| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PDPK1 | 2BIYA | O15530 | 72 | 359 | 556.0 | ATP:1373 | ATPlike | Active | DFGin | 6.6186 | 15.0949 | BLAminus | -141.33, -175.84 | 82.91, 67.67 | -104.99, 1.58 | 283.05, 104.18 | -61.63, -33.06 | in-in | in | 8.6731 | Saltbr-in | 2.5745 | HRD-in | -63.52, -52.73 | 78.44, -11.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8201 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.22, 130.12 | APE9-dihe-na | 106.71, 171.13 | APE8-dihe-in | -96.94, 126.07 | APE8-rot-in | 299.07 | APE67-dihe-in | -62.15, -19.51 | -52.23, -44.36 | APE12-dist-in | 12.8679 | APE11-dist-in | 12.8691 | APE10-dist-in | 7.2677 | APE9-dist-in | 4.7446 | S241A | None | None | XRAY | 1.95 | 0.186 | 0.23 | A | 310.0 | 288.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 2biy | AGC_PDPK1_HUMAN | AGC | 1.8e-84 | 288.8 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3HRCA | O15530 | 76 | 359 | 556.0 | ATP:1373 | ATPlike | Active | DFGin | 6.4861 | 14.8331 | BLAminus | -136.91, -178.17 | 71.81, 74.55 | -104.54, 6.98 | 286.89, 102.51 | -65.47, -24.41 | in-in | in | 8.4211 | Saltbr-in | 3.1591 | HRD-in | -77.24, -54.93 | 76.93, -11.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.87 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.25, 162.0 | APE9-dihe-na | 130.63, -171.63 | APE8-dihe-in | -125.01, 129.68 | APE8-rot-in | 292.48 | APE67-dihe-in | -58.92, -25.29 | -45.32, -48.7 | APE12-dist-in | 7.4085 | APE11-dist-in | 10.582 | APE10-dist-in | 4.9259 | APE9-dist-in | 3.4793 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.91 | 0.182 | 0.207 | A | 311.0 | 280.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 3hrc | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4RRVA | O15530 | 76 | 359 | 556.0 | ATP:60401 | ATPlike | Active | DFGin | 6.5481 | 14.9984 | BLAminus | -136.55, -175.99 | 74.63, 72.8 | -106.52, 5.78 | 286.61, 100.18 | -68.12, -17.88 | in-in | in | 8.5198 | Saltbr-in | 2.956 | HRD-in | -71.77, -54.29 | 78.75, -11.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9375 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.13, 162.83 | APE9-dihe-na | 132.08, -169.67 | APE8-dihe-in | -127.24, 132.02 | APE8-rot-in | 298.33 | APE67-dihe-in | -59.21, -24.3 | -51.83, -46.04 | APE12-dist-in | 7.2806 | APE11-dist-in | 10.5025 | APE10-dist-in | 4.943 | APE9-dist-in | 3.5694 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.412 | 0.135 | 0.163 | A | 311.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4rrv | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5ACKA | O15530 | 73 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.6153 | 14.8606 | BLAminus | -135.34, 179.84 | 72.22, 79.01 | -106.01, 4.14 | 287.93, 97.64 | -67.02, -18.73 | in-in | in | 8.4184 | Saltbr-in | 2.5825 | HRD-in | -74.68, -53.67 | 78.01, -12.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9064 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.4, 162.51 | APE9-dihe-na | 136.44, -168.07 | APE8-dihe-in | -132.35, 133.52 | APE8-rot-in | 296.36 | APE67-dihe-in | -62.96, -23.95 | -54.34, -43.19 | APE12-dist-in | 7.3257 | APE11-dist-in | 10.5222 | APE10-dist-in | 4.9779 | APE9-dist-in | 3.5575 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.24 | 0.143 | 0.166 | A | 311.0 | 287.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5ack | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVPA | O15530 | 75 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3028 | 14.9979 | BLAminus | -144.92, -168.82 | 66.06, 77.78 | -108.23, 11.17 | 281.99, 93.22 | -63.04, -32.41 | in-in | in | 9.539 | Saltbr-in | 3.1581 | HRD-in | -77.47, -51.83 | 79.92, -12.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8481 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.64, 166.02 | APE9-dihe-na | 141.61, 177.5 | APE8-dihe-in | -123.02, 134.29 | APE8-rot-in | 296.02 | APE67-dihe-in | -68.65, -16.53 | -46.89, -50.92 | APE12-dist-in | 7.9068 | APE11-dist-in | 10.6706 | APE10-dist-in | 5.166 | APE9-dist-in | 3.7049 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | A | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVPB | O15530 | 74 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3283 | 14.5498 | BLAminus | -137.23, -179.71 | 80.14, 74.16 | -105.47, 15.38 | 295.0, 84.83 | -59.91, -31.47 | in-in | in | 9.2741 | Saltbr-in | 3.3024 | HRD-in | -80.68, -44.41 | 73.96, -16.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7443 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.8, 152.43 | APE9-dihe-na | 134.43, -173.75 | APE8-dihe-in | -120.09, 128.28 | APE8-rot-in | 302.93 | APE67-dihe-in | -67.56, -25.72 | -44.99, -47.55 | APE12-dist-in | 7.8719 | APE11-dist-in | 11.0112 | APE10-dist-in | 5.3751 | APE9-dist-in | 3.7868 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | B | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVPC | O15530 | 75 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3906 | 14.6076 | BLAminus | -132.15, -176.81 | 71.98, 84.02 | -116.53, 7.62 | 291.47, 90.46 | -60.24, -24.5 | in-in | in | 9.3044 | Saltbr-in | 3.0866 | HRD-in | -75.92, -52.06 | 78.45, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8228 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.81, 168.64 | APE9-dihe-na | 131.92, -176.79 | APE8-dihe-in | -126.79, 133.21 | APE8-rot-in | 299.13 | APE67-dihe-in | -67.64, -15.8 | -51.62, -50.49 | APE12-dist-in | 7.6523 | APE11-dist-in | 10.8632 | APE10-dist-in | 5.1235 | APE9-dist-in | 3.6447 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | C | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVPD | O15530 | 74 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3336 | 14.4328 | BLAminus | -146.99, -174.22 | 74.22, 81.56 | -113.84, 4.02 | 287.97, 93.59 | -56.11, -25.73 | in-in | in | 9.3044 | Saltbr-in | 3.2517 | HRD-in | -82.38, -50.18 | 78.4, -12.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8357 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.65, 165.17 | APE9-dihe-na | 129.1, -166.82 | APE8-dihe-in | -132.84, 129.79 | APE8-rot-in | 300.06 | APE67-dihe-in | -65.46, -17.03 | -48.9, -48.47 | APE12-dist-in | 8.2282 | APE11-dist-in | 10.8909 | APE10-dist-in | 5.3485 | APE9-dist-in | 3.6459 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | D | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4CT2A | O15530 | 75 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.5509 | 14.8668 | BLAminus | -136.23, -174.98 | 70.54, 70.07 | -102.02, 6.41 | 290.69, 95.78 | -63.73, -21.59 | in-in | in | 8.2523 | Saltbr-in | 2.6427 | HRD-in | -73.2, -54.84 | 77.37, -9.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9649 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.02, 163.59 | APE9-dihe-na | 137.39, -170.05 | APE8-dihe-in | -132.12, 131.72 | APE8-rot-in | 295.26 | APE67-dihe-in | -63.06, -17.27 | -51.84, -45.87 | APE12-dist-in | 7.1628 | APE11-dist-in | 10.5242 | APE10-dist-in | 4.9787 | APE9-dist-in | 3.5273 | L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.25 | 0.194 | 0.226 | A | 311.0 | 280.0 | 5 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4ct2 | AGC_PDPK1_HUMAN | AGC | 9.5e-84 | 286.4 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5MRDA | O15530 | 76 | 359 | 556.0 | ATP:405 | ATPlike | Active | DFGin | 6.4288 | 14.7004 | BLAminus | -133.69, -177.11 | 74.21, 73.9 | -105.88, 9.0 | 289.39, 99.64 | -68.32, -19.62 | in-in | in | 8.3463 | Saltbr-in | 2.6673 | HRD-in | -74.32, -53.19 | 77.26, -10.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9416 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.86, 160.68 | APE9-dihe-na | 136.11, -166.87 | APE8-dihe-in | -131.1, 132.63 | APE8-rot-in | 296.36 | APE67-dihe-in | -62.36, -23.28 | -53.02, -44.84 | APE12-dist-in | 7.3524 | APE11-dist-in | 10.4975 | APE10-dist-in | 4.9095 | APE9-dist-in | 3.5424 | K76S,L113V,I118V,I119N,V124I,T128Q,R131K,T148C | SEP241 | SEP241 | XRAY | 1.41 | 0.142 | 0.174 | A | 310.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5mrd | AGC_PDPK1_HUMAN | AGC | 1.7e-83 | 285.6 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3HRFA | O15530 | 75 | 359 | 556.0 | ATP:1373,P47:1374 | ATPlike,Allosteric | Active | DFGin | 6.5137 | 14.7842 | BLAminus | -133.77, -176.11 | 75.25, 77.12 | -110.83, 6.58 | 287.55, 100.98 | -63.85, -22.79 | in-in | in | 8.3869 | Saltbr-in | 2.7006 | HRD-in | -73.67, -53.98 | 76.59, -10.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9232 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.42, 166.15 | APE9-dihe-na | 124.75, -165.6 | APE8-dihe-in | -127.97, 128.5 | APE8-rot-in | 295.31 | APE67-dihe-in | -62.28, -24.12 | -44.34, -47.42 | APE12-dist-in | 7.3513 | APE11-dist-in | 10.5457 | APE10-dist-in | 4.8669 | APE9-dist-in | 3.4806 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.9 | 0.165 | 0.177 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 3hrf | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4A06A | O15530 | 75 | 359 | 556.0 | ATP:500,A06:600 | ATPlike,Allosteric | Active | DFGin | 6.5121 | 14.757 | BLAminus | -135.73, -177.17 | 74.25, 74.67 | -110.25, 11.82 | 284.97, 101.73 | -68.23, -22.46 | in-in | in | 8.3192 | Saltbr-in | 2.8636 | HRD-in | -73.73, -51.84 | 74.62, -10.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9204 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.65, 165.25 | APE9-dihe-na | 128.95, -173.35 | APE8-dihe-in | -120.15, 131.51 | APE8-rot-in | 299.31 | APE67-dihe-in | -59.46, -27.29 | -45.75, -47.91 | APE12-dist-in | 7.336 | APE11-dist-in | 10.4473 | APE10-dist-in | 4.8734 | APE9-dist-in | 3.5088 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.0 | 0.161 | 0.198 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4a06 | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4AW0A | O15530 | 75 | 359 | 556.0 | ATP:500,MJF:600 | ATPlike,Allosteric | Active | DFGin | 6.5313 | 14.9926 | BLAminus | -134.84, 177.25 | 78.73, 76.19 | -106.3, 8.53 | 283.51, 97.11 | -69.63, -19.36 | in-in | in | 8.5954 | Saltbr-in | 3.0091 | HRD-in | -83.05, -53.03 | 79.45, -12.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9336 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.69, 159.04 | APE9-dihe-na | 139.48, -167.8 | APE8-dihe-in | -131.87, 132.42 | APE8-rot-in | 295.45 | APE67-dihe-in | -61.29, -25.28 | -54.74, -42.17 | APE12-dist-in | 7.5089 | APE11-dist-in | 10.6011 | APE10-dist-in | 5.0264 | APE9-dist-in | 3.5797 | Y288G,Q292A | SEP241 | SEP241,CME260 | XRAY | 1.43 | 0.171 | 0.188 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4aw0 | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4AW1A | O15530 | 66 | 359 | 556.0 | ATP:1360,21O:1361 | ATPlike,Allosteric | Active | DFGin | 6.325 | 14.155 | BLAminus | -137.24, -178.23 | 68.96, 84.69 | -105.37, 17.06 | 286.01, 86.79 | -62.77, -26.7 | in-in | in | 8.5758 | Saltbr-in | 2.8639 | HRD-in | -81.18, -54.06 | 78.32, -13.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8487 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.98, 160.2 | APE9-dihe-na | 130.22, -162.57 | APE8-dihe-in | -126.98, 128.72 | APE8-rot-in | 295.96 | APE67-dihe-in | -57.45, -24.35 | -48.01, -47.7 | APE12-dist-in | 7.6532 | APE11-dist-in | 10.8523 | APE10-dist-in | 5.0751 | APE9-dist-in | 3.5856 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.68 | 0.165 | 0.186 | A | 311.0 | 287.0 | 5 | 30 | 25 | 5 | [[82, 342]] | 1.0 | 4aw1 | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4RQKA | O15530 | 74 | 359 | 556.0 | ATP:403,R1S:404 | ATPlike,Allosteric | Active | DFGin | 6.4608 | 14.7857 | BLAminus | -139.06, -177.03 | 75.27, 72.83 | -105.25, 7.36 | 287.3, 98.33 | -64.7, -21.38 | in-in | in | 8.4643 | Saltbr-in | 2.9412 | HRD-in | -73.98, -52.31 | 74.79, -9.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8799 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.64, 164.69 | APE9-dihe-na | 126.87, -171.23 | APE8-dihe-in | -124.75, 130.48 | APE8-rot-in | 298.57 | APE67-dihe-in | -59.79, -23.66 | -48.31, -47.88 | APE12-dist-in | 7.2437 | APE11-dist-in | 10.4657 | APE10-dist-in | 4.9176 | APE9-dist-in | 3.5437 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.55 | 0.133 | 0.167 | A | 311.0 | 286.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4rqk | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4RQVA | O15530 | 71 | 359 | 556.0 | ATP:405,R2S:406 | ATPlike,Allosteric | Active | DFGin | 6.4916 | 14.9536 | BLAminus | -139.41, -174.88 | 74.87, 69.78 | -102.0, 7.85 | 285.85, 94.73 | -65.11, -21.56 | in-in | in | 8.2557 | Saltbr-in | 2.7717 | HRD-in | -72.94, -52.57 | 74.87, -10.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9156 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.07, 164.19 | APE9-dihe-na | 130.69, -171.7 | APE8-dihe-in | -126.67, 130.74 | APE8-rot-in | 297.63 | APE67-dihe-in | -61.47, -23.77 | -49.17, -46.26 | APE12-dist-in | 7.2532 | APE11-dist-in | 10.4876 | APE10-dist-in | 4.9687 | APE9-dist-in | 3.5133 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.502 | 0.133 | 0.166 | A | 311.0 | 289.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4rqv | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVOA | O15530 | 73 | 359 | 556.0 | ATP:401,78W:402 | ATPlike,Allosteric | Active | DFGin | 6.581 | 15.0047 | BLAminus | -134.78, 179.9 | 79.12, 70.17 | -103.55, 0.25 | 286.72, 100.66 | -64.63, -19.63 | in-in | in | 8.5884 | Saltbr-in | 2.6313 | HRD-in | -71.89, -54.41 | 77.65, -9.82 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9194 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.78, 162.52 | APE9-dihe-na | 134.75, -167.11 | APE8-dihe-in | -130.46, 134.12 | APE8-rot-in | 296.12 | APE67-dihe-in | -62.26, -22.94 | -53.92, -45.37 | APE12-dist-in | 7.4502 | APE11-dist-in | 10.5584 | APE10-dist-in | 4.9836 | APE9-dist-in | 3.5527 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.09 | 0.136 | 0.157 | A | 311.0 | 287.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvo | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4XX9A | O15530 | 71 | 359 | 556.0 | ATP:401,RF4:402,RF4:403 | ATPlike,Allosteric,Allosteric | Active | DFGin | 6.5134 | 14.9881 | BLAminus | -138.47, -176.21 | 74.83, 73.76 | -104.66, 7.86 | 282.59, 98.49 | -68.99, -20.43 | in-in | in | 8.4422 | Saltbr-in | 2.9225 | HRD-in | -73.71, -50.51 | 73.32, -9.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8949 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.41, 162.37 | APE9-dihe-na | 129.79, -167.49 | APE8-dihe-in | -129.09, 132.1 | APE8-rot-in | 295.95 | APE67-dihe-in | -59.66, -23.23 | -49.94, -47.34 | APE12-dist-in | 7.3717 | APE11-dist-in | 10.5754 | APE10-dist-in | 4.9467 | APE9-dist-in | 3.5452 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.4 | 0.13 | 0.165 | A | 310.0 | 289.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4xx9 | AGC_PDPK1_HUMAN | AGC | 6.8e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4A07A | O15530 | 75 | 359 | 556.0 | ATP:500,AZ7:600,AZ7:700 | ATPlike,Allosteric,Allosteric | Active | DFGin | 6.6546 | 14.7523 | BLAminus | -135.35, -178.9 | 76.01, 72.4 | -108.94, 8.63 | 286.31, 98.68 | -64.37, -21.88 | in-in | in | 8.6213 | Saltbr-in | 2.919 | HRD-in | -76.19, -54.82 | 80.07, -12.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9107 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.16, 162.52 | APE9-dihe-na | 132.15, -164.48 | APE8-dihe-in | -133.89, 130.56 | APE8-rot-in | 295.87 | APE67-dihe-in | -62.13, -24.83 | -47.31, -46.9 | APE12-dist-in | 7.3216 | APE11-dist-in | 10.4272 | APE10-dist-in | 4.9977 | APE9-dist-in | 3.5816 | Y288G,Q292A | SEP241 | SEP241,CSS260 | XRAY | 1.85 | 0.161 | 0.2 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4a07 | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 8DQTA | O15530 | 70 | 359 | 556.0 | U35:401,U35:402,U35:403 | Allosteric,Allosteric,Allosteric | Active | DFGin | 6.5386 | 15.228 | BLAminus | -137.99, -177.67 | 76.39, 75.41 | -107.03, 7.63 | 286.75, 95.91 | -68.77, -18.63 | in-in | in | 8.5573 | Saltbr-in | 2.9067 | HRD-in | -74.31, -48.93 | 74.07, -13.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9489 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -143.2, 161.34 | APE9-dihe-na | 132.87, -165.96 | APE8-dihe-in | -131.33, 133.45 | APE8-rot-in | 295.53 | APE67-dihe-in | -61.71, -24.62 | -51.87, -45.17 | APE12-dist-in | 7.2521 | APE11-dist-in | 10.4342 | APE10-dist-in | 4.9085 | APE9-dist-in | 3.5907 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.31 | 0.2 | 0.224 | A | 311.0 | 290.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 8dqt | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3OTUA | O15530 | 77 | 359 | 556.0 | J30:1,BI4:360 | Allosteric,Type1.5_Front | Active | DFGin | 6.407 | 14.9865 | BLAminus | -147.19, -166.49 | 62.44, 61.65 | -95.64, 10.19 | 290.91, 105.88 | -63.28, -24.6 | in-in | in | 8.3704 | Saltbr-in | 3.3366 | HRD-in | -67.23, -53.13 | 82.11, -16.