| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| MAPK8 | 3O2MA | P45983 | 7 | 364 | 427.0 | 46A:60701 | Allosteric | Active | DFGin | 6.41 | 14.2667 | BLAminus | -152.63, 162.08 | 80.49, 93.8 | -114.77, 18.61 | 304.8, 107.67 | -61.69, -39.94 | in-in | in | 8.7422 | Saltbr-in | 2.6189 | HRD-in | -69.47, -52.78 | 72.9, -13.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7753 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -72.53, -31.31 | APE9-dihe-na | -91.45, 126.81 | APE8-dihe-in | -59.5, 135.65 | APE8-rot-in | 301.85 | APE67-dihe-in | -63.02, -13.15 | -75.49, -27.8 | APE12-dist-in | 11.2068 | APE11-dist-in | 12.7825 | APE10-dist-in | 7.434 | APE9-dist-in | 5.5284 | T183E,Y185E | None | None | XRAY | 2.7 | 0.233 | 0.266 | A | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o2m | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3O2MB | P45983 | 7 | 364 | 427.0 | 46A:60701 | Allosteric | Active | DFGin | 6.4326 | 14.024 | BLAminus | -142.38, 178.22 | 61.31, 93.12 | -105.38, 24.63 | 305.62, 107.49 | -54.81, -31.65 | in-in | in | 9.0593 | Saltbr-in | 2.7002 | HRD-in | -67.22, -47.31 | 66.21, -6.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9293 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -49.13, -35.19 | APE9-dihe-na | -86.25, 135.93 | APE8-dihe-in | -71.9, 130.6 | APE8-rot-in | 296.5 | APE67-dihe-in | -57.01, -19.27 | -49.25, -52.93 | APE12-dist-in | 11.5641 | APE11-dist-in | 12.8788 | APE10-dist-in | 7.9595 | APE9-dist-in | 5.5407 | T183E,Y185E | None | None | XRAY | 2.7 | 0.233 | 0.266 | B | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o2m | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VUIA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.2788 | 13.6367 | BLAminus | -161.71, 166.24 | 49.14, 98.79 | -100.93, 7.58 | 304.49, 111.2 | -57.41, -21.38 | in-in | in | 8.4447 | Saltbr-in | 2.7506 | HRD-in | -80.72, -34.44 | 66.81, -22.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -102.67, -34.53 | APE9-dihe-na | -81.58, 139.5 | APE8-dihe-in | -52.39, 128.3 | APE8-rot-in | 307.22 | APE67-dihe-in | -66.42, -12.33 | -38.87, -57.39 | APE12-dist-in | 13.5866 | APE11-dist-in | 13.1455 | APE10-dist-in | 7.2945 | APE9-dist-in | 4.5897 | C79V,C116S,C163A,C245S | None | None | XRAY | 2.8 | 0.22 | 0.282 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vui | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.7 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VUHA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.2446 | 13.5359 | BLAminus | -148.39, 170.84 | 44.38, 107.19 | -110.71, 10.86 | 305.1, 110.58 | -49.1, -34.53 | in-in | in | 8.3464 | Saltbr-in | 2.8139 | HRD-in | -67.84, -45.56 | 77.42, -28.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6841 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -82.33, -19.09 | APE9-dihe-na | -84.3, 142.26 | APE8-dihe-in | -58.96, 126.9 | APE8-rot-in | 301.88 | APE67-dihe-in | -66.35, -10.47 | -35.08, -59.67 | APE12-dist-in | 13.3098 | APE11-dist-in | 12.8591 | APE10-dist-in | 7.1419 | APE9-dist-in | 4.9243 | C116S,C163A,C245S | None | None | XRAY | 2.7 | 0.197 | 0.256 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vuh | CMGC_MAPK8_HUMAN | CMGC | 3e-84 | 288.7 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VUDA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.321 | 13.1923 | BLAminus | -128.97, 166.57 | 47.01, 116.8 | -121.87, 36.87 | 302.27, 89.43 | -73.6, -27.82 | in-in | in | 8.3203 | Saltbr-in | 2.7057 | HRD-in | -64.61, -34.78 | 67.2, -26.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.4829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -80.25, -55.44 | APE9-dihe-na | -80.77, 154.38 | APE8-dihe-in | -65.03, 131.96 | APE8-rot-in | 311.85 | APE67-dihe-in | -68.72, -34.8 | -46.83, -54.0 | APE12-dist-in | 13.3511 | APE11-dist-in | 12.8752 | APE10-dist-in | 6.8198 | APE9-dist-in | 4.9827 | C245S | None | None | XRAY | 3.5 | 0.204 | 0.293 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vud | CMGC_MAPK8_HUMAN | CMGC | 5.6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VUGA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.241 | 13.6703 | BLAminus | -151.25, 155.67 | 63.84, 102.6 | -110.8, 4.88 | 299.0, 108.74 | -61.2, -37.22 | in-in | in | 8.4642 | Saltbr-in | 2.6149 | HRD-in | -84.82, -38.91 | 70.88, -35.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6276 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -99.41, -25.55 | APE9-dihe-na | -88.01, 136.95 | APE8-dihe-in | -41.17, 111.55 | APE8-rot-in | 298.57 | APE67-dihe-in | -72.82, -30.6 | -28.21, -48.81 | APE12-dist-in | 13.4113 | APE11-dist-in | 12.8679 | APE10-dist-in | 7.0446 | APE9-dist-in | 4.8127 | C116S,C245S | None | None | XRAY | 3.24 | 0.195 | 0.284 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vug | CMGC_MAPK8_HUMAN | CMGC | 1.1e-84 | 290.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VUKA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 5.846 | 13.3361 | BLAminus | -160.02, 162.58 | 68.67, 104.55 | -110.92, -0.02 | 303.39, 88.83 | -56.44, -11.87 | in-in | in | 8.0975 | Saltbr-in | 2.7544 | HRD-in | -73.52, -45.64 | 80.08, -26.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7264 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.92, -26.67 | APE9-dihe-na | -92.92, 137.67 | APE8-dihe-in | -49.6, 127.14 | APE8-rot-in | 331.83 | APE67-dihe-in | -67.5, -4.18 | -38.21, -62.31 | APE12-dist-in | 13.399 | APE11-dist-in | 12.8977 | APE10-dist-in | 7.1315 | APE9-dist-in | 4.9417 | C79V,C116S,C137V,C163A,C245S | None | None | XRAY | 2.95 | 0.229 | 0.302 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vuk | CMGC_MAPK8_HUMAN | CMGC | 4.2e-83 | 285.0 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | AF-P45983-K1A | P45983 | 18 | 329 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.4146 | 13.6432 | BLAminus | -143.36, 178.91 | 71.76, 59.86 | -79.25, 6.67 | 305.71, 110.21 | -57.24, -28.48 | in-in | in | 8.7613 | Saltbr-in | 2.7045 | HRD-in | -68.06, -45.26 | 66.86, -8.1 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -79.62, -32.38 | APE9-dihe-na | -74.54, 148.67 | APE8-dihe-in | -64.82, 122.89 | APE8-rot-in | 305.16 | APE67-dihe-in | -66.57, -21.46 | -45.8, -48.81 | APE12-dist-in | 12.8637 | APE11-dist-in | 12.5239 | APE10-dist-in | 6.8143 | APE9-dist-in | 4.4072 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 312.0 | 312.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | AF-P45983-K1 | CMGC_MAPK8_HUMAN | CMGC | 2.4e-84 | 288.9 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | AF-P45983-K3A | P45983 | 18 | 329 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.1015 | 14.4206 | BLAminus | -131.11, 176.97 | 65.27, 65.06 | -73.24, 10.87 | 295.36, 94.81 | -61.15, -20.86 | in-in | in | 9.583 | Saltbr-in | 2.7357 | HRD-in | -74.19, -48.13 | 61.63, 17.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8487 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -76.5, 167.97 | APE9-dihe-na | 65.01, 133.8 | APE8-dihe-in | -55.56, 132.77 | APE8-rot-in | 297.67 | APE67-dihe-in | -67.94, -21.16 | -47.15, -46.41 | APE12-dist-in | 12.7744 | APE11-dist-in | 11.0959 | APE10-dist-in | 6.4288 | APE9-dist-in | 3.1656 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 312.0 | 312.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | AF-P45983-K3 | CMGC_MAPK8_HUMAN | CMGC | 2.4e-84 | 288.9 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3O17A | P45983 | 7 | 363 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.1281 | 13.9918 | BLAminus | -143.08, -155.15 | 4.86, 119.05 | -115.61, 15.13 | 291.48, 95.12 | -55.48, -42.85 | in-in | in | 8.9255 | Saltbr-in | 2.9771 | HRD-in | -88.38, -43.35 | 58.03, 10.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.3731 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -76.55, -54.88 | APE9-dihe-na | -56.03, 107.98 | APE8-dihe-in | -41.53, 122.11 | APE8-rot-in | 303.39 | APE67-dihe-in | -26.7, -32.66 | -31.75, -85.44 | APE12-dist-in | 10.5963 | APE11-dist-in | 11.6428 | APE10-dist-in | 6.8427 | APE9-dist-in | 4.5653 | T183E,Y185E | None | None | XRAY | 3.0 | 0.263 | 0.308 | A | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o17 | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3O17B | P45983 | 7 | 363 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.3772 | 13.3535 | BLAminus | -141.52, 176.46 | 56.9, 126.68 | -136.61, 6.27 | 299.25, 120.4 | -50.46, -23.38 | in-in | in | 9.2139 | Saltbr-in | 3.0929 | HRD-in | -88.24, -52.87 | 72.9, -9.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.4939 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -59.17, -32.26 | APE9-dihe-na | -88.08, 142.34 | APE8-dihe-in | -62.23, 117.26 | APE8-rot-in | 321.66 | APE67-dihe-in | -47.49, -37.82 | -30.24, -67.12 | APE12-dist-in | 11.7384 | APE11-dist-in | 12.4339 | APE10-dist-in | 7.0415 | APE9-dist-in | 4.5416 | T183E,Y185E | None | None | XRAY | 3.0 | 0.263 | 0.308 | B | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o17 | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2G01A | P45983 | 10 | 364 | 427.0 | 73Q:60901 | Type1 | Active | DFGin | 5.9935 | 14.6114 | BLAminus | -138.21, 160.8 | 78.02, 123.65 | -129.29, 5.43 | 293.89, 44.0 | -38.65, -23.81 | out-in | out | 10.3783 | Saltbr-in | 3.5583 | HRD-in | -86.8, -31.67 | 38.11, 34.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6571 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.24, -50.25 | APE9-dihe-na | -79.72, 72.99 | APE8-dihe-in | -7.98, 107.48 | APE8-rot-in | 347.58 | APE67-dihe-in | -48.8, -23.78 | -62.13, -32.37 | APE12-dist-in | 12.1688 | APE11-dist-in | 12.9249 | APE10-dist-in | 7.5972 | APE9-dist-in | 4.5707 | T183E,Y185E | None | None | XRAY | 3.5 | 0.296 | 0.354 | A | 370.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2g01 | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2H96A | P45983 | 7 | 364 | 427.0 | 893:60901 | Type1 | Active | DFGin | 5.7466 | 14.0711 | BLAminus | -142.02, 170.57 | 47.6, 140.71 | -141.49, -1.15 | 291.84, 115.53 | -55.85, -8.38 | in-in | in | 9.1022 | Saltbr-in | 2.8225 | HRD-in | -85.69, -41.32 | 64.83, 4.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -74.81, -40.52 | APE9-dihe-na | -68.31, 154.87 | APE8-dihe-in | -75.38, 102.01 | APE8-rot-in | 313.08 | APE67-dihe-in | -53.52, -10.26 | -11.43, -68.01 | APE12-dist-in | 11.968 | APE11-dist-in | 12.5208 | APE10-dist-in | 7.0412 | APE9-dist-in | 4.4506 | T183E,Y185E | None | None | XRAY | 3.0 | 0.243 | 0.278 | A | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2h96 | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2H96B | P45983 | 7 | 364 | 427.0 | 893:60902 | Type1 | Active | DFGin | 5.8069 | 14.0678 | BLAminus | -144.72, 174.09 | 54.02, 123.29 | -119.24, -14.41 | 278.05, 179.66 | -39.96, -62.74 | in-in | in | 9.0689 | Saltbr-in | 2.9733 | HRD-in | -74.32, -61.93 | 80.7, -10.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8668 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.3, -36.87 | APE9-dihe-na | -83.37, 136.31 | APE8-dihe-in | -75.86, 124.1 | APE8-rot-in | 311.58 | APE67-dihe-in | -48.77, -30.54 | -42.37, -58.0 | APE12-dist-in | 11.8616 | APE11-dist-in | 12.7575 | APE10-dist-in | 7.2009 | APE9-dist-in | 5.2463 | T183E,Y185E | None | None | XRAY | 3.0 | 0.243 | 0.278 | B | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2h96 | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2NO3A | P45983 | 8 | 364 | 427.0 | 859:901 | Type1 | Active | DFGin | 5.8629 | 13.8896 | BLAminus | -141.07, 148.97 | 75.82, 137.69 | -138.71, 16.78 | 294.85, 98.43 | -54.01, -64.02 | in-in | in | 8.4814 | Saltbr-in | 2.7915 | HRD-in | -92.56, -31.18 | 61.32, -24.