9.6038 APE11-dist-in 8.5277 APE10-dist-in 5.4138 APE9-dist-in 3.7385 None SEP261 SEP261 XRAY 1.86 0.16 0.194 A 329.0 273.0 0 26 26 0 [[38, 290]] 1.0 6ykd CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2OBJA P11309 33 305 313.0 VRV:400 Type1 Active DFGin 5.8483 14.3418 BLAminus -135.1, 165.89 65.58, 81.59 -93.29, 20.74 291.15, 68.53 -60.11, -19.32 in-in in 8.6835 Saltbr-in 2.448 HRD-naA -67.98, -46.96 66.7, 2.66 in-in-in SNCiii in-in ActLoopNT-in 2.9077 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.26, 30.91 APE9-dihe-na -92.97, -164.42 APE8-dihe-in -76.75, 121.77 APE8-rot-in 305.59 APE67-dihe-in -61.67, -9.38 -55.68, -49.65 APE12-dist-in 9.4446 APE11-dist-in 8.5058 APE10-dist-in 5.3383 APE9-dist-in 3.7537 None SEP261 SEP261 XRAY 2.5 0.205 0.246 A 333.0 273.0 0 26 26 0 [[38, 290]] 1.0 2obj CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3BGPA P11309 33 305 313.0 VX1:314 Type1 Active DFGin 5.9426 14.4251 BLAminus -126.41, 157.1 77.54, 91.73 -104.16, 28.82 293.34, 70.26 -65.15, -26.7 in-in in 8.6312 Saltbr-in 2.6289 HRD-naA -72.43, -49.43 73.8, -3.17 in-in-in SNCiii in-in ActLoopNT-in 2.7729 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.31, 13.68 APE9-dihe-na -86.06, -170.88 APE8-dihe-in -67.89, 136.06 APE8-rot-in 304.87 APE67-dihe-in -64.78, -12.46 -73.3, -44.0 APE12-dist-in 9.3655 APE11-dist-in 8.5615 APE10-dist-in 4.9825 APE9-dist-in 3.9275 None SEP261 SEP261 XRAY 2.8 0.213 0.261 A 333.0 273.0 0 26 26 0 [[38, 290]] 1.0 3bgp CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3BGQA P11309 33 305 313.0 VX2:314 Type1 Active DFGin 6.3949 14.8556 BLAminus -129.22, 172.22 56.92, 80.34 -93.96, 24.94 287.45, 64.49 -68.32, -10.99 in-in in 8.4273 Saltbr-in 2.6592 HRD-naA -70.11, -48.13 67.03, 6.04 in-in-in SNCiii in-in ActLoopNT-in 2.9262 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.69, 26.46 APE9-dihe-na -85.59, -155.16 APE8-dihe-in -92.08, 118.01 APE8-rot-in 308.33 APE67-dihe-in -63.18, -11.49 -49.18, -49.37 APE12-dist-in 9.6074 APE11-dist-in 8.5858 APE10-dist-in 5.4106 APE9-dist-in 3.6395 None SEP261 SEP261 XRAY 2.0 0.213 0.23 A 333.0 273.0 0 26 26 0 [[38, 290]] 1.0 3bgq CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3BGZA P11309 33 305 313.0 VX3:314 Type1 Active DFGin 6.223 14.5079 BLAminus -126.99, 169.09 64.54, 79.92 -92.02, 15.99 284.89, 75.21 -68.7, -13.09 in-in in 8.7342 Saltbr-in 2.7258 HRD-naA -68.01, -47.53 72.06, 3.12 in-in-in SNCiii in-in ActLoopNT-in 2.8055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.26, 35.08 APE9-dihe-na -86.26, -142.72 APE8-dihe-in -103.04, 122.93 APE8-rot-in 309.34 APE67-dihe-in -67.64, -10.68 -55.55, -46.74 APE12-dist-in 9.5335 APE11-dist-in 8.6464 APE10-dist-in 5.6709 APE9-dist-in 3.6886 None SEP261 SEP261 XRAY 2.4 0.196 0.233 A 333.0 268.0 5 26 26 0 [[38, 290]] 1.0 3bgz CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3WE8A P11309 33 305 313.0 RUI:401 Type1 Active DFGin 6.0765 14.5621 BLAminus -133.3, 170.64 67.13, 73.63 -87.77, 10.99 287.95, 77.91 -66.1, -8.31 in-in in 8.9805 Saltbr-in 2.6432 HRD-naA -75.68, -43.45 65.63, 6.85 in-in-in SNCiii in-in ActLoopNT-in 2.8418 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.96, 25.34 APE9-dihe-na -83.21, -158.59 APE8-dihe-in -86.86, 122.45 APE8-rot-in 300.85 APE67-dihe-in -73.76, -3.38 -61.05, -39.9 APE12-dist-in 9.8003 APE11-dist-in 8.6353 APE10-dist-in 5.6029 APE9-dist-in 3.7476 R250G None None XRAY 1.954 0.16 0.177 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3we8 CAMK_PIM1_HUMAN CAMK 9.2e-65 224.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4AS0A P11309 33 305 313.0 RPS:1306 Type1 Active DFGin 6.2392 14.7972 BLAminus -125.08, 170.08 63.9, 84.56 -93.79, 23.62 287.71, 77.4 -74.79, -13.31 in-in in 8.9969 Saltbr-in 2.4858 HRD-naA -73.68, -44.47 70.76, -1.79 in-in-in SNCiii in-in ActLoopNT-in 2.8952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.05, 33.62 APE9-dihe-na -96.04, -155.25 APE8-dihe-in -91.93, 124.92 APE8-rot-in 312.41 APE67-dihe-in -67.91, -14.18 -64.04, -41.51 APE12-dist-in 9.5865 APE11-dist-in 8.5215 APE10-dist-in 5.3972 APE9-dist-in 4.1789 None None None XRAY 2.3 0.172 0.201 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 4as0 CAMK_PIM1_HUMAN CAMK 9.2e-65 224.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5TURA P11309 34 306 313.0 7LK:401 Type1 Active DFGin 6.061 14.49 BLAminus -136.79, 174.59 58.79, 85.71 -98.08, 24.51 288.61, 83.41 -77.7, -2.74 in-in in 8.7582 Saltbr-in 2.6156 HRD-naA -76.1, -44.31 69.09, 5.73 in-in-in SNCiii in-in ActLoopNT-in 2.7428 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.99, 42.91 APE9-dihe-na -110.95, -154.07 APE8-dihe-in -91.19, 125.87 APE8-rot-in 304.26 APE67-dihe-in -69.95, -16.95 -69.94, -33.83 APE12-dist-in 9.7357 APE11-dist-in 8.7982 APE10-dist-in 5.3539 APE9-dist-in 3.9645 None None None XRAY 2.948 0.209 0.248 A 404.0 270.0 3 26 26 0 [[38, 290]] 1.0 5tur CAMK_PIM1_HUMAN CAMK 8.9e-65 224.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2J2IB P11309 33 305 313.0 LY4:1307 Type1 Active DFGin 6.3491 14.7879 BLAminus -124.69, 164.2 69.56, 81.11 -88.57, 16.71 287.44, 78.04 -63.89, -22.24 in-in in 8.7154 Saltbr-in 2.8844 HRD-naA -68.27, -48.73 73.43, 1.94 in-in-in SNCiii in-in ActLoopNT-in 2.8048 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.68, 17.7 APE9-dihe-na -79.18, -163.88 APE8-dihe-in -85.23, 122.14 APE8-rot-in 304.09 APE67-dihe-in -70.03, -11.09 -55.65, -47.61 APE12-dist-in 9.3137 APE11-dist-in 8.7009 APE10-dist-in 5.4569 APE9-dist-in 3.9641 R250G None None XRAY 1.9 0.18 0.2 B 312.0 273.0 0 26 26 0 [[38, 290]] 1.0 2j2i CAMK_PIM1_HUMAN CAMK 1.5e-64 223.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7QB2A P11309 33 305 313.0 A7X:402 Type1 Active DFGin 6.2608 14.4336 BLAminus -125.87, 176.63 53.43, 82.5 -86.6, 20.72 284.17, 73.36 -70.8, -10.08 in-in in 8.6566 Saltbr-in 2.6079 HRD-naA -76.36, -48.43 70.95, 3.72 in-in-in SNCiii in-in ActLoopNT-in 2.6919 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.34, 22.15 APE9-dihe-na -86.92, -149.81 APE8-dihe-in -97.03, 122.97 APE8-rot-in 300.26 APE67-dihe-in -69.31, -7.68 -64.45, -41.13 APE12-dist-in 9.9263 APE11-dist-in 8.6524 APE10-dist-in 4.9748 APE9-dist-in 3.7444 R250G SEP261 SEP261 XRAY 2.53 0.159 0.202 A 312.0 273.0 0 26 26 0 [[38, 290]] 1.0 7qb2 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7QFMA P11309 33 305 313.0 AY3:402 Type1 Active DFGin 6.2031 14.458 BLAminus -124.14, 177.11 57.14, 79.43 -85.98, 19.87 284.85, 75.66 -69.01, -15.13 in-in in 8.7647 Saltbr-in 2.6921 HRD-naA -73.09, -45.9 66.81, 9.42 in-in-in SNCiii in-in ActLoopNT-in 2.846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 26.43 APE9-dihe-na -81.47, -151.25 APE8-dihe-in -97.97, 122.34 APE8-rot-in 302.11 APE67-dihe-in -71.87, -9.27 -61.74, -39.67 APE12-dist-in 9.9106 APE11-dist-in 8.6095 APE10-dist-in 5.3753 APE9-dist-in 3.6137 R250G SEP261 SEP261 XRAY 1.95 0.159 0.178 A 312.0 271.0 2 26 26 0 [[38, 290]] 1.0 7qfm CAMK_PIM1_HUMAN CAMK 1.5e-64 223.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3JPVA P11309 33 305 313.0 1DR:313 Type1 Active DFGin 6.1479 14.441 BLAminus -120.08, 164.67 68.13, 86.84 -92.5, 13.59 289.99, 74.69 -67.43, -13.65 in-in in 9.0034 Saltbr-in 2.5634 HRD-naA -72.55, -46.96 72.58, 4.93 in-in-in SNCiii in-in ActLoopNT-in 2.8888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.51, 21.98 APE9-dihe-na -83.62, -150.17 APE8-dihe-in -98.9, 116.73 APE8-rot-in 306.83 APE67-dihe-in -67.26, -10.5 -54.29, -42.64 APE12-dist-in 9.8235 APE11-dist-in 8.4389 APE10-dist-in 5.4133 APE9-dist-in 3.7639 None None None XRAY 2.35 0.176 0.226 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 3jpv CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3MA3A P11309 37 305 313.0 01I:313 Type1 Active DFGin 6.0181 14.2367 BLAminus -126.51, 170.48 60.71, 85.71 -91.62, 21.05 288.87, 82.52 -71.65, -14.95 in-in in 8.9174 Saltbr-in 2.6909 HRD-naA -71.5, -42.79 64.42, 10.83 in-in-in SNCiii in-in ActLoopNT-in 2.754 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.06, 17.84 APE9-dihe-na -81.84, -163.49 APE8-dihe-in -85.13, 123.05 APE8-rot-in 304.03 APE67-dihe-in -65.07, -11.91 -66.26, -41.53 APE12-dist-in 9.8117 APE11-dist-in 8.4025 APE10-dist-in 5.2207 APE9-dist-in 3.8789 None SEP261 SEP261 XRAY 2.3 0.172 0.233 A 313.0 267.0 2 26 26 0 [[38, 290]] 1.0 3ma3 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3QF9A P11309 32 305 313.0 NM8:313 Type1 Active DFGin 6.0701 14.424 BLAminus -120.87, 169.05 67.22, 78.8 -88.89, 16.3 288.42, 76.0 -67.55, -12.21 in-in in 8.8485 Saltbr-in 2.5791 HRD-naA -70.76, -46.92 73.96, 4.53 in-in-in SNCiii in-in ActLoopNT-in 2.8907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.62, 24.45 APE9-dihe-na -83.53, -155.23 APE8-dihe-in -93.29, 124.33 APE8-rot-in 299.27 APE67-dihe-in -72.17, -10.84 -63.75, -37.33 APE12-dist-in 9.804 APE11-dist-in 8.4801 APE10-dist-in 5.3666 APE9-dist-in 3.6712 R250G None None XRAY 2.2 0.188 0.227 A 313.0 274.0 0 26 26 0 [[38, 290]] 1.0 3qf9 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4GW8A P11309 33 305 313.0 3RA:401 Type1 Active DFGin 6.2361 14.6142 BLAminus -126.36, 165.58 62.03, 83.71 -89.36, 16.13 285.86, 76.28 -67.97, -17.62 in-in in 8.7369 Saltbr-in 2.7149 HRD-naA -74.23, -46.85 73.75, 9.79 in-in-in SNCiii in-in ActLoopNT-in 2.8877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.85, 8.01 APE9-dihe-na -80.24, -160.25 APE8-dihe-in -87.85, 121.5 APE8-rot-in 304.03 APE67-dihe-in -71.21, -12.4 -59.35, -38.89 APE12-dist-in 9.4824 APE11-dist-in 8.2992 APE10-dist-in 4.4436 APE9-dist-in 3.7427 R250G None None XRAY 2.0 0.178 0.213 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 4gw8 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6PCWA P11309 32 305 313.0 O97:500 Type1 Active DFGin 6.1281 14.5651 BLAminus -128.69, 170.24 60.89, 83.86 -89.77, 15.97 285.56, 79.53 -66.69, -14.24 in-in in 8.7913 Saltbr-in 2.6314 HRD-naA -73.35, -47.8 66.65, 11.24 in-in-in SNCiii in-in ActLoopNT-in 2.8121 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.44, 8.45 APE9-dihe-na -84.75, -155.07 APE8-dihe-in -92.6, 123.69 APE8-rot-in 306.23 APE67-dihe-in -72.6, -7.76 -62.22, -39.85 APE12-dist-in 9.4745 APE11-dist-in 8.4917 APE10-dist-in 4.5618 APE9-dist-in 3.6262 None None None XRAY 2.2 0.177 0.226 A 313.0 273.0 1 26 26 0 [[38, 290]] 1.0 6pcw CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6PDIA P11309 32 305 313.0 OCJ:501 Type1 Active DFGin 6.1283 14.4792 BLAminus -126.87, 170.77 61.93, 81.48 -89.41, 13.26 285.32, 82.24 -64.21, -18.32 in-in in 8.8112 Saltbr-in 2.6199 HRD-naA -69.88, -49.72 68.62, 9.34 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.35, 18.43 APE9-dihe-na -84.8, -157.57 APE8-dihe-in -92.5, 120.51 APE8-rot-in 302.8 APE67-dihe-in -73.34, -11.57 -60.21, -38.03 APE12-dist-in 9.5818 APE11-dist-in 8.3694 APE10-dist-in 4.9704 APE9-dist-in 3.6699 None None None XRAY 1.85 0.163 0.193 A 313.0 274.0 0 26 26 0 [[38, 290]] 1.0 6pdi CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6PDNA P11309 32 305 313.0 OD4:900 Type1 Active DFGin 6.303 14.6787 BLAminus -127.91, 168.34 63.69, 84.1 -90.47, 15.7 284.14, 84.0 -75.26, -13.52 in-in in 8.8267 Saltbr-in 2.587 HRD-naA -70.55, -51.59 71.07, 6.03 in-in-in SNCiii in-in ActLoopNT-in 2.792 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.78, 23.66 APE9-dihe-na -88.42, -164.96 APE8-dihe-in -87.14, 123.03 APE8-rot-in 304.39 APE67-dihe-in -74.69, -11.36 -61.92, -39.09 APE12-dist-in 9.5899 APE11-dist-in 8.4061 APE10-dist-in 5.0533 APE9-dist-in 3.7386 None SEP261 SEP261 XRAY 2.4 0.19 0.223 A 313.0 270.0 4 26 26 0 [[38, 290]] 1.0 6pdn CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6PDOA P11309 35 305 313.0 OD1:501 Type1 Active DFGin 6.1292 14.2926 BLAminus -134.81, 169.87 61.89, 85.2 -91.49, 10.5 286.61, 82.45 -62.88, -17.93 in-in in 8.5877 Saltbr-in 2.7516 HRD-naA -69.22, -51.16 69.51, 6.24 in-in-in SNCiii in-in ActLoopNT-in 2.7835 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.34, 22.85 APE9-dihe-na -86.44, -166.55 APE8-dihe-in -83.99, 120.38 APE8-rot-in 303.74 APE67-dihe-in -70.14, -12.44 -58.32, -42.49 APE12-dist-in 9.5734 APE11-dist-in 8.3618 APE10-dist-in 4.7473 APE9-dist-in 3.7884 None None None XRAY 2.4 0.177 0.223 A 313.0 267.0 4 26 26 0 [[38, 290]] 1.0 6pdo CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6PDPA P11309 36 305 313.0 OBY:502 Type1 Active DFGin 6.1497 14.2213 BLAminus -129.84, 173.21 59.86, 93.48 -102.79, 22.43 282.95, 82.01 -70.26, -12.41 in-in in 8.422 Saltbr-in 2.7863 HRD-naA -67.94, -55.57 82.45, -11.52 in-in-in SNCiii in-in ActLoopNT-in 2.8844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.22, 34.63 APE9-dihe-na -88.55, -154.18 APE8-dihe-in -92.87, 123.61 APE8-rot-in 300.67 APE67-dihe-in -66.54, -13.53 -62.56, -42.85 APE12-dist-in 9.7024 APE11-dist-in 8.577 APE10-dist-in 5.7129 APE9-dist-in 4.1106 None None None XRAY 2.5 0.195 0.23 A 313.0 268.0 2 26 26 0 [[38, 290]] 1.0 6pdp CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6QXKB P11309 35 305 313.0 JKW:401 Type1 Active DFGin 6.1014 14.6091 BLAminus -124.57, 170.74 63.53, 81.45 -86.73, 15.75 286.17, 80.26 -64.12, -13.74 in-in in 8.945 Saltbr-in 2.6481 HRD-naA -69.55, -43.65 65.58, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.8414 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.01, 26.44 APE9-dihe-na -78.6, -156.19 APE8-dihe-in -94.84, 121.84 APE8-rot-in 303.08 APE67-dihe-in -71.43, -12.21 -59.33, -38.29 APE12-dist-in 9.8192 APE11-dist-in 8.4888 APE10-dist-in 5.4191 APE9-dist-in 3.6144 None None None XRAY 2.1 0.177 0.201 B 313.0 269.0 2 26 26 0 [[38, 290]] 1.0 6qxk CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R0HA P11309 33 305 313.0 8UB:403 Type1 Active DFGin 6.1948 14.5044 BLAminus -130.64, 169.15 64.03, 75.42 -86.88, 14.36 285.23, 74.81 -64.53, -17.19 in-in in 8.7633 Saltbr-in 2.7368 HRD-naA -71.57, -46.79 68.26, 11.15 in-in-in SNCiii in-in ActLoopNT-in 2.836 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.99, 20.76 APE9-dihe-na -80.37, -156.78 APE8-dihe-in -90.68, 121.72 APE8-rot-in 301.93 APE67-dihe-in -72.4, -8.98 -63.85, -37.03 APE12-dist-in 9.5338 APE11-dist-in 8.4986 APE10-dist-in 5.275 APE9-dist-in 3.6981 R250G SEP261 SEP261 XRAY 1.88 0.155 0.174 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r0h CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R0QA P11309 33 305 313.0 XGB:402 Type1 Active DFGin 6.1107 14.4727 BLAminus -124.88, 175.93 64.13, 67.05 -83.42, 11.36 282.83, 73.71 -70.16, -12.5 in-in in 8.8722 Saltbr-in 2.6597 HRD-naA -75.58, -44.16 66.56, 9.98 in-in-in SNCiii in-in ActLoopNT-in 2.8238 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.86, 18.75 APE9-dihe-na -80.22, -154.78 APE8-dihe-in -92.21, 122.35 APE8-rot-in 302.64 APE67-dihe-in -70.96, -8.32 -63.59, -38.0 APE12-dist-in 9.7252 APE11-dist-in 8.5877 APE10-dist-in 5.3973 APE9-dist-in 3.7047 R250G SEP261 SEP261 XRAY 1.7 0.166 0.177 A 313.0 267.0 6 26 26 0 [[38, 290]] 1.0 8r0q CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R0WA P11309 33 305 313.0 XGF:405 Type1 Active DFGin 5.9965 14.3841 BLAminus -131.73, 166.77 65.97, 82.46 -89.79, 16.41 289.35, 79.56 -63.02, -16.4 in-in in 8.8117 Saltbr-in 2.6426 HRD-naA -73.15, -45.35 65.43, 10.88 in-in-in SNCiii in-in ActLoopNT-in 2.8554 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.23, 17.26 APE9-dihe-na -81.93, -156.28 APE8-dihe-in -91.39, 121.88 APE8-rot-in 296.84 APE67-dihe-in -71.92, -8.94 -64.52, -38.27 APE12-dist-in 9.5591 APE11-dist-in 8.4794 APE10-dist-in 5.1163 APE9-dist-in 3.7129 R250G SEP261 SEP261 XRAY 1.95 0.167 0.201 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r0w CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R0YA P11309 33 305 313.0 XH3:402 Type1 Active DFGin 6.1278 14.5374 BLAminus -126.73, 169.7 64.58, 82.54 -91.76, 17.79 287.7, 78.06 -67.67, -13.51 in-in in 8.9569 Saltbr-in 2.6397 HRD-naA -71.78, -46.47 66.88, 6.9 in-in-in SNCiii in-in ActLoopNT-in 2.8623 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.85, 18.81 APE9-dihe-na -78.72, -154.37 APE8-dihe-in -95.58, 121.63 APE8-rot-in 303.84 APE67-dihe-in -73.42, -9.78 -59.84, -39.22 APE12-dist-in 9.539 APE11-dist-in 8.5542 APE10-dist-in 5.1289 APE9-dist-in 3.718 R250G SEP261 SEP261 XRAY 2.05 0.176 0.19 A 313.0 271.0 2 26 26 0 [[38, 290]] 1.0 8r0y CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R10A P11309 33 305 313.0 XGQ:401 Type1 Active DFGin 6.0079 14.5901 BLAminus -125.35, 178.02 53.25, 82.24 -86.16, 17.78 284.81, 76.38 -68.05, -10.88 in-in in 8.8956 Saltbr-in 2.6351 HRD-naA -73.59, -46.61 66.3, 8.94 in-in-in SNCiii in-in ActLoopNT-in 2.8079 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.14, 17.84 APE9-dihe-na -81.41, -153.47 APE8-dihe-in -91.91, 123.95 APE8-rot-in 303.23 APE67-dihe-in -72.41, -8.02 -63.66, -38.07 APE12-dist-in 9.9235 APE11-dist-in 8.4791 APE10-dist-in 5.2127 APE9-dist-in 3.6321 R250G SEP261 SEP261 XRAY 2.2 0.171 0.202 A 313.0 263.0 10 26 26 0 [[38, 290]] 1.0 8r10 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R18A P11309 33 305 313.0 XGK:402 Type1 Active DFGin 6.0344 14.3517 BLAminus -124.11, 175.65 61.57, 82.15 -90.26, 19.65 285.44, 75.92 -71.89, -10.87 in-in in 8.8263 Saltbr-in 2.5902 HRD-naA -75.08, -45.72 63.91, 12.1 in-in-in SNCiii in-in ActLoopNT-in 2.8326 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.79, 24.66 APE9-dihe-na -82.08, -152.26 APE8-dihe-in -93.08, 122.4 APE8-rot-in 301.75 APE67-dihe-in -73.31, -7.85 -63.76, -37.55 APE12-dist-in 9.8399 APE11-dist-in 8.5947 APE10-dist-in 5.5183 APE9-dist-in 3.68 R250G SEP261 SEP261 XRAY 1.89 0.161 0.186 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r18 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R1KA P11309 33 305 313.0 XHI:403 Type1 Active DFGin 6.2459 14.5708 BLAminus -130.32, 173.36 62.94, 72.15 -85.85, 16.37 285.53, 75.29 -71.64, -12.67 in-in in 8.7619 Saltbr-in 2.5021 HRD-naA -71.16, -48.89 70.04, 11.26 in-in-in SNCiii in-in ActLoopNT-in 2.8665 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.08, 4.88 APE9-dihe-na -84.34, -155.09 APE8-dihe-in -91.8, 121.7 APE8-rot-in 300.68 APE67-dihe-in -73.09, -10.26 -62.22, -37.87 APE12-dist-in 9.5411 APE11-dist-in 8.5475 APE10-dist-in 4.4357 APE9-dist-in 3.6882 R250G SEP261 SEP261 XRAY 1.95 0.177 0.192 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r1k CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R1NA P11309 34 305 313.0 XIT:401 Type1 Active DFGin 6.0573 14.5468 BLAminus -128.21, 174.49 58.15, 82.23 -87.85, 19.59 286.58, 72.67 -72.06, -10.27 in-in in 8.9084 Saltbr-in 2.7552 HRD-naA -72.06, -45.87 66.94, 8.6 in-in-in SNCiii in-in ActLoopNT-in 2.7691 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.59, 26.14 APE9-dihe-na -82.46, -153.43 APE8-dihe-in -96.65, 123.51 APE8-rot-in 298.16 APE67-dihe-in -70.63, -8.19 -63.53, -39.8 APE12-dist-in 9.783 APE11-dist-in 8.6205 APE10-dist-in 5.2058 APE9-dist-in 3.5907 R250G SEP261 SEP261 XRAY 2.21 0.163 0.192 A 313.0 272.0 0 26 26 0 [[38, 290]] 1.0 8r1n CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R1PA P11309 33 305 313.0 XIP:401 Type1 Active DFGin 6.0662 14.6184 BLAminus -128.97, 176.78 55.64, 82.37 -89.27, 14.78 284.77, 74.77 -64.96, -11.11 in-in in 8.8719 Saltbr-in 2.5719 HRD-naA -73.78, -46.66 71.64, 3.78 in-in-in SNCiii in-in ActLoopNT-in 2.8165 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.36, 22.63 APE9-dihe-na -86.45, -148.42 APE8-dihe-in -100.33, 122.66 APE8-rot-in 304.21 APE67-dihe-in -71.49, -6.91 -61.13, -41.84 APE12-dist-in 9.7904 APE11-dist-in 8.549 APE10-dist-in 4.924 APE9-dist-in 3.7558 R250G SEP261 SEP261 XRAY 2.45 0.178 0.206 A 313.0 269.0 4 26 26 0 [[38, 290]] 1.0 8r1p CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R1TA P11309 33 305 313.0 XIJ:402 Type1 Active DFGin 6.1286 14.5004 BLAminus -125.46, 175.2 59.64, 82.38 -89.86, 18.41 286.56, 77.1 -71.67, -11.65 in-in in 8.8527 Saltbr-in 2.6881 HRD-naA -72.26, -44.66 65.09, 8.72 in-in-in SNCiii in-in ActLoopNT-in 2.792 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.98, 13.92 APE9-dihe-na -81.53, -153.62 APE8-dihe-in -94.64, 124.09 APE8-rot-in 299.63 APE67-dihe-in -71.25, -8.49 -63.99, -39.26 APE12-dist-in 9.7963 APE11-dist-in 8.6337 APE10-dist-in 4.9525 APE9-dist-in 3.6603 R250G SEP261 SEP261 XRAY 2.0 0.16 0.179 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r1t CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R1WA P11309 33 305 313.0 XIW:402 Type1 Active DFGin 6.0093 14.6266 BLAminus -126.26, 175.45 55.83, 87.17 -92.67, 17.42 288.58, 76.06 -64.09, -13.07 in-in in 9.0119 Saltbr-in 2.6417 HRD-naA -70.36, -47.52 67.35, 8.76 in-in-in SNCiii in-in ActLoopNT-in 2.7892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.05, 16.58 APE9-dihe-na -79.71, -155.45 APE8-dihe-in -91.51, 124.54 APE8-rot-in 299.68 APE67-dihe-in -71.95, -9.45 -64.13, -40.15 APE12-dist-in 9.7391 APE11-dist-in 8.5662 APE10-dist-in 5.1338 APE9-dist-in 3.6453 R250G SEP261 SEP261 XRAY 2.15 0.176 0.204 A 313.0 270.0 3 26 26 0 [[38, 290]] 1.0 8r1w CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R25A P11309 33 305 313.0 XJL:402 Type1 Active DFGin 6.2238 14.6031 BLAminus -130.14, 174.3 56.41, 81.8 -90.04, 19.15 286.56, 75.38 -70.08, -10.25 in-in in 9.0651 Saltbr-in 2.4738 HRD-naA -71.77, -46.38 67.37, 8.2 in-in-in SNCiii in-in ActLoopNT-in 2.8145 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.33, 17.96 APE9-dihe-na -81.3, -151.78 APE8-dihe-in -98.77, 123.36 APE8-rot-in 301.63 APE67-dihe-in -70.17, -10.17 -64.54, -39.25 APE12-dist-in 9.6803 APE11-dist-in 8.6865 APE10-dist-in 4.9632 APE9-dist-in 3.6548 R250G SEP261 SEP261 XRAY 2.1 0.178 0.208 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r25 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8R27A P11309 33 305 313.0 XJW:402 Type1 Active DFGin 6.0133 14.3845 BLAminus -125.88, 174.13 60.12, 79.82 -86.61, 17.63 284.74, 75.1 -73.25, -8.78 in-in in 8.8799 Saltbr-in 2.7031 HRD-naA -74.94, -45.68 65.39, 9.33 in-in-in SNCiii in-in ActLoopNT-in 2.8424 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.2, 23.86 APE9-dihe-na -82.24, -153.87 APE8-dihe-in -93.36, 121.12 APE8-rot-in 300.79 APE67-dihe-in -70.77, -7.65 -61.34, -41.5 APE12-dist-in 9.7823 APE11-dist-in 8.5259 APE10-dist-in 5.2562 APE9-dist-in 3.6976 R250G SEP261 SEP261 XRAY 1.95 0.166 0.192 A 313.0 272.0 1 26 26 0 [[38, 290]] 1.0 8r27 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2BIKB P11309 33 305 313.0 BI1:1306 Type1 Active DFGin 6.2085 14.8544 BLAminus -129.68, 166.2 65.31, 82.3 -90.49, 20.51 284.24, 80.72 -71.93, -11.81 in-in in 8.7316 Saltbr-in 2.7718 HRD-naA -71.08, -48.28 72.24, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.8318 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.84, 26.95 APE9-dihe-na -83.77, -163.0 APE8-dihe-in -86.27, 123.71 APE8-rot-in 311.31 APE67-dihe-in -70.32, -9.34 -58.19, -44.58 APE12-dist-in 9.5525 APE11-dist-in 8.6863 APE10-dist-in 5.6274 APE9-dist-in 3.928 None SEP261 SEP261 XRAY 1.8 0.159 0.183 B 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 2bik CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2BILB P11309 33 306 313.0 