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7953 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.97, 157.81 | APE9-dihe-na | 151.4, -176.81 | APE8-dihe-in | -123.26, 126.19 | APE8-rot-in | 294.94 | APE67-dihe-in | -53.95, -30.51 | -40.25, -53.87 | APE12-dist-in | 7.7118 | APE11-dist-in | 10.3288 | APE10-dist-in | 5.2437 | APE9-dist-in | 4.1303 | T148C | SEP241 | SEP241 | XRAY | 2.101 | 0.197 | 0.24 | A | 316.0 | 277.0 | 6 | 30 | 25 | 5 | [[82, 342]] | 1.0 | 3otu | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | AF-O15530-K1A | O15530 | 74 | 350 | 556.0 | No_ligand | No_ligand | Active | DFGin | 6.307 | 14.7525 | BLAminus | -134.14, -175.03 | 67.73, 56.76 | -81.0, 7.09 | 290.02, 100.1 | -62.73, -31.75 | in-in | in | 8.4785 | Saltbr-in | 2.6917 | HRD-in | -71.22, -49.98 | 68.85, -15.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9019 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -143.76, 160.45 | APE9-dihe-na | 125.82, -178.56 | APE8-dihe-in | -110.7, 135.78 | APE8-rot-in | 301.58 | APE67-dihe-in | -71.92, -18.9 | -54.44, -36.21 | APE12-dist-in | 7.4783 | APE11-dist-in | 10.7463 | APE10-dist-in | 5.0363 | APE9-dist-in | 3.4837 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 277.0 | 277.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | AF-O15530-K1 | AGC_PDPK1_HUMAN | AGC | 8.4e-85 | 289.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | AF-O15530-K3A | O15530 | 74 | 350 | 556.0 | No_ligand | No_ligand | Active | DFGin | 6.0234 | 14.6473 | BLAminus | -139.54, -179.29 | 63.97, 66.91 | -82.88, 11.22 | 294.97, 97.73 | -59.7, -35.74 | in-in | in | 8.7295 | Saltbr-in | 2.6551 | HRD-in | -73.34, -47.9 | 67.59, -9.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8048 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.66, 143.7 | APE9-dihe-na | 124.83, 164.09 | APE8-dihe-in | -82.81, 130.45 | APE8-rot-in | 291.03 | APE67-dihe-in | -71.92, -16.19 | -51.02, -35.4 | APE12-dist-in | 8.3871 | APE11-dist-in | 11.0601 | APE10-dist-in | 5.2904 | APE9-dist-in | 4.3622 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 277.0 | 277.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | AF-O15530-K3 | AGC_PDPK1_HUMAN | AGC | 8.4e-85 | 289.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3SC1A | O15530 | 73 | 359 | 556.0 | 3S1:900 | Type1 | Active | DFGin | 6.4332 | 14.1153 | BLAminus | -125.85, 175.62 | 82.13, 80.63 | -113.39, 8.45 | 290.85, 87.77 | -53.07, -47.22 | in-in | in | 8.7083 | Saltbr-in | 3.2163 | HRD-in | -72.93, -48.81 | 80.48, -8.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8508 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -100.12, -172.48 | APE9-dihe-na | 115.93, 147.74 | APE8-dihe-in | -93.61, 137.68 | APE8-rot-in | 299.7 | APE67-dihe-in | -55.26, -32.91 | -54.79, -48.8 | APE12-dist-in | 8.7388 | APE11-dist-in | 10.6062 | APE10-dist-in | 5.4107 | APE9-dist-in | 3.9864 | None | SEP241 | SEP241 | XRAY | 2.7 | 0.2 | 0.237 | A | 311.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3sc1 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3RCJA | O15530 | 77 | 358 | 556.0 | 3RC:0 | Type1 | Active | DFGin | 6.5504 | 14.3915 | BLAminus | -128.99, -167.62 | 59.76, 67.13 | -93.27, 12.1 | 286.78, 86.8 | -60.54, -37.27 | in-in | in | 8.539 | Saltbr-in | 2.7862 | HRD-in | -65.85, -49.34 | 77.48, -8.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.08, 164.56 | APE9-dihe-na | 127.57, -173.24 | APE8-dihe-in | -123.98, 130.3 | APE8-rot-in | 296.56 | APE67-dihe-in | -63.09, -20.07 | -49.59, -44.96 | APE12-dist-in | 7.8304 | APE11-dist-in | 10.7456 | APE10-dist-in | 5.0252 | APE9-dist-in | 3.6456 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.7 | 0.217 | 0.198 | A | 311.0 | 282.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 3rcj | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVLA | O15530 | 74 | 359 | 556.0 | 537:401 | Type1 | Active | DFGin | 6.5959 | 14.602 | BLAminus | -130.64, -179.01 | 78.07, 78.29 | -107.64, 5.9 | 287.24, 98.42 | -64.3, -24.0 | in-in | in | 8.2927 | Saltbr-in | 2.5582 | HRD-in | -74.44, -52.48 | 78.34, -12.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9059 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.91, 163.01 | APE9-dihe-na | 134.48, -168.83 | APE8-dihe-in | -131.23, 133.97 | APE8-rot-in | 296.05 | APE67-dihe-in | -61.17, -24.01 | -50.83, -47.55 | APE12-dist-in | 7.3206 | APE11-dist-in | 10.4705 | APE10-dist-in | 4.8806 | APE9-dist-in | 3.5651 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.4 | 0.154 | 0.178 | A | 311.0 | 286.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvl | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVMA | O15530 | 76 | 359 | 556.0 | ADE:401 | Type1 | Active | DFGin | 6.5146 | 14.8576 | BLAminus | -134.29, -178.73 | 78.5, 76.19 | -107.92, 3.05 | 284.81, 100.85 | -68.49, -15.39 | in-in | in | 8.3988 | Saltbr-in | 2.9222 | HRD-in | -74.83, -53.98 | 76.68, -6.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9138 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.77, 160.72 | APE9-dihe-na | 136.54, -165.87 | APE8-dihe-in | -131.32, 134.23 | APE8-rot-in | 298.42 | APE67-dihe-in | -62.0, -21.56 | -53.2, -46.03 | APE12-dist-in | 7.4265 | APE11-dist-in | 10.5567 | APE10-dist-in | 4.9493 | APE9-dist-in | 3.5336 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.26 | 0.135 | 0.155 | A | 311.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvm | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5LVNA | O15530 | 75 | 359 | 556.0 | ADN:402 | Type1 | Active | DFGin | 6.4926 | 14.7837 | BLAminus | -138.56, -175.41 | 73.41, 75.09 | -105.63, 5.44 | 285.54, 101.95 | -63.79, -19.6 | in-in | in | 8.4347 | Saltbr-in | 2.7393 | HRD-in | -74.59, -52.51 | 78.18, -12.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8995 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.48, 161.66 | APE9-dihe-na | 136.02, -164.27 | APE8-dihe-in | -134.21, 135.25 | APE8-rot-in | 295.47 | APE67-dihe-in | -61.9, -23.15 | -53.94, -45.84 | APE12-dist-in | 7.4385 | APE11-dist-in | 10.5331 | APE10-dist-in | 4.8932 | APE9-dist-in | 3.5664 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.379 | 0.135 | 0.162 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvn | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1H1WA | O15530 | 71 | 359 | 556.0 | ATP:1373 | ATPlike | Inactive | DFGin | 6.6116 | 14.931 | BLAminus | -145.26, -169.97 | 71.92, 72.18 | -105.82, -0.04 | 289.27, 102.08 | -58.33, -31.92 | in-in | in | 8.5808 | Saltbr-in | 2.7103 | HRD-in | -71.45, -48.32 | 74.08, -8.04 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8395 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.69, 112.94 | APE9-dihe-na | -63.98, -168.66 | APE8-dihe-in | -54.13, 124.0 | APE8-rot-in | 301.59 | APE67-dihe-in | -62.54, -19.03 | -38.83, -50.46 | APE12-dist-in | 8.922 | APE11-dist-out | 5.528 | APE10-dist-out | 10.2978 | APE9-dist-in | 3.7994 | None | SEP241 | SEP241 | XRAY | 2.0 | 0.196 | 0.223 | A | 289.0 | 285.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 1h1w | AGC_PDPK1_HUMAN | AGC | 9.8e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXA | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.5961 | 14.1691 | BLAminus | -138.52, -175.65 | 62.9, 74.02 | -93.7, 13.51 | 275.9, 89.61 | -62.84, -23.94 | in-in | in | 8.8135 | Saltbr-in | 2.5558 | HRD-in | -68.79, -51.77 | 77.65, -2.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8365 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -110.22, 106.38 | APE9-dihe-na | -61.01, -163.77 | APE8-dihe-in | -59.2, 130.87 | APE8-rot-in | 313.64 | APE67-dihe-in | -68.86, -21.58 | -48.76, -40.32 | APE12-dist-in | 9.226 | APE11-dist-out | 5.7837 | APE10-dist-out | 10.5309 | APE9-dist-in | 3.9835 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | A | 316.0 | 284.0 | 1 | 30 | 29 | 1 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXB | O15530 | 77 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.6597 | 14.1548 | BLAminus | -140.69, -175.67 | 59.43, 71.11 | -92.21, 14.29 | 279.78, 86.28 | -63.72, -16.63 | in-in | in | 8.802 | Saltbr-in | 2.5641 | HRD-in | -68.32, -50.05 | 78.21, -3.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8222 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -111.03, 106.62 | APE9-dihe-na | -60.26, -162.55 | APE8-dihe-in | -59.71, 131.44 | APE8-rot-in | 313.93 | APE67-dihe-in | -67.3, -21.72 | -51.61, -39.66 | APE12-dist-in | 9.2384 | APE11-dist-out | 5.8005 | APE10-dist-out | 10.5524 | APE9-dist-in | 3.9081 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | B | 316.0 | 281.0 | 2 | 30 | 28 | 2 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXC | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.6298 | 14.0961 | BLAminus | -135.92, -176.39 | 63.79, 71.64 | -93.36, 13.73 | 280.67, 86.49 | -62.67, -20.94 | in-in | in | 8.7824 | Saltbr-in | 2.5509 | HRD-in | -66.06, -52.0 | 76.42, -2.2 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8354 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -110.22, 106.64 | APE9-dihe-na | -60.77, -161.89 | APE8-dihe-in | -59.91, 131.8 | APE8-rot-in | 311.89 | APE67-dihe-in | -63.47, -22.82 | -49.61, -43.91 | APE12-dist-in | 9.1653 | APE11-dist-out | 5.8015 | APE10-dist-out | 10.55 | APE9-dist-in | 3.9841 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | C | 316.0 | 284.0 | 1 | 30 | 29 | 1 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXD | O15530 | 76 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.5711 | 14.146 | BLAminus | -134.45, -170.09 | 60.8, 71.91 | -91.57, 12.91 | 278.05, 86.51 | -67.5, -17.43 | in-in | in | 8.7987 | Saltbr-in | 2.5834 | HRD-in | -66.01, -50.34 | 77.25, -1.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8418 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -110.2, 105.71 | APE9-dihe-na | -59.39, -160.44 | APE8-dihe-in | -60.94, 132.03 | APE8-rot-in | 313.43 | APE67-dihe-in | -67.95, -22.9 | -52.31, -39.76 | APE12-dist-in | 9.2273 | APE11-dist-out | 5.7904 | APE10-dist-out | 10.5469 | APE9-dist-in | 3.9121 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | D | 316.0 | 283.0 | 1 | 30 | 29 | 1 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXE | O15530 | 76 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.3816 | 14.9206 | BLAminus | -125.38, -158.75 | 61.49, 56.01 | -85.03, 10.36 | 279.31, 82.03 | -55.13, -32.27 | in-in | in | 9.2368 | Saltbr-in | 3.2715 | HRD-in | -67.18, -49.37 | 73.61, -2.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9678 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nooi | APE10-dihe-na | -112.75, 120.85 | APE9-dihe-na | -80.18, -170.48 | APE8-dihe-in | -52.91, 130.32 | APE8-rot-in | 309.26 | APE67-dihe-in | -61.57, -27.92 | -56.84, -38.07 | APE12-dist-none | 999.0 | APE11-dist-out | 5.4882 | APE10-dist-out | 10.2693 | APE9-dist-in | 4.4822 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | E | 316.0 | 274.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXF | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.3677 | 14.9155 | BLAminus | -124.96, -165.04 | 64.25, 56.63 | -90.23, 13.81 | 273.61, 91.31 | -58.82, -32.5 | in-none | in | 9.2317 | Saltbr-none | 999.0 | HRD-in | -66.95, -49.19 | 76.54, -9.89 | none-in-out | SNCnio | in-out | ActLoopNT-in | 2.9816 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -112.23, 117.01 | APE9-dihe-na | -74.75, -174.06 | APE8-dihe-in | -40.45, 117.92 | APE8-rot-in | 309.94 | APE67-dihe-in | -62.78, -29.13 | -41.21, -44.42 | APE12-dist-in | 8.1177 | APE11-dist-out | 5.4885 | APE10-dist-out | 10.2748 | APE9-dist-in | 4.4634 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | F | 316.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXG | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.4182 | 15.1625 | BLAminus | -124.35, -160.11 | 59.71, 58.4 | -85.01, 8.33 | 270.63, 86.47 | -58.24, -35.05 | in-in | in | 9.2322 | Saltbr-in | 3.2566 | HRD-in | -66.57, -49.64 | 76.01, -6.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0259 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -113.59, 119.71 | APE9-dihe-na | -80.06, -167.69 | APE8-dihe-in | -52.92, 132.86 | APE8-rot-in | 313.01 | APE67-dihe-in | -62.53, -35.87 | -56.69, -38.23 | APE12-dist-in | 8.4931 | APE11-dist-out | 5.4816 | APE10-dist-out | 10.2289 | APE9-dist-in | 4.3614 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | G | 316.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORXH | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.4702 | 14.8365 | BLAminus | -123.34, -162.32 | 62.45, 60.25 | -89.76, 14.7 | 283.48, 85.4 | -55.85, -32.26 | in-in | in | 9.2345 | Saltbr-in | 3.2833 | HRD-in | -67.42, -48.8 | 75.62, -9.07 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9802 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -112.9, 122.93 | APE9-dihe-na | -81.65, -170.32 | APE8-dihe-in | -53.77, 133.41 | APE8-rot-in | 303.61 | APE67-dihe-in | -61.23, -30.63 | -57.13, -39.02 | APE12-dist-in | 8.3784 | APE11-dist-out | 5.4961 | APE10-dist-out | 10.1982 | APE9-dist-in | 4.4177 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | H | 316.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORZA | O15530 | 74 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6225 | 14.6052 | BLAminus | -134.96, -167.36 | 70.2, 66.13 | -101.26, 0.99 | 293.7, 88.7 | -61.05, -29.24 | in-in | in | 8.2152 | Saltbr-in | 2.8103 | HRD-in | -65.12, -49.46 | 75.7, -10.07 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8327 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -134.38, 111.86 | APE9-dihe-na | -60.27, -174.97 | APE8-dihe-in | -55.74, 132.42 | APE8-rot-in | 303.15 | APE67-dihe-in | -56.98, -32.17 | -55.27, -42.37 | APE12-dist-in | 11.5493 | APE11-dist-out | 6.544 | APE10-dist-out | 10.866 | APE9-dist-in | 4.1173 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | A | 316.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3orz | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORZB | O15530 | 73 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6476 | 14.7764 | BLAminus | -139.38, -168.66 | 74.13, 69.92 | -111.18, 3.04 | 284.6, 93.64 | -63.39, -24.83 | in-in | in | 8.2923 | Saltbr-in | 2.7592 | HRD-in | -64.66, -48.81 | 76.86, -10.42 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8659 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.43, 114.97 | APE9-dihe-na | -62.67, -167.65 | APE8-dihe-in | -63.67, 131.38 | APE8-rot-in | 299.84 | APE67-dihe-in | -54.64, -32.97 | -56.45, -39.98 | APE12-dist-in | 11.638 | APE11-dist-out | 6.3971 | APE10-dist-out | 10.7873 | APE9-dist-in | 4.0869 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | B | 316.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3orz | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORZC | O15530 | 74 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6668 | 14.6791 | BLAminus | -134.07, -170.51 | 76.79, 69.39 | -110.34, 1.38 | 287.93, 89.81 | -56.71, -30.43 | in-in | in | 8.2245 | Saltbr-in | 2.8037 | HRD-in | -64.4, -49.76 | 78.61, -9.94 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8049 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -134.53, 111.0 | APE9-dihe-na | -58.83, -174.56 | APE8-dihe-in | -56.66, 132.63 | APE8-rot-in | 302.29 | APE67-dihe-in | -56.84, -32.58 | -55.43, -42.03 | APE12-dist-in | 11.7307 | APE11-dist-out | 6.55 | APE10-dist-out | 10.875 | APE9-dist-in | 4.0824 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | C | 316.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3orz | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3ORZD | O15530 | 73 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6487 | 14.7735 | BLAminus | -139.63, -168.42 | 74.39, 69.06 | -110.33, 3.29 | 285.32, 93.06 | -63.48, -24.84 | in-in | in | 8.3101 | Saltbr-in | 2.754 | HRD-in | -64.65, -47.43 | 73.97, -9.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8768 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -126.78, 121.12 | APE9-dihe-na | -63.33, -166.44 | APE8-dihe-in | -63.66, 131.18 | APE8-rot-in | 301.29 | APE67-dihe-in | -54.43, -33.46 | -55.31, -40.36 | APE12-dist-in | 11.5839 | APE11-dist-out | 6.4058 | APE10-dist-out | 10.8417 | APE9-dist-in | 4.0404 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | D | 316.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3orz | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1Z5MA | O15530 | 74 | 359 | 556.0 | LI8:501 | Type1 | Inactive | DFGin | 6.9657 | 14.6691 | BLAminus | -143.06, -166.04 | 70.1, 70.4 | -106.54, 10.63 | 285.55, 95.37 | -57.95, -38.82 | in-in | in | 8.979 | Saltbr-in | 2.8616 | HRD-in | -60.53, -42.76 | 63.99, 3.