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.5506 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -47.4, -34.85 | APE9-dihe-na | -77.56, 142.56 | APE8-dihe-in | -59.37, 120.51 | APE8-rot-in | 310.95 | APE67-dihe-in | -29.44, -22.2 | -32.85, -87.31 | APE12-dist-in | 11.9332 | APE11-dist-in | 12.0435 | APE10-dist-in | 6.6597 | APE9-dist-in | 4.8178 | T183E,Y185E | None | None | XRAY | 3.2 | 0.233 | 0.276 | A | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2no3 | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2NO3B | P45983 | 7 | 363 | 427.0 | 859:902 | Type1 | Active | DFGin | 6.4988 | 14.1591 | BLAminus | -157.78, 177.02 | 69.64, 114.69 | -132.65, 1.82 | 296.08, 106.12 | -53.25, -7.72 | in-in | in | 9.1606 | Saltbr-in | 3.0003 | HRD-in | -57.79, -52.24 | 74.94, -7.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1052 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -98.63, -57.06 | APE9-dihe-na | -57.37, 144.61 | APE8-dihe-in | -64.67, 111.29 | APE8-rot-in | 358.49 | APE67-dihe-in | -34.54, -28.75 | -26.01, -79.7 | APE12-dist-in | 12.833 | APE11-dist-in | 13.3757 | APE10-dist-in | 7.5425 | APE9-dist-in | 4.8072 | T183E,Y185E | None | None | XRAY | 3.2 | 0.233 | 0.276 | B | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2no3 | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 6ZR5A | P45983 | 3 | 362 | 427.0 | ANP:60402 | ATPlike | Inactive | DFGin | 3.8172 | 14.2258 | ABAminus | -84.03, -42.55 | -114.88, 174.79 | -114.82, 8.54 | 299.13, 101.86 | 79.5, -168.62 | out-out | out | 10.0023 | Saltbr-out | 5.0314 | HRD-in | -56.29, -55.44 | 70.4, -2.27 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8722 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 107.14 | APE8-rot-out | 87.08 | APE67-dihe-in | -67.28, -21.26 | -101.91, 26.36 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.699 | 0.186 | 0.256 | A | 366.0 | 348.0 | 12 | 27 | 15 | 12 | [[26, 321]] | 1.0 | 6zr5 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 6ZR5B | P45983 | 4 | 362 | 427.0 | ANP:60400 | ATPlike | Inactive | DFGin | 3.867 | 14.0721 | ABAminus | -85.51, -41.13 | -110.19, 172.79 | -115.96, 8.05 | 294.61, 92.39 | 79.48, -170.78 | out-out | out | 10.0205 | Saltbr-out | 4.2237 | HRD-in | -59.93, -50.9 | 67.15, -3.15 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8489 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioo | APE10-dihe-na | -100.6, 89.98 | APE9-dihe-na | -140.16, 151.66 | APE8-dihe-in | -87.57, 109.71 | APE8-rot-in | 298.46 | APE67-dihe-in | -73.45, -13.54 | -100.12, 16.22 | APE12-dist-out | 17.5514 | APE11-dist-in | 12.8984 | APE10-dist-out | 16.3414 | APE9-dist-out | 11.496 | None | None | None | XRAY | 2.699 | 0.186 | 0.256 | B | 366.0 | 359.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 6zr5 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2XRWA | P45983 | 2 | 364 | 427.0 | ANP:61367 | ATPlike | Inactive | DFGin | 3.8162 | 13.9414 | ABAminus | -85.3, -24.5 | -153.59, -177.02 | -115.68, 7.02 | 304.14, 97.05 | 88.01, -156.78 | in-out | in | 9.886 | Saltbr-out | 4.6349 | HRD-in | -83.3, -58.4 | 77.36, -14.29 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.45, -23.57 | 999.0, -3.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.33 | 0.166 | 0.187 | A | 371.0 | 347.0 | 16 | 27 | 11 | 16 | [[26, 321]] | 1.0 | 2xrw | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2XS0A | P45983 | 6 | 365 | 427.0 | ANP:1367 | ATPlike | Inactive | DFGin | 3.7537 | 14.0806 | ABAminus | -75.25, -22.88 | -148.14, -178.22 | -116.01, 26.92 | 303.04, 86.85 | 61.81, -161.42 | in-out | in | 9.7349 | Saltbr-out | 5.5498 | HRD-in | -69.33, -60.51 | 78.49, -20.02 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoo | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 173.45 | APE8-rot-out | 188.87 | APE67-dihe-out | -73.26, -26.46 | -135.55, 95.92 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T183V,Y185F | None | None | XRAY | 2.6 | 0.194 | 0.246 | A | 386.0 | 346.0 | 14 | 27 | 13 | 14 | [[26, 321]] | 1.0 | 2xs0 | CMGC_MAPK8_HUMAN | CMGC | 4.5e-83 | 284.9 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4UX9A | P45983 | 8 | 363 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.5081 | 13.5979 | ABAminus | -106.9, -65.56 | -75.5, 125.74 | -123.36, 16.47 | 304.33, 124.23 | -68.62, -34.25 | in-out | in | 8.8495 | Saltbr-out | 3.6733 | HRD-in | -62.88, -46.37 | 73.76, -28.18 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.694 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -77.3, -23.46 | APE9-dihe-na | -71.58, 140.2 | APE8-dihe-in | -64.86, 127.48 | APE8-rot-in | 308.5 | APE67-dihe-in | -60.43, -26.76 | -33.69, -61.49 | APE12-dist-in | 11.784 | APE11-dist-in | 12.4258 | APE10-dist-in | 6.6314 | APE9-dist-in | 4.5326 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | A | 364.0 | 343.0 | 7 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 4ux9 | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4UX9C | P45983 | 8 | 363 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.9564 | 13.7764 | ABAminus | -110.49, -64.95 | -89.1, 120.63 | -119.14, 21.23 | 309.02, 115.06 | -68.23, -26.49 | in-out | in | 8.9193 | Saltbr-out | 3.6356 | HRD-in | -66.22, -47.15 | 71.23, -16.82 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.5691 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -79.69, -26.4 | APE9-dihe-na | -76.07, 142.18 | APE8-dihe-in | -66.37, 127.01 | APE8-rot-in | 305.02 | APE67-dihe-in | -64.57, -24.76 | -35.27, -55.26 | APE12-dist-none | 999.0 | APE11-dist-in | 12.0054 | APE10-dist-in | 6.5305 | APE9-dist-in | 4.6212 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | C | 364.0 | 333.0 | 15 | 27 | 20 | 7 | [[26, 321]] | 1.0 | 4ux9 | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4UX9D | P45983 | 9 | 364 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.7553 | 13.4065 | ABAminus | -120.6, -55.98 | -93.07, 108.1 | -98.68, 25.97 | 301.07, 117.04 | -64.8, -33.9 | in-in | in | 9.3656 | Saltbr-in | 2.7382 | HRD-in | -59.8, -49.61 | 70.57, -12.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.6695 | ActLoopCT-out | nonTYR | APEdihe_aaioo | APEdist_oioo | APE10-dihe-na | -95.31, 105.19 | APE9-dihe-na | -74.34, -56.46 | APE8-dihe-in | -76.71, 134.72 | APE8-rot-out | 95.68 | APE67-dihe-out | -66.63, -26.9 | -139.86, 50.27 | APE12-dist-out | 14.0313 | APE11-dist-in | 13.438 | APE10-dist-out | 10.8234 | APE9-dist-out | 13.5554 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | D | 364.0 | 344.0 | 9 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 4ux9 | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8R5EA | P45983 | 5 | 363 | 427.0 | ANP:402,Y6K:403 | ATPlike,Allosteric | Inactive | DFGin | 4.2147 | 13.8837 | ABAminus | -92.07, -26.65 | -133.67, 178.16 | -123.93, 6.5 | 294.94, 97.33 | 89.15, -162.77 | in-out | in | 9.5208 | Saltbr-out | 4.8419 | HRD-in | -77.17, -59.97 | 76.05, -10.25 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.7895 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -62.14, 143.17 | APE9-dihe-na | -120.32, 118.65 | APE8-dihe-in | -75.39, 123.94 | APE8-rot-in | 299.29 | APE67-dihe-in | -61.41, -23.9 | -115.12, 4.11 | APE12-dist-out | 18.7072 | APE11-dist-out | 15.3251 | APE10-dist-out | 16.6803 | APE9-dist-out | 11.2441 | None | None | None | XRAY | 1.7 | 0.177 | 0.222 | A | 366.0 | 359.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 8r5e | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 1UKHA | P45983 | 9 | 363 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.009 | 13.5918 | ABAminus | -71.05, -50.54 | -134.57, 170.42 | -88.05, 19.73 | 310.31, 96.24 | 54.55, -119.32 | in-in | in | 8.7257 | Saltbr-in | 3.5395 | HRD-in | -32.35, -66.36 | 74.83, -11.73 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, -21.95 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.35 | 0.229 | 0.245 | A | 369.0 | 321.0 | 22 | 27 | 10 | 17 | [[26, 321]] | 1.0 | 1ukh | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4YR8A | P45983 | 8 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 3.746 | 13.6511 | ABAminus | -92.48, -36.82 | -128.7, -177.95 | -116.24, 9.95 | 302.59, 109.3 | 79.22, -159.79 | in-in | in | 9.397 | Saltbr-in | 2.7167 | HRD-in | -91.12, -57.47 | 70.8, -11.5 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 120.35 | APE8-dihe-in | -90.35, 105.5 | APE8-rot-out | 50.94 | APE67-dihe-in | -67.62, -16.88 | -108.83, 0.82 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.1748 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | A | 371.0 | 320.0 | 17 | 27 | 14 | 13 | [[26, 321]] | 1.0 | 4yr8 | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4YR8C | P45983 | 10 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.3451 | 13.3914 | ABAminus | -88.52, -41.45 | -131.53, -175.1 | -114.96, 11.59 | 302.69, 109.92 | 79.73, 999.0 | in-in | in | 8.8736 | Saltbr-in | 2.6944 | HRD-in | -68.29, -62.18 | 77.05, -0.67 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanni | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 118.23 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.66, -18.42 | -99.29, -2.8 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | C | 371.0 | 318.0 | 21 | 27 | 11 | 16 | [[26, 321]] | 1.0 | 4yr8 | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4YR8E | P45983 | 7 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 3.7276 | 14.1372 | ABAminus | -86.08, -36.9 | -129.28, 170.42 | -104.47, 7.33 | 299.61, 110.26 | 81.64, -165.5 | out-out | out | 10.093 | Saltbr-out | 3.6951 | HRD-in | -78.61, -55.83 | 65.3, 1.9 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8909 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -50.39 | APE8-dihe-in | -79.39, 102.65 | APE8-rot-out | 53.21 | APE67-dihe-in | -61.82, -18.77 | -109.31, -0.43 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.7944 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | E | 371.0 | 317.0 | 17 | 27 | 15 | 12 | [[26, 321]] | 1.0 | 4yr8 | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4YR8F | P45983 | 10 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.6068 | 13.3341 | ABAminus | -92.28, -40.63 | -125.1, 178.19 | -117.35, 11.6 | 304.63, 110.41 | 81.03, 999.0 | in-in | in | 8.5474 | Saltbr-in | 2.4139 | HRD-in | -61.32, -58.08 | 77.0, -3.6 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanni | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 114.52 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.79, -18.18 | -101.48, -2.27 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | F | 371.0 | 300.0 | 38 | 27 | 11 | 16 | [[26, 321]] | 1.0 | 4yr8 | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 6F5EB | P45983 | 7 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.2446 | 14.401 | ABAminus | -85.23, -40.02 | -143.49, -172.1 | -102.9, -4.9 | 292.34, 110.9 | 97.56, -150.23 | in-in | in | 9.2523 | Saltbr-in | 3.1606 | HRD-in | -56.05, -56.91 | 72.46, 7.42 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9127 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, 112.0 | APE9-dihe-na | -95.81, 149.23 | APE8-dihe-out | -71.37, -38.95 | APE8-rot-in | 293.49 | APE67-dihe-in | -53.11, -31.53 | -58.04, -34.44 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 14.7564 | APE9-dist-out | 11.1737 | None | None | None | XRAY | 2.7 | 0.202 | 0.226 | B | 373.0 | 346.0 | 10 | 27 | 23 | 4 | [[26, 321]] | 1.0 | 6f5e | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8X5MA | P45983 | 7 | 363 | 427.0 | Y4O:401 | Type1 | Inactive | DFGin | 3.8295 | 13.7211 | ABAminus | -82.03, -35.59 | -145.84, 177.75 | -109.61, 10.51 | 302.7, 100.16 | 80.95, -155.06 | in-in | in | 9.1059 | Saltbr-in | 2.7679 | HRD-in | -69.78, -60.93 | 77.08, -7.13 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.2374 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 140.93 | APE8-dihe-in | -94.27, 100.92 | APE8-rot-in | 297.8 | APE67-dihe-in | -57.39, -30.56 | -110.37, 11.17 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.1596 | None | None | CSO163 | XRAY | 2.0 | 0.195 | 0.234 | A | 363.0 | 341.0 | 16 | 27 | 15 | 12 | [[26, 321]] | 1.0 | 8x5m | CMGC_MAPK8_HUMAN | CMGC | 7.9e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PT8A | P45983 | 7 | 363 | 427.0 | A3O:401 | Type1 | Inactive | DFGin | 3.5115 | 13.6408 | ABAminus | -86.46, -36.69 | -113.24, 157.51 | -107.14, 5.23 | 297.22, 84.35 | 63.56, -136.9 | in-out | in | 9.7221 | Saltbr-out | 5.4719 | HRD-in | -69.36, -62.04 | 67.14, -1.26 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.2593 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nioo | APE10-dihe-na | -78.69, 132.14 | APE9-dihe-na | -97.09, 6.93 | APE8-dihe-in | -119.44, 125.16 | APE8-rot-out | 77.92 | APE67-dihe-in | -61.62, -35.67 | -102.35, -19.0 | APE12-dist-none | 999.0 | APE11-dist-in | 10.0559 | APE10-dist-out | 10.1664 | APE9-dist-out | 11.4072 | None | None | None | XRAY | 2.78 | 0.219 | 0.218 | A | 366.0 | 353.0 | 2 | 27 | 25 | 2 | [[26, 321]] | 1.0 | 8pt8 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PT8B | P45983 | 8 | 363 | 427.0 | A3O:401 | Type1 | Inactive | DFGin | 3.7083 | 13.5603 | ABAminus | -87.46, -36.99 | -114.07, 158.6 | -107.2, 3.96 | 306.69, 95.61 | 61.75, -138.76 | out-out | out | 10.0137 | Saltbr-out | 4.7072 | HRD-in | -65.17, -60.14 | 69.69, -8.9 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.0336 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_iioo | APE10-dihe-na | -125.68, 169.43 | APE9-dihe-na | -89.29, -51.47 | APE8-dihe-out | 50.18, 54.05 | APE8-rot-out | 80.12 | APE67-dihe-in | -59.08, -31.41 | -75.35, -27.98 | APE12-dist-in | 11.3425 | APE11-dist-in | 8.5237 | APE10-dist-out | 11.6714 | APE9-dist-out | 8.6343 | None | None | None | XRAY | 2.78 | 0.219 | 0.218 | B | 366.0 | 354.