| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PDGFRA | AF-P16234-K1A | P16234 | 585 | 960 | 1089.0 | No_ligand | No_ligand | Active | DFGin | 6.6997 | 13.6749 | BLAminus | -137.69, -178.12 | 65.56, 55.38 | -76.94, 17.55 | 294.68, 89.62 | -62.07, -30.49 | in-in | in | 7.3733 | Saltbr-in | 2.6326 | HRD-in | -76.76, -43.79 | 66.53, -13.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9412 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.33, 108.79 | APE9-dihe-in | -125.4, 152.2 | APE8-dihe-in | -75.15, 89.08 | APE8-rot-na | 36.01 | APE67-dihe-in | -66.01, -16.63 | -47.84, -37.12 | APE12-dist-na | 14.0618 | APE11-dist-na | 7.9646 | APE10-dist-na | 9.9372 | APE9-dist-in | 5.9594 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 376.0 | 376.0 | 0 | 30 | 30 | 0 | [[593, 952]] | 1.0 | AF-P16234-K1 | TYR_PDGFRA_HUMAN | TYR | 7.7e-106 | 359.3 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | AF-P16234-K3A | P16234 | 585 | 960 | 1089.0 | No_ligand | No_ligand | Active | DFGin | 6.6303 | 13.2587 | BLAminus | -128.58, 177.17 | 60.47, 65.55 | -71.97, 11.95 | 293.94, 94.32 | -62.2, -32.16 | in-in | in | 7.8236 | Saltbr-in | 2.7054 | HRD-in | -82.85, -43.12 | 66.78, -5.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9021 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -63.73, 118.36 | APE9-dihe-in | -107.5, 147.11 | APE8-dihe-in | -82.35, 65.15 | APE8-rot-na | 33.41 | APE67-dihe-in | -66.83, -20.14 | -51.1, -37.81 | APE12-dist-na | 14.3911 | APE11-dist-na | 8.9234 | APE10-dist-na | 12.0386 | APE9-dist-in | 7.1492 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 376.0 | 376.0 | 0 | 30 | 30 | 0 | [[593, 952]] | 1.0 | AF-P16234-K3 | TYR_PDGFRA_HUMAN | TYR | 7.7e-106 | 359.3 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 8PQHA | P16234 | 555 | 971 | 1089.0 | 9JI:1001 | Type1 | Active | DFGin | 7.1176 | 13.5042 | BLAminus | -137.77, -173.06 | 54.37, 84.67 | -94.17, 27.12 | 292.06, 83.63 | -63.26, -46.8 | in-in | in | 7.9228 | Saltbr-in | 3.2447 | HRD-in | -71.43, -45.05 | 70.07, -2.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9791 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -118.37, 127.86 | APE9-dihe-in | -120.13, 154.51 | APE8-dihe-in | -81.88, 68.37 | APE8-rot-na | 25.31 | APE67-dihe-in | -67.91, -9.11 | -50.35, -46.55 | APE12-dist-na | 6.6948 | APE11-dist-na | 11.7329 | APE10-dist-na | 11.1167 | APE9-dist-in | 7.073 | T674I | None | None | XRAY | 2.5 | 0.22 | 0.249 | A | 352.0 | 321.0 | 23 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 8pqh | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 8PQIA | P16234 | 567 | 969 | 1089.0 | 9OO:1001 | Type1 | Active | DFGin | 6.9059 | 13.5927 | BLAminus | -132.24, 178.87 | 62.52, 88.22 | -103.25, 28.49 | 291.7, 71.46 | -68.1, -30.59 | in-in | in | 7.9933 | Saltbr-in | 2.898 | HRD-in | -71.63, -43.38 | 66.22, 2.