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.6826 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -142.8, 123.87 | APE9-dihe-na | -69.98, -168.75 | APE8-dihe-in | -47.59, 126.16 | APE8-rot-in | 298.44 | APE67-dihe-in | -75.58, -18.39 | -37.0, -46.81 | APE12-dist-in | 8.5442 | APE11-dist-out | 6.2855 | APE10-dist-out | 10.4569 | APE9-dist-in | 4.0502 | None | SEP241 | SEP241 | XRAY | 2.17 | 0.232 | 0.269 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 1z5m | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 2PE0A | O15530 | 74 | 359 | 556.0 | 39Z:501 | Type1 | Inactive | DFGin | 6.4474 | 14.3844 | BLAminus | -129.98, -179.46 | 78.75, 74.81 | -106.99, 5.13 | 286.59, 90.93 | -55.7, -29.7 | in-in | in | 8.7227 | Saltbr-in | 2.7831 | HRD-in | -72.01, -55.71 | 78.26, -0.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8174 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -117.01, 133.16 | APE9-dihe-na | -80.12, -143.18 | APE8-dihe-in | -90.02, 137.86 | APE8-rot-in | 307.83 | APE67-dihe-in | -64.54, -15.21 | -51.36, -49.75 | APE12-dist-in | 9.1401 | APE11-dist-out | 5.5127 | APE10-dist-out | 10.1028 | APE9-dist-in | 3.7888 | None | SEP241 | SEP241 | XRAY | 2.35 | 0.202 | 0.24 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2pe0 | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 2PE1A | O15530 | 74 | 359 | 556.0 | 517:501 | Type1 | Inactive | DFGin | 6.6447 | 14.6824 | BLAminus | -139.4, -175.86 | 73.15, 71.4 | -105.21, 7.65 | 286.89, 93.63 | -52.89, -40.97 | in-in | in | 8.8829 | Saltbr-in | 2.5948 | HRD-in | -69.74, -56.95 | 81.13, 2.35 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8564 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -114.84, 143.11 | APE9-dihe-na | -79.47, -134.7 | APE8-dihe-in | -90.68, 136.03 | APE8-rot-in | 300.98 | APE67-dihe-in | -68.92, -11.38 | -43.74, -52.34 | APE12-dist-in | 9.1167 | APE11-dist-out | 5.7014 | APE10-dist-out | 10.3798 | APE9-dist-in | 3.6055 | None | SEP241 | SEP241 | XRAY | 2.14 | 0.224 | 0.282 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2pe1 | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 2PE2A | O15530 | 74 | 359 | 556.0 | 464:501 | Type1 | Inactive | DFGin | 6.5908 | 14.4155 | BLAminus | -135.75, -175.91 | 78.63, 72.01 | -109.62, 0.43 | 287.28, 93.19 | -54.2, -35.84 | in-in | in | 8.5622 | Saltbr-in | 2.5509 | HRD-in | -75.76, -49.83 | 75.8, -8.69 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7244 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.61, 128.36 | APE9-dihe-na | -70.67, -166.57 | APE8-dihe-in | -59.34, 134.44 | APE8-rot-in | 302.45 | APE67-dihe-in | -67.69, -11.47 | -51.51, -47.62 | APE12-dist-in | 8.9817 | APE11-dist-out | 5.5266 | APE10-dist-out | 10.3125 | APE9-dist-in | 3.7381 | None | SEP241 | SEP241 | XRAY | 2.13 | 0.189 | 0.215 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2pe2 | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NUSA | O15530 | 73 | 358 | 556.0 | JNZ:374 | Type1 | Inactive | DFGin | 6.6661 | 14.0143 | BLAminus | -134.94, -176.79 | 67.79, 79.24 | -106.97, 14.51 | 293.69, 91.17 | -56.65, -43.75 | in-in | in | 8.6145 | Saltbr-in | 3.1048 | HRD-in | -75.65, -54.6 | 82.78, -6.2 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8741 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -129.47, 126.95 | APE9-dihe-na | -67.17, -145.64 | APE8-dihe-in | -85.86, 130.62 | APE8-rot-in | 299.93 | APE67-dihe-in | -70.26, -18.43 | -47.43, -45.34 | APE12-dist-in | 9.4758 | APE11-dist-out | 6.257 | APE10-dist-out | 10.2994 | APE9-dist-in | 4.0295 | None | SEP241 | SEP241 | XRAY | 2.75 | 0.177 | 0.236 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nus | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NUUA | O15530 | 73 | 358 | 556.0 | JOZ:361 | Type1 | Inactive | DFGin | 6.8153 | 14.418 | BLAminus | -135.1, 176.45 | 77.67, 76.35 | -106.62, 4.54 | 289.58, 95.96 | -54.87, -35.17 | in-in | in | 8.6632 | Saltbr-in | 2.6457 | HRD-in | -75.97, -55.36 | 84.01, -8.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8245 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -123.64, 126.08 | APE9-dihe-na | -69.19, -150.37 | APE8-dihe-in | -79.82, 127.26 | APE8-rot-in | 298.22 | APE67-dihe-in | -66.17, -14.72 | -39.18, -51.46 | APE12-dist-in | 8.929 | APE11-dist-out | 5.8492 | APE10-dist-out | 10.298 | APE9-dist-in | 3.9915 | None | SEP241 | SEP241 | XRAY | 1.98 | 0.189 | 0.239 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nuu | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NUYA | O15530 | 73 | 358 | 556.0 | JPZ:370 | Type1 | Inactive | DFGin | 6.7298 | 14.5499 | BLAminus | -136.81, -175.62 | 72.08, 77.54 | -106.37, 8.07 | 285.95, 95.42 | -50.93, -42.82 | in-in | in | 8.7638 | Saltbr-in | 2.731 | HRD-in | -78.09, -53.76 | 79.66, -9.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8966 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.52, 118.04 | APE9-dihe-na | -67.36, -159.8 | APE8-dihe-in | -67.79, 132.38 | APE8-rot-in | 304.86 | APE67-dihe-in | -62.4, -17.72 | -54.87, -44.81 | APE12-dist-in | 9.4109 | APE11-dist-out | 5.8201 | APE10-dist-out | 10.2784 | APE9-dist-in | 3.9709 | None | SEP241 | SEP241 | XRAY | 2.1 | 0.187 | 0.225 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nuy | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1UU9A | O15530 | 72 | 357 | 556.0 | BI3:1370 | Type1 | Inactive | DFGin | 6.6788 | 14.783 | BLAminus | -137.61, -169.2 | 68.82, 72.55 | -103.82, -0.34 | 285.88, 98.86 | -59.49, -32.23 | in-in | in | 8.3257 | Saltbr-in | 2.6975 | HRD-in | -73.71, -52.28 | 77.02, -6.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8778 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.15, 123.88 | APE9-dihe-na | -73.46, -162.02 | APE8-dihe-in | -55.23, 126.59 | APE8-rot-in | 305.35 | APE67-dihe-in | -59.52, -20.56 | -41.52, -52.97 | APE12-dist-in | 9.3386 | APE11-dist-out | 5.5023 | APE10-dist-out | 10.2727 | APE9-dist-in | 3.7767 | None | SEP241 | SEP241 | XRAY | 1.95 | 0.176 | 0.224 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 1uu9 | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1UVRA | O15530 | 71 | 359 | 556.0 | BI8:1372 | Type1 | Inactive | DFGin | 6.5811 | 14.4064 | BLAminus | -141.7, -169.27 | 62.75, 72.58 | -105.41, 8.55 | 300.9, 81.55 | -59.95, -35.71 | in-in | in | 8.5947 | Saltbr-in | 2.9835 | HRD-in | -62.43, -49.82 | 76.81, -6.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9337 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -133.17, 120.18 | APE9-dihe-na | -60.87, -168.42 | APE8-dihe-in | -53.67, 135.35 | APE8-rot-in | 308.99 | APE67-dihe-in | -63.6, -1.85 | -44.81, -56.98 | APE12-dist-in | 7.2881 | APE11-dist-out | 6.6429 | APE10-dist-out | 10.6143 | APE9-dist-in | 4.0897 | None | SEP241 | SEP241 | XRAY | 2.81 | 0.176 | 0.248 | A | 289.0 | 285.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 1uvr | AGC_PDPK1_HUMAN | AGC | 9.8e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NUNA | O15530 | 71 | 358 | 556.0 | JMZ:361 | Type1 | Inactive | DFGin | 6.4722 | 14.2209 | BLAminus | -136.64, 178.66 | 75.33, 84.73 | -114.4, 16.28 | 293.69, 90.85 | -60.42, -36.06 | in-in | in | 8.6724 | Saltbr-in | 2.7874 | HRD-in | -68.71, -51.25 | 77.84, -3.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8357 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -115.38, 127.64 | APE9-dihe-na | -69.91, -151.05 | APE8-dihe-in | -80.37, 125.09 | APE8-rot-in | 310.77 | APE67-dihe-in | -66.15, -18.43 | -42.77, -46.09 | APE12-dist-in | 8.9686 | APE11-dist-out | 5.8965 | APE10-dist-out | 10.4173 | APE9-dist-in | 4.3142 | None | SEP241 | SEP241 | XRAY | 2.2 | 0.18 | 0.227 | A | 292.0 | 279.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nun | AGC_PDPK1_HUMAN | AGC | 1e-84 | 289.6 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 2XCHA | O15530 | 73 | 359 | 556.0 | CKG:1360 | Type1 | Inactive | DFGin | 6.7339 | 14.5287 | BLAminus | -129.58, 177.2 | 73.14, 77.15 | -102.2, 9.9 | 285.13, 96.86 | -57.37, -39.89 | in-in | in | 8.6981 | Saltbr-in | 2.571 | HRD-in | -76.48, -53.27 | 78.53, -7.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.893 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -122.55, 124.18 | APE9-dihe-na | -77.48, -153.81 | APE8-dihe-in | -63.6, 127.96 | APE8-rot-in | 306.17 | APE67-dihe-in | -61.93, -18.13 | -48.28, -49.39 | APE12-dist-in | 9.2863 | APE11-dist-out | 5.6905 | APE10-dist-out | 10.3423 | APE9-dist-in | 3.8907 | None | SEP241 | SEP241 | XRAY | 2.0 | 0.191 | 0.226 | A | 309.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 2xch | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5HKMA | O15530 | 76 | 358 | 556.0 | 61Y:403 | Type1 | Inactive | DFGin | 6.428 | 14.1502 | BLAminus | -122.57, -157.08 | 51.69, 73.85 | -100.67, 14.09 | 281.12, 81.43 | -62.59, -33.63 | in-in | in | 8.6492 | Saltbr-in | 2.8074 | HRD-in | -66.63, -45.86 | 63.42, -2.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7614 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -140.98, 122.73 | APE9-dihe-na | -75.89, -160.0 | APE8-dihe-in | -62.57, 122.86 | APE8-rot-in | 309.65 | APE67-dihe-in | -56.46, -24.28 | -29.66, -64.05 | APE12-dist-in | 9.6471 | APE11-dist-out | 5.8023 | APE10-dist-out | 10.2714 | APE9-dist-in | 3.7976 | None | SEP241 | SEP241 | XRAY | 2.1 | 0.228 | 0.273 | A | 309.0 | 273.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 5hkm | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5HNGA | O15530 | 71 | 359 | 556.0 | 62O:403 | Type1 | Inactive | DFGin | 6.5015 | 14.356 | BLAminus | -131.37, -170.36 | 61.15, 71.88 | -92.77, 10.44 | 287.92, 92.83 | -55.25, -43.3 | in-in | in | 8.828 | Saltbr-in | 2.8729 | HRD-in | -61.06, -47.37 | 70.67, -1.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7991 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -117.82, 119.15 | APE9-dihe-na | -68.32, -153.72 | APE8-dihe-in | -67.95, 131.45 | APE8-rot-in | 305.81 | APE67-dihe-in | -63.0, -22.16 | -48.07, -47.57 | APE12-dist-in | 9.0259 | APE11-dist-out | 5.7457 | APE10-dist-out | 10.5212 | APE9-dist-in | 4.0322 | None | SEP241 | SEP241 | XRAY | 3.01 | 0.176 | 0.243 | A | 309.0 | 281.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 5hng | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5HO7A | O15530 | 71 | 359 | 556.0 | 63L:701 | Type1 | Inactive | DFGin | 6.4996 | 13.9982 | BLAminus | -138.45, -177.98 | 79.97, 72.22 | -103.24, 8.72 | 293.52, 91.58 | -60.99, -44.96 | in-in | in | 8.5843 | Saltbr-in | 3.0686 | HRD-in | -62.96, -39.76 | 64.33, -4.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9376 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -122.91, 120.25 | APE9-dihe-na | -71.94, -150.13 | APE8-dihe-in | -74.96, 128.19 | APE8-rot-in | 303.71 | APE67-dihe-in | -61.52, -27.36 | -46.49, -48.45 | APE12-dist-in | 9.4591 | APE11-dist-out | 6.0158 | APE10-dist-out | 10.3175 | APE9-dist-in | 4.1229 | None | SEP241 | SEP241 | XRAY | 3.0 | 0.175 | 0.233 | A | 309.0 | 281.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 5ho7 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 5HO8A | O15530 | 71 | 358 | 556.0 | 63E:701 | Type1 | Inactive | DFGin | 6.3257 | 13.7271 | BLAminus | -137.78, 179.62 | 80.28, 69.7 | -100.25, 11.3 | 296.62, 94.66 | -58.72, -47.18 | in-in | in | 8.7434 | Saltbr-in | 3.0233 | HRD-in | -65.39, -42.86 | 64.55, -6.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8667 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -124.41, 121.86 | APE9-dihe-na | -70.34, -152.74 | APE8-dihe-in | -66.74, 122.4 | APE8-rot-in | 293.45 | APE67-dihe-in | -65.08, -24.35 | -41.28, -45.91 | APE12-dist-in | 9.1451 | APE11-dist-out | 5.9265 | APE10-dist-out | 10.2379 | APE9-dist-in | 4.0594 | None | SEP241 | SEP241 | XRAY | 2.7 | 0.184 | 0.229 | A | 309.0 | 279.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5ho8 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1OKYA | O15530 | 72 | 360 | 556.0 | STU:1368 | Type1 | Inactive | DFGin | 6.1532 | 14.4616 | BLAminus | -148.97, -170.84 | 70.56, 80.45 | -102.75, 23.82 | 286.84, 96.04 | -69.28, -20.21 | in-in | in | 8.6718 | Saltbr-in | 2.6729 | HRD-in | -67.69, -57.78 | 80.28, 0.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9341 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -113.7, -80.59 | APE9-dihe-na | 115.49, 169.91 | APE8-dihe-in | -54.49, 123.73 | APE8-rot-in | 316.76 | APE67-dihe-in | -63.35, -17.55 | -42.07, -50.54 | APE12-dist-in | 9.2892 | APE11-dist-out | 5.5558 | APE10-dist-out | 9.7186 | APE9-dist-in | 4.222 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.219 | 0.255 | A | 310.0 | 283.0 | 6 | 30 | 24 | 6 | [[82, 342]] | 1.0 | 1oky | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1OKZA | O15530 | 73 | 359 | 556.0 | UCN:1370 | Type1 | Inactive | DFGin | 6.5441 | 14.1675 | BLAminus | -141.57, -164.78 | 67.55, 76.85 | -103.78, 11.05 | 287.85, 85.4 | -63.67, 2.06 | in-in | in | 8.7271 | Saltbr-in | 2.7175 | HRD-in | -70.44, -54.0 | 75.32, 3.69 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9208 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -147.16, 105.01 | APE9-dihe-na | -62.12, -140.62 | APE8-dihe-in | -78.85, 125.76 | APE8-rot-in | 304.75 | APE67-dihe-in | -63.07, -21.46 | -38.09, -52.99 | APE12-dist-in | 9.5567 | APE11-dist-out | 6.099 | APE10-dist-out | 10.4075 | APE9-dist-in | 4.1656 | None | SEP241 | SEP241 | XRAY | 2.51 | 0.19 | 0.257 | A | 310.0 | 278.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 1okz | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1UU3A | O15530 | 73 | 360 | 556.0 | LY4:1374 | Type1 | Inactive | DFGin | 6.5956 | 14.9714 | BLAminus | -134.47, -173.45 | 74.38, 73.99 | -109.66, 0.57 | 283.46, 101.61 | -63.98, -27.2 | in-in | in | 8.2752 | Saltbr-in | 2.8167 | HRD-in | -64.65, -55.05 | 74.86, -6.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8643 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -122.92, 125.5 | APE9-dihe-na | -77.61, -163.62 | APE8-dihe-in | -56.98, 127.76 | APE8-rot-in | 299.91 | APE67-dihe-in | -61.39, -22.49 | -53.63, -41.57 | APE12-dist-in | 9.2019 | APE11-dist-out | 5.4661 | APE10-dist-out | 10.4073 | APE9-dist-in | 4.0483 | None | SEP241 | SEP241 | XRAY | 1.7 | 0.174 | 0.202 | A | 310.0 | 278.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 1uu3 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1UU7A | O15530 | 73 | 359 | 556.0 | BI2:1364 | Type1 | Inactive | DFGin | 6.5571 | 14.7415 | BLAminus | -136.5, -171.94 | 74.29, 73.79 | -109.8, -2.64 | 287.37, 96.13 | -53.85, -39.14 | in-in | in | 8.463 | Saltbr-in | 2.8801 | HRD-in | -68.07, -51.28 | 73.99, -8.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8332 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.82, 121.67 | APE9-dihe-na | -67.64, -173.23 | APE8-dihe-in | -49.06, 125.05 | APE8-rot-in | 301.64 | APE67-dihe-in | -67.12, -19.88 | -49.14, -41.33 | APE12-dist-in | 8.9136 | APE11-dist-out | 5.317 | APE10-dist-out | 10.2667 | APE9-dist-in | 3.9105 | None | SEP241 | SEP241 | XRAY | 1.9 | 0.235 | 0.279 | A | 310.0 | 282.0 | 5 | 30 | 25 | 5 | [[82, 342]] | 1.0 | 1uu7 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 1UU8A | O15530 | 72 | 358 | 556.0 | BI1:1368 | Type1 | Inactive | DFGin | 6.6469 | 14.4714 | BLAminus | -136.37, -165.37 | 63.01, 71.98 | -101.9, 2.54 | 288.65, 101.81 | -58.08, -33.97 | in-in | in | 8.8152 | Saltbr-in | 2.7275 | HRD-in | -71.97, -53.07 | 75.47, 11.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8428 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -142.67, 117.85 | APE9-dihe-na | -65.71, -160.29 | APE8-dihe-in | -63.31, 129.15 | APE8-rot-in | 297.13 | APE67-dihe-in | -68.38, -3.88 | -40.88, -48.91 | APE12-dist-in | 9.2375 | APE11-dist-out | 5.6529 | APE10-dist-out | 10.0877 | APE9-dist-in | 3.759 | None | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.258 | A | 310.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 1uu8 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NAYA | O15530 | 76 | 362 | 556.0 | MP6:1 | Type1 | Inactive | DFGin | 6.7641 | 14.6579 | BLAminus | -146.79, -173.04 | 72.2, 70.67 | -103.69, 5.05 | 296.95, 109.64 | -60.79, -27.91 | in-in | in | 8.5567 | Saltbr-in | 2.5649 | HRD-in | -62.07, -50.65 | 74.17, -9.68 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.74 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -127.84, 118.23 | APE9-dihe-na | -69.99, -167.96 | APE8-dihe-in | -54.98, 129.37 | APE8-rot-in | 302.57 | APE67-dihe-in | -65.83, -27.98 | -54.2, -37.6 | APE12-dist-in | 8.6002 | APE11-dist-out | 5.6186 | APE10-dist-out | 10.5309 | APE9-dist-in | 3.8392 | None | SEP241 | SEP241 | XRAY | 2.6 | 0.211 | 0.274 | A | 311.