BI1:1307 Type1 Active DFGin 5.907 14.6412 BLAminus -131.58, 166.0 69.48, 82.95 -91.3, 19.54 286.18, 78.18 -74.97, -10.91 in-in in 8.7854 Saltbr-in 2.6353 HRD-naA -70.92, -50.11 73.56, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.8565 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.49, 48.23 APE9-dihe-na -87.89, -146.11 APE8-dihe-in -91.43, 121.08 APE8-rot-in 306.95 APE67-dihe-in -71.1, -13.65 -55.02, -40.77 APE12-dist-in 9.4619 APE11-dist-in 8.2518 APE10-dist-in 6.34 APE9-dist-in 3.8583 None None None XRAY 2.55 0.195 0.248 B 313.0 274.0 0 26 26 0 [[38, 290]] 1.0 2bil CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2BZHB P11309 32 306 313.0 HB1:1307 Type1 Active DFGin 6.241 14.7174 BLAminus -128.91, 169.67 62.16, 81.6 -86.25, 13.92 287.87, 80.39 -66.46, -13.69 in-in in 8.8333 Saltbr-in 2.7881 HRD-naA -70.2, -46.33 68.04, 6.62 in-in-in SNCiii in-in ActLoopNT-in 2.86 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.94, 27.94 APE9-dihe-na -80.38, -157.42 APE8-dihe-in -90.55, 119.15 APE8-rot-in 302.06 APE67-dihe-in -68.66, -8.15 -56.91, -42.45 APE12-dist-in 9.5819 APE11-dist-in 8.5307 APE10-dist-in 5.5946 APE9-dist-in 3.6731 R250G None None XRAY 1.9 0.159 0.19 B 313.0 275.0 0 26 26 0 [[38, 290]] 1.0 2bzh CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2BZIB P11309 33 305 313.0 DW2:1306 Type1 Active DFGin 6.2667 14.8353 BLAminus -123.34, 165.34 66.36, 86.11 -93.21, 22.23 286.33, 78.94 -70.39, -16.59 in-in in 8.8727 Saltbr-in 2.7797 HRD-naA -72.04, -45.2 68.6, 5.31 in-in-in SNCiii in-in ActLoopNT-in 2.857 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.77, 39.69 APE9-dihe-na -92.21, -159.18 APE8-dihe-in -82.89, 124.01 APE8-rot-in 305.62 APE67-dihe-in -65.59, -13.31 -61.02, -47.85 APE12-dist-in 9.4556 APE11-dist-in 8.486 APE10-dist-in 5.6923 APE9-dist-in 3.9382 R250G SEP261 SEP261 XRAY 1.9 0.218 0.265 B 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 2bzi CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2BZJA P11309 33 305 313.0 ME3:1306 Type1 Active DFGin 6.2938 14.8461 BLAminus -129.09, 166.61 64.15, 83.62 -93.36, 13.13 283.19, 80.4 -68.93, -14.93 in-in in 8.9144 Saltbr-in 2.5247 HRD-naA -66.52, -47.22 65.13, 9.09 in-in-in SNCiii in-in ActLoopNT-in 2.7732 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -114.4, 32.87 APE9-dihe-na -91.23, -169.99 APE8-dihe-in -72.16, 120.4 APE8-rot-in 307.22 APE67-dihe-in -77.22, -2.13 -52.79, -48.09 APE12-dist-in 9.3195 APE11-dist-in 8.7496 APE10-dist-in 5.5282 APE9-dist-in 3.9837 R250G None None XRAY 2.05 0.185 0.221 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 2bzj CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2C3IB P11309 37 305 313.0 IYZ:1306 Type1 Active DFGin 6.3264 14.7526 BLAminus -127.31, 169.9 65.35, 81.96 -93.82, 15.98 286.0, 76.19 -64.86, -18.96 in-in in 8.5925 Saltbr-in 2.708 HRD-naA -73.6, -47.48 67.75, 10.67 in-in-in SNCiii in-in ActLoopNT-in 2.9203 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.67, 24.77 APE9-dihe-na -79.26, -156.38 APE8-dihe-in -92.5, 121.61 APE8-rot-in 301.77 APE67-dihe-in -67.73, -10.57 -57.93, -41.83 APE12-dist-in 9.5195 APE11-dist-in 8.5652 APE10-dist-in 5.3265 APE9-dist-in 3.7771 R250G None None XRAY 1.9 0.187 0.219 B 313.0 266.0 3 26 26 0 [[38, 290]] 1.0 2c3i CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 2OI4X P11309 32 306 313.0 JM1:1000 Type1 Active DFGin 6.3452 14.8125 BLAminus -127.98, 160.81 73.35, 71.74 -86.12, 11.96 287.24, 83.24 -76.7, -11.05 in-in in 9.0524 Saltbr-in 2.725 HRD-naA -64.97, -46.27 67.59, 4.83 in-in-in SNCiii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.16, 42.39 APE9-dihe-na -92.81, -143.09 APE8-dihe-in -99.99, 118.85 APE8-rot-in 297.17 APE67-dihe-in -72.38, -14.41 -46.73, -45.08 APE12-dist-in 9.4593 APE11-dist-in 8.8662 APE10-dist-in 5.9919 APE9-dist-in 3.671 R250G None None XRAY 2.2 0.192 0.244 X 313.0 275.0 0 26 26 0 [[38, 290]] 1.0 2oi4 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3BWFA P11309 33 305 313.0 DWC:315 Type1 Active DFGin 6.1521 14.7614 BLAminus -130.15, 160.75 70.46, 85.62 -95.56, 18.11 287.26, 79.6 -68.63, -18.22 in-in in 9.0395 Saltbr-in 2.6434 HRD-naA -63.89, -51.3 70.35, 5.77 in-in-in SNCiii in-in ActLoopNT-in 2.7913 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.65, 13.48 APE9-dihe-na -90.68, -158.0 APE8-dihe-in -83.6, 122.9 APE8-rot-in 307.99 APE67-dihe-in -60.33, -14.69 -56.04, -57.34 APE12-dist-in 9.2482 APE11-dist-in 8.6585 APE10-dist-in 5.0955 APE9-dist-in 3.9038 R250G None None XRAY 2.35 0.171 0.225 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 3bwf CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5MZLA P11309 33 305 313.0 8ET:401 Type1 Active DFGin 6.0702 14.4143 BLAminus -131.62, 169.01 61.49, 83.12 -91.63, 17.39 285.49, 78.9 -67.71, -14.16 in-in in 8.7664 Saltbr-in 2.5894 HRD-naA -71.92, -48.75 69.25, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.7988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.79, 22.06 APE9-dihe-na -80.91, -155.94 APE8-dihe-in -90.97, 120.03 APE8-rot-in 302.78 APE67-dihe-in -70.3, -10.66 -61.44, -39.24 APE12-dist-in 9.7338 APE11-dist-in 8.5092 APE10-dist-in 5.304 APE9-dist-in 3.6957 R250G None None XRAY 1.955 0.158 0.183 A 313.0 269.0 4 26 26 0 [[38, 290]] 1.0 5mzl CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4NA P11309 33 305 313.0 8M8:401 Type1 Active DFGin 6.1249 14.6169 BLAminus -129.29, 170.82 62.47, 79.55 -88.93, 16.9 284.33, 80.08 -68.56, -10.77 in-in in 8.9316 Saltbr-in 2.5396 HRD-naA -74.48, -44.52 65.43, 11.21 in-in-in SNCiii in-in ActLoopNT-in 2.7939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.35, 17.93 APE9-dihe-na -79.41, -153.04 APE8-dihe-in -96.16, 122.12 APE8-rot-in 301.83 APE67-dihe-in -69.32, -12.36 -62.25, -40.05 APE12-dist-in 9.5995 APE11-dist-in 8.5712 APE10-dist-in 5.2029 APE9-dist-in 3.7045 R250G None None XRAY 2.09 0.161 0.188 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4n CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4OA P11309 33 305 313.0 8MB:401 Type1 Active DFGin 6.0998 14.6005 BLAminus -128.07, 170.32 63.44, 81.51 -90.0, 20.39 288.36, 74.25 -70.54, -10.71 in-in in 8.8244 Saltbr-in 2.5204 HRD-naA -74.44, -43.81 65.23, 5.78 in-in-in SNCiii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.86, 22.33 APE9-dihe-na -84.24, -148.33 APE8-dihe-in -98.01, 118.97 APE8-rot-in 304.06 APE67-dihe-in -72.76, -7.0 -59.82, -38.64 APE12-dist-in 9.676 APE11-dist-in 8.6398 APE10-dist-in 5.1918 APE9-dist-in 3.7491 R250G None None XRAY 2.22 0.182 0.196 A 313.0 271.0 2 26 26 0 [[38, 290]] 1.0 5n4o CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4RA P11309 33 305 313.0 8MQ:402 Type1 Active DFGin 6.1615 14.6842 BLAminus -127.95, 172.44 62.9, 73.52 -86.51, 10.58 283.66, 75.96 -65.07, -11.8 in-in in 8.8652 Saltbr-in 2.7964 HRD-naA -74.57, -43.89 66.05, 7.98 in-in-in SNCiii in-in ActLoopNT-in 2.8278 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.44, 14.9 APE9-dihe-na -80.8, -159.32 APE8-dihe-in -87.99, 122.23 APE8-rot-in 303.81 APE67-dihe-in -72.42, -8.25 -61.99, -38.57 APE12-dist-in 9.6804 APE11-dist-in 8.5666 APE10-dist-in 5.225 APE9-dist-in 3.6808 R250G None None XRAY 2.13 0.162 0.193 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4r CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4UA P11309 34 305 313.0 8MZ:401 Type1 Active DFGin 6.1707 14.6229 BLAminus -127.06, 173.77 59.59, 86.28 -91.8, 19.55 284.63, 76.39 -67.81, -14.94 in-in in 8.939 Saltbr-in 2.6625 HRD-naA -76.79, -43.95 67.64, 10.17 in-in-in SNCiii in-in ActLoopNT-in 2.7659 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.95, 11.58 APE9-dihe-na -74.78, -161.25 APE8-dihe-in -87.42, 123.39 APE8-rot-in 302.63 APE67-dihe-in -68.48, -11.24 -64.0, -41.0 APE12-dist-in 9.5659 APE11-dist-in 8.4312 APE10-dist-in 5.1177 APE9-dist-in 3.6356 R250G None None XRAY 2.202 0.165 0.198 A 313.0 272.0 0 26 26 0 [[38, 290]] 1.0 5n4u CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4VA P11309 33 305 313.0 8MW:401 Type1 Active DFGin 6.1863 14.5848 BLAminus -124.08, 176.44 56.8, 80.25 -87.01, 16.92 283.21, 72.16 -68.4, -12.83 in-in in 8.8997 Saltbr-in 2.6276 HRD-naA -74.68, -46.5 67.92, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.8775 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.8, 18.81 APE9-dihe-na -79.43, -156.57 APE8-dihe-in -90.82, 123.02 APE8-rot-in 301.39 APE67-dihe-in -72.01, -7.09 -64.55, -37.95 APE12-dist-in 9.8641 APE11-dist-in 8.5735 APE10-dist-in 5.3957 APE9-dist-in 3.6541 R250G None None XRAY 1.85 0.165 0.187 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4v CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4XA P11309 33 305 313.0 8MT:401 Type1 Active DFGin 6.1755 14.6336 BLAminus -130.04, 168.92 67.47, 77.08 -88.95, 14.23 284.67, 77.55 -69.57, -11.46 in-in in 8.8767 Saltbr-in 2.7977 HRD-naA -75.83, -47.71 70.47, 10.64 in-in-in SNCiii in-in ActLoopNT-in 2.8155 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.28, 25.38 APE9-dihe-na -81.19, -156.58 APE8-dihe-in -90.87, 123.23 APE8-rot-in 301.93 APE67-dihe-in -70.8, -10.69 -63.86, -38.58 APE12-dist-in 9.6753 APE11-dist-in 8.5636 APE10-dist-in 5.5271 APE9-dist-in 3.6878 R250G None None XRAY 2.2 0.178 0.215 A 313.0 272.0 1 26 26 0 [[38, 290]] 1.0 5n4x CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4YA P11309 33 305 313.0 8N5:401 Type1 Active DFGin 6.0422 14.7244 BLAminus -130.6, 168.91 64.51, 83.34 -90.72, 17.65 288.76, 80.39 -65.28, -8.11 in-in in 9.034 Saltbr-in 2.9653 HRD-naA -68.66, -50.14 72.28, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.849 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.0, 26.36 APE9-dihe-na -86.43, -160.39 APE8-dihe-in -83.05, 121.49 APE8-rot-in 308.67 APE67-dihe-in -70.07, -12.6 -65.48, -36.81 APE12-dist-in 9.8289 APE11-dist-in 8.5102 APE10-dist-in 5.511 APE9-dist-in 3.916 R250G None None XRAY 2.56 0.177 0.218 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4y CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N4ZA P11309 34 305 313.0 8MK:401 Type1 Active DFGin 6.0929 14.5863 BLAminus -128.45, 169.26 63.69, 88.15 -96.51, 19.04 288.58, 75.49 -67.41, -11.99 in-in in 8.9657 Saltbr-in 2.5723 HRD-naA -72.17, -46.94 66.82, 8.56 in-in-in SNCiii in-in ActLoopNT-in 2.8563 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.32, 24.78 APE9-dihe-na -81.23, -155.7 APE8-dihe-in -89.42, 121.2 APE8-rot-in 306.52 APE67-dihe-in -67.82, -10.0 -59.95, -43.55 APE12-dist-in 9.5784 APE11-dist-in 8.5279 APE10-dist-in 5.3815 APE9-dist-in 3.7131 R250G None None XRAY 2.257 0.18 0.208 A 313.0 272.0 0 26 26 0 [[38, 290]] 1.0 5n4z CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N50A P11309 33 305 313.0 8MN:401 Type1 Active DFGin 6.0402 14.6666 BLAminus -127.77, 166.5 68.05, 82.07 -89.1, 18.46 287.73, 79.6 -66.42, -13.96 in-in in 8.9208 Saltbr-in 2.5541 HRD-naA -72.47, -47.69 66.88, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.8127 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.17, 14.92 APE9-dihe-na -76.58, -153.55 APE8-dihe-in -94.04, 123.44 APE8-rot-in 302.17 APE67-dihe-in -70.74, -9.3 -65.25, -38.14 APE12-dist-in 9.5673 APE11-dist-in 8.4941 APE10-dist-in 5.16 APE9-dist-in 3.6772 R250G None None XRAY 1.92 0.16 0.18 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n50 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N51A P11309 33 305 313.0 8N8:401 Type1 Active DFGin 6.14 14.6258 BLAminus -127.02, 176.35 56.56, 82.77 -90.34, 20.5 285.79, 74.98 -67.87, -15.26 in-in in 8.787 Saltbr-in 2.6446 HRD-naA -74.16, -46.81 67.83, 8.58 in-in-in SNCiii in-in ActLoopNT-in 2.8023 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.83, 20.8 APE9-dihe-na -83.46, -153.2 APE8-dihe-in -92.57, 121.76 APE8-rot-in 302.99 APE67-dihe-in -70.78, -10.06 -61.78, -40.18 APE12-dist-in 9.7216 APE11-dist-in 8.5406 APE10-dist-in 5.1634 APE9-dist-in 3.7372 R250G SEP261 SEP261 XRAY 2.118 0.182 0.207 A 313.0 269.0 4 26 26 0 [[38, 290]] 1.0 5n51 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N52A P11309 33 305 313.0 8N2:401 Type1 Active DFGin 6.0542 14.4946 BLAminus -128.92, 172.68 61.78, 83.49 -88.53, 18.1 285.87, 76.88 -62.86, -14.96 in-in in 8.8791 Saltbr-in 2.8 HRD-naA -72.66, -45.02 65.77, 9.07 in-in-in SNCiii in-in ActLoopNT-in 2.8047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.64, 23.49 APE9-dihe-na -83.54, -155.05 APE8-dihe-in -91.57, 124.16 APE8-rot-in 301.67 APE67-dihe-in -71.63, -7.35 -64.67, -40.35 APE12-dist-in 9.7762 APE11-dist-in 8.5757 APE10-dist-in 5.2818 APE9-dist-in 3.6764 R250G None None XRAY 2.252 0.172 0.21 A 313.0 268.0 5 26 26 0 [[38, 290]] 1.0 5n52 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N5LA P11309 33 305 313.0 8NZ:401 Type1 Active DFGin 6.1605 14.53 BLAminus -127.06, 174.1 60.7, 73.46 -86.15, 14.2 284.46, 73.6 -71.56, -14.64 in-in in 8.9176 Saltbr-in 2.7811 HRD-naA -74.26, -45.32 66.26, 11.22 in-in-in SNCiii in-in ActLoopNT-in 2.8951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.1, 16.72 APE9-dihe-na -75.29, -159.06 APE8-dihe-in -90.45, 122.93 APE8-rot-in 300.5 APE67-dihe-in -72.6, -9.34 -63.53, -38.45 APE12-dist-in 9.6906 APE11-dist-in 8.485 APE10-dist-in 5.2932 APE9-dist-in 3.5687 R250G SEP261 SEP261 XRAY 1.97 0.162 0.195 A 313.0 272.0 1 26 26 0 [[38, 290]] 1.0 5n5l CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5N5MA P11309 33 305 313.0 8O8:401 Type1 Active DFGin 6.0953 14.7209 BLAminus -128.4, 173.39 60.49, 81.96 -90.76, 15.73 290.29, 74.98 -68.5, -8.46 in-in in 9.0069 Saltbr-in 2.7752 HRD-naA -74.58, -47.17 67.22, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.8408 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.85, 20.79 APE9-dihe-na -81.68, -154.64 APE8-dihe-in -91.98, 123.1 APE8-rot-in 303.04 APE67-dihe-in -72.34, -6.29 -62.86, -39.4 APE12-dist-in 9.6452 APE11-dist-in 8.5152 APE10-dist-in 5.2422 APE9-dist-in 3.6671 R250G SEP261 SEP261 XRAY 2.21 0.168 0.205 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n5m CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 5NDTA P11309 33 305 313.0 8UB:402 Type1 Active DFGin 6.114 14.7046 BLAminus -128.77, 171.81 63.42, 78.28 -87.87, 17.81 284.74, 79.81 -71.9, -9.72 in-in in 8.8817 Saltbr-in 2.6322 HRD-naA -72.09, -45.67 67.68, 10.44 in-in-in SNCiii in-in ActLoopNT-in 2.837 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.91, 24.5 APE9-dihe-na -81.02, -156.58 APE8-dihe-in -91.09, 121.22 APE8-rot-in 302.75 APE67-dihe-in -68.43, -10.6 -60.72, -41.46 APE12-dist-in 9.788 APE11-dist-in 8.5839 APE10-dist-in 5.4022 APE9-dist-in 3.7192 R250G None None XRAY 1.985 0.162 0.194 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5ndt CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7Z6UA P11309 33 305 313.0 IJB:402 Type1 Active DFGin 6.2708 14.4925 BLAminus -123.62, 176.91 53.69, 81.97 -85.84, 21.16 285.55, 68.27 -70.71, -12.85 in-in in 8.7429 Saltbr-in 2.7682 HRD-naA -72.34, -45.38 65.34, 4.41 in-in-in SNCiii in-in ActLoopNT-in 2.7594 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.54, 10.63 APE9-dihe-na -83.63, -150.44 APE8-dihe-in -98.54, 120.92 APE8-rot-in 299.64 APE67-dihe-in -72.4, -8.48 -60.83, -39.47 APE12-dist-in 9.7699 APE11-dist-in 8.6298 APE10-dist-in 4.6662 APE9-dist-in 3.71 R250G SEP261 SEP261 XRAY 2.28 0.163 0.191 A 313.0 268.0 5 26 26 0 [[38, 290]] 1.0 7z6u CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3CXWA P11309 33 306 313.0 7CP:501 Type1 Active DFGin 6.1536 14.6175 BLAminus -123.7, 175.96 66.3, 77.59 -92.53, 20.47 286.96, 76.96 -73.25, -11.74 in-in in 8.9096 Saltbr-in 2.6276 HRD-naA -73.02, -49.99 67.21, 12.05 in-in-in SNCiii in-in ActLoopNT-in 2.8094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.29, 21.64 APE9-dihe-na -81.37, -152.87 APE8-dihe-in -93.72, 121.7 APE8-rot-in 305.98 APE67-dihe-in -70.04, -11.91 -61.57, -39.54 APE12-dist-in 9.572 APE11-dist-in 8.3971 APE10-dist-in 5.2889 APE9-dist-in 3.6214 R250G None None XRAY 2.1 0.166 0.206 A 314.0 272.0 2 26 26 0 [[38, 290]] 1.0 3cxw CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3CY2A P11309 33 305 313.0 MB9:501 Type1 Active DFGin 6.1626 14.6449 BLAminus -126.41, 176.21 64.46, 78.27 -92.72, 18.89 288.13, 73.75 -67.98, -11.93 in-in in 8.9051 Saltbr-in 2.5685 HRD-naA -71.13, -52.84 70.37, 7.17 in-in-in SNCiii in-in ActLoopNT-in 2.8534 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.27, 21.57 APE9-dihe-na -78.39, -153.2 APE8-dihe-in -93.22, 122.03 APE8-rot-in 307.28 APE67-dihe-in -67.99, -12.82 -60.45, -42.49 APE12-dist-in 9.5435 APE11-dist-in 8.4795 APE10-dist-in 5.3954 APE9-dist-in 3.5574 R250G None None XRAY 2.01 0.169 0.199 A 314.0 271.0 2 26 26 0 [[38, 290]] 1.0 3cy2 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3CY3A P11309 33 305 313.0 JN5:501 Type1 Active DFGin 6.3033 14.4186 BLAminus -119.65, 175.12 56.83, 74.92 -82.21, 12.5 285.74, 75.76 -70.58, -7.45 in-in in 8.7561 Saltbr-in 2.5596 HRD-naA -67.55, -45.89 68.27, 6.37 in-in-in SNCiii in-in ActLoopNT-in 2.8172 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.11, 26.07 APE9-dihe-na -79.4, -161.09 APE8-dihe-in -89.18, 123.7 APE8-rot-in 304.7 APE67-dihe-in -65.31, -15.75 -62.09, -40.0 APE12-dist-in 9.6746 APE11-dist-in 8.4856 APE10-dist-in 5.5666 APE9-dist-in 3.6228 R250G SEP261 SEP261 XRAY 2.15 0.165 0.205 A 314.0 271.0 2 26 26 0 [[38, 290]] 1.0 3cy3 CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4RPVA P11309 33 305 313.0 3UR:401 Type1 Active DFGin 5.9582 14.8542 BLAminus -145.63, 161.43 69.99, 88.37 -103.98, 21.07 280.48, 100.64 -81.25, 11.11 in-in in 8.9443 Saltbr-in 2.804 HRD-naA -54.49, -51.71 77.62, -1.62 in-in-in SNCiii in-in ActLoopNT-in 2.6013 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.21, 30.75 APE9-dihe-na -100.7, -169.57 APE8-dihe-in -63.18, 128.08 APE8-rot-in 302.06 APE67-dihe-in -40.53, -14.86 -60.72, -74.04 APE12-dist-in 9.5906 APE11-dist-in 8.8948 APE10-dist-in 5.655 APE9-dist-in 4.1527 None None None XRAY 3.05 0.229 0.273 A 410.0 273.0 0 26 26 0 [[38, 290]] 1.0 4rpv CAMK_PIM1_HUMAN CAMK 9.3e-65 224.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 8AFRA P11309 33 305 313.0 M0F:401 Type1 Active DFGin 6.0243 14.4056 BLAminus -126.46, 177.16 55.61, 83.44 -89.48, 19.88 284.93, 74.96 -67.33, -13.52 in-in in 8.8307 Saltbr-in 2.6484 HRD-naA -72.52, -48.51 66.56, 10.77 in-in-in SNCiii in-in ActLoopNT-in 2.8149 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.4, 19.87 APE9-dihe-na -78.39, -149.93 APE8-dihe-in -97.85, 123.61 APE8-rot-in 301.25 APE67-dihe-in -68.16, -10.25 -64.9, -40.75 APE12-dist-in 9.7271 APE11-dist-in 8.4666 APE10-dist-in 5.304 APE9-dist-in 3.645 R250G SEP261 SEP261 XRAY 2.15 0.166 0.191 A 309.0 264.0 7 26 26 0 [[38, 290]] 1.0 8afr CAMK_PIM1_HUMAN CAMK 3.1e-62 216.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4ALUA P11309 33 306 313.0 79O:1308 Type1 Active DFGin 6.0396 14.4546 BLAminus -129.3, 164.2 71.61, 87.87 -98.95, 24.33 283.93, 80.99 -80.29, 2.07 in-in in 8.7471 Saltbr-in 2.5495 HRD-naA -75.13, -46.19 78.28, -3.97 in-in-in SNCiii in-in ActLoopNT-in 2.8293 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.43, 41.36 APE9-dihe-na -93.61, -144.58 APE8-dihe-in -101.6, 125.74 APE8-rot-in 300.81 APE67-dihe-in -62.7, -19.8 -64.97, -44.76 APE12-dist-in 9.6233 APE11-dist-in 8.6017 APE10-dist-in 5.7263 APE9-dist-in 3.7807 None None None XRAY 2.6 0.184 0.248 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 4alu CAMK_PIM1_HUMAN CAMK 2.7e-64 222.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3T9IA P11309 33 306 313.0 3T9:401 Type1.5_Back Active DFGin 6.5428 14.2947 BLAminus -132.77, 172.96 59.67, 82.28 -96.48, 17.83 287.7, 76.66 -65.3, -19.74 in-in in 8.4349 Saltbr-in 2.7571 HRD-naA -69.28, -50.32 73.93, -9.03 in-in-in SNCiii in-in ActLoopNT-in 2.8337 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.31, 28.32 APE9-dihe-na -97.99, -160.13 APE8-dihe-in -83.72, 117.37 APE8-rot-in 302.02 APE67-dihe-in -69.04, -9.18 -56.37, -42.61 APE12-dist-in 9.7353 APE11-dist-in 8.6561 APE10-dist-in 5.1983 APE9-dist-in 4.2807 None SEP261 SEP261 XRAY 2.6 0.165 0.227 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 3t9i CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6AYDA P11309 34 305 313.0 C2J:401 Type1.5_Back Active DFGin 6.2253 14.5726 BLAminus -129.9, 167.94 69.26, 93.71 -101.76, 29.48 284.65, 86.99 -77.7, -11.94 in-in in 8.4989 Saltbr-in 2.6944 HRD-naA -64.89, -48.59 73.72, 7.41 in-in-in SNCiii in-in ActLoopNT-in 2.7192 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.07, 29.72 APE9-dihe-na -90.29, -149.58 APE8-dihe-in -90.3, 121.0 APE8-rot-in 309.33 APE67-dihe-in -70.19, -4.08 -54.85, -49.52 APE12-dist-in 9.7574 APE11-dist-in 8.5952 APE10-dist-in 5.4358 APE9-dist-in 4.0665 R250G None None XRAY 3.0 0.171 0.23 A 334.0 272.0 0 26 26 0 [[38, 290]] 1.0 6ayd CAMK_PIM1_HUMAN CAMK 1.9e-64 223.