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8201 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -98.65, 130.26 | APE9-dihe-in | -117.66, 147.18 | APE8-dihe-in | -84.02, 76.87 | APE8-rot-na | 33.16 | APE67-dihe-in | -69.02, -9.85 | -66.15, -32.32 | APE12-dist-na | 999.0 | APE11-dist-na | 9.4755 | APE10-dist-na | 11.4786 | APE9-dist-in | 7.1354 | T674I | None | None | XRAY | 2.6 | 0.232 | 0.254 | A | 352.0 | 299.0 | 32 | 30 | 20 | 10 | [[593, 952]] | 1.0 | 8pqi | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 6JOIA | P16234 | 569 | 973 | 1089.0 | 6T2:1001 | Type1 | Inactive | DFGin | 5.8932 | 12.4237 | BLAplus | -149.03, 179.69 | 59.48, 39.87 | -90.32, -0.87 | 38.91, 91.7 | -108.94, 138.34 | in-out | in | 7.8145 | Saltbr-out | 4.0493 | HRD-in | -63.69, -47.81 | 78.72, -13.59 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.07, 131.06 | APE9-dihe-in | -119.74, 141.05 | APE8-dihe-in | -77.37, 79.89 | APE8-rot-na | 19.31 | APE67-dihe-in | -62.19, -30.0 | -59.33, -40.19 | APE12-dist-na | 999.0 | APE11-dist-na | 13.197 | APE10-dist-na | 15.7508 | APE9-dist-in | 7.4573 | T674I | None | None | XRAY | 3.1 | 0.224 | 0.244 | A | 375.0 | 296.0 | 37 | 30 | 15 | 15 | [[593, 952]] | 1.0 | 6joi | TYR_PDGFRA_HUMAN | TYR | 2.2e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 8XRRA | A0A0B4J203 | 338 | 730 | 849.0 | A1LV8:61001 | Type1 | Inactive | DFGin | 6.0782 | 12.8103 | BLBminus | -136.82, -170.16 | 60.75, 77.27 | -91.15, -163.07 | 294.15, 83.07 | 112.28, -36.82 | in-in | in | 7.2816 | Saltbr-in | 2.8565 | HRD-in | -63.02, -44.11 | 69.37, 4.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9784 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.33, 138.03 | APE9-dihe-in | -122.05, 151.58 | APE8-dihe-in | -77.69, 73.7 | APE8-rot-na | 29.73 | APE67-dihe-in | -63.37, -4.92 | -54.48, -47.94 | APE12-dist-na | 999.0 | APE11-dist-na | 8.1413 | APE10-dist-na | 10.8954 | APE9-dist-in | 6.9028 | None | None | None | XRAY | 2.57 | 0.238 | 0.26 | A | 356.0 | 285.0 | 36 | 30 | 19 | 11 | [[353, 712]] | 1.0 | 8xrr | TYR_PDGFRA_HUMAN | TYR | 3.7e-106 | 360.5 | 1.0 | 260.0 | 260.0 | 595 | 596 | 597 | 599 | 601 | 387 | 404 | 408 | 575 | 577 | 576 | 578.0 | 637 | 625 | 620 | 619 | 618 | 617 | 616 | 615 | 614 | 435 | receptor protein-tyrosine kinase |
| PDGFRA | 9GZHA | P16234 | 583 | 958 | 1089.0 | A1IRC:1001 | Type2 | Inactive | DFGout | 15.6481 | 9.5759 | BBAminus | -142.99, 176.85 | -144.44, 111.57 | -68.84, -35.83 | 280.23, 92.0 | 59.84, -119.26 | in-in | in | 7.8509 | Saltbr-in | 2.9454 | HRD-in | -72.49, -49.27 | 74.96, -9.55 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.0825 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -107.38, 139.27 | APE9-dihe-in | -132.11, 144.36 | APE8-dihe-in | -77.41, 71.6 | APE8-rot-na | 33.5 | APE67-dihe-in | -62.63, -15.56 | -62.2, -45.12 | APE12-dist-na | 15.5208 | APE11-dist-na | 11.6099 | APE10-dist-na | 11.6095 | APE9-dist-in | 7.5857 | T674I | None | None | XRAY | 2.2 | 0.183 | 0.215 | A | 355.0 | 282.0 | 22 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 9gzh | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 5GRNA | P16234 | 583 | 958 | 1089.0 | 748:1001 | Type2 | Inactive | DFGout | 16.3718 | 10.5289 | BBAminus | -143.58, -173.72 | -146.28, 106.78 | -54.79, -37.05 | 281.52, 58.25 | 60.16, -122.4 | in-in | in | 7.9371 | Saltbr-in | 2.7389 | HRD-in | -77.42, -50.02 | 77.14, -8.21 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.3417 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -107.12, 130.75 | APE9-dihe-in | -120.55, 