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3nay | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NAYB | O15530 | 76 | 362 | 556.0 | MP6:2 | Type1 | Inactive | DFGin | 6.8794 | 14.3665 | BLAminus | -131.67, -178.35 | 72.0, 77.09 | -107.77, 17.41 | 299.66, 102.49 | -69.46, -28.42 | in-in | in | 8.3299 | Saltbr-in | 2.8238 | HRD-in | -70.5, -49.88 | 76.39, -13.79 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8417 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 114.84, 100.21 | APE9-dihe-na | -68.09, -163.03 | APE8-dihe-in | -59.66, 125.08 | APE8-rot-in | 300.78 | APE67-dihe-in | -68.69, -23.52 | -42.99, -40.54 | APE12-dist-in | 8.7294 | APE11-dist-out | 5.8365 | APE10-dist-out | 10.6017 | APE9-dist-in | 3.8844 | None | SEP241 | SEP241 | XRAY | 2.6 | 0.211 | 0.274 | B | 311.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3nay | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3RWPA | O15530 | 73 | 359 | 556.0 | ABQ:360 | Type1 | Inactive | DFGin | 6.6301 | 14.6122 | BLAminus | -138.06, -171.84 | 73.21, 68.9 | -101.84, 0.77 | 284.24, 99.91 | -67.12, -24.97 | in-in | in | 8.4872 | Saltbr-in | 2.668 | HRD-in | -72.19, -48.95 | 75.52, -7.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8439 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -116.4, 122.62 | APE9-dihe-na | -64.5, -165.33 | APE8-dihe-in | -62.97, 132.8 | APE8-rot-in | 302.69 | APE67-dihe-in | -57.73, -26.43 | -57.73, -39.86 | APE12-dist-in | 9.571 | APE11-dist-out | 5.748 | APE10-dist-out | 10.613 | APE9-dist-in | 4.2017 | None | SEP241 | SEP241 | XRAY | 1.92 | 0.174 | 0.213 | A | 311.0 | 278.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3rwp | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3RWQA | O15530 | 72 | 359 | 556.0 | 3RW:1 | Type1 | Inactive | DFGin | 6.5891 | 14.463 | BLAminus | -143.65, -172.61 | 68.52, 70.31 | -102.07, 3.38 | 289.03, 95.5 | -56.64, -39.2 | in-in | in | 8.5646 | Saltbr-in | 2.7282 | HRD-in | -70.4, -52.28 | 81.8, -9.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.02 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -127.88, 122.18 | APE9-dihe-na | -69.74, -149.03 | APE8-dihe-in | -75.72, 125.93 | APE8-rot-in | 318.02 | APE67-dihe-in | -73.55, -21.89 | -37.75, -44.68 | APE12-dist-in | 9.2067 | APE11-dist-out | 5.8786 | APE10-dist-out | 10.5237 | APE9-dist-in | 4.0165 | None | SEP241 | SEP241 | XRAY | 2.55 | 0.196 | 0.256 | A | 311.0 | 284.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 3rwq | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3H9OA | O15530 | 75 | 359 | 556.0 | 9BD:1 | Type1 | Inactive | DFGin | 6.5678 | 14.261 | BLAminus | -131.94, -168.71 | 66.62, 79.57 | -104.6, 18.2 | 283.3, 82.81 | -72.27, -11.03 | in-in | in | 8.8763 | Saltbr-in | 2.5436 | HRD-in | -78.26, -52.42 | 80.3, -1.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8097 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 77.5, 119.89 | APE9-dihe-na | -89.12, -112.65 | APE8-dihe-in | -101.23, 134.92 | APE8-rot-in | 301.13 | APE67-dihe-in | -62.27, -18.27 | -50.83, -50.03 | APE12-dist-in | 9.6432 | APE11-dist-out | 6.2678 | APE10-dist-out | 10.1736 | APE9-dist-in | 3.934 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.211 | 0.256 | A | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3h9o | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 2R7BA | O15530 | 75 | 359 | 556.0 | 253:701 | Type1 | Inactive | DFGin | 6.1992 | 14.366 | BLAminus | -133.94, -179.49 | 77.82, 81.49 | -108.24, 22.02 | 291.13, 86.98 | -68.69, -10.97 | in-in | in | 8.8662 | Saltbr-in | 2.5883 | HRD-in | -75.75, -47.44 | 52.14, 30.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7982 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 148.51, 113.35 | APE9-dihe-na | -77.58, -157.1 | APE8-dihe-in | -58.21, 135.29 | APE8-rot-in | 301.99 | APE67-dihe-in | -57.75, -20.67 | -44.89, -55.44 | APE12-dist-in | 9.1968 | APE11-dist-out | 5.7727 | APE10-dist-out | 9.8875 | APE9-dist-in | 4.0959 | None | SEP241 | SEP241 | XRAY | 2.7 | 0.225 | 0.25 | A | 312.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2r7b | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3IONA | O15530 | 75 | 359 | 556.0 | 8H1:1 | Type1 | Inactive | DFGin | 6.3855 | 14.0119 | BLAminus | -129.57, -169.56 | 64.12, 80.16 | -106.23, 22.91 | 285.85, 87.72 | -68.81, -24.37 | in-in | in | 8.9313 | Saltbr-in | 3.3369 | HRD-in | -74.01, -54.84 | 77.47, 1.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7001 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoi | APE10-dihe-na | 999.0, 132.89 | APE9-dihe-na | -88.46, -116.13 | APE8-dihe-in | -104.9, 134.52 | APE8-rot-in | 307.56 | APE67-dihe-in | -73.92, -18.65 | -45.98, -45.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 10.0803 | APE9-dist-in | 3.6029 | None | None | None | XRAY | 2.4 | 0.246 | 0.282 | A | 312.0 | 274.0 | 11 | 30 | 19 | 11 | [[82, 342]] | 1.0 | 3ion | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3IOPA | O15530 | 75 | 359 | 556.0 | 8I1:1 | Type1 | Inactive | DFGin | 6.6057 | 14.3164 | BLAminus | -125.3, -165.97 | 58.12, 80.1 | -105.24, 23.38 | 285.73, 86.81 | -73.19, -11.32 | in-in | in | 8.8064 | Saltbr-in | 2.6809 | HRD-in | -71.7, -52.98 | 78.46, -5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8075 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 67.02, 113.91 | APE9-dihe-na | -74.5, -127.28 | APE8-dihe-in | -97.61, 129.5 | APE8-rot-in | 303.0 | APE67-dihe-in | -63.74, -18.61 | -44.16, -50.92 | APE12-dist-in | 9.5697 | APE11-dist-out | 5.9687 | APE10-dist-out | 10.4647 | APE9-dist-in | 3.7908 | None | SEP241 | SEP241 | XRAY | 2.2 | 0.24 | 0.278 | A | 312.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3iop | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QCQA | O15530 | 73 | 358 | 556.0 | 3Q0:370 | Type1 | Inactive | DFGin | 6.286 | 13.9428 | BLAminus | -130.07, -172.39 | 67.81, 84.85 | -116.19, 10.14 | 290.92, 91.68 | -60.0, -35.96 | in-in | in | 8.6682 | Saltbr-in | 2.8169 | HRD-in | -76.77, -43.93 | 72.04, -4.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9565 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -127.34, 117.15 | APE9-dihe-na | -68.0, -161.08 | APE8-dihe-in | -59.72, 132.52 | APE8-rot-in | 308.25 | APE67-dihe-in | -73.95, -13.03 | -56.44, -42.24 | APE12-dist-in | 9.3219 | APE11-dist-out | 6.2157 | APE10-dist-out | 10.3256 | APE9-dist-in | 4.2085 | None | SEP241 | SEP241 | XRAY | 2.501 | 0.181 | 0.251 | A | 312.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qcq | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QCSA | O15530 | 73 | 358 | 556.0 | 3Q1:370 | Type1 | Inactive | DFGin | 6.4977 | 14.3423 | BLAminus | -129.15, -172.55 | 69.95, 84.25 | -118.54, 4.81 | 283.02, 93.04 | -59.77, -28.42 | in-in | in | 8.591 | Saltbr-in | 2.8075 | HRD-in | -71.62, -47.65 | 74.15, -7.51 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8349 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -125.7, 120.85 | APE9-dihe-na | -72.97, -164.1 | APE8-dihe-in | -54.02, 130.58 | APE8-rot-in | 312.22 | APE67-dihe-in | -61.81, -24.07 | -54.55, -47.19 | APE12-dist-in | 9.2353 | APE11-dist-out | 6.3341 | APE10-dist-out | 10.5363 | APE9-dist-in | 4.4067 | None | SEP241 | SEP241 | XRAY | 2.487 | 0.182 | 0.251 | A | 312.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qcs | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3PWYA | O15530 | 71 | 359 | 556.0 | SYP:1 | Type1 | Inactive | DFGin | 6.477 | 14.4835 | BLAminus | -124.65, -178.35 | 67.96, 96.3 | -130.58, 11.45 | 300.55, 97.42 | -64.93, -31.03 | in-in | in | 8.587 | Saltbr-in | 2.6927 | HRD-in | -58.86, -48.53 | 68.39, -3.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.761 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -116.65, 129.21 | APE9-dihe-na | -78.78, -151.6 | APE8-dihe-in | -77.12, 126.15 | APE8-rot-in | 307.61 | APE67-dihe-in | -78.87, -27.54 | -44.08, -37.51 | APE12-dist-in | 10.3267 | APE11-dist-out | 5.848 | APE10-dist-out | 10.5798 | APE9-dist-in | 3.8548 | E166C,C260S | None | None | XRAY | 3.5 | 0.226 | 0.276 | A | 311.0 | 281.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3pwy | AGC_PDPK1_HUMAN | AGC | 9.5e-84 | 286.4 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 2XCKA | O15530 | 76 | 359 | 556.0 | MH4:1360 | Type1 | Inactive | DFGin | 6.7771 | 14.7278 | BLAminus | -138.18, -175.27 | 71.05, 75.56 | -104.69, 7.11 | 286.41, 101.4 | -56.07, -44.06 | in-in | in | 8.7216 | Saltbr-in | 2.7225 | HRD-in | -74.69, -54.88 | 79.61, -3.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.891 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -108.24, 134.08 | APE9-dihe-na | -87.44, -159.07 | APE8-dihe-in | -56.55, 126.47 | APE8-rot-in | 304.89 | APE67-dihe-in | -62.34, -18.12 | -47.8, -48.47 | APE12-dist-in | 9.3328 | APE11-dist-out | 5.5135 | APE10-dist-out | 10.4019 | APE9-dist-in | 3.8752 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.195 | 0.24 | A | 309.0 | 276.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 2xck | AGC_PDPK1_HUMAN | AGC | 1.8e-83 | 285.5 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QCXA | O15530 | 73 | 358 | 556.0 | 3Q2:370 | Type1.5_Back | Inactive | DFGin | 6.5656 | 14.4479 | BLAminus | -128.85, -170.97 | 71.83, 79.3 | -115.33, 7.3 | 284.13, 92.7 | -60.73, -28.9 | in-in | in | 8.4024 | Saltbr-in | 2.7064 | HRD-in | -68.18, -50.11 | 76.96, -14.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8031 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -135.89, 122.06 | APE9-dihe-na | -67.11, -167.83 | APE8-dihe-in | -62.01, 135.81 | APE8-rot-in | 308.12 | APE67-dihe-in | -61.25, -24.88 | -55.14, -44.7 | APE12-dist-in | 9.4652 | APE11-dist-out | 6.3732 | APE10-dist-out | 10.3227 | APE9-dist-in | 4.269 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.184 | 0.225 | A | 312.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qcx | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QCYA | O15530 | 73 | 358 | 556.0 | 3Q3:371 | Type1.5_Front | Inactive | DFGin | 6.3885 | 14.5918 | BLAminus | -136.93, -173.16 | 70.99, 75.14 | -110.32, 14.26 | 284.13, 86.28 | -62.73, -28.34 | in-in | in | 8.4189 | Saltbr-in | 2.559 | HRD-in | -71.32, -53.51 | 82.01, -8.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.825 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoi | APE10-dihe-na | 999.0, 125.83 | APE9-dihe-na | -76.07, -148.77 | APE8-dihe-in | -79.07, 127.11 | APE8-rot-in | 312.38 | APE67-dihe-in | -58.65, -24.48 | -40.2, -55.49 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 10.317 | APE9-dist-in | 4.4989 | None | SEP241 | SEP241 | XRAY | 2.2 | 0.181 | 0.212 | A | 312.0 | 275.0 | 11 | 30 | 19 | 11 | [[82, 342]] | 1.0 | 3qcy | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QD3A | O15530 | 71 | 358 | 556.0 | 3Q5:360 | Type1.5_Front | Inactive | DFGin | 6.6397 | 14.7756 | BLAminus | -136.15, -173.35 | 75.08, 78.84 | -114.86, 7.79 | 284.21, 92.48 | -60.8, -30.07 | in-in | in | 8.4699 | Saltbr-in | 2.5474 | HRD-in | -69.84, -52.9 | 76.92, -8.58 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8112 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -114.87, 124.76 | APE9-dihe-na | -70.78, -165.19 | APE8-dihe-in | -61.65, 129.32 | APE8-rot-in | 306.27 | APE67-dihe-in | -62.1, -22.78 | -46.86, -49.49 | APE12-dist-in | 8.9916 | APE11-dist-out | 5.7339 | APE10-dist-out | 10.4141 | APE9-dist-in | 4.0376 | None | SEP241 | SEP241 | XRAY | 2.0 | 0.185 | 0.211 | A | 312.0 | 279.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qd3 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3NAXA | O15530 | 76 | 360 | 556.0 | MP7:363 | Type2 | Inactive | DFGout | 15.1303 | 9.5196 | BBAminus | -103.03, 154.8 | -117.91, 140.31 | -115.35, 34.44 | 271.6, 90.85 | 93.28, 8.79 | out-out | out | 17.0845 | Saltbr-out | 10.2575 | HRD-in | -72.23, -50.17 | 78.89, -10.91 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.8524 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.19, -19.08 | 999.0, -56.98 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.75 | 0.166 | 0.195 | A | 311.0 | 278.0 | 7 | 30 | 23 | 7 | [[82, 342]] | 1.0 | 3nax | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QC4A | O15530 | 76 | 359 | 556.0 | MP7:60001 | Type2 | Inactive | DFGout | 15.1445 | 8.4181 | BBAminus | -116.84, 146.54 | -96.89, 143.53 | -123.04, 29.2 | 249.8, 111.12 | 113.47, -5.45 | out-out | out | 19.868 | Saltbr-out | 17.8176 | HRD-in | -79.45, -51.8 | 76.86, -8.13 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.035 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.28, 161.52 | APE9-dihe-na | 127.76, -165.1 | APE8-dihe-in | -132.92, 137.19 | APE8-rot-in | 293.31 | APE67-dihe-in | -63.51, -29.78 | -55.77, -40.56 | APE12-dist-in | 7.6463 | APE11-dist-in | 10.8912 | APE10-dist-in | 5.0977 | APE9-dist-in | 3.6028 | E303A,K304A | SEP241 | SEP241 | XRAY | 1.8 | 0.174 | 0.213 | A | 314.0 | 277.0 | 7 | 30 | 23 | 7 | [[82, 342]] | 1.0 | 3qc4 | AGC_PDPK1_HUMAN | AGC | 5.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QC4B | O15530 | 51 | 359 | 556.0 | MP7:60002 | Type2 | Inactive | DFGout | 15.5034 | 8.2994 | None | -106.7, 145.77 | -96.8, 153.42 | -131.45, 34.1 | 235.15, 115.54 | 107.65, 4.91 | out-out | out | 18.0578 | Saltbr-out | 15.1697 | HRD-in | -74.82, -53.49 | 77.73, -9.15 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9345 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.95, 158.08 | APE9-dihe-na | 130.3, -155.43 | APE8-dihe-in | -143.11, 135.86 | APE8-rot-in | 293.55 | APE67-dihe-in | -66.08, -20.71 | -55.87, -43.65 | APE12-dist-in | 7.6714 | APE11-dist-in | 10.9464 | APE10-dist-in | 5.0678 | APE9-dist-in | 3.5388 | E303A,K304A | SEP241 | SEP241 | XRAY | 1.8 | 0.174 | 0.213 | B | 314.0 | 274.0 | 15 | 30 | 23 | 7 | [[82, 342]] | 1.0 | 3qc4 | AGC_PDPK1_HUMAN | AGC | 5.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 4CT1A | O15530 | 76 | 359 | 556.0 | ATP:500,31S:600 | ATPlike,Allosteric | None | DFGin | 6.6022 | 14.9785 | BLAminus | -141.71, -172.51 | 72.43, 72.08 | -107.06, 8.07 | 284.9, 97.13 | -62.67, -20.12 | in-none | in | 8.1463 | Saltbr-none | 999.0 | HRD-in | -74.62, -54.47 | 79.43, -8.97 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.9992 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -143.29, 160.89 | APE9-dihe-na | 137.85, -171.95 | APE8-dihe-in | -126.26, 129.35 | APE8-rot-in | 296.2 | APE67-dihe-in | -61.08, -24.26 | -47.64, -46.5 | APE12-dist-in | 7.3566 | APE11-dist-in | 10.4885 | APE10-dist-in | 5.0182 | APE9-dist-in | 3.4798 | L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.85 | 0.172 | 0.215 | A | 311.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4ct1 | AGC_PDPK1_HUMAN | AGC | 9.5e-84 | 286.4 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QD0A | O15530 | 73 | 358 | 556.0 | 3Q4:370 | Type1.5_Front | None | DFGin | 6.5836 | 14.7913 | BLAminus | -135.89, -173.14 | 73.55, 73.02 | -106.35, 12.12 | 281.49, 88.39 | -54.84, -35.9 | in-in | in | 8.5258 | Saltbr-in | 2.5731 | HRD-in | -72.98, -50.98 | 74.13, -9.69 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8508 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -154.13 | APE8-dihe-in | -74.4, 123.75 | APE8-rot-in | 309.46 | APE67-dihe-in | -59.36, -28.41 | -43.01, -50.59 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 4.7652 | None | SEP241 | SEP241 | XRAY | 1.99 | 0.191 | 0.231 | A | 312.0 | 274.0 | 12 | 30 | 18 | 12 | [[82, 342]] | 1.0 | 3qd0 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | 3QD4A | O15530 | 71 | 358 | 556.0 | 3Q6:360 | Type1.5_Front | None | DFGin | 6.4034 | 14.6264 | BLAminus | -137.72, -173.39 | 72.99, 75.84 | -110.69, 10.4 | 285.12, 91.81 | -64.41, -29.28 | in-in | in | 8.5579 | Saltbr-in | 2.7898 | HRD-in | -69.09, -51.69 | 76.33, -7.4 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9076 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -153.49 | APE8-dihe-in | -83.46, 122.24 | APE8-rot-in | 298.92 | APE67-dihe-in | -62.96, -22.94 | -34.73, -56.97 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 4.1203 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.199 | 0.244 | A | 312.0 | 276.0 | 12 | 30 | 18 | 12 | [[82, 342]] | 1.0 | 3qd4 | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PDPK1 | PDPK1_HUMAN | 2BIYA | O15530 | 72 | 359 | 556.0 | ATP:1373 | ATPlike | Active | DFGin | 6.6186 | 15.0949 | BLAminus | -141.33, -175.84 | 82.91, 67.67 | -104.99, 1.58 | 283.05, 104.18 | -61.63, -33.06 | in-in | in | 8.6731 | Saltbr-in | 2.5745 | HRD-in | -63.52, -52.73 | 78.44, -11.