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4RBLA P11309 33 305 313.0 3O7:401 Type1 Inactive DFGin 6.1855 14.6322 ABAminus -123.28, -49.04 -102.92, 101.34 -86.59, 10.95 288.26, 82.24 -66.9, -9.47 in-in in 8.7086 Saltbr-in 2.5498 HRD-naA -76.77, -47.35 72.65, 1.38 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.2, 7.15 APE9-dihe-na -86.69, -159.73 APE8-dihe-in -86.44, 135.53 APE8-rot-in 335.24 APE67-dihe-in -50.84, -15.83 -62.51, -62.82 APE12-dist-in 9.2624 APE11-dist-in 8.5648 APE10-dist-in 4.3791 APE9-dist-in 3.874 None SEP261 SEP261 XRAY 2.55 0.191 0.249 A 289.0 272.0 1 26 26 0 [[38, 290]] 1.0 4rbl CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4RC2A P11309 33 305 313.0 3O8:401 Type1 Inactive DFGin 6.1514 14.4868 ABAminus -124.35, -31.66 -113.65, 105.77 -88.14, 13.2 287.98, 83.78 -66.51, -15.85 in-in in 8.8722 Saltbr-in 2.534 HRD-naA -72.15, -49.17 67.29, 8.38 in-in-in SNCiii in-in ActLoopNT-in 2.7926 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.36, 8.25 APE9-dihe-na -77.04, -152.99 APE8-dihe-in -93.85, 131.35 APE8-rot-in 322.71 APE67-dihe-in -71.49, -6.88 -57.98, -44.79 APE12-dist-in 9.4324 APE11-dist-in 8.5203 APE10-dist-in 4.7174 APE9-dist-in 3.8077 None SEP261 SEP261 XRAY 2.096 0.21 0.246 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 4rc2 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4RC3A P11309 33 305 313.0 3OA:401 Type1 Inactive DFGin 6.1312 14.7301 ABAminus -124.18, -44.55 -102.49, 107.8 -86.08, 9.84 283.97, 82.66 -66.94, -13.06 in-in in 8.9316 Saltbr-in 2.7278 HRD-naA -74.64, -46.7 68.78, 5.57 in-in-in SNCiii in-in ActLoopNT-in 2.7168 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.55, 7.68 APE9-dihe-na -87.91, -151.36 APE8-dihe-in -94.35, 131.18 APE8-rot-in 325.68 APE67-dihe-in -63.89, -8.14 -60.26, -51.45 APE12-dist-in 9.479 APE11-dist-in 8.6351 APE10-dist-in 4.6757 APE9-dist-in 3.9424 None SEP261 SEP261 XRAY 2.338 0.192 0.222 A 289.0 272.0 1 26 26 0 [[38, 290]] 1.0 4rc3 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4RC4A P11309 33 305 313.0 3OK:401 Type1 Inactive DFGin 6.1945 14.5075 ABAminus -123.13, -33.74 -113.37, 104.45 -91.23, 9.07 284.92, 83.68 -71.27, -6.47 in-in in 8.6118 Saltbr-in 2.7351 HRD-naA -68.9, -48.63 75.17, 7.81 in-in-in SNCiii in-in ActLoopNT-in 2.8636 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.62, -3.25 APE9-dihe-na -70.99, -164.38 APE8-dihe-in -82.7, 141.94 APE8-rot-in 331.47 APE67-dihe-in -56.62, -19.58 -59.05, -56.98 APE12-dist-in 9.1914 APE11-dist-in 8.5877 APE10-dist-in 4.5075 APE9-dist-in 3.8584 None SEP261 SEP261 XRAY 2.651 0.191 0.241 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 4rc4 CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4I41A P11309 33 305 313.0 MIX:500,MIX:501 Type1,Allosteric Inactive DFGin 6.1399 14.4159 ABAminus -121.87, -36.78 -115.75, 100.81 -88.41, 10.15 289.07, 75.39 -54.5, -25.74 in-in in 8.6342 Saltbr-in 2.7561 HRD-naA -69.84, -46.43 70.52, 12.32 in-in-out SNCiio in-out ActLoopNT-in 2.9176 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -124.01, -14.74 APE9-dihe-na -57.33, 178.24 APE8-dihe-in -71.04, 142.33 APE8-rot-out 6.4 APE67-dihe-in -51.91, -16.42 -63.07, -52.85 APE12-dist-in 9.1226 APE11-dist-in 8.5821 APE10-dist-in 4.5899 APE9-dist-in 3.8828 None SEP261 SEP261 XRAY 2.7 0.2 0.249 A 281.0 273.0 0 26 26 0 [[38, 290]] 1.0 4i41 CAMK_PIM1_HUMAN CAMK 2.7e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 7OOXA P11309 1 305 313.0 No_ligand No_ligand Inactive DFGin 6.0077 14.4258 BLAminus -128.2, 171.48 64.26, 84.06 -90.51, 19.09 289.76, 88.29 -67.14, -14.45 in-in in 8.8933 Saltbr-in 2.5304 HRD-naA -69.11, -49.22 70.21, 6.96 in-in-out SNCiio in-out ActLoopNT-in 2.8525 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -112.93, -2.13 APE9-dihe-na -73.5, 169.82 APE8-dihe-in -80.91, 158.93 APE8-rot-out 67.73 APE67-dihe-in -74.5, -10.73 -58.29, -40.88 APE12-dist-in 9.6067 APE11-dist-in 8.8847 APE10-dist-in 4.9932 APE9-dist-in 5.4364 None None None XRAY 1.97 0.181 0.222 A 313.0 284.0 0 26 26 0 [[38, 290]] 1.0 7oox CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 3DCVA P11309 32 305 313.0 55E:500 Type1 Inactive DFGin 6.4113 14.6785 BLAminus -130.48, 168.13 69.03, 78.23 -92.76, 18.93 285.58, 71.29 -63.83, -15.25 in-in in 8.3124 Saltbr-in 2.5592 HRD-naA -64.55, -50.54 72.29, 1.73 in-in-out SNCiio in-out ActLoopNT-in 2.876 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -106.61, -25.99 APE9-dihe-na -54.65, -172.57 APE8-dihe-in -80.08, 136.57 APE8-rot-out 118.16 APE67-dihe-in -59.26, -8.45 -62.5, -57.95 APE12-dist-in 9.5381 APE11-dist-in 8.9721 APE10-dist-in 4.6762 APE9-dist-in 3.8897 None SEP261 SEP261 XRAY 2.7 0.182 0.234 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 3dcv CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 6KZIA P11309 33 305 313.0 RTX:401 Type1 Inactive DFGin 6.0118 14.7309 BLBminus -130.32, 166.69 73.68, 82.71 -88.65, -171.62 289.43, 86.65 20.03, 81.34 in-in in 8.9794 Saltbr-in 2.742 HRD-naA -68.55, -45.07 65.35, 8.38 in-in-in SNCiii in-in ActLoopNT-in 2.7184 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.04, 49.18 APE9-dihe-na -108.43, -149.21 APE8-dihe-in -96.99, 121.09 APE8-rot-in 319.52 APE67-dihe-in -60.06, -16.31 -54.82, -52.12 APE12-dist-in 9.3829 APE11-dist-in 8.3363 APE10-dist-in 5.48 APE9-dist-in 4.0226 None SEP261 SEP261 XRAY 2.8 0.173 0.233 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6kzi CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4IAAA P11309 33 305 313.0 RTZ:401 Type1 Inactive DFGin 6.018 14.534 None -118.73, -143.64 -58.0, 140.84 -105.0, 12.55 279.89, 91.42 -63.74, -38.82 in-in in 8.9764 Saltbr-in 2.4263 HRD-naA -66.74, -45.93 76.57, 1.9 in-in-in SNCiii in-in ActLoopNT-in 2.8243 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -101.97, 36.36 APE9-dihe-na -102.7, -148.72 APE8-dihe-in -99.25, 120.44 APE8-rot-in 325.38 APE67-dihe-in -56.81, -14.63 -51.76, -61.55 APE12-dist-in 9.3212 APE11-dist-in 8.4746 APE10-dist-in 4.9412 APE9-dist-in 4.319 None SEP261 SEP261 XRAY 2.85 0.187 0.231 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 4iaa CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 4XH6A P11309 33 305 313.0 HUL:401 Type1 Inactive DFGin 6.0669 14.6256 None -113.12, -75.74 -81.94, 104.4 -86.86, 17.15 286.29, 78.0 -66.66, -16.93 in-in in 8.963 Saltbr-in 2.6759 HRD-naA -71.75, -47.81 68.98, 9.54 in-in-in SNCiii in-in ActLoopNT-in 2.8264 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.53, 35.49 APE9-dihe-na -89.22, -153.74 APE8-dihe-in -92.85, 123.83 APE8-rot-in 304.19 APE67-dihe-in -63.31, -10.32 -62.77, -45.27 APE12-dist-in 9.5688 APE11-dist-in 8.4688 APE10-dist-in 5.5301 APE9-dist-in 3.7526 None None None XRAY 2.04 0.202 0.226 A 294.0 273.0 0 26 26 0 [[38, 290]] 1.0 4xh6 CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1

CAMK_PIM1 (Serine/threonine-protein kinase pim-1)

Total number of chains: 198
Active chains: 188
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 190 96.0% AF-P11309-K1A
DFGin ABAminus 5 2.5% 4RC2A
DFGin None 2 1.0% 4XH6A
DFGin BLBminus 1 0.5% 6KZIA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PIM1 PIM1_HUMAN 1YXTA P11309 33 306 313.0 ANP:322 ATPlike Active DFGin 6.0285 14.2451 BLAminus -131.81, 176.98 66.39, 83.69 -99.64, 19.64 287.53, 80.25 -65.72, -15.35 in-in in 8.3094 Saltbr-in 2.8936 HRD-naA -67.95, -50.18 66.45, 4.68 in-in-in SNCiii in-in ActLoopNT-in 2.8088 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.69, 12.99 APE9-dihe-na -80.03, -158.46 APE8-dihe-in -83.46, 121.7 APE8-rot-in 308.53 APE67-dihe-in -70.36, -3.81 -49.69, -52.76 APE12-dist-in 9.7291 APE11-dist-in 8.6653 APE10-dist-in 5.2788 APE9-dist-in 3.8051 None None None XRAY 2.0 0.183 0.216 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxt Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXUA P11309 33 305 313.0 AMP:550 ATPlike Active DFGin 6.0455 14.5804 BLAminus -128.48, 170.01 62.85, 77.77 -90.35, 20.24 287.6, 77.99 -74.7, 1.63 in-in in 8.5131 Saltbr-in 2.4861 HRD-naA -60.24, -50.74 67.33, 4.52 in-in-in SNCiii in-in ActLoopNT-in 2.8925 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.18, 25.46 APE9-dihe-na -90.91, -158.18 APE8-dihe-in -86.5, 120.86 APE8-rot-in 310.09 APE67-dihe-in -63.06, -9.2 -60.21, -45.83 APE12-dist-in 9.9588 APE11-dist-in 8.8348 APE10-dist-in 5.6887 APE9-dist-in 3.8693 None None None XRAY 2.24 0.231 0.276 A 293.0 273.0 0 26 26 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXUB P11309 33 305 313.0 AMP:650 ATPlike Active DFGin 6.1203 14.6734 BLAminus -120.37, 167.93 65.74, 85.44 -95.36, 14.03 285.37, 78.45 -64.71, -9.22 in-in in 8.6002 Saltbr-in 2.814 HRD-naA -59.51, -51.25 68.06, 6.92 in-in-in SNCiii in-in ActLoopNT-in 2.9988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.12, 36.18 APE9-dihe-na -84.74, -152.35 APE8-dihe-in -93.27, 122.65 APE8-rot-in 302.12 APE67-dihe-in -68.21, -7.03 -55.31, -45.11 APE12-dist-in 9.8003 APE11-dist-in 8.5338 APE10-dist-in 5.4571 APE9-dist-in 3.8415 None None None XRAY 2.24 0.231 0.276 B 293.0 273.0 0 26 26 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXUC P11309 34 305 313.0 AMP:750 ATPlike Active DFGin 6.1096 14.7409 BLAminus -134.94, 167.86 62.59, 83.1 -95.62, 21.45 280.06, 80.63 -81.83, 7.92 in-in in 8.7162 Saltbr-in 2.6122 HRD-naA -67.31, -48.53 67.93, 5.85 in-in-in SNCiii in-in ActLoopNT-in 2.8989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.01, 44.98 APE9-dihe-na -103.92, -155.25 APE8-dihe-in -86.11, 117.99 APE8-rot-in 310.09 APE67-dihe-in -68.22, -9.23 -52.45, -45.39 APE12-dist-in 9.6966 APE11-dist-in 8.6541 APE10-dist-in 5.6036 APE9-dist-in 3.8474 None None None XRAY 2.24 0.231 0.276 C 293.0 272.0 0 26 26 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXUD P11309 33 305 313.0 AMP:850 ATPlike Active DFGin 6.2355 14.5561 BLAminus -126.04, 169.08 67.7, 73.28 -88.52, 13.94 289.01, 78.99 -70.28, -2.85 in-in in 8.7886 Saltbr-in 2.4658 HRD-naA -64.06, -51.29 66.47, 10.4 in-in-in SNCiii in-in ActLoopNT-in 2.9168 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.8, 31.82 APE9-dihe-na -93.66, -159.09 APE8-dihe-in -85.99, 118.35 APE8-rot-in 303.12 APE67-dihe-in -71.66, -13.36 -52.91, -39.75 APE12-dist-in 9.8955 APE11-dist-in 8.6446 APE10-dist-in 5.4567 APE9-dist-in 3.827 None None None XRAY 2.24 0.231 0.276 D 293.0 273.0 0 26 26 0 [[38, 290]] 1.0 1yxu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1XR1A P11309 32 308 313.0 ANP:501 ATPlike Active DFGin 5.8877 14.2143 BLAminus -138.05, 176.98 59.78, 85.31 -96.55, 16.88 287.93, 82.19 -61.38, -7.19 in-in in 8.717 Saltbr-in 2.833 HRD-naA -59.95, -51.82 71.23, 5.72 in-in-in SNCiii in-in ActLoopNT-in 2.7525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.05, 45.66 APE9-dihe-na -114.17, -171.15 APE8-dihe-in -64.11, 112.97 APE8-rot-in 299.41 APE67-dihe-in -49.28, -12.21 -42.84, -67.53 APE12-dist-in 9.6083 APE11-dist-in 8.6947 APE10-dist-in 5.5225 APE9-dist-in 4.0703 None None None XRAY 2.1 0.267 0.301 A 300.0 277.0 0 26 26 0 [[38, 290]] 1.0 1xr1 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3A99A P11309 33 305 313.0 ANP:501 ATPlike Active DFGin 5.9337 14.254 BLAminus -128.38, 171.59 60.85, 87.29 -96.61, 22.08 288.57, 75.78 -65.84, -9.23 in-in in 8.7536 Saltbr-in 2.6044 HRD-naA -66.86, -47.45 66.12, 8.26 in-in-in SNCiii in-in ActLoopNT-in 2.8889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.19, 26.41 APE9-dihe-na -87.51, -159.07 APE8-dihe-in -85.64, 119.66 APE8-rot-in 305.41 APE67-dihe-in -70.7, -5.81 -56.65, -39.81 APE12-dist-in 9.6122 APE11-dist-in 8.4607 APE10-dist-in 5.2903 APE9-dist-in 3.7779 None None None XRAY 1.6 0.187 0.206 A 320.0 273.0 0 26 26 0 [[38, 290]] 1.0 3a99 Homo sapiens CAMK_PIM1_HUMAN CAMK 4.3e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2BZKB P11309 33 305 313.0 ANP:1306 ATPlike Active DFGin 6.1262 14.4434 BLAminus -123.86, 174.78 64.57, 79.13 -87.5, 17.23 286.98, 86.61 -67.5, -17.62 in-in in 8.7809 Saltbr-in 2.7266 HRD-naA -70.49, -48.81 68.36, 6.4 in-in-in SNCiii in-in ActLoopNT-in 2.8129 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.63, 10.91 APE9-dihe-na -77.79, -156.22 APE8-dihe-in -90.85, 124.06 APE8-rot-in 315.85 APE67-dihe-in -68.94, -10.63 -60.69, -42.64 APE12-dist-in 9.4641 APE11-dist-in 8.4783 APE10-dist-in 4.8507 APE9-dist-in 3.7821 R250G None None XRAY 2.45 0.191 0.225 B 313.0 268.0 5 26 26 0 [[38, 290]] 1.0 2bzk Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXSA P11309 33 306 313.0 No_ligand No_ligand Active DFGin 6.0435 14.6911 BLAminus -127.76, 171.69 59.08, 88.63 -95.69, 24.45 285.74, 79.92 -71.89, -12.05 in-in in 8.8359 Saltbr-in 2.5148 HRD-naA -69.25, -46.6 65.7, 9.18 in-in-in SNCiii in-in ActLoopNT-in 2.8874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.7, 28.09 APE9-dihe-na -94.38, -153.78 APE8-dihe-in -89.3, 121.74 APE8-rot-in 312.97 APE67-dihe-in -69.81, -9.24 -57.4, -43.57 APE12-dist-in 9.6115 APE11-dist-in 8.495 APE10-dist-in 5.3233 APE9-dist-in 3.8299 P123M None None XRAY 2.2 0.197 0.237 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxs Homo sapiens CAMK_PIM1_HUMAN CAMK 5.7e-66 228.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN AF-P11309-K1A P11309 30 298 313.0 No_ligand No_ligand Active DFGin 5.9244 14.426 BLAminus -123.59, 173.12 59.42, 75.84 -84.42, 19.94 286.93, 72.18 -59.74, -40.02 in-in in 8.502 Saltbr-in 2.6923 HRD-naA -69.93, -42.11 63.25, -11.96 in-in-in SNCiii in-in ActLoopNT-in 2.8371 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.01, 20.91 APE9-dihe-na -84.17, 176.91 APE8-dihe-in -67.72, 122.1 APE8-rot-in 305.72 APE67-dihe-in -69.25, -16.84 -56.89, -41.09 APE12-dist-in 9.5789 APE11-dist-in 8.723 APE10-dist-in 4.8295 APE9-dist-in 3.8227 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 26 26 0 [[38, 290]] 1.0 AF-P11309-K1 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.3e-65 226.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN AF-P11309-K3A P11309 30 298 313.0 No_ligand No_ligand Active DFGin 5.794 14.2839 BLAminus -126.38, 175.52 54.92, 81.68 -85.76, 15.39 286.52, 75.42 -58.44, -43.23 in-in in 8.4804 Saltbr-in 2.6753 HRD-naA -72.55, -35.61 62.65, -28.81 in-in-in SNCiii in-in ActLoopNT-in 2.818 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.76, 133.51 APE9-dihe-na 135.29, -179.73 APE8-dihe-in -78.77, 123.98 APE8-rot-in 299.06 APE67-dihe-in -67.9, -19.52 -59.41, -42.11 APE12-dist-in 10.2793 APE11-dist-in 9.2154 APE10-dist-in 4.16 APE9-dist-in 4.4335 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 26 26 0 [[38, 290]] 1.0 AF-P11309-K3 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.3e-65 226.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YWVA P11309 33 306 313.0 No_ligand No_ligand Active DFGin 6.1075 14.6848 BLAminus -128.69, 170.23 59.45, 82.37 -93.38, 16.91 284.75, 80.98 -65.5, -15.92 in-in in 8.8752 Saltbr-in 2.4035 HRD-naA -68.35, -45.31 66.91, 0.56 in-in-in SNCiii in-in ActLoopNT-in 2.9161 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.63, 18.4 APE9-dihe-na -83.53, -173.89 APE8-dihe-in -74.3, 128.16 APE8-rot-in 308.34 APE67-dihe-in -66.79, -7.76 -58.38, -49.12 APE12-dist-in 9.4097 APE11-dist-in 8.6884 APE10-dist-in 5.159 APE9-dist-in 3.9453 None None None XRAY 2.0 0.213 0.239 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1ywv Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1XQZA P11309 32 308 313.0 No_ligand No_ligand Active DFGin 6.113 14.3232 BLAminus -132.59, 173.59 55.58, 88.87 -95.24, 18.48 288.46, 74.92 -59.23, -7.62 in-in in 8.4544 Saltbr-in 2.8339 HRD-naA -64.93, -53.25 74.7, 0.79 in-in-in SNCiii in-in ActLoopNT-in 2.8964 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.51, 32.32 APE9-dihe-na -92.62, -159.59 APE8-dihe-in -84.16, 115.96 APE8-rot-in 305.78 APE67-dihe-in -51.85, -11.5 -41.07, -65.14 APE12-dist-in 9.6322 APE11-dist-in 8.7408 APE10-dist-in 5.5845 APE9-dist-in 3.8829 None None None XRAY 2.1 0.249 0.297 A 300.0 277.0 0 26 26 0 [[38, 290]] 1.0 1xqz Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7VSYA P11309 33 305 313.0 No_ligand No_ligand Active DFGin 6.1466 14.8353 BLAminus -134.49, 172.31 56.25, 85.19 -90.8, 13.5 283.59, 75.74 -71.18, -5.96 in-in in 8.9886 Saltbr-in 2.572 HRD-naA -72.16, -48.61 72.01, 2.74 in-in-in SNCiii in-in ActLoopNT-in 2.8186 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.2, 35.54 APE9-dihe-na -94.69, -147.72 APE8-dihe-in -96.93, 120.22 APE8-rot-in 307.41 APE67-dihe-in -68.94, -11.56 -54.86, -45.03 APE12-dist-in 10.1896 APE11-dist-in 8.7411 APE10-dist-in 5.5966 APE9-dist-in 3.8972 N82K None None XRAY 2.141 0.198 0.22 A 326.0 273.0 0 26 26 0 [[38, 290]] 1.0 7vsy Homo sapiens CAMK_PIM1_HUMAN CAMK 4.5e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4JX3A P11309 33 306 313.0 No_ligand No_ligand Active DFGin 6.2546 14.8623 BLAminus -127.82, 159.43 82.11, 81.67 -96.33, 22.05 278.91, 78.81 -66.22, -18.54 in-in in 9.0351 Saltbr-in 2.8635 HRD-naA -65.27, -47.76 69.76, -1.05 in-in-in SNCiii in-in ActLoopNT-in 2.647 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.67, 50.36 APE9-dihe-na -106.43, -151.13 APE8-dihe-in -91.89, 110.71 APE8-rot-in 312.27 APE67-dihe-in -55.41, -25.98 -43.33, -53.94 APE12-dist-in 9.6927 APE11-dist-in 8.5235 APE10-dist-in 5.6535 APE9-dist-in 4.0695 None None None XRAY 2.5 0.222 0.249 A 326.0 274.0 0 26 26 0 [[38, 290]] 1.0 4jx3 Homo sapiens CAMK_PIM1_HUMAN CAMK 4.6e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7OOVA P11309 33 305 313.0 No_ligand No_ligand Active DFGin 6.203 14.5695 BLAminus -122.84, 171.74 65.68, 80.45 -90.31, 16.43 288.09, 76.06 -72.31, -11.34 in-in in 8.7995 Saltbr-in 2.608 HRD-naA -67.33, -47.42 68.65, 9.26 in-in-in SNCiii in-in ActLoopNT-in 2.8419 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.94, 17.29 APE9-dihe-na -81.04, -164.98 APE8-dihe-in -82.61, 126.44 APE8-rot-in 309.83 APE67-dihe-in -78.03, -5.17 -57.01, -47.48 APE12-dist-in 9.5122 APE11-dist-in 8.789 APE10-dist-in 5.4863 APE9-dist-in 3.8884 None None None XRAY 1.96 0.163 0.195 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 7oov Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7OOWA P11309 33 305 313.0 No_ligand No_ligand Active DFGin 6.3063 14.7477 BLAminus -122.68, 175.54 62.53, 73.89 -87.93, 12.78 283.68, 73.03 -76.55, -12.97 in-in in 8.7425 Saltbr-in 2.6023 HRD-naA -68.81, -49.98 73.35, 5.62 in-in-in SNCiii in-in ActLoopNT-in 2.9105 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.14, 32.43 APE9-dihe-na -87.5, -147.91 APE8-dihe-in -98.97, 121.57 APE8-rot-in 305.26 APE67-dihe-in -77.55, -5.21 -53.13, -44.92 APE12-dist-in 9.5933 APE11-dist-in 8.9762 APE10-dist-in 5.5753 APE9-dist-in 3.7722 None None None XRAY 1.95 0.161 0.184 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 7oow Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5TOEA P11309 34 306 313.0 7GK:401 Type1 Active DFGin 6.0724 14.6604 BLAminus -139.61, 170.18 66.65, 79.11 -92.13, 15.86 288.09, 73.32 -71.9, -3.59 in-in in 8.9752 Saltbr-in 2.649 HRD-naA -71.41, -51.31 74.77, 4.24 in-in-in SNCiii in-in ActLoopNT-in 2.7859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.61, 20.8 APE9-dihe-na -92.31, -158.45 APE8-dihe-in -81.21, 122.35 APE8-rot-in 309.79 APE67-dihe-in -65.59, -11.22 -66.85, -44.0 APE12-dist-in 9.6842 APE11-dist-in 8.6635 APE10-dist-in 5.3884 APE9-dist-in 3.9063 None None None XRAY 2.301 0.194 0.233 A 273.0 272.0 1 26 26 0 [[38, 290]] 1.0 5toe Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YHSA P11309 33 305 313.0 STU:306 Type1 Active DFGin 6.3607 14.5116 BLAminus -129.35, 165.16 65.09, 87.92 -99.2, 21.71 283.47, 69.45 -67.38, -11.76 in-in in 8.5242 Saltbr-in 2.8992 HRD-naA -65.05, -49.56 68.79, 3.6 in-in-in SNCiii in-in ActLoopNT-in 2.9031 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.4, 26.1 APE9-dihe-na -84.03, -156.82 APE8-dihe-in -85.78, 122.63 APE8-rot-in 304.34 APE67-dihe-in -62.69, -6.01 -56.85, -49.38 APE12-dist-in 9.327 APE11-dist-in 8.5203 APE10-dist-in 5.5084 APE9-dist-in 3.8321 None SEP261 CME161,SEP261 XRAY 2.15 0.233 0.233 A 273.0 269.0 4 26 26 0 [[38, 290]] 1.0 1yhs Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YI3A P11309 33 305 313.0 LY2:306 Type1 Active DFGin 6.2916 14.7641 BLAminus -128.81, 164.98 60.01, 85.31 -95.12, 30.71 287.86, 62.33 -66.19, -20.32 in-in in 7.7949 Saltbr-in 2.7333 HRD-naA -63.25, -48.22 66.78, 7.96 in-in-in SNCiii in-in ActLoopNT-in 2.8372 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.69, 36.2 APE9-dihe-na -99.79, -161.83 APE8-dihe-in -81.08, 117.39 APE8-rot-in 309.96 APE67-dihe-in -55.73, -11.01 -50.65, -56.8 APE12-dist-in 9.4522 APE11-dist-in 8.685 APE10-dist-in 5.2315 APE9-dist-in 4.0187 None SEP261 CME161,SEP261 XRAY 2.5 0.208 0.259 A 273.0 269.0 4 26 26 0 [[38, 290]] 1.0 1yi3 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YI4A P11309 33 305 313.0 ADN:306 Type1 Active DFGin 6.0722 14.6981 BLAminus -134.71, 164.97 59.13, 80.78 -89.82, 21.93 287.09, 72.06 -64.68, -12.33 in-in in 8.788 Saltbr-in 2.7168 HRD-naA -68.53, -44.87 69.57, -1.62 in-in-in SNCiii in-in ActLoopNT-in 2.9339 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.9, 36.65 APE9-dihe-na -82.94, -132.28 APE8-dihe-in -114.84, 117.13 APE8-rot-in 309.09 APE67-dihe-in -54.56, -19.23 -51.71, -52.26 APE12-dist-in 9.605 APE11-dist-in 8.6743 APE10-dist-in 5.878 APE9-dist-in 4.1822 None SEP261 CME161,SEP261 XRAY 2.4 0.21 0.246 A 273.0 269.0 4 26 26 0 [[38, 290]] 1.0 1yi4 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3C4EA P11309 33 305 313.0 C4E:306 Type1 Active DFGin 6.0215 14.7761 BLAminus -128.35, 166.0 69.48, 82.58 -93.7, 21.6 286.61, 78.83 -72.51, -9.22 in-in in 8.8865 Saltbr-in 2.7325 HRD-naA -67.91, -51.23 70.69, 5.52 in-in-in SNCiii in-in ActLoopNT-in 2.8123 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.94, 10.44 APE9-dihe-na -76.24, -163.31 APE8-dihe-in -81.86, 120.75 APE8-rot-in 311.66 APE67-dihe-in -66.61, -7.38 -59.14, -42.78 APE12-dist-in 9.659 APE11-dist-in 8.5496 APE10-dist-in 5.1757 APE9-dist-in 3.7908 None None None XRAY 1.98 0.216 0.245 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3c4e Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3C4EB P11309 33 305 313.0 C4E:306 Type1 Active DFGin 6.0749 14.7907 BLAminus -125.63, 166.99 68.65, 82.63 -92.11, 15.76 285.08, 79.16 -64.7, -9.12 in-in in 8.8733 Saltbr-in 2.9369 HRD-naA -73.69, -46.03 62.22, 13.94 in-in-in SNCiii in-in ActLoopNT-in 2.8715 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.74, 17.74 APE9-dihe-na -78.68, -151.78 APE8-dihe-in -92.25, 117.75 APE8-rot-in 301.9 APE67-dihe-in -69.85, -9.71 -53.08, -43.68 APE12-dist-in 9.7383 APE11-dist-in 8.5606 APE10-dist-in 5.43 APE9-dist-in 3.6989 None None None XRAY 1.98 0.216 0.245 B 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3c4e Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3C4EC P11309 34 305 313.0 C4E:306 Type1 Active DFGin 6.0604 14.7651 BLAminus -128.73, 171.78 61.45, 83.06 -93.51, 22.09 285.2, 77.36 -74.45, -9.29 in-in in 9.0241 Saltbr-in 2.46 HRD-naA -74.89, -48.06 74.46, 0.4 in-in-in SNCiii in-in ActLoopNT-in 2.9066 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.43, 22.53 APE9-dihe-na -88.97, -156.05 APE8-dihe-in -88.82, 119.66 APE8-rot-in 306.87 APE67-dihe-in -73.65, -3.54 -57.42, -41.13 APE12-dist-in 9.7009 APE11-dist-in 8.436 APE10-dist-in 5.1657 APE9-dist-in 3.9214 None None None XRAY 1.98 0.216 0.245 C 273.0 272.0 0 26 26 0 [[38, 290]] 1.0 3c4e Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3C4ED P11309 33 305 313.0 C4E:306 Type1 Active DFGin 6.3092 14.7094 BLAminus -130.13, 172.88 59.98, 79.45 -88.47, 15.36 281.95, 81.3 -75.02, -5.99 in-in in 8.7901 Saltbr-in 2.4435 HRD-naA -70.24, -47.69 69.35, 4.35 in-in-in SNCiii in-in ActLoopNT-in 2.8326 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.82, 22.76 APE9-dihe-na -80.15, -163.14 APE8-dihe-in -81.97, 115.05 APE8-rot-in 309.18 APE67-dihe-in -70.46, -13.8 -51.69, -41.7 APE12-dist-in 9.7262 APE11-dist-in 8.5833 APE10-dist-in 5.5064 APE9-dist-in 3.7583 None None None XRAY 1.98 0.216 0.245 D 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3c4e Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4K1BA P11309 33 305 313.0 1OC:402 Type1 Active DFGin 6.0427 14.6126 BLAminus -132.6, 164.86 70.11, 79.62 -92.82, 21.53 288.39, 81.35 -65.25, -17.96 in-in in 8.8563 Saltbr-in 2.6319 HRD-naA -70.69, -51.38 75.39, 5.68 in-in-in SNCiii in-in ActLoopNT-in 2.8194 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.17, 19.78 APE9-dihe-na -83.3, -161.37 APE8-dihe-in -81.98, 126.09 APE8-rot-in 308.93 APE67-dihe-in -65.14, -9.59 -61.45, -45.63 APE12-dist-in 9.5986 APE11-dist-in 8.6775 APE10-dist-in 5.2847 APE9-dist-in 3.8229 None None None XRAY 2.082 0.172 0.199 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 4k1b Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6NO8A P11309 33 305 313.0 KUY:401 Type1 Active DFGin 6.245 14.4648 BLAminus -136.93, 161.07 71.64, 80.45 -96.46, 11.0 281.89, 88.38 -60.27, -17.64 in-in in 8.6572 Saltbr-in 2.6047 HRD-naA -78.06, -49.34 70.05, 6.39 in-in-in SNCiii in-in ActLoopNT-in 2.8128 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.3, 11.35 APE9-dihe-na -78.95, -162.34 APE8-dihe-in -79.37, 127.44 APE8-rot-in 316.96 APE67-dihe-in -61.79, -7.22 -64.64, -48.15 APE12-dist-in 9.6679 APE11-dist-in 8.7765 APE10-dist-in 5.2156 APE9-dist-in 3.7941 None None None XRAY 2.377 0.187 0.232 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 6no8 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6NO9A