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 8pt8 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PT8C | P45983 | 7 | 362 | 427.0 | A3O:401 | Type1 | Inactive | DFGin | 4.333 | 13.6339 | ABAminus | -100.64, -42.98 | -112.04, 163.18 | -107.79, 3.91 | 318.61, 83.5 | 62.89, -142.35 | in-out | in | 9.3615 | Saltbr-out | 6.3544 | HRD-in | -65.16, -58.91 | 71.32, -6.19 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.1345 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -0.16 | APE9-dihe-na | -89.45, -4.71 | APE8-dihe-in | -89.37, 113.03 | APE8-rot-out | 66.41 | APE67-dihe-in | -51.88, -31.5 | -134.08, -10.25 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 11.551 | APE9-dist-out | 11.4356 | None | None | None | XRAY | 2.78 | 0.219 | 0.218 | C | 366.0 | 353.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 8pt8 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PT9A | P45983 | 8 | 363 | 427.0 | DVI:401 | Type1 | Inactive | DFGin | 3.6725 | 13.8445 | ABAminus | -82.42, -42.96 | -101.44, 156.25 | -107.65, 10.42 | 293.61, 64.96 | 107.26, -173.51 | out-in | out | 10.2179 | Saltbr-in | 3.1648 | HRD-in | -86.93, -57.09 | 73.38, 1.77 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.3496 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_iooo | APE10-dihe-na | -132.39, 130.51 | APE9-dihe-na | -63.89, -49.36 | APE8-dihe-out | 47.93, 60.73 | APE8-rot-out | 86.13 | APE67-dihe-in | -60.85, -39.95 | -75.12, -7.36 | APE12-dist-in | 10.0694 | APE11-dist-out | 6.9139 | APE10-dist-out | 10.6396 | APE9-dist-out | 8.438 | None | None | None | XRAY | 2.7 | 0.215 | 0.225 | A | 366.0 | 353.0 | 2 | 27 | 25 | 2 | [[26, 321]] | 1.0 | 8pt9 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PT9B | P45983 | 7 | 363 | 427.0 | DVI:401 | Type1 | Inactive | DFGin | 3.6022 | 13.3587 | ABAminus | -78.87, -38.7 | -110.84, 150.53 | -102.26, 4.03 | 302.35, 93.73 | 66.71, -148.92 | in-out | in | 9.405 | Saltbr-out | 4.004 | HRD-in | -82.54, -61.31 | 64.36, 5.02 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nioo | APE10-dihe-na | -99.2, 123.92 | APE9-dihe-na | -85.67, -7.28 | APE8-dihe-in | -87.66, 94.6 | APE8-rot-out | 69.53 | APE67-dihe-in | -57.65, -34.34 | -84.42, -14.13 | APE12-dist-none | 999.0 | APE11-dist-in | 9.9637 | APE10-dist-out | 10.6502 | APE9-dist-out | 11.067 | None | None | None | XRAY | 2.7 | 0.215 | 0.225 | B | 366.0 | 351.0 | 5 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 8pt9 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PT9C | P45983 | 8 | 362 | 427.0 | DVI:401 | Type1 | Inactive | DFGin | 3.804 | 14.2556 | ABAminus | -88.85, -34.33 | -106.1, 147.38 | -98.39, 6.8 | 298.91, 67.63 | 59.14, -132.88 | out-out | out | 10.1832 | Saltbr-out | 3.8904 | HRD-in | -79.93, -61.89 | 65.26, 3.23 | out-out-out | SNCooo | out-out | ActLoopNT-out | 4.6788 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -169.35 | APE9-dihe-na | -94.15, 7.09 | APE8-dihe-in | -84.28, 82.63 | APE8-rot-out | 73.62 | APE67-dihe-in | -62.72, -39.65 | -92.57, -5.37 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 11.9341 | APE9-dist-out | 11.2227 | None | None | None | XRAY | 2.7 | 0.215 | 0.225 | C | 366.0 | 352.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 8pt9 | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PTAA | P45983 | 8 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.923 | 14.4771 | ABAminus | -80.58, -61.37 | -103.85, 165.38 | -100.79, 23.99 | 295.77, 91.74 | 73.84, -149.47 | in-in | in | 9.7897 | Saltbr-in | 3.1262 | HRD-in | -78.59, -61.53 | 62.23, 7.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.4702 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iooo | APE10-dihe-na | -130.45, 138.38 | APE9-dihe-na | -101.99, 109.25 | APE8-dihe-in | -118.89, 112.23 | APE8-rot-out | 53.5 | APE67-dihe-in | -51.79, -30.07 | -95.29, -17.54 | APE12-dist-in | 10.569 | APE11-dist-out | 7.0333 | APE10-dist-out | 10.1833 | APE9-dist-out | 8.5978 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | A | 366.0 | 354.0 | 2 | 27 | 25 | 2 | [[26, 321]] | 1.0 | 8pta | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PTAB | P45983 | 7 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.5773 | 13.1788 | ABAminus | -81.24, -57.35 | -101.3, 158.61 | -105.36, 14.2 | 308.93, 93.28 | 64.59, -148.13 | in-in | in | 9.3658 | Saltbr-in | 3.5356 | HRD-in | -77.41, -61.25 | 61.49, 9.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -112.33, 168.25 | APE9-dihe-na | -116.9, 36.67 | APE8-dihe-in | -104.63, 91.0 | APE8-rot-out | 52.55 | APE67-dihe-in | -56.88, -29.41 | -95.02, -21.65 | APE12-dist-in | 11.7839 | APE11-dist-in | 9.1521 | APE10-dist-out | 11.2421 | APE9-dist-out | 10.2145 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | B | 366.0 | 352.0 | 5 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 8pta | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 8PTAC | P45983 | 8 | 361 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.8263 | 14.0885 | ABAminus | -83.97, -56.35 | -97.04, 154.46 | -105.76, 13.83 | 294.99, 32.04 | 63.79, -147.27 | in-out | in | 9.7228 | Saltbr-out | 4.5276 | HRD-in | -77.01, -60.9 | 63.25, 7.56 | out-out-out | SNCooo | out-out | ActLoopNT-out | 4.6109 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -137.59 | APE9-dihe-na | -94.11, 17.64 | APE8-dihe-in | -81.48, 63.35 | APE8-rot-out | 71.39 | APE67-dihe-in | -58.68, -26.77 | -108.19, -24.77 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 12.4666 | APE9-dist-out | 10.7804 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | C | 366.0 | 351.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 8pta | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 1UKIA | P45983 | 9 | 363 | 427.0 | 537:0 | Type1 | Inactive | DFGin | 4.7042 | 13.1142 | ABAminus | -77.11, -62.2 | -116.68, -161.07 | -126.7, 15.2 | 318.68, 71.9 | 41.91, -116.91 | in-in | in | 9.1687 | Saltbr-in | 2.9158 | HRD-in | -66.76, -57.64 | 78.15, -46.3 | in-out-out | SNCioo | out-out | ActLoopNT-out | 5.4563 | ActLoopCT-out | nonTYR | APEdihe_aanio | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 77.25 | APE8-rot-in | 304.87 | APE67-dihe-out | -76.75, -17.12 | 155.56, -17.08 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.221 | 0.241 | A | 369.0 | 328.0 | 18 | 27 | 14 | 13 | [[26, 321]] | 1.0 | 1uki | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4E73A | P45983 | 8 | 361 | 427.0 | 0NR:60401 | Type1 | Inactive | DFGin | 3.9405 | 13.7141 | ABAminus | -80.5, -42.58 | -144.32, -163.84 | -110.6, 6.62 | 304.02, 132.42 | 68.66, -151.79 | in-in | in | 9.1157 | Saltbr-in | 2.603 | HRD-in | -76.2, -63.12 | 71.21, -5.48 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -70.49, -32.11 | 999.0, 34.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.27 | 0.249 | 0.282 | A | 369.0 | 318.0 | 23 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4e73 | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4G1WA | P45983 | 8 | 361 | 427.0 | G1W:60401 | Type1 | Inactive | DFGin | 4.1305 | 13.7474 | ABAminus | -75.19, -46.06 | -145.01, -166.31 | -101.8, 11.35 | 310.93, 129.6 | 54.15, -150.73 | in-in | in | 9.5121 | Saltbr-in | 2.8152 | HRD-in | -74.24, -60.52 | 76.29, -17.95 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 110.92 | APE8-rot-in | 305.3 | APE67-dihe-in | -68.41, -20.62 | -111.33, 3.9 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.45 | 0.233 | 0.297 | A | 369.0 | 322.0 | 22 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4g1w | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4HYSA | P45983 | 8 | 361 | 427.0 | 1BJ:60401 | Type1 | Inactive | DFGin | 4.1442 | 13.7039 | ABAminus | -65.58, -42.99 | -148.13, -172.29 | -105.42, 11.47 | 305.84, 116.47 | 62.72, -152.88 | in-in | in | 9.1693 | Saltbr-in | 2.5418 | HRD-in | -81.1, -55.52 | 80.05, -13.7 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 85.27 | APE8-rot-in | 300.61 | APE67-dihe-in | -75.95, -19.65 | -89.11, 15.51 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.415 | 0.249 | 0.295 | A | 369.0 | 321.0 | 23 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4hys | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4HYUA | P45983 | 8 | 361 | 427.0 | 1BK:60401 | Type1 | Inactive | DFGin | 4.0678 | 13.5935 | ABAminus | -80.82, -40.1 | -141.28, -176.81 | -103.55, 4.37 | 303.13, 103.89 | 67.61, -155.32 | in-in | in | 9.276 | Saltbr-in | 2.7839 | HRD-in | -63.72, -62.24 | 77.82, -3.04 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 97.87 | APE8-rot-in | 304.34 | APE67-dihe-in | -66.69, -21.83 | -103.0, 8.43 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.152 | 0.231 | 0.269 | A | 369.0 | 322.0 | 22 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4hyu | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4IZYA | P45983 | 8 | 361 | 427.0 | 1J2:60401 | Type1 | Inactive | DFGin | 3.8819 | 13.4843 | ABAminus | -76.71, -38.87 | -145.64, -179.24 | -102.44, 14.51 | 311.23, 93.45 | 52.84, -142.09 | in-in | in | 9.149 | Saltbr-in | 2.7383 | HRD-in | -72.23, -60.13 | 78.79, -8.13 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 111.06 | APE8-rot-in | 300.16 | APE67-dihe-in | -67.83, -22.42 | -106.79, 8.95 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.3 | 0.239 | 0.261 | A | 369.0 | 322.0 | 22 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4izy | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3PZEA | P45983 | 7 | 362 | 427.0 | CFK:1 | Type1 | Inactive | DFGin | 4.1379 | 13.9068 | ABAminus | -81.12, -32.94 | -131.86, 179.29 | -115.73, 16.97 | 304.08, 91.38 | 65.8, -99.93 | in-in | in | 8.7987 | Saltbr-in | 2.79 | HRD-in | -65.45, -61.37 | 74.31, -21.03 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 43.07 | APE8-dihe-out | -90.42, -23.2 | APE8-rot-in | 308.55 | APE67-dihe-in | -65.57, -26.71 | -47.05, -33.16 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.1182 | None | None | None | XRAY | 2.0 | 0.206 | 0.24 | A | 358.0 | 347.0 | 9 | 27 | 18 | 9 | [[26, 321]] | 1.0 | 3pze | CMGC_MAPK8_HUMAN | CMGC | 4.1e-84 | 288.3 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4L7FA | P45983 | 7 | 362 | 427.0 | 1V5:60401 | Type1 | Inactive | DFGin | 4.168 | 13.9028 | ABAminus | -92.73, -21.27 | -136.46, -179.9 | -126.51, 2.69 | 298.75, 92.07 | 123.75, 92.84 | in-in | in | 9.571 | Saltbr-in | 2.7172 | HRD-in | -73.68, -60.59 | 73.9, -18.64 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, 56.52 | APE9-dihe-na | -75.12, 136.19 | APE8-dihe-in | -88.12, 112.11 | APE8-rot-in | 306.44 | APE67-dihe-in | -64.04, -21.62 | -99.03, -5.95 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 14.8393 | APE9-dist-out | 11.6873 | None | None | None | XRAY | 1.95 | 0.162 | 0.198 | A | 367.0 | 343.0 | 13 | 27 | 14 | 13 | [[26, 321]] | 1.0 | 4l7f | CMGC_MAPK8_HUMAN | CMGC | 4.4e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3ELJA | P45983 | 7 | 364 | 427.0 | GS7:365 | Type1 | Inactive | DFGin | 4.2607 | 13.8455 | ABAminus | -96.2, -23.23 | -129.0, 175.64 | -123.66, 12.92 | 303.89, 93.13 | 80.21, -148.51 | in-in | in | 9.2759 | Saltbr-in | 3.4358 | HRD-in | -62.88, -61.88 | 76.44, -14.77 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -113.33, 122.34 | APE9-dihe-na | -76.53, 136.67 | APE8-dihe-in | -80.59, 119.63 | APE8-rot-in | 296.46 | APE67-dihe-in | -59.78, -20.24 | -110.49, 3.47 | APE12-dist-out | 20.996 | APE11-dist-out | 15.8219 | APE10-dist-out | 16.3336 | APE9-dist-out | 11.4349 | None | None | None | XRAY | 1.8 | 0.188 | 0.215 | A | 369.0 | 347.0 | 6 | 27 | 21 | 6 | [[26, 321]] | 1.0 | 3elj | CMGC_MAPK8_HUMAN | CMGC | 4.5e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4AWIA | P45983 | 8 | 364 | 427.0 | AQ2:1365 | Type1 | Inactive | DFGin | 4.4603 | 13.936 | ABAminus | -87.42, -26.01 | -133.81, 169.02 | -108.8, 6.11 | 295.82, 101.28 | 92.5, -161.91 | in-in | in | 8.9051 | Saltbr-in | 2.7425 | HRD-in | -70.34, -61.6 | 77.73, -9.92 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -85.55, 146.28 | APE9-dihe-na | -95.6, 128.29 | APE8-dihe-in | -89.62, 121.11 | APE8-rot-in | 309.81 | APE67-dihe-in | -66.82, -18.55 | -120.34, 14.07 | APE12-dist-out | 18.8339 | APE11-dist-out | 14.9052 | APE10-dist-out | 16.4247 | APE9-dist-out | 11.46 | None | None | None | XRAY | 1.91 | 0.188 | 0.219 | A | 369.0 | 352.0 | 5 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 4awi | CMGC_MAPK8_HUMAN | CMGC | 4.5e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 5LW1B | P45983 | 8 | 362 | 427.0 | ADN:60401 | Type1 | Inactive | DFGin | 4.4197 | 14.4478 | ABAminus | -83.29, -51.84 | -118.5, -177.73 | -115.08, 20.0 | 298.98, 87.21 | 71.2, -159.63 | out-out | out | 10.4298 | Saltbr-out | 3.8124 | HRD-in | -68.61, -60.19 | 64.51, 12.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.4773 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -136.58, 144.4 | APE9-dihe-na | -122.04, 105.79 | APE8-dihe-out | -71.41, -33.58 | APE8-rot-in | 307.18 | APE67-dihe-in | -61.62, -32.85 | -63.18, -22.53 | APE12-dist-out | 20.0348 | APE11-dist-out | 18.2025 | APE10-dist-out | 13.7638 | APE9-dist-out | 11.7502 | None | None | None | XRAY | 3.2 | 0.177 | 0.212 | B | 373.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 5lw1 | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 5LW1E | P45983 | 8 | 362 | 427.0 | ADN:60401 | Type1 | Inactive | DFGin | 4.1748 | 14.0755 | ABAminus | -82.51, -53.19 | -119.45, -176.34 | -115.64, 20.66 | 300.14, 87.37 | 72.63, -160.31 | in-out | in | 9.9432 | Saltbr-out | 4.611 | HRD-in | -68.12, -61.52 | 63.83, 14.63 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8826 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -137.31, 145.55 | APE9-dihe-na | -120.94, 104.94 | APE8-dihe-out | -71.75, -32.64 | APE8-rot-in | 307.04 | APE67-dihe-in | -62.19, -31.77 | -62.28, -22.63 | APE12-dist-out | 20.0912 | APE11-dist-out | 18.3879 | APE10-dist-out | 14.0865 | APE9-dist-out | 12.0009 | None | None | None | XRAY | 3.2 | 0.177 | 0.212 | E | 373.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 5lw1 | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 5LW1H | P45983 | 8 | 362 | 427.0 | ADN:60401 | Type1 | Inactive | DFGin | 4.1303 | 14.3776 | ABAminus | -82.43, -51.23 | -118.2, -176.9 | -114.7, 20.75 | 298.45, 87.29 | 72.11, -159.03 | out-out | out | 10.2847 | Saltbr-out | 3.7377 | HRD-in | -69.31, -61.29 | 63.64, 13.39 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.4743 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -136.56, 144.9 | APE9-dihe-na | -119.98, 105.48 | APE8-dihe-out | -71.78, -33.35 | APE8-rot-in | 307.69 | APE67-dihe-in | -61.37, -31.81 | -63.06, -22.73 | APE12-dist-out | 20.0957 | APE11-dist-out | 18.3691 | APE10-dist-out | 13.9653 | APE9-dist-out | 11.9943 | None | None | None | XRAY | 3.2 | 0.177 | 0.212 | H | 373.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 5lw1 | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4QTDA | P45983 | 6 | 363 | 427.0 | 38Z:424,ANP:425 | Type1,Allosteric | Inactive | DFGin | 4.2787 | 13.95 | ABAminus | -89.69, -21.2 | -135.34, 171.77 | -115.48, 9.24 | 298.02, 89.8 | 87.52, -156.74 | in-out | in | 9.5926 | Saltbr-out | 4.1531 | HRD-in | -75.36, -55.62 | 72.51, -12.26 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.6893 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -117.32, 137.81 | APE9-dihe-na | -80.42, 132.23 | APE8-dihe-in | -83.54, 120.1 | APE8-rot-in | 296.41 | APE67-dihe-in | -61.39, -20.52 | -109.55, -3.05 | APE12-dist-out | 21.1401 | APE11-dist-out | 16.032 | APE10-dist-out | 16.5166 | APE9-dist-out | 11.1471 | None | None | None | XRAY | 1.5 | 0.167 | 0.192 | A | 364.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 4qtd | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 9FT9A | P45983 | 7 | 363 | 427.0 | ANP:401 | ATPlike | Inactive | DFGin | 6.2012 | 13.6807 | BLAminus | -138.37, -170.04 | 58.94, 78.24 | -92.66, 22.82 | 315.32, 103.73 | -63.89, -26.18 | in-out | in | 8.5419 | Saltbr-out | 3.8425 | HRD-in | -66.92, -47.02 | 65.13, 0.51 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8271 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioo | APE10-dihe-na | -150.17, 156.5 | APE9-dihe-na | -75.27, -52.01 | APE8-dihe-in | -88.35, 100.07 | APE8-rot-in | 310.81 | APE67-dihe-in | -64.72, -11.39 | -102.84, 1.94 | APE12-dist-out | 5.9095 | APE11-dist-in | 10.5805 | APE10-dist-out | 8.0786 | APE9-dist-out | 10.9491 | None | None | None | XRAY | 2.35 | 0.234 | 0.27 | A | 360.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 9ft9 | CMGC_MAPK8_HUMAN | CMGC | 4.1e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3V3VA | P45983 | 7 | 363 | 427.0 | MYU:401 | Type1 | Inactive | DFGin | 6.8274 | 13.7856 | BLAminus | -143.77, -172.33 | 52.69, 90.19 | -99.08, 8.98 | 306.34, 125.67 | -39.78, -30.71 | in-in | in | 8.0358 | Saltbr-in | 2.8823 | HRD-in | -67.72, -38.9 | 75.22, -25.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.605 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -111.93, -15.72 | APE9-dihe-na | -81.89, 141.96 | APE8-dihe-in | -63.44, 127.02 | APE8-rot-out | 31.94 | APE67-dihe-in | -66.37, -23.13 | -30.24, -61.71 | APE12-dist-in | 12.8042 | APE11-dist-in | 12.8097 | APE10-dist-in | 7.6481 | APE9-dist-in | 5.1004 | None | None | None | XRAY | 2.7 | 0.229 | 0.266 | A | 379.0 | 351.0 | 6 | 27 | 23 | 4 | [[26, 321]] | 1.0 | 3v3v | CMGC_MAPK8_HUMAN | CMGC | 3.3e-84 | 288.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2GMXA | P45983 | 8 | 364 | 427.0 | 877:60901 | Type1 | Inactive | DFGin | 6.4145 | 15.103 | BLAminus | -169.49, -165.44 | 17.67, 94.27 | -93.05, 32.73 | 281.95, 52.09 | -74.74, -22.92 | in-in | in | 9.2457 | Saltbr-in | 3.4507 | HRD-in | -84.23, -59.06 | 73.39, 47.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7327 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -71.92, -33.15 | APE9-dihe-na | -81.6, 112.65 | APE8-dihe-in | -25.7, 132.77 | APE8-rot-out | 32.67 | APE67-dihe-in | -46.1, -17.73 | -58.05, -70.61 | APE12-dist-in | 10.542 | APE11-dist-in | 13.1827 | APE10-dist-in | 7.8512 | APE9-dist-in | 4.9448 | T183E,Y185E | None | None | XRAY | 3.5 | 0.278 | 0.351 | A | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2gmx | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 4UX9B | P45983 | 8 | 362 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.8269 | 14.0009 | None | -95.23, -79.97 | -82.17, 124.02 | -113.22, 13.68 | 297.81, 107.19 | -60.29, -32.64 | in-in | in | 8.6029 | Saltbr-in | 2.9418 | HRD-in | -59.44, -53.0 | 79.08, -24.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.5822 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -58.47, -40.48 | APE9-dihe-na | -78.17, 138.93 | APE8-dihe-in | -64.59, 122.35 | APE8-rot-in | 308.57 | APE67-dihe-in | -67.83, -19.56 | -32.59, -57.13 | APE12-dist-in | 12.3608 | APE11-dist-in | 12.1486 | APE10-dist-in | 6.5271 | APE9-dist-in | 4.6911 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | B | 364.0 | 327.0 | 14 | 27 | 21 | 6 | [[26, 321]] | 1.0 | 4ux9 | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2G01B | P45983 | 9 | 364 | 427.0 | 73Q:61001 | Type1 | Inactive | DFGin | 5.7329 | 14.7118 | None | -124.05, -159.93 | 70.3, -99.04 | 78.28, -8.58 | 269.85, 26.32 | -60.64, -29.84 | in-in | in | 9.3096 | Saltbr-in | 3.522 | HRD-in | -75.33, -51.61 | 81.6, -31.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0497 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -55.32, -77.05 | APE9-dihe-na | -50.72, 131.97 | APE8-dihe-in | -62.41, 127.97 | APE8-rot-out | 179.45 | APE67-dihe-in | -34.47, -20.37 | -26.15, -85.34 | APE12-dist-in | 12.6428 | APE11-dist-in | 12.8438 | APE10-dist-in | 7.3262 | APE9-dist-in | 4.7568 | T183E,Y185E | None | None | XRAY | 3.5 | 0.296 | 0.354 | B | 370.0 | 356.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2g01 | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 2GMXB | P45983 | 7 | 364 | 427.0 | 877:61001 | Type1 | Inactive | DFGin | 5.6113 | 13.9429 | None | -106.95, -175.57 | 54.48, -113.25 | 110.31, -6.6 | 279.44, 165.75 | -41.3, -39.48 | in-out | in | 8.4562 | Saltbr-out | 4.4993 | HRD-in | -77.53, -48.43 | 77.05, -21.57 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8017 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -70.75, -77.84 | APE9-dihe-na | -45.43, 98.08 | APE8-dihe-in | -37.04, 123.81 | APE8-rot-in | 354.32 | APE67-dihe-in | -25.17, -38.2 | -26.5, -90.08 | APE12-dist-in | 11.7738 | APE11-dist-in | 12.5874 | APE10-dist-in | 7.2474 | APE9-dist-in | 4.4727 | T183E,Y185E | None | None | XRAY | 3.5 | 0.278 | 0.351 | B | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2gmx | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VULA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | None | DFGin | 5.1102 | 13.7682 | BLAminus | -85.93, 163.21 | 85.46, 126.64 | -150.76, 1.53 | 338.77, 110.45 | -63.64, 22.92 | in-in | in | 9.4027 | Saltbr-in | 3.0531 | HRD-in | -77.29, -39.59 | 61.8, -14.75 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.6801 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -129.09, 14.97 | 999.0, -38.05 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | C79V,C116S,C137V,C163A,C213V,C245S | None | None | XRAY | 2.81 | 0.252 | 0.315 | A | 370.0 | 344.0 | 14 | 27 | 13 | 14 | [[26, 321]] | 1.0 | 3vul | CMGC_MAPK8_HUMAN | CMGC | 2.6e-81 | 279.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | 3VUMA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | None | DFGin | 5.0561 | 13.607 | BLAminus | -112.58, 170.27 | 77.92, 128.69 | -145.25, 34.84 | 350.71, 122.87 | -58.09, -36.69 | in-in | in | 9.0374 | Saltbr-in | 2.9813 | HRD-in | -72.36, -43.79 | 70.87, -4.2 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9289 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -69.29, -4.06 | 999.0, -24.38 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | C41V,C79V,C116S,C137V,C163A,C213V,C245S | None | None | XRAY | 2.69 | 0.192 | 0.255 | A | 370.0 | 344.0 | 14 | 27 | 13 | 14 | [[26, 321]] | 1.0 | 3vum | CMGC_MAPK8_HUMAN | CMGC | 2.8e-81 | 279.0 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| MAPK8 | MK08_HUMAN | 3O2MA | P45983 | 7 | 364 | 427.0 | 46A:60701 | Allosteric | Active | DFGin | 6.41 | 14.2667 | BLAminus | -152.63, 162.08 | 80.49, 93.8 | -114.77, 18.61 | 304.8, 107.67 | -61.69, -39.94 | in-in | in | 8.7422 | Saltbr-in | 2.6189 | HRD-in | -69.47, -52.78 | 72.9, -13.