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8201 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.22, 130.12 | APE9-dihe-na | 106.71, 171.13 | APE8-dihe-in | -96.94, 126.07 | APE8-rot-in | 299.07 | APE67-dihe-in | -62.15, -19.51 | -52.23, -44.36 | APE12-dist-in | 12.8679 | APE11-dist-in | 12.8691 | APE10-dist-in | 7.2677 | APE9-dist-in | 4.7446 | S241A | None | None | XRAY | 1.95 | 0.186 | 0.23 | A | 310.0 | 288.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 2biy | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.8e-84 | 288.8 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3HRCA | O15530 | 76 | 359 | 556.0 | ATP:1373 | ATPlike | Active | DFGin | 6.4861 | 14.8331 | BLAminus | -136.91, -178.17 | 71.81, 74.55 | -104.54, 6.98 | 286.89, 102.51 | -65.47, -24.41 | in-in | in | 8.4211 | Saltbr-in | 3.1591 | HRD-in | -77.24, -54.93 | 76.93, -11.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.87 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.25, 162.0 | APE9-dihe-na | 130.63, -171.63 | APE8-dihe-in | -125.01, 129.68 | APE8-rot-in | 292.48 | APE67-dihe-in | -58.92, -25.29 | -45.32, -48.7 | APE12-dist-in | 7.4085 | APE11-dist-in | 10.582 | APE10-dist-in | 4.9259 | APE9-dist-in | 3.4793 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.91 | 0.182 | 0.207 | A | 311.0 | 280.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 3hrc | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4RRVA | O15530 | 76 | 359 | 556.0 | ATP:60401 | ATPlike | Active | DFGin | 6.5481 | 14.9984 | BLAminus | -136.55, -175.99 | 74.63, 72.8 | -106.52, 5.78 | 286.61, 100.18 | -68.12, -17.88 | in-in | in | 8.5198 | Saltbr-in | 2.956 | HRD-in | -71.77, -54.29 | 78.75, -11.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9375 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.13, 162.83 | APE9-dihe-na | 132.08, -169.67 | APE8-dihe-in | -127.24, 132.02 | APE8-rot-in | 298.33 | APE67-dihe-in | -59.21, -24.3 | -51.83, -46.04 | APE12-dist-in | 7.2806 | APE11-dist-in | 10.5025 | APE10-dist-in | 4.943 | APE9-dist-in | 3.5694 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.412 | 0.135 | 0.163 | A | 311.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4rrv | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5ACKA | O15530 | 73 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.6153 | 14.8606 | BLAminus | -135.34, 179.84 | 72.22, 79.01 | -106.01, 4.14 | 287.93, 97.64 | -67.02, -18.73 | in-in | in | 8.4184 | Saltbr-in | 2.5825 | HRD-in | -74.68, -53.67 | 78.01, -12.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9064 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.4, 162.51 | APE9-dihe-na | 136.44, -168.07 | APE8-dihe-in | -132.35, 133.52 | APE8-rot-in | 296.36 | APE67-dihe-in | -62.96, -23.95 | -54.34, -43.19 | APE12-dist-in | 7.3257 | APE11-dist-in | 10.5222 | APE10-dist-in | 4.9779 | APE9-dist-in | 3.5575 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.24 | 0.143 | 0.166 | A | 311.0 | 287.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5ack | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVPA | O15530 | 75 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3028 | 14.9979 | BLAminus | -144.92, -168.82 | 66.06, 77.78 | -108.23, 11.17 | 281.99, 93.22 | -63.04, -32.41 | in-in | in | 9.539 | Saltbr-in | 3.1581 | HRD-in | -77.47, -51.83 | 79.92, -12.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8481 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.64, 166.02 | APE9-dihe-na | 141.61, 177.5 | APE8-dihe-in | -123.02, 134.29 | APE8-rot-in | 296.02 | APE67-dihe-in | -68.65, -16.53 | -46.89, -50.92 | APE12-dist-in | 7.9068 | APE11-dist-in | 10.6706 | APE10-dist-in | 5.166 | APE9-dist-in | 3.7049 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | A | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVPB | O15530 | 74 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3283 | 14.5498 | BLAminus | -137.23, -179.71 | 80.14, 74.16 | -105.47, 15.38 | 295.0, 84.83 | -59.91, -31.47 | in-in | in | 9.2741 | Saltbr-in | 3.3024 | HRD-in | -80.68, -44.41 | 73.96, -16.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7443 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.8, 152.43 | APE9-dihe-na | 134.43, -173.75 | APE8-dihe-in | -120.09, 128.28 | APE8-rot-in | 302.93 | APE67-dihe-in | -67.56, -25.72 | -44.99, -47.55 | APE12-dist-in | 7.8719 | APE11-dist-in | 11.0112 | APE10-dist-in | 5.3751 | APE9-dist-in | 3.7868 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | B | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVPC | O15530 | 75 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3906 | 14.6076 | BLAminus | -132.15, -176.81 | 71.98, 84.02 | -116.53, 7.62 | 291.47, 90.46 | -60.24, -24.5 | in-in | in | 9.3044 | Saltbr-in | 3.0866 | HRD-in | -75.92, -52.06 | 78.45, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8228 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.81, 168.64 | APE9-dihe-na | 131.92, -176.79 | APE8-dihe-in | -126.79, 133.21 | APE8-rot-in | 299.13 | APE67-dihe-in | -67.64, -15.8 | -51.62, -50.49 | APE12-dist-in | 7.6523 | APE11-dist-in | 10.8632 | APE10-dist-in | 5.1235 | APE9-dist-in | 3.6447 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | C | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVPD | O15530 | 74 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3336 | 14.4328 | BLAminus | -146.99, -174.22 | 74.22, 81.56 | -113.84, 4.02 | 287.97, 93.59 | -56.11, -25.73 | in-in | in | 9.3044 | Saltbr-in | 3.2517 | HRD-in | -82.38, -50.18 | 78.4, -12.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8357 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.65, 165.17 | APE9-dihe-na | 129.1, -166.82 | APE8-dihe-in | -132.84, 129.79 | APE8-rot-in | 300.06 | APE67-dihe-in | -65.46, -17.03 | -48.9, -48.47 | APE12-dist-in | 8.2282 | APE11-dist-in | 10.8909 | APE10-dist-in | 5.3485 | APE9-dist-in | 3.6459 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | D | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4CT2A | O15530 | 75 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.5509 | 14.8668 | BLAminus | -136.23, -174.98 | 70.54, 70.07 | -102.02, 6.41 | 290.69, 95.78 | -63.73, -21.59 | in-in | in | 8.2523 | Saltbr-in | 2.6427 | HRD-in | -73.2, -54.84 | 77.37, -9.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9649 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.02, 163.59 | APE9-dihe-na | 137.39, -170.05 | APE8-dihe-in | -132.12, 131.72 | APE8-rot-in | 295.26 | APE67-dihe-in | -63.06, -17.27 | -51.84, -45.87 | APE12-dist-in | 7.1628 | APE11-dist-in | 10.5242 | APE10-dist-in | 4.9787 | APE9-dist-in | 3.5273 | L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.25 | 0.194 | 0.226 | A | 311.0 | 280.0 | 5 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4ct2 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.5e-84 | 286.4 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5MRDA | O15530 | 76 | 359 | 556.0 | ATP:405 | ATPlike | Active | DFGin | 6.4288 | 14.7004 | BLAminus | -133.69, -177.11 | 74.21, 73.9 | -105.88, 9.0 | 289.39, 99.64 | -68.32, -19.62 | in-in | in | 8.3463 | Saltbr-in | 2.6673 | HRD-in | -74.32, -53.19 | 77.26, -10.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9416 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.86, 160.68 | APE9-dihe-na | 136.11, -166.87 | APE8-dihe-in | -131.1, 132.63 | APE8-rot-in | 296.36 | APE67-dihe-in | -62.36, -23.28 | -53.02, -44.84 | APE12-dist-in | 7.3524 | APE11-dist-in | 10.4975 | APE10-dist-in | 4.9095 | APE9-dist-in | 3.5424 | K76S,L113V,I118V,I119N,V124I,T128Q,R131K,T148C | SEP241 | SEP241 | XRAY | 1.41 | 0.142 | 0.174 | A | 310.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5mrd | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.7e-83 | 285.6 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3HRFA | O15530 | 75 | 359 | 556.0 | ATP:1373,P47:1374 | ATPlike,Allosteric | Active | DFGin | 6.5137 | 14.7842 | BLAminus | -133.77, -176.11 | 75.25, 77.12 | -110.83, 6.58 | 287.55, 100.98 | -63.85, -22.79 | in-in | in | 8.3869 | Saltbr-in | 2.7006 | HRD-in | -73.67, -53.98 | 76.59, -10.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9232 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.42, 166.15 | APE9-dihe-na | 124.75, -165.6 | APE8-dihe-in | -127.97, 128.5 | APE8-rot-in | 295.31 | APE67-dihe-in | -62.28, -24.12 | -44.34, -47.42 | APE12-dist-in | 7.3513 | APE11-dist-in | 10.5457 | APE10-dist-in | 4.8669 | APE9-dist-in | 3.4806 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.9 | 0.165 | 0.177 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 3hrf | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4A06A | O15530 | 75 | 359 | 556.0 | ATP:500,A06:600 | ATPlike,Allosteric | Active | DFGin | 6.5121 | 14.757 | BLAminus | -135.73, -177.17 | 74.25, 74.67 | -110.25, 11.82 | 284.97, 101.73 | -68.23, -22.46 | in-in | in | 8.3192 | Saltbr-in | 2.8636 | HRD-in | -73.73, -51.84 | 74.62, -10.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9204 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.65, 165.25 | APE9-dihe-na | 128.95, -173.35 | APE8-dihe-in | -120.15, 131.51 | APE8-rot-in | 299.31 | APE67-dihe-in | -59.46, -27.29 | -45.75, -47.91 | APE12-dist-in | 7.336 | APE11-dist-in | 10.4473 | APE10-dist-in | 4.8734 | APE9-dist-in | 3.5088 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.0 | 0.161 | 0.198 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4a06 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4AW0A | O15530 | 75 | 359 | 556.0 | ATP:500,MJF:600 | ATPlike,Allosteric | Active | DFGin | 6.5313 | 14.9926 | BLAminus | -134.84, 177.25 | 78.73, 76.19 | -106.3, 8.53 | 283.51, 97.11 | -69.63, -19.36 | in-in | in | 8.5954 | Saltbr-in | 3.0091 | HRD-in | -83.05, -53.03 | 79.45, -12.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9336 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.69, 159.04 | APE9-dihe-na | 139.48, -167.8 | APE8-dihe-in | -131.87, 132.42 | APE8-rot-in | 295.45 | APE67-dihe-in | -61.29, -25.28 | -54.74, -42.17 | APE12-dist-in | 7.5089 | APE11-dist-in | 10.6011 | APE10-dist-in | 5.0264 | APE9-dist-in | 3.5797 | Y288G,Q292A | SEP241 | SEP241,CME260 | XRAY | 1.43 | 0.171 | 0.188 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4aw0 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4AW1A | O15530 | 66 | 359 | 556.0 | ATP:1360,21O:1361 | ATPlike,Allosteric | Active | DFGin | 6.325 | 14.155 | BLAminus | -137.24, -178.23 | 68.96, 84.69 | -105.37, 17.06 | 286.01, 86.79 | -62.77, -26.7 | in-in | in | 8.5758 | Saltbr-in | 2.8639 | HRD-in | -81.18, -54.06 | 78.32, -13.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8487 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.98, 160.2 | APE9-dihe-na | 130.22, -162.57 | APE8-dihe-in | -126.98, 128.72 | APE8-rot-in | 295.96 | APE67-dihe-in | -57.45, -24.35 | -48.01, -47.7 | APE12-dist-in | 7.6532 | APE11-dist-in | 10.8523 | APE10-dist-in | 5.0751 | APE9-dist-in | 3.5856 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.68 | 0.165 | 0.186 | A | 311.0 | 287.0 | 5 | 30 | 25 | 5 | [[82, 342]] | 1.0 | 4aw1 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4RQKA | O15530 | 74 | 359 | 556.0 | ATP:403,R1S:404 | ATPlike,Allosteric | Active | DFGin | 6.4608 | 14.7857 | BLAminus | -139.06, -177.03 | 75.27, 72.83 | -105.25, 7.36 | 287.3, 98.33 | -64.7, -21.38 | in-in | in | 8.4643 | Saltbr-in | 2.9412 | HRD-in | -73.98, -52.31 | 74.79, -9.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8799 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.64, 164.69 | APE9-dihe-na | 126.87, -171.23 | APE8-dihe-in | -124.75, 130.48 | APE8-rot-in | 298.57 | APE67-dihe-in | -59.79, -23.66 | -48.31, -47.88 | APE12-dist-in | 7.2437 | APE11-dist-in | 10.4657 | APE10-dist-in | 4.9176 | APE9-dist-in | 3.5437 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.55 | 0.133 | 0.167 | A | 311.0 | 286.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4rqk | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4RQVA | O15530 | 71 | 359 | 556.0 | ATP:405,R2S:406 | ATPlike,Allosteric | Active | DFGin | 6.4916 | 14.9536 | BLAminus | -139.41, -174.88 | 74.87, 69.78 | -102.0, 7.85 | 285.85, 94.73 | -65.11, -21.56 | in-in | in | 8.2557 | Saltbr-in | 2.7717 | HRD-in | -72.94, -52.57 | 74.87, -10.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9156 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.07, 164.19 | APE9-dihe-na | 130.69, -171.7 | APE8-dihe-in | -126.67, 130.74 | APE8-rot-in | 297.63 | APE67-dihe-in | -61.47, -23.77 | -49.17, -46.26 | APE12-dist-in | 7.2532 | APE11-dist-in | 10.4876 | APE10-dist-in | 4.9687 | APE9-dist-in | 3.5133 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.502 | 0.133 | 0.166 | A | 311.0 | 289.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4rqv | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVOA | O15530 | 73 | 359 | 556.0 | ATP:401,78W:402 | ATPlike,Allosteric | Active | DFGin | 6.581 | 15.0047 | BLAminus | -134.78, 179.9 | 79.12, 70.17 | -103.55, 0.25 | 286.72, 100.66 | -64.63, -19.63 | in-in | in | 8.5884 | Saltbr-in | 2.6313 | HRD-in | -71.89, -54.41 | 77.65, -9.82 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9194 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.78, 162.52 | APE9-dihe-na | 134.75, -167.11 | APE8-dihe-in | -130.46, 134.12 | APE8-rot-in | 296.12 | APE67-dihe-in | -62.26, -22.94 | -53.92, -45.37 | APE12-dist-in | 7.4502 | APE11-dist-in | 10.5584 | APE10-dist-in | 4.9836 | APE9-dist-in | 3.5527 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.09 | 0.136 | 0.157 | A | 311.0 | 287.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvo | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4XX9A | O15530 | 71 | 359 | 556.0 | ATP:401,RF4:402,RF4:403 | ATPlike,Allosteric,Allosteric | Active | DFGin | 6.5134 | 14.9881 | BLAminus | -138.47, -176.21 | 74.83, 73.76 | -104.66, 7.86 | 282.59, 98.49 | -68.99, -20.43 | in-in | in | 8.4422 | Saltbr-in | 2.9225 | HRD-in | -73.71, -50.51 | 73.32, -9.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8949 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.41, 162.37 | APE9-dihe-na | 129.79, -167.49 | APE8-dihe-in | -129.09, 132.1 | APE8-rot-in | 295.95 | APE67-dihe-in | -59.66, -23.23 | -49.94, -47.34 | APE12-dist-in | 7.3717 | APE11-dist-in | 10.5754 | APE10-dist-in | 4.9467 | APE9-dist-in | 3.5452 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.4 | 0.13 | 0.165 | A | 310.0 | 289.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4xx9 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.8e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4A07A | O15530 | 75 | 359 | 556.0 | ATP:500,AZ7:600,AZ7:700 | ATPlike,Allosteric,Allosteric | Active | DFGin | 6.6546 | 14.7523 | BLAminus | -135.35, -178.9 | 76.01, 72.4 | -108.94, 8.63 | 286.31, 98.68 | -64.37, -21.88 | in-in | in | 8.6213 | Saltbr-in | 2.919 | HRD-in | -76.19, -54.82 | 80.07, -12.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9107 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.16, 162.52 | APE9-dihe-na | 132.15, -164.48 | APE8-dihe-in | -133.89, 130.56 | APE8-rot-in | 295.87 | APE67-dihe-in | -62.13, -24.83 | -47.31, -46.9 | APE12-dist-in | 7.3216 | APE11-dist-in | 10.4272 | APE10-dist-in | 4.9977 | APE9-dist-in | 3.5816 | Y288G,Q292A | SEP241 | SEP241,CSS260 | XRAY | 1.85 | 0.161 | 0.2 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4a07 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 8DQTA | O15530 | 70 | 359 | 556.0 | U35:401,U35:402,U35:403 | Allosteric,Allosteric,Allosteric | Active | DFGin | 6.5386 | 15.228 | BLAminus | -137.99, -177.67 | 76.39, 75.41 | -107.03, 7.63 | 286.75, 95.91 | -68.77, -18.63 | in-in | in | 8.5573 | Saltbr-in | 2.9067 | HRD-in | -74.31, -48.93 | 74.07, -13.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9489 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -143.2, 161.34 | APE9-dihe-na | 132.87, -165.96 | APE8-dihe-in | -131.33, 133.45 | APE8-rot-in | 295.53 | APE67-dihe-in | -61.71, -24.62 | -51.87, -45.17 | APE12-dist-in | 7.2521 | APE11-dist-in | 10.4342 | APE10-dist-in | 4.9085 | APE9-dist-in | 3.5907 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.31 | 0.2 | 0.224 | A | 311.0 | 290.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 8dqt | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3OTUA | O15530 | 77 | 359 | 556.0 | J30:1,BI4:360 | Allosteric,Type1.5_Front | Active | DFGin | 6.407 | 14.9865 | BLAminus | -147.19, -166.49 | 62.44, 61.65 | -95.64, 10.19 | 290.91, 105.88 | -63.28, -24.6 | in-in | in | 8.3704 | Saltbr-in | 3.3366 | HRD-in | -67.23, -53.13 | 82.11, -16.