P11309 33 305 313.0 KUV:504 Type1 Active DFGin 6.1556 14.4327 BLAminus -126.34, 166.87 60.03, 83.92 -89.43, 21.76 289.02, 78.21 -70.19, -16.22 in-in in 8.6109 Saltbr-in 2.4384 HRD-naA -72.3, -46.64 69.8, 3.74 in-in-in SNCiii in-in ActLoopNT-in 2.8144 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.26, 10.84 APE9-dihe-na -76.6, -153.49 APE8-dihe-in -92.15, 125.02 APE8-rot-in 306.25 APE67-dihe-in -69.76, -6.68 -64.44, -39.96 APE12-dist-in 9.6794 APE11-dist-in 8.7289 APE10-dist-in 5.0813 APE9-dist-in 3.6717 None None None XRAY 1.712 0.17 0.205 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 6no9 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.4e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4K0YA P11309 33 306 313.0 1OA:401 Type1 Active DFGin 6.292 14.3895 BLAminus -121.94, 171.4 62.4, 86.58 -95.92, 17.62 287.73, 79.01 -70.57, -9.06 in-in in 8.9044 Saltbr-in 2.5085 HRD-naA -73.78, -47.42 68.19, 7.19 in-in-in SNCiii in-in ActLoopNT-in 2.7966 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.37, 25.39 APE9-dihe-na -84.39, -155.13 APE8-dihe-in -90.58, 120.54 APE8-rot-in 303.27 APE67-dihe-in -71.06, -6.6 -61.16, -38.44 APE12-dist-in 9.6715 APE11-dist-in 8.6212 APE10-dist-in 5.5489 APE9-dist-in 3.6456 None None None XRAY 1.954 0.177 0.214 A 274.0 274.0 0 26 26 0 [[38, 290]] 1.0 4k0y Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5TELA P11309 33 306 313.0 7AJ:402 Type1 Active DFGin 6.1394 14.6282 BLAminus -138.92, 170.35 61.02, 78.29 -89.18, 17.43 286.77, 73.8 -69.83, -8.87 in-in in 8.9252 Saltbr-in 2.5481 HRD-naA -74.49, -48.42 69.85, 6.32 in-in-in SNCiii in-in ActLoopNT-in 2.8228 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.37, 35.58 APE9-dihe-na -94.48, -159.56 APE8-dihe-in -83.62, 124.38 APE8-rot-in 309.44 APE67-dihe-in -63.92, -12.31 -66.13, -42.06 APE12-dist-in 9.6957 APE11-dist-in 8.6914 APE10-dist-in 5.4702 APE9-dist-in 3.9726 None None None XRAY 2.214 0.182 0.207 A 274.0 273.0 1 26 26 0 [[38, 290]] 1.0 5tel Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5TEXA P11309 33 306 313.0 7AU:402 Type1 Active DFGin 6.0104 14.8294 BLAminus -138.39, 174.01 63.47, 82.62 -93.78, 16.92 290.32, 76.89 -70.47, -10.69 in-in in 9.269 Saltbr-in 2.8453 HRD-naA -75.68, -50.36 69.23, 7.58 in-in-in SNCiii in-in ActLoopNT-in 2.8374 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.29, 24.17 APE9-dihe-na -86.25, -152.07 APE8-dihe-in -90.77, 121.09 APE8-rot-in 307.82 APE67-dihe-in -67.29, -11.31 -64.01, -39.58 APE12-dist-in 9.6917 APE11-dist-in 8.5519 APE10-dist-in 5.4035 APE9-dist-in 3.8882 None None None XRAY 2.149 0.184 0.217 A 274.0 274.0 0 26 26 0 [[38, 290]] 1.0 5tex Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6VRUA P11309 34 306 313.0 ROY:402 Type1 Active DFGin 6.2493 14.7341 BLAminus -126.97, 167.03 70.01, 79.24 -93.65, 20.02 287.24, 69.33 -68.9, -13.34 in-in in 8.636 Saltbr-in 2.498 HRD-naA -74.69, -47.82 68.45, 8.0 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.88, 21.88 APE9-dihe-na -81.69, -157.22 APE8-dihe-in -91.46, 126.79 APE8-rot-in 307.71 APE67-dihe-in -66.96, -7.81 -67.63, -41.62 APE12-dist-in 9.5785 APE11-dist-in 8.5741 APE10-dist-in 5.2117 APE9-dist-in 3.7056 None None None XRAY 2.07 0.179 0.202 A 274.0 273.0 0 26 26 0 [[38, 290]] 1.0 6vru Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6VRVA P11309 35 305 313.0 WFY:401 Type1 Active DFGin 6.31 14.7748 BLAminus -128.18, 168.1 70.4, 82.6 -93.17, 16.82 287.59, 75.85 -67.39, -13.62 in-in in 8.7763 Saltbr-in 2.5274 HRD-naA -73.57, -42.57 66.05, 10.02 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.71, 32.21 APE9-dihe-na -87.53, -152.73 APE8-dihe-in -95.97, 120.66 APE8-rot-in 293.39 APE67-dihe-in -72.79, -2.49 -61.51, -35.74 APE12-dist-in 9.5715 APE11-dist-in 8.5796 APE10-dist-in 5.6753 APE9-dist-in 3.7577 None None None XRAY 1.74 0.173 0.197 A 274.0 271.0 0 26 26 0 [[38, 290]] 1.0 6vrv Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.3 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4DTKA P11309 33 305 313.0 7LI:408 Type1 Active DFGin 6.1421 14.6613 BLAminus -128.39, 173.69 63.23, 87.87 -95.85, 17.29 285.67, 80.15 -64.1, -18.22 in-in in 8.8606 Saltbr-in 2.5881 HRD-naA -66.25, -50.01 70.2, 5.45 in-in-in SNCiii in-in ActLoopNT-in 2.8698 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.52, 26.77 APE9-dihe-na -86.23, -154.0 APE8-dihe-in -89.22, 120.59 APE8-rot-in 306.1 APE67-dihe-in -65.85, -11.4 -53.32, -45.84 APE12-dist-in 9.7014 APE11-dist-in 8.5854 APE10-dist-in 5.4744 APE9-dist-in 3.6925 None None None XRAY 1.86 0.166 0.182 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 4dtk Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KGDA P11309 33 305 313.0 6SL:420 Type1 Active DFGin 6.1941 14.5978 BLAminus -129.0, 173.16 59.49, 81.21 -91.39, 15.51 283.61, 78.67 -67.75, -14.27 in-in in 8.8183 Saltbr-in 2.7249 HRD-naA -68.62, -47.74 69.23, 3.07 in-in-in SNCiii in-in ActLoopNT-in 2.8548 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.77, 31.72 APE9-dihe-na -89.5, -153.75 APE8-dihe-in -91.96, 121.37 APE8-rot-in 309.6 APE67-dihe-in -67.17, -11.15 -55.07, -44.24 APE12-dist-in 9.602 APE11-dist-in 8.6734 APE10-dist-in 5.6063 APE9-dist-in 3.7255 None None None XRAY 1.98 0.163 0.184 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgd Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KGEA P11309 33 305 313.0 6SN:416 Type1 Active DFGin 6.1855 14.6068 BLAminus -127.16, 171.98 58.94, 83.36 -93.06, 16.77 283.0, 80.17 -66.19, -15.51 in-in in 8.8007 Saltbr-in 2.6657 HRD-naA -68.2, -48.81 68.27, 3.74 in-in-in SNCiii in-in ActLoopNT-in 2.8389 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.87, 31.34 APE9-dihe-na -88.89, -156.61 APE8-dihe-in -88.29, 120.88 APE8-rot-in 311.55 APE67-dihe-in -66.51, -12.56 -54.59, -43.9 APE12-dist-in 9.6589 APE11-dist-in 8.6942 APE10-dist-in 5.6243 APE9-dist-in 3.7446 None None None XRAY 2.23 0.196 0.208 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kge Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KGGA P11309 33 305 313.0 6SO:423 Type1 Active DFGin 6.0952 14.601 BLAminus -129.17, 178.0 55.81, 74.89 -86.97, 13.61 281.87, 79.94 -67.04, -14.98 in-in in 8.9363 Saltbr-in 2.6656 HRD-naA -69.61, -46.82 68.9, 2.47 in-in-in SNCiii in-in ActLoopNT-in 2.883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.69, 27.94 APE9-dihe-na -86.85, -153.1 APE8-dihe-in -91.39, 121.35 APE8-rot-in 307.73 APE67-dihe-in -68.33, -11.23 -55.33, -42.82 APE12-dist-in 9.8085 APE11-dist-in 8.7335 APE10-dist-in 5.6043 APE9-dist-in 3.6841 None None None XRAY 1.95 0.159 0.17 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgg Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KGIA P11309 33 305 313.0 6SF:414 Type1 Active DFGin 6.1959 14.6781 BLAminus -128.85, 173.72 58.37, 80.83 -91.15, 15.65 283.15, 78.86 -67.29, -15.19 in-in in 8.8975 Saltbr-in 2.6991 HRD-naA -66.85, -48.52 69.49, 3.32 in-in-in SNCiii in-in ActLoopNT-in 2.8537 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.48, 30.3 APE9-dihe-na -88.67, -155.26 APE8-dihe-in -89.24, 121.14 APE8-rot-in 310.96 APE67-dihe-in -66.24, -12.88 -55.29, -44.34 APE12-dist-in 9.7233 APE11-dist-in 8.7346 APE10-dist-in 5.6424 APE9-dist-in 3.7397 None None None XRAY 2.13 0.173 0.186 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgi Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KGKA P11309 33 305 313.0 6SD:407 Type1 Active DFGin 6.3082 14.8602 BLAminus -128.4, 171.34 59.1, 83.1 -92.34, 16.26 283.46, 79.02 -66.84, -16.78 in-in in 8.9281 Saltbr-in 2.7226 HRD-naA -66.62, -48.72 69.73, 2.6 in-in-in SNCiii in-in ActLoopNT-in 2.8541 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.74, 32.55 APE9-dihe-na -90.23, -157.96 APE8-dihe-in -86.86, 120.62 APE8-rot-in 311.8 APE67-dihe-in -66.57, -13.56 -54.03, -44.15 APE12-dist-in 9.7032 APE11-dist-in 8.8498 APE10-dist-in 5.6821 APE9-dist-in 3.7634 None None None XRAY 2.66 0.188 0.206 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kgk Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6BSKA P11309 33 305 313.0 MVG:405 Type1 Active DFGin 6.1061 14.5261 BLAminus -127.81, 171.26 61.28, 88.13 -94.14, 14.55 285.4, 81.12 -65.15, -15.23 in-in in 8.7334 Saltbr-in 2.6534 HRD-naA -65.0, -51.26 70.65, 3.06 in-in-in SNCiii in-in ActLoopNT-in 2.8175 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.1, 36.25 APE9-dihe-na -95.43, -156.67 APE8-dihe-in -85.65, 120.06 APE8-rot-in 311.62 APE67-dihe-in -68.39, -14.22 -55.35, -43.45 APE12-dist-in 9.8022 APE11-dist-in 8.5486 APE10-dist-in 5.6356 APE9-dist-in 3.7924 None None None XRAY 2.573 0.171 0.196 A 276.0 273.0 0 26 26 0 [[38, 290]] 1.0 6bsk Homo sapiens CAMK_PIM1_HUMAN CAMK 2.5e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4K18A P11309 32 308 313.0 1OB:402 Type1 Active DFGin 6.0917 14.4411 BLAminus -127.16, 170.25 67.68, 77.49 -90.65, 24.19 290.3, 84.83 -68.81, -16.15 in-in in 8.7657 Saltbr-in 2.6128 HRD-naA -73.4, -51.44 75.59, 3.74 in-in-in SNCiii in-in ActLoopNT-in 2.8538 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.67, 18.39 APE9-dihe-na -83.8, -157.76 APE8-dihe-in -87.59, 123.77 APE8-rot-in 308.05 APE67-dihe-in -70.86, -5.11 -63.89, -39.96 APE12-dist-in 9.7914 APE11-dist-in 8.8029 APE10-dist-in 5.401 APE9-dist-in 3.9252 None None None XRAY 2.051 0.186 0.22 A 277.0 277.0 0 26 26 0 [[38, 290]] 1.0 4k18 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.6e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5IISA P11309 32 305 313.0 6CB:402 Type1 Active DFGin 6.3878 14.7567 BLAminus -128.84, 173.3 61.28, 84.09 -98.54, 16.15 284.91, 73.79 -69.44, -13.21 in-in in 8.2803 Saltbr-in 2.7008 HRD-naA -69.32, -50.23 68.69, 7.8 in-in-in SNCiii in-in ActLoopNT-in 2.9101 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.03, 27.99 APE9-dihe-na -88.44, -153.73 APE8-dihe-in -93.14, 121.31 APE8-rot-in 307.37 APE67-dihe-in -67.36, -12.92 -53.81, -44.97 APE12-dist-in 9.4712 APE11-dist-in 8.5316 APE10-dist-in 5.2689 APE9-dist-in 3.6397 None SEP261 SEP261 XRAY 2.1 0.172 0.193 A 277.0 274.0 0 26 26 0 [[38, 290]] 1.0 5iis Homo sapiens CAMK_PIM1_HUMAN CAMK 2.6e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4TY1A P11309 33 305 313.0 38W:401 Type1 Active DFGin 6.387 14.5113 BLAminus -133.05, 165.34 66.19, 78.61 -90.98, 18.04 289.04, 69.92 -66.35, -17.07 in-in in 8.0757 Saltbr-in 2.8545 HRD-naA -75.5, -52.3 76.47, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.8796 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.39, -3.83 APE9-dihe-na -80.99, -152.88 APE8-dihe-in -92.77, 125.02 APE8-rot-in 308.7 APE67-dihe-in -59.27, -21.7 -50.58, -57.32 APE12-dist-in 9.5504 APE11-dist-in 8.7416 APE10-dist-in 4.3675 APE9-dist-in 3.6288 None None None XRAY 2.7 0.183 0.237 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4ty1 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4WRSA P11309 33 305 313.0 3U1:403 Type1 Active DFGin 6.1624 14.6882 BLAminus -131.19, 168.19 62.17, 84.39 -94.94, 19.3 284.32, 75.21 -73.2, -12.05 in-in in 8.9033 Saltbr-in 2.6155 HRD-naA -70.39, -48.07 69.42, 8.56 in-in-in SNCiii in-in ActLoopNT-in 2.9235 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.6, 16.03 APE9-dihe-na -86.28, -152.26 APE8-dihe-in -92.85, 128.8 APE8-rot-in 308.26 APE67-dihe-in -65.67, -10.81 -62.91, -47.38 APE12-dist-in 9.4769 APE11-dist-in 8.6179 APE10-dist-in 4.9364 APE9-dist-in 3.7627 None None None XRAY 2.2 0.18 0.208 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4wrs Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4WSYA P11309 33 305 313.0 3U5:401 Type1 Active DFGin 6.1044 14.6207 BLAminus -127.31, -178.18 57.57, 65.12 -84.25, 18.54 286.02, 73.35 -69.75, -14.58 in-in in 8.9086 Saltbr-in 2.7849 HRD-naA -70.92, -47.77 70.77, 0.48 in-in-in SNCiii in-in ActLoopNT-in 2.9139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.56, 17.45 APE9-dihe-na -80.04, -158.16 APE8-dihe-in -87.23, 129.67 APE8-rot-in 306.6 APE67-dihe-in -63.98, -11.76 -66.05, -47.25 APE12-dist-in 9.5 APE11-dist-in 8.5775 APE10-dist-in 5.3469 APE9-dist-in 3.7953 None None None XRAY 2.3 0.184 0.224 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4wsy Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4WT6A P11309 33 305 313.0 3U6:401 Type1 Active DFGin 6.2247 14.7413 BLAminus -129.31, 179.15 54.14, 72.7 -88.4, 20.56 284.51, 71.19 -73.36, -15.22 in-in in 8.4691 Saltbr-in 2.6562 HRD-naA -72.36, -44.25 65.88, 2.27 in-in-in SNCiii in-in ActLoopNT-in 2.9723 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.26, 22.96 APE9-dihe-na -91.6, -154.03 APE8-dihe-in -92.19, 127.1 APE8-rot-in 312.31 APE67-dihe-in -65.83, -13.24 -60.93, -48.29 APE12-dist-in 9.496 APE11-dist-in 8.6131 APE10-dist-in 5.0588 APE9-dist-in 3.9979 None None None XRAY 2.3 0.178 0.211 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4wt6 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5EOLA P11309 33 305 313.0 5QO:401 Type1 Active DFGin 6.2561 14.6307 BLAminus -125.24, 171.83 59.51, 79.96 -92.44, 22.49 285.02, 73.25 -70.93, -14.06 in-in in 8.7627 Saltbr-in 2.5732 HRD-naA -73.1, -47.95 68.92, 3.14 in-in-in SNCiii in-in ActLoopNT-in 2.8417 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.99, 8.97 APE9-dihe-na -79.78, -148.56 APE8-dihe-in -97.04, 122.04 APE8-rot-in 309.05 APE67-dihe-in -66.69, -11.1 -58.67, -42.55 APE12-dist-in 9.5827 APE11-dist-in 8.513 APE10-dist-in 4.9128 APE9-dist-in 3.6325 None None None XRAY 2.2 0.196 0.223 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 5eol Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5IPJA P11309 33 305 313.0 6CD:401 Type1 Active DFGin 6.1587 14.6449 BLAminus -129.06, 166.2 63.4, 89.79 -98.28, 24.16 286.53, 74.98 -69.52, -15.68 in-in in 8.8615 Saltbr-in 2.6437 HRD-naA -72.25, -47.9 67.86, 13.58 in-in-in SNCiii in-in ActLoopNT-in 2.8528 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.03, 18.83 APE9-dihe-na -86.4, -154.92 APE8-dihe-in -92.64, 123.62 APE8-rot-in 306.86 APE67-dihe-in -66.21, -11.28 -62.03, -43.15 APE12-dist-in 9.5154 APE11-dist-in 8.5252 APE10-dist-in 4.9669 APE9-dist-in 3.5939 None None None XRAY 2.1 0.181 0.221 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 5ipj Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KZIA P11309 33 305 313.0 6YN:401 Type1 Active DFGin 6.2318 14.4593 BLAminus -125.28, 171.61 59.7, 76.37 -89.66, 23.41 287.5, 74.51 -76.32, -14.48 in-in in 8.5633 Saltbr-in 2.6219 HRD-naA -74.51, -47.69 70.34, 4.33 in-in-in SNCiii in-in ActLoopNT-in 2.7817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.16, 14.87 APE9-dihe-na -85.38, -150.81 APE8-dihe-in -98.45, 122.78 APE8-rot-in 307.97 APE67-dihe-in -69.43, -12.03 -61.1, -42.73 APE12-dist-in 9.6227 APE11-dist-in 8.7118 APE10-dist-in 4.9438 APE9-dist-in 3.8102 None None None XRAY 2.1 0.179 0.205 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 5kzi Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6MT0A P11309 33 305 313.0 JYG:401 Type1 Active DFGin 6.1797 14.6437 BLAminus -129.1, 162.88 69.48, 92.17 -101.8, 22.17 287.32, 75.1 -69.24, -17.14 in-in in 8.6669 Saltbr-in 2.7291 HRD-naA -70.67, -47.42 66.78, 12.82 in-in-in SNCiii in-in ActLoopNT-in 2.8517 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -118.16, 8.39 APE9-dihe-na -79.87, -163.75 APE8-dihe-in -86.85, 127.4 APE8-rot-in 308.59 APE67-dihe-in -66.88, -11.27 -60.5, -47.04 APE12-dist-in 9.3772 APE11-dist-in 8.5534 APE10-dist-in 4.6116 APE9-dist-in 3.5443 None None None XRAY 2.2 0.18 0.208 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 6mt0 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4MTAA P11309 33 305 313.0 2D2:401 Type1 Active DFGin 6.2759 14.3366 BLAminus -121.41, 177.86 55.53, 82.62 -93.46, 16.76 281.52, 74.78 -72.09, -10.86 in-in in 8.719 Saltbr-in 2.6113 HRD-naA -62.2, -48.48 67.49, 3.7 in-in-in SNCiii in-in ActLoopNT-in 2.7947 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.11, 24.3 APE9-dihe-na -85.34, -152.54 APE8-dihe-in -92.96, 123.11 APE8-rot-in 306.26 APE67-dihe-in -67.9, -13.27 -54.99, -44.77 APE12-dist-in 9.5277 APE11-dist-in 8.5158 APE10-dist-in 5.416 APE9-dist-in 3.5754 None None None XRAY 2.2 0.16 0.192 A 286.0 273.0 0 26 26 0 [[38, 290]] 1.0 4mta Homo sapiens CAMK_PIM1_HUMAN CAMK 2.9e-65 226.1 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5C1QB P11309 33 305 313.0 4YK:401 Type1 Active DFGin 5.891 13.333 BLAminus -134.33, 156.38 72.1, 106.74 -112.64, 17.25 301.94, 90.76 -59.71, -41.8 in-in in 8.6215 Saltbr-in 2.5933 HRD-naA -64.46, -50.63 69.52, -24.55 in-in-in SNCiii in-in ActLoopNT-in 2.8007 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.39, 56.57 APE9-dihe-na -121.47, -173.24 APE8-dihe-in -77.48, 148.97 APE8-rot-in 348.38 APE67-dihe-in -42.36, -34.75 -61.79, -66.84 APE12-dist-in 9.4062 APE11-dist-in 8.2515 APE10-dist-in 5.3773 APE9-dist-in 4.9262 None None None XRAY 3.0 0.178 0.246 B 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 5c1q Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L11A P11309 33 305 313.0 E2C:401 Type1 Active DFGin 6.1626 14.9671 BLAminus -125.67, 168.03 67.88, 78.16 -84.6, 16.39 285.76, 87.64 -71.05, -19.61 in-in in 8.9964 Saltbr-in 2.7022 HRD-naA -66.89, -52.69 70.36, 8.44 in-in-in SNCiii in-in ActLoopNT-in 2.767 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.89, 29.6 APE9-dihe-na -84.12, -156.34 APE8-dihe-in -92.4, 128.66 APE8-rot-in 306.74 APE67-dihe-in -67.11, -6.47 -60.7, -48.56 APE12-dist-in 9.3558 APE11-dist-in 8.3863 APE10-dist-in 5.4313 APE9-dist-in 3.7089 None SEP261 SEP261 XRAY 2.05 0.214 0.24 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l11 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L12A P11309 33 305 313.0 E2R:401 Type1 Active DFGin 6.2158 14.7026 BLAminus -127.05, 170.42 68.23, 81.09 -92.51, 16.44 287.76, 81.55 -64.97, -20.04 in-in in 8.983 Saltbr-in 2.7221 HRD-naA -72.18, -48.09 70.82, 3.37 in-in-in SNCiii in-in ActLoopNT-in 2.8382 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.36, 18.6 APE9-dihe-na -85.64, -160.05 APE8-dihe-in -87.61, 125.01 APE8-rot-in 307.11 APE67-dihe-in -68.37, -12.11 -58.28, -46.28 APE12-dist-in 9.3781 APE11-dist-in 8.5814 APE10-dist-in 5.0596 APE9-dist-in 3.8326 None SEP261 SEP261 XRAY 1.87 0.197 0.21 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l12 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L13A P11309 33 305 313.0 E2F:401 Type1 Active DFGin 6.1902 14.7858 BLAminus -130.24, 168.2 68.46, 80.68 -89.17, 16.05 288.1, 80.31 -69.01, -19.61 in-in in 9.1055 Saltbr-in 2.9362 HRD-naA -68.46, -51.8 71.9, 8.52 in-in-in SNCiii in-in ActLoopNT-in 2.7778 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.76, 29.56 APE9-dihe-na -92.34, -153.25 APE8-dihe-in -98.43, 124.2 APE8-rot-in 303.55 APE67-dihe-in -68.48, -12.49 -58.68, -45.06 APE12-dist-in 9.5 APE11-dist-in 8.5109 APE10-dist-in 5.0987 APE9-dist-in 3.6586 None SEP261 SEP261 XRAY 2.24 0.18 0.214 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l13 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L14A P11309 33 305 313.0 E2L:401 Type1 Active DFGin 6.2009 14.8938 BLAminus -126.69, 169.11 67.27, 79.53 -86.62, 19.33 288.75, 82.28 -66.99, -22.84 in-in in 9.0448 Saltbr-in 2.8364 HRD-naA -67.72, -50.1 68.21, 9.79 in-in-in SNCiii in-in ActLoopNT-in 2.8055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.83, 24.46 APE9-dihe-na -89.25, -158.62 APE8-dihe-in -92.28, 125.41 APE8-rot-in 306.06 APE67-dihe-in -68.05, -12.07 -60.25, -45.14 APE12-dist-in 9.5091 APE11-dist-in 8.5175 APE10-dist-in 5.0735 APE9-dist-in 3.7712 None SEP261 SEP261 XRAY 1.95 0.193 0.209 A 289.0 271.0 2 26 26 0 [[38, 290]] 1.0 6l14 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L15A P11309 33 305 313.0 E2O:401 Type1 Active DFGin 6.3499 14.598 BLAminus -131.83, 163.47 71.59, 79.35 -89.78, 14.2 284.41, 77.37 -65.48, -21.82 in-in in 8.235 Saltbr-in 2.5656 HRD-naA -64.16, -54.27 75.51, 4.04 in-in-in SNCiii in-in ActLoopNT-in 2.7413 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.69, 27.17 APE9-dihe-na -98.51, -154.05 APE8-dihe-in -93.58, 128.93 APE8-rot-in 316.57 APE67-dihe-in -60.96, -21.44 -58.79, -53.8 APE12-dist-in 9.4071 APE11-dist-in 8.6356 APE10-dist-in 4.9291 APE9-dist-in 3.916 None SEP261 SEP261 XRAY 2.6 0.184 0.221 A 289.0 270.0 3 26 26 0 [[38, 290]] 1.0 6l15 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L16A P11309 33 305 313.0 E2U:401 Type1 Active DFGin 6.3278 14.74 BLAminus -130.86, 166.29 65.26, 82.88 -91.87, 18.01 283.01, 76.97 -72.19, -13.53 in-in in 8.7021 Saltbr-in 2.4147 HRD-naA -67.28, -47.47 67.45, 11.65 in-in-in SNCiii in-in ActLoopNT-in 2.8263 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.92, 16.39 APE9-dihe-na -84.74, -155.75 APE8-dihe-in -95.92, 129.43 APE8-rot-in 310.51 APE67-dihe-in -64.98, -15.76 -62.83, -46.58 APE12-dist-in 9.3102 APE11-dist-in 8.5215 APE10-dist-in 4.7385 APE9-dist-in 3.7782 None SEP261 SEP261 XRAY 2.1 0.199 0.218 A 289.0 270.0 3 26 26 0 [[38, 290]] 1.0 6l16 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6L17A P11309 33 305 313.0 E2X:401 Type1 Active DFGin 6.3235 14.6531 BLAminus -129.55, 165.34 65.87, 81.97 -92.53, 17.46 286.99, 73.6 -66.81, -14.75 in-in in 8.3978 Saltbr-in 2.601 HRD-naA -68.49, -49.87 68.95, 13.18 in-in-in SNCiii in-in ActLoopNT-in 2.8216 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.96, 18.29 APE9-dihe-na -82.73, -153.32 APE8-dihe-in -94.04, 120.15 APE8-rot-in 303.42 APE67-dihe-in -68.29, -9.26 -56.68, -41.93 APE12-dist-in 9.5105 APE11-dist-in 8.5589 APE10-dist-in 5.2242 APE9-dist-in 3.7004 None SEP261 SEP261 XRAY 1.75 0.185 0.205 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6l17 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7XSVA P11309 32 305 313.0 I4M:401 Type1 Active DFGin 6.058 14.3167 BLAminus -136.35, 175.71 54.46, 80.4 -90.61, 15.51 289.45, 76.26 -61.12, -29.45 in-in in 8.1673 Saltbr-in 2.4868 HRD-naA -80.1, -41.91 69.45, -9.52 in-in-in SNCiii in-in ActLoopNT-in 2.7914 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.82, 18.64 APE9-dihe-na -91.64, 171.14 APE8-dihe-in -71.59, 144.23 APE8-rot-in 295.24 APE67-dihe-in -74.83, -31.12 -57.05, -23.4 APE12-dist-in 8.859 APE11-dist-in 8.4261 APE10-dist-in 4.6305 APE9-dist-in 4.8183 None SEP261 SEP261 XRAY 2.66 0.197 0.233 A 289.0 274.0 0 26 26 0 [[38, 290]] 1.0 7xsv Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5KCXA P11309 34 305 313.0 6S3:403 Type1 Active DFGin 6.2209 14.9168 BLAminus -132.88, 167.48 63.01, 80.22 -91.16, 17.8 283.48, 68.85 -71.72, -7.39 in-in in 8.8485 Saltbr-in 2.5228 HRD-naA -73.28, -48.22 75.07, 1.67 in-in-in SNCiii in-in ActLoopNT-in 2.8307 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.64, 15.26 APE9-dihe-na -83.36, -157.62 APE8-dihe-in -86.75, 121.87 APE8-rot-in 307.36 APE67-dihe-in -65.54, -9.34 -59.93, -45.42 APE12-dist-in 9.6483 APE11-dist-in 8.6086 APE10-dist-in 5.2518 APE9-dist-in 3.8637 None None None XRAY 2.2 0.19 0.211 A 291.0 272.0 0 26 26 0 [[38, 290]] 1.0 5kcx Homo sapiens CAMK_PIM1_HUMAN CAMK 3.1e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4MBIA P11309 33 306 313.0 26K:401 Type1 Active DFGin 6.1239 14.4723 BLAminus -131.89, 168.18 61.53, 68.36 -79.59, 15.15 287.22, 79.02 -64.78, -12.91 in-in in 8.6887 Saltbr-in 2.7726 HRD-naA -75.96, -48.7 66.71, 16.19 in-in-in SNCiii in-in ActLoopNT-in 2.7522 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.73, 31.55 APE9-dihe-na -87.7, -149.18 APE8-dihe-in -95.91, 132.2 APE8-rot-in 306.67 APE67-dihe-in -76.77, -11.58 -65.7, -39.07 APE12-dist-in 9.5635 APE11-dist-in 8.4731 APE10-dist-in 5.1024 APE9-dist-in 3.6425 None None None XRAY 2.3 0.215 0.246 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 4mbi Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4MBLA P11309 33 306 313.0 26L:401 Type1 Active DFGin 6.3571 14.6471 BLAminus -140.97, 162.32 61.82, 87.23 -100.32, 23.61 288.64, 85.04 -75.88, -10.71 in-in in 8.4627 Saltbr-in 2.705 HRD-naA -66.61, -53.32 68.87, 14.83 in-in-in SNCiii in-in ActLoopNT-in 2.7923 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.99, 40.01 APE9-dihe-na -114.3, -171.32 APE8-dihe-in -75.76, 118.27 APE8-rot-in 314.72 APE67-dihe-in -58.14, -19.65 -55.56, -49.63 APE12-dist-in 9.0327 APE11-dist-in 8.6582 APE10-dist-in 4.8819 APE9-dist-in 4.1912 None None None XRAY 2.6 0.202 0.242 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 4mbl Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXVA P11309 33 306 313.0 LI6:323 Type1 Active DFGin 6.1534 14.6197 BLAminus -131.19, 171.32 56.28, 85.76 -94.29, 14.73 284.91, 75.06 -64.34, -11.63 in-in in 8.8928 Saltbr-in 2.5423 HRD-naA -66.61, -47.26 65.08, 9.89 in-in-in SNCiii in-in ActLoopNT-in 2.9207 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.55, 31.12 APE9-dihe-na -89.85, -157.25 APE8-dihe-in -87.05, 122.1 APE8-rot-in 305.25 APE67-dihe-in -67.3, -11.88 -57.54, -43.12 APE12-dist-in 9.6965 APE11-dist-in 8.4898 APE10-dist-in 5.4378 APE9-dist-in 3.7355 None None None XRAY 2.0 0.189 0.211 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxv Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1YXXA P11309 33 306 313.0 LI7:323 Type1 Active DFGin 6.1644 14.4349 BLAminus -118.82, 172.49 62.96, 83.76 -93.84, 24.35 282.94, 80.67 -77.24, -2.76 in-in in 8.8737 Saltbr-in 2.4462 HRD-naA -72.3, -43.39 62.78, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.9232 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.23, 43.27 APE9-dihe-na -100.31, -154.93 APE8-dihe-in -89.78, 124.47 APE8-rot-in 309.92 APE67-dihe-in -69.42, -9.61 -60.64, -40.01 APE12-dist-in 9.7437 APE11-dist-in 8.4051 APE10-dist-in 5.643 APE9-dist-in 3.8007 None None None XRAY 2.0 0.219 0.251 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 1yxx Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2O3PA P11309 33 306 313.0 QUE:501 Type1 Active DFGin 6.2383 14.5362 BLAminus -130.88, 170.78 53.54, 90.02 -97.28, 20.48 282.33, 78.83 -71.95, -12.75 in-in in 8.6674 Saltbr-in 2.2959 HRD-naA -68.04, -46.2 63.08, 8.81 in-in-in SNCiii in-in ActLoopNT-in 2.8581 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.42, 29.49 APE9-dihe-na -90.86, -153.23 APE8-dihe-in -86.96, 125.45 APE8-rot-in 306.17 APE67-dihe-in -64.91, -8.64 -61.09, -46.67 APE12-dist-in 9.6614 APE11-dist-in 8.5306 APE10-dist-in 5.4294 APE9-dist-in 3.8478 None None None XRAY 2.24 0.189 0.22 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o3p Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2O63A P11309 33 306 313.0 MYC:501 Type1 Active DFGin 6.0925 14.4288 BLAminus -133.37, 172.38 63.28, 75.17 -88.32, 15.11 286.1, 77.55 -67.51, -7.66 in-in in 8.5833 Saltbr-in 2.552 HRD-naA -71.09, -45.59 61.3, 13.27 in-in-in SNCiii in-in ActLoopNT-in 2.9029 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.73, 31.74 APE9-dihe-na -90.0, -152.24 APE8-dihe-in -91.1, 122.3 APE8-rot-in 305.54 APE67-dihe-in -66.75, -10.3 -56.16, -45.71 APE12-dist-in 9.8969 APE11-dist-in 8.6251 APE10-dist-in 5.6381 APE9-dist-in 3.7828 None None None XRAY 2.0 0.194 0.218 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o63 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2O64A P11309 33 306 313.0 MYU:501 Type1 Active DFGin 6.2715 14.6755 BLAminus -128.75, 172.17 61.57, 79.87 -92.44, 15.52 285.23, 76.88 -62.99, -16.57 in-in in 8.4121 Saltbr-in 2.672 HRD-naA -65.21, -51.23 71.84, 4.17 in-in-in SNCiii in-in ActLoopNT-in 2.9535 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.67, 34.14 APE9-dihe-na -99.78, -147.67 APE8-dihe-in -92.72, 124.85 APE8-rot-in 309.85 APE67-dihe-in -64.3, -15.3 -61.26, -48.06 APE12-dist-in 9.6056 APE11-dist-in 8.584 APE10-dist-in 5.4192 APE9-dist-in 3.9479 None None None XRAY 2.44 0.191 0.23 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o64 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2O65A P11309 33 306 313.0 MYF:501 Type1 Active DFGin 5.7731 14.2228 BLAminus -134.9, 170.04 60.08, 89.22 -101.35, 10.62 287.34, 92.73 -63.96, -9.9 in-in in 8.7039 Saltbr-in 2.4715 HRD-naA -65.14, -47.59 70.03, -4.07 in-in-in SNCiii in-in ActLoopNT-in 2.9803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.66, 34.64 APE9-dihe-na -104.35, -148.26 APE8-dihe-in -83.11, 121.1 APE8-rot-in 316.59 APE67-dihe-in -62.15, -16.44 -57.04, -47.52 APE12-dist-in 9.9881 APE11-dist-in 8.6279 APE10-dist-in 5.2887 APE9-dist-in 4.1355 None None None XRAY 2.85 0.21 0.262 A 293.0 274.0 0 26 26 0 [[38, 290]] 1.0 2o65 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3JXWA P11309 33 306 313.0 LXG:1000 Type1 Active DFGin 6.2103 14.5966 BLAminus -134.41, 162.67 73.18, 86.78 -94.42, 16.28 283.72, 78.67 -67.2, -7.05 in-in in 8.9431 Saltbr-in 2.7638 HRD-naA -66.64, -45.65 67.32, 6.42 in-in-in SNCiii in-in ActLoopNT-in 2.7858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.1, 39.58 APE9-dihe-na -109.74, -153.05 APE8-dihe-in -85.54, 118.8 APE8-rot-in 317.48 APE67-dihe-in -60.88, -20.58 -50.76, -58.31 APE12-dist-in 9.5275 APE11-dist-in 8.5452 APE10-dist-in 5.4917 APE9-dist-in 4.2563 None None None XRAY 2.8 0.219 0.266 A 294.0 274.0 0 26 26 0 [[38, 290]] 1.0 3jxw Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3JY0A P11309 33 307 313.0 LYG:1000 Type1 Active DFGin 5.9655 14.4592 BLAminus -136.0, 169.05 67.14, 86.13 -88.57, 12.42 285.25, 84.28 -62.59, -9.01 in-in in 8.897 Saltbr-in 2.5785 HRD-naA -73.59, -52.32 72.38, 9.82 in-in-in SNCiii in-in ActLoopNT-in 2.7783 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.33, 17.31 APE9-dihe-na -90.28, -146.77 APE8-dihe-in -93.89, 122.92 APE8-rot-in 318.19 APE67-dihe-in -68.56, -0.09 -56.36, -49.84 APE12-dist-in 9.7621 APE11-dist-in 8.4913 APE10-dist-in 4.9707 APE9-dist-in 3.8014 None None None XRAY 2.4 0.226 0.257 A 294.0 275.0 0 26 26 0 [[38, 290]] 1.0 3jy0 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3JYAA P11309 33 306 313.0 LWG:1000 Type1 Active DFGin 6.2096 14.5113 BLAminus -132.92, 173.52 45.25, 85.32 -90.21, 14.37 285.74, 75.57 -67.67, -13.84 in-in in 9.0619 Saltbr-in 2.4726 HRD-naA -71.42, -47.46 64.92, 10.13 in-in-in SNCiii in-in ActLoopNT-in 2.7063 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.34, 26.83 APE9-dihe-na -88.37, -156.09 APE8-dihe-in -89.17, 119.95 APE8-rot-in 305.54 APE67-dihe-in -68.16, -12.31 -55.92, -42.85 APE12-dist-in 9.5401 APE11-dist-in 8.4965 APE10-dist-in 5.3913 APE9-dist-in 3.7507 None None None XRAY 2.1 0.234 0.257 A 294.0 274.0 0 26 26 0 [[38, 290]] 1.0 3jya Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5O11A P11309 34 305 313.0 3NG:401 Type1 Active DFGin 6.1285 14.6109 BLAminus -127.88, 174.91 62.14, 80.5 -88.8, 17.09 290.86, 80.03 -61.06, -19.7 in-in in 8.8564 Saltbr-in 2.6066 HRD-naA -68.12, -50.16 69.42, 1.48 in-in-in SNCiii in-in ActLoopNT-in 2.8771 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.35, 8.9 APE9-dihe-na -86.78, -150.83 APE8-dihe-in -93.81, 133.37 APE8-rot-in 308.93 APE67-dihe-in -69.86, -10.11 -67.48, -44.09 APE12-dist-in 9.7422 APE11-dist-in 8.7304 APE10-dist-in 4.8611 APE9-dist-in 3.817 None SEP261 CME161,SEP261 XRAY 2.4 0.167 0.212 A 298.0 270.0 2 26 26 0 [[38, 290]] 1.0 5o11 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5O12A P11309 34 305 313.0 1RO:401 Type1 Active DFGin 6.2318 14.4999 BLAminus -126.26, 172.57 61.88, 84.82 -89.13, 24.53 288.01, 80.82 -77.95, -15.0 in-in in 8.881 Saltbr-in 2.7 HRD-naA -70.16, -50.1 71.34, 2.69 in-in-in SNCiii in-in ActLoopNT-in 2.8956 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.86, 30.76 APE9-dihe-na -86.98, -148.45 APE8-dihe-in -99.72, 127.71 APE8-rot-in 312.69 APE67-dihe-in -67.78, -9.89 -65.97, -45.8 APE12-dist-in 9.5158 APE11-dist-in 8.4456 APE10-dist-in 5.6506 APE9-dist-in 3.7177 None SEP261 CME161,SEP261 XRAY 2.4 0.179 0.223 A 298.0 266.0 6 26 26 0 [[38, 290]] 1.0 5o12 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5O13A P11309 34 305 313.0 9G5:401 Type1 Active DFGin 6.232 14.5703 BLAminus -126.22, 173.43 61.18, 82.34 -90.65, 15.63 288.81, 77.08 -66.25, -16.88 in-in in 8.8079 Saltbr-in 2.6206 HRD-naA -66.53, -48.7 66.86, 2.99 in-in-in SNCiii in-in ActLoopNT-in 2.8173 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.42, 11.87 APE9-dihe-na -70.23, -134.62 APE8-dihe-in -110.38, 131.64 APE8-rot-in 317.06 APE67-dihe-in -70.9, -10.23 -68.47, -45.42 APE12-dist-in 9.6816 APE11-dist-in 8.5431 APE10-dist-in 5.4383 APE9-dist-in 4.0623 None SEP261 CSX161,SEP261 XRAY 2.44 0.162 0.214 A 298.0 272.0 0 26 26 0 [[38, 290]] 1.0 5o13 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5DGZA P11309 33 305 313.0 L20:401 Type1 Active DFGin 6.3283 14.8412 BLAminus -128.71, 169.75 60.97, 88.72 -102.55, 22.85 284.63, 77.63 -73.84, -14.69 in-in in 8.5704 Saltbr-in 2.5393 HRD-naA -79.61, -44.74 68.32, 8.97 in-in-in SNCiii in-in ActLoopNT-in 2.9586 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.12, 19.6 APE9-dihe-na -84.49, -168.79 APE8-dihe-in -78.12, 137.4 APE8-rot-in 353.29 APE67-dihe-in -67.56, -8.39 -54.96, -54.27 APE12-dist-in 9.4821 APE11-dist-in 8.7924 APE10-dist-in 5.0905 APE9-dist-in 3.8694 None None None XRAY 2.502 0.182 0.213 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5dgz Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5DHJA P11309 33 305 313.0 5E5:401 Type1 Active DFGin 6.2772 14.6413 BLAminus -132.48, 165.98 68.77, 75.26 -89.6, 23.34 285.29, 75.18 -66.63, -15.53 in-in in 8.6776 Saltbr-in 2.5997 HRD-naA -74.9, -49.69 73.89, 5.62 in-in-in SNCiii in-in ActLoopNT-in 2.8008 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.14, 28.7 APE9-dihe-na -93.46, -149.0 APE8-dihe-in -88.51, 125.57 APE8-rot-in 319.11 APE67-dihe-in -63.27, -9.53 -60.93, -48.3 APE12-dist-in 9.6899 APE11-dist-in 8.7094 APE10-dist-in 5.5758 APE9-dist-in 3.8895 None None None XRAY 2.457 0.191 0.25 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5dhj Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5DIAA P11309 33 305 313.0 5E6:401 Type1 Active DFGin 6.1094 14.3642 BLAminus -131.51, 162.73 65.64, 95.79 -106.0, 22.43 288.31, 75.68 -70.61, -13.53 in-in in 8.8932 Saltbr-in 2.6632 HRD-naA -70.21, -53.43 79.23, -0.98 in-in-in SNCiii in-in ActLoopNT-in 2.8151 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.54, 25.72 APE9-dihe-na -78.57, -156.72 APE8-dihe-in -91.47, 121.1 APE8-rot-in 309.49 APE67-dihe-in -70.58, -6.62 -58.72, -40.2 APE12-dist-in 9.6002 APE11-dist-in 8.6495 APE10-dist-in 5.4875 APE9-dist-in 3.7674 None None None XRAY 1.964 0.198 0.229 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5dia Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5V80A P11309 33 305 313.0 971:402 Type1 Active DFGin 6.2933 14.711 BLAminus -125.21, 168.1 67.15, 84.62 -97.5, 21.56 283.85, 73.58 -74.5, -9.73 in-in in 8.8229 Saltbr-in 2.4892 HRD-naA -71.2, -48.76 73.46, -4.54 in-in-in SNCiii in-in ActLoopNT-in 2.8494 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 17.28 APE9-dihe-na -81.45, -156.95 APE8-dihe-in -91.64, 124.53 APE8-rot-in 310.44 APE67-dihe-in -65.24, -8.9 -57.42, -46.72 APE12-dist-in 9.6206 APE11-dist-in 8.7016 APE10-dist-in 5.1963 APE9-dist-in 3.9237 None None None XRAY 2.252 0.177 0.212 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5v80 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5V82A P11309 34 306 313.0 96Y:401 Type1 Active DFGin 6.2131 14.4118 BLAminus -125.78, 171.27 64.15, 78.85 -91.71, 19.69 286.42, 77.38 -68.31, -20.73 in-in in 8.8236 Saltbr-in 2.5709 HRD-naA -70.88, -47.55 68.67, 4.77 in-in-in SNCiii in-in ActLoopNT-in 2.7889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.07, 17.68 APE9-dihe-na -81.71, -152.79 APE8-dihe-in -94.55, 121.67 APE8-rot-in 301.55 APE67-dihe-in -68.27, -8.9 -60.36, -41.63 APE12-dist-in 9.7433 APE11-dist-in 8.6739 APE10-dist-in 5.1826 APE9-dist-in 3.5857 None None None XRAY 1.888 0.182 0.199 A 299.0 273.0 0 26 26 0 [[38, 290]] 1.0 5v82 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3UIXA P11309 37 305 313.0 Q17:400 Type1 Active DFGin 6.1591 14.8214 BLAminus -133.2, 170.02 65.66, 77.49 -86.97, 13.03 288.74, 81.94 -68.85, -14.59 in-in in 9.0654 Saltbr-in 2.8853 HRD-naA -68.2, -50.15 66.82, 5.77 in-in-in SNCiii in-in ActLoopNT-in 2.7993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.4, 30.15 APE9-dihe-na -90.24, -149.24 APE8-dihe-in -93.32, 120.98 APE8-rot-in 306.79 APE67-dihe-in -70.28, -11.9 -58.72, -40.96 APE12-dist-in 9.6064 APE11-dist-in 8.5237 APE10-dist-in 5.4885 APE9-dist-in 3.7562 None None None XRAY 2.2 0.168 0.201 A 298.0 266.0 3 26 26 0 [[38, 290]] 1.0 3uix Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3UMWA P11309 37 304 313.0 596:400 Type1 Active DFGin 6.2909 14.5837 BLAminus -128.68, 168.78 67.21, 80.33 -91.49, 18.98 287.81, 74.46 -67.02, -11.8 in-in in 8.4885 Saltbr-in 2.8503 HRD-naA -69.92, -48.57 70.74, 4.13 in-in-in SNCiii in-in ActLoopNT-in 2.8096 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.82, 23.54 APE9-dihe-na -81.68, -155.27 APE8-dihe-in -92.32, 121.26 APE8-rot-in 306.5 APE67-dihe-in -69.25, -11.28 -53.65, -48.44 APE12-dist-in 9.1537 APE11-dist-in 8.5631 APE10-dist-in 5.5517 APE9-dist-in 3.7718 None None None XRAY 2.08 0.175 0.2 A 298.0 264.0 4 26 26 0 [[38, 290]] 1.0 3umw Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3UMXA P11309 37 304 313.0 Q18:400 Type1 Active DFGin 6.3211 14.6927 BLAminus -128.18, 168.05 66.13, 83.77 -95.39, 17.61 280.32, 78.57 -66.8, -16.44 in-in in 8.4362 Saltbr-in 2.9518 HRD-naA -70.86, -46.1 72.14, -3.21 in-in-in SNCiii in-in ActLoopNT-in 2.9654 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.18, 34.19 APE9-dihe-na -90.9, -156.14 APE8-dihe-in -92.65, 120.83 APE8-rot-in 316.33 APE67-dihe-in -56.49, -20.39 -55.25, -56.16 APE12-dist-in 9.0182 APE11-dist-in 8.6132 APE10-dist-in 5.466 APE9-dist-in 3.9429 None None None XRAY 2.55 0.18 0.229 A 298.0 261.0 7 26 26 0 [[38, 290]] 1.0 3umx Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4ENXA P11309 37 305 313.0 Z20:402 Type1 Active DFGin 6.0724 14.2577 BLAminus -124.23, 174.95 56.93, 87.82 -99.36, 21.71 285.95, 80.74 -78.01, -5.47 in-in in 8.7919 Saltbr-in 2.4703 HRD-naA -68.51, -45.47 67.84, 12.31 in-in-in SNCiii in-in ActLoopNT-in 2.803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.34, 41.24 APE9-dihe-na -101.41, -153.2 APE8-dihe-in -90.61, 127.01 APE8-rot-in 310.22 APE67-dihe-in -64.59, -15.43 -67.29, -43.92 APE12-dist-in 9.2342 APE11-dist-in 8.6621 APE10-dist-in 5.4211 APE9-dist-in 3.7373 None None None XRAY 2.8 0.192 0.233 A 298.0 266.0 3 26 26 0 [[38, 290]] 1.0 4enx Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4ENYA P11309 37 305 313.0 J19:404 Type1 Active DFGin 6.1683 14.409 BLAminus -126.77, 176.31 56.15, 81.83 -92.01, 22.92 285.19, 76.91 -75.2, -11.55 in-in in 8.8121 Saltbr-in 2.6741 HRD-naA -67.09, -45.67 67.16, 8.93 in-in-in SNCiii in-in ActLoopNT-in 2.7579 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.12, 33.6 APE9-dihe-na -103.74, -163.7 APE8-dihe-in -76.76, 123.85 APE8-rot-in 309.22 APE67-dihe-in -67.99, -11.42 -63.9, -43.13 APE12-dist-in 9.4542 APE11-dist-in 8.6678 APE10-dist-in 5.2094 APE9-dist-in 3.8101 None None None XRAY 2.801 0.175 0.224 A 298.0 261.0 8 26 26 0 [[38, 290]] 1.0 4eny Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4LL5A P11309 34 305 313.0 SK8:401 Type1 Active DFGin 6.1536 14.9413 BLAminus -130.09, 167.4 64.64, 85.24 -96.78, 19.13 285.46, 79.08 -67.1, -17.77 in-in in 8.9048 Saltbr-in 2.9074 HRD-naA -72.89, -48.94 71.1, 5.66 in-in-in SNCiii in-in ActLoopNT-in 2.8583 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.97, 33.17 APE9-dihe-na -91.19, -159.67 APE8-dihe-in -86.75, 127.22 APE8-rot-in 309.08 APE67-dihe-in -69.44, -9.3 -64.52, -42.1 APE12-dist-in 9.5929 APE11-dist-in 8.6246 APE10-dist-in 5.5027 APE9-dist-in 3.7227 None None None XRAY 2.0 0.169 0.189 A 298.0 268.0 4 26 26 0 [[38, 290]] 1.0 4ll5 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4LM5A P11309 35 305 313.0 Q17:401 Type1 Active DFGin 6.1717 14.8472 BLAminus -129.33, 170.23 65.43, 81.43 -93.64, 15.07 286.04, 82.64 -63.86, -18.24 in-in in 9.1345 Saltbr-in 2.7309 HRD-naA -69.11, -47.25 68.05, 2.81 in-in-in SNCiii in-in ActLoopNT-in 2.8293 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.68, 24.87 APE9-dihe-na -83.15, -151.88 APE8-dihe-in -95.39, 124.37 APE8-rot-in 310.14 APE67-dihe-in -64.57, -11.11 -60.82, -46.98 APE12-dist-in 9.5104 APE11-dist-in 8.5146 APE10-dist-in 5.4234 APE9-dist-in 3.7127 None None CSO161 XRAY 2.25 0.158 0.198 A 298.0 265.0 6 26 26 0 [[38, 290]] 1.0 4lm5 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4LMUA P11309 36 304 313.0 QUE:401 Type1 Active DFGin 6.1615 14.4307 BLAminus -125.85, 174.43 58.26, 85.32 -97.42, 18.39 285.76, 76.14 -68.38, -9.73 in-in in 8.702 Saltbr-in 2.3854 HRD-naA -71.42, -45.75 68.18, 3.07 in-in-in SNCiii in-in ActLoopNT-in 2.8482 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.78, 30.35 APE9-dihe-na -86.53, -151.77 APE8-dihe-in -97.13, 122.66 APE8-rot-in 306.98 APE67-dihe-in -65.32, -7.73 -59.99, -46.55 APE12-dist-in 9.4521 APE11-dist-in 8.6168 APE10-dist-in 5.5144 APE9-dist-in 3.8345 None None None XRAY 2.38 0.172 0.204 A 298.0 265.0 4 26 26 0 [[38, 290]] 1.0 4lmu Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5VUAB P11309 36 305 313.0 8GX:403 Type1 Active DFGin 6.2674 14.6306 BLAminus -131.5, 169.5 65.68, 85.46 -98.43, 24.84 284.2, 75.16 -72.94, -9.76 in-in in 8.4537 Saltbr-in 2.8407 HRD-naA -72.0, -46.73 70.73, 2.09 in-in-in SNCiii in-in ActLoopNT-in 2.8479 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.51, 33.95 APE9-dihe-na -87.15, -156.37 APE8-dihe-in -92.0, 123.34 APE8-rot-in 311.17 APE67-dihe-in -66.19, -11.92 -56.69, -48.02 APE12-dist-in 9.2638 APE11-dist-in 8.5434 APE10-dist-in 5.6059 APE9-dist-in 3.7837 None None None XRAY 2.2 0.167 0.196 B 298.0 270.0 0 26 26 0 [[38, 290]] 1.0 5vua Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5VUBB P11309 36 305 313.0 8GU:402 Type1 Active DFGin 6.2652 14.6046 BLAminus -124.74, 173.14 60.11, 84.16 -95.33, 18.9 286.57, 72.73 -67.18, -11.28 in-in in 8.585 Saltbr-in 2.3633 HRD-naA -74.43, -46.89 71.06, 5.3 in-in-in SNCiii in-in ActLoopNT-in 2.8541 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.25, 31.18 APE9-dihe-na -85.43, -151.45 APE8-dihe-in -96.33, 120.96 APE8-rot-in 305.35 APE67-dihe-in -68.9, -7.9 -56.39, -44.27 APE12-dist-in 9.3708 APE11-dist-in 8.5694 APE10-dist-in 5.5734 APE9-dist-in 3.6525 None None CSO161 XRAY 2.0 0.161 0.184 B 298.0 270.0 0 26 26 0 [[38, 290]] 1.0 5vub Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5VUCB P11309 36 305 313.0 8GR:402 Type1 Active DFGin 6.2599 14.5902 BLAminus -130.18, 165.22 63.78, 87.26 -96.8, 21.67 286.89, 72.33 -70.38, -11.1 in-in in 8.2713 Saltbr-in 2.7802 HRD-naA -75.49, -49.39 71.96, 7.41 in-in-in SNCiii in-in ActLoopNT-in 2.9022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.01, 27.32 APE9-dihe-na -81.89, -157.57 APE8-dihe-in -92.9, 123.77 APE8-rot-in 305.96 APE67-dihe-in -68.92, -9.19 -62.84, -43.07 APE12-dist-in 9.1928 APE11-dist-in 8.5586 APE10-dist-in 5.4339 APE9-dist-in 3.7674 None None CSO161 XRAY 2.0 0.176 0.199 B 298.0 270.0 0 26 26 0 [[38, 290]] 1.0 5vuc Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3R00A P11309 33 306 313.0 UNJ:1 Type1 Active DFGin 6.0775 14.5853 BLAminus -129.23, 179.95 62.78, 78.65 -92.67, 17.69 284.89, 76.92 -65.27, -12.58 in-in in 8.9851 Saltbr-in 2.6149 HRD-naA -69.03, -46.16 61.18, 15.3 in-in-in SNCiii in-in ActLoopNT-in 2.8737 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.83, 36.17 APE9-dihe-na -94.5, -143.14 APE8-dihe-in -99.32, 120.22 APE8-rot-in 298.64 APE67-dihe-in -66.4, -11.74 -58.9, -42.32 APE12-dist-in 9.8111 APE11-dist-in 8.5314 APE10-dist-in 5.6392 APE9-dist-in 3.7189 None None None XRAY 2.1 0.175 0.216 A 299.0 274.0 0 26 26 0 [[38, 290]] 1.0 3r00 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3R01A P11309 33 306 313.0 UNE:1 Type1 Active DFGin 6.1709 14.6386 BLAminus -135.6, 167.7 70.77, 75.77 -84.82, 17.16 285.86, 84.24 -68.67, -10.33 in-in in 8.8032 Saltbr-in 2.8831 HRD-naA -70.35, -49.23 74.71, 2.68 in-in-in SNCiii in-in ActLoopNT-in 2.8788 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.59, 35.76 APE9-dihe-na -87.25, -132.26 APE8-dihe-in -117.56, 118.78 APE8-rot-in 316.73 APE67-dihe-in -73.58, -11.68 -54.47, -42.96 APE12-dist-in 9.7376 APE11-dist-in 8.5085 APE10-dist-in 5.818 APE9-dist-in 3.9243 None None None XRAY 2.6 0.219 0.287 A 299.0 274.0 0 26 26 0 [[38, 290]] 1.0 3r01 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3R02A P11309 35 305 313.0 UNM:555 Type1 Active DFGin 6.1751 14.5657 BLAminus -128.64, 175.57 56.97, 87.35 -90.49, 17.56 285.73, 81.34 -74.51, -7.05 in-in in 9.0281 Saltbr-in 2.6339 HRD-naA -75.58, -44.47 72.61, 3.3 in-in-in SNCiii in-in ActLoopNT-in 2.8106 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.47, 29.58 APE9-dihe-na -87.11, -147.11 APE8-dihe-in -98.53, 121.85 APE8-rot-in 301.03 APE67-dihe-in -70.13, -7.69 -53.51, -42.81 APE12-dist-in 9.8451 APE11-dist-in 8.5843 APE10-dist-in 5.7937 APE9-dist-in 3.7583 None None None XRAY 1.95 0.168 0.189 A 299.0 271.0 0 26 26 0 [[38, 290]] 1.0 3r02 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3R04A P11309 35 305 313.0 UNQ:555 Type1 Active DFGin 6.1113 14.4928 BLAminus -119.88, 174.34 65.61, 74.31 -82.3, 14.36 287.66, 74.37 -62.06, -16.62 in-in in 8.9281 Saltbr-in 2.6342 HRD-naA -74.82, -45.09 62.9, 11.66 in-in-in SNCiii in-in ActLoopNT-in 2.8523 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.54, 31.05 APE9-dihe-na -88.35, -143.56 APE8-dihe-in -101.19, 121.66 APE8-rot-in 294.82 APE67-dihe-in -73.54, -5.15 -62.57, -37.68 APE12-dist-in 9.8484 APE11-dist-in 8.5024 APE10-dist-in 5.6442 APE9-dist-in 3.7219 None None None XRAY 1.7 0.179 0.206 A 299.0 271.0 0 26 26 0 [[38, 290]] 1.0 3r04 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VBQA P11309 35 305 313.0 0F5:555 Type1 Active DFGin 6.1979 14.5767 BLAminus -127.7, 179.22 57.68, 76.69 -85.86, 12.59 286.24, 73.15 -68.96, -5.86 in-in in 8.7676 Saltbr-in 2.64 HRD-naA -70.31, -44.96 66.03, 8.09 in-in-in SNCiii in-in ActLoopNT-in 2.8903 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.65, 27.89 APE9-dihe-na -90.08, -142.39 APE8-dihe-in -98.6, 121.83 APE8-rot-in 304.23 APE67-dihe-in -72.3, -7.09 -58.75, -37.63 APE12-dist-in 9.8116 APE11-dist-in 8.5951 APE10-dist-in 5.6985 APE9-dist-in 3.7029 None None None XRAY 1.85 0.206 0.206 A 299.0 271.0 0 26 26 0 [[38, 290]] 1.0 3vbq Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VBTA P11309 35 305 313.0 0F9:1 Type1 Active DFGin 6.1544 14.4155 BLAminus -130.27, 172.67 63.33, 71.31 -82.69, 17.12 286.5, 71.57 -76.38, -5.32 in-in in 8.7106 Saltbr-in 2.6583 HRD-naA -67.81, -46.73 67.69, 4.14 in-in-in SNCiii in-in ActLoopNT-in 2.8556 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.09, 27.22 APE9-dihe-na -88.86, -143.07 APE8-dihe-in -97.4, 123.61 APE8-rot-in 305.69 APE67-dihe-in -63.29, -9.77 -57.85, -48.3 APE12-dist-in 9.4897 APE11-dist-in 8.3934 APE10-dist-in 5.6037 APE9-dist-in 3.764 None None None XRAY 2.23 0.273 0.273 A 299.0 267.0 4 26 26 0 [[38, 290]] 1.0 3vbt Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VBVA P11309 35 305 313.0 0FK:1 Type1 Active DFGin 6.1684 14.5244 BLAminus -132.06, 170.0 63.81, 81.21 -91.04, 16.51 285.74, 75.33 -71.88, -8.41 in-in in 8.8343 Saltbr-in 2.6332 HRD-naA -65.91, -47.52 66.96, 5.14 in-in-in SNCiii in-in ActLoopNT-in 2.8482 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.35, 27.86 APE9-dihe-na -84.91, -139.46 APE8-dihe-in -108.06, 126.97 APE8-rot-in 303.82 APE67-dihe-in -70.7, -8.74 -60.57, -44.13 APE12-dist-in 9.4986 APE11-dist-in 8.4391 APE10-dist-in 5.6633 APE9-dist-in 3.6721 None None None XRAY 2.08 0.245 0.245 A 299.0 268.0 3 26 26 0 [[38, 290]] 1.0 3vbv Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VBWA P11309 35 305 313.0 0FN:1 Type1 Active DFGin 6.0586 14.28 BLAminus -127.49, 167.57 67.98, 79.4 -86.02, 16.62 293.39, 81.3 -60.91, -19.46 in-in in 8.8607 Saltbr-in 2.8787 HRD-naA -70.94, -49.39 81.06, -4.45 in-in-in SNCiii in-in ActLoopNT-in 2.7981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.47, 33.12 APE9-dihe-na -84.03, -133.93 APE8-dihe-in -105.55, 127.02 APE8-rot-in 315.81 APE67-dihe-in -63.23, -11.02 -61.62, -47.09 APE12-dist-in 9.5414 APE11-dist-in 8.3432 APE10-dist-in 5.6723 APE9-dist-in 3.8503 None None None XRAY 2.48 0.299 0.299 A 299.0 264.0 7 26 26 0 [[38, 290]] 1.0 3vbw Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VBXA P11309 35 305 313.0 0FO:1 Type1 Active DFGin 6.0578 14.5368 BLAminus -132.08, 169.91 71.33, 70.33 -85.72, 14.8 288.27, 79.72 -65.16, -16.66 in-in in 8.9539 Saltbr-in 2.6816 HRD-naA -64.87, -49.91 70.18, 2.86 in-in-in SNCiii in-in ActLoopNT-in 2.7949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.29, 28.64 APE9-dihe-na -87.57, -146.06 APE8-dihe-in -95.38, 125.1 APE8-rot-in 301.97 APE67-dihe-in -65.7, -15.04 -61.83, -41.49 APE12-dist-in 9.426 APE11-dist-in 8.3985 APE10-dist-in 5.5184 APE9-dist-in 3.8074 None None None XRAY 2.03 0.258 0.258 A 299.0 268.0 3 26 26 0 [[38, 290]] 1.0 3vbx Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VBYA P11309 35 305 313.0 0FR:1 Type1 Active DFGin 6.1427 14.6314 BLAminus -131.01, 169.0 66.5, 79.73 -89.48, 18.31 287.57, 72.75 -74.21, -13.52 in-in in 8.9517 Saltbr-in 2.7609 HRD-naA -68.42, -44.76 63.69, 3.49 in-in-in SNCiii in-in ActLoopNT-in 2.7963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.13, 34.14 APE9-dihe-na -92.9, -153.09 APE8-dihe-in -93.99, 123.58 APE8-rot-in 305.15 APE67-dihe-in -72.64, -2.35 -57.97, -45.41 APE12-dist-in 9.3282 APE11-dist-in 8.3473 APE10-dist-in 5.5122 APE9-dist-in 3.8248 None None None XRAY 2.27 0.261 0.261 A 299.0 267.0 4 26 26 0 [[38, 290]] 1.0 3vby Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3VC4A P11309 33 306 313.0 0FS:1 Type1 Active DFGin 6.0756 14.6091 BLAminus -139.74, 164.89 72.09, 84.05 -96.17, 20.14 288.43, 67.45 -72.44, -2.97 in-in in 9.0297 Saltbr-in 2.6612 HRD-naA -61.2, -51.03 71.16, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.7242 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.23, 31.29 APE9-dihe-na -95.97, -149.39 APE8-dihe-in -93.38, 121.01 APE8-rot-in 311.86 APE67-dihe-in -66.44, -6.52 -55.27, -50.39 APE12-dist-in 9.953 APE11-dist-in 8.5606 APE10-dist-in 5.4613 APE9-dist-in 3.8012 None None None XRAY 2.23 0.319 0.319 A 299.0 274.0 0 26 26 0 [[38, 290]] 1.0 3vc4 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3F2AA P11309 32 308 313.0 985:1 Type1 Active DFGin 6.0885 14.3121 BLAminus -128.57, 176.64 59.08, 83.27 -93.92, 21.71 288.01, 71.24 -68.66, -6.64 in-in in 8.7442 Saltbr-in 2.7888 HRD-naA -68.81, -50.19 71.47, 2.55 in-in-in SNCiii in-in ActLoopNT-in 2.8314 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.81, 27.99 APE9-dihe-na -90.31, -146.93 APE8-dihe-in -92.75, 125.96 APE8-rot-in 310.85 APE67-dihe-in -59.77, -4.55 -52.49, -57.5 APE12-dist-in 9.8822 APE11-dist-in 8.7738 APE10-dist-in 5.5518 APE9-dist-in 3.6432 None SEP261 SEP261 XRAY 1.9 0.256 0.282 A 300.0 277.0 0 26 26 0 [[38, 290]] 1.0 3f2a Homo sapiens CAMK_PIM1_HUMAN CAMK 3.4e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2XIXA P11309 33 306 313.0 XIX:1307 Type1 Active DFGin 6.198 14.4047 BLAminus -127.72, 172.47 53.38, 85.02 -93.57, 22.7 288.78, 75.96 -73.48, -9.49 in-in in 8.7954 Saltbr-in 2.6185 HRD-naA -70.78, -45.87 74.83, 0.99 in-in-in SNCiii in-in ActLoopNT-in 2.79 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.52, 26.26 APE9-dihe-na -83.36, -151.06 APE8-dihe-in -94.01, 119.49 APE8-rot-in 303.81 APE67-dihe-in -72.45, -16.36 -55.92, -38.22 APE12-dist-in 9.7148 APE11-dist-in 8.6346 APE10-dist-in 5.6984 APE9-dist-in 3.6685 None SEP261,SEP276 SEP261,SEP276 XRAY 2.4 0.173 0.214 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xix Homo sapiens CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2XIYA P11309 33 306 313.0 XIY:1307 Type1 Active DFGin 6.3046 14.5836 BLAminus -122.45, 177.21 60.39, 73.41 -90.27, 13.91 284.0, 74.82 -69.72, -11.86 in-in in 9.0115 Saltbr-in 2.5935 HRD-naA -65.92, -48.71 70.04, 1.22 in-in-in SNCiii in-in ActLoopNT-in 2.7462 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.76, 20.93 APE9-dihe-na -80.08, -150.81 APE8-dihe-in -97.46, 126.22 APE8-rot-in 306.41 APE67-dihe-in -71.61, -13.32 -59.57, -41.49 APE12-dist-in 9.8366 APE11-dist-in 8.6241 APE10-dist-in 5.5581 APE9-dist-in 3.6392 None SEP261 SEP261 XRAY 2.2 0.172 0.201 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xiy Homo sapiens CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2XIZA P11309 33 306 313.0 XIZ:1307 Type1 Active DFGin 6.1763 14.5485 BLAminus -122.54, 175.77 58.35, 84.58 -93.18, 17.46 282.52, 76.08 -67.84, -13.59 in-in in 8.8664 Saltbr-in 2.5793 HRD-naA -67.92, -44.32 48.8, 19.99 in-in-in SNCiii in-in ActLoopNT-in 2.8687 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.12, 25.76 APE9-dihe-na -79.92, -145.43 APE8-dihe-in -101.02, 126.08 APE8-rot-in 309.36 APE67-dihe-in -71.71, -14.75 -59.22, -39.66 APE12-dist-in 9.7528 APE11-dist-in 8.6841 APE10-dist-in 5.6508 APE9-dist-in 3.6837 None SEP261 SEP261 XRAY 2.21 0.258 0.286 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xiz Homo sapiens CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2XJ0A P11309 33 307 313.0 XJ0:1307 Type1 Active DFGin 5.9294 13.6758 BLAminus -134.6, 165.43 58.42, 101.5 -112.27, 25.85 290.56, 60.01 -70.79, -14.26 in-in in 8.6795 Saltbr-in 2.9659 HRD-naA -62.77, -42.06 61.42, 5.55 in-in-in SNCiii in-in ActLoopNT-in 2.9811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 10.17 APE9-dihe-na -82.33, -169.45 APE8-dihe-in -68.0, 130.83 APE8-rot-in 305.92 APE67-dihe-in -52.49, -21.01 -63.78, -52.51 APE12-dist-in 9.7715 APE11-dist-in 8.4681 APE10-dist-in 4.9761 APE9-dist-in 3.8973 None None None XRAY 3.1 0.218 0.263 A 301.0 275.0 0 26 26 0 [[38, 290]] 1.0 2xj0 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2XJ1A P11309 33 306 313.0 XJ1:1307 Type1 Active DFGin 6.2498 14.2958 BLAminus -129.27, 177.63 56.13, 82.39 -92.13, 21.02 283.59, 76.59 -73.33, -11.63 in-in in 8.8725 Saltbr-in 2.7085 HRD-naA -72.25, -47.05 68.39, 1.49 in-in-in SNCiii in-in ActLoopNT-in 2.6939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.13, 25.06 APE9-dihe-na -81.21, -153.15 APE8-dihe-in -95.3, 123.79 APE8-rot-in 303.34 APE67-dihe-in -71.81, -9.27 -59.4, -42.14 APE12-dist-in 9.8771 APE11-dist-in 8.5709 APE10-dist-in 5.6004 APE9-dist-in 3.6104 None SEP261 SEP261 XRAY 2.13 0.178 0.212 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xj1 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2XJ2A P11309 33 306 313.0 985:1001 Type1 Active DFGin 6.1572 14.3889 BLAminus -121.97, 176.14 56.84, 82.15 -90.5, 18.96 286.44, 74.76 -71.88, -10.32 in-in in 8.8085 Saltbr-in 2.6446 HRD-naA -70.41, -47.45 68.26, 1.41 in-in-in SNCiii in-in ActLoopNT-in 2.7186 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.43, 24.44 APE9-dihe-na -81.03, -149.66 APE8-dihe-in -95.09, 121.86 APE8-rot-in 305.59 APE67-dihe-in -74.97, -11.2 -56.65, -40.34 APE12-dist-in 9.8346 APE11-dist-in 8.6692 APE10-dist-in 5.671 APE9-dist-in 3.522 None SEP261 SEP261 XRAY 2.2 0.169 0.202 A 301.0 274.0 0 26 26 0 [[38, 290]] 1.0 2xj2 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.5e-65 225.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4A7CA P11309 32 305 313.0 E46:1306 Type1 Active DFGin 6.1794 14.789 BLAminus -131.67, 167.73 66.77, 79.73 -90.97, 18.69 290.12, 73.93 -69.69, -11.45 in-in in 8.9034 Saltbr-in 2.5501 HRD-naA -69.9, -49.4 70.62, 3.17 in-in-in SNCiii in-in ActLoopNT-in 2.7677 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.97, 35.42 APE9-dihe-na -90.39, -152.55 APE8-dihe-in -91.86, 121.24 APE8-rot-in 305.64 APE67-dihe-in -69.15, -9.02 -58.09, -44.18 APE12-dist-in 9.5612 APE11-dist-in 8.6243 APE10-dist-in 5.6568 APE9-dist-in 3.8767 None SEP261 SEP261 XRAY 2.3 0.171 0.207 A 308.0 274.0 0 26 26 0 [[38, 290]] 1.0 4a7c Homo sapiens CAMK_PIM1_HUMAN CAMK 3.8e-65 225.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 1XWSA P11309 33 305 313.0 BI1:1001 Type1 Active DFGin 6.1159 14.9341 BLAminus -129.52, 166.95 66.18, 81.14 -88.91, 13.45 284.44, 80.6 -63.86, -15.19 in-in in 8.8578 Saltbr-in 2.8112 HRD-naA -69.66, -47.71 69.42, 1.43 in-in-in SNCiii in-in ActLoopNT-in 2.84 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.43, 26.37 APE9-dihe-na -77.62, -162.66 APE8-dihe-in -79.83, 125.2 APE8-rot-in 307.07 APE67-dihe-in -74.93, -11.45 -55.08, -43.34 APE12-dist-in 9.7063 APE11-dist-in 8.7658 APE10-dist-in 5.8681 APE9-dist-in 3.8449 None None None XRAY 1.8 0.182 0.213 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 1xws Homo sapiens CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4BZNA P11309 33 305 313.0 UGX:1306 Type1 Active DFGin 6.1991 14.5084 BLAminus -123.83, 168.52 64.99, 88.0 -96.39, 24.65 289.87, 72.27 -71.02, -12.29 in-in in 8.3963 Saltbr-in 2.5786 HRD-naA -70.91, -47.25 68.09, 6.65 in-in-in SNCiii in-in ActLoopNT-in 2.868 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.83, 29.38 APE9-dihe-na -84.39, -152.15 APE8-dihe-in -95.81, 123.59 APE8-rot-in 305.15 APE67-dihe-in -71.92, -8.16 -59.74, -41.18 APE12-dist-in 9.3592 APE11-dist-in 8.4435 APE10-dist-in 5.5192 APE9-dist-in 3.6102 None SEP261 SEP261 XRAY 1.9 0.178 0.199 A 314.0 273.0 0 26 26 0 [[38, 290]] 1.0 4bzn Homo sapiens CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4BZOA P11309 33 305 313.0 676:1306 Type1 Active DFGin 6.254 14.7622 BLAminus -127.92, 165.55 68.25, 84.97 -95.87, 20.96 286.29, 72.86 -74.22, -6.71 in-in in 8.4398 Saltbr-in 2.622 HRD-naA -71.06, -49.33 68.13, 9.04 in-in-in SNCiii in-in ActLoopNT-in 2.8672 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.68, 32.17 APE9-dihe-na -87.85, -152.26 APE8-dihe-in -92.39, 123.96 APE8-rot-in 304.04 APE67-dihe-in -67.43, -9.74 -60.54, -43.52 APE12-dist-in 9.6012 APE11-dist-in 8.5854 APE10-dist-in 5.5358 APE9-dist-in 3.6618 None SEP261 SEP261 XRAY 2.1 0.183 0.216 A 314.0 273.0 0 26 26 0 [[38, 290]] 1.0 4bzo Homo sapiens CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7ZUNA P11309 33 305 313.0 JYO:401 Type1 Active DFGin 6.2197 14.2081 BLAminus -133.16, 165.47 67.55, 84.83 -98.38, 21.66 289.12, 75.62 -70.0, -22.74 in-in in 8.2062 Saltbr-in 2.792 HRD-naA -67.79, -58.14 75.87, 8.23 in-in-in SNCiii in-in ActLoopNT-in 2.8668 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.98, 24.87 APE9-dihe-na -93.48, -164.33 APE8-dihe-in -86.18, 121.45 APE8-rot-in 312.27 APE67-dihe-in -61.31, -13.56 -57.48, -51.41 APE12-dist-in 9.4299 APE11-dist-in 8.4442 APE10-dist-in 5.0492 APE9-dist-in 3.8725 None SEP261 SEP261 XRAY 2.5 0.177 0.235 A 314.0 270.0 3 26 26 0 [[38, 290]] 1.0 7zun Homo sapiens CAMK_PIM1_HUMAN CAMK 4e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4XHKB P11309 32 305 313.0 3YR:401 Type1 Active DFGin 6.2265 14.5249 BLAminus -126.44, 167.48 62.73, 73.24 -76.02, 8.65 289.12, 83.25 -72.3, -9.91 in-in in 8.8608 Saltbr-in 2.6139 HRD-naA -68.85, -46.46 65.48, 11.28 in-in-in SNCiii in-in ActLoopNT-in 2.8772 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.53, 24.82 APE9-dihe-na -81.56, -148.04 APE8-dihe-in -105.73, 126.46 APE8-rot-in 298.97 APE67-dihe-in -77.31, -6.66 -69.47, -34.63 APE12-dist-in 9.5732 APE11-dist-in 8.6835 APE10-dist-in 5.642 APE9-dist-in 3.7202 None SEP261 SEP261 XRAY 1.9 0.158 0.184 B 315.0 270.0 4 26 26 0 [[38, 290]] 1.0 4xhk Homo sapiens CAMK_PIM1_HUMAN CAMK 4.1e-65 225.6 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4JX7A P11309 33 306 313.0 1N6:401 Type1 Active DFGin 6.2835 14.7533 BLAminus -127.31, 170.34 63.68, 81.99 -92.92, 12.24 283.66, 75.72 -67.48, -14.52 in-in in 8.8428 Saltbr-in 2.7677 HRD-naA -66.3, -47.17 67.1, 1.58 in-in-in SNCiii in-in ActLoopNT-in 2.7336 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.4, 25.92 APE9-dihe-na -85.09, -149.75 APE8-dihe-in -93.53, 123.68 APE8-rot-in 312.23 APE67-dihe-in -66.8, -17.18 -56.19, -45.11 APE12-dist-in 9.7559 APE11-dist-in 8.5902 APE10-dist-in 5.6048 APE9-dist-in 3.9044 None None None XRAY 2.4 0.193 0.228 A 326.0 274.0 0 26 26 0 [[38, 290]] 1.0 4jx7 Homo sapiens CAMK_PIM1_HUMAN CAMK 4.6e-65 225.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4ALVA P11309 33 306 313.0 R9P:1308 Type1 Active DFGin 6.0359 14.4757 BLAminus -137.53, 165.69 68.25, 83.91 -91.38, 16.23 287.59, 75.48 -60.65, -18.54 in-in in 8.6626 Saltbr-in 2.3403 HRD-naA -75.94, -45.06 66.41, 17.82 in-in-in SNCiii in-in ActLoopNT-in 2.9682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.01, 38.02 APE9-dihe-na -89.15, -139.06 APE8-dihe-in -112.86, 124.4 APE8-rot-in 319.08 APE67-dihe-in -51.23, -17.72 -57.73, -58.1 APE12-dist-in 9.4151 APE11-dist-in 8.6868 APE10-dist-in 5.7072 APE9-dist-in 3.6859 None None None XRAY 2.59 0.195 0.256 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 4alv Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4ALWA P11309 34 306 313.0 HY7:1308 Type1 Active DFGin 6.0045 14.5947 BLAminus -122.86, 171.92 71.12, 81.46 -94.23, 18.88 291.83, 80.43 -59.13, -19.56 in-in in 8.8614 Saltbr-in 2.6093 HRD-naA -72.84, -43.49 62.9, 3.06 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.98, 32.2 APE9-dihe-na -91.86, -145.44 APE8-dihe-in -92.13, 124.7 APE8-rot-in 302.73 APE67-dihe-in -76.25, -2.93 -59.68, -41.94 APE12-dist-in 9.6324 APE11-dist-in 8.5086 APE10-dist-in 5.7436 APE9-dist-in 3.771 None None None XRAY 1.92 0.158 0.207 A 328.0 273.0 0 26 26 0 [[38, 290]] 1.0 4alw Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4N6YA P11309 32 305 313.0 2HV:401 Type1 Active DFGin 6.2593 14.8808 BLAminus -123.98, 165.51 60.84, 90.41 -100.85, 18.31 286.86, 79.6 -74.61, -13.5 in-in in 8.7605 Saltbr-in 2.7094 HRD-naA -69.76, -50.01 73.25, 2.39 in-in-in SNCiii in-in ActLoopNT-in 2.9037 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.48, 35.75 APE9-dihe-na -98.87, -155.99 APE8-dihe-in -86.09, 125.72 APE8-rot-in 310.58 APE67-dihe-in -66.86, -9.74 -54.28, -49.47 APE12-dist-in 9.3871 APE11-dist-in 8.4414 APE10-dist-in 5.4013 APE9-dist-in 3.7697 None SEP261 SEP261 XRAY 2.6 0.159 0.212 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 4n6y Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4N6ZA P11309 33 305 313.0 2HW:401 Type1 Active DFGin 6.463 14.6459 BLAminus -126.99, 169.95 59.29, 83.89 -97.92, 18.69 285.67, 67.47 -72.35, -9.24 in-in in 8.2536 Saltbr-in 2.7291 HRD-naA -69.23, -47.57 69.1, 0.1 in-in-in SNCiii in-in ActLoopNT-in 2.9924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.18, 25.75 APE9-dihe-na -86.3, -154.15 APE8-dihe-in -92.66, 118.79 APE8-rot-in 308.24 APE67-dihe-in -66.17, -14.41 -51.57, -45.87 APE12-dist-in 9.4646 APE11-dist-in 8.5132 APE10-dist-in 5.3789 APE9-dist-in 3.6943 None SEP261 SEP261 XRAY 2.2 0.161 0.189 A 328.0 273.0 0 26 26 0 [[38, 290]] 1.0 4n6z Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4N70A P11309 32 306 313.0 2HX:401 Type1 Active DFGin 6.1649 14.5694 BLAminus -137.89, 169.53 64.36, 80.83 -93.88, 21.26 288.11, 67.53 -75.41, -5.31 in-in in 8.6245 Saltbr-in 2.6005 HRD-naA -69.13, -48.86 67.14, 6.63 in-in-in SNCiii in-in ActLoopNT-in 2.8242 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.37, 33.23 APE9-dihe-na -89.84, -146.82 APE8-dihe-in -98.54, 120.46 APE8-rot-in 304.86 APE67-dihe-in -67.47, -8.0 -60.04, -43.4 APE12-dist-in 9.5943 APE11-dist-in 8.6595 APE10-dist-in 5.7234 APE9-dist-in 3.7572 None SEP261 SEP261 XRAY 2.1 0.169 0.208 A 328.0 275.0 0 26 26 0 [[38, 290]] 1.0 4n70 Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5DWRA P11309 33 306 313.0 5H7:401 Type1 Active DFGin 6.2423 14.6643 BLAminus -131.54, 168.2 64.5, 84.97 -98.37, 18.01 285.62, 75.32 -66.32, -15.3 in-in in 8.5476 Saltbr-in 2.6698 HRD-naA -72.01, -47.63 67.32, 6.26 in-in-in SNCiii in-in ActLoopNT-in 2.9583 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.09, 26.57 APE9-dihe-na -84.89, -152.84 APE8-dihe-in -93.58, 121.01 APE8-rot-in 307.85 APE67-dihe-in -68.04, -7.01 -54.84, -45.5 APE12-dist-in 9.522 APE11-dist-in 8.5314 APE10-dist-in 5.4179 APE9-dist-in 3.6508 None SEP261 SEP261 XRAY 2.0 0.175 0.202 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 5dwr Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6YKDA P11309 33 305 313.0 OWB:60400 Type1 Active DFGin 6.1577 14.6899 BLAminus -121.19, 171.99 65.51, 79.7 -90.44, 14.31 281.37, 83.04 -61.46, -20.23 in-in in 8.9313 Saltbr-in 2.6812 HRD-naA -69.86, -48.77 63.9, 14.36 in-in-in SNCiii in-in ActLoopNT-in 2.8682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.12, 24.2 APE9-dihe-na -86.9, -151.63 APE8-dihe-in -93.7, 123.39 APE8-rot-in 303.13 APE67-dihe-in -72.97, -5.5 -60.57, -42.11 APE12-dist-in 9.6038 APE11-dist-in 8.5277 APE10-dist-in 5.4138 APE9-dist-in 3.7385 None SEP261 SEP261 XRAY 1.86 0.16 0.194 A 329.0 273.0 0 26 26 0 [[38, 290]] 1.0 6ykd Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2OBJA P11309 33 305 313.0 VRV:400 Type1 Active DFGin 5.8483 14.3418 BLAminus -135.1, 165.89 65.58, 81.59 -93.29, 20.74 291.15, 68.53 -60.11, -19.32 in-in in 8.6835 Saltbr-in 2.448 HRD-naA -67.98, -46.96 66.7, 2.66 in-in-in SNCiii in-in ActLoopNT-in 2.9077 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.26, 30.91 APE9-dihe-na -92.97, -164.42 APE8-dihe-in -76.75, 121.77 APE8-rot-in 305.59 APE67-dihe-in -61.67, -9.38 -55.68, -49.65 APE12-dist-in 9.4446 APE11-dist-in 8.5058 APE10-dist-in 5.3383 APE9-dist-in 3.7537 None SEP261 SEP261 XRAY 2.5 0.205 0.246 A 333.0 273.0 0 26 26 0 [[38, 290]] 1.0 2obj Homo sapiens CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3BGPA P11309 33 305 313.0 VX1:314 Type1 Active DFGin 5.9426 14.4251 BLAminus -126.41, 157.1 77.54, 91.73 -104.16, 28.82 293.34, 70.26 -65.15, -26.7 in-in in 8.6312 Saltbr-in 2.6289 HRD-naA -72.43, -49.43 73.8, -3.17 in-in-in SNCiii in-in ActLoopNT-in 2.7729 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.31, 13.68 APE9-dihe-na -86.06, -170.88 APE8-dihe-in -67.89, 136.06 APE8-rot-in 304.87 APE67-dihe-in -64.78, -12.46 -73.3, -44.0 APE12-dist-in 9.3655 APE11-dist-in 8.5615 APE10-dist-in 4.9825 APE9-dist-in 3.9275 None SEP261 SEP261 XRAY 2.8 0.213 0.261 A 333.0 273.0 0 26 26 0 [[38, 290]] 1.0 3bgp Homo sapiens CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3BGQA P11309 33 305 313.0 VX2:314 Type1 Active DFGin 6.3949 14.8556 BLAminus -129.22, 172.22 56.92, 80.34 -93.96, 24.94 287.45, 64.49 -68.32, -10.99 in-in in 8.4273 Saltbr-in 2.6592 HRD-naA -70.11, -48.13 67.03, 6.04 in-in-in SNCiii in-in ActLoopNT-in 2.9262 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.69, 26.46 APE9-dihe-na -85.59, -155.16 APE8-dihe-in -92.08, 118.01 APE8-rot-in 308.33 APE67-dihe-in -63.18, -11.49 -49.18, -49.37 APE12-dist-in 9.6074 APE11-dist-in 8.5858 APE10-dist-in 5.4106 APE9-dist-in 3.6395 None SEP261 SEP261 XRAY 2.0 0.213 0.23 A 333.0 273.0 0 26 26 0 [[38, 290]] 1.0 3bgq Homo sapiens CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3BGZA P11309 33 305 313.0 VX3:314 Type1 Active DFGin 6.223 14.5079 BLAminus -126.99, 169.09 64.54, 79.92 -92.02, 15.99 284.89, 75.21 -68.7, -13.09 in-in in 8.7342 Saltbr-in 2.7258 HRD-naA -68.01, -47.53 72.06, 3.12 in-in-in SNCiii in-in ActLoopNT-in 2.8055 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.26, 35.08 APE9-dihe-na -86.26, -142.72 APE8-dihe-in -103.04, 122.93 APE8-rot-in 309.34 APE67-dihe-in -67.64, -10.68 -55.55, -46.74 APE12-dist-in 9.5335 APE11-dist-in 8.6464 APE10-dist-in 5.6709 APE9-dist-in 3.6886 None SEP261 SEP261 XRAY 2.4 0.196 0.233 A 333.0 268.0 5 26 26 0 [[38, 290]] 1.0 3bgz Homo sapiens CAMK_PIM1_HUMAN CAMK 4.9e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3WE8A P11309 33 305 313.0 RUI:401 Type1 Active DFGin 6.0765 14.5621 BLAminus -133.3, 170.64 67.13, 73.63 -87.77, 10.99 287.95, 77.91 -66.1, -8.31 in-in in 8.9805 Saltbr-in 2.6432 HRD-naA -75.68, -43.45 65.63, 6.85 in-in-in SNCiii in-in ActLoopNT-in 2.8418 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.96, 25.34 APE9-dihe-na -83.21, -158.59 APE8-dihe-in -86.86, 122.45 APE8-rot-in 300.85 APE67-dihe-in -73.76, -3.38 -61.05, -39.9 APE12-dist-in 9.8003 APE11-dist-in 8.6353 APE10-dist-in 5.6029 APE9-dist-in 3.7476 R250G None None XRAY 1.954 0.16 0.177 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 3we8 Homo sapiens CAMK_PIM1_HUMAN CAMK 9.2e-65 224.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4AS0A P11309 33 305 313.0 RPS:1306 Type1 Active DFGin 6.2392 14.7972 BLAminus -125.08, 170.08 63.9, 84.56 -93.79, 23.62 287.71, 77.4 -74.79, -13.31 in-in in 8.9969 Saltbr-in 2.4858 HRD-naA -73.68, -44.47 70.76, -1.79 in-in-in SNCiii in-in ActLoopNT-in 2.8952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.05, 33.62 APE9-dihe-na -96.04, -155.25 APE8-dihe-in -91.93, 124.92 APE8-rot-in 312.41 APE67-dihe-in -67.91, -14.18 -64.04, -41.51 APE12-dist-in 9.5865 APE11-dist-in 8.5215 APE10-dist-in 5.3972 APE9-dist-in 4.1789 None None None XRAY 2.3 0.172 0.201 A 273.0 273.0 0 26 26 0 [[38, 290]] 1.0 4as0 Homo sapiens CAMK_PIM1_HUMAN CAMK 9.2e-65 224.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5TURA P11309 34 306 313.0 7LK:401 Type1 Active DFGin 6.061 14.49 BLAminus -136.79, 174.59 58.79, 85.71 -98.08, 24.51 288.61, 83.41 -77.7, -2.74 in-in in 8.7582 Saltbr-in 2.6156 HRD-naA -76.1, -44.31 69.09, 5.73 in-in-in SNCiii in-in ActLoopNT-in 2.7428 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.99, 42.91 APE9-dihe-na -110.95, -154.07 APE8-dihe-in -91.19, 125.87 APE8-rot-in 304.26 APE67-dihe-in -69.95, -16.95 -69.94, -33.83 APE12-dist-in 9.7357 APE11-dist-in 8.7982 APE10-dist-in 5.3539 APE9-dist-in 3.9645 None None None XRAY 2.948 0.209 0.248 A 404.0 270.0 3 26 26 0 [[38, 290]] 1.0 5tur Homo sapiens CAMK_PIM1_HUMAN CAMK 8.9e-65 224.