148.05 | APE8-dihe-in | -80.95, 69.87 | APE8-rot-na | 36.32 | APE67-dihe-in | -65.74, -12.4 | -60.52, -41.33 | APE12-dist-na | 15.1679 | APE11-dist-na | 11.2852 | APE10-dist-na | 11.4357 | APE9-dist-in | 7.6446 | None | None | None | XRAY | 1.77 | 0.158 | 0.179 | A | 356.0 | 286.0 | 18 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 5grn | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 6JOLA | P16234 | 583 | 957 | 1089.0 | STI:1001 | Type2 | Inactive | DFGout | 16.377 | 10.1801 | BBAminus | -142.0, 174.77 | -141.65, 105.94 | -59.47, -37.67 | 274.19, 66.43 | 59.87, -122.37 | in-in | in | 7.9131 | Saltbr-in | 2.7813 | HRD-in | -68.97, -54.53 | 78.87, -11.97 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.9266 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.21, 134.53 | APE9-dihe-in | -124.89, 147.83 | APE8-dihe-in | -86.42, 79.14 | APE8-rot-na | 35.14 | APE67-dihe-in | -66.62, -11.35 | -62.29, -37.28 | APE12-dist-na | 16.0066 | APE11-dist-na | 12.1566 | APE10-dist-na | 11.9857 | APE9-dist-in | 7.6302 | None | None | None | XRAY | 1.9 | 0.215 | 0.236 | A | 356.0 | 279.0 | 24 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6jol | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 8PQKA | P16234 | 554 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 15.5834 | 8.1772 | None | -154.9, 179.4 | -116.45, 101.18 | -96.78, 25.45 | 224.18, 59.38 | -62.44, -23.73 | in-in | in | 7.7684 | Saltbr-in | 2.5801 | HRD-in | -75.59, -53.47 | 73.99, -2.28 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.7619 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -124.57, 123.17 | APE9-dihe-in | -122.51, 149.52 | APE8-dihe-in | -78.18, 70.07 | APE8-rot-na | 31.79 | APE67-dihe-in | -62.15, -17.78 | -60.4, -41.22 | APE12-dist-na | 19.4466 | APE11-dist-na | 15.06 | APE10-dist-na | 13.5403 | APE9-dist-in | 7.4476 | T674I | None | None | XRAY | 2.0 | 0.197 | 0.222 | A | 352.0 | 322.0 | 17 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 8pqk | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 6A32A | P16234 | 554 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 16.6148 | 8.4618 | None | -149.24, -176.86 | -118.22, 104.49 | -91.23, 25.57 | 218.48, 75.46 | -61.15, -35.43 | in-in | in | 8.2677 | Saltbr-in | 2.3994 | HRD-in | -77.45, -54.11 | 74.43, 2.58 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.5149 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.41, 128.42 | APE9-dihe-in | -113.39, 143.39 | APE8-dihe-in | -83.41, 71.44 | APE8-rot-na | 35.27 | APE67-dihe-in | -66.73, -17.33 | -56.98, -40.55 | APE12-dist-na | 17.2193 | APE11-dist-na | 14.1538 | APE10-dist-na | 12.9888 | APE9-dist-in | 7.2815 | T674I | None | None | XRAY | 1.87 | 0.205 | 0.24 | A | 356.0 | 336.0 | 12 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6a32 | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 8PQJA | P16234 | 553 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 15.7273 | 8.2369 | None | -151.0, -178.54 | -115.21, 108.13 | -99.29, 20.66 | 220.99, 51.76 | -57.16, -27.12 | in-in | in | 7.805 | Saltbr-in | 2.6763 | HRD-in | -70.62, -57.5 | 76.76, 1.26 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8216 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -126.61, 120.89 | APE9-dihe-in | -120.18, 150.45 | APE8-dihe-in | -75.53, 66.41 | APE8-rot-na | 31.49 | APE67-dihe-in | -62.28, -19.29 | -62.48, -36.33 | APE12-dist-na | 19.3874 | APE11-dist-na | 15.0565 | APE10-dist-na | 13.613 | APE9-dist-in | 7.4582 | None | None | None | XRAY | 1.82 | 0.185 | 0.215 | A | 352.0 | 329.0 | 14 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 8pqj | TYR_PDGFRA_HUMAN | TYR | 8.8e-107 | 362.