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7953 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.97, 157.81 | APE9-dihe-na | 151.4, -176.81 | APE8-dihe-in | -123.26, 126.19 | APE8-rot-in | 294.94 | APE67-dihe-in | -53.95, -30.51 | -40.25, -53.87 | APE12-dist-in | 7.7118 | APE11-dist-in | 10.3288 | APE10-dist-in | 5.2437 | APE9-dist-in | 4.1303 | T148C | SEP241 | SEP241 | XRAY | 2.101 | 0.197 | 0.24 | A | 316.0 | 277.0 | 6 | 30 | 25 | 5 | [[82, 342]] | 1.0 | 3otu | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | AF-O15530-K1A | O15530 | 74 | 350 | 556.0 | No_ligand | No_ligand | Active | DFGin | 6.307 | 14.7525 | BLAminus | -134.14, -175.03 | 67.73, 56.76 | -81.0, 7.09 | 290.02, 100.1 | -62.73, -31.75 | in-in | in | 8.4785 | Saltbr-in | 2.6917 | HRD-in | -71.22, -49.98 | 68.85, -15.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9019 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -143.76, 160.45 | APE9-dihe-na | 125.82, -178.56 | APE8-dihe-in | -110.7, 135.78 | APE8-rot-in | 301.58 | APE67-dihe-in | -71.92, -18.9 | -54.44, -36.21 | APE12-dist-in | 7.4783 | APE11-dist-in | 10.7463 | APE10-dist-in | 5.0363 | APE9-dist-in | 3.4837 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 277.0 | 277.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | AF-O15530-K1 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 8.4e-85 | 289.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | AF-O15530-K3A | O15530 | 74 | 350 | 556.0 | No_ligand | No_ligand | Active | DFGin | 6.0234 | 14.6473 | BLAminus | -139.54, -179.29 | 63.97, 66.91 | -82.88, 11.22 | 294.97, 97.73 | -59.7, -35.74 | in-in | in | 8.7295 | Saltbr-in | 2.6551 | HRD-in | -73.34, -47.9 | 67.59, -9.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8048 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.66, 143.7 | APE9-dihe-na | 124.83, 164.09 | APE8-dihe-in | -82.81, 130.45 | APE8-rot-in | 291.03 | APE67-dihe-in | -71.92, -16.19 | -51.02, -35.4 | APE12-dist-in | 8.3871 | APE11-dist-in | 11.0601 | APE10-dist-in | 5.2904 | APE9-dist-in | 4.3622 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 277.0 | 277.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | AF-O15530-K3 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 8.4e-85 | 289.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3SC1A | O15530 | 73 | 359 | 556.0 | 3S1:900 | Type1 | Active | DFGin | 6.4332 | 14.1153 | BLAminus | -125.85, 175.62 | 82.13, 80.63 | -113.39, 8.45 | 290.85, 87.77 | -53.07, -47.22 | in-in | in | 8.7083 | Saltbr-in | 3.2163 | HRD-in | -72.93, -48.81 | 80.48, -8.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8508 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -100.12, -172.48 | APE9-dihe-na | 115.93, 147.74 | APE8-dihe-in | -93.61, 137.68 | APE8-rot-in | 299.7 | APE67-dihe-in | -55.26, -32.91 | -54.79, -48.8 | APE12-dist-in | 8.7388 | APE11-dist-in | 10.6062 | APE10-dist-in | 5.4107 | APE9-dist-in | 3.9864 | None | SEP241 | SEP241 | XRAY | 2.7 | 0.2 | 0.237 | A | 311.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3sc1 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3RCJA | O15530 | 77 | 358 | 556.0 | 3RC:0 | Type1 | Active | DFGin | 6.5504 | 14.3915 | BLAminus | -128.99, -167.62 | 59.76, 67.13 | -93.27, 12.1 | 286.78, 86.8 | -60.54, -37.27 | in-in | in | 8.539 | Saltbr-in | 2.7862 | HRD-in | -65.85, -49.34 | 77.48, -8.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.08, 164.56 | APE9-dihe-na | 127.57, -173.24 | APE8-dihe-in | -123.98, 130.3 | APE8-rot-in | 296.56 | APE67-dihe-in | -63.09, -20.07 | -49.59, -44.96 | APE12-dist-in | 7.8304 | APE11-dist-in | 10.7456 | APE10-dist-in | 5.0252 | APE9-dist-in | 3.6456 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.7 | 0.217 | 0.198 | A | 311.0 | 282.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 3rcj | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVLA | O15530 | 74 | 359 | 556.0 | 537:401 | Type1 | Active | DFGin | 6.5959 | 14.602 | BLAminus | -130.64, -179.01 | 78.07, 78.29 | -107.64, 5.9 | 287.24, 98.42 | -64.3, -24.0 | in-in | in | 8.2927 | Saltbr-in | 2.5582 | HRD-in | -74.44, -52.48 | 78.34, -12.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9059 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.91, 163.01 | APE9-dihe-na | 134.48, -168.83 | APE8-dihe-in | -131.23, 133.97 | APE8-rot-in | 296.05 | APE67-dihe-in | -61.17, -24.01 | -50.83, -47.55 | APE12-dist-in | 7.3206 | APE11-dist-in | 10.4705 | APE10-dist-in | 4.8806 | APE9-dist-in | 3.5651 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.4 | 0.154 | 0.178 | A | 311.0 | 286.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvl | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVMA | O15530 | 76 | 359 | 556.0 | ADE:401 | Type1 | Active | DFGin | 6.5146 | 14.8576 | BLAminus | -134.29, -178.73 | 78.5, 76.19 | -107.92, 3.05 | 284.81, 100.85 | -68.49, -15.39 | in-in | in | 8.3988 | Saltbr-in | 2.9222 | HRD-in | -74.83, -53.98 | 76.68, -6.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9138 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.77, 160.72 | APE9-dihe-na | 136.54, -165.87 | APE8-dihe-in | -131.32, 134.23 | APE8-rot-in | 298.42 | APE67-dihe-in | -62.0, -21.56 | -53.2, -46.03 | APE12-dist-in | 7.4265 | APE11-dist-in | 10.5567 | APE10-dist-in | 4.9493 | APE9-dist-in | 3.5336 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.26 | 0.135 | 0.155 | A | 311.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvm | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5LVNA | O15530 | 75 | 359 | 556.0 | ADN:402 | Type1 | Active | DFGin | 6.4926 | 14.7837 | BLAminus | -138.56, -175.41 | 73.41, 75.09 | -105.63, 5.44 | 285.54, 101.95 | -63.79, -19.6 | in-in | in | 8.4347 | Saltbr-in | 2.7393 | HRD-in | -74.59, -52.51 | 78.18, -12.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8995 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.48, 161.66 | APE9-dihe-na | 136.02, -164.27 | APE8-dihe-in | -134.21, 135.25 | APE8-rot-in | 295.47 | APE67-dihe-in | -61.9, -23.15 | -53.94, -45.84 | APE12-dist-in | 7.4385 | APE11-dist-in | 10.5331 | APE10-dist-in | 4.8932 | APE9-dist-in | 3.5664 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.379 | 0.135 | 0.162 | A | 311.0 | 285.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 5lvn | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1H1WA | O15530 | 71 | 359 | 556.0 | ATP:1373 | ATPlike | Inactive | DFGin | 6.6116 | 14.931 | BLAminus | -145.26, -169.97 | 71.92, 72.18 | -105.82, -0.04 | 289.27, 102.08 | -58.33, -31.92 | in-in | in | 8.5808 | Saltbr-in | 2.7103 | HRD-in | -71.45, -48.32 | 74.08, -8.04 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8395 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.69, 112.94 | APE9-dihe-na | -63.98, -168.66 | APE8-dihe-in | -54.13, 124.0 | APE8-rot-in | 301.59 | APE67-dihe-in | -62.54, -19.03 | -38.83, -50.46 | APE12-dist-in | 8.922 | APE11-dist-out | 5.528 | APE10-dist-out | 10.2978 | APE9-dist-in | 3.7994 | None | SEP241 | SEP241 | XRAY | 2.0 | 0.196 | 0.223 | A | 289.0 | 285.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 1h1w | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.8e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXA | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.5961 | 14.1691 | BLAminus | -138.52, -175.65 | 62.9, 74.02 | -93.7, 13.51 | 275.9, 89.61 | -62.84, -23.94 | in-in | in | 8.8135 | Saltbr-in | 2.5558 | HRD-in | -68.79, -51.77 | 77.65, -2.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8365 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -110.22, 106.38 | APE9-dihe-na | -61.01, -163.77 | APE8-dihe-in | -59.2, 130.87 | APE8-rot-in | 313.64 | APE67-dihe-in | -68.86, -21.58 | -48.76, -40.32 | APE12-dist-in | 9.226 | APE11-dist-out | 5.7837 | APE10-dist-out | 10.5309 | APE9-dist-in | 3.9835 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | A | 316.0 | 284.0 | 1 | 30 | 29 | 1 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXB | O15530 | 77 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.6597 | 14.1548 | BLAminus | -140.69, -175.67 | 59.43, 71.11 | -92.21, 14.29 | 279.78, 86.28 | -63.72, -16.63 | in-in | in | 8.802 | Saltbr-in | 2.5641 | HRD-in | -68.32, -50.05 | 78.21, -3.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8222 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -111.03, 106.62 | APE9-dihe-na | -60.26, -162.55 | APE8-dihe-in | -59.71, 131.44 | APE8-rot-in | 313.93 | APE67-dihe-in | -67.3, -21.72 | -51.61, -39.66 | APE12-dist-in | 9.2384 | APE11-dist-out | 5.8005 | APE10-dist-out | 10.5524 | APE9-dist-in | 3.9081 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | B | 316.0 | 281.0 | 2 | 30 | 28 | 2 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXC | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.6298 | 14.0961 | BLAminus | -135.92, -176.39 | 63.79, 71.64 | -93.36, 13.73 | 280.67, 86.49 | -62.67, -20.94 | in-in | in | 8.7824 | Saltbr-in | 2.5509 | HRD-in | -66.06, -52.0 | 76.42, -2.2 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8354 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -110.22, 106.64 | APE9-dihe-na | -60.77, -161.89 | APE8-dihe-in | -59.91, 131.8 | APE8-rot-in | 311.89 | APE67-dihe-in | -63.47, -22.82 | -49.61, -43.91 | APE12-dist-in | 9.1653 | APE11-dist-out | 5.8015 | APE10-dist-out | 10.55 | APE9-dist-in | 3.9841 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | C | 316.0 | 284.0 | 1 | 30 | 29 | 1 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXD | O15530 | 76 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.5711 | 14.146 | BLAminus | -134.45, -170.09 | 60.8, 71.91 | -91.57, 12.91 | 278.05, 86.51 | -67.5, -17.43 | in-in | in | 8.7987 | Saltbr-in | 2.5834 | HRD-in | -66.01, -50.34 | 77.25, -1.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8418 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -110.2, 105.71 | APE9-dihe-na | -59.39, -160.44 | APE8-dihe-in | -60.94, 132.03 | APE8-rot-in | 313.43 | APE67-dihe-in | -67.95, -22.9 | -52.31, -39.76 | APE12-dist-in | 9.2273 | APE11-dist-out | 5.7904 | APE10-dist-out | 10.5469 | APE9-dist-in | 3.9121 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | D | 316.0 | 283.0 | 1 | 30 | 29 | 1 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXE | O15530 | 76 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.3816 | 14.9206 | BLAminus | -125.38, -158.75 | 61.49, 56.01 | -85.03, 10.36 | 279.31, 82.03 | -55.13, -32.27 | in-in | in | 9.2368 | Saltbr-in | 3.2715 | HRD-in | -67.18, -49.37 | 73.61, -2.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9678 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nooi | APE10-dihe-na | -112.75, 120.85 | APE9-dihe-na | -80.18, -170.48 | APE8-dihe-in | -52.91, 130.32 | APE8-rot-in | 309.26 | APE67-dihe-in | -61.57, -27.92 | -56.84, -38.07 | APE12-dist-none | 999.0 | APE11-dist-out | 5.4882 | APE10-dist-out | 10.2693 | APE9-dist-in | 4.4822 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | E | 316.0 | 274.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXF | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.3677 | 14.9155 | BLAminus | -124.96, -165.04 | 64.25, 56.63 | -90.23, 13.81 | 273.61, 91.31 | -58.82, -32.5 | in-none | in | 9.2317 | Saltbr-none | 999.0 | HRD-in | -66.95, -49.19 | 76.54, -9.89 | none-in-out | SNCnio | in-out | ActLoopNT-in | 2.9816 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -112.23, 117.01 | APE9-dihe-na | -74.75, -174.06 | APE8-dihe-in | -40.45, 117.92 | APE8-rot-in | 309.94 | APE67-dihe-in | -62.78, -29.13 | -41.21, -44.42 | APE12-dist-in | 8.1177 | APE11-dist-out | 5.4885 | APE10-dist-out | 10.2748 | APE9-dist-in | 4.4634 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | F | 316.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXG | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.4182 | 15.1625 | BLAminus | -124.35, -160.11 | 59.71, 58.4 | -85.01, 8.33 | 270.63, 86.47 | -58.24, -35.05 | in-in | in | 9.2322 | Saltbr-in | 3.2566 | HRD-in | -66.57, -49.64 | 76.01, -6.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0259 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -113.59, 119.71 | APE9-dihe-na | -80.06, -167.69 | APE8-dihe-in | -52.92, 132.86 | APE8-rot-in | 313.01 | APE67-dihe-in | -62.53, -35.87 | -56.69, -38.23 | APE12-dist-in | 8.4931 | APE11-dist-out | 5.4816 | APE10-dist-out | 10.2289 | APE9-dist-in | 4.3614 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | G | 316.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORXH | O15530 | 75 | 359 | 556.0 | 1F8:1 | Allosteric | Inactive | DFGin | 6.4702 | 14.8365 | BLAminus | -123.34, -162.32 | 62.45, 60.25 | -89.76, 14.7 | 283.48, 85.4 | -55.85, -32.26 | in-in | in | 9.2345 | Saltbr-in | 3.2833 | HRD-in | -67.42, -48.8 | 75.62, -9.07 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9802 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -112.9, 122.93 | APE9-dihe-na | -81.65, -170.32 | APE8-dihe-in | -53.77, 133.41 | APE8-rot-in | 303.61 | APE67-dihe-in | -61.23, -30.63 | -57.13, -39.02 | APE12-dist-in | 8.3784 | APE11-dist-out | 5.4961 | APE10-dist-out | 10.1982 | APE9-dist-in | 4.4177 | T148C | SEP241 | SEP241 | XRAY | 2.204 | 0.209 | 0.243 | H | 316.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 3orx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORZA | O15530 | 74 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6225 | 14.6052 | BLAminus | -134.96, -167.36 | 70.2, 66.13 | -101.26, 0.99 | 293.7, 88.7 | -61.05, -29.24 | in-in | in | 8.2152 | Saltbr-in | 2.8103 | HRD-in | -65.12, -49.46 | 75.7, -10.07 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8327 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -134.38, 111.86 | APE9-dihe-na | -60.27, -174.97 | APE8-dihe-in | -55.74, 132.42 | APE8-rot-in | 303.15 | APE67-dihe-in | -56.98, -32.17 | -55.27, -42.37 | APE12-dist-in | 11.5493 | APE11-dist-out | 6.544 | APE10-dist-out | 10.866 | APE9-dist-in | 4.1173 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | A | 316.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3orz | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORZB | O15530 | 73 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6476 | 14.7764 | BLAminus | -139.38, -168.66 | 74.13, 69.92 | -111.18, 3.04 | 284.6, 93.64 | -63.39, -24.83 | in-in | in | 8.2923 | Saltbr-in | 2.7592 | HRD-in | -64.66, -48.81 | 76.86, -10.42 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8659 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.43, 114.97 | APE9-dihe-na | -62.67, -167.65 | APE8-dihe-in | -63.67, 131.38 | APE8-rot-in | 299.84 | APE67-dihe-in | -54.64, -32.97 | -56.45, -39.98 | APE12-dist-in | 11.638 | APE11-dist-out | 6.3971 | APE10-dist-out | 10.7873 | APE9-dist-in | 4.0869 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | B | 316.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3orz | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORZC | O15530 | 74 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6668 | 14.6791 | BLAminus | -134.07, -170.51 | 76.79, 69.39 | -110.34, 1.38 | 287.93, 89.81 | -56.71, -30.43 | in-in | in | 8.2245 | Saltbr-in | 2.8037 | HRD-in | -64.4, -49.76 | 78.61, -9.94 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8049 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -134.53, 111.0 | APE9-dihe-na | -58.83, -174.56 | APE8-dihe-in | -56.66, 132.63 | APE8-rot-in | 302.29 | APE67-dihe-in | -56.84, -32.58 | -55.43, -42.03 | APE12-dist-in | 11.7307 | APE11-dist-out | 6.55 | APE10-dist-out | 10.875 | APE9-dist-in | 4.0824 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | C | 316.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3orz | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3ORZD | O15530 | 73 | 359 | 556.0 | 2A2:1,BI4:360 | Allosteric,Type1 | Inactive | DFGin | 6.6487 | 14.7735 | BLAminus | -139.63, -168.42 | 74.39, 69.06 | -110.33, 3.29 | 285.32, 93.06 | -63.48, -24.84 | in-in | in | 8.3101 | Saltbr-in | 2.754 | HRD-in | -64.65, -47.43 | 73.97, -9.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8768 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -126.78, 121.12 | APE9-dihe-na | -63.33, -166.44 | APE8-dihe-in | -63.66, 131.18 | APE8-rot-in | 301.29 | APE67-dihe-in | -54.43, -33.46 | -55.31, -40.36 | APE12-dist-in | 11.5839 | APE11-dist-out | 6.4058 | APE10-dist-out | 10.8417 | APE9-dist-in | 4.0404 | T148C | SEP241 | SEP241 | XRAY | 2.0 | 0.22 | 0.265 | D | 316.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3orz | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 7.9e-85 | 290.0 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1Z5MA | O15530 | 74 | 359 | 556.0 | LI8:501 | Type1 | Inactive | DFGin | 6.9657 | 14.6691 | BLAminus | -143.06, -166.04 | 70.1, 70.4 | -106.54, 10.63 | 285.55, 95.37 | -57.95, -38.82 | in-in | in | 8.979 | Saltbr-in | 2.8616 | HRD-in | -60.53, -42.76 | 63.99, 3.