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2J2IB P11309 33 305 313.0 LY4:1307 Type1 Active DFGin 6.3491 14.7879 BLAminus -124.69, 164.2 69.56, 81.11 -88.57, 16.71 287.44, 78.04 -63.89, -22.24 in-in in 8.7154 Saltbr-in 2.8844 HRD-naA -68.27, -48.73 73.43, 1.94 in-in-in SNCiii in-in ActLoopNT-in 2.8048 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.68, 17.7 APE9-dihe-na -79.18, -163.88 APE8-dihe-in -85.23, 122.14 APE8-rot-in 304.09 APE67-dihe-in -70.03, -11.09 -55.65, -47.61 APE12-dist-in 9.3137 APE11-dist-in 8.7009 APE10-dist-in 5.4569 APE9-dist-in 3.9641 R250G None None XRAY 1.9 0.18 0.2 B 312.0 273.0 0 26 26 0 [[38, 290]] 1.0 2j2i Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7QB2A P11309 33 305 313.0 A7X:402 Type1 Active DFGin 6.2608 14.4336 BLAminus -125.87, 176.63 53.43, 82.5 -86.6, 20.72 284.17, 73.36 -70.8, -10.08 in-in in 8.6566 Saltbr-in 2.6079 HRD-naA -76.36, -48.43 70.95, 3.72 in-in-in SNCiii in-in ActLoopNT-in 2.6919 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.34, 22.15 APE9-dihe-na -86.92, -149.81 APE8-dihe-in -97.03, 122.97 APE8-rot-in 300.26 APE67-dihe-in -69.31, -7.68 -64.45, -41.13 APE12-dist-in 9.9263 APE11-dist-in 8.6524 APE10-dist-in 4.9748 APE9-dist-in 3.7444 R250G SEP261 SEP261 XRAY 2.53 0.159 0.202 A 312.0 273.0 0 26 26 0 [[38, 290]] 1.0 7qb2 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7QFMA P11309 33 305 313.0 AY3:402 Type1 Active DFGin 6.2031 14.458 BLAminus -124.14, 177.11 57.14, 79.43 -85.98, 19.87 284.85, 75.66 -69.01, -15.13 in-in in 8.7647 Saltbr-in 2.6921 HRD-naA -73.09, -45.9 66.81, 9.42 in-in-in SNCiii in-in ActLoopNT-in 2.846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 26.43 APE9-dihe-na -81.47, -151.25 APE8-dihe-in -97.97, 122.34 APE8-rot-in 302.11 APE67-dihe-in -71.87, -9.27 -61.74, -39.67 APE12-dist-in 9.9106 APE11-dist-in 8.6095 APE10-dist-in 5.3753 APE9-dist-in 3.6137 R250G SEP261 SEP261 XRAY 1.95 0.159 0.178 A 312.0 271.0 2 26 26 0 [[38, 290]] 1.0 7qfm Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.8 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3JPVA P11309 33 305 313.0 1DR:313 Type1 Active DFGin 6.1479 14.441 BLAminus -120.08, 164.67 68.13, 86.84 -92.5, 13.59 289.99, 74.69 -67.43, -13.65 in-in in 9.0034 Saltbr-in 2.5634 HRD-naA -72.55, -46.96 72.58, 4.93 in-in-in SNCiii in-in ActLoopNT-in 2.8888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.51, 21.98 APE9-dihe-na -83.62, -150.17 APE8-dihe-in -98.9, 116.73 APE8-rot-in 306.83 APE67-dihe-in -67.26, -10.5 -54.29, -42.64 APE12-dist-in 9.8235 APE11-dist-in 8.4389 APE10-dist-in 5.4133 APE9-dist-in 3.7639 None None None XRAY 2.35 0.176 0.226 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 3jpv Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3MA3A P11309 37 305 313.0 01I:313 Type1 Active DFGin 6.0181 14.2367 BLAminus -126.51, 170.48 60.71, 85.71 -91.62, 21.05 288.87, 82.52 -71.65, -14.95 in-in in 8.9174 Saltbr-in 2.6909 HRD-naA -71.5, -42.79 64.42, 10.83 in-in-in SNCiii in-in ActLoopNT-in 2.754 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.06, 17.84 APE9-dihe-na -81.84, -163.49 APE8-dihe-in -85.13, 123.05 APE8-rot-in 304.03 APE67-dihe-in -65.07, -11.91 -66.26, -41.53 APE12-dist-in 9.8117 APE11-dist-in 8.4025 APE10-dist-in 5.2207 APE9-dist-in 3.8789 None SEP261 SEP261 XRAY 2.3 0.172 0.233 A 313.0 267.0 2 26 26 0 [[38, 290]] 1.0 3ma3 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3QF9A P11309 32 305 313.0 NM8:313 Type1 Active DFGin 6.0701 14.424 BLAminus -120.87, 169.05 67.22, 78.8 -88.89, 16.3 288.42, 76.0 -67.55, -12.21 in-in in 8.8485 Saltbr-in 2.5791 HRD-naA -70.76, -46.92 73.96, 4.53 in-in-in SNCiii in-in ActLoopNT-in 2.8907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.62, 24.45 APE9-dihe-na -83.53, -155.23 APE8-dihe-in -93.29, 124.33 APE8-rot-in 299.27 APE67-dihe-in -72.17, -10.84 -63.75, -37.33 APE12-dist-in 9.804 APE11-dist-in 8.4801 APE10-dist-in 5.3666 APE9-dist-in 3.6712 R250G None None XRAY 2.2 0.188 0.227 A 313.0 274.0 0 26 26 0 [[38, 290]] 1.0 3qf9 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4GW8A P11309 33 305 313.0 3RA:401 Type1 Active DFGin 6.2361 14.6142 BLAminus -126.36, 165.58 62.03, 83.71 -89.36, 16.13 285.86, 76.28 -67.97, -17.62 in-in in 8.7369 Saltbr-in 2.7149 HRD-naA -74.23, -46.85 73.75, 9.79 in-in-in SNCiii in-in ActLoopNT-in 2.8877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.85, 8.01 APE9-dihe-na -80.24, -160.25 APE8-dihe-in -87.85, 121.5 APE8-rot-in 304.03 APE67-dihe-in -71.21, -12.4 -59.35, -38.89 APE12-dist-in 9.4824 APE11-dist-in 8.2992 APE10-dist-in 4.4436 APE9-dist-in 3.7427 R250G None None XRAY 2.0 0.178 0.213 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 4gw8 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6PCWA P11309 32 305 313.0 O97:500 Type1 Active DFGin 6.1281 14.5651 BLAminus -128.69, 170.24 60.89, 83.86 -89.77, 15.97 285.56, 79.53 -66.69, -14.24 in-in in 8.7913 Saltbr-in 2.6314 HRD-naA -73.35, -47.8 66.65, 11.24 in-in-in SNCiii in-in ActLoopNT-in 2.8121 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.44, 8.45 APE9-dihe-na -84.75, -155.07 APE8-dihe-in -92.6, 123.69 APE8-rot-in 306.23 APE67-dihe-in -72.6, -7.76 -62.22, -39.85 APE12-dist-in 9.4745 APE11-dist-in 8.4917 APE10-dist-in 4.5618 APE9-dist-in 3.6262 None None None XRAY 2.2 0.177 0.226 A 313.0 273.0 1 26 26 0 [[38, 290]] 1.0 6pcw Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6PDIA P11309 32 305 313.0 OCJ:501 Type1 Active DFGin 6.1283 14.4792 BLAminus -126.87, 170.77 61.93, 81.48 -89.41, 13.26 285.32, 82.24 -64.21, -18.32 in-in in 8.8112 Saltbr-in 2.6199 HRD-naA -69.88, -49.72 68.62, 9.34 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.35, 18.43 APE9-dihe-na -84.8, -157.57 APE8-dihe-in -92.5, 120.51 APE8-rot-in 302.8 APE67-dihe-in -73.34, -11.57 -60.21, -38.03 APE12-dist-in 9.5818 APE11-dist-in 8.3694 APE10-dist-in 4.9704 APE9-dist-in 3.6699 None None None XRAY 1.85 0.163 0.193 A 313.0 274.0 0 26 26 0 [[38, 290]] 1.0 6pdi Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6PDNA P11309 32 305 313.0 OD4:900 Type1 Active DFGin 6.303 14.6787 BLAminus -127.91, 168.34 63.69, 84.1 -90.47, 15.7 284.14, 84.0 -75.26, -13.52 in-in in 8.8267 Saltbr-in 2.587 HRD-naA -70.55, -51.59 71.07, 6.03 in-in-in SNCiii in-in ActLoopNT-in 2.792 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.78, 23.66 APE9-dihe-na -88.42, -164.96 APE8-dihe-in -87.14, 123.03 APE8-rot-in 304.39 APE67-dihe-in -74.69, -11.36 -61.92, -39.09 APE12-dist-in 9.5899 APE11-dist-in 8.4061 APE10-dist-in 5.0533 APE9-dist-in 3.7386 None SEP261 SEP261 XRAY 2.4 0.19 0.223 A 313.0 270.0 4 26 26 0 [[38, 290]] 1.0 6pdn Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6PDOA P11309 35 305 313.0 OD1:501 Type1 Active DFGin 6.1292 14.2926 BLAminus -134.81, 169.87 61.89, 85.2 -91.49, 10.5 286.61, 82.45 -62.88, -17.93 in-in in 8.5877 Saltbr-in 2.7516 HRD-naA -69.22, -51.16 69.51, 6.24 in-in-in SNCiii in-in ActLoopNT-in 2.7835 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -122.34, 22.85 APE9-dihe-na -86.44, -166.55 APE8-dihe-in -83.99, 120.38 APE8-rot-in 303.74 APE67-dihe-in -70.14, -12.44 -58.32, -42.49 APE12-dist-in 9.5734 APE11-dist-in 8.3618 APE10-dist-in 4.7473 APE9-dist-in 3.7884 None None None XRAY 2.4 0.177 0.223 A 313.0 267.0 4 26 26 0 [[38, 290]] 1.0 6pdo Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6PDPA P11309 36 305 313.0 OBY:502 Type1 Active DFGin 6.1497 14.2213 BLAminus -129.84, 173.21 59.86, 93.48 -102.79, 22.43 282.95, 82.01 -70.26, -12.41 in-in in 8.422 Saltbr-in 2.7863 HRD-naA -67.94, -55.57 82.45, -11.52 in-in-in SNCiii in-in ActLoopNT-in 2.8844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.22, 34.63 APE9-dihe-na -88.55, -154.18 APE8-dihe-in -92.87, 123.61 APE8-rot-in 300.67 APE67-dihe-in -66.54, -13.53 -62.56, -42.85 APE12-dist-in 9.7024 APE11-dist-in 8.577 APE10-dist-in 5.7129 APE9-dist-in 4.1106 None None None XRAY 2.5 0.195 0.23 A 313.0 268.0 2 26 26 0 [[38, 290]] 1.0 6pdp Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6QXKB P11309 35 305 313.0 JKW:401 Type1 Active DFGin 6.1014 14.6091 BLAminus -124.57, 170.74 63.53, 81.45 -86.73, 15.75 286.17, 80.26 -64.12, -13.74 in-in in 8.945 Saltbr-in 2.6481 HRD-naA -69.55, -43.65 65.58, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.8414 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.01, 26.44 APE9-dihe-na -78.6, -156.19 APE8-dihe-in -94.84, 121.84 APE8-rot-in 303.08 APE67-dihe-in -71.43, -12.21 -59.33, -38.29 APE12-dist-in 9.8192 APE11-dist-in 8.4888 APE10-dist-in 5.4191 APE9-dist-in 3.6144 None None None XRAY 2.1 0.177 0.201 B 313.0 269.0 2 26 26 0 [[38, 290]] 1.0 6qxk Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R0HA P11309 33 305 313.0 8UB:403 Type1 Active DFGin 6.1948 14.5044 BLAminus -130.64, 169.15 64.03, 75.42 -86.88, 14.36 285.23, 74.81 -64.53, -17.19 in-in in 8.7633 Saltbr-in 2.7368 HRD-naA -71.57, -46.79 68.26, 11.15 in-in-in SNCiii in-in ActLoopNT-in 2.836 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.99, 20.76 APE9-dihe-na -80.37, -156.78 APE8-dihe-in -90.68, 121.72 APE8-rot-in 301.93 APE67-dihe-in -72.4, -8.98 -63.85, -37.03 APE12-dist-in 9.5338 APE11-dist-in 8.4986 APE10-dist-in 5.275 APE9-dist-in 3.6981 R250G SEP261 SEP261 XRAY 1.88 0.155 0.174 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r0h Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R0QA P11309 33 305 313.0 XGB:402 Type1 Active DFGin 6.1107 14.4727 BLAminus -124.88, 175.93 64.13, 67.05 -83.42, 11.36 282.83, 73.71 -70.16, -12.5 in-in in 8.8722 Saltbr-in 2.6597 HRD-naA -75.58, -44.16 66.56, 9.98 in-in-in SNCiii in-in ActLoopNT-in 2.8238 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.86, 18.75 APE9-dihe-na -80.22, -154.78 APE8-dihe-in -92.21, 122.35 APE8-rot-in 302.64 APE67-dihe-in -70.96, -8.32 -63.59, -38.0 APE12-dist-in 9.7252 APE11-dist-in 8.5877 APE10-dist-in 5.3973 APE9-dist-in 3.7047 R250G SEP261 SEP261 XRAY 1.7 0.166 0.177 A 313.0 267.0 6 26 26 0 [[38, 290]] 1.0 8r0q Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R0WA P11309 33 305 313.0 XGF:405 Type1 Active DFGin 5.9965 14.3841 BLAminus -131.73, 166.77 65.97, 82.46 -89.79, 16.41 289.35, 79.56 -63.02, -16.4 in-in in 8.8117 Saltbr-in 2.6426 HRD-naA -73.15, -45.35 65.43, 10.88 in-in-in SNCiii in-in ActLoopNT-in 2.8554 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.23, 17.26 APE9-dihe-na -81.93, -156.28 APE8-dihe-in -91.39, 121.88 APE8-rot-in 296.84 APE67-dihe-in -71.92, -8.94 -64.52, -38.27 APE12-dist-in 9.5591 APE11-dist-in 8.4794 APE10-dist-in 5.1163 APE9-dist-in 3.7129 R250G SEP261 SEP261 XRAY 1.95 0.167 0.201 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r0w Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R0YA P11309 33 305 313.0 XH3:402 Type1 Active DFGin 6.1278 14.5374 BLAminus -126.73, 169.7 64.58, 82.54 -91.76, 17.79 287.7, 78.06 -67.67, -13.51 in-in in 8.9569 Saltbr-in 2.6397 HRD-naA -71.78, -46.47 66.88, 6.9 in-in-in SNCiii in-in ActLoopNT-in 2.8623 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.85, 18.81 APE9-dihe-na -78.72, -154.37 APE8-dihe-in -95.58, 121.63 APE8-rot-in 303.84 APE67-dihe-in -73.42, -9.78 -59.84, -39.22 APE12-dist-in 9.539 APE11-dist-in 8.5542 APE10-dist-in 5.1289 APE9-dist-in 3.718 R250G SEP261 SEP261 XRAY 2.05 0.176 0.19 A 313.0 271.0 2 26 26 0 [[38, 290]] 1.0 8r0y Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R10A P11309 33 305 313.0 XGQ:401 Type1 Active DFGin 6.0079 14.5901 BLAminus -125.35, 178.02 53.25, 82.24 -86.16, 17.78 284.81, 76.38 -68.05, -10.88 in-in in 8.8956 Saltbr-in 2.6351 HRD-naA -73.59, -46.61 66.3, 8.94 in-in-in SNCiii in-in ActLoopNT-in 2.8079 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.14, 17.84 APE9-dihe-na -81.41, -153.47 APE8-dihe-in -91.91, 123.95 APE8-rot-in 303.23 APE67-dihe-in -72.41, -8.02 -63.66, -38.07 APE12-dist-in 9.9235 APE11-dist-in 8.4791 APE10-dist-in 5.2127 APE9-dist-in 3.6321 R250G SEP261 SEP261 XRAY 2.2 0.171 0.202 A 313.0 263.0 10 26 26 0 [[38, 290]] 1.0 8r10 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R18A P11309 33 305 313.0 XGK:402 Type1 Active DFGin 6.0344 14.3517 BLAminus -124.11, 175.65 61.57, 82.15 -90.26, 19.65 285.44, 75.92 -71.89, -10.87 in-in in 8.8263 Saltbr-in 2.5902 HRD-naA -75.08, -45.72 63.91, 12.1 in-in-in SNCiii in-in ActLoopNT-in 2.8326 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.79, 24.66 APE9-dihe-na -82.08, -152.26 APE8-dihe-in -93.08, 122.4 APE8-rot-in 301.75 APE67-dihe-in -73.31, -7.85 -63.76, -37.55 APE12-dist-in 9.8399 APE11-dist-in 8.5947 APE10-dist-in 5.5183 APE9-dist-in 3.68 R250G SEP261 SEP261 XRAY 1.89 0.161 0.186 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r18 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R1KA P11309 33 305 313.0 XHI:403 Type1 Active DFGin 6.2459 14.5708 BLAminus -130.32, 173.36 62.94, 72.15 -85.85, 16.37 285.53, 75.29 -71.64, -12.67 in-in in 8.7619 Saltbr-in 2.5021 HRD-naA -71.16, -48.89 70.04, 11.26 in-in-in SNCiii in-in ActLoopNT-in 2.8665 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.08, 4.88 APE9-dihe-na -84.34, -155.09 APE8-dihe-in -91.8, 121.7 APE8-rot-in 300.68 APE67-dihe-in -73.09, -10.26 -62.22, -37.87 APE12-dist-in 9.5411 APE11-dist-in 8.5475 APE10-dist-in 4.4357 APE9-dist-in 3.6882 R250G SEP261 SEP261 XRAY 1.95 0.177 0.192 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r1k Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R1NA P11309 34 305 313.0 XIT:401 Type1 Active DFGin 6.0573 14.5468 BLAminus -128.21, 174.49 58.15, 82.23 -87.85, 19.59 286.58, 72.67 -72.06, -10.27 in-in in 8.9084 Saltbr-in 2.7552 HRD-naA -72.06, -45.87 66.94, 8.6 in-in-in SNCiii in-in ActLoopNT-in 2.7691 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.59, 26.14 APE9-dihe-na -82.46, -153.43 APE8-dihe-in -96.65, 123.51 APE8-rot-in 298.16 APE67-dihe-in -70.63, -8.19 -63.53, -39.8 APE12-dist-in 9.783 APE11-dist-in 8.6205 APE10-dist-in 5.2058 APE9-dist-in 3.5907 R250G SEP261 SEP261 XRAY 2.21 0.163 0.192 A 313.0 272.0 0 26 26 0 [[38, 290]] 1.0 8r1n Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R1PA P11309 33 305 313.0 XIP:401 Type1 Active DFGin 6.0662 14.6184 BLAminus -128.97, 176.78 55.64, 82.37 -89.27, 14.78 284.77, 74.77 -64.96, -11.11 in-in in 8.8719 Saltbr-in 2.5719 HRD-naA -73.78, -46.66 71.64, 3.78 in-in-in SNCiii in-in ActLoopNT-in 2.8165 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.36, 22.63 APE9-dihe-na -86.45, -148.42 APE8-dihe-in -100.33, 122.66 APE8-rot-in 304.21 APE67-dihe-in -71.49, -6.91 -61.13, -41.84 APE12-dist-in 9.7904 APE11-dist-in 8.549 APE10-dist-in 4.924 APE9-dist-in 3.7558 R250G SEP261 SEP261 XRAY 2.45 0.178 0.206 A 313.0 269.0 4 26 26 0 [[38, 290]] 1.0 8r1p Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R1TA P11309 33 305 313.0 XIJ:402 Type1 Active DFGin 6.1286 14.5004 BLAminus -125.46, 175.2 59.64, 82.38 -89.86, 18.41 286.56, 77.1 -71.67, -11.65 in-in in 8.8527 Saltbr-in 2.6881 HRD-naA -72.26, -44.66 65.09, 8.72 in-in-in SNCiii in-in ActLoopNT-in 2.792 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.98, 13.92 APE9-dihe-na -81.53, -153.62 APE8-dihe-in -94.64, 124.09 APE8-rot-in 299.63 APE67-dihe-in -71.25, -8.49 -63.99, -39.26 APE12-dist-in 9.7963 APE11-dist-in 8.6337 APE10-dist-in 4.9525 APE9-dist-in 3.6603 R250G SEP261 SEP261 XRAY 2.0 0.16 0.179 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r1t Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R1WA P11309 33 305 313.0 XIW:402 Type1 Active DFGin 6.0093 14.6266 BLAminus -126.26, 175.45 55.83, 87.17 -92.67, 17.42 288.58, 76.06 -64.09, -13.07 in-in in 9.0119 Saltbr-in 2.6417 HRD-naA -70.36, -47.52 67.35, 8.76 in-in-in SNCiii in-in ActLoopNT-in 2.7892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.05, 16.58 APE9-dihe-na -79.71, -155.45 APE8-dihe-in -91.51, 124.54 APE8-rot-in 299.68 APE67-dihe-in -71.95, -9.45 -64.13, -40.15 APE12-dist-in 9.7391 APE11-dist-in 8.5662 APE10-dist-in 5.1338 APE9-dist-in 3.6453 R250G SEP261 SEP261 XRAY 2.15 0.176 0.204 A 313.0 270.0 3 26 26 0 [[38, 290]] 1.0 8r1w Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R25A P11309 33 305 313.0 XJL:402 Type1 Active DFGin 6.2238 14.6031 BLAminus -130.14, 174.3 56.41, 81.8 -90.04, 19.15 286.56, 75.38 -70.08, -10.25 in-in in 9.0651 Saltbr-in 2.4738 HRD-naA -71.77, -46.38 67.37, 8.2 in-in-in SNCiii in-in ActLoopNT-in 2.8145 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.33, 17.96 APE9-dihe-na -81.3, -151.78 APE8-dihe-in -98.77, 123.36 APE8-rot-in 301.63 APE67-dihe-in -70.17, -10.17 -64.54, -39.25 APE12-dist-in 9.6803 APE11-dist-in 8.6865 APE10-dist-in 4.9632 APE9-dist-in 3.6548 R250G SEP261 SEP261 XRAY 2.1 0.178 0.208 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 8r25 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8R27A P11309 33 305 313.0 XJW:402 Type1 Active DFGin 6.0133 14.3845 BLAminus -125.88, 174.13 60.12, 79.82 -86.61, 17.63 284.74, 75.1 -73.25, -8.78 in-in in 8.8799 Saltbr-in 2.7031 HRD-naA -74.94, -45.68 65.39, 9.33 in-in-in SNCiii in-in ActLoopNT-in 2.8424 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.2, 23.86 APE9-dihe-na -82.24, -153.87 APE8-dihe-in -93.36, 121.12 APE8-rot-in 300.79 APE67-dihe-in -70.77, -7.65 -61.34, -41.5 APE12-dist-in 9.7823 APE11-dist-in 8.5259 APE10-dist-in 5.2562 APE9-dist-in 3.6976 R250G SEP261 SEP261 XRAY 1.95 0.166 0.192 A 313.0 272.0 1 26 26 0 [[38, 290]] 1.0 8r27 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2BIKB P11309 33 305 313.0 BI1:1306 Type1 Active DFGin 6.2085 14.8544 BLAminus -129.68, 166.2 65.31, 82.3 -90.49, 20.51 284.24, 80.72 -71.93, -11.81 in-in in 8.7316 Saltbr-in 2.7718 HRD-naA -71.08, -48.28 72.24, 3.48 in-in-in SNCiii in-in ActLoopNT-in 2.8318 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.84, 26.95 APE9-dihe-na -83.77, -163.0 APE8-dihe-in -86.27, 123.71 APE8-rot-in 311.31 APE67-dihe-in -70.32, -9.34 -58.19, -44.58 APE12-dist-in 9.5525 APE11-dist-in 8.6863 APE10-dist-in 5.6274 APE9-dist-in 3.928 None SEP261 SEP261 XRAY 1.8 0.159 0.183 B 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 2bik Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2BILB P11309 33 306 313.0 BI1:1307 Type1 Active DFGin 5.907 14.6412 BLAminus -131.58, 166.0 69.48, 82.95 -91.3, 19.54 286.18, 78.18 -74.97, -10.91 in-in in 8.7854 Saltbr-in 2.6353 HRD-naA -70.92, -50.11 73.56, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.8565 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.49, 48.23 APE9-dihe-na -87.89, -146.11 APE8-dihe-in -91.43, 121.08 APE8-rot-in 306.95 APE67-dihe-in -71.1, -13.65 -55.02, -40.77 APE12-dist-in 9.4619 APE11-dist-in 8.2518 APE10-dist-in 6.34 APE9-dist-in 3.8583 None None None XRAY 2.55 0.195 0.248 B 313.0 274.0 0 26 26 0 [[38, 290]] 1.0 2bil Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2BZHB P11309 32 306 313.0 HB1:1307 Type1 Active DFGin 6.241 14.7174 BLAminus -128.91, 169.67 62.16, 81.6 -86.25, 13.92 287.87, 80.39 -66.46, -13.69 in-in in 8.8333 Saltbr-in 2.7881 HRD-naA -70.2, -46.33 68.04, 6.62 in-in-in SNCiii in-in ActLoopNT-in 2.86 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.94, 27.94 APE9-dihe-na -80.38, -157.42 APE8-dihe-in -90.55, 119.15 APE8-rot-in 302.06 APE67-dihe-in -68.66, -8.15 -56.91, -42.45 APE12-dist-in 9.5819 APE11-dist-in 8.5307 APE10-dist-in 5.5946 APE9-dist-in 3.6731 R250G None None XRAY 1.9 0.159 0.19 B 313.0 275.0 0 26 26 0 [[38, 290]] 1.0 2bzh Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2BZIB P11309 33 305 313.0 DW2:1306 Type1 Active DFGin 6.2667 14.8353 BLAminus -123.34, 165.34 66.36, 86.11 -93.21, 22.23 286.33, 78.94 -70.39, -16.59 in-in in 8.8727 Saltbr-in 2.7797 HRD-naA -72.04, -45.2 68.6, 5.31 in-in-in SNCiii in-in ActLoopNT-in 2.857 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.77, 39.69 APE9-dihe-na -92.21, -159.18 APE8-dihe-in -82.89, 124.01 APE8-rot-in 305.62 APE67-dihe-in -65.59, -13.31 -61.02, -47.85 APE12-dist-in 9.4556 APE11-dist-in 8.486 APE10-dist-in 5.6923 APE9-dist-in 3.9382 R250G SEP261 SEP261 XRAY 1.9 0.218 0.265 B 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 2bzi Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2BZJA P11309 33 305 313.0 ME3:1306 Type1 Active DFGin 6.2938 14.8461 BLAminus -129.09, 166.61 64.15, 83.62 -93.36, 13.13 283.19, 80.4 -68.93, -14.93 in-in in 8.9144 Saltbr-in 2.5247 HRD-naA -66.52, -47.22 65.13, 9.09 in-in-in SNCiii in-in ActLoopNT-in 2.7732 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -114.4, 32.87 APE9-dihe-na -91.23, -169.99 APE8-dihe-in -72.16, 120.4 APE8-rot-in 307.22 APE67-dihe-in -77.22, -2.13 -52.79, -48.09 APE12-dist-in 9.3195 APE11-dist-in 8.7496 APE10-dist-in 5.5282 APE9-dist-in 3.9837 R250G None None XRAY 2.05 0.185 0.221 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 2bzj Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2C3IB P11309 37 305 313.0 IYZ:1306 Type1 Active DFGin 6.3264 14.7526 BLAminus -127.31, 169.9 65.35, 81.96 -93.82, 15.98 286.0, 76.19 -64.86, -18.96 in-in in 8.5925 Saltbr-in 2.708 HRD-naA -73.6, -47.48 67.75, 10.67 in-in-in SNCiii in-in ActLoopNT-in 2.9203 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.67, 24.77 APE9-dihe-na -79.26, -156.38 APE8-dihe-in -92.5, 121.61 APE8-rot-in 301.77 APE67-dihe-in -67.73, -10.57 -57.93, -41.83 APE12-dist-in 9.5195 APE11-dist-in 8.5652 APE10-dist-in 5.3265 APE9-dist-in 3.7771 R250G None None XRAY 1.9 0.187 0.219 B 313.0 266.0 3 26 26 0 [[38, 290]] 1.0 2c3i Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 2OI4X P11309 32 306 313.0 JM1:1000 Type1 Active DFGin 6.3452 14.8125 BLAminus -127.98, 160.81 73.35, 71.74 -86.12, 11.96 287.24, 83.24 -76.7, -11.05 in-in in 9.0524 Saltbr-in 2.725 HRD-naA -64.97, -46.27 67.59, 4.83 in-in-in SNCiii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.16, 42.39 APE9-dihe-na -92.81, -143.09 APE8-dihe-in -99.99, 118.85 APE8-rot-in 297.17 APE67-dihe-in -72.38, -14.41 -46.73, -45.08 APE12-dist-in 9.4593 APE11-dist-in 8.8662 APE10-dist-in 5.9919 APE9-dist-in 3.671 R250G None None XRAY 2.2 0.192 0.244 X 313.0 275.0 0 26 26 0 [[38, 290]] 1.0 2oi4 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3BWFA P11309 33 305 313.0 DWC:315 Type1 Active DFGin 6.1521 14.7614 BLAminus -130.15, 160.75 70.46, 85.62 -95.56, 18.11 287.26, 79.6 -68.63, -18.22 in-in in 9.0395 Saltbr-in 2.6434 HRD-naA -63.89, -51.3 70.35, 5.77 in-in-in SNCiii in-in ActLoopNT-in 2.7913 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.65, 13.48 APE9-dihe-na -90.68, -158.0 APE8-dihe-in -83.6, 122.9 APE8-rot-in 307.99 APE67-dihe-in -60.33, -14.69 -56.04, -57.34 APE12-dist-in 9.2482 APE11-dist-in 8.6585 APE10-dist-in 5.0955 APE9-dist-in 3.9038 R250G None None XRAY 2.35 0.171 0.225 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 3bwf Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5MZLA P11309 33 305 313.0 8ET:401 Type1 Active DFGin 6.0702 14.4143 BLAminus -131.62, 169.01 61.49, 83.12 -91.63, 17.39 285.49, 78.9 -67.71, -14.16 in-in in 8.7664 Saltbr-in 2.5894 HRD-naA -71.92, -48.75 69.25, 10.18 in-in-in SNCiii