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 5K5XA | P16234 | 554 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 15.8713 | 8.3345 | None | -153.24, -177.14 | -114.02, 113.86 | -108.1, 22.87 | 215.74, 54.5 | -59.52, -34.36 | in-in | in | 7.7455 | Saltbr-in | 2.4976 | HRD-in | -70.35, -55.34 | 73.06, -5.1 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.9506 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.49, 130.42 | APE9-dihe-in | -117.78, 136.58 | APE8-dihe-in | -73.77, 63.63 | APE8-rot-na | 32.36 | APE67-dihe-in | -68.21, -12.54 | -54.21, -40.36 | APE12-dist-na | 18.4802 | APE11-dist-na | 15.1785 | APE10-dist-na | 13.332 | APE9-dist-in | 7.4009 | None | None | None | XRAY | 2.168 | 0.193 | 0.224 | A | 356.0 | 345.0 | 3 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 5k5x | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 6JOKA | P16234 | 556 | 973 | 1089.0 | B49:1001 | Type1 | Inactive | DFGout | 17.3303 | 10.1516 | None | -157.96, 162.23 | -90.74, 118.75 | -83.04, 4.75 | 220.32, 127.42 | -60.76, -49.9 | in-out | in | 7.8064 | Saltbr-out | 4.6095 | HRD-in | -71.4, -52.83 | 71.29, -1.66 | out-out-in | SNCooi | out-in | ActLoopNT-out | 16.719 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -133.37, 126.64 | APE9-dihe-in | -119.51, 140.56 | APE8-dihe-in | -75.53, 69.74 | APE8-rot-na | 31.06 | APE67-dihe-in | -63.68, -19.63 | -58.21, -43.02 | APE12-dist-na | 17.5027 | APE11-dist-na | 14.289 | APE10-dist-na | 13.1977 | APE9-dist-in | 7.2863 | None | None | None | XRAY | 3.8 | 0.259 | 0.282 | A | 356.0 | 338.0 | 8 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6jok | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | 6JOJA | P16234 | 554 | 973 | 1089.0 | 6T2:1001 | Type1 | Inactive | None | 20.3126 | 15.0063 | None | -134.96, -163.27 | -129.94, 169.75 | -62.88, -45.52 | 197.17, 82.33 | 72.34, -174.07 | in-in | in | 7.904 | Saltbr-in | 2.5098 | HRD-in | -72.82, -51.47 | 79.17, -0.33 | in-out-in | SNCioi | out-in | ActLoopNT-out | 18.4772 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.85, 133.76 | APE9-dihe-in | -123.13, 133.08 | APE8-dihe-in | -84.33, 80.22 | APE8-rot-na | 30.95 | APE67-dihe-in | -63.18, -24.53 | -59.42, -37.34 | APE12-dist-na | 16.2106 | APE11-dist-na | 14.5332 | APE10-dist-na | 11.8148 | APE9-dist-in | 7.0278 | None | None | None | XRAY | 2.6 | 0.224 | 0.233 | A | 356.0 | 338.0 | 10 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6joj | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PDGFRA | PGFRA_HUMAN | AF-P16234-K1A | P16234 | 585 | 960 | 1089.0 | No_ligand | No_ligand | Active | DFGin | 6.6997 | 13.6749 | BLAminus | -137.69, -178.12 | 65.56, 55.38 | -76.94, 17.55 | 294.68, 89.62 | -62.07, -30.49 | in-in | in | 7.3733 | Saltbr-in | 2.6326 | HRD-in | -76.76, -43.79 | 66.53, -13.