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.6826 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -142.8, 123.87 | APE9-dihe-na | -69.98, -168.75 | APE8-dihe-in | -47.59, 126.16 | APE8-rot-in | 298.44 | APE67-dihe-in | -75.58, -18.39 | -37.0, -46.81 | APE12-dist-in | 8.5442 | APE11-dist-out | 6.2855 | APE10-dist-out | 10.4569 | APE9-dist-in | 4.0502 | None | SEP241 | SEP241 | XRAY | 2.17 | 0.232 | 0.269 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 1z5m | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 2PE0A | O15530 | 74 | 359 | 556.0 | 39Z:501 | Type1 | Inactive | DFGin | 6.4474 | 14.3844 | BLAminus | -129.98, -179.46 | 78.75, 74.81 | -106.99, 5.13 | 286.59, 90.93 | -55.7, -29.7 | in-in | in | 8.7227 | Saltbr-in | 2.7831 | HRD-in | -72.01, -55.71 | 78.26, -0.88 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8174 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -117.01, 133.16 | APE9-dihe-na | -80.12, -143.18 | APE8-dihe-in | -90.02, 137.86 | APE8-rot-in | 307.83 | APE67-dihe-in | -64.54, -15.21 | -51.36, -49.75 | APE12-dist-in | 9.1401 | APE11-dist-out | 5.5127 | APE10-dist-out | 10.1028 | APE9-dist-in | 3.7888 | None | SEP241 | SEP241 | XRAY | 2.35 | 0.202 | 0.24 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2pe0 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 2PE1A | O15530 | 74 | 359 | 556.0 | 517:501 | Type1 | Inactive | DFGin | 6.6447 | 14.6824 | BLAminus | -139.4, -175.86 | 73.15, 71.4 | -105.21, 7.65 | 286.89, 93.63 | -52.89, -40.97 | in-in | in | 8.8829 | Saltbr-in | 2.5948 | HRD-in | -69.74, -56.95 | 81.13, 2.35 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8564 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -114.84, 143.11 | APE9-dihe-na | -79.47, -134.7 | APE8-dihe-in | -90.68, 136.03 | APE8-rot-in | 300.98 | APE67-dihe-in | -68.92, -11.38 | -43.74, -52.34 | APE12-dist-in | 9.1167 | APE11-dist-out | 5.7014 | APE10-dist-out | 10.3798 | APE9-dist-in | 3.6055 | None | SEP241 | SEP241 | XRAY | 2.14 | 0.224 | 0.282 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2pe1 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 2PE2A | O15530 | 74 | 359 | 556.0 | 464:501 | Type1 | Inactive | DFGin | 6.5908 | 14.4155 | BLAminus | -135.75, -175.91 | 78.63, 72.01 | -109.62, 0.43 | 287.28, 93.19 | -54.2, -35.84 | in-in | in | 8.5622 | Saltbr-in | 2.5509 | HRD-in | -75.76, -49.83 | 75.8, -8.69 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7244 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.61, 128.36 | APE9-dihe-na | -70.67, -166.57 | APE8-dihe-in | -59.34, 134.44 | APE8-rot-in | 302.45 | APE67-dihe-in | -67.69, -11.47 | -51.51, -47.62 | APE12-dist-in | 8.9817 | APE11-dist-out | 5.5266 | APE10-dist-out | 10.3125 | APE9-dist-in | 3.7381 | None | SEP241 | SEP241 | XRAY | 2.13 | 0.189 | 0.215 | A | 286.0 | 276.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2pe2 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NUSA | O15530 | 73 | 358 | 556.0 | JNZ:374 | Type1 | Inactive | DFGin | 6.6661 | 14.0143 | BLAminus | -134.94, -176.79 | 67.79, 79.24 | -106.97, 14.51 | 293.69, 91.17 | -56.65, -43.75 | in-in | in | 8.6145 | Saltbr-in | 3.1048 | HRD-in | -75.65, -54.6 | 82.78, -6.2 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8741 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -129.47, 126.95 | APE9-dihe-na | -67.17, -145.64 | APE8-dihe-in | -85.86, 130.62 | APE8-rot-in | 299.93 | APE67-dihe-in | -70.26, -18.43 | -47.43, -45.34 | APE12-dist-in | 9.4758 | APE11-dist-out | 6.257 | APE10-dist-out | 10.2994 | APE9-dist-in | 4.0295 | None | SEP241 | SEP241 | XRAY | 2.75 | 0.177 | 0.236 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nus | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NUUA | O15530 | 73 | 358 | 556.0 | JOZ:361 | Type1 | Inactive | DFGin | 6.8153 | 14.418 | BLAminus | -135.1, 176.45 | 77.67, 76.35 | -106.62, 4.54 | 289.58, 95.96 | -54.87, -35.17 | in-in | in | 8.6632 | Saltbr-in | 2.6457 | HRD-in | -75.97, -55.36 | 84.01, -8.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8245 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -123.64, 126.08 | APE9-dihe-na | -69.19, -150.37 | APE8-dihe-in | -79.82, 127.26 | APE8-rot-in | 298.22 | APE67-dihe-in | -66.17, -14.72 | -39.18, -51.46 | APE12-dist-in | 8.929 | APE11-dist-out | 5.8492 | APE10-dist-out | 10.298 | APE9-dist-in | 3.9915 | None | SEP241 | SEP241 | XRAY | 1.98 | 0.189 | 0.239 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nuu | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NUYA | O15530 | 73 | 358 | 556.0 | JPZ:370 | Type1 | Inactive | DFGin | 6.7298 | 14.5499 | BLAminus | -136.81, -175.62 | 72.08, 77.54 | -106.37, 8.07 | 285.95, 95.42 | -50.93, -42.82 | in-in | in | 8.7638 | Saltbr-in | 2.731 | HRD-in | -78.09, -53.76 | 79.66, -9.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8966 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.52, 118.04 | APE9-dihe-na | -67.36, -159.8 | APE8-dihe-in | -67.79, 132.38 | APE8-rot-in | 304.86 | APE67-dihe-in | -62.4, -17.72 | -54.87, -44.81 | APE12-dist-in | 9.4109 | APE11-dist-out | 5.8201 | APE10-dist-out | 10.2784 | APE9-dist-in | 3.9709 | None | SEP241 | SEP241 | XRAY | 2.1 | 0.187 | 0.225 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nuy | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1UU9A | O15530 | 72 | 357 | 556.0 | BI3:1370 | Type1 | Inactive | DFGin | 6.6788 | 14.783 | BLAminus | -137.61, -169.2 | 68.82, 72.55 | -103.82, -0.34 | 285.88, 98.86 | -59.49, -32.23 | in-in | in | 8.3257 | Saltbr-in | 2.6975 | HRD-in | -73.71, -52.28 | 77.02, -6.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8778 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.15, 123.88 | APE9-dihe-na | -73.46, -162.02 | APE8-dihe-in | -55.23, 126.59 | APE8-rot-in | 305.35 | APE67-dihe-in | -59.52, -20.56 | -41.52, -52.97 | APE12-dist-in | 9.3386 | APE11-dist-out | 5.5023 | APE10-dist-out | 10.2727 | APE9-dist-in | 3.7767 | None | SEP241 | SEP241 | XRAY | 1.95 | 0.176 | 0.224 | A | 286.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 1uu9 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.4e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1UVRA | O15530 | 71 | 359 | 556.0 | BI8:1372 | Type1 | Inactive | DFGin | 6.5811 | 14.4064 | BLAminus | -141.7, -169.27 | 62.75, 72.58 | -105.41, 8.55 | 300.9, 81.55 | -59.95, -35.71 | in-in | in | 8.5947 | Saltbr-in | 2.9835 | HRD-in | -62.43, -49.82 | 76.81, -6.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9337 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -133.17, 120.18 | APE9-dihe-na | -60.87, -168.42 | APE8-dihe-in | -53.67, 135.35 | APE8-rot-in | 308.99 | APE67-dihe-in | -63.6, -1.85 | -44.81, -56.98 | APE12-dist-in | 7.2881 | APE11-dist-out | 6.6429 | APE10-dist-out | 10.6143 | APE9-dist-in | 4.0897 | None | SEP241 | SEP241 | XRAY | 2.81 | 0.176 | 0.248 | A | 289.0 | 285.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 1uvr | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.8e-85 | 289.7 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NUNA | O15530 | 71 | 358 | 556.0 | JMZ:361 | Type1 | Inactive | DFGin | 6.4722 | 14.2209 | BLAminus | -136.64, 178.66 | 75.33, 84.73 | -114.4, 16.28 | 293.69, 90.85 | -60.42, -36.06 | in-in | in | 8.6724 | Saltbr-in | 2.7874 | HRD-in | -68.71, -51.25 | 77.84, -3.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8357 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -115.38, 127.64 | APE9-dihe-na | -69.91, -151.05 | APE8-dihe-in | -80.37, 125.09 | APE8-rot-in | 310.77 | APE67-dihe-in | -66.15, -18.43 | -42.77, -46.09 | APE12-dist-in | 8.9686 | APE11-dist-out | 5.8965 | APE10-dist-out | 10.4173 | APE9-dist-in | 4.3142 | None | SEP241 | SEP241 | XRAY | 2.2 | 0.18 | 0.227 | A | 292.0 | 279.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3nun | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1e-84 | 289.6 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 2XCHA | O15530 | 73 | 359 | 556.0 | CKG:1360 | Type1 | Inactive | DFGin | 6.7339 | 14.5287 | BLAminus | -129.58, 177.2 | 73.14, 77.15 | -102.2, 9.9 | 285.13, 96.86 | -57.37, -39.89 | in-in | in | 8.6981 | Saltbr-in | 2.571 | HRD-in | -76.48, -53.27 | 78.53, -7.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.893 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -122.55, 124.18 | APE9-dihe-na | -77.48, -153.81 | APE8-dihe-in | -63.6, 127.96 | APE8-rot-in | 306.17 | APE67-dihe-in | -61.93, -18.13 | -48.28, -49.39 | APE12-dist-in | 9.2863 | APE11-dist-out | 5.6905 | APE10-dist-out | 10.3423 | APE9-dist-in | 3.8907 | None | SEP241 | SEP241 | XRAY | 2.0 | 0.191 | 0.226 | A | 309.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 2xch | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5HKMA | O15530 | 76 | 358 | 556.0 | 61Y:403 | Type1 | Inactive | DFGin | 6.428 | 14.1502 | BLAminus | -122.57, -157.08 | 51.69, 73.85 | -100.67, 14.09 | 281.12, 81.43 | -62.59, -33.63 | in-in | in | 8.6492 | Saltbr-in | 2.8074 | HRD-in | -66.63, -45.86 | 63.42, -2.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7614 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -140.98, 122.73 | APE9-dihe-na | -75.89, -160.0 | APE8-dihe-in | -62.57, 122.86 | APE8-rot-in | 309.65 | APE67-dihe-in | -56.46, -24.28 | -29.66, -64.05 | APE12-dist-in | 9.6471 | APE11-dist-out | 5.8023 | APE10-dist-out | 10.2714 | APE9-dist-in | 3.7976 | None | SEP241 | SEP241 | XRAY | 2.1 | 0.228 | 0.273 | A | 309.0 | 273.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 5hkm | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5HNGA | O15530 | 71 | 359 | 556.0 | 62O:403 | Type1 | Inactive | DFGin | 6.5015 | 14.356 | BLAminus | -131.37, -170.36 | 61.15, 71.88 | -92.77, 10.44 | 287.92, 92.83 | -55.25, -43.3 | in-in | in | 8.828 | Saltbr-in | 2.8729 | HRD-in | -61.06, -47.37 | 70.67, -1.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7991 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -117.82, 119.15 | APE9-dihe-na | -68.32, -153.72 | APE8-dihe-in | -67.95, 131.45 | APE8-rot-in | 305.81 | APE67-dihe-in | -63.0, -22.16 | -48.07, -47.57 | APE12-dist-in | 9.0259 | APE11-dist-out | 5.7457 | APE10-dist-out | 10.5212 | APE9-dist-in | 4.0322 | None | SEP241 | SEP241 | XRAY | 3.01 | 0.176 | 0.243 | A | 309.0 | 281.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 5hng | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5HO7A | O15530 | 71 | 359 | 556.0 | 63L:701 | Type1 | Inactive | DFGin | 6.4996 | 13.9982 | BLAminus | -138.45, -177.98 | 79.97, 72.22 | -103.24, 8.72 | 293.52, 91.58 | -60.99, -44.96 | in-in | in | 8.5843 | Saltbr-in | 3.0686 | HRD-in | -62.96, -39.76 | 64.33, -4.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9376 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -122.91, 120.25 | APE9-dihe-na | -71.94, -150.13 | APE8-dihe-in | -74.96, 128.19 | APE8-rot-in | 303.71 | APE67-dihe-in | -61.52, -27.36 | -46.49, -48.45 | APE12-dist-in | 9.4591 | APE11-dist-out | 6.0158 | APE10-dist-out | 10.3175 | APE9-dist-in | 4.1229 | None | SEP241 | SEP241 | XRAY | 3.0 | 0.175 | 0.233 | A | 309.0 | 281.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 5ho7 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 5HO8A | O15530 | 71 | 358 | 556.0 | 63E:701 | Type1 | Inactive | DFGin | 6.3257 | 13.7271 | BLAminus | -137.78, 179.62 | 80.28, 69.7 | -100.25, 11.3 | 296.62, 94.66 | -58.72, -47.18 | in-in | in | 8.7434 | Saltbr-in | 3.0233 | HRD-in | -65.39, -42.86 | 64.55, -6.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8667 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -124.41, 121.86 | APE9-dihe-na | -70.34, -152.74 | APE8-dihe-in | -66.74, 122.4 | APE8-rot-in | 293.45 | APE67-dihe-in | -65.08, -24.35 | -41.28, -45.91 | APE12-dist-in | 9.1451 | APE11-dist-out | 5.9265 | APE10-dist-out | 10.2379 | APE9-dist-in | 4.0594 | None | SEP241 | SEP241 | XRAY | 2.7 | 0.184 | 0.229 | A | 309.0 | 279.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5ho8 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1OKYA | O15530 | 72 | 360 | 556.0 | STU:1368 | Type1 | Inactive | DFGin | 6.1532 | 14.4616 | BLAminus | -148.97, -170.84 | 70.56, 80.45 | -102.75, 23.82 | 286.84, 96.04 | -69.28, -20.21 | in-in | in | 8.6718 | Saltbr-in | 2.6729 | HRD-in | -67.69, -57.78 | 80.28, 0.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9341 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -113.7, -80.59 | APE9-dihe-na | 115.49, 169.91 | APE8-dihe-in | -54.49, 123.73 | APE8-rot-in | 316.76 | APE67-dihe-in | -63.35, -17.55 | -42.07, -50.54 | APE12-dist-in | 9.2892 | APE11-dist-out | 5.5558 | APE10-dist-out | 9.7186 | APE9-dist-in | 4.222 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.219 | 0.255 | A | 310.0 | 283.0 | 6 | 30 | 24 | 6 | [[82, 342]] | 1.0 | 1oky | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1OKZA | O15530 | 73 | 359 | 556.0 | UCN:1370 | Type1 | Inactive | DFGin | 6.5441 | 14.1675 | BLAminus | -141.57, -164.78 | 67.55, 76.85 | -103.78, 11.05 | 287.85, 85.4 | -63.67, 2.06 | in-in | in | 8.7271 | Saltbr-in | 2.7175 | HRD-in | -70.44, -54.0 | 75.32, 3.69 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9208 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -147.16, 105.01 | APE9-dihe-na | -62.12, -140.62 | APE8-dihe-in | -78.85, 125.76 | APE8-rot-in | 304.75 | APE67-dihe-in | -63.07, -21.46 | -38.09, -52.99 | APE12-dist-in | 9.5567 | APE11-dist-out | 6.099 | APE10-dist-out | 10.4075 | APE9-dist-in | 4.1656 | None | SEP241 | SEP241 | XRAY | 2.51 | 0.19 | 0.257 | A | 310.0 | 278.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 1okz | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1UU3A | O15530 | 73 | 360 | 556.0 | LY4:1374 | Type1 | Inactive | DFGin | 6.5956 | 14.9714 | BLAminus | -134.47, -173.45 | 74.38, 73.99 | -109.66, 0.57 | 283.46, 101.61 | -63.98, -27.2 | in-in | in | 8.2752 | Saltbr-in | 2.8167 | HRD-in | -64.65, -55.05 | 74.86, -6.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8643 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -122.92, 125.5 | APE9-dihe-na | -77.61, -163.62 | APE8-dihe-in | -56.98, 127.76 | APE8-rot-in | 299.91 | APE67-dihe-in | -61.39, -22.49 | -53.63, -41.57 | APE12-dist-in | 9.2019 | APE11-dist-out | 5.4661 | APE10-dist-out | 10.4073 | APE9-dist-in | 4.0483 | None | SEP241 | SEP241 | XRAY | 1.7 | 0.174 | 0.202 | A | 310.0 | 278.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 1uu3 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1UU7A | O15530 | 73 | 359 | 556.0 | BI2:1364 | Type1 | Inactive | DFGin | 6.5571 | 14.7415 | BLAminus | -136.5, -171.94 | 74.29, 73.79 | -109.8, -2.64 | 287.37, 96.13 | -53.85, -39.14 | in-in | in | 8.463 | Saltbr-in | 2.8801 | HRD-in | -68.07, -51.28 | 73.99, -8.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8332 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -131.82, 121.67 | APE9-dihe-na | -67.64, -173.23 | APE8-dihe-in | -49.06, 125.05 | APE8-rot-in | 301.64 | APE67-dihe-in | -67.12, -19.88 | -49.14, -41.33 | APE12-dist-in | 8.9136 | APE11-dist-out | 5.317 | APE10-dist-out | 10.2667 | APE9-dist-in | 3.9105 | None | SEP241 | SEP241 | XRAY | 1.9 | 0.235 | 0.279 | A | 310.0 | 282.0 | 5 | 30 | 25 | 5 | [[82, 342]] | 1.0 | 1uu7 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 1UU8A | O15530 | 72 | 358 | 556.0 | BI1:1368 | Type1 | Inactive | DFGin | 6.6469 | 14.4714 | BLAminus | -136.37, -165.37 | 63.01, 71.98 | -101.9, 2.54 | 288.65, 101.81 | -58.08, -33.97 | in-in | in | 8.8152 | Saltbr-in | 2.7275 | HRD-in | -71.97, -53.07 | 75.47, 11.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8428 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -142.67, 117.85 | APE9-dihe-na | -65.71, -160.29 | APE8-dihe-in | -63.31, 129.15 | APE8-rot-in | 297.13 | APE67-dihe-in | -68.38, -3.88 | -40.88, -48.91 | APE12-dist-in | 9.2375 | APE11-dist-out | 5.6529 | APE10-dist-out | 10.0877 | APE9-dist-in | 3.759 | None | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.258 | A | 310.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 1uu8 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NAYA | O15530 | 76 | 362 | 556.0 | MP6:1 | Type1 | Inactive | DFGin | 6.7641 | 14.6579 | BLAminus | -146.79, -173.04 | 72.2, 70.67 | -103.69, 5.05 | 296.95, 109.64 | -60.79, -27.91 | in-in | in | 8.5567 | Saltbr-in | 2.5649 | HRD-in | -62.07, -50.65 | 74.17, -9.68 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.74 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -127.84, 118.23 | APE9-dihe-na | -69.99, -167.96 | APE8-dihe-in | -54.98, 129.37 | APE8-rot-in | 302.57 | APE67-dihe-in | -65.83, -27.98 | -54.2, -37.6 | APE12-dist-in | 8.6002 | APE11-dist-out | 5.6186 | APE10-dist-out | 10.5309 | APE9-dist-in | 3.8392 | None | SEP241 | SEP241 | XRAY | 2.6 | 0.211 | 0.274 | A | 311.