in-in ActLoopNT-in 2.7988 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.79, 22.06 APE9-dihe-na -80.91, -155.94 APE8-dihe-in -90.97, 120.03 APE8-rot-in 302.78 APE67-dihe-in -70.3, -10.66 -61.44, -39.24 APE12-dist-in 9.7338 APE11-dist-in 8.5092 APE10-dist-in 5.304 APE9-dist-in 3.6957 R250G None None XRAY 1.955 0.158 0.183 A 313.0 269.0 4 26 26 0 [[38, 290]] 1.0 5mzl Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4NA P11309 33 305 313.0 8M8:401 Type1 Active DFGin 6.1249 14.6169 BLAminus -129.29, 170.82 62.47, 79.55 -88.93, 16.9 284.33, 80.08 -68.56, -10.77 in-in in 8.9316 Saltbr-in 2.5396 HRD-naA -74.48, -44.52 65.43, 11.21 in-in-in SNCiii in-in ActLoopNT-in 2.7939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.35, 17.93 APE9-dihe-na -79.41, -153.04 APE8-dihe-in -96.16, 122.12 APE8-rot-in 301.83 APE67-dihe-in -69.32, -12.36 -62.25, -40.05 APE12-dist-in 9.5995 APE11-dist-in 8.5712 APE10-dist-in 5.2029 APE9-dist-in 3.7045 R250G None None XRAY 2.09 0.161 0.188 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4n Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4OA P11309 33 305 313.0 8MB:401 Type1 Active DFGin 6.0998 14.6005 BLAminus -128.07, 170.32 63.44, 81.51 -90.0, 20.39 288.36, 74.25 -70.54, -10.71 in-in in 8.8244 Saltbr-in 2.5204 HRD-naA -74.44, -43.81 65.23, 5.78 in-in-in SNCiii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.86, 22.33 APE9-dihe-na -84.24, -148.33 APE8-dihe-in -98.01, 118.97 APE8-rot-in 304.06 APE67-dihe-in -72.76, -7.0 -59.82, -38.64 APE12-dist-in 9.676 APE11-dist-in 8.6398 APE10-dist-in 5.1918 APE9-dist-in 3.7491 R250G None None XRAY 2.22 0.182 0.196 A 313.0 271.0 2 26 26 0 [[38, 290]] 1.0 5n4o Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4RA P11309 33 305 313.0 8MQ:402 Type1 Active DFGin 6.1615 14.6842 BLAminus -127.95, 172.44 62.9, 73.52 -86.51, 10.58 283.66, 75.96 -65.07, -11.8 in-in in 8.8652 Saltbr-in 2.7964 HRD-naA -74.57, -43.89 66.05, 7.98 in-in-in SNCiii in-in ActLoopNT-in 2.8278 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.44, 14.9 APE9-dihe-na -80.8, -159.32 APE8-dihe-in -87.99, 122.23 APE8-rot-in 303.81 APE67-dihe-in -72.42, -8.25 -61.99, -38.57 APE12-dist-in 9.6804 APE11-dist-in 8.5666 APE10-dist-in 5.225 APE9-dist-in 3.6808 R250G None None XRAY 2.13 0.162 0.193 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4r Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4UA P11309 34 305 313.0 8MZ:401 Type1 Active DFGin 6.1707 14.6229 BLAminus -127.06, 173.77 59.59, 86.28 -91.8, 19.55 284.63, 76.39 -67.81, -14.94 in-in in 8.939 Saltbr-in 2.6625 HRD-naA -76.79, -43.95 67.64, 10.17 in-in-in SNCiii in-in ActLoopNT-in 2.7659 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.95, 11.58 APE9-dihe-na -74.78, -161.25 APE8-dihe-in -87.42, 123.39 APE8-rot-in 302.63 APE67-dihe-in -68.48, -11.24 -64.0, -41.0 APE12-dist-in 9.5659 APE11-dist-in 8.4312 APE10-dist-in 5.1177 APE9-dist-in 3.6356 R250G None None XRAY 2.202 0.165 0.198 A 313.0 272.0 0 26 26 0 [[38, 290]] 1.0 5n4u Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4VA P11309 33 305 313.0 8MW:401 Type1 Active DFGin 6.1863 14.5848 BLAminus -124.08, 176.44 56.8, 80.25 -87.01, 16.92 283.21, 72.16 -68.4, -12.83 in-in in 8.8997 Saltbr-in 2.6276 HRD-naA -74.68, -46.5 67.92, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.8775 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.8, 18.81 APE9-dihe-na -79.43, -156.57 APE8-dihe-in -90.82, 123.02 APE8-rot-in 301.39 APE67-dihe-in -72.01, -7.09 -64.55, -37.95 APE12-dist-in 9.8641 APE11-dist-in 8.5735 APE10-dist-in 5.3957 APE9-dist-in 3.6541 R250G None None XRAY 1.85 0.165 0.187 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4v Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4XA P11309 33 305 313.0 8MT:401 Type1 Active DFGin 6.1755 14.6336 BLAminus -130.04, 168.92 67.47, 77.08 -88.95, 14.23 284.67, 77.55 -69.57, -11.46 in-in in 8.8767 Saltbr-in 2.7977 HRD-naA -75.83, -47.71 70.47, 10.64 in-in-in SNCiii in-in ActLoopNT-in 2.8155 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.28, 25.38 APE9-dihe-na -81.19, -156.58 APE8-dihe-in -90.87, 123.23 APE8-rot-in 301.93 APE67-dihe-in -70.8, -10.69 -63.86, -38.58 APE12-dist-in 9.6753 APE11-dist-in 8.5636 APE10-dist-in 5.5271 APE9-dist-in 3.6878 R250G None None XRAY 2.2 0.178 0.215 A 313.0 272.0 1 26 26 0 [[38, 290]] 1.0 5n4x Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4YA P11309 33 305 313.0 8N5:401 Type1 Active DFGin 6.0422 14.7244 BLAminus -130.6, 168.91 64.51, 83.34 -90.72, 17.65 288.76, 80.39 -65.28, -8.11 in-in in 9.034 Saltbr-in 2.9653 HRD-naA -68.66, -50.14 72.28, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.849 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.0, 26.36 APE9-dihe-na -86.43, -160.39 APE8-dihe-in -83.05, 121.49 APE8-rot-in 308.67 APE67-dihe-in -70.07, -12.6 -65.48, -36.81 APE12-dist-in 9.8289 APE11-dist-in 8.5102 APE10-dist-in 5.511 APE9-dist-in 3.916 R250G None None XRAY 2.56 0.177 0.218 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n4y Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N4ZA P11309 34 305 313.0 8MK:401 Type1 Active DFGin 6.0929 14.5863 BLAminus -128.45, 169.26 63.69, 88.15 -96.51, 19.04 288.58, 75.49 -67.41, -11.99 in-in in 8.9657 Saltbr-in 2.5723 HRD-naA -72.17, -46.94 66.82, 8.56 in-in-in SNCiii in-in ActLoopNT-in 2.8563 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.32, 24.78 APE9-dihe-na -81.23, -155.7 APE8-dihe-in -89.42, 121.2 APE8-rot-in 306.52 APE67-dihe-in -67.82, -10.0 -59.95, -43.55 APE12-dist-in 9.5784 APE11-dist-in 8.5279 APE10-dist-in 5.3815 APE9-dist-in 3.7131 R250G None None XRAY 2.257 0.18 0.208 A 313.0 272.0 0 26 26 0 [[38, 290]] 1.0 5n4z Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N50A P11309 33 305 313.0 8MN:401 Type1 Active DFGin 6.0402 14.6666 BLAminus -127.77, 166.5 68.05, 82.07 -89.1, 18.46 287.73, 79.6 -66.42, -13.96 in-in in 8.9208 Saltbr-in 2.5541 HRD-naA -72.47, -47.69 66.88, 11.1 in-in-in SNCiii in-in ActLoopNT-in 2.8127 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.17, 14.92 APE9-dihe-na -76.58, -153.55 APE8-dihe-in -94.04, 123.44 APE8-rot-in 302.17 APE67-dihe-in -70.74, -9.3 -65.25, -38.14 APE12-dist-in 9.5673 APE11-dist-in 8.4941 APE10-dist-in 5.16 APE9-dist-in 3.6772 R250G None None XRAY 1.92 0.16 0.18 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n50 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N51A P11309 33 305 313.0 8N8:401 Type1 Active DFGin 6.14 14.6258 BLAminus -127.02, 176.35 56.56, 82.77 -90.34, 20.5 285.79, 74.98 -67.87, -15.26 in-in in 8.787 Saltbr-in 2.6446 HRD-naA -74.16, -46.81 67.83, 8.58 in-in-in SNCiii in-in ActLoopNT-in 2.8023 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.83, 20.8 APE9-dihe-na -83.46, -153.2 APE8-dihe-in -92.57, 121.76 APE8-rot-in 302.99 APE67-dihe-in -70.78, -10.06 -61.78, -40.18 APE12-dist-in 9.7216 APE11-dist-in 8.5406 APE10-dist-in 5.1634 APE9-dist-in 3.7372 R250G SEP261 SEP261 XRAY 2.118 0.182 0.207 A 313.0 269.0 4 26 26 0 [[38, 290]] 1.0 5n51 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N52A P11309 33 305 313.0 8N2:401 Type1 Active DFGin 6.0542 14.4946 BLAminus -128.92, 172.68 61.78, 83.49 -88.53, 18.1 285.87, 76.88 -62.86, -14.96 in-in in 8.8791 Saltbr-in 2.8 HRD-naA -72.66, -45.02 65.77, 9.07 in-in-in SNCiii in-in ActLoopNT-in 2.8047 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.64, 23.49 APE9-dihe-na -83.54, -155.05 APE8-dihe-in -91.57, 124.16 APE8-rot-in 301.67 APE67-dihe-in -71.63, -7.35 -64.67, -40.35 APE12-dist-in 9.7762 APE11-dist-in 8.5757 APE10-dist-in 5.2818 APE9-dist-in 3.6764 R250G None None XRAY 2.252 0.172 0.21 A 313.0 268.0 5 26 26 0 [[38, 290]] 1.0 5n52 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N5LA P11309 33 305 313.0 8NZ:401 Type1 Active DFGin 6.1605 14.53 BLAminus -127.06, 174.1 60.7, 73.46 -86.15, 14.2 284.46, 73.6 -71.56, -14.64 in-in in 8.9176 Saltbr-in 2.7811 HRD-naA -74.26, -45.32 66.26, 11.22 in-in-in SNCiii in-in ActLoopNT-in 2.8951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.1, 16.72 APE9-dihe-na -75.29, -159.06 APE8-dihe-in -90.45, 122.93 APE8-rot-in 300.5 APE67-dihe-in -72.6, -9.34 -63.53, -38.45 APE12-dist-in 9.6906 APE11-dist-in 8.485 APE10-dist-in 5.2932 APE9-dist-in 3.5687 R250G SEP261 SEP261 XRAY 1.97 0.162 0.195 A 313.0 272.0 1 26 26 0 [[38, 290]] 1.0 5n5l Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5N5MA P11309 33 305 313.0 8O8:401 Type1 Active DFGin 6.0953 14.7209 BLAminus -128.4, 173.39 60.49, 81.96 -90.76, 15.73 290.29, 74.98 -68.5, -8.46 in-in in 9.0069 Saltbr-in 2.7752 HRD-naA -74.58, -47.17 67.22, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.8408 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.85, 20.79 APE9-dihe-na -81.68, -154.64 APE8-dihe-in -91.98, 123.1 APE8-rot-in 303.04 APE67-dihe-in -72.34, -6.29 -62.86, -39.4 APE12-dist-in 9.6452 APE11-dist-in 8.5152 APE10-dist-in 5.2422 APE9-dist-in 3.6671 R250G SEP261 SEP261 XRAY 2.21 0.168 0.205 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5n5m Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 5NDTA P11309 33 305 313.0 8UB:402 Type1 Active DFGin 6.114 14.7046 BLAminus -128.77, 171.81 63.42, 78.28 -87.87, 17.81 284.74, 79.81 -71.9, -9.72 in-in in 8.8817 Saltbr-in 2.6322 HRD-naA -72.09, -45.67 67.68, 10.44 in-in-in SNCiii in-in ActLoopNT-in 2.837 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.91, 24.5 APE9-dihe-na -81.02, -156.58 APE8-dihe-in -91.09, 121.22 APE8-rot-in 302.75 APE67-dihe-in -68.43, -10.6 -60.72, -41.46 APE12-dist-in 9.788 APE11-dist-in 8.5839 APE10-dist-in 5.4022 APE9-dist-in 3.7192 R250G None None XRAY 1.985 0.162 0.194 A 313.0 273.0 0 26 26 0 [[38, 290]] 1.0 5ndt Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7Z6UA P11309 33 305 313.0 IJB:402 Type1 Active DFGin 6.2708 14.4925 BLAminus -123.62, 176.91 53.69, 81.97 -85.84, 21.16 285.55, 68.27 -70.71, -12.85 in-in in 8.7429 Saltbr-in 2.7682 HRD-naA -72.34, -45.38 65.34, 4.41 in-in-in SNCiii in-in ActLoopNT-in 2.7594 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.54, 10.63 APE9-dihe-na -83.63, -150.44 APE8-dihe-in -98.54, 120.92 APE8-rot-in 299.64 APE67-dihe-in -72.4, -8.48 -60.83, -39.47 APE12-dist-in 9.7699 APE11-dist-in 8.6298 APE10-dist-in 4.6662 APE9-dist-in 3.71 R250G SEP261 SEP261 XRAY 2.28 0.163 0.191 A 313.0 268.0 5 26 26 0 [[38, 290]] 1.0 7z6u Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3CXWA P11309 33 306 313.0 7CP:501 Type1 Active DFGin 6.1536 14.6175 BLAminus -123.7, 175.96 66.3, 77.59 -92.53, 20.47 286.96, 76.96 -73.25, -11.74 in-in in 8.9096 Saltbr-in 2.6276 HRD-naA -73.02, -49.99 67.21, 12.05 in-in-in SNCiii in-in ActLoopNT-in 2.8094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.29, 21.64 APE9-dihe-na -81.37, -152.87 APE8-dihe-in -93.72, 121.7 APE8-rot-in 305.98 APE67-dihe-in -70.04, -11.91 -61.57, -39.54 APE12-dist-in 9.572 APE11-dist-in 8.3971 APE10-dist-in 5.2889 APE9-dist-in 3.6214 R250G None None XRAY 2.1 0.166 0.206 A 314.0 272.0 2 26 26 0 [[38, 290]] 1.0 3cxw Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3CY2A P11309 33 305 313.0 MB9:501 Type1 Active DFGin 6.1626 14.6449 BLAminus -126.41, 176.21 64.46, 78.27 -92.72, 18.89 288.13, 73.75 -67.98, -11.93 in-in in 8.9051 Saltbr-in 2.5685 HRD-naA -71.13, -52.84 70.37, 7.17 in-in-in SNCiii in-in ActLoopNT-in 2.8534 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.27, 21.57 APE9-dihe-na -78.39, -153.2 APE8-dihe-in -93.22, 122.03 APE8-rot-in 307.28 APE67-dihe-in -67.99, -12.82 -60.45, -42.49 APE12-dist-in 9.5435 APE11-dist-in 8.4795 APE10-dist-in 5.3954 APE9-dist-in 3.5574 R250G None None XRAY 2.01 0.169 0.199 A 314.0 271.0 2 26 26 0 [[38, 290]] 1.0 3cy2 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3CY3A P11309 33 305 313.0 JN5:501 Type1 Active DFGin 6.3033 14.4186 BLAminus -119.65, 175.12 56.83, 74.92 -82.21, 12.5 285.74, 75.76 -70.58, -7.45 in-in in 8.7561 Saltbr-in 2.5596 HRD-naA -67.55, -45.89 68.27, 6.37 in-in-in SNCiii in-in ActLoopNT-in 2.8172 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.11, 26.07 APE9-dihe-na -79.4, -161.09 APE8-dihe-in -89.18, 123.7 APE8-rot-in 304.7 APE67-dihe-in -65.31, -15.75 -62.09, -40.0 APE12-dist-in 9.6746 APE11-dist-in 8.4856 APE10-dist-in 5.5666 APE9-dist-in 3.6228 R250G SEP261 SEP261 XRAY 2.15 0.165 0.205 A 314.0 271.0 2 26 26 0 [[38, 290]] 1.0 3cy3 Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4RPVA P11309 33 305 313.0 3UR:401 Type1 Active DFGin 5.9582 14.8542 BLAminus -145.63, 161.43 69.99, 88.37 -103.98, 21.07 280.48, 100.64 -81.25, 11.11 in-in in 8.9443 Saltbr-in 2.804 HRD-naA -54.49, -51.71 77.62, -1.62 in-in-in SNCiii in-in ActLoopNT-in 2.6013 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.21, 30.75 APE9-dihe-na -100.7, -169.57 APE8-dihe-in -63.18, 128.08 APE8-rot-in 302.06 APE67-dihe-in -40.53, -14.86 -60.72, -74.04 APE12-dist-in 9.5906 APE11-dist-in 8.8948 APE10-dist-in 5.655 APE9-dist-in 4.1527 None None None XRAY 3.05 0.229 0.273 A 410.0 273.0 0 26 26 0 [[38, 290]] 1.0 4rpv Homo sapiens CAMK_PIM1_HUMAN CAMK 9.3e-65 224.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 8AFRA P11309 33 305 313.0 M0F:401 Type1 Active DFGin 6.0243 14.4056 BLAminus -126.46, 177.16 55.61, 83.44 -89.48, 19.88 284.93, 74.96 -67.33, -13.52 in-in in 8.8307 Saltbr-in 2.6484 HRD-naA -72.52, -48.51 66.56, 10.77 in-in-in SNCiii in-in ActLoopNT-in 2.8149 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.4, 19.87 APE9-dihe-na -78.39, -149.93 APE8-dihe-in -97.85, 123.61 APE8-rot-in 301.25 APE67-dihe-in -68.16, -10.25 -64.9, -40.75 APE12-dist-in 9.7271 APE11-dist-in 8.4666 APE10-dist-in 5.304 APE9-dist-in 3.645 R250G SEP261 SEP261 XRAY 2.15 0.166 0.191 A 309.0 264.0 7 26 26 0 [[38, 290]] 1.0 8afr Homo sapiens CAMK_PIM1_HUMAN CAMK 3.1e-62 216.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4ALUA P11309 33 306 313.0 79O:1308 Type1 Active DFGin 6.0396 14.4546 BLAminus -129.3, 164.2 71.61, 87.87 -98.95, 24.33 283.93, 80.99 -80.29, 2.07 in-in in 8.7471 Saltbr-in 2.5495 HRD-naA -75.13, -46.19 78.28, -3.97 in-in-in SNCiii in-in ActLoopNT-in 2.8293 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.43, 41.36 APE9-dihe-na -93.61, -144.58 APE8-dihe-in -101.6, 125.74 APE8-rot-in 300.81 APE67-dihe-in -62.7, -19.8 -64.97, -44.76 APE12-dist-in 9.6233 APE11-dist-in 8.6017 APE10-dist-in 5.7263 APE9-dist-in 3.7807 None None None XRAY 2.6 0.184 0.248 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 4alu Homo sapiens CAMK_PIM1_HUMAN CAMK 2.7e-64 222.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3T9IA P11309 33 306 313.0 3T9:401 Type1.5_Back Active DFGin 6.5428 14.2947 BLAminus -132.77, 172.96 59.67, 82.28 -96.48, 17.83 287.7, 76.66 -65.3, -19.74 in-in in 8.4349 Saltbr-in 2.7571 HRD-naA -69.28, -50.32 73.93, -9.03 in-in-in SNCiii in-in ActLoopNT-in 2.8337 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.31, 28.32 APE9-dihe-na -97.99, -160.13 APE8-dihe-in -83.72, 117.37 APE8-rot-in 302.02 APE67-dihe-in -69.04, -9.18 -56.37, -42.61 APE12-dist-in 9.7353 APE11-dist-in 8.6561 APE10-dist-in 5.1983 APE9-dist-in 4.2807 None SEP261 SEP261 XRAY 2.6 0.165 0.227 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 3t9i Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6AYDA P11309 34 305 313.0 C2J:401 Type1.5_Back Active DFGin 6.2253 14.5726 BLAminus -129.9, 167.94 69.26, 93.71 -101.76, 29.48 284.65, 86.99 -77.7, -11.94 in-in in 8.4989 Saltbr-in 2.6944 HRD-naA -64.89, -48.59 73.72, 7.41 in-in-in SNCiii in-in ActLoopNT-in 2.7192 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.07, 29.72 APE9-dihe-na -90.29, -149.58 APE8-dihe-in -90.3, 121.0 APE8-rot-in 309.33 APE67-dihe-in -70.19, -4.08 -54.85, -49.52 APE12-dist-in 9.7574 APE11-dist-in 8.5952 APE10-dist-in 5.4358 APE9-dist-in 4.0665 R250G None None XRAY 3.0 0.171 0.23 A 334.0 272.0 0 26 26 0 [[38, 290]] 1.0 6ayd Homo sapiens CAMK_PIM1_HUMAN CAMK 1.9e-64 223.5 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4RBLA P11309 33 305 313.0 3O7:401 Type1 Inactive DFGin 6.1855 14.6322 ABAminus -123.28, -49.04 -102.92, 101.34 -86.59, 10.95 288.26, 82.24 -66.9, -9.47 in-in in 8.7086 Saltbr-in 2.5498 HRD-naA -76.77, -47.35 72.65, 1.38 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.2, 7.15 APE9-dihe-na -86.69, -159.73 APE8-dihe-in -86.44, 135.53 APE8-rot-in 335.24 APE67-dihe-in -50.84, -15.83 -62.51, -62.82 APE12-dist-in 9.2624 APE11-dist-in 8.5648 APE10-dist-in 4.3791 APE9-dist-in 3.874 None SEP261 SEP261 XRAY 2.55 0.191 0.249 A 289.0 272.0 1 26 26 0 [[38, 290]] 1.0 4rbl Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4RC2A P11309 33 305 313.0 3O8:401 Type1 Inactive DFGin 6.1514 14.4868 ABAminus -124.35, -31.66 -113.65, 105.77 -88.14, 13.2 287.98, 83.78 -66.51, -15.85 in-in in 8.8722 Saltbr-in 2.534 HRD-naA -72.15, -49.17 67.29, 8.38 in-in-in SNCiii in-in ActLoopNT-in 2.7926 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.36, 8.25 APE9-dihe-na -77.04, -152.99 APE8-dihe-in -93.85, 131.35 APE8-rot-in 322.71 APE67-dihe-in -71.49, -6.88 -57.98, -44.79 APE12-dist-in 9.4324 APE11-dist-in 8.5203 APE10-dist-in 4.7174 APE9-dist-in 3.8077 None SEP261 SEP261 XRAY 2.096 0.21 0.246 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 4rc2 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4RC3A P11309 33 305 313.0 3OA:401 Type1 Inactive DFGin 6.1312 14.7301 ABAminus -124.18, -44.55 -102.49, 107.8 -86.08, 9.84 283.97, 82.66 -66.94, -13.06 in-in in 8.9316 Saltbr-in 2.7278 HRD-naA -74.64, -46.7 68.78, 5.57 in-in-in SNCiii in-in ActLoopNT-in 2.7168 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.55, 7.68 APE9-dihe-na -87.91, -151.36 APE8-dihe-in -94.35, 131.18 APE8-rot-in 325.68 APE67-dihe-in -63.89, -8.14 -60.26, -51.45 APE12-dist-in 9.479 APE11-dist-in 8.6351 APE10-dist-in 4.6757 APE9-dist-in 3.9424 None SEP261 SEP261 XRAY 2.338 0.192 0.222 A 289.0 272.0 1 26 26 0 [[38, 290]] 1.0 4rc3 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4RC4A P11309 33 305 313.0 3OK:401 Type1 Inactive DFGin 6.1945 14.5075 ABAminus -123.13, -33.74 -113.37, 104.45 -91.23, 9.07 284.92, 83.68 -71.27, -6.47 in-in in 8.6118 Saltbr-in 2.7351 HRD-naA -68.9, -48.63 75.17, 7.81 in-in-in SNCiii in-in ActLoopNT-in 2.8636 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.62, -3.25 APE9-dihe-na -70.99, -164.38 APE8-dihe-in -82.7, 141.94 APE8-rot-in 331.47 APE67-dihe-in -56.62, -19.58 -59.05, -56.98 APE12-dist-in 9.1914 APE11-dist-in 8.5877 APE10-dist-in 4.5075 APE9-dist-in 3.8584 None SEP261 SEP261 XRAY 2.651 0.191 0.241 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 4rc4 Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4I41A P11309 33 305 313.0 MIX:500,MIX:501 Type1,Allosteric Inactive DFGin 6.1399 14.4159 ABAminus -121.87, -36.78 -115.75, 100.81 -88.41, 10.15 289.07, 75.39 -54.5, -25.74 in-in in 8.6342 Saltbr-in 2.7561 HRD-naA -69.84, -46.43 70.52, 12.32 in-in-out SNCiio in-out ActLoopNT-in 2.9176 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -124.01, -14.74 APE9-dihe-na -57.33, 178.24 APE8-dihe-in -71.04, 142.33 APE8-rot-out 6.4 APE67-dihe-in -51.91, -16.42 -63.07, -52.85 APE12-dist-in 9.1226 APE11-dist-in 8.5821 APE10-dist-in 4.5899 APE9-dist-in 3.8828 None SEP261 SEP261 XRAY 2.7 0.2 0.249 A 281.0 273.0 0 26 26 0 [[38, 290]] 1.0 4i41 Homo sapiens CAMK_PIM1_HUMAN CAMK 2.7e-65 226.2 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 7OOXA P11309 1 305 313.0 No_ligand No_ligand Inactive DFGin 6.0077 14.4258 BLAminus -128.2, 171.48 64.26, 84.06 -90.51, 19.09 289.76, 88.29 -67.14, -14.45 in-in in 8.8933 Saltbr-in 2.5304 HRD-naA -69.11, -49.22 70.21, 6.96 in-in-out SNCiio in-out ActLoopNT-in 2.8525 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -112.93, -2.13 APE9-dihe-na -73.5, 169.82 APE8-dihe-in -80.91, 158.93 APE8-rot-out 67.73 APE67-dihe-in -74.5, -10.73 -58.29, -40.88 APE12-dist-in 9.6067 APE11-dist-in 8.8847 APE10-dist-in 4.9932 APE9-dist-in 5.4364 None None None XRAY 1.97 0.181 0.222 A 313.0 284.0 0 26 26 0 [[38, 290]] 1.0 7oox Homo sapiens CAMK_PIM1_HUMAN CAMK 1.5e-64 223.7 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 3DCVA P11309 32 305 313.0 55E:500 Type1 Inactive DFGin 6.4113 14.6785 BLAminus -130.48, 168.13 69.03, 78.23 -92.76, 18.93 285.58, 71.29 -63.83, -15.25 in-in in 8.3124 Saltbr-in 2.5592 HRD-naA -64.55, -50.54 72.29, 1.73 in-in-out SNCiio in-out ActLoopNT-in 2.876 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -106.61, -25.99 APE9-dihe-na -54.65, -172.57 APE8-dihe-in -80.08, 136.57 APE8-rot-out 118.16 APE67-dihe-in -59.26, -8.45 -62.5, -57.95 APE12-dist-in 9.5381 APE11-dist-in 8.9721 APE10-dist-in 4.6762 APE9-dist-in 3.8897 None SEP261 SEP261 XRAY 2.7 0.182 0.234 A 328.0 274.0 0 26 26 0 [[38, 290]] 1.0 3dcv Homo sapiens CAMK_PIM1_HUMAN CAMK 4.7e-65 225.4 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 6KZIA P11309 33 305 313.0 RTX:401 Type1 Inactive DFGin 6.0118 14.7309 BLBminus -130.32, 166.69 73.68, 82.71 -88.65, -171.62 289.43, 86.65 20.03, 81.34 in-in in 8.9794 Saltbr-in 2.742 HRD-naA -68.55, -45.07 65.35, 8.38 in-in-in SNCiii in-in ActLoopNT-in 2.7184 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.04, 49.18 APE9-dihe-na -108.43, -149.21 APE8-dihe-in -96.99, 121.09 APE8-rot-in 319.52 APE67-dihe-in -60.06, -16.31 -54.82, -52.12 APE12-dist-in 9.3829 APE11-dist-in 8.3363 APE10-dist-in 5.48 APE9-dist-in 4.0226 None SEP261 SEP261 XRAY 2.8 0.173 0.233 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 6kzi Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4IAAA P11309 33 305 313.0 RTZ:401 Type1 Inactive DFGin 6.018 14.534 None -118.73, -143.64 -58.0, 140.84 -105.0, 12.55 279.89, 91.42 -63.74, -38.82 in-in in 8.9764 Saltbr-in 2.4263 HRD-naA -66.74, -45.93 76.57, 1.9 in-in-in SNCiii in-in ActLoopNT-in 2.8243 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -101.97, 36.36 APE9-dihe-na -102.7, -148.72 APE8-dihe-in -99.25, 120.44 APE8-rot-in 325.38 APE67-dihe-in -56.81, -14.63 -51.76, -61.55 APE12-dist-in 9.3212 APE11-dist-in 8.4746 APE10-dist-in 4.9412 APE9-dist-in 4.319 None SEP261 SEP261 XRAY 2.85 0.187 0.231 A 289.0 273.0 0 26 26 0 [[38, 290]] 1.0 4iaa Homo sapiens CAMK_PIM1_HUMAN CAMK 3e-65 226.0 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1
PIM1 PIM1_HUMAN 4XH6A P11309 33 305 313.0 HUL:401 Type1 Inactive DFGin 6.0669 14.6256 None -113.12, -75.74 -81.94, 104.4 -86.86, 17.15 286.29, 78.0 -66.66, -16.93 in-in in 8.963 Saltbr-in 2.6759 HRD-naA -71.75, -47.81 68.98, 9.54 in-in-in SNCiii in-in ActLoopNT-in 2.8264 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.53, 35.49 APE9-dihe-na -89.22, -153.74 APE8-dihe-in -92.85, 123.83 APE8-rot-in 304.19 APE67-dihe-in -63.31, -10.32 -62.77, -45.27 APE12-dist-in 9.5688 APE11-dist-in 8.4688 APE10-dist-in 5.5301 APE9-dist-in 3.7526 None None None XRAY 2.04 0.202 0.226 A 294.0 273.0 0 26 26 0 [[38, 290]] 1.0 4xh6 Homo sapiens CAMK_PIM1_HUMAN CAMK 3.2e-65 225.9 1.0 256.0 256.0 185 186 187 189 191 67 89 93 164 166 165 167.0 224 211 206 205 204 203 202 201 200 121 Serine/threonine-protein kinase pim-1

CAMK_PIM1 (Serine/threonine-protein kinase pim-1)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name