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9412 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.33, 108.79 | APE9-dihe-in | -125.4, 152.2 | APE8-dihe-in | -75.15, 89.08 | APE8-rot-na | 36.01 | APE67-dihe-in | -66.01, -16.63 | -47.84, -37.12 | APE12-dist-na | 14.0618 | APE11-dist-na | 7.9646 | APE10-dist-na | 9.9372 | APE9-dist-in | 5.9594 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 376.0 | 376.0 | 0 | 30 | 30 | 0 | [[593, 952]] | 1.0 | AF-P16234-K1 | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 7.7e-106 | 359.3 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | AF-P16234-K3A | P16234 | 585 | 960 | 1089.0 | No_ligand | No_ligand | Active | DFGin | 6.6303 | 13.2587 | BLAminus | -128.58, 177.17 | 60.47, 65.55 | -71.97, 11.95 | 293.94, 94.32 | -62.2, -32.16 | in-in | in | 7.8236 | Saltbr-in | 2.7054 | HRD-in | -82.85, -43.12 | 66.78, -5.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9021 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -63.73, 118.36 | APE9-dihe-in | -107.5, 147.11 | APE8-dihe-in | -82.35, 65.15 | APE8-rot-na | 33.41 | APE67-dihe-in | -66.83, -20.14 | -51.1, -37.81 | APE12-dist-na | 14.3911 | APE11-dist-na | 8.9234 | APE10-dist-na | 12.0386 | APE9-dist-in | 7.1492 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 376.0 | 376.0 | 0 | 30 | 30 | 0 | [[593, 952]] | 1.0 | AF-P16234-K3 | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 7.7e-106 | 359.3 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 8PQHA | P16234 | 555 | 971 | 1089.0 | 9JI:1001 | Type1 | Active | DFGin | 7.1176 | 13.5042 | BLAminus | -137.77, -173.06 | 54.37, 84.67 | -94.17, 27.12 | 292.06, 83.63 | -63.26, -46.8 | in-in | in | 7.9228 | Saltbr-in | 3.2447 | HRD-in | -71.43, -45.05 | 70.07, -2.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9791 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -118.37, 127.86 | APE9-dihe-in | -120.13, 154.51 | APE8-dihe-in | -81.88, 68.37 | APE8-rot-na | 25.31 | APE67-dihe-in | -67.91, -9.11 | -50.35, -46.55 | APE12-dist-na | 6.6948 | APE11-dist-na | 11.7329 | APE10-dist-na | 11.1167 | APE9-dist-in | 7.073 | T674I | None | None | XRAY | 2.5 | 0.22 | 0.249 | A | 352.0 | 321.0 | 23 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 8pqh | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 8PQIA | P16234 | 567 | 969 | 1089.0 | 9OO:1001 | Type1 | Active | DFGin | 6.9059 | 13.5927 | BLAminus | -132.24, 178.87 | 62.52, 88.22 | -103.25, 28.49 | 291.7, 71.46 | -68.1, -30.59 | in-in | in | 7.9933 | Saltbr-in | 2.898 | HRD-in | -71.63, -43.38 | 66.22, 2.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8201 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -98.65, 130.26 | APE9-dihe-in | -117.66, 147.18 | APE8-dihe-in | -84.02, 76.87 | APE8-rot-na | 33.16 | APE67-dihe-in | -69.02, -9.85 | -66.15, -32.32 | APE12-dist-na | 999.0 | APE11-dist-na | 9.4755 | APE10-dist-na | 11.4786 | APE9-dist-in | 7.1354 | T674I | None | None | XRAY | 2.6 | 0.232 | 0.254 | A | 352.0 | 299.0 | 32 | 30 | 20 | 10 | [[593, 952]] | 1.0 | 8pqi | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 6JOIA | P16234 | 569 | 973 | 1089.0 | 6T2:1001 | Type1 | Inactive | DFGin | 5.8932 | 12.4237 | BLAplus | -149.03, 179.69 | 59.48, 39.87 | -90.32, -0.87 | 38.91, 91.7 | -108.94, 138.34 | in-out | in | 7.8145 | Saltbr-out | 4.0493 | HRD-in | -63.69, -47.81 | 78.72, -13.59 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.07, 131.06 | APE9-dihe-in | -119.74, 141.05 | APE8-dihe-in | -77.37, 79.89 | APE8-rot-na | 19.31 | APE67-dihe-in | -62.19, -30.0 | -59.33, -40.19 | APE12-dist-na | 999.0 | APE11-dist-na | 13.197 | APE10-dist-na | 15.7508 | APE9-dist-in | 7.4573 | T674I | None | None | XRAY | 3.1 | 0.224 | 0.244 | A | 375.0 | 296.0 | 37 | 30 | 15 | 15 | [[593, 952]] | 1.0 | 6joi | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 2.2e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | A0A0B4J203_HUMAN | 8XRRA | A0A0B4J203 | 338 | 730 | 849.0 | A1LV8:61001 | Type1 | Inactive | DFGin | 6.0782 | 12.8103 | BLBminus | -136.82, -170.16 | 60.75, 77.27 | -91.15, -163.07 | 294.15, 83.07 | 112.28, -36.82 | in-in | in | 7.2816 | Saltbr-in | 2.8565 | HRD-in | -63.02, -44.11 | 69.37, 4.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9784 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.33, 138.03 | APE9-dihe-in | -122.05, 151.58 | APE8-dihe-in | -77.69, 73.7 | APE8-rot-na | 29.73 | APE67-dihe-in | -63.37, -4.92 | -54.48, -47.94 | APE12-dist-na | 999.0 | APE11-dist-na | 8.1413 | APE10-dist-na | 10.8954 | APE9-dist-in | 6.9028 | None | None | None | XRAY | 2.57 | 0.238 | 0.26 | A | 356.0 | 285.0 | 36 | 30 | 19 | 11 | [[353, 712]] | 1.0 | 8xrr | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 3.7e-106 | 360.5 | 1.0 | 260.0 | 260.0 | 595 | 596 | 597 | 599 | 601 | 387 | 404 | 408 | 575 | 577 | 576 | 578.0 | 637 | 625 | 620 | 619 | 618 | 617 | 616 | 615 | 614 | 435 | receptor protein-tyrosine kinase |
| PDGFRA | PGFRA_HUMAN | 9GZHA | P16234 | 583 | 958 | 1089.0 | A1IRC:1001 | Type2 | Inactive | DFGout | 15.6481 | 9.5759 | BBAminus | -142.99, 176.85 | -144.44, 111.57 | -68.84, -35.83 | 280.23, 92.0 | 59.84, -119.26 | in-in | in | 7.8509 | Saltbr-in | 2.9454 | HRD-in | -72.49, -49.27 | 74.96, -9.55 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.0825 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -107.38, 139.27 | APE9-dihe-in | -132.11, 144.36 | APE8-dihe-in | -77.41, 71.6 | APE8-rot-na | 33.5 | APE67-dihe-in | -62.63, -15.56 | -62.2, -45.12 | APE12-dist-na | 15.5208 | APE11-dist-na | 11.6099 | APE10-dist-na | 11.6095 | APE9-dist-in | 7.5857 | T674I | None | None | XRAY | 2.2 | 0.183 | 0.215 | A | 355.0 | 282.0 | 22 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 9gzh | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 5GRNA | P16234 | 583 | 958 | 1089.0 | 748:1001 | Type2 | Inactive | DFGout | 16.3718 | 10.5289 | BBAminus | -143.58, -173.72 | -146.28, 106.78 | -54.79, -37.05 | 281.52, 58.25 | 60.16, -122.4 | in-in | in | 7.9371 | Saltbr-in | 2.7389 | HRD-in | -77.42, -50.02 | 77.14, -8.21 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.3417 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -107.12, 130.75 | APE9-dihe-in | -120.55, 148.05 | APE8-dihe-in | -80.95, 69.87 | APE8-rot-na | 36.32 | APE67-dihe-in | -65.74, -12.4 | -60.52, -41.33 | APE12-dist-na | 15.1679 | APE11-dist-na | 11.2852 | APE10-dist-na | 11.4357 | APE9-dist-in | 7.6446 | None | None | None | XRAY | 1.77 | 0.158 | 0.179 | A | 356.0 | 286.0 | 18 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 5grn | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 6JOLA | P16234 | 583 | 957 | 1089.0 | STI:1001 | Type2 | Inactive | DFGout | 16.377 | 10.1801 | BBAminus | -142.0, 174.77 | -141.65, 105.94 | -59.47, -37.67 | 274.19, 66.43 | 59.87, -122.37 | in-in | in | 7.9131 | Saltbr-in | 2.7813 | HRD-in | -68.97, -54.53 | 78.87, -11.97 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.9266 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.21, 134.53 | APE9-dihe-in | -124.89, 147.83 | APE8-dihe-in | -86.42, 79.14 | APE8-rot-na | 35.14 | APE67-dihe-in | -66.62, -11.35 | -62.29, -37.28 | APE12-dist-na | 16.0066 | APE11-dist-na | 12.1566 | APE10-dist-na | 11.9857 | APE9-dist-in | 7.6302 | None | None | None | XRAY | 1.9 | 0.215 | 0.236 | A | 356.0 | 279.0 | 24 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6jol | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 8PQKA | P16234 | 554 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 15.5834 | 8.1772 | None | -154.9, 179.4 | -116.45, 101.18 | -96.78, 25.45 | 224.18, 59.38 | -62.44, -23.73 | in-in | in | 7.7684 | Saltbr-in | 2.5801 | HRD-in | -75.59, -53.47 | 73.99, -2.28 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.7619 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -124.57, 123.17 | APE9-dihe-in | -122.51, 149.52 | APE8-dihe-in | -78.18, 70.07 | APE8-rot-na | 31.79 | APE67-dihe-in | -62.15, -17.78 | -60.4, -41.22 | APE12-dist-na | 19.4466 | APE11-dist-na | 15.06 | APE10-dist-na | 13.5403 | APE9-dist-in | 7.4476 | T674I | None | None | XRAY | 2.0 | 0.197 | 0.222 | A | 352.0 | 322.0 | 17 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 8pqk | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 6A32A | P16234 | 554 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 16.6148 | 8.4618 | None | -149.24, -176.86 | -118.22, 104.49 | -91.23, 25.57 | 218.48, 75.46 | -61.15, -35.43 | in-in | in | 8.2677 | Saltbr-in | 2.3994 | HRD-in | -77.45, -54.11 | 74.43, 2.58 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.5149 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.41, 128.42 | APE9-dihe-in | -113.39, 143.39 | APE8-dihe-in | -83.41, 71.44 | APE8-rot-na | 35.27 | APE67-dihe-in | -66.73, -17.33 | -56.98, -40.55 | APE12-dist-na | 17.2193 | APE11-dist-na | 14.1538 | APE10-dist-na | 12.9888 | APE9-dist-in | 7.2815 | T674I | None | None | XRAY | 1.87 | 0.205 | 0.24 | A | 356.0 | 336.0 | 12 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6a32 | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 1.8e-106 | 361.