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7753 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -72.53, -31.31 | APE9-dihe-na | -91.45, 126.81 | APE8-dihe-in | -59.5, 135.65 | APE8-rot-in | 301.85 | APE67-dihe-in | -63.02, -13.15 | -75.49, -27.8 | APE12-dist-in | 11.2068 | APE11-dist-in | 12.7825 | APE10-dist-in | 7.434 | APE9-dist-in | 5.5284 | T183E,Y185E | None | None | XRAY | 2.7 | 0.233 | 0.266 | A | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o2m | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3O2MB | P45983 | 7 | 364 | 427.0 | 46A:60701 | Allosteric | Active | DFGin | 6.4326 | 14.024 | BLAminus | -142.38, 178.22 | 61.31, 93.12 | -105.38, 24.63 | 305.62, 107.49 | -54.81, -31.65 | in-in | in | 9.0593 | Saltbr-in | 2.7002 | HRD-in | -67.22, -47.31 | 66.21, -6.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9293 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -49.13, -35.19 | APE9-dihe-na | -86.25, 135.93 | APE8-dihe-in | -71.9, 130.6 | APE8-rot-in | 296.5 | APE67-dihe-in | -57.01, -19.27 | -49.25, -52.93 | APE12-dist-in | 11.5641 | APE11-dist-in | 12.8788 | APE10-dist-in | 7.9595 | APE9-dist-in | 5.5407 | T183E,Y185E | None | None | XRAY | 2.7 | 0.233 | 0.266 | B | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o2m | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VUIA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.2788 | 13.6367 | BLAminus | -161.71, 166.24 | 49.14, 98.79 | -100.93, 7.58 | 304.49, 111.2 | -57.41, -21.38 | in-in | in | 8.4447 | Saltbr-in | 2.7506 | HRD-in | -80.72, -34.44 | 66.81, -22.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -102.67, -34.53 | APE9-dihe-na | -81.58, 139.5 | APE8-dihe-in | -52.39, 128.3 | APE8-rot-in | 307.22 | APE67-dihe-in | -66.42, -12.33 | -38.87, -57.39 | APE12-dist-in | 13.5866 | APE11-dist-in | 13.1455 | APE10-dist-in | 7.2945 | APE9-dist-in | 4.5897 | C79V,C116S,C163A,C245S | None | None | XRAY | 2.8 | 0.22 | 0.282 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vui | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.7 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VUHA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.2446 | 13.5359 | BLAminus | -148.39, 170.84 | 44.38, 107.19 | -110.71, 10.86 | 305.1, 110.58 | -49.1, -34.53 | in-in | in | 8.3464 | Saltbr-in | 2.8139 | HRD-in | -67.84, -45.56 | 77.42, -28.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6841 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -82.33, -19.09 | APE9-dihe-na | -84.3, 142.26 | APE8-dihe-in | -58.96, 126.9 | APE8-rot-in | 301.88 | APE67-dihe-in | -66.35, -10.47 | -35.08, -59.67 | APE12-dist-in | 13.3098 | APE11-dist-in | 12.8591 | APE10-dist-in | 7.1419 | APE9-dist-in | 4.9243 | C116S,C163A,C245S | None | None | XRAY | 2.7 | 0.197 | 0.256 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vuh | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 3e-84 | 288.7 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VUDA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.321 | 13.1923 | BLAminus | -128.97, 166.57 | 47.01, 116.8 | -121.87, 36.87 | 302.27, 89.43 | -73.6, -27.82 | in-in | in | 8.3203 | Saltbr-in | 2.7057 | HRD-in | -64.61, -34.78 | 67.2, -26.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.4829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -80.25, -55.44 | APE9-dihe-na | -80.77, 154.38 | APE8-dihe-in | -65.03, 131.96 | APE8-rot-in | 311.85 | APE67-dihe-in | -68.72, -34.8 | -46.83, -54.0 | APE12-dist-in | 13.3511 | APE11-dist-in | 12.8752 | APE10-dist-in | 6.8198 | APE9-dist-in | 4.9827 | C245S | None | None | XRAY | 3.5 | 0.204 | 0.293 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vud | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 5.6e-85 | 291.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VUGA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.241 | 13.6703 | BLAminus | -151.25, 155.67 | 63.84, 102.6 | -110.8, 4.88 | 299.0, 108.74 | -61.2, -37.22 | in-in | in | 8.4642 | Saltbr-in | 2.6149 | HRD-in | -84.82, -38.91 | 70.88, -35.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6276 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -99.41, -25.55 | APE9-dihe-na | -88.01, 136.95 | APE8-dihe-in | -41.17, 111.55 | APE8-rot-in | 298.57 | APE67-dihe-in | -72.82, -30.6 | -28.21, -48.81 | APE12-dist-in | 13.4113 | APE11-dist-in | 12.8679 | APE10-dist-in | 7.0446 | APE9-dist-in | 4.8127 | C116S,C245S | None | None | XRAY | 3.24 | 0.195 | 0.284 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vug | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 1.1e-84 | 290.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VUKA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | Active | DFGin | 5.846 | 13.3361 | BLAminus | -160.02, 162.58 | 68.67, 104.55 | -110.92, -0.02 | 303.39, 88.83 | -56.44, -11.87 | in-in | in | 8.0975 | Saltbr-in | 2.7544 | HRD-in | -73.52, -45.64 | 80.08, -26.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7264 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.92, -26.67 | APE9-dihe-na | -92.92, 137.67 | APE8-dihe-in | -49.6, 127.14 | APE8-rot-in | 331.83 | APE67-dihe-in | -67.5, -4.18 | -38.21, -62.31 | APE12-dist-in | 13.399 | APE11-dist-in | 12.8977 | APE10-dist-in | 7.1315 | APE9-dist-in | 4.9417 | C79V,C116S,C137V,C163A,C245S | None | None | XRAY | 2.95 | 0.229 | 0.302 | A | 370.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 3vuk | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.2e-83 | 285.0 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | AF-P45983-K1A | P45983 | 18 | 329 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.4146 | 13.6432 | BLAminus | -143.36, 178.91 | 71.76, 59.86 | -79.25, 6.67 | 305.71, 110.21 | -57.24, -28.48 | in-in | in | 8.7613 | Saltbr-in | 2.7045 | HRD-in | -68.06, -45.26 | 66.86, -8.1 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -79.62, -32.38 | APE9-dihe-na | -74.54, 148.67 | APE8-dihe-in | -64.82, 122.89 | APE8-rot-in | 305.16 | APE67-dihe-in | -66.57, -21.46 | -45.8, -48.81 | APE12-dist-in | 12.8637 | APE11-dist-in | 12.5239 | APE10-dist-in | 6.8143 | APE9-dist-in | 4.4072 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 312.0 | 312.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | AF-P45983-K1 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.4e-84 | 288.9 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | AF-P45983-K3A | P45983 | 18 | 329 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.1015 | 14.4206 | BLAminus | -131.11, 176.97 | 65.27, 65.06 | -73.24, 10.87 | 295.36, 94.81 | -61.15, -20.86 | in-in | in | 9.583 | Saltbr-in | 2.7357 | HRD-in | -74.19, -48.13 | 61.63, 17.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8487 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -76.5, 167.97 | APE9-dihe-na | 65.01, 133.8 | APE8-dihe-in | -55.56, 132.77 | APE8-rot-in | 297.67 | APE67-dihe-in | -67.94, -21.16 | -47.15, -46.41 | APE12-dist-in | 12.7744 | APE11-dist-in | 11.0959 | APE10-dist-in | 6.4288 | APE9-dist-in | 3.1656 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 312.0 | 312.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | AF-P45983-K3 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.4e-84 | 288.9 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3O17A | P45983 | 7 | 363 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.1281 | 13.9918 | BLAminus | -143.08, -155.15 | 4.86, 119.05 | -115.61, 15.13 | 291.48, 95.12 | -55.48, -42.85 | in-in | in | 8.9255 | Saltbr-in | 2.9771 | HRD-in | -88.38, -43.35 | 58.03, 10.08 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.3731 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -76.55, -54.88 | APE9-dihe-na | -56.03, 107.98 | APE8-dihe-in | -41.53, 122.11 | APE8-rot-in | 303.39 | APE67-dihe-in | -26.7, -32.66 | -31.75, -85.44 | APE12-dist-in | 10.5963 | APE11-dist-in | 11.6428 | APE10-dist-in | 6.8427 | APE9-dist-in | 4.5653 | T183E,Y185E | None | None | XRAY | 3.0 | 0.263 | 0.308 | A | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o17 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3O17B | P45983 | 7 | 363 | 427.0 | No_ligand | No_ligand | Active | DFGin | 6.3772 | 13.3535 | BLAminus | -141.52, 176.46 | 56.9, 126.68 | -136.61, 6.27 | 299.25, 120.4 | -50.46, -23.38 | in-in | in | 9.2139 | Saltbr-in | 3.0929 | HRD-in | -88.24, -52.87 | 72.9, -9.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.4939 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -59.17, -32.26 | APE9-dihe-na | -88.08, 142.34 | APE8-dihe-in | -62.23, 117.26 | APE8-rot-in | 321.66 | APE67-dihe-in | -47.49, -37.82 | -30.24, -67.12 | APE12-dist-in | 11.7384 | APE11-dist-in | 12.4339 | APE10-dist-in | 7.0415 | APE9-dist-in | 4.5416 | T183E,Y185E | None | None | XRAY | 3.0 | 0.263 | 0.308 | B | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 3o17 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 1.6e-83 | 286.4 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2G01A | P45983 | 10 | 364 | 427.0 | 73Q:60901 | Type1 | Active | DFGin | 5.9935 | 14.6114 | BLAminus | -138.21, 160.8 | 78.02, 123.65 | -129.29, 5.43 | 293.89, 44.0 | -38.65, -23.81 | out-in | out | 10.3783 | Saltbr-in | 3.5583 | HRD-in | -86.8, -31.67 | 38.11, 34.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6571 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.24, -50.25 | APE9-dihe-na | -79.72, 72.99 | APE8-dihe-in | -7.98, 107.48 | APE8-rot-in | 347.58 | APE67-dihe-in | -48.8, -23.78 | -62.13, -32.37 | APE12-dist-in | 12.1688 | APE11-dist-in | 12.9249 | APE10-dist-in | 7.5972 | APE9-dist-in | 4.5707 | T183E,Y185E | None | None | XRAY | 3.5 | 0.296 | 0.354 | A | 370.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2g01 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2H96A | P45983 | 7 | 364 | 427.0 | 893:60901 | Type1 | Active | DFGin | 5.7466 | 14.0711 | BLAminus | -142.02, 170.57 | 47.6, 140.71 | -141.49, -1.15 | 291.84, 115.53 | -55.85, -8.38 | in-in | in | 9.1022 | Saltbr-in | 2.8225 | HRD-in | -85.69, -41.32 | 64.83, 4.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -74.81, -40.52 | APE9-dihe-na | -68.31, 154.87 | APE8-dihe-in | -75.38, 102.01 | APE8-rot-in | 313.08 | APE67-dihe-in | -53.52, -10.26 | -11.43, -68.01 | APE12-dist-in | 11.968 | APE11-dist-in | 12.5208 | APE10-dist-in | 7.0412 | APE9-dist-in | 4.4506 | T183E,Y185E | None | None | XRAY | 3.0 | 0.243 | 0.278 | A | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2h96 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2H96B | P45983 | 7 | 364 | 427.0 | 893:60902 | Type1 | Active | DFGin | 5.8069 | 14.0678 | BLAminus | -144.72, 174.09 | 54.02, 123.29 | -119.24, -14.41 | 278.05, 179.66 | -39.96, -62.74 | in-in | in | 9.0689 | Saltbr-in | 2.9733 | HRD-in | -74.32, -61.93 | 80.7, -10.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8668 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.3, -36.87 | APE9-dihe-na | -83.37, 136.31 | APE8-dihe-in | -75.86, 124.1 | APE8-rot-in | 311.58 | APE67-dihe-in | -48.77, -30.54 | -42.37, -58.0 | APE12-dist-in | 11.8616 | APE11-dist-in | 12.7575 | APE10-dist-in | 7.2009 | APE9-dist-in | 5.2463 | T183E,Y185E | None | None | XRAY | 3.0 | 0.243 | 0.278 | B | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2h96 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2NO3A | P45983 | 8 | 364 | 427.0 | 859:901 | Type1 | Active | DFGin | 5.8629 | 13.8896 | BLAminus | -141.07, 148.97 | 75.82, 137.69 | -138.71, 16.78 | 294.85, 98.43 | -54.01, -64.02 | in-in | in | 8.4814 | Saltbr-in | 2.7915 | HRD-in | -92.56, -31.18 | 61.32, -24.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.5506 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -47.4, -34.85 | APE9-dihe-na | -77.56, 142.56 | APE8-dihe-in | -59.37, 120.51 | APE8-rot-in | 310.95 | APE67-dihe-in | -29.44, -22.2 | -32.85, -87.31 | APE12-dist-in | 11.9332 | APE11-dist-in | 12.0435 | APE10-dist-in | 6.6597 | APE9-dist-in | 4.8178 | T183E,Y185E | None | None | XRAY | 3.2 | 0.233 | 0.276 | A | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2no3 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2NO3B | P45983 | 7 | 363 | 427.0 | 859:902 | Type1 | Active | DFGin | 6.4988 | 14.1591 | BLAminus | -157.78, 177.02 | 69.64, 114.69 | -132.65, 1.82 | 296.08, 106.12 | -53.25, -7.72 | in-in | in | 9.1606 | Saltbr-in | 3.0003 | HRD-in | -57.79, -52.24 | 74.94, -7.