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3nay | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NAYB | O15530 | 76 | 362 | 556.0 | MP6:2 | Type1 | Inactive | DFGin | 6.8794 | 14.3665 | BLAminus | -131.67, -178.35 | 72.0, 77.09 | -107.77, 17.41 | 299.66, 102.49 | -69.46, -28.42 | in-in | in | 8.3299 | Saltbr-in | 2.8238 | HRD-in | -70.5, -49.88 | 76.39, -13.79 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8417 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 114.84, 100.21 | APE9-dihe-na | -68.09, -163.03 | APE8-dihe-in | -59.66, 125.08 | APE8-rot-in | 300.78 | APE67-dihe-in | -68.69, -23.52 | -42.99, -40.54 | APE12-dist-in | 8.7294 | APE11-dist-out | 5.8365 | APE10-dist-out | 10.6017 | APE9-dist-in | 3.8844 | None | SEP241 | SEP241 | XRAY | 2.6 | 0.211 | 0.274 | B | 311.0 | 279.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3nay | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3RWPA | O15530 | 73 | 359 | 556.0 | ABQ:360 | Type1 | Inactive | DFGin | 6.6301 | 14.6122 | BLAminus | -138.06, -171.84 | 73.21, 68.9 | -101.84, 0.77 | 284.24, 99.91 | -67.12, -24.97 | in-in | in | 8.4872 | Saltbr-in | 2.668 | HRD-in | -72.19, -48.95 | 75.52, -7.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8439 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -116.4, 122.62 | APE9-dihe-na | -64.5, -165.33 | APE8-dihe-in | -62.97, 132.8 | APE8-rot-in | 302.69 | APE67-dihe-in | -57.73, -26.43 | -57.73, -39.86 | APE12-dist-in | 9.571 | APE11-dist-out | 5.748 | APE10-dist-out | 10.613 | APE9-dist-in | 4.2017 | None | SEP241 | SEP241 | XRAY | 1.92 | 0.174 | 0.213 | A | 311.0 | 278.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3rwp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3RWQA | O15530 | 72 | 359 | 556.0 | 3RW:1 | Type1 | Inactive | DFGin | 6.5891 | 14.463 | BLAminus | -143.65, -172.61 | 68.52, 70.31 | -102.07, 3.38 | 289.03, 95.5 | -56.64, -39.2 | in-in | in | 8.5646 | Saltbr-in | 2.7282 | HRD-in | -70.4, -52.28 | 81.8, -9.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.02 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -127.88, 122.18 | APE9-dihe-na | -69.74, -149.03 | APE8-dihe-in | -75.72, 125.93 | APE8-rot-in | 318.02 | APE67-dihe-in | -73.55, -21.89 | -37.75, -44.68 | APE12-dist-in | 9.2067 | APE11-dist-out | 5.8786 | APE10-dist-out | 10.5237 | APE9-dist-in | 4.0165 | None | SEP241 | SEP241 | XRAY | 2.55 | 0.196 | 0.256 | A | 311.0 | 284.0 | 4 | 30 | 26 | 4 | [[82, 342]] | 1.0 | 3rwq | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3H9OA | O15530 | 75 | 359 | 556.0 | 9BD:1 | Type1 | Inactive | DFGin | 6.5678 | 14.261 | BLAminus | -131.94, -168.71 | 66.62, 79.57 | -104.6, 18.2 | 283.3, 82.81 | -72.27, -11.03 | in-in | in | 8.8763 | Saltbr-in | 2.5436 | HRD-in | -78.26, -52.42 | 80.3, -1.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8097 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 77.5, 119.89 | APE9-dihe-na | -89.12, -112.65 | APE8-dihe-in | -101.23, 134.92 | APE8-rot-in | 301.13 | APE67-dihe-in | -62.27, -18.27 | -50.83, -50.03 | APE12-dist-in | 9.6432 | APE11-dist-out | 6.2678 | APE10-dist-out | 10.1736 | APE9-dist-in | 3.934 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.211 | 0.256 | A | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3h9o | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 2R7BA | O15530 | 75 | 359 | 556.0 | 253:701 | Type1 | Inactive | DFGin | 6.1992 | 14.366 | BLAminus | -133.94, -179.49 | 77.82, 81.49 | -108.24, 22.02 | 291.13, 86.98 | -68.69, -10.97 | in-in | in | 8.8662 | Saltbr-in | 2.5883 | HRD-in | -75.75, -47.44 | 52.14, 30.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7982 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 148.51, 113.35 | APE9-dihe-na | -77.58, -157.1 | APE8-dihe-in | -58.21, 135.29 | APE8-rot-in | 301.99 | APE67-dihe-in | -57.75, -20.67 | -44.89, -55.44 | APE12-dist-in | 9.1968 | APE11-dist-out | 5.7727 | APE10-dist-out | 9.8875 | APE9-dist-in | 4.0959 | None | SEP241 | SEP241 | XRAY | 2.7 | 0.225 | 0.25 | A | 312.0 | 275.0 | 10 | 30 | 20 | 10 | [[82, 342]] | 1.0 | 2r7b | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3IONA | O15530 | 75 | 359 | 556.0 | 8H1:1 | Type1 | Inactive | DFGin | 6.3855 | 14.0119 | BLAminus | -129.57, -169.56 | 64.12, 80.16 | -106.23, 22.91 | 285.85, 87.72 | -68.81, -24.37 | in-in | in | 8.9313 | Saltbr-in | 3.3369 | HRD-in | -74.01, -54.84 | 77.47, 1.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7001 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoi | APE10-dihe-na | 999.0, 132.89 | APE9-dihe-na | -88.46, -116.13 | APE8-dihe-in | -104.9, 134.52 | APE8-rot-in | 307.56 | APE67-dihe-in | -73.92, -18.65 | -45.98, -45.06 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 10.0803 | APE9-dist-in | 3.6029 | None | None | None | XRAY | 2.4 | 0.246 | 0.282 | A | 312.0 | 274.0 | 11 | 30 | 19 | 11 | [[82, 342]] | 1.0 | 3ion | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3IOPA | O15530 | 75 | 359 | 556.0 | 8I1:1 | Type1 | Inactive | DFGin | 6.6057 | 14.3164 | BLAminus | -125.3, -165.97 | 58.12, 80.1 | -105.24, 23.38 | 285.73, 86.81 | -73.19, -11.32 | in-in | in | 8.8064 | Saltbr-in | 2.6809 | HRD-in | -71.7, -52.98 | 78.46, -5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8075 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | 67.02, 113.91 | APE9-dihe-na | -74.5, -127.28 | APE8-dihe-in | -97.61, 129.5 | APE8-rot-in | 303.0 | APE67-dihe-in | -63.74, -18.61 | -44.16, -50.92 | APE12-dist-in | 9.5697 | APE11-dist-out | 5.9687 | APE10-dist-out | 10.4647 | APE9-dist-in | 3.7908 | None | SEP241 | SEP241 | XRAY | 2.2 | 0.24 | 0.278 | A | 312.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3iop | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QCQA | O15530 | 73 | 358 | 556.0 | 3Q0:370 | Type1 | Inactive | DFGin | 6.286 | 13.9428 | BLAminus | -130.07, -172.39 | 67.81, 84.85 | -116.19, 10.14 | 290.92, 91.68 | -60.0, -35.96 | in-in | in | 8.6682 | Saltbr-in | 2.8169 | HRD-in | -76.77, -43.93 | 72.04, -4.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9565 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -127.34, 117.15 | APE9-dihe-na | -68.0, -161.08 | APE8-dihe-in | -59.72, 132.52 | APE8-rot-in | 308.25 | APE67-dihe-in | -73.95, -13.03 | -56.44, -42.24 | APE12-dist-in | 9.3219 | APE11-dist-out | 6.2157 | APE10-dist-out | 10.3256 | APE9-dist-in | 4.2085 | None | SEP241 | SEP241 | XRAY | 2.501 | 0.181 | 0.251 | A | 312.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qcq | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QCSA | O15530 | 73 | 358 | 556.0 | 3Q1:370 | Type1 | Inactive | DFGin | 6.4977 | 14.3423 | BLAminus | -129.15, -172.55 | 69.95, 84.25 | -118.54, 4.81 | 283.02, 93.04 | -59.77, -28.42 | in-in | in | 8.591 | Saltbr-in | 2.8075 | HRD-in | -71.62, -47.65 | 74.15, -7.51 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8349 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -125.7, 120.85 | APE9-dihe-na | -72.97, -164.1 | APE8-dihe-in | -54.02, 130.58 | APE8-rot-in | 312.22 | APE67-dihe-in | -61.81, -24.07 | -54.55, -47.19 | APE12-dist-in | 9.2353 | APE11-dist-out | 6.3341 | APE10-dist-out | 10.5363 | APE9-dist-in | 4.4067 | None | SEP241 | SEP241 | XRAY | 2.487 | 0.182 | 0.251 | A | 312.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qcs | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3PWYA | O15530 | 71 | 359 | 556.0 | SYP:1 | Type1 | Inactive | DFGin | 6.477 | 14.4835 | BLAminus | -124.65, -178.35 | 67.96, 96.3 | -130.58, 11.45 | 300.55, 97.42 | -64.93, -31.03 | in-in | in | 8.587 | Saltbr-in | 2.6927 | HRD-in | -58.86, -48.53 | 68.39, -3.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.761 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -116.65, 129.21 | APE9-dihe-na | -78.78, -151.6 | APE8-dihe-in | -77.12, 126.15 | APE8-rot-in | 307.61 | APE67-dihe-in | -78.87, -27.54 | -44.08, -37.51 | APE12-dist-in | 10.3267 | APE11-dist-out | 5.848 | APE10-dist-out | 10.5798 | APE9-dist-in | 3.8548 | E166C,C260S | None | None | XRAY | 3.5 | 0.226 | 0.276 | A | 311.0 | 281.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 3pwy | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.5e-84 | 286.4 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 2XCKA | O15530 | 76 | 359 | 556.0 | MH4:1360 | Type1 | Inactive | DFGin | 6.7771 | 14.7278 | BLAminus | -138.18, -175.27 | 71.05, 75.56 | -104.69, 7.11 | 286.41, 101.4 | -56.07, -44.06 | in-in | in | 8.7216 | Saltbr-in | 2.7225 | HRD-in | -74.69, -54.88 | 79.61, -3.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.891 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -108.24, 134.08 | APE9-dihe-na | -87.44, -159.07 | APE8-dihe-in | -56.55, 126.47 | APE8-rot-in | 304.89 | APE67-dihe-in | -62.34, -18.12 | -47.8, -48.47 | APE12-dist-in | 9.3328 | APE11-dist-out | 5.5135 | APE10-dist-out | 10.4019 | APE9-dist-in | 3.8752 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.195 | 0.24 | A | 309.0 | 276.0 | 8 | 30 | 22 | 8 | [[82, 342]] | 1.0 | 2xck | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.8e-83 | 285.5 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QCXA | O15530 | 73 | 358 | 556.0 | 3Q2:370 | Type1.5_Back | Inactive | DFGin | 6.5656 | 14.4479 | BLAminus | -128.85, -170.97 | 71.83, 79.3 | -115.33, 7.3 | 284.13, 92.7 | -60.73, -28.9 | in-in | in | 8.4024 | Saltbr-in | 2.7064 | HRD-in | -68.18, -50.11 | 76.96, -14.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8031 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -135.89, 122.06 | APE9-dihe-na | -67.11, -167.83 | APE8-dihe-in | -62.01, 135.81 | APE8-rot-in | 308.12 | APE67-dihe-in | -61.25, -24.88 | -55.14, -44.7 | APE12-dist-in | 9.4652 | APE11-dist-out | 6.3732 | APE10-dist-out | 10.3227 | APE9-dist-in | 4.269 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.184 | 0.225 | A | 312.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qcx | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QCYA | O15530 | 73 | 358 | 556.0 | 3Q3:371 | Type1.5_Front | Inactive | DFGin | 6.3885 | 14.5918 | BLAminus | -136.93, -173.16 | 70.99, 75.14 | -110.32, 14.26 | 284.13, 86.28 | -62.73, -28.34 | in-in | in | 8.4189 | Saltbr-in | 2.559 | HRD-in | -71.32, -53.51 | 82.01, -8.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.825 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoi | APE10-dihe-na | 999.0, 125.83 | APE9-dihe-na | -76.07, -148.77 | APE8-dihe-in | -79.07, 127.11 | APE8-rot-in | 312.38 | APE67-dihe-in | -58.65, -24.48 | -40.2, -55.49 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 10.317 | APE9-dist-in | 4.4989 | None | SEP241 | SEP241 | XRAY | 2.2 | 0.181 | 0.212 | A | 312.0 | 275.0 | 11 | 30 | 19 | 11 | [[82, 342]] | 1.0 | 3qcy | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QD3A | O15530 | 71 | 358 | 556.0 | 3Q5:360 | Type1.5_Front | Inactive | DFGin | 6.6397 | 14.7756 | BLAminus | -136.15, -173.35 | 75.08, 78.84 | -114.86, 7.79 | 284.21, 92.48 | -60.8, -30.07 | in-in | in | 8.4699 | Saltbr-in | 2.5474 | HRD-in | -69.84, -52.9 | 76.92, -8.58 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8112 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -114.87, 124.76 | APE9-dihe-na | -70.78, -165.19 | APE8-dihe-in | -61.65, 129.32 | APE8-rot-in | 306.27 | APE67-dihe-in | -62.1, -22.78 | -46.86, -49.49 | APE12-dist-in | 8.9916 | APE11-dist-out | 5.7339 | APE10-dist-out | 10.4141 | APE9-dist-in | 4.0376 | None | SEP241 | SEP241 | XRAY | 2.0 | 0.185 | 0.211 | A | 312.0 | 279.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 3qd3 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3NAXA | O15530 | 76 | 360 | 556.0 | MP7:363 | Type2 | Inactive | DFGout | 15.1303 | 9.5196 | BBAminus | -103.03, 154.8 | -117.91, 140.31 | -115.35, 34.44 | 271.6, 90.85 | 93.28, 8.79 | out-out | out | 17.0845 | Saltbr-out | 10.2575 | HRD-in | -72.23, -50.17 | 78.89, -10.91 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.8524 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.19, -19.08 | 999.0, -56.98 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.75 | 0.166 | 0.195 | A | 311.0 | 278.0 | 7 | 30 | 23 | 7 | [[82, 342]] | 1.0 | 3nax | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QC4A | O15530 | 76 | 359 | 556.0 | MP7:60001 | Type2 | Inactive | DFGout | 15.1445 | 8.4181 | BBAminus | -116.84, 146.54 | -96.89, 143.53 | -123.04, 29.2 | 249.8, 111.12 | 113.47, -5.45 | out-out | out | 19.868 | Saltbr-out | 17.8176 | HRD-in | -79.45, -51.8 | 76.86, -8.13 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.035 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.28, 161.52 | APE9-dihe-na | 127.76, -165.1 | APE8-dihe-in | -132.92, 137.19 | APE8-rot-in | 293.31 | APE67-dihe-in | -63.51, -29.78 | -55.77, -40.56 | APE12-dist-in | 7.6463 | APE11-dist-in | 10.8912 | APE10-dist-in | 5.0977 | APE9-dist-in | 3.6028 | E303A,K304A | SEP241 | SEP241 | XRAY | 1.8 | 0.174 | 0.213 | A | 314.0 | 277.0 | 7 | 30 | 23 | 7 | [[82, 342]] | 1.0 | 3qc4 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 5.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QC4B | O15530 | 51 | 359 | 556.0 | MP7:60002 | Type2 | Inactive | DFGout | 15.5034 | 8.2994 | None | -106.7, 145.77 | -96.8, 153.42 | -131.45, 34.1 | 235.15, 115.54 | 107.65, 4.91 | out-out | out | 18.0578 | Saltbr-out | 15.1697 | HRD-in | -74.82, -53.49 | 77.73, -9.15 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9345 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.95, 158.08 | APE9-dihe-na | 130.3, -155.43 | APE8-dihe-in | -143.11, 135.86 | APE8-rot-in | 293.55 | APE67-dihe-in | -66.08, -20.71 | -55.87, -43.65 | APE12-dist-in | 7.6714 | APE11-dist-in | 10.9464 | APE10-dist-in | 5.0678 | APE9-dist-in | 3.5388 | E303A,K304A | SEP241 | SEP241 | XRAY | 1.8 | 0.174 | 0.213 | B | 314.0 | 274.0 | 15 | 30 | 23 | 7 | [[82, 342]] | 1.0 | 3qc4 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 5.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 4CT1A | O15530 | 76 | 359 | 556.0 | ATP:500,31S:600 | ATPlike,Allosteric | None | DFGin | 6.6022 | 14.9785 | BLAminus | -141.71, -172.51 | 72.43, 72.08 | -107.06, 8.07 | 284.9, 97.13 | -62.67, -20.12 | in-none | in | 8.1463 | Saltbr-none | 999.0 | HRD-in | -74.62, -54.47 | 79.43, -8.97 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.9992 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -143.29, 160.89 | APE9-dihe-na | 137.85, -171.95 | APE8-dihe-in | -126.26, 129.35 | APE8-rot-in | 296.2 | APE67-dihe-in | -61.08, -24.26 | -47.64, -46.5 | APE12-dist-in | 7.3566 | APE11-dist-in | 10.4885 | APE10-dist-in | 5.0182 | APE9-dist-in | 3.4798 | L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A | SEP241 | SEP241 | XRAY | 1.85 | 0.172 | 0.215 | A | 311.0 | 284.0 | 0 | 30 | 30 | 0 | [[82, 342]] | 1.0 | 4ct1 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 9.5e-84 | 286.4 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QD0A | O15530 | 73 | 358 | 556.0 | 3Q4:370 | Type1.5_Front | None | DFGin | 6.5836 | 14.7913 | BLAminus | -135.89, -173.14 | 73.55, 73.02 | -106.35, 12.12 | 281.49, 88.39 | -54.84, -35.9 | in-in | in | 8.5258 | Saltbr-in | 2.5731 | HRD-in | -72.98, -50.98 | 74.13, -9.69 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8508 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -154.13 | APE8-dihe-in | -74.4, 123.75 | APE8-rot-in | 309.46 | APE67-dihe-in | -59.36, -28.41 | -43.01, -50.59 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 4.7652 | None | SEP241 | SEP241 | XRAY | 1.99 | 0.191 | 0.231 | A | 312.0 | 274.0 | 12 | 30 | 18 | 12 | [[82, 342]] | 1.0 | 3qd0 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| PDPK1 | PDPK1_HUMAN | 3QD4A | O15530 | 71 | 358 | 556.0 | 3Q6:360 | Type1.5_Front | None | DFGin | 6.4034 | 14.6264 | BLAminus | -137.72, -173.39 | 72.99, 75.84 | -110.69, 10.4 | 285.12, 91.81 | -64.41, -29.28 | in-in | in | 8.5579 | Saltbr-in | 2.7898 | HRD-in | -69.09, -51.69 | 76.33, -7.4 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9076 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnni | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -153.49 | APE8-dihe-in | -83.46, 122.24 | APE8-rot-in | 298.92 | APE67-dihe-in | -62.96, -22.94 | -34.73, -56.97 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-in | 4.1203 | None | SEP241 | SEP241 | XRAY | 2.3 | 0.199 | 0.244 | A | 312.0 | 276.0 | 12 | 30 | 18 | 12 | [[82, 342]] | 1.0 | 3qd4 | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 1.3e-84 | 289.3 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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