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 8PQJA | P16234 | 553 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 15.7273 | 8.2369 | None | -151.0, -178.54 | -115.21, 108.13 | -99.29, 20.66 | 220.99, 51.76 | -57.16, -27.12 | in-in | in | 7.805 | Saltbr-in | 2.6763 | HRD-in | -70.62, -57.5 | 76.76, 1.26 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8216 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -126.61, 120.89 | APE9-dihe-in | -120.18, 150.45 | APE8-dihe-in | -75.53, 66.41 | APE8-rot-na | 31.49 | APE67-dihe-in | -62.28, -19.29 | -62.48, -36.33 | APE12-dist-na | 19.3874 | APE11-dist-na | 15.0565 | APE10-dist-na | 13.613 | APE9-dist-in | 7.4582 | None | None | None | XRAY | 1.82 | 0.185 | 0.215 | A | 352.0 | 329.0 | 14 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 8pqj | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 8.8e-107 | 362.4 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 5K5XA | P16234 | 554 | 973 | 1089.0 | No_ligand | No_ligand | Inactive | DFGout | 15.8713 | 8.3345 | None | -153.24, -177.14 | -114.02, 113.86 | -108.1, 22.87 | 215.74, 54.5 | -59.52, -34.36 | in-in | in | 7.7455 | Saltbr-in | 2.4976 | HRD-in | -70.35, -55.34 | 73.06, -5.1 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.9506 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.49, 130.42 | APE9-dihe-in | -117.78, 136.58 | APE8-dihe-in | -73.77, 63.63 | APE8-rot-na | 32.36 | APE67-dihe-in | -68.21, -12.54 | -54.21, -40.36 | APE12-dist-na | 18.4802 | APE11-dist-na | 15.1785 | APE10-dist-na | 13.332 | APE9-dist-in | 7.4009 | None | None | None | XRAY | 2.168 | 0.193 | 0.224 | A | 356.0 | 345.0 | 3 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 5k5x | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 6JOKA | P16234 | 556 | 973 | 1089.0 | B49:1001 | Type1 | Inactive | DFGout | 17.3303 | 10.1516 | None | -157.96, 162.23 | -90.74, 118.75 | -83.04, 4.75 | 220.32, 127.42 | -60.76, -49.9 | in-out | in | 7.8064 | Saltbr-out | 4.6095 | HRD-in | -71.4, -52.83 | 71.29, -1.66 | out-out-in | SNCooi | out-in | ActLoopNT-out | 16.719 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -133.37, 126.64 | APE9-dihe-in | -119.51, 140.56 | APE8-dihe-in | -75.53, 69.74 | APE8-rot-na | 31.06 | APE67-dihe-in | -63.68, -19.63 | -58.21, -43.02 | APE12-dist-na | 17.5027 | APE11-dist-na | 14.289 | APE10-dist-na | 13.1977 | APE9-dist-in | 7.2863 | None | None | None | XRAY | 3.8 | 0.259 | 0.282 | A | 356.0 | 338.0 | 8 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6jok | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| PDGFRA | PGFRA_HUMAN | 6JOJA | P16234 | 554 | 973 | 1089.0 | 6T2:1001 | Type1 | Inactive | None | 20.3126 | 15.0063 | None | -134.96, -163.27 | -129.94, 169.75 | -62.88, -45.52 | 197.17, 82.33 | 72.34, -174.07 | in-in | in | 7.904 | Saltbr-in | 2.5098 | HRD-in | -72.82, -51.47 | 79.17, -0.33 | in-out-in | SNCioi | out-in | ActLoopNT-out | 18.4772 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -112.85, 133.76 | APE9-dihe-in | -123.13, 133.08 | APE8-dihe-in | -84.33, 80.22 | APE8-rot-na | 30.95 | APE67-dihe-in | -63.18, -24.53 | -59.42, -37.34 | APE12-dist-na | 16.2106 | APE11-dist-na | 14.5332 | APE10-dist-na | 11.8148 | APE9-dist-in | 7.0278 | None | None | None | XRAY | 2.6 | 0.224 | 0.233 | A | 356.0 | 338.0 | 10 | 30 | 30 | 0 | [[593, 952]] | 1.0 | 6joj | Homo sapiens | TYR_PDGFRA_HUMAN | TYR | 9.2e-107 | 362.5 | 1.0 | 260.0 | 260.0 | 835 | 836 | 837 | 839 | 841 | 627 | 644 | 648 | 815 | 817 | 816 | 818.0 | 877 | 865 | 860 | 859 | 858 | 857 | 856 | 855 | 854 | 675 | Platelet-derived growth factor receptor alpha |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|