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1052 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -98.63, -57.06 | APE9-dihe-na | -57.37, 144.61 | APE8-dihe-in | -64.67, 111.29 | APE8-rot-in | 358.49 | APE67-dihe-in | -34.54, -28.75 | -26.01, -79.7 | APE12-dist-in | 12.833 | APE11-dist-in | 13.3757 | APE10-dist-in | 7.5425 | APE9-dist-in | 4.8072 | T183E,Y185E | None | None | XRAY | 3.2 | 0.233 | 0.276 | B | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2no3 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 6ZR5A | P45983 | 3 | 362 | 427.0 | ANP:60402 | ATPlike | Inactive | DFGin | 3.8172 | 14.2258 | ABAminus | -84.03, -42.55 | -114.88, 174.79 | -114.82, 8.54 | 299.13, 101.86 | 79.5, -168.62 | out-out | out | 10.0023 | Saltbr-out | 5.0314 | HRD-in | -56.29, -55.44 | 70.4, -2.27 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8722 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 107.14 | APE8-rot-out | 87.08 | APE67-dihe-in | -67.28, -21.26 | -101.91, 26.36 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.699 | 0.186 | 0.256 | A | 366.0 | 348.0 | 12 | 27 | 15 | 12 | [[26, 321]] | 1.0 | 6zr5 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 6ZR5B | P45983 | 4 | 362 | 427.0 | ANP:60400 | ATPlike | Inactive | DFGin | 3.867 | 14.0721 | ABAminus | -85.51, -41.13 | -110.19, 172.79 | -115.96, 8.05 | 294.61, 92.39 | 79.48, -170.78 | out-out | out | 10.0205 | Saltbr-out | 4.2237 | HRD-in | -59.93, -50.9 | 67.15, -3.15 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8489 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioo | APE10-dihe-na | -100.6, 89.98 | APE9-dihe-na | -140.16, 151.66 | APE8-dihe-in | -87.57, 109.71 | APE8-rot-in | 298.46 | APE67-dihe-in | -73.45, -13.54 | -100.12, 16.22 | APE12-dist-out | 17.5514 | APE11-dist-in | 12.8984 | APE10-dist-out | 16.3414 | APE9-dist-out | 11.496 | None | None | None | XRAY | 2.699 | 0.186 | 0.256 | B | 366.0 | 359.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 6zr5 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2XRWA | P45983 | 2 | 364 | 427.0 | ANP:61367 | ATPlike | Inactive | DFGin | 3.8162 | 13.9414 | ABAminus | -85.3, -24.5 | -153.59, -177.02 | -115.68, 7.02 | 304.14, 97.05 | 88.01, -156.78 | in-out | in | 9.886 | Saltbr-out | 4.6349 | HRD-in | -83.3, -58.4 | 77.36, -14.29 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -64.45, -23.57 | 999.0, -3.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.33 | 0.166 | 0.187 | A | 371.0 | 347.0 | 16 | 27 | 11 | 16 | [[26, 321]] | 1.0 | 2xrw | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2XS0A | P45983 | 6 | 365 | 427.0 | ANP:1367 | ATPlike | Inactive | DFGin | 3.7537 | 14.0806 | ABAminus | -75.25, -22.88 | -148.14, -178.22 | -116.01, 26.92 | 303.04, 86.85 | 61.81, -161.42 | in-out | in | 9.7349 | Saltbr-out | 5.5498 | HRD-in | -69.33, -60.51 | 78.49, -20.02 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoo | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 173.45 | APE8-rot-out | 188.87 | APE67-dihe-out | -73.26, -26.46 | -135.55, 95.92 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T183V,Y185F | None | None | XRAY | 2.6 | 0.194 | 0.246 | A | 386.0 | 346.0 | 14 | 27 | 13 | 14 | [[26, 321]] | 1.0 | 2xs0 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.5e-83 | 284.9 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4UX9A | P45983 | 8 | 363 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.5081 | 13.5979 | ABAminus | -106.9, -65.56 | -75.5, 125.74 | -123.36, 16.47 | 304.33, 124.23 | -68.62, -34.25 | in-out | in | 8.8495 | Saltbr-out | 3.6733 | HRD-in | -62.88, -46.37 | 73.76, -28.18 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.694 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -77.3, -23.46 | APE9-dihe-na | -71.58, 140.2 | APE8-dihe-in | -64.86, 127.48 | APE8-rot-in | 308.5 | APE67-dihe-in | -60.43, -26.76 | -33.69, -61.49 | APE12-dist-in | 11.784 | APE11-dist-in | 12.4258 | APE10-dist-in | 6.6314 | APE9-dist-in | 4.5326 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | A | 364.0 | 343.0 | 7 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 4ux9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4UX9C | P45983 | 8 | 363 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.9564 | 13.7764 | ABAminus | -110.49, -64.95 | -89.1, 120.63 | -119.14, 21.23 | 309.02, 115.06 | -68.23, -26.49 | in-out | in | 8.9193 | Saltbr-out | 3.6356 | HRD-in | -66.22, -47.15 | 71.23, -16.82 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.5691 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -79.69, -26.4 | APE9-dihe-na | -76.07, 142.18 | APE8-dihe-in | -66.37, 127.01 | APE8-rot-in | 305.02 | APE67-dihe-in | -64.57, -24.76 | -35.27, -55.26 | APE12-dist-none | 999.0 | APE11-dist-in | 12.0054 | APE10-dist-in | 6.5305 | APE9-dist-in | 4.6212 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | C | 364.0 | 333.0 | 15 | 27 | 20 | 7 | [[26, 321]] | 1.0 | 4ux9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4UX9D | P45983 | 9 | 364 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.7553 | 13.4065 | ABAminus | -120.6, -55.98 | -93.07, 108.1 | -98.68, 25.97 | 301.07, 117.04 | -64.8, -33.9 | in-in | in | 9.3656 | Saltbr-in | 2.7382 | HRD-in | -59.8, -49.61 | 70.57, -12.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.6695 | ActLoopCT-out | nonTYR | APEdihe_aaioo | APEdist_oioo | APE10-dihe-na | -95.31, 105.19 | APE9-dihe-na | -74.34, -56.46 | APE8-dihe-in | -76.71, 134.72 | APE8-rot-out | 95.68 | APE67-dihe-out | -66.63, -26.9 | -139.86, 50.27 | APE12-dist-out | 14.0313 | APE11-dist-in | 13.438 | APE10-dist-out | 10.8234 | APE9-dist-out | 13.5554 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | D | 364.0 | 344.0 | 9 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 4ux9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8R5EA | P45983 | 5 | 363 | 427.0 | ANP:402,Y6K:403 | ATPlike,Allosteric | Inactive | DFGin | 4.2147 | 13.8837 | ABAminus | -92.07, -26.65 | -133.67, 178.16 | -123.93, 6.5 | 294.94, 97.33 | 89.15, -162.77 | in-out | in | 9.5208 | Saltbr-out | 4.8419 | HRD-in | -77.17, -59.97 | 76.05, -10.25 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.7895 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -62.14, 143.17 | APE9-dihe-na | -120.32, 118.65 | APE8-dihe-in | -75.39, 123.94 | APE8-rot-in | 299.29 | APE67-dihe-in | -61.41, -23.9 | -115.12, 4.11 | APE12-dist-out | 18.7072 | APE11-dist-out | 15.3251 | APE10-dist-out | 16.6803 | APE9-dist-out | 11.2441 | None | None | None | XRAY | 1.7 | 0.177 | 0.222 | A | 366.0 | 359.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 8r5e | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 1UKHA | P45983 | 9 | 363 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.009 | 13.5918 | ABAminus | -71.05, -50.54 | -134.57, 170.42 | -88.05, 19.73 | 310.31, 96.24 | 54.55, -119.32 | in-in | in | 8.7257 | Saltbr-in | 3.5395 | HRD-in | -32.35, -66.36 | 74.83, -11.73 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | 999.0, -21.95 | 999.0, 999.0 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.35 | 0.229 | 0.245 | A | 369.0 | 321.0 | 22 | 27 | 10 | 17 | [[26, 321]] | 1.0 | 1ukh | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4YR8A | P45983 | 8 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 3.746 | 13.6511 | ABAminus | -92.48, -36.82 | -128.7, -177.95 | -116.24, 9.95 | 302.59, 109.3 | 79.22, -159.79 | in-in | in | 9.397 | Saltbr-in | 2.7167 | HRD-in | -91.12, -57.47 | 70.8, -11.5 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 120.35 | APE8-dihe-in | -90.35, 105.5 | APE8-rot-out | 50.94 | APE67-dihe-in | -67.62, -16.88 | -108.83, 0.82 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.1748 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | A | 371.0 | 320.0 | 17 | 27 | 14 | 13 | [[26, 321]] | 1.0 | 4yr8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4YR8C | P45983 | 10 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.3451 | 13.3914 | ABAminus | -88.52, -41.45 | -131.53, -175.1 | -114.96, 11.59 | 302.69, 109.92 | 79.73, 999.0 | in-in | in | 8.8736 | Saltbr-in | 2.6944 | HRD-in | -68.29, -62.18 | 77.05, -0.67 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanni | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 118.23 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.66, -18.42 | -99.29, -2.8 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | C | 371.0 | 318.0 | 21 | 27 | 11 | 16 | [[26, 321]] | 1.0 | 4yr8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4YR8E | P45983 | 7 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 3.7276 | 14.1372 | ABAminus | -86.08, -36.9 | -129.28, 170.42 | -104.47, 7.33 | 299.61, 110.26 | 81.64, -165.5 | out-out | out | 10.093 | Saltbr-out | 3.6951 | HRD-in | -78.61, -55.83 | 65.3, 1.9 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8909 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -50.39 | APE8-dihe-in | -79.39, 102.65 | APE8-rot-out | 53.21 | APE67-dihe-in | -61.82, -18.77 | -109.31, -0.43 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.7944 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | E | 371.0 | 317.0 | 17 | 27 | 15 | 12 | [[26, 321]] | 1.0 | 4yr8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4YR8F | P45983 | 10 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.6068 | 13.3341 | ABAminus | -92.28, -40.63 | -125.1, 178.19 | -117.35, 11.6 | 304.63, 110.41 | 81.03, 999.0 | in-in | in | 8.5474 | Saltbr-in | 2.4139 | HRD-in | -61.32, -58.08 | 77.0, -3.6 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanni | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 114.52 | APE8-rot-none | 999.0 | APE67-dihe-in | -64.79, -18.18 | -101.48, -2.27 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.4 | 0.218 | 0.239 | F | 371.0 | 300.0 | 38 | 27 | 11 | 16 | [[26, 321]] | 1.0 | 4yr8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.5e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 6F5EB | P45983 | 7 | 362 | 427.0 | No_ligand | No_ligand | Inactive | DFGin | 4.2446 | 14.401 | ABAminus | -85.23, -40.02 | -143.49, -172.1 | -102.9, -4.9 | 292.34, 110.9 | 97.56, -150.23 | in-in | in | 9.2523 | Saltbr-in | 3.1606 | HRD-in | -56.05, -56.91 | 72.46, 7.42 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9127 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | APE10-dihe-na | 999.0, 112.0 | APE9-dihe-na | -95.81, 149.23 | APE8-dihe-out | -71.37, -38.95 | APE8-rot-in | 293.49 | APE67-dihe-in | -53.11, -31.53 | -58.04, -34.44 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 14.7564 | APE9-dist-out | 11.1737 | None | None | None | XRAY | 2.7 | 0.202 | 0.226 | B | 373.0 | 346.0 | 10 | 27 | 23 | 4 | [[26, 321]] | 1.0 | 6f5e | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8X5MA | P45983 | 7 | 363 | 427.0 | Y4O:401 | Type1 | Inactive | DFGin | 3.8295 | 13.7211 | ABAminus | -82.03, -35.59 | -145.84, 177.75 | -109.61, 10.51 | 302.7, 100.16 | 80.95, -155.06 | in-in | in | 9.1059 | Saltbr-in | 2.7679 | HRD-in | -69.78, -60.93 | 77.08, -7.13 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.2374 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 140.93 | APE8-dihe-in | -94.27, 100.92 | APE8-rot-in | 297.8 | APE67-dihe-in | -57.39, -30.56 | -110.37, 11.17 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 12.1596 | None | None | CSO163 | XRAY | 2.0 | 0.195 | 0.234 | A | 363.0 | 341.0 | 16 | 27 | 15 | 12 | [[26, 321]] | 1.0 | 8x5m | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 7.9e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PT8A | P45983 | 7 | 363 | 427.0 | A3O:401 | Type1 | Inactive | DFGin | 3.5115 | 13.6408 | ABAminus | -86.46, -36.69 | -113.24, 157.51 | -107.14, 5.23 | 297.22, 84.35 | 63.56, -136.9 | in-out | in | 9.7221 | Saltbr-out | 5.4719 | HRD-in | -69.36, -62.04 | 67.14, -1.26 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.2593 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nioo | APE10-dihe-na | -78.69, 132.14 | APE9-dihe-na | -97.09, 6.93 | APE8-dihe-in | -119.44, 125.16 | APE8-rot-out | 77.92 | APE67-dihe-in | -61.62, -35.67 | -102.35, -19.0 | APE12-dist-none | 999.0 | APE11-dist-in | 10.0559 | APE10-dist-out | 10.1664 | APE9-dist-out | 11.4072 | None | None | None | XRAY | 2.78 | 0.219 | 0.218 | A | 366.0 | 353.0 | 2 | 27 | 25 | 2 | [[26, 321]] | 1.0 | 8pt8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PT8B | P45983 | 8 | 363 | 427.0 | A3O:401 | Type1 | Inactive | DFGin | 3.7083 | 13.5603 | ABAminus | -87.46, -36.99 | -114.07, 158.6 | -107.2, 3.96 | 306.69, 95.61 | 61.75, -138.76 | out-out | out | 10.0137 | Saltbr-out | 4.7072 | HRD-in | -65.17, -60.14 | 69.69, -8.9 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.0336 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_iioo | APE10-dihe-na | -125.68, 169.43 | APE9-dihe-na | -89.29, -51.47 | APE8-dihe-out | 50.18, 54.05 | APE8-rot-out | 80.12 | APE67-dihe-in | -59.08, -31.41 | -75.35, -27.98 | APE12-dist-in | 11.3425 | APE11-dist-in | 8.5237 | APE10-dist-out | 11.6714 | APE9-dist-out | 8.6343 | None | None | None | XRAY | 2.78 | 0.219 | 0.218 | B | 366.0 | 354.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 8pt8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PT8C | P45983 | 7 | 362 | 427.0 | A3O:401 | Type1 | Inactive | DFGin | 4.333 | 13.6339 | ABAminus | -100.64, -42.98 | -112.04, 163.18 | -107.79, 3.91 | 318.61, 83.5 | 62.89, -142.35 | in-out | in | 9.3615 | Saltbr-out | 6.3544 | HRD-in | -65.16, -58.91 | 71.32, -6.19 | out-out-out | SNCooo | out-out | ActLoopNT-out | 5.1345 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -0.16 | APE9-dihe-na | -89.45, -4.71 | APE8-dihe-in | -89.37, 113.03 | APE8-rot-out | 66.41 | APE67-dihe-in | -51.88, -31.5 | -134.08, -10.25 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 11.551 | APE9-dist-out | 11.4356 | None | None | None | XRAY | 2.78 | 0.219 | 0.218 | C | 366.0 | 353.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 8pt8 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PT9A | P45983 | 8 | 363 | 427.0 | DVI:401 | Type1 | Inactive | DFGin | 3.6725 | 13.8445 | ABAminus | -82.42, -42.96 | -101.44, 156.25 | -107.65, 10.42 | 293.61, 64.96 | 107.26, -173.51 | out-in | out | 10.2179 | Saltbr-in | 3.1648 | HRD-in | -86.93, -57.09 | 73.38, 1.77 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.3496 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_iooo | APE10-dihe-na | -132.39, 130.51 | APE9-dihe-na | -63.89, -49.36 | APE8-dihe-out | 47.93, 60.73 | APE8-rot-out | 86.13 | APE67-dihe-in | -60.85, -39.95 | -75.12, -7.36 | APE12-dist-in | 10.0694 | APE11-dist-out | 6.9139 | APE10-dist-out | 10.6396 | APE9-dist-out | 8.438 | None | None | None | XRAY | 2.7 | 0.215 | 0.225 | A | 366.0 | 353.0 | 2 | 27 | 25 | 2 | [[26, 321]] | 1.0 | 8pt9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PT9B | P45983 | 7 | 363 | 427.0 | DVI:401 | Type1 | Inactive | DFGin | 3.6022 | 13.3587 | ABAminus | -78.87, -38.7 | -110.84, 150.53 | -102.26, 4.03 | 302.35, 93.73 | 66.71, -148.92 | in-out | in | 9.405 | Saltbr-out | 4.004 | HRD-in | -82.54, -61.31 | 64.36, 5.02 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nioo | APE10-dihe-na | -99.2, 123.92 | APE9-dihe-na | -85.67, -7.28 | APE8-dihe-in | -87.66, 94.6 | APE8-rot-out | 69.53 | APE67-dihe-in | -57.65, -34.34 | -84.42, -14.13 | APE12-dist-none | 999.0 | APE11-dist-in | 9.9637 | APE10-dist-out | 10.6502 | APE9-dist-out | 11.067 | None | None | None | XRAY | 2.7 | 0.215 | 0.225 | B | 366.0 | 351.0 | 5 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 8pt9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PT9C | P45983 | 8 | 362 | 427.0 | DVI:401 | Type1 | Inactive | DFGin | 3.804 | 14.2556 | ABAminus | -88.85, -34.33 | -106.1, 147.38 | -98.39, 6.8 | 298.91, 67.63 | 59.14, -132.88 | out-out | out | 10.1832 | Saltbr-out | 3.8904 | HRD-in | -79.93, -61.89 | 65.26, 3.23 | out-out-out | SNCooo | out-out | ActLoopNT-out | 4.6788 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -169.35 | APE9-dihe-na | -94.15, 7.09 | APE8-dihe-in | -84.28, 82.63 | APE8-rot-out | 73.62 | APE67-dihe-in | -62.72, -39.65 | -92.57, -5.37 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 11.9341 | APE9-dist-out | 11.2227 | None | None | None | XRAY | 2.7 | 0.215 | 0.225 | C | 366.0 | 352.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 8pt9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PTAA | P45983 | 8 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.923 | 14.4771 | ABAminus | -80.58, -61.37 | -103.85, 165.38 | -100.79, 23.99 | 295.77, 91.74 | 73.84, -149.47 | in-in | in | 9.7897 | Saltbr-in | 3.1262 | HRD-in | -78.59, -61.53 | 62.23, 7.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.4702 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iooo | APE10-dihe-na | -130.45, 138.38 | APE9-dihe-na | -101.99, 109.25 | APE8-dihe-in | -118.89, 112.23 | APE8-rot-out | 53.5 | APE67-dihe-in | -51.79, -30.07 | -95.29, -17.54 | APE12-dist-in | 10.569 | APE11-dist-out | 7.0333 | APE10-dist-out | 10.1833 | APE9-dist-out | 8.5978 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | A | 366.0 | 354.0 | 2 | 27 | 25 | 2 | [[26, 321]] | 1.0 | 8pta | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PTAB | P45983 | 7 | 363 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.5773 | 13.1788 | ABAminus | -81.24, -57.35 | -101.3, 158.61 | -105.36, 14.2 | 308.93, 93.28 | 64.59, -148.13 | in-in | in | 9.3658 | Saltbr-in | 3.5356 | HRD-in | -77.41, -61.25 | 61.49, 9.23 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -112.33, 168.25 | APE9-dihe-na | -116.9, 36.67 | APE8-dihe-in | -104.63, 91.0 | APE8-rot-out | 52.55 | APE67-dihe-in | -56.88, -29.41 | -95.02, -21.65 | APE12-dist-in | 11.7839 | APE11-dist-in | 9.1521 | APE10-dist-out | 11.2421 | APE9-dist-out | 10.2145 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | B | 366.0 | 352.0 | 5 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 8pta | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 8PTAC | P45983 | 8 | 361 | 427.0 | CIF:401 | Type1 | Inactive | DFGin | 3.8263 | 14.0885 | ABAminus | -83.97, -56.35 | -97.04, 154.46 | -105.76, 13.83 | 294.99, 32.04 | 63.79, -147.27 | in-out | in | 9.7228 | Saltbr-out | 4.5276 | HRD-in | -77.01, -60.9 | 63.25, 7.56 | out-out-out | SNCooo | out-out | ActLoopNT-out | 4.6109 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_nnoo | APE10-dihe-na | 999.0, -137.59 | APE9-dihe-na | -94.11, 17.64 | APE8-dihe-in | -81.48, 63.35 | APE8-rot-out | 71.39 | APE67-dihe-in | -58.68, -26.77 | -108.19, -24.77 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 12.4666 | APE9-dist-out | 10.7804 | None | None | None | XRAY | 2.41 | 0.224 | 0.226 | C | 366.0 | 351.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 8pta | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.1e-85 | 290.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 1UKIA | P45983 | 9 | 363 | 427.0 | 537:0 | Type1 | Inactive | DFGin | 4.7042 | 13.1142 | ABAminus | -77.11, -62.2 | -116.68, -161.07 | -126.7, 15.2 | 318.68, 71.9 | 41.91, -116.91 | in-in | in | 9.1687 | Saltbr-in | 2.9158 | HRD-in | -66.76, -57.64 | 78.15, -46.3 | in-out-out | SNCioo | out-out | ActLoopNT-out | 5.4563 | ActLoopCT-out | nonTYR | APEdihe_aanio | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 77.25 | APE8-rot-in | 304.87 | APE67-dihe-out | -76.75, -17.12 | 155.56, -17.08 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.7 | 0.221 | 0.241 | A | 369.0 | 328.0 | 18 | 27 | 14 | 13 | [[26, 321]] | 1.0 | 1uki | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4E73A | P45983 | 8 | 361 | 427.0 | 0NR:60401 | Type1 | Inactive | DFGin | 3.9405 | 13.7141 | ABAminus | -80.5, -42.58 | -144.32, -163.84 | -110.6, 6.62 | 304.02, 132.42 | 68.66, -151.79 | in-in | in | 9.1157 | Saltbr-in | 2.603 | HRD-in | -76.2, -63.12 | 71.21, -5.48 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -70.49, -32.11 | 999.0, 34.81 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.27 | 0.249 | 0.282 | A | 369.0 | 318.0 | 23 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4e73 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4G1WA | P45983 | 8 | 361 | 427.0 | G1W:60401 | Type1 | Inactive | DFGin | 4.1305 | 13.7474 | ABAminus | -75.19, -46.06 | -145.01, -166.31 | -101.8, 11.35 | 310.93, 129.6 | 54.15, -150.73 | in-in | in | 9.5121 | Saltbr-in | 2.8152 | HRD-in | -74.24, -60.52 | 76.29, -17.95 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 110.92 | APE8-rot-in | 305.3 | APE67-dihe-in | -68.41, -20.62 | -111.33, 3.9 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.45 | 0.233 | 0.297 | A | 369.0 | 322.0 | 22 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4g1w | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4HYSA | P45983 | 8 | 361 | 427.0 | 1BJ:60401 | Type1 | Inactive | DFGin | 4.1442 | 13.7039 | ABAminus | -65.58, -42.99 | -148.13, -172.29 | -105.42, 11.47 | 305.84, 116.47 | 62.72, -152.88 | in-in | in | 9.1693 | Saltbr-in | 2.5418 | HRD-in | -81.1, -55.52 | 80.05, -13.7 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 85.27 | APE8-rot-in | 300.61 | APE67-dihe-in | -75.95, -19.65 | -89.11, 15.51 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.415 | 0.249 | 0.295 | A | 369.0 | 321.0 | 23 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4hys | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4HYUA | P45983 | 8 | 361 | 427.0 | 1BK:60401 | Type1 | Inactive | DFGin | 4.0678 | 13.5935 | ABAminus | -80.82, -40.1 | -141.28, -176.81 | -103.55, 4.37 | 303.13, 103.89 | 67.61, -155.32 | in-in | in | 9.276 | Saltbr-in | 2.7839 | HRD-in | -63.72, -62.24 | 77.82, -3.04 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 97.87 | APE8-rot-in | 304.34 | APE67-dihe-in | -66.69, -21.83 | -103.0, 8.43 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.152 | 0.231 | 0.269 | A | 369.0 | 322.0 | 22 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4hyu | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4IZYA | P45983 | 8 | 361 | 427.0 | 1J2:60401 | Type1 | Inactive | DFGin | 3.8819 | 13.4843 | ABAminus | -76.71, -38.87 | -145.64, -179.24 | -102.44, 14.51 | 311.23, 93.45 | 52.84, -142.09 | in-in | in | 9.149 | Saltbr-in | 2.7383 | HRD-in | -72.23, -60.13 | 78.79, -8.13 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 111.06 | APE8-rot-in | 300.16 | APE67-dihe-in | -67.83, -22.42 | -106.79, 8.95 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 2.3 | 0.239 | 0.261 | A | 369.0 | 322.0 | 22 | 27 | 12 | 15 | [[26, 321]] | 1.0 | 4izy | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 8.3e-85 | 290.5 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3PZEA | P45983 | 7 | 362 | 427.0 | CFK:1 | Type1 | Inactive | DFGin | 4.1379 | 13.9068 | ABAminus | -81.12, -32.94 | -131.86, 179.29 | -115.73, 16.97 | 304.08, 91.38 | 65.8, -99.93 | in-in | in | 8.7987 | Saltbr-in | 2.79 | HRD-in | -65.45, -61.37 | 74.31, -21.03 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 43.07 | APE8-dihe-out | -90.42, -23.2 | APE8-rot-in | 308.55 | APE67-dihe-in | -65.57, -26.71 | -47.05, -33.16 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.1182 | None | None | None | XRAY | 2.0 | 0.206 | 0.24 | A | 358.0 | 347.0 | 9 | 27 | 18 | 9 | [[26, 321]] | 1.0 | 3pze | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.1e-84 | 288.3 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4L7FA | P45983 | 7 | 362 | 427.0 | 1V5:60401 | Type1 | Inactive | DFGin | 4.168 | 13.9028 | ABAminus | -92.73, -21.27 | -136.46, -179.9 | -126.51, 2.69 | 298.75, 92.07 | 123.75, 92.84 | in-in | in | 9.571 | Saltbr-in | 2.7172 | HRD-in | -73.68, -60.59 | 73.9, -18.64 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnoo | APE10-dihe-na | 999.0, 56.52 | APE9-dihe-na | -75.12, 136.19 | APE8-dihe-in | -88.12, 112.11 | APE8-rot-in | 306.44 | APE67-dihe-in | -64.04, -21.62 | -99.03, -5.95 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 14.8393 | APE9-dist-out | 11.6873 | None | None | None | XRAY | 1.95 | 0.162 | 0.198 | A | 367.0 | 343.0 | 13 | 27 | 14 | 13 | [[26, 321]] | 1.0 | 4l7f | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.4e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3ELJA | P45983 | 7 | 364 | 427.0 | GS7:365 | Type1 | Inactive | DFGin | 4.2607 | 13.8455 | ABAminus | -96.2, -23.23 | -129.0, 175.64 | -123.66, 12.92 | 303.89, 93.13 | 80.21, -148.51 | in-in | in | 9.2759 | Saltbr-in | 3.4358 | HRD-in | -62.88, -61.88 | 76.44, -14.77 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -113.33, 122.34 | APE9-dihe-na | -76.53, 136.67 | APE8-dihe-in | -80.59, 119.63 | APE8-rot-in | 296.46 | APE67-dihe-in | -59.78, -20.24 | -110.49, 3.47 | APE12-dist-out | 20.996 | APE11-dist-out | 15.8219 | APE10-dist-out | 16.3336 | APE9-dist-out | 11.4349 | None | None | None | XRAY | 1.8 | 0.188 | 0.215 | A | 369.0 | 347.0 | 6 | 27 | 21 | 6 | [[26, 321]] | 1.0 | 3elj | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.5e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4AWIA | P45983 | 8 | 364 | 427.0 | AQ2:1365 | Type1 | Inactive | DFGin | 4.4603 | 13.936 | ABAminus | -87.42, -26.01 | -133.81, 169.02 | -108.8, 6.11 | 295.82, 101.28 | 92.5, -161.91 | in-in | in | 8.9051 | Saltbr-in | 2.7425 | HRD-in | -70.34, -61.6 | 77.73, -9.92 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -85.55, 146.28 | APE9-dihe-na | -95.6, 128.29 | APE8-dihe-in | -89.62, 121.11 | APE8-rot-in | 309.81 | APE67-dihe-in | -66.82, -18.55 | -120.34, 14.07 | APE12-dist-out | 18.8339 | APE11-dist-out | 14.9052 | APE10-dist-out | 16.4247 | APE9-dist-out | 11.46 | None | None | None | XRAY | 1.91 | 0.188 | 0.219 | A | 369.0 | 352.0 | 5 | 27 | 22 | 5 | [[26, 321]] | 1.0 | 4awi | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.5e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 5LW1B | P45983 | 8 | 362 | 427.0 | ADN:60401 | Type1 | Inactive | DFGin | 4.4197 | 14.4478 | ABAminus | -83.29, -51.84 | -118.5, -177.73 | -115.08, 20.0 | 298.98, 87.21 | 71.2, -159.63 | out-out | out | 10.4298 | Saltbr-out | 3.8124 | HRD-in | -68.61, -60.19 | 64.51, 12.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.4773 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -136.58, 144.4 | APE9-dihe-na | -122.04, 105.79 | APE8-dihe-out | -71.41, -33.58 | APE8-rot-in | 307.18 | APE67-dihe-in | -61.62, -32.85 | -63.18, -22.53 | APE12-dist-out | 20.0348 | APE11-dist-out | 18.2025 | APE10-dist-out | 13.7638 | APE9-dist-out | 11.7502 | None | None | None | XRAY | 3.2 | 0.177 | 0.212 | B | 373.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 5lw1 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 5LW1E | P45983 | 8 | 362 | 427.0 | ADN:60401 | Type1 | Inactive | DFGin | 4.1748 | 14.0755 | ABAminus | -82.51, -53.19 | -119.45, -176.34 | -115.64, 20.66 | 300.14, 87.37 | 72.63, -160.31 | in-out | in | 9.9432 | Saltbr-out | 4.611 | HRD-in | -68.12, -61.52 | 63.83, 14.63 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8826 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -137.31, 145.55 | APE9-dihe-na | -120.94, 104.94 | APE8-dihe-out | -71.75, -32.64 | APE8-rot-in | 307.04 | APE67-dihe-in | -62.19, -31.77 | -62.28, -22.63 | APE12-dist-out | 20.0912 | APE11-dist-out | 18.3879 | APE10-dist-out | 14.0865 | APE9-dist-out | 12.0009 | None | None | None | XRAY | 3.2 | 0.177 | 0.212 | E | 373.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 5lw1 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 5LW1H | P45983 | 8 | 362 | 427.0 | ADN:60401 | Type1 | Inactive | DFGin | 4.1303 | 14.3776 | ABAminus | -82.43, -51.23 | -118.2, -176.9 | -114.7, 20.75 | 298.45, 87.29 | 72.11, -159.03 | out-out | out | 10.2847 | Saltbr-out | 3.7377 | HRD-in | -69.31, -61.29 | 63.64, 13.39 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.4743 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -136.56, 144.9 | APE9-dihe-na | -119.98, 105.48 | APE8-dihe-out | -71.78, -33.35 | APE8-rot-in | 307.69 | APE67-dihe-in | -61.37, -31.81 | -63.06, -22.73 | APE12-dist-out | 20.0957 | APE11-dist-out | 18.3691 | APE10-dist-out | 13.9653 | APE9-dist-out | 11.9943 | None | None | None | XRAY | 3.2 | 0.177 | 0.212 | H | 373.0 | 355.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 5lw1 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.7e-84 | 288.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4QTDA | P45983 | 6 | 363 | 427.0 | 38Z:424,ANP:425 | Type1,Allosteric | Inactive | DFGin | 4.2787 | 13.95 | ABAminus | -89.69, -21.2 | -135.34, 171.77 | -115.48, 9.24 | 298.02, 89.8 | 87.52, -156.74 | in-out | in | 9.5926 | Saltbr-out | 4.1531 | HRD-in | -75.36, -55.62 | 72.51, -12.26 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.6893 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -117.32, 137.81 | APE9-dihe-na | -80.42, 132.23 | APE8-dihe-in | -83.54, 120.1 | APE8-rot-in | 296.41 | APE67-dihe-in | -61.39, -20.52 | -109.55, -3.05 | APE12-dist-out | 21.1401 | APE11-dist-out | 16.032 | APE10-dist-out | 16.5166 | APE9-dist-out | 11.1471 | None | None | None | XRAY | 1.5 | 0.167 | 0.192 | A | 364.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 4qtd | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 9FT9A | P45983 | 7 | 363 | 427.0 | ANP:401 | ATPlike | Inactive | DFGin | 6.2012 | 13.6807 | BLAminus | -138.37, -170.04 | 58.94, 78.24 | -92.66, 22.82 | 315.32, 103.73 | -63.89, -26.18 | in-out | in | 8.5419 | Saltbr-out | 3.8425 | HRD-in | -66.92, -47.02 | 65.13, 0.51 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8271 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oioo | APE10-dihe-na | -150.17, 156.5 | APE9-dihe-na | -75.27, -52.01 | APE8-dihe-in | -88.35, 100.07 | APE8-rot-in | 310.81 | APE67-dihe-in | -64.72, -11.39 | -102.84, 1.94 | APE12-dist-out | 5.9095 | APE11-dist-in | 10.5805 | APE10-dist-out | 8.0786 | APE9-dist-out | 10.9491 | None | None | None | XRAY | 2.35 | 0.234 | 0.27 | A | 360.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 9ft9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.1e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3V3VA | P45983 | 7 | 363 | 427.0 | MYU:401 | Type1 | Inactive | DFGin | 6.8274 | 13.7856 | BLAminus | -143.77, -172.33 | 52.69, 90.19 | -99.08, 8.98 | 306.34, 125.67 | -39.78, -30.71 | in-in | in | 8.0358 | Saltbr-in | 2.8823 | HRD-in | -67.72, -38.9 | 75.22, -25.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.605 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -111.93, -15.72 | APE9-dihe-na | -81.89, 141.96 | APE8-dihe-in | -63.44, 127.02 | APE8-rot-out | 31.94 | APE67-dihe-in | -66.37, -23.13 | -30.24, -61.71 | APE12-dist-in | 12.8042 | APE11-dist-in | 12.8097 | APE10-dist-in | 7.6481 | APE9-dist-in | 5.1004 | None | None | None | XRAY | 2.7 | 0.229 | 0.266 | A | 379.0 | 351.0 | 6 | 27 | 23 | 4 | [[26, 321]] | 1.0 | 3v3v | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 3.3e-84 | 288.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2GMXA | P45983 | 8 | 364 | 427.0 | 877:60901 | Type1 | Inactive | DFGin | 6.4145 | 15.103 | BLAminus | -169.49, -165.44 | 17.67, 94.27 | -93.05, 32.73 | 281.95, 52.09 | -74.74, -22.92 | in-in | in | 9.2457 | Saltbr-in | 3.4507 | HRD-in | -84.23, -59.06 | 73.39, 47.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7327 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -71.92, -33.15 | APE9-dihe-na | -81.6, 112.65 | APE8-dihe-in | -25.7, 132.77 | APE8-rot-out | 32.67 | APE67-dihe-in | -46.1, -17.73 | -58.05, -70.61 | APE12-dist-in | 10.542 | APE11-dist-in | 13.1827 | APE10-dist-in | 7.8512 | APE9-dist-in | 4.9448 | T183E,Y185E | None | None | XRAY | 3.5 | 0.278 | 0.351 | A | 370.0 | 357.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2gmx | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 4UX9B | P45983 | 8 | 362 | 427.0 | ANP:1000 | ATPlike | Inactive | DFGin | 6.8269 | 14.0009 | None | -95.23, -79.97 | -82.17, 124.02 | -113.22, 13.68 | 297.81, 107.19 | -60.29, -32.64 | in-in | in | 8.6029 | Saltbr-in | 2.9418 | HRD-in | -59.44, -53.0 | 79.08, -24.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.5822 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -58.47, -40.48 | APE9-dihe-na | -78.17, 138.93 | APE8-dihe-in | -64.59, 122.35 | APE8-rot-in | 308.57 | APE67-dihe-in | -67.83, -19.56 | -32.59, -57.13 | APE12-dist-in | 12.3608 | APE11-dist-in | 12.1486 | APE10-dist-in | 6.5271 | APE9-dist-in | 4.6911 | None | None | None | XRAY | 2.34 | 0.202 | 0.24 | B | 364.0 | 327.0 | 14 | 27 | 21 | 6 | [[26, 321]] | 1.0 | 4ux9 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2G01B | P45983 | 9 | 364 | 427.0 | 73Q:61001 | Type1 | Inactive | DFGin | 5.7329 | 14.7118 | None | -124.05, -159.93 | 70.3, -99.04 | 78.28, -8.58 | 269.85, 26.32 | -60.64, -29.84 | in-in | in | 9.3096 | Saltbr-in | 3.522 | HRD-in | -75.33, -51.61 | 81.6, -31.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0497 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -55.32, -77.05 | APE9-dihe-na | -50.72, 131.97 | APE8-dihe-in | -62.41, 127.97 | APE8-rot-out | 179.45 | APE67-dihe-in | -34.47, -20.37 | -26.15, -85.34 | APE12-dist-in | 12.6428 | APE11-dist-in | 12.8438 | APE10-dist-in | 7.3262 | APE9-dist-in | 4.7568 | T183E,Y185E | None | None | XRAY | 3.5 | 0.296 | 0.354 | B | 370.0 | 356.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2g01 | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 2GMXB | P45983 | 7 | 364 | 427.0 | 877:61001 | Type1 | Inactive | DFGin | 5.6113 | 13.9429 | None | -106.95, -175.57 | 54.48, -113.25 | 110.31, -6.6 | 279.44, 165.75 | -41.3, -39.48 | in-out | in | 8.4562 | Saltbr-out | 4.4993 | HRD-in | -77.53, -48.43 | 77.05, -21.57 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8017 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -70.75, -77.84 | APE9-dihe-na | -45.43, 98.08 | APE8-dihe-in | -37.04, 123.81 | APE8-rot-in | 354.32 | APE67-dihe-in | -25.17, -38.2 | -26.5, -90.08 | APE12-dist-in | 11.7738 | APE11-dist-in | 12.5874 | APE10-dist-in | 7.2474 | APE9-dist-in | 4.4727 | T183E,Y185E | None | None | XRAY | 3.5 | 0.278 | 0.351 | B | 370.0 | 358.0 | 0 | 27 | 27 | 0 | [[26, 321]] | 1.0 | 2gmx | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-83 | 285.6 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VULA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | None | DFGin | 5.1102 | 13.7682 | BLAminus | -85.93, 163.21 | 85.46, 126.64 | -150.76, 1.53 | 338.77, 110.45 | -63.64, 22.92 | in-in | in | 9.4027 | Saltbr-in | 3.0531 | HRD-in | -77.29, -39.59 | 61.8, -14.75 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.6801 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -129.09, 14.97 | 999.0, -38.05 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | C79V,C116S,C137V,C163A,C213V,C245S | None | None | XRAY | 2.81 | 0.252 | 0.315 | A | 370.0 | 344.0 | 14 | 27 | 13 | 14 | [[26, 321]] | 1.0 | 3vul | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.6e-81 | 279.1 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| MAPK8 | MK08_HUMAN | 3VUMA | P45983 | 7 | 364 | 427.0 | No_ligand | No_ligand | None | DFGin | 5.0561 | 13.607 | BLAminus | -112.58, 170.27 | 77.92, 128.69 | -145.25, 34.84 | 350.71, 122.87 | -58.09, -36.69 | in-in | in | 9.0374 | Saltbr-in | 2.9813 | HRD-in | -72.36, -43.79 | 70.87, -4.2 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9289 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -69.29, -4.06 | 999.0, -24.38 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | C41V,C79V,C116S,C137V,C163A,C213V,C245S | None | None | XRAY | 2.69 | 0.192 | 0.255 | A | 370.0 | 344.0 | 14 | 27 | 13 | 14 | [[26, 321]] | 1.0 | 